ZA200810680B - Treating psychological conditions using muscarinic receptor m1 antagonists - Google Patents
Treating psychological conditions using muscarinic receptor m1 antagonistsInfo
- Publication number
- ZA200810680B ZA200810680B ZA2008/10680A ZA200810680A ZA200810680B ZA 200810680 B ZA200810680 B ZA 200810680B ZA 2008/10680 A ZA2008/10680 A ZA 2008/10680A ZA 200810680 A ZA200810680 A ZA 200810680A ZA 200810680 B ZA200810680 B ZA 200810680B
- Authority
- ZA
- South Africa
- Prior art keywords
- antagonists
- muscarinic receptor
- psychological conditions
- treating psychological
- treating
- Prior art date
Links
- 102000007207 Muscarinic M1 Receptor Human genes 0.000 title 1
- 108010008406 Muscarinic M1 Receptor Proteins 0.000 title 1
- 239000005557 antagonist Substances 0.000 title 1
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Emergency Medicine (AREA)
- Pain & Pain Management (AREA)
- Psychology (AREA)
- Reproductive Health (AREA)
- Nutrition Science (AREA)
- Hospice & Palliative Care (AREA)
- Rheumatology (AREA)
- Child & Adolescent Psychology (AREA)
- Anesthesiology (AREA)
- Gynecology & Obstetrics (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US80506606P | 2006-06-16 | 2006-06-16 | |
| US82922506P | 2006-10-12 | 2006-10-12 | |
| US11/763,145 US7893053B2 (en) | 2006-06-16 | 2007-06-14 | Treating psychological conditions using muscarinic receptor M1 antagonists |
| PCT/US2007/071356 WO2007147123A1 (en) | 2006-06-16 | 2007-06-15 | Treating psychological conditions using muscarinic receptor m1 antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200810680B true ZA200810680B (en) | 2011-04-28 |
Family
ID=38832129
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA2008/10680A ZA200810680B (en) | 2006-06-16 | 2008-12-18 | Treating psychological conditions using muscarinic receptor m1 antagonists |
| ZA2010/08538A ZA201008538B (en) | 2006-06-16 | 2010-11-29 | Treating psychological conditions using muscarinic receptor m1 antagonists |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA2010/08538A ZA201008538B (en) | 2006-06-16 | 2010-11-29 | Treating psychological conditions using muscarinic receptor m1 antagonists |
Country Status (15)
| Country | Link |
|---|---|
| US (2) | US7893053B2 (enExample) |
| EP (2) | EP2032127B1 (enExample) |
| JP (2) | JP4874397B2 (enExample) |
| KR (1) | KR101408650B1 (enExample) |
| CN (1) | CN103041389A (enExample) |
| AU (1) | AU2007260631B2 (enExample) |
| BR (1) | BRPI0713733A2 (enExample) |
| CA (1) | CA2655131C (enExample) |
| IL (1) | IL195857A (enExample) |
| MX (1) | MX2008015887A (enExample) |
| NZ (1) | NZ573570A (enExample) |
| RU (1) | RU2012152922A (enExample) |
| SG (1) | SG172712A1 (enExample) |
| WO (1) | WO2007147123A1 (enExample) |
| ZA (2) | ZA200810680B (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7893053B2 (en) * | 2006-06-16 | 2011-02-22 | Theracos, Inc. | Treating psychological conditions using muscarinic receptor M1 antagonists |
| US8748419B2 (en) | 2006-06-16 | 2014-06-10 | Theracos, Inc. | Treating obesity with muscarinic receptor M1 antagonists |
| WO2010006249A1 (en) * | 2008-07-10 | 2010-01-14 | Tyrx Pharma, Inc. | Sustained release formulations of psychoactive drugs |
| WO2010028130A2 (en) * | 2008-09-03 | 2010-03-11 | Concert Pharmaceuticals, Inc. | Antidepressant compounds |
| US20110021507A1 (en) * | 2009-07-22 | 2011-01-27 | Theracos, Inc. | Inhibiting antipsychotic-induced weight gain |
| EP2510949A4 (en) * | 2009-12-11 | 2013-11-13 | Astellas Pharma Inc | THERAPEUTICS FOR FIBROMYALGIA |
| PL2632468T3 (pl) * | 2010-10-25 | 2018-04-30 | University Of Manitoba | Kompozycje terapeutyczne do leczenia symetrycznej polineuropatii cukrzycowej |
| WO2020206410A1 (en) * | 2019-04-04 | 2020-10-08 | University Of Maryland, Baltimore | Methods of using muscarinic antagonists in the treatment of depression |
Family Cites Families (66)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1795183B1 (de) | 1968-08-20 | 1972-07-20 | Thomae Gmbh Dr K | 5,11-Dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-on-derivate und Arzneimittel |
| US4172831A (en) | 1974-11-26 | 1979-10-30 | Lilly Industries Limited | Thieno-benzodiazepines |
| US3953430A (en) | 1975-02-24 | 1976-04-27 | American Cyanamid Company | Substituted benzodiazepin-10-ones and method of use |
| US4168269A (en) | 1978-04-12 | 1979-09-18 | American Cyanamid Company | Substituted thieno-benzodiazepines |
| US4536518A (en) | 1979-11-01 | 1985-08-20 | Pfizer Inc. | Antidepressant derivatives of cis-4-phenyl-1,2,3,4-tetrahydro-1-naphthalenamine |
| US4381301A (en) | 1980-05-07 | 1983-04-26 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Substituted tricyclic thieno compounds, their synthesis, their use, their compositions and their medicaments |
