DK1644350T3 - Sullfamatbenzothiophenderivater som steroidsulfataseinhibitorer - Google Patents
Sullfamatbenzothiophenderivater som steroidsulfataseinhibitorerInfo
- Publication number
- DK1644350T3 DK1644350T3 DK03816954T DK03816954T DK1644350T3 DK 1644350 T3 DK1644350 T3 DK 1644350T3 DK 03816954 T DK03816954 T DK 03816954T DK 03816954 T DK03816954 T DK 03816954T DK 1644350 T3 DK1644350 T3 DK 1644350T3
- Authority
- DK
- Denmark
- Prior art keywords
- steroid sulfatase
- benzothiophene derivatives
- sulfatase inhibitors
- sulfamate benzothiophene
- sulfamate
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/34—Gestagens
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/76—Dibenzothiophenes
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Immunology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Materials For Photolithography (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/EP2003/008811 WO2004101545A1 (en) | 2003-05-16 | 2003-05-16 | Sulfamate benzothiophene derivatives as steroid sulfatase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1644350T3 true DK1644350T3 (da) | 2009-11-23 |
Family
ID=33442621
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK03816954T DK1644350T3 (da) | 2003-05-16 | 2003-05-16 | Sullfamatbenzothiophenderivater som steroidsulfataseinhibitorer |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US7476691B2 (da) |
| EP (1) | EP1644350B1 (da) |
| JP (1) | JP4757497B2 (da) |
| CN (2) | CN100491370C (da) |
| AP (1) | AP2066A (da) |
| AT (1) | ATE435221T1 (da) |
| AU (1) | AU2003260390B2 (da) |
| BR (1) | BR0318295A (da) |
| CA (1) | CA2525684C (da) |
| CY (1) | CY1109371T1 (da) |
| DE (1) | DE60328233D1 (da) |
| DK (1) | DK1644350T3 (da) |
| ES (1) | ES2329241T3 (da) |
| HK (1) | HK1087115A1 (da) |
| IL (1) | IL171763A (da) |
| MX (1) | MXPA05012300A (da) |
| NO (1) | NO20055749L (da) |
| NZ (1) | NZ544013A (da) |
| PT (1) | PT1644350E (da) |
| SI (1) | SI1644350T1 (da) |
| TN (1) | TNSN05291A1 (da) |
| WO (1) | WO2004101545A1 (da) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| OA13336A (en) | 2003-12-15 | 2006-04-13 | Theramex | 1-N-phenyl-amino-1H-imidazole derivatives and pharmaceutical compositions containing them. |
| GB0511190D0 (en) * | 2005-06-01 | 2005-07-06 | Sterix Ltd | Use |
| AU2007271486A1 (en) * | 2006-07-05 | 2008-01-10 | Merck Patent Gmbh | Sulfamate benzothiophene derivatives |
| WO2008067892A1 (de) * | 2006-12-04 | 2008-06-12 | Merck Patent Gmbh | Sulfamat-benzothiophen-derivate |
| BRPI0817045A2 (pt) * | 2007-09-17 | 2015-03-24 | Preglem Sa | Tratamento de condições estrogênio-dependentes em mulheres pré-menopáusicas |
| JP2011157371A (ja) * | 2011-03-17 | 2011-08-18 | Lab Theramex | ステロイドスルファターゼ阻害剤としてのベンゾチオフェンスルファミン酸塩誘導体 |
| CN115805103B (zh) * | 2021-09-14 | 2024-04-09 | 万华化学集团股份有限公司 | 一种失活钛硅分子筛的再生方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9118478D0 (en) * | 1991-08-29 | 1991-10-16 | Imperial College | Steroid sulphatase inhibitors |
| US6248780B1 (en) * | 1998-10-01 | 2001-06-19 | Duquesne University Of The Holy Ghost | Compounds for the treatment of estrogen-dependent illnesses and methods for making and using the same |
-
2003
- 2003-05-16 ES ES03816954T patent/ES2329241T3/es not_active Expired - Lifetime
- 2003-05-16 BR BRPI0318295-9A patent/BR0318295A/pt not_active IP Right Cessation
- 2003-05-16 US US10/555,780 patent/US7476691B2/en not_active Expired - Fee Related
- 2003-05-16 NZ NZ544013A patent/NZ544013A/en not_active IP Right Cessation
- 2003-05-16 PT PT03816954T patent/PT1644350E/pt unknown
- 2003-05-16 SI SI200331665T patent/SI1644350T1/sl unknown
- 2003-05-16 AT AT03816954T patent/ATE435221T1/de active
- 2003-05-16 DK DK03816954T patent/DK1644350T3/da active
- 2003-05-16 CN CNB038264706A patent/CN100491370C/zh not_active Expired - Fee Related
- 2003-05-16 DE DE60328233T patent/DE60328233D1/de not_active Expired - Lifetime
- 2003-05-16 JP JP2004571781A patent/JP4757497B2/ja not_active Expired - Fee Related
