ZA958995B - Derivatives of acid pyrazolones and pyrazoles their preparation process the intermediates obtained their use as medicaments and the pharmaceutical compositions containing them - Google Patents

Derivatives of acid pyrazolones and pyrazoles their preparation process the intermediates obtained their use as medicaments and the pharmaceutical compositions containing them

Info

Publication number
ZA958995B
ZA958995B ZA958995A ZA958995A ZA958995B ZA 958995 B ZA958995 B ZA 958995B ZA 958995 A ZA958995 A ZA 958995A ZA 958995 A ZA958995 A ZA 958995A ZA 958995 B ZA958995 B ZA 958995B
Authority
ZA
South Africa
Prior art keywords
pyrazolones
pyrazoles
medicaments
derivatives
acid
Prior art date
Application number
ZA958995A
Inventor
Michel Fortin
Jidong Zhang
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of ZA958995B publication Critical patent/ZA958995B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ZA958995A 1994-10-24 1995-10-24 Derivatives of acid pyrazolones and pyrazoles their preparation process the intermediates obtained their use as medicaments and the pharmaceutical compositions containing them ZA958995B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9412676A FR2725988B1 (en) 1994-10-24 1994-10-24 NEW DERIVATIVES OF PYRAZOLONES AND ACID PYRAZOLES, THEIR PROCESS OF PREPARATION, THE NEW INTERMEDIARIES OBTAINED, THEIR APPLICATION AS MEDICINAL PRODUCTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Publications (1)

Publication Number Publication Date
ZA958995B true ZA958995B (en) 1996-10-24

Family

ID=9468134

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA958995A ZA958995B (en) 1994-10-24 1995-10-24 Derivatives of acid pyrazolones and pyrazoles their preparation process the intermediates obtained their use as medicaments and the pharmaceutical compositions containing them

Country Status (5)

Country Link
AU (1) AU3808595A (en)
FR (1) FR2725988B1 (en)
IL (1) IL115653A0 (en)
WO (1) WO1996012706A1 (en)
ZA (1) ZA958995B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2740135B1 (en) * 1995-10-20 1997-12-19 Roussel Uclaf NOVEL ACID PYRAZOLES DERIVATIVES, THEIR PREPARATION PROCESS, THEIR USE AS MEDICAMENTS, THEIR NEW USE AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
DE19645313A1 (en) 1996-11-04 1998-05-07 Basf Ag Substituted 3-benzylpyrazoles
DE19653024A1 (en) * 1996-12-19 1998-06-25 Merck Patent Gmbh Endothelin receptor antagonists
WO2005090313A1 (en) 2004-03-18 2005-09-29 Pfizer Limited N-(1-arylpyrazol-4l)sulfonamides and their use as parasiticides
DE102008020113A1 (en) 2008-04-23 2009-10-29 Bayer Schering Pharma Aktiengesellschaft Substituted dihydropyrazolones and their use
DE102005019712A1 (en) 2005-04-28 2006-11-09 Bayer Healthcare Ag Dipyridyl-dihydropyrazolone and its use
NL2000351C2 (en) 2005-12-22 2007-09-11 Pfizer Prod Inc Estrogen modulators.
DE102006050513A1 (en) 2006-10-26 2008-04-30 Bayer Healthcare Ag New substituted dihydropyrazolone derivatives are hypoxia-inducible transcription factor-prolyl-4-hydroxylase inhibitors useful to treat/prevent e.g. cardiovascular diseases, heart-circulation diseases, heart failure and anemia
DE102006050515A1 (en) 2006-10-26 2008-04-30 Bayer Healthcare Ag New substituted dipyridiyl-dihydropyrazolone derivatives are hypoxia-inducible transcription factor-prolyl-4-hydroxylase inhibitors useful to treat/prevent e.g. cardiovascular diseases, heart-circulation diseases, heart failure and anemia
DE102006050516A1 (en) 2006-10-26 2008-04-30 Bayer Healthcare Ag New pyrazol-3-one compounds are hypoxia-inducible transcription factor-prolyl-4-hydroxylase inhibitors useful e.g. to treat and/or prophylaxis heart-circulation diseases, heart failure, anemia, chronic kidney diseases and renal failure
DE102007044032A1 (en) 2007-09-14 2009-03-19 Bayer Healthcare Ag New substituted heteroaryl compounds are hypoxia-inducible factor prolyl-4-hydroxylase inhibitors useful to treat and/or prevent e.g. circulatory heart diseases, heart failure, anemia, chronic kidney diseases and renal failure
DE102007048447A1 (en) 2007-10-10 2009-04-16 Bayer Healthcare Ag New substituted dihydropyrazole-3-thione compounds are hypoxia inducible factor-prolyl-4-hydroxylase inhibitor, useful for preparing medicament to treat and/or prevent e.g. cardiovascular diseases, wound healing and anemia
DE102010044131A1 (en) 2010-11-18 2012-05-24 Bayer Schering Pharma Aktiengesellschaft Substituted sodium 1H-pyrazole-5-olate
AU2015217450A1 (en) 2014-02-14 2016-08-11 Inception 2, Inc. Pyrazolone compounds and uses thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2672891B1 (en) * 1991-02-20 1994-02-18 Synthelabo DERIVATIVES OF 3-PYRAZOLONES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION.
NZ247440A (en) * 1992-05-06 1995-04-27 Squibb & Sons Inc Phenyl sulphonamide derivatives, preparation and pharmaceutical compositions thereof
WO1994002474A1 (en) * 1992-07-17 1994-02-03 Smithkline Beecham Corporation Endothelin receptor antagonists

Also Published As

Publication number Publication date
AU3808595A (en) 1996-05-15
WO1996012706A1 (en) 1996-05-02
IL115653A0 (en) 1996-01-19
FR2725988B1 (en) 1997-01-24
FR2725988A1 (en) 1996-04-26

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