AR013160A1 - POLYMORPHIC FORM OF AN ANTAGONIST RECEIVER OF TACHYQUININE, PHARMACEUTICAL COMPOSITION, USE OF THE SAME FOR THE PREPARATION OF MEDICINES. - Google Patents
POLYMORPHIC FORM OF AN ANTAGONIST RECEIVER OF TACHYQUININE, PHARMACEUTICAL COMPOSITION, USE OF THE SAME FOR THE PREPARATION OF MEDICINES.Info
- Publication number
- AR013160A1 AR013160A1 ARP980103199A AR013160A1 AR 013160 A1 AR013160 A1 AR 013160A1 AR P980103199 A ARP980103199 A AR P980103199A AR 013160 A1 AR013160 A1 AR 013160A1
- Authority
- AR
- Argentina
- Prior art keywords
- phenyl
- preparation
- polymorphic form
- tachyquinine
- antagonist
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Abstract
Forma polimorfica del compuesto 2-(R)-(1-(R)-(3,5-bis(trifluormetil)fenil) etoxi)-3-(S)-(4-fluor)fenil-4-(3-(5-oxo-1H,4H-1,2,4-triazol)metilmorfolina,antagonista receptor de taquiquinina util en el tratamiento o prevencion de los desordenes delsistema nervioso central, enfermedades inflamatorias, doloro migrana, asma y emesis. La misma tiene ventajas con respecto a las otras formas de2-(R)-(1-(R)-(3,5-bis(trifluormetil)fenil)etoxi)-3-(S)-(4-fluor)fenil)-4-(3-(5-oxo-1H,4H-1,2,4-triazo l)metil-morfolina en términos de estabilidad termodinámica y conveniencia para inclusion en formulacionesfarmacéuticas, composicionfarmacéutica, uso de dicha forma para preparar medicamentos, procedimientos para su preparacion y prod uctos producidos pordichos procedimientos.Polymorphic form of compound 2- (R) - (1- (R) - (3,5-bis (trifluormethyl) phenyl) ethoxy) -3- (S) - (4-fluor) phenyl-4- (3- ( 5-oxo-1H, 4H-1,2,4-triazole) methylmorpholine, a tachykinin receptor antagonist useful in the treatment or prevention of central nervous system disorders, inflammatory diseases, migraine pain, asthma, and emesis. relative to the other forms of 2- (R) - (1- (R) - (3,5-bis (trifluormethyl) phenyl) ethoxy) -3- (S) - (4-fluor) phenyl) -4- (3 - (5-oxo-1H, 4H-1,2,4-triazo l) methyl-morpholine in terms of thermodynamic stability and suitability for inclusion in pharmaceutical, compositional-pharmaceutical formulations, use of said form to prepare drugs, procedures for their preparation and prod ucts produced by said procedures.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US5160097P | 1997-07-02 | 1997-07-02 | |
GBGB9800216.5A GB9800216D0 (en) | 1998-01-07 | 1998-01-07 | Polymorphic form of a tachykinin receptor antagonist |
Publications (1)
Publication Number | Publication Date |
---|---|
AR013160A1 true AR013160A1 (en) | 2000-12-13 |
Family
ID=10824888
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP980103199 AR013160A1 (en) | 1997-07-02 | 1998-07-01 | POLYMORPHIC FORM OF AN ANTAGONIST RECEIVER OF TACHYQUININE, PHARMACEUTICAL COMPOSITION, USE OF THE SAME FOR THE PREPARATION OF MEDICINES. |
Country Status (6)
Country | Link |
---|---|
AR (1) | AR013160A1 (en) |
CO (1) | CO4940431A1 (en) |
GB (1) | GB9800216D0 (en) |
MY (1) | MY126509A (en) |
RS (1) | RS49980B (en) |
UA (1) | UA57089C2 (en) |
-
1998
- 1998-01-07 GB GBGB9800216.5A patent/GB9800216D0/en not_active Ceased
- 1998-01-07 UA UA99127240A patent/UA57089C2/en unknown
- 1998-07-01 AR ARP980103199 patent/AR013160A1/en active IP Right Grant
- 1998-07-01 RS YUP-721/99A patent/RS49980B/en unknown
- 1998-07-01 MY MYPI98003007A patent/MY126509A/en unknown
- 1998-07-03 CO CO98037640A patent/CO4940431A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
CO4940431A1 (en) | 2000-07-24 |
RS49980B (en) | 2008-09-29 |
UA57089C2 (en) | 2003-06-16 |
GB9800216D0 (en) | 1998-03-04 |
MY126509A (en) | 2006-10-31 |
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