AR008395A1 - Compuesto derivado de pirimidina, composicion farmaceutica que lo comprende, procedimiento para prepararlo, y compuesto intermediario util parallevar a cabo dicho procedimiento. - Google Patents

Compuesto derivado de pirimidina, composicion farmaceutica que lo comprende, procedimiento para prepararlo, y compuesto intermediario util parallevar a cabo dicho procedimiento.

Info

Publication number
AR008395A1
AR008395A1 ARP970102801A ARP970102801A AR008395A1 AR 008395 A1 AR008395 A1 AR 008395A1 AR P970102801 A ARP970102801 A AR P970102801A AR P970102801 A ARP970102801 A AR P970102801A AR 008395 A1 AR008395 A1 AR 008395A1
Authority
AR
Argentina
Prior art keywords
procedure
pharmaceutical composition
pirimidine
understands
prepare
Prior art date
Application number
ARP970102801A
Other languages
English (en)
Original Assignee
Astra Pharma Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9614360.7A external-priority patent/GB9614360D0/en
Priority claimed from GBGB9626884.2A external-priority patent/GB9626884D0/en
Application filed by Astra Pharma Prod filed Critical Astra Pharma Prod
Publication of AR008395A1 publication Critical patent/AR008395A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D491/00Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Un compuesto derivado de pirimidina que tiene la formula I donde R, Ar1, W, X, Y y Z son como se definen en la memoria descriptiva. Además, se dan aconocer una composicion farmacéutica que comprende a dicho compuesto, un procedimiento para prepararlo, y un compuesto intermediario util para llevar acabo dicho procedimiento.
ARP970102801A 1996-07-09 1997-06-25 Compuesto derivado de pirimidina, composicion farmaceutica que lo comprende, procedimiento para prepararlo, y compuesto intermediario util parallevar a cabo dicho procedimiento. AR008395A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9614360.7A GB9614360D0 (en) 1996-07-09 1996-07-09 Compounds
GBGB9626884.2A GB9626884D0 (en) 1996-12-24 1996-12-24 Compounds

Publications (1)

Publication Number Publication Date
AR008395A1 true AR008395A1 (es) 2000-01-19

Family

ID=26309668

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP970102801A AR008395A1 (es) 1996-07-09 1997-06-25 Compuesto derivado de pirimidina, composicion farmaceutica que lo comprende, procedimiento para prepararlo, y compuesto intermediario util parallevar a cabo dicho procedimiento.

Country Status (16)

Country Link
EP (1) EP0915879A1 (es)
JP (1) JP2000516206A (es)
KR (1) KR20000023644A (es)
AR (1) AR008395A1 (es)
AU (1) AU708882B2 (es)
BR (1) BR9710215A (es)
CA (1) CA2260057A1 (es)
CZ (1) CZ3699A3 (es)
EE (1) EE9900012A (es)
ID (1) ID18889A (es)
IL (1) IL127690A0 (es)
IS (1) IS4932A (es)
NO (1) NO990072D0 (es)
PL (1) PL331090A1 (es)
TR (1) TR199900013T2 (es)
WO (1) WO1998001449A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003015776A1 (en) 2001-08-13 2003-02-27 Janssen Pharmaceutica N.V. 2,4,5-trisubstituted thiazolyl derivatives and their antiinflammatory activity
EP2504871B1 (en) 2009-11-24 2017-03-22 Novaled GmbH Organic electronic device comprising an organic semiconducting material
WO2014084612A1 (ko) * 2012-11-30 2014-06-05 주식회사 엘지화학 신규한 화합물 및 이를 이용한 유기 전자 소자
KR102153040B1 (ko) 2013-11-28 2020-09-07 삼성전자주식회사 축합환 화합물 및 이를 포함한 유기 발광 소자
CN108484606B (zh) * 2018-03-16 2020-03-06 江南大学 一种嘧啶并[4,5-f]喹唑啉类化合物及其应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1670577A1 (de) * 1967-10-05 1971-05-19 Akad Wissenschaften Ddr Verfahren zur Herstellung von 5-oxo-5.6.7.8-tetrahydro-chinazelinen
US4272535A (en) * 1978-07-31 1981-06-09 Schering Corporation 2,4-[1H,3H,5H]-(1)-Benzopyrano-[2,3-d]-pyrimidinediones and their use as anti-allergy agents
US4762843A (en) * 1986-09-15 1988-08-09 Warner-Lambert Company Hetero [f] fused carbocyclic pyridines as dopaminergic agents
US5597823A (en) * 1995-01-27 1997-01-28 Abbott Laboratories Tricyclic substituted hexahydrobenz [e]isoindole alpha-1 adrenergic antagonists

Also Published As

Publication number Publication date
JP2000516206A (ja) 2000-12-05
CA2260057A1 (en) 1998-01-15
PL331090A1 (en) 1999-06-21
EE9900012A (et) 1999-06-15
IL127690A0 (en) 1999-10-28
ID18889A (id) 1998-05-20
WO1998001449A1 (en) 1998-01-15
EP0915879A1 (en) 1999-05-19
NO990072D0 (no) 1999-01-08
AU3711697A (en) 1998-02-02
TR199900013T2 (xx) 1999-04-21
KR20000023644A (ko) 2000-04-25
IS4932A (is) 1998-12-23
CZ3699A3 (cs) 1999-06-16
AU708882B2 (en) 1999-08-12
BR9710215A (pt) 1999-08-10

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