AR023617A1 - Utilizacion del (2s)-1-[(2r,3s)-5-cloro-3-(2-clorofenil)-1-(3,4-dimetoxibencensulfonil)-3-hidroxi-2,3-dihidro-1h-indol-2-carbonil]pirrolidin-2-carboxamidapara la preparacion de medicamentos utiles en el tratamiento del fenomeno de raynaud - Google Patents
Utilizacion del (2s)-1-[(2r,3s)-5-cloro-3-(2-clorofenil)-1-(3,4-dimetoxibencensulfonil)-3-hidroxi-2,3-dihidro-1h-indol-2-carbonil]pirrolidin-2-carboxamidapara la preparacion de medicamentos utiles en el tratamiento del fenomeno de raynaudInfo
- Publication number
- AR023617A1 AR023617A1 ARP000101990A ARP000101990A AR023617A1 AR 023617 A1 AR023617 A1 AR 023617A1 AR P000101990 A ARP000101990 A AR P000101990A AR P000101990 A ARP000101990 A AR P000101990A AR 023617 A1 AR023617 A1 AR 023617A1
- Authority
- AR
- Argentina
- Prior art keywords
- dihydro
- preparation
- treatment
- dimetoxibencensulfonil
- chlorophenil
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
Abstract
Utilizacion del (2S)-1-[(2R,3S)-5-cloro-3-(2-clorofenil)-1-(3,4-dimetoxibencensulfonil)-3-hidroxi-2,3-dihidro-1H-indol-2-carbonil]pirrolidin-2-carboxamida,de sus solvatos y/o hidratos farmacéuticamente aceptables, para la preparacion de medicamentosutiles en el tratamiento o la prevencion del fenomeno deRaynaud.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9905434A FR2792834A1 (fr) | 1999-04-29 | 1999-04-29 | Utilisation du sr 49059, de ses solvats et/ou hydrates pharmaceutiquement acceptables, pour la preparation de medicaments utiles dans le traitement ou la prevention du phenomene de raynaud |
Publications (1)
Publication Number | Publication Date |
---|---|
AR023617A1 true AR023617A1 (es) | 2002-09-04 |
Family
ID=9545016
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP000101990A AR023617A1 (es) | 1999-04-29 | 2000-04-27 | Utilizacion del (2s)-1-[(2r,3s)-5-cloro-3-(2-clorofenil)-1-(3,4-dimetoxibencensulfonil)-3-hidroxi-2,3-dihidro-1h-indol-2-carbonil]pirrolidin-2-carboxamidapara la preparacion de medicamentos utiles en el tratamiento del fenomeno de raynaud |
Country Status (4)
Country | Link |
---|---|
AR (1) | AR023617A1 (es) |
AU (1) | AU4303500A (es) |
FR (1) | FR2792834A1 (es) |
WO (1) | WO2000066117A1 (es) |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2679903B1 (fr) * | 1991-08-02 | 1993-12-03 | Elf Sanofi | Derives de la n-sulfonyl indoline portant une fonction amidique, leur preparation, les compositions pharmaceutiques en contenant. |
US5338755A (en) * | 1990-07-31 | 1994-08-16 | Elf Sanofi | N-sulfonylindoline derivatives, their preparation and the pharmaceutical compositions in which they are present |
FR2714378B1 (fr) * | 1993-12-24 | 1996-03-15 | Sanofi Sa | Dérivés de l'indol-2-one substitués en 3 par un groupe azoté, leur préparation, les compositions pharmaceutiques en contenant. |
FR2775598A1 (fr) * | 1998-03-06 | 1999-09-10 | Sanofi Sa | Compositions pharmaceutiques contenant en association un antagoniste selectif des recepteurs v1a de l'arginine-vasopressine et un antagoniste selectif des recepteur v2 de l'arginine-vasopressine |
-
1999
- 1999-04-29 FR FR9905434A patent/FR2792834A1/fr not_active Withdrawn
-
2000
- 2000-04-25 WO PCT/FR2000/001085 patent/WO2000066117A1/fr active Application Filing
- 2000-04-25 AU AU43035/00A patent/AU4303500A/en not_active Abandoned
- 2000-04-27 AR ARP000101990A patent/AR023617A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
FR2792834A1 (fr) | 2000-11-03 |
WO2000066117A1 (fr) | 2000-11-09 |
AU4303500A (en) | 2000-11-17 |
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