AR010307A1 - Derivado de la eritromicina a, composicion farmaceutica y preparacion antibacteriana que lo contienen. - Google Patents

Derivado de la eritromicina a, composicion farmaceutica y preparacion antibacteriana que lo contienen.

Info

Publication number
AR010307A1
AR010307A1 ARP970105505A ARP970105505A AR010307A1 AR 010307 A1 AR010307 A1 AR 010307A1 AR P970105505 A ARP970105505 A AR P970105505A AR P970105505 A ARP970105505 A AR P970105505A AR 010307 A1 AR010307 A1 AR 010307A1
Authority
AR
Argentina
Prior art keywords
group
erythromycin
derived
pharmaceutical composition
preparation containing
Prior art date
Application number
ARP970105505A
Other languages
English (en)
Original Assignee
Taieb Alain
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taieb Alain filed Critical Taieb Alain
Publication of AR010307A1 publication Critical patent/AR010307A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

Un derivado de eritromicina A representado por la formula (1) donde n es un numero entero de 1 a 4, R1 es un grupo representado por la formula II, un gruporepresentado por la formula III, un piridilacetilo, un grupo cicloalquilmetilo o un grupo 1,2-bi(etoxicarbonil)vinilo, R2 es el mismo grupo R1, un átomo dehidrogeno, un alquilo, alcanoílo, R1 y R2 juntos forman un grupo de la formula =CH-R14, o R1 y R2 forman junto al nitrogeno al que están unidos un grupo IV...sigue el resumen.
ARP970105505A 1996-11-27 1997-11-25 Derivado de la eritromicina a, composicion farmaceutica y preparacion antibacteriana que lo contienen. AR010307A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP31580596 1996-11-27

Publications (1)

Publication Number Publication Date
AR010307A1 true AR010307A1 (es) 2000-06-07

Family

ID=18069775

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP970105505A AR010307A1 (es) 1996-11-27 1997-11-25 Derivado de la eritromicina a, composicion farmaceutica y preparacion antibacteriana que lo contienen.

Country Status (14)

Country Link
US (1) US6191118B1 (es)
EP (1) EP0945459A4 (es)
JP (1) JP4077882B2 (es)
KR (1) KR20000069138A (es)
CN (1) CN1238777A (es)
AR (1) AR010307A1 (es)
AU (1) AU720921B2 (es)
BR (1) BR9713302A (es)
CA (1) CA2272620A1 (es)
CZ (1) CZ180799A3 (es)
HU (1) HUP0000198A3 (es)
IL (1) IL129946A0 (es)
WO (1) WO1998023628A1 (es)
ZA (1) ZA9710648B (es)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2004514643A (ja) * 1997-10-29 2004-05-20 大正製薬株式会社 エリスロマイシンa誘導体
ATE344269T1 (de) 1998-12-10 2006-11-15 Pfizer Prod Inc Carbamat und carbazat ketolid antibiotika
WO2000071557A1 (en) 1999-05-24 2000-11-30 Pfizer Products Inc. 13-methyl-erythromycin derivatives
EP1146051A3 (en) * 2000-04-10 2001-10-31 Pfizer Products Inc. Erythromycin A derivatives
US20020115621A1 (en) * 2000-08-07 2002-08-22 Wei-Gu Su Macrolide antibiotics
JP2002173498A (ja) * 2000-09-27 2002-06-21 Hokuriku Seiyaku Co Ltd エリスロマイシン誘導体
US6472372B1 (en) * 2000-12-06 2002-10-29 Ortho-Mcneil Pharmaceuticals, Inc. 6-O-Carbamoyl ketolide antibacterials
WO2003004509A2 (en) * 2001-07-03 2003-01-16 Chiron Corporation C12 modified erythromycin macrolides and ketolides having antibacterial activity
US6825172B2 (en) 2002-05-31 2004-11-30 Janssen Pharmaceutica, Nv 3-descladinosyl-6-O-carbamoyl and 6-O-carbonoyl macrolide antibacterial agents
EP1618119A2 (en) 2003-04-25 2006-01-25 Chiron Corporation Pyridyl substituted ketolide antibiotics
US7163924B2 (en) 2003-04-25 2007-01-16 Chiron Corporation Ketolide derivatives
AU2003263482A1 (en) * 2003-09-25 2005-04-14 Ranbaxy Laboratories Limited 3'-n-substituted-3-o-substituted erythronolide a derivatives
DE10357532A1 (de) * 2003-12-08 2005-07-07 Basf Ag Verwendung von Polymerisaten auf Basis von N-Vinylcaprolactam für die Haarkosmetik
US20080207536A1 (en) * 2004-07-28 2008-08-28 Ranbaxy Laboratories Limited Antibacterial Agents
BRPI0514381A (pt) * 2004-07-30 2008-06-10 Palumed Sa compostos hìbridos de aminoquinolina-antibiótico, composições farmacêuticas, método de preparação e uso destes
FR2874922A1 (fr) * 2004-07-30 2006-03-10 Palumed Sa Molecules hybrides qa ou q est une aminoquinoleine et a est un residu antibiotique, leur synthese et leurs utilisations en tant qu'agent antibacterien
FR2873695A1 (fr) * 2004-07-30 2006-02-03 Palumed Sa Molecules hybrides qa ou q est une aminoquinoleine et a est un antibiotique ou un inhibiteur de resistance), leur synthese et leurs utilisations en tant qu'agent antibacterien
EP1836211B1 (en) * 2004-12-21 2010-03-03 Pfizer Products Inc. Macrolides
CN100577678C (zh) * 2006-06-19 2010-01-06 中国医学科学院药物研究所 大环内酯类药物双侧链红霉素a衍生物、合成方法和用途
US8293715B2 (en) * 2007-08-06 2012-10-23 Taisho Pharmaceutical Co., Ltd. 10a-Azalide compound crosslinked at 10a- and 12-positions
WO2009139181A1 (ja) 2008-05-15 2009-11-19 大正製薬株式会社 4員環構造を有する10a-アザライド化合物
US10260000B2 (en) * 2012-01-23 2019-04-16 Macdermid Acumen, Inc. Etching of plastic using acidic solutions containing trivalent manganese

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4331803A (en) 1980-06-04 1982-05-25 Taisho Pharmaceutical Co., Ltd. Novel erythromycin compounds
US4742049A (en) 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
US5523399A (en) 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives
WO1993021199A1 (en) 1992-04-22 1993-10-28 Taisho Pharmaceutical Co., Ltd. 5-o-desosaminylerythronolide a derivative

Also Published As

Publication number Publication date
HUP0000198A2 (hu) 2000-08-28
KR20000069138A (ko) 2000-11-25
EP0945459A1 (en) 1999-09-29
US6191118B1 (en) 2001-02-20
AU4473097A (en) 1998-06-22
CA2272620A1 (en) 1998-06-04
AU720921B2 (en) 2000-06-15
ZA9710648B (en) 1998-06-23
CZ180799A3 (cs) 1999-09-15
IL129946A0 (en) 2000-02-29
BR9713302A (pt) 2000-03-21
EP0945459A4 (en) 2000-02-09
HUP0000198A3 (en) 2000-09-28
WO1998023628A1 (fr) 1998-06-04
JP4077882B2 (ja) 2008-04-23
CN1238777A (zh) 1999-12-15

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