ZA200606564B - Pyrolle-3-carboxamide derivatives for the treatment of obesity - Google Patents
Pyrolle-3-carboxamide derivatives for the treatment of obesity Download PDFInfo
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Classifications
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- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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Landscapes
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- Anesthesiology (AREA)
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- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0403780.0A GB0403780D0 (en) | 2004-02-20 | 2004-02-20 | Therapeutic agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200606564B true ZA200606564B (en) | 2008-01-30 |
Family
ID=32040068
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200606564A ZA200606564B (en) | 2004-02-20 | 2006-08-07 | Pyrolle-3-carboxamide derivatives for the treatment of obesity |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20080051433A1 (zh) |
| EP (1) | EP1718610A1 (zh) |
| JP (1) | JP4176805B2 (zh) |
| CN (1) | CN1918121A (zh) |
| AU (1) | AU2005214143B2 (zh) |
| CA (1) | CA2559398A1 (zh) |
| GB (1) | GB0403780D0 (zh) |
| WO (1) | WO2005080328A1 (zh) |
| ZA (1) | ZA200606564B (zh) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1574211A1 (en) * | 2004-03-09 | 2005-09-14 | Inserm | Use of antagonists of the CB1 receptor for the manufacture of a composition useful for the treatment of hepatic diseases |
| EP1928827B1 (en) | 2005-09-27 | 2012-08-22 | Myriad Genetics, Inc. | Pyrrole derivatives as therapeutic compounds |
| AR056560A1 (es) | 2005-10-06 | 2007-10-10 | Astrazeneca Ab | Pirrolopiridinonas como moduladores cb1 |
| BRPI0715160A2 (pt) | 2006-08-08 | 2013-06-11 | Sanofi Aventis | imidazolidina-2,4-dionas substituÍdas por arilamimoaril-alquil-, processo para preparÁ-las, medicamentos compeendendo estes compostos, e seu uso |
| EP2025674A1 (de) | 2007-08-15 | 2009-02-18 | sanofi-aventis | Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| FR2926554B1 (fr) | 2008-01-22 | 2010-03-12 | Sanofi Aventis | Derives de carboxamides azabicycliques, leur preparation et leur application en therapeutique |
| FR2930939B1 (fr) | 2008-05-09 | 2010-07-30 | Sanofi Aventis | Derives de pyrrole, leur preparation et leur application en therapeutique |
| AR072707A1 (es) | 2008-07-09 | 2010-09-15 | Sanofi Aventis | Compuestos heterociclicos, procesos para su preparacion, medicamentos que comprenden estos compuestos y el uso de los mismos |
| WO2010068601A1 (en) | 2008-12-08 | 2010-06-17 | Sanofi-Aventis | A crystalline heteroaromatic fluoroglycoside hydrate, processes for making, methods of use and pharmaceutical compositions thereof |
| SG178880A1 (en) | 2009-08-26 | 2012-04-27 | Sanofi Sa | Novel crystalline heteroaromatic fluoroglycoside hydrates, pharmaceuticals comprising these compounds and their use |
| EP2582709B1 (de) | 2010-06-18 | 2018-01-24 | Sanofi | Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen |
| WO2012120056A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
| WO2012120050A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Neue substituierte phenyl-oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
| WO2012120051A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Mit adamantan- oder noradamantan substituierte benzyl-oxathiazinderivate, diese verbindungen enthaltende arzneimittel und deren verwendung |
| WO2012120058A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Mit benzyl- oder heteromethylengruppen substituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
| US8710050B2 (en) | 2011-03-08 | 2014-04-29 | Sanofi | Di and tri- substituted oxathiazine derivatives, method for the production, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof |
| US8828995B2 (en) | 2011-03-08 | 2014-09-09 | Sanofi | Branched oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof |
| WO2012120057A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Neue substituierte phenyl-oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
| WO2012120052A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung |
| WO2012120054A1 (de) | 2011-03-08 | 2012-09-13 | Sanofi | Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung |
| EP3206683A4 (en) * | 2014-10-16 | 2018-06-13 | The Board of Trustees of the Leland Stanford Junior University | Novel methods, compounds, and compositions for anesthesia |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MXPA02009258A (es) * | 2000-03-23 | 2005-04-19 | Solvay Pharm Bv | Derivados de 4,5-dihidro-1h-pirazol que tienen actividad antagonistica de cannabis-1. |
| EP1432679A1 (en) * | 2001-09-24 | 2004-06-30 | Bayer Pharmaceuticals Corporation | Preparation and use of pyrrole derivatives for treating obesity |
| GB0230088D0 (en) * | 2002-12-24 | 2003-01-29 | Astrazeneca Ab | Therapeutic agents |
| CN100395234C (zh) * | 2003-01-02 | 2008-06-18 | 霍夫曼-拉罗奇有限公司 | 新cb1受体反激动剂 |
| GB0302671D0 (en) * | 2003-02-06 | 2003-03-12 | Astrazeneca Ab | Pharmaceutical formulations |
-
2004
- 2004-02-20 GB GBGB0403780.0A patent/GB0403780D0/en not_active Ceased
-
2005
- 2005-02-17 US US10/588,518 patent/US20080051433A1/en not_active Abandoned
- 2005-02-17 JP JP2006553667A patent/JP4176805B2/ja not_active Expired - Fee Related
- 2005-02-17 EP EP05708389A patent/EP1718610A1/en not_active Withdrawn
- 2005-02-17 WO PCT/GB2005/000588 patent/WO2005080328A1/en active Application Filing
- 2005-02-17 CN CNA2005800049731A patent/CN1918121A/zh active Pending
- 2005-02-17 CA CA002559398A patent/CA2559398A1/en not_active Abandoned
- 2005-02-17 AU AU2005214143A patent/AU2005214143B2/en not_active Ceased
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2006
- 2006-08-07 ZA ZA200606564A patent/ZA200606564B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP1718610A1 (en) | 2006-11-08 |
| WO2005080328A1 (en) | 2005-09-01 |
| CN1918121A (zh) | 2007-02-21 |
| CA2559398A1 (en) | 2005-09-01 |
| AU2005214143B2 (en) | 2008-02-21 |
| JP4176805B2 (ja) | 2008-11-05 |
| GB0403780D0 (en) | 2004-03-24 |
| AU2005214143A1 (en) | 2005-09-01 |
| JP2007523147A (ja) | 2007-08-16 |
| US20080051433A1 (en) | 2008-02-28 |
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