AR051674A1 - Farmacos y profarmacos utiles para el tratamiento de equilibrio energetico en rumiantes - Google Patents

Farmacos y profarmacos utiles para el tratamiento de equilibrio energetico en rumiantes

Info

Publication number
AR051674A1
AR051674A1 ARP050104842A ARP050104842A AR051674A1 AR 051674 A1 AR051674 A1 AR 051674A1 AR P050104842 A ARP050104842 A AR P050104842A AR P050104842 A ARP050104842 A AR P050104842A AR 051674 A1 AR051674 A1 AR 051674A1
Authority
AR
Argentina
Prior art keywords
ruminants
compound
isomer
energy balance
negative energy
Prior art date
Application number
ARP050104842A
Other languages
English (en)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of AR051674A1 publication Critical patent/AR051674A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/472Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00General protective or antinoxious agents
    • A61P39/02Antidotes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Nutrition Science (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Toxicology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

El uso de un compuesto de formula (1), un isomero del mismo, un profármaco de dicho compuesto o isomero o una sal farmacéuticamente aceptable de dicho compuesto, isomero o profármaco, en la fabricacion de un medicamento para el tratamiento paliativo, profiláctico o curativo de equilibrio energético negativo en rumiantes. El uso de un compuesto de formula (1), en la fabricacion de un medicamento para el tratamiento paliativo, profiláctico o curativo de la enfermedad de la enfermedad del rumiante asociada con equilibrio energético negativo en rumiantes, en el que, preferiblemente la enfermedad de los rumiantes asociada con equilibrio energético negativo en rumiantes se selecciona de: esteatosis, hepática, distocia, disfuncion inmunitaria, inmunodeficiencia, envenenamiento, cetosis primaria, cetosis secundaria, síndrome de la vaca que no puede sostenerse por sí misma, dispepsia, inapetencia, placenta retenida, abomaso desplazado, mastitis, (endo-)-metritis, esterilidad, baja fertilidad y cojera.
ARP050104842A 2004-11-18 2005-11-17 Farmacos y profarmacos utiles para el tratamiento de equilibrio energetico en rumiantes AR051674A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US62910904P 2004-11-18 2004-11-18

Publications (1)

Publication Number Publication Date
AR051674A1 true AR051674A1 (es) 2007-01-31

Family

ID=35695821

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP050104842A AR051674A1 (es) 2004-11-18 2005-11-17 Farmacos y profarmacos utiles para el tratamiento de equilibrio energetico en rumiantes

Country Status (8)

Country Link
US (1) US20080096916A1 (es)
EP (1) EP1824484A1 (es)
JP (1) JP2008520643A (es)
AR (1) AR051674A1 (es)
AU (1) AU2005305593A1 (es)
CA (1) CA2587690A1 (es)
TW (1) TW200631579A (es)
WO (1) WO2006054166A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2007210076A1 (en) * 2006-01-30 2007-08-09 Irm Llc Polycyclic 1, 2, 3, 4 -tetrahydro- isoquinoline derivatives and compositions comprising them as PPAR modulators
US8791105B2 (en) 2010-07-14 2014-07-29 Kansas State University Research Foundation Methods for alleviating chronic pain and improving performance of cattle undergoing dehorning or castration

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI52797C (fi) * 1971-03-17 1977-12-12 Rumen Chemie Ag Lisärehu märehtijöitä varten.
AU779266B2 (en) * 2000-05-11 2005-01-13 Banyu Pharmaceutical Co., Ltd. N-acyltetrahydroisoquinoline derivatives
US6867224B2 (en) * 2002-03-07 2005-03-15 Warner-Lambert Company Compounds that modulate PPAR activity and methods of preparation
DE60306636T2 (de) * 2002-04-09 2007-07-05 Eli Lilly And Co., Indianapolis Wachstumhormonsekretionsförderer
US6987118B2 (en) * 2003-05-21 2006-01-17 Pfizer Inc. Tetrahydroisoquinoline derivatives as PPAR-alpha activators

Also Published As

Publication number Publication date
WO2006054166A1 (en) 2006-05-26
EP1824484A1 (en) 2007-08-29
AU2005305593A1 (en) 2006-05-26
US20080096916A1 (en) 2008-04-24
CA2587690A1 (en) 2006-05-26
JP2008520643A (ja) 2008-06-19
TW200631579A (en) 2006-09-16

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