ZA200507258B - 4, 6-, or 7-hydroxyindoles having n-oxide groups and the use thereof as therapeutic agents - Google Patents
4, 6-, or 7-hydroxyindoles having n-oxide groups and the use thereof as therapeutic agents Download PDFInfo
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- ZA200507258B ZA200507258B ZA200507258A ZA200507258A ZA200507258B ZA 200507258 B ZA200507258 B ZA 200507258B ZA 200507258 A ZA200507258 A ZA 200507258A ZA 200507258 A ZA200507258 A ZA 200507258A ZA 200507258 B ZA200507258 B ZA 200507258B
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
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- Public Health (AREA)
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- Pulmonology (AREA)
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- Diabetes (AREA)
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- Virology (AREA)
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- Dermatology (AREA)
- Cardiology (AREA)
- Endocrinology (AREA)
- Heart & Thoracic Surgery (AREA)
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Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10318611A DE10318611A1 (de) | 2003-04-24 | 2003-04-24 | 4-, 6- oder 7-Hydroxyindole mit N-Oxidgruppen und deren Verwendung als Therapeutika |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200507258B true ZA200507258B (en) | 2006-06-28 |
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| Application Number | Title | Priority Date | Filing Date |
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| ZA200507258A ZA200507258B (en) | 2003-04-24 | 2005-09-09 | 4, 6-, or 7-hydroxyindoles having n-oxide groups and the use thereof as therapeutic agents |
Country Status (16)
Families Citing this family (7)
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|---|---|---|---|---|
| TW200738677A (en) * | 2005-06-27 | 2007-10-16 | Elbion Ag | Nitro-substituted hydroxyindoles, their use as inhibitors of phosphodiesterase 4, and processes for preparing them |
| US8067433B2 (en) | 2005-11-09 | 2011-11-29 | Zalicus Inc. | Methods, compositions, and kits for the treatment of ophthalmic disorders |
| WO2008019357A2 (en) * | 2006-08-07 | 2008-02-14 | Ironwood Pharmaceuticals, Inc. | Indole compounds |
| SI2124944T1 (sl) * | 2007-03-14 | 2012-05-31 | Ranbaxy Lab Ltd | Derivati pirazolo b piridina kot inhibitorji fosfodiesteraze |
| AR084433A1 (es) | 2010-12-22 | 2013-05-15 | Ironwood Pharmaceuticals Inc | Inhibidores de la faah y composiciones farmaceuticas que los contienen |
| CR20200464A (es) | 2018-03-08 | 2021-04-14 | Incyte Corp | Compuestos diólicos de aminopirazina como inhibidores de pi3k-y |
| WO2020010003A1 (en) | 2018-07-02 | 2020-01-09 | Incyte Corporation | AMINOPYRAZINE DERIVATIVES AS PI3K-γ INHIBITORS |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19636150A1 (de) | 1996-09-06 | 1998-03-12 | Asta Medica Ag | N-substituierte Indol-3-glyoxylamide mit antiasthmatischer, antiallergischer und immunsuppressiver/immunmodulierender Wirkung |
| DE19814838C2 (de) | 1998-04-02 | 2001-01-18 | Asta Medica Ag | Indolyl-3-glyoxylsäure-Derivate mit Antitumorwirkung |
| DK1076657T3 (da) | 1998-04-28 | 2004-11-08 | Elbion Ag | Hidtil ukendte hydroxyindoler, deres anvendelse som inhibitorer for phosphodiesterase 4 og fremgangsmåde til deres fremstilling |
| DE19962300A1 (de) * | 1999-12-23 | 2001-06-28 | Asta Medica Ag | Substituierte N-Benzyl-Indol-3-yl-glyoxylsäure-Derivate mit Antitumorwirkung |
| IL160810A0 (en) | 2001-09-13 | 2004-08-31 | Synta Pharmaceuticals Corp | 1-glyoxlylamide indolizines for treating cancer |
| US20040116462A1 (en) | 2002-12-12 | 2004-06-17 | Mitsunori Ono | Indolizine compounds |
| DE10253426B4 (de) * | 2002-11-15 | 2005-09-22 | Elbion Ag | Neue Hydroxyindole, deren Verwendung als Inhibitoren der Phosphodiesterase 4 und Verfahren zu deren Herstellung |
| DE10318609A1 (de) * | 2003-04-24 | 2004-11-11 | Elbion Ag | 5-Hydroxyindole mit N-Oxidgruppen und deren Verwendung als Therapeutika |
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2003
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2004
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- 2004-04-21 TW TW093111114A patent/TW200503693A/zh unknown
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- 2004-04-23 EP EP04729109A patent/EP1615912A1/de not_active Withdrawn
- 2004-04-23 KR KR1020057020097A patent/KR20060021831A/ko not_active Withdrawn
- 2004-04-23 MX MXPA05011437A patent/MXPA05011437A/es unknown
- 2004-04-23 RU RU2005136431/04A patent/RU2005136431A/ru not_active Application Discontinuation
- 2004-04-23 CN CNA2004800110345A patent/CN1777600A/zh active Pending
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2005
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2006
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Also Published As
| Publication number | Publication date |
|---|---|
| MXPA05011437A (es) | 2005-12-12 |
| AU2004232482A1 (en) | 2004-11-04 |
| US20060128758A1 (en) | 2006-06-15 |
| NO20055517L (no) | 2006-01-18 |
| EP1615912A1 (de) | 2006-01-18 |
| BRPI0409793A (pt) | 2006-05-30 |
| CN1777600A (zh) | 2006-05-24 |
| US20040242643A1 (en) | 2004-12-02 |
| CA2523048A1 (en) | 2004-11-04 |
| US7067536B2 (en) | 2006-06-27 |
| NO20055517D0 (no) | 2005-11-22 |
| TW200503693A (en) | 2005-02-01 |
| KR20060021831A (ko) | 2006-03-08 |
| RU2005136431A (ru) | 2006-03-20 |
| WO2004094405A1 (de) | 2004-11-04 |
| JP2006524208A (ja) | 2006-10-26 |
| DE10318611A1 (de) | 2004-11-11 |
| AR044081A1 (es) | 2005-08-24 |
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