AR033305A1 - Procedimiento para preparar un aminoacido biciclico - Google Patents

Procedimiento para preparar un aminoacido biciclico

Info

Publication number
AR033305A1
AR033305A1 ARP020101609A ARP020101609A AR033305A1 AR 033305 A1 AR033305 A1 AR 033305A1 AR P020101609 A ARP020101609 A AR P020101609A AR P020101609 A ARP020101609 A AR P020101609A AR 033305 A1 AR033305 A1 AR 033305A1
Authority
AR
Argentina
Prior art keywords
procedure
bicycle
prepare
amino acid
aminomethylbicyclo
Prior art date
Application number
ARP020101609A
Other languages
English (en)
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of AR033305A1 publication Critical patent/AR033305A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/12Formation of amino and carboxyl groups
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00Systems containing two condensed rings
    • C07C2602/02Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/14All rings being cycloaliphatic
    • C07C2602/20All rings being cycloaliphatic the ring system containing seven carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

La presente se refiere a un procedimiento para preparar ácido (1,3,5)-(3-aminometilbiciclo[3.2.0]hept-3-il)acético, o una de sus sales de adicion de ácidos. En el esquema (1) de reaccion se muestra una realizacion del procedimiento.
ARP020101609A 2001-05-04 2002-05-02 Procedimiento para preparar un aminoacido biciclico AR033305A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB0110935A GB2375109A (en) 2001-05-04 2001-05-04 Process for preparing bicyclic amino acid

Publications (1)

Publication Number Publication Date
AR033305A1 true AR033305A1 (es) 2003-12-10

Family

ID=9914014

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP020101609A AR033305A1 (es) 2001-05-04 2002-05-02 Procedimiento para preparar un aminoacido biciclico

Country Status (4)

Country Link
US (1) US20030083520A1 (es)
AR (1) AR033305A1 (es)
GB (1) GB2375109A (es)
WO (1) WO2002090318A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003297927A1 (en) 2002-12-11 2004-06-30 Xenoport, Inc. Prodrugs of fused gaba analogs, pharmaceutical compositions and uses thereof
US20040162351A1 (en) * 2002-12-11 2004-08-19 Gallop Mark A. Orally administered dosage forms of fused GABA analog prodrugs having reduced toxicity
US9066853B2 (en) 2013-01-15 2015-06-30 Warsaw Orthopedic, Inc. Clonidine compounds in a biodegradable fiber

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN2000000224A (es) * 1999-10-20 2001-04-11 Warner Lambert Co Aminoacidos biciclicos como agentes farmaceuticos

Also Published As

Publication number Publication date
WO2002090318A1 (en) 2002-11-14
US20030083520A1 (en) 2003-05-01
GB0110935D0 (en) 2001-06-27
GB2375109A (en) 2002-11-06

Similar Documents

Publication Publication Date Title
ATE370109T1 (de) Festphasenherstellung von 18f-markierten aminosäuren
DK1870417T3 (da) Peptidacceptor-ligeringsmetoder
BR0015622A (pt) Processo de limpeza que utiliza ondas ultra-sÈnicas
DE50208306D1 (de) Verfahren zur Herstellung von nicht-proteinogenen L-Aminosäuren
BR0000897A (pt) Processo para a produção fermentativa de l-aminoácidos usando-se bactéria corineforme
MXPA03004986A (es) Proceso para preparar polimeros de emulsion con alta pureza.
AR021232A1 (es) Procedimiento de preparacion de metionina.
NO20030182L (no) Dermalt påföringssystem for aminolevulinsyre
CY1113871T1 (el) Διαδικασια παρασκευης γκαμπαπεντινης
IT1319234B1 (it) Processo di preparazione di gabapentina.
BR0313795A (pt) Processo para a hidrogenação enantiosseletiva de aminoálcoois
ECSP045215A (es) Metabolitos del ácido (3-{[4-terc-butilbencil)-(piridin-3-sulfonil)amino]metil}fenoxi) acético
NO20040388L (no) Fremgangsmåte for fremstilling av beraprost og salter derav, samt forbindelser som er mellomprodukter i fremgangsmåten
BR0012631A (pt) Processo para a preparação de compostos de amina
AR036623A1 (es) Proceso para la preparacion de repaglinida
BR0212390A (pt) Processo para a preparação de cilastatina
BR0316702A (pt) xprocesso para preparação de (s)-pantoprazol
AR033305A1 (es) Procedimiento para preparar un aminoacido biciclico
BRPI0409095A (pt) processos de sìntese do ácido (2s)-indolina-2-carboxìlico, e aplicação para a sìntese do perindopril
ES2185967T3 (es) Procedimiento para preparar derivados acidos beta-amino-alfa-hidroxi.
BR0001342A (pt) Processo para a produção de l-aminoácidos por meio de fermentação usando bactérias corineformes
BR0315055A (pt) Diamidas de ácido pirimidin-4,6-dicarboxìilco para a inibição seletiva de colagenases
BR0314838A (pt) Sistema de liberação controlada, e, processo para preparar comprimidos de liberação controlada de temozolomida
NO20014885D0 (no) Fremgangsmåte til fremstilling av en amidforbindelse
AU2003287173A1 (en) Process for synthesizing l-y-methylene glutamic acid and analogs