ZA200908631B - N-Oxides of venlafaxine and O-Desmethylvenlafaxine as prodrugs - Google Patents

N-Oxides of venlafaxine and O-Desmethylvenlafaxine as prodrugs

Info

Publication number
ZA200908631B
ZA200908631B ZA200908631A ZA200908631A ZA200908631B ZA 200908631 B ZA200908631 B ZA 200908631B ZA 200908631 A ZA200908631 A ZA 200908631A ZA 200908631 A ZA200908631 A ZA 200908631A ZA 200908631 B ZA200908631 B ZA 200908631B
Authority
ZA
South Africa
Prior art keywords
desmethylvenlafaxine
venlafaxine
prodrugs
oxides
Prior art date
Application number
ZA200908631A
Inventor
Lechoslaw A Turski
Axel Stoit
Cornelis G Kruse
Sander Vader
Martinus Th M Tulp
Original Assignee
Solvay Pharm Bv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Solvay Pharm Bv filed Critical Solvay Pharm Bv
Publication of ZA200908631B publication Critical patent/ZA200908631B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C291/00Compounds containing carbon and nitrogen and having functional groups not covered by groups C07C201/00 - C07C281/00
    • C07C291/02Compounds containing carbon and nitrogen and having functional groups not covered by groups C07C201/00 - C07C281/00 containing nitrogen-oxide bonds
    • C07C291/04Compounds containing carbon and nitrogen and having functional groups not covered by groups C07C201/00 - C07C281/00 containing nitrogen-oxide bonds containing amino-oxide bonds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/12Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14The ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ZA200908631A 2007-06-26 2009-12-04 N-Oxides of venlafaxine and O-Desmethylvenlafaxine as prodrugs ZA200908631B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP07111028 2007-06-26

Publications (1)

Publication Number Publication Date
ZA200908631B true ZA200908631B (en) 2010-08-25

Family

ID=38626380

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200908631A ZA200908631B (en) 2007-06-26 2009-12-04 N-Oxides of venlafaxine and O-Desmethylvenlafaxine as prodrugs

Country Status (6)

Country Link
JP (1) JP2010531326A (en)
CN (1) CN101939293A (en)
AR (1) AR068978A1 (en)
BR (1) BRPI0813658A2 (en)
TW (1) TW200916092A (en)
ZA (1) ZA200908631B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI490189B (en) * 2011-05-16 2015-07-01 江蘇豪森醫藥集團有限公司 O-demethylation of venlafaxine hydrochloride hydrate and their preparation method
CN103570669B (en) * 2013-10-31 2015-07-22 吉林大学 Brain-targeted O-desmethylvenlafaxine phenolic ester prodrug and preparation method and applications thereof
CN111072505A (en) * 2019-12-27 2020-04-28 合肥华方医药科技有限公司 Preparation method of venlafaxine impurity

Also Published As

Publication number Publication date
CN101939293A (en) 2011-01-05
TW200916092A (en) 2009-04-16
AR068978A1 (en) 2009-12-23
JP2010531326A (en) 2010-09-24
BRPI0813658A2 (en) 2016-10-18

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