ZA200204485B - Fused tri-heterocyclic compounds. - Google Patents

Fused tri-heterocyclic compounds.

Info

Publication number
ZA200204485B
ZA200204485B ZA200204485A ZA200204485A ZA200204485B ZA 200204485 B ZA200204485 B ZA 200204485B ZA 200204485 A ZA200204485 A ZA 200204485A ZA 200204485 A ZA200204485 A ZA 200204485A ZA 200204485 B ZA200204485 B ZA 200204485B
Authority
ZA
South Africa
Prior art keywords
heterocyclic compounds
fused tri
tri
fused
heterocyclic
Prior art date
Application number
ZA200204485A
Other languages
English (en)
Inventor
Lee Fang Yu
Lee Fang Chen
Yang Chang An
Ma Wei Yong
Xiao Xu Hua
Xu Ai Wu
Wu Qiu Ye
Original Assignee
Yung Shin Pharmaceutical Ind
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to EP02011934A priority Critical patent/EP1270008B1/en
Priority to JP2002157957A priority patent/JP2003104987A/ja
Priority to CN02122155A priority patent/CN1389463A/zh
Priority to US10/161,215 priority patent/US6887997B2/en
Application filed by Yung Shin Pharmaceutical Ind filed Critical Yung Shin Pharmaceutical Ind
Priority to AU45802/02A priority patent/AU4580202A/en
Priority to ZA200204485A priority patent/ZA200204485B/xx
Priority to CA002389634A priority patent/CA2389634A1/en
Publication of ZA200204485B publication Critical patent/ZA200204485B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ZA200204485A 2001-05-31 2002-06-05 Fused tri-heterocyclic compounds. ZA200204485B (en)

Priority Applications (7)

Application Number Priority Date Filing Date Title
EP02011934A EP1270008B1 (en) 2001-05-31 2002-05-29 Fused tricyclic analogues of guanosine for treating tumors
JP2002157957A JP2003104987A (ja) 2001-05-31 2002-05-30 縮合三環性複素環化合物
CN02122155A CN1389463A (zh) 2001-05-31 2002-05-31 稠合的三杂环化合物
US10/161,215 US6887997B2 (en) 2001-05-31 2002-05-31 9H-imidazo[1,2-a]purin-9-one compounds
AU45802/02A AU4580202A (en) 2001-05-31 2002-06-05 Fused tri-heterocyclic compounds
ZA200204485A ZA200204485B (en) 2001-05-31 2002-06-05 Fused tri-heterocyclic compounds.
CA002389634A CA2389634A1 (en) 2001-05-31 2002-06-06 Fused tri-heterocyclic compounds

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US29508601P 2001-05-31 2001-05-31
ZA200204485A ZA200204485B (en) 2001-05-31 2002-06-05 Fused tri-heterocyclic compounds.
CA002389634A CA2389634A1 (en) 2001-05-31 2002-06-06 Fused tri-heterocyclic compounds

Publications (1)

Publication Number Publication Date
ZA200204485B true ZA200204485B (en) 2003-08-27

Family

ID=32995168

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200204485A ZA200204485B (en) 2001-05-31 2002-06-05 Fused tri-heterocyclic compounds.

Country Status (7)

Country Link
US (1) US6887997B2 (ja)
EP (1) EP1270008B1 (ja)
JP (1) JP2003104987A (ja)
CN (1) CN1389463A (ja)
AU (1) AU4580202A (ja)
CA (1) CA2389634A1 (ja)
ZA (1) ZA200204485B (ja)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN100516049C (zh) * 2004-11-16 2009-07-22 永信药品工业股份有限公司 抗血管生成药n2-(取代的芳基甲基)-3-(取代的苯基)吲唑的合成

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE109154T1 (de) * 1988-08-25 1994-08-15 Yoshitomi Pharmaceutical 2'-methylidenpyrimidin-nukleoside, ihre verwendung und verfahren zu ihrer herstellung.
US5591722A (en) * 1989-09-15 1997-01-07 Southern Research Institute 2'-deoxy-4'-thioribonucleosides and their antiviral activity
US5412088A (en) * 1989-11-20 1995-05-02 Rutgers, The State University 6-O-substituted guanosine derivatives
EP0693072B9 (en) * 1993-04-08 2004-09-15 The Trustees of Columbia University in the City of New York Method for the synthesis of 4- and/or 5-(di)substituted 2-aminoimidazoles from 2-aminoimidazoles and aldehydes
US5521294A (en) * 1995-01-18 1996-05-28 Eli Lilly And Company 2,2-difluoro-3-carbamoyl ribose sulfonate compounds and process for the preparation of beta nucleosides

Also Published As

Publication number Publication date
EP1270008A3 (en) 2003-01-15
EP1270008A2 (en) 2003-01-02
CA2389634A1 (en) 2003-12-06
US20030105116A1 (en) 2003-06-05
AU4580202A (en) 2002-12-05
JP2003104987A (ja) 2003-04-09
US6887997B2 (en) 2005-05-03
EP1270008B1 (en) 2006-07-12
CN1389463A (zh) 2003-01-08

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