AR023617A1 - Utilizacion del (2s)-1-[(2r,3s)-5-cloro-3-(2-clorofenil)-1-(3,4-dimetoxibencensulfonil)-3-hidroxi-2,3-dihidro-1h-indol-2-carbonil]pirrolidin-2-carboxamidapara la preparacion de medicamentos utiles en el tratamiento del fenomeno de raynaud - Google Patents

Utilizacion del (2s)-1-[(2r,3s)-5-cloro-3-(2-clorofenil)-1-(3,4-dimetoxibencensulfonil)-3-hidroxi-2,3-dihidro-1h-indol-2-carbonil]pirrolidin-2-carboxamidapara la preparacion de medicamentos utiles en el tratamiento del fenomeno de raynaud

Info

Publication number
AR023617A1
AR023617A1 ARP000101990A ARP000101990A AR023617A1 AR 023617 A1 AR023617 A1 AR 023617A1 AR P000101990 A ARP000101990 A AR P000101990A AR P000101990 A ARP000101990 A AR P000101990A AR 023617 A1 AR023617 A1 AR 023617A1
Authority
AR
Argentina
Prior art keywords
dihydro
preparation
treatment
dimetoxibencensulfonil
chlorophenil
Prior art date
Application number
ARP000101990A
Other languages
English (en)
Original Assignee
Addario Ezio Nicola D
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Addario Ezio Nicola D filed Critical Addario Ezio Nicola D
Publication of AR023617A1 publication Critical patent/AR023617A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A61K31/404Indoles, e.g. pindolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)

Abstract

Utilizacion del (2S)-1-[(2R,3S)-5-cloro-3-(2-clorofenil)-1-(3,4-dimetoxibencensulfonil)-3-hidroxi-2,3-dihidro-1H-indol-2-carbonil]pirrolidin-2-carboxamida,de sus solvatos y/o hidratos farmacéuticamente aceptables, para la preparacion de medicamentosutiles en el tratamiento o la prevencion del fenomeno deRaynaud.
ARP000101990A 1999-04-29 2000-04-27 Utilizacion del (2s)-1-[(2r,3s)-5-cloro-3-(2-clorofenil)-1-(3,4-dimetoxibencensulfonil)-3-hidroxi-2,3-dihidro-1h-indol-2-carbonil]pirrolidin-2-carboxamidapara la preparacion de medicamentos utiles en el tratamiento del fenomeno de raynaud AR023617A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9905434A FR2792834A1 (fr) 1999-04-29 1999-04-29 Utilisation du sr 49059, de ses solvats et/ou hydrates pharmaceutiquement acceptables, pour la preparation de medicaments utiles dans le traitement ou la prevention du phenomene de raynaud

Publications (1)

Publication Number Publication Date
AR023617A1 true AR023617A1 (es) 2002-09-04

Family

ID=9545016

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP000101990A AR023617A1 (es) 1999-04-29 2000-04-27 Utilizacion del (2s)-1-[(2r,3s)-5-cloro-3-(2-clorofenil)-1-(3,4-dimetoxibencensulfonil)-3-hidroxi-2,3-dihidro-1h-indol-2-carbonil]pirrolidin-2-carboxamidapara la preparacion de medicamentos utiles en el tratamiento del fenomeno de raynaud

Country Status (4)

Country Link
AR (1) AR023617A1 (es)
AU (1) AU4303500A (es)
FR (1) FR2792834A1 (es)
WO (1) WO2000066117A1 (es)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2679903B1 (fr) * 1991-08-02 1993-12-03 Elf Sanofi Derives de la n-sulfonyl indoline portant une fonction amidique, leur preparation, les compositions pharmaceutiques en contenant.
US5338755A (en) * 1990-07-31 1994-08-16 Elf Sanofi N-sulfonylindoline derivatives, their preparation and the pharmaceutical compositions in which they are present
FR2714378B1 (fr) * 1993-12-24 1996-03-15 Sanofi Sa Dérivés de l'indol-2-one substitués en 3 par un groupe azoté, leur préparation, les compositions pharmaceutiques en contenant.
FR2775598A1 (fr) * 1998-03-06 1999-09-10 Sanofi Sa Compositions pharmaceutiques contenant en association un antagoniste selectif des recepteurs v1a de l'arginine-vasopressine et un antagoniste selectif des recepteur v2 de l'arginine-vasopressine

Also Published As

Publication number Publication date
FR2792834A1 (fr) 2000-11-03
WO2000066117A1 (fr) 2000-11-09
AU4303500A (en) 2000-11-17

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DE60121048D1 (de) PYRAZINOi1'2':1,6öPYRIDOi3,4-BöINDOLDERIVATE