YU28495A - NEW AMINO ACID DERIVATIVES A PROCEDURE FOR THEIR PREPARATION AND THE PHARMACEUTICAL PRODUCTS CONTAINING THESE COMPOUNDS (II) - Google Patents
NEW AMINO ACID DERIVATIVES A PROCEDURE FOR THEIR PREPARATION AND THE PHARMACEUTICAL PRODUCTS CONTAINING THESE COMPOUNDS (II)Info
- Publication number
- YU28495A YU28495A YU28495A YU28495A YU28495A YU 28495 A YU28495 A YU 28495A YU 28495 A YU28495 A YU 28495A YU 28495 A YU28495 A YU 28495A YU 28495 A YU28495 A YU 28495A
- Authority
- YU
- Yugoslavia
- Prior art keywords
- preparation
- amino acid
- acid derivatives
- compounds
- procedure
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
- C07K5/06165—Dipeptides with the first amino acid being heterocyclic and Pro-amino acid; Derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- General Health & Medical Sciences (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Life Sciences & Earth Sciences (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
NOVI DERIVATI AMINO KISELINE POSTUPAK ZA NJIHOVO PRIPREMANJE I FARMACEUTSKI PREPARATI KOJI SADRŽE OVA JEDINJENJA (II) - Pronalazak se odnosi na nove derivate amino kiseline, opšte formule R'-R^-A'-B i njihove farmaceutski prihvatljive soli, u kojoj grupa B označava -A2- NR2R3 ili R5, pri čemu R 1 Al A2 p2 R3 OS r6 p7 r8 ,M,M,n,n,n,ri,n,ri,R9, X, Y, Z, t i u imaju značenja navedena u opisu, kao i njihovo pripremanje i primenu. Nova jedinjenja su dragoceni antagonisti neurokinina (tahikinina).The invention relates to new amino acid derivatives, of general formula R'-R ^ -A'-B and their pharmaceutically acceptable salts, in which group B denotes -A2- NR2R3 or R5, wherein R 1 Al A2 p2 R3 OS r6 p7 r8, M, M, n, n, n, ri, n, ri, R9, X, Y, Z, tiu have the meanings given in description, as well as their preparation and application. The new compounds are valuable antagonists of neurokinin (tachykinin).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE4416255 | 1994-05-07 | ||
DE4445939A DE4445939A1 (en) | 1994-05-07 | 1994-12-22 | Novel amino acid derivatives, process for their preparation and pharmaceutical compositions containing them (II) |
Publications (1)
Publication Number | Publication Date |
---|---|
YU28495A true YU28495A (en) | 1998-05-15 |
Family
ID=6517628
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
YU28495A YU28495A (en) | 1994-05-07 | 1995-05-05 | NEW AMINO ACID DERIVATIVES A PROCEDURE FOR THEIR PREPARATION AND THE PHARMACEUTICAL PRODUCTS CONTAINING THESE COMPOUNDS (II) |
Country Status (6)
Country | Link |
---|---|
KR (1) | KR970702876A (en) |
CO (1) | CO4960643A1 (en) |
DE (1) | DE4445939A1 (en) |
PE (1) | PE14996A1 (en) |
YU (1) | YU28495A (en) |
ZA (1) | ZA953628B (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE19541283A1 (en) * | 1995-11-06 | 1997-05-07 | Boehringer Ingelheim Kg | Novel amino acid derivatives, processes for their preparation and pharmaceutical compositions containing these compounds |
-
1994
- 1994-12-22 DE DE4445939A patent/DE4445939A1/en not_active Withdrawn
-
1995
- 1995-05-04 CO CO95018565A patent/CO4960643A1/en unknown
- 1995-05-05 YU YU28495A patent/YU28495A/en unknown
- 1995-05-05 PE PE1995267931A patent/PE14996A1/en not_active Application Discontinuation
- 1995-05-05 ZA ZA953628A patent/ZA953628B/en unknown
-
1996
- 1996-11-07 KR KR1019960706283A patent/KR970702876A/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
ZA953628B (en) | 1995-11-07 |
KR970702876A (en) | 1997-06-10 |
DE4445939A1 (en) | 1995-11-09 |
CO4960643A1 (en) | 2000-09-25 |
PE14996A1 (en) | 1996-05-08 |
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