| US4933438A (en) | 1984-02-29 | 1990-06-12 | University Of Florida | Brain-specific analogues of centrally acting amines |
| US6150354A (en) | 1987-01-15 | 2000-11-21 | Bonnie Davis | Compounds for the treatment of Alzheimer's disease |
| US4839104A (en) | 1987-06-11 | 1989-06-13 | Pfizer, Inc. | Process for preparing sertraline intermediates |
| US4904731A (en) * | 1987-09-04 | 1990-02-27 | Shell Oil Company | Polymeric composition |
| US4952128A (en) * | 1987-09-22 | 1990-08-28 | Chicopee | Transverse web forming apparatus |
| EP0386145A1 (de) | 1987-12-22 | 1990-09-12 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Thienotricyclen zur behandlung von erkrankungen der bronchien |
| US5114976A (en) | 1989-01-06 | 1992-05-19 | Norden Michael J | Method for treating certain psychiatric disorders and certain psychiatric symptoms |
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| US4940731A (en) | 1989-08-30 | 1990-07-10 | Pfizer Inc. | Method of treating premature ejaculation using sertraline |
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| WO1992020327A1 (en) | 1991-05-14 | 1992-11-26 | Ernir Snorrason | Treatment of fatigue syndrome with cholinesterase inhibitors |
| IT1250421B (it) | 1991-05-30 | 1995-04-07 | Recordati Chem Pharm | Composizione farmaceutica a rilascio controllato con proprieta' bio-adesive. |
| US5324832A (en) | 1991-07-03 | 1994-06-28 | The United States Of America As Represented By The Department Of Health And Human Services | Muscarinic antagonists |
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| FR2710265B1 (fr) | 1993-09-22 | 1995-10-20 | Adir | Composition pharmaceutique bioadhésive pour la libération contrôlée de principes actifs. |
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| US6548084B2 (en) | 1995-07-20 | 2003-04-15 | Smithkline Beecham Plc | Controlled release compositions |
| US6245347B1 (en) | 1995-07-28 | 2001-06-12 | Zars, Inc. | Methods and apparatus for improved administration of pharmaceutically active compounds |
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-
2007
- 2007-06-14 US US11/763,145 patent/US7893053B2/en not_active Expired - Fee Related
- 2007-06-15 JP JP2009530697A patent/JP4874397B2/ja not_active Expired - Fee Related
- 2007-06-15 NZ NZ573570A patent/NZ573570A/en not_active IP Right Cessation
- 2007-06-15 BR BRPI0713733-8A patent/BRPI0713733A2/pt not_active IP Right Cessation
- 2007-06-15 EP EP07784456.1A patent/EP2032127B1/en not_active Not-in-force
- 2007-06-15 KR KR1020097000753A patent/KR101408650B1/ko not_active Expired - Fee Related
- 2007-06-15 CN CN2012103367136A patent/CN103041389A/zh active Pending
- 2007-06-15 SG SG2011043882A patent/SG172712A1/en unknown
- 2007-06-15 MX MX2008015887A patent/MX2008015887A/es active IP Right Grant
- 2007-06-15 AU AU2007260631A patent/AU2007260631B2/en not_active Ceased
- 2007-06-15 CA CA2655131A patent/CA2655131C/en not_active Expired - Fee Related
- 2007-06-15 WO PCT/US2007/071356 patent/WO2007147123A1/en not_active Ceased
- 2007-06-15 EP EP12194224.7A patent/EP2666358A1/en not_active Withdrawn
-
2008
- 2008-12-11 IL IL195857A patent/IL195857A/en active IP Right Grant
- 2008-12-18 ZA ZA2008/10680A patent/ZA200810680B/en unknown
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2010
- 2010-11-29 ZA ZA2010/08538A patent/ZA201008538B/en unknown
-
2011
- 2011-01-11 US US13/004,837 patent/US8735389B2/en not_active Expired - Fee Related
- 2011-10-11 JP JP2011224234A patent/JP5491475B2/ja not_active Expired - Fee Related
-
2012
- 2012-12-07 RU RU2012152922/15A patent/RU2012152922A/ru not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| BRPI0713733A2 (pt) | 2012-10-30 |
| IL195857A (en) | 2016-02-29 |
| RU2012152922A (ru) | 2014-06-20 |
| ZA201008538B (en) | 2014-01-29 |
| WO2007147123A1 (en) | 2007-12-21 |
| CA2655131A1 (en) | 2007-12-21 |
| EP2666358A1 (en) | 2013-11-27 |
| KR20090036114A (ko) | 2009-04-13 |
| US20110195952A1 (en) | 2011-08-11 |
| AU2007260631B2 (en) | 2013-02-14 |
| JP4874397B2 (ja) | 2012-02-15 |
| JP2009542819A (ja) | 2009-12-03 |
| US8735389B2 (en) | 2014-05-27 |
| NZ573570A (en) | 2012-01-12 |
| EP2032127A4 (en) | 2009-11-25 |
| JP2012036212A (ja) | 2012-02-23 |
| EP2032127A1 (en) | 2009-03-11 |
| JP5491475B2 (ja) | 2014-05-14 |
| CN103041389A (zh) | 2013-04-17 |
| AU2007260631A1 (en) | 2007-12-21 |
| CA2655131C (en) | 2015-08-04 |
| IL195857A0 (en) | 2009-09-22 |
| US20070293480A1 (en) | 2007-12-20 |
| MX2008015887A (es) | 2009-02-06 |
| EP2032127B1 (en) | 2014-07-23 |
| KR101408650B1 (ko) | 2014-06-20 |
| US7893053B2 (en) | 2011-02-22 |
| SG172712A1 (en) | 2011-07-28 |
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