- 2003-05-16 CN CNA2009100023017A patent/CN101508691A/zh active Pending
- 2003-05-16 EP EP03816954A patent/EP1644350B1/en not_active Expired - Lifetime
- 2003-05-16 AP AP2005003468A patent/AP2066A/en active
- 2003-05-16 CA CA2525684A patent/CA2525684C/en not_active Expired - Fee Related
- 2003-05-16 AU AU2003260390A patent/AU2003260390B2/en not_active Ceased
- 2003-05-16 MX MXPA05012300A patent/MXPA05012300A/es active IP Right Grant
- 2003-05-16 WO PCT/EP2003/008811 patent/WO2004101545A1/en active Application Filing
-
2005
- 2005-11-03 IL IL171763A patent/IL171763A/en not_active IP Right Cessation
- 2005-11-15 TN TNP2005000291A patent/TNSN05291A1/en unknown
- 2005-12-05 NO NO20055749A patent/NO20055749L/no not_active Application Discontinuation
-
2006
- 2006-06-29 HK HK06107352.1A patent/HK1087115A1/xx not_active IP Right Cessation
-
2009
- 2009-09-09 CY CY20091100937T patent/CY1109371T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CY1109371T1 (el) | 2014-07-02 |
| AU2003260390B2 (en) | 2010-05-20 |
| CN100491370C (zh) | 2009-05-27 |
| CN101508691A (zh) | 2009-08-19 |
| ATE435221T1 (de) | 2009-07-15 |
| HK1087115A1 (en) | 2006-10-06 |
| WO2004101545A1 (en) | 2004-11-25 |
| EP1644350B1 (en) | 2009-07-01 |
| CA2525684A1 (en) | 2004-11-25 |
| NO20055749L (no) | 2005-12-14 |
| SI1644350T1 (sl) | 2009-12-31 |
| DE60328233D1 (de) | 2009-08-13 |
| CN1771243A (zh) | 2006-05-10 |
| TNSN05291A1 (en) | 2007-07-10 |
| AP2005003468A0 (en) | 2005-12-31 |
| JP4757497B2 (ja) | 2011-08-24 |
| NO20055749D0 (no) | 2005-12-05 |
| US7476691B2 (en) | 2009-01-13 |
| BR0318295A (pt) | 2006-07-11 |
| IL171763A (en) | 2013-09-30 |
| AU2003260390A1 (en) | 2004-12-03 |
| ES2329241T3 (es) | 2009-11-24 |
| NZ544013A (en) | 2009-04-30 |
| CA2525684C (en) | 2015-01-06 |
| AP2066A (en) | 2009-11-27 |
| MXPA05012300A (es) | 2006-01-30 |
| US20070021492A1 (en) | 2007-01-25 |
| EP1644350A1 (en) | 2006-04-12 |
| JP2006525947A (ja) | 2006-11-16 |
| PT1644350E (pt) | 2009-09-02 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK1789041T3 (da) | Aryl-pyridinderivater som 11-beta-HSD1-inhibitorer | |
| DK1797042T3 (da) | Indozolonderivater som 11B-HSD1-inhibitorer | |
| DK1585749T3 (da) | Diazepinoindol-derivater som kinaseinhibitorer | |
| DK2094263T3 (da) | 2-adamantyl-butyramidderivater som selektive 11 beta-hsd1-inhibitorer | |
| DK1828167T3 (da) | Acrylamidderivater som antibiotiske midler | |
| NO20050665L (no) | Pyrrolidonderivater som MAOE inhibitoere | |
| NO20050426L (no) | Arylkarbonylderivater som terapeutiske midler | |
| DK1960352T3 (da) | 2-adamantylurinstof-derivater som selektive 11beta-hsd1 inhibitorer | |
| NO20034307L (no) | Cyklopropylindol-derivater som selektive serotonin- gjenopptaksinhibitorer | |
| DK1863787T3 (da) | Hydrogeneret benzo[c]thiophenderivater som immunmodulatorer | |
| DK1740569T3 (da) | Imidazol-derivater som TAFla-inhibitorer | |
| DK1848430T3 (da) | Nye benzylamin-derivativer som cetp-inhibitors | |
| DK1959951T3 (da) | Heteroaryl-substituerede piperidinderivater som L-CPT1-inhibitorer | |
| DK1663232T3 (da) | Benzimidazolderivater som human chymase-inhibitorer | |
| NO20044654L (no) | Piperidinoylpiperidiner som 5-HTIF-agonister | |
| DK1763517T3 (da) | Pyrimidinderivater som 11beta-HSD1-inhibitorer | |
| IS2656B (is) | Nýjar besímídasólafleiður | |
| DK1492785T3 (da) | 2-hydroxy-3-heteroarylindol-derivater som GSK3-inhibitorer | |
| ATE394399T1 (de) | Tetrahydropyridoindolderivate | |
| ATE383361T1 (de) | Pyrrazolopyrimidinderivate | |
| DK2078001T3 (da) | Diazepan-acetamidderivater som selektive 11-HSD1-inhibitorer | |
| ATE396724T1 (de) | 1h-thieno 2,3-c-pyrazol-derivate als kinase-i- hemmer | |
| DK1709018T3 (da) | Acylaminothiazolderivater og anvendelse deraf som beta-amyloid-hæmmere | |
| DK1660090T3 (da) | Quinazolin-analoger som receptor-tyrosinkinase-inhibitorer | |
| NO20030842L (no) | Fenoksybenzylaminderivater som selektive serotonin- gjenopptaksinhibitorer |