YU12396A - PROCEDURE FOR PREPARATION OF LORAKARBEG MONOHYDRATE - Google Patents

PROCEDURE FOR PREPARATION OF LORAKARBEG MONOHYDRATE

Info

Publication number
YU12396A
YU12396A YU12396A YU12396A YU12396A YU 12396 A YU12396 A YU 12396A YU 12396 A YU12396 A YU 12396A YU 12396 A YU12396 A YU 12396A YU 12396 A YU12396 A YU 12396A
Authority
YU
Yugoslavia
Prior art keywords
compound
formula
monohydrate
lorakarbeg
procedure
Prior art date
Application number
YU12396A
Other languages
Serbo-Croatian (sh)
Inventor
Henning
Stout
Original Assignee
Eli Lilly Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly Company filed Critical Eli Lilly Company
Priority to YU12396A priority Critical patent/YU12396A/en
Publication of YU12396A publication Critical patent/YU12396A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Ovaj pronalazak obezbedjuje postupak za pripremanje kristalnog anhidratnog oblika jedinjenja formule (I)koji obuhvata izlaganje kristalnog anhidratnog oblika jedinjenja formule (I) relativnoj vlažnosti od oko 90 do oko 100%, a takodje obezbedjuje postupak za pripremanje kristalnog anhidratnog oblika jedinjenja formule (I) koji obuhvata sušenje kristalnog izopropanolatnog oblika jedinjenja formule (I) na temperaturi od oko 50В°C do oko 100В°C, i postupak za pripremanje kristalnog monohidratnog oblika jedinjenja formule (I) koji obuhvata izlaganje kristalnog anhidratnog oblika jedinjenja formule (I) relativnoj vlažnosti od oko 90 do oko 100%.The present invention provides a process for preparing a crystalline anhydrous form of a compound of formula (I) comprising exposing a crystalline anhydrous form of a compound of formula (I) to a relative humidity of about 90 to about 100%, and also provides a process for preparing a crystalline anhydrous form of a compound of formula (I) which comprising drying the crystalline isopropanolate form of the compound of formula (I) at a temperature of from about 50V ° C to about 100V ° C, and a process for preparing the crystalline monohydrate form of the compound of formula (I) comprising exposing the crystalline anhydrous form of the compound of formula (I) to a relative humidity of about 90 to about 100%.

YU12396A 1996-02-29 1996-02-29 PROCEDURE FOR PREPARATION OF LORAKARBEG MONOHYDRATE YU12396A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
YU12396A YU12396A (en) 1996-02-29 1996-02-29 PROCEDURE FOR PREPARATION OF LORAKARBEG MONOHYDRATE

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
YU12396A YU12396A (en) 1996-02-29 1996-02-29 PROCEDURE FOR PREPARATION OF LORAKARBEG MONOHYDRATE

Publications (1)

Publication Number Publication Date
YU12396A true YU12396A (en) 1998-07-10

Family

ID=47595852

Family Applications (1)

Application Number Title Priority Date Filing Date
YU12396A YU12396A (en) 1996-02-29 1996-02-29 PROCEDURE FOR PREPARATION OF LORAKARBEG MONOHYDRATE

Country Status (1)

Country Link
YU (1) YU12396A (en)

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