ZA200105473B - Utilisation of 2-substituted 1,2-benzisothiazole derivatives and 3-substituted tetrahydropyridopyrimidinone derivatives for the prophylaxis and therapy of cerebral ischaemia. - Google Patents
Utilisation of 2-substituted 1,2-benzisothiazole derivatives and 3-substituted tetrahydropyridopyrimidinone derivatives for the prophylaxis and therapy of cerebral ischaemia.Info
- Publication number
- ZA200105473B ZA200105473B ZA200105473A ZA200105473A ZA200105473B ZA 200105473 B ZA200105473 B ZA 200105473B ZA 200105473 A ZA200105473 A ZA 200105473A ZA 200105473 A ZA200105473 A ZA 200105473A ZA 200105473 B ZA200105473 B ZA 200105473B
- Authority
- ZA
- South Africa
- Prior art keywords
- substituted
- derivatives
- utilisation
- prophylaxis
- therapy
- Prior art date
Links
- -1 2-substituted 1,2-benzisothiazole Chemical class 0.000 title 2
- 206010008120 Cerebral ischaemia Diseases 0.000 title 1
- 238000011321 prophylaxis Methods 0.000 title 1
- 238000002560 therapeutic procedure Methods 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
- Steroid Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19900544A DE19900544A1 (en) | 1999-01-11 | 1999-01-11 | Use of compounds of formula I for the prophylaxis and therapy of cerebral ischemia |
Publications (1)
Publication Number | Publication Date |
---|---|
ZA200105473B true ZA200105473B (en) | 2002-10-03 |
Family
ID=7893835
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA200105473A ZA200105473B (en) | 1999-01-11 | 2001-07-03 | Utilisation of 2-substituted 1,2-benzisothiazole derivatives and 3-substituted tetrahydropyridopyrimidinone derivatives for the prophylaxis and therapy of cerebral ischaemia. |
Country Status (19)
Country | Link |
---|---|
EP (1) | EP1140099A1 (en) |
JP (1) | JP2002534467A (en) |
KR (1) | KR20010101440A (en) |
CN (1) | CN1333685A (en) |
AR (1) | AR029741A1 (en) |
AU (1) | AU2285100A (en) |
BG (1) | BG105688A (en) |
BR (1) | BR9916888A (en) |
CA (1) | CA2359390A1 (en) |
DE (1) | DE19900544A1 (en) |
HU (1) | HUP0200520A3 (en) |
IL (1) | IL144145A0 (en) |
MX (1) | MXPA01006966A (en) |
NO (1) | NO20013408L (en) |
PL (1) | PL348916A1 (en) |
SK (1) | SK9682001A3 (en) |
TR (1) | TR200102009T2 (en) |
WO (1) | WO2000041697A1 (en) |
ZA (1) | ZA200105473B (en) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1560488B1 (en) | 2002-11-05 | 2010-09-01 | Glaxo Group Limited | Antibacterial agents |
EP1667979A4 (en) * | 2003-09-23 | 2007-04-18 | Merck & Co Inc | Isoquinoline potassium channel inhibitors |
BRPI0615248A2 (en) * | 2005-08-26 | 2009-07-14 | Shionogi & Co | derivative having ppar agonist activity |
KR20100063087A (en) * | 2007-09-20 | 2010-06-10 | 코텍스 파마슈티칼스, 인크. | 3-substituted 1,2,3-triazin-4-one's and 3-substituted 1,3-pyrimidinone's for enhancing glutamatergic synaptic responses |
MA41168A (en) | 2014-12-17 | 2017-10-24 | Acraf | NEW ANTIBACTERIAL COMPOUNDS |
CN108484594B (en) * | 2018-02-09 | 2020-08-04 | 福建医科大学 | Alkoxy substituted tetrahydropyridopyrimidine compound or available salt thereof, and preparation method and application thereof |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3620643A1 (en) * | 1985-06-22 | 1987-01-22 | Sandoz Ag | Thiazoles, their preparation and use |
DE3831888A1 (en) * | 1988-09-20 | 1990-03-29 | Troponwerke Gmbh & Co Kg | MEDICINES FOR TREATING APOPLEXIA CEREBRI |
JP3036789B2 (en) * | 1990-06-22 | 2000-04-24 | 三井化学株式会社 | Novel heterocyclic compounds and pharmaceutical compositions |
DE19746612A1 (en) * | 1997-10-22 | 1999-04-29 | Basf Ag | New 2-substituted 1,2-benzisothiazole derivatives |
DE19747063A1 (en) * | 1997-10-24 | 1999-04-29 | Basf Ag | New 3-substituted tetrahydropyridopyrimidinone derivatives |
-
1999
- 1999-01-11 DE DE19900544A patent/DE19900544A1/en not_active Withdrawn
- 1999-12-22 EP EP99966990A patent/EP1140099A1/en not_active Withdrawn
- 1999-12-22 MX MXPA01006966A patent/MXPA01006966A/en unknown
- 1999-12-22 KR KR1020017008690A patent/KR20010101440A/en not_active Application Discontinuation
- 1999-12-22 PL PL99348916A patent/PL348916A1/en not_active Application Discontinuation
- 1999-12-22 JP JP2000593308A patent/JP2002534467A/en active Pending
- 1999-12-22 CN CN99815452A patent/CN1333685A/en active Pending
- 1999-12-22 IL IL14414599A patent/IL144145A0/en unknown
- 1999-12-22 HU HU0200520A patent/HUP0200520A3/en unknown
- 1999-12-22 WO PCT/EP1999/010275 patent/WO2000041697A1/en not_active Application Discontinuation
- 1999-12-22 CA CA002359390A patent/CA2359390A1/en not_active Abandoned
- 1999-12-22 AU AU22851/00A patent/AU2285100A/en not_active Abandoned
- 1999-12-22 TR TR2001/02009T patent/TR200102009T2/en unknown
- 1999-12-22 BR BR9916888-0A patent/BR9916888A/en not_active IP Right Cessation
- 1999-12-22 SK SK968-2001A patent/SK9682001A3/en unknown
-
2000
- 2000-01-06 AR ARP000100036A patent/AR029741A1/en unknown
-
2001
- 2001-07-03 ZA ZA200105473A patent/ZA200105473B/en unknown
- 2001-07-10 NO NO20013408A patent/NO20013408L/en not_active Application Discontinuation
- 2001-07-10 BG BG105688A patent/BG105688A/en unknown
Also Published As
Publication number | Publication date |
---|---|
HUP0200520A2 (en) | 2002-07-29 |
BR9916888A (en) | 2001-11-20 |
DE19900544A1 (en) | 2000-07-13 |
AR029741A1 (en) | 2003-07-16 |
CA2359390A1 (en) | 2000-07-20 |
JP2002534467A (en) | 2002-10-15 |
KR20010101440A (en) | 2001-11-14 |
BG105688A (en) | 2002-02-28 |
WO2000041697A1 (en) | 2000-07-20 |
MXPA01006966A (en) | 2002-04-10 |
AU2285100A (en) | 2000-08-01 |
CN1333685A (en) | 2002-01-30 |
HUP0200520A3 (en) | 2003-04-28 |
TR200102009T2 (en) | 2002-01-21 |
NO20013408L (en) | 2001-08-21 |
IL144145A0 (en) | 2002-05-23 |
NO20013408D0 (en) | 2001-07-10 |
PL348916A1 (en) | 2002-06-17 |
SK9682001A3 (en) | 2002-03-05 |
EP1140099A1 (en) | 2001-10-10 |
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