WO2019203755A3 - Forme pharmaceutique orale solide comprenant de la linagliptine - Google Patents
Forme pharmaceutique orale solide comprenant de la linagliptine Download PDFInfo
- Publication number
- WO2019203755A3 WO2019203755A3 PCT/TR2018/050812 TR2018050812W WO2019203755A3 WO 2019203755 A3 WO2019203755 A3 WO 2019203755A3 TR 2018050812 W TR2018050812 W TR 2018050812W WO 2019203755 A3 WO2019203755 A3 WO 2019203755A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- linagliptin
- dosage form
- oral dosage
- solid oral
- binder
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
- A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La présente invention concerne une forme pharmaceutique orale solide comprenant de la linagliptine et au moins un liant.
Priority Applications (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CA3085455A CA3085455C (fr) | 2017-12-15 | 2018-12-14 | Forme pharmaceutique orale solide comprenant de la linagliptine |
EP18914956.0A EP3723761A4 (fr) | 2017-12-15 | 2018-12-14 | Forme pharmaceutique orale solide comprenant de la linagliptine |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
TR2017/20515 | 2017-12-15 | ||
TR2017/20515A TR201720515A2 (tr) | 2017-12-15 | 2017-12-15 | Li̇nagli̇pti̇n i̇çeren bi̇r kati oral dozaj formu |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2019203755A2 WO2019203755A2 (fr) | 2019-10-24 |
WO2019203755A3 true WO2019203755A3 (fr) | 2020-01-16 |
Family
ID=67900883
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/TR2018/050812 WO2019203755A2 (fr) | 2017-12-15 | 2018-12-14 | Forme pharmaceutique orale solide comprenant de la linagliptine |
Country Status (4)
Country | Link |
---|---|
EP (1) | EP3723761A4 (fr) |
CA (1) | CA3085455C (fr) |
TR (1) | TR201720515A2 (fr) |
WO (1) | WO2019203755A2 (fr) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2022173406A1 (fr) * | 2021-02-15 | 2022-08-18 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Procédé pour formulations de linagliptine ou d'un sel pharmaceutiquement acceptable de celle-ci |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN106138059A (zh) * | 2015-03-27 | 2016-11-23 | 天津汉瑞药业有限公司 | 一种稳定的利格列汀药物组合物 |
EP3156048A1 (fr) * | 2015-10-13 | 2017-04-19 | Galenicum Health S.L. | Composition pharmaceutique stable de linagliptine sous forme de comprimé à libération immédiate |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
UY32427A (es) * | 2009-02-13 | 2010-09-30 | Boheringer Ingelheim Internat Gmbh | Composicion farmaceutica, forma farmaceutica, procedimiento para su preparacion, metodos de tratamiento y usos de la misma |
WO2013128379A2 (fr) | 2012-02-27 | 2013-09-06 | Dr. Reddy's Laboratories Limited | Formes polymorphes cristallines de linagliptine |
EP2908806A1 (fr) * | 2012-10-09 | 2015-08-26 | Boehringer Ingelheim International GmbH | Utilisation de matière à fabriquer les comprimés dont on ajuste sélectivement l'humidité dans la production de comprimés mécaniquement stables qui contiennent au moins une substance active formant un hydrate et/ou un adjuvant lié à la stabilité mécanique des comprimés, en particulier des comprimés contenant de l'arginine |
WO2014080383A1 (fr) * | 2012-11-26 | 2014-05-30 | Ranbaxy Laboratories Limited | Composition pharmaceutique d'inhibiteurs de la dipeptidyl-peptidase-iv (dpp-iv) en association avec d'autres antidiabétiques |
WO2014080384A1 (fr) | 2012-11-26 | 2014-05-30 | Ranbaxy Laboratories Limited | Composition pharmaceutique de linagliptine |
-
2017
- 2017-12-15 TR TR2017/20515A patent/TR201720515A2/tr unknown
-
2018
- 2018-12-14 CA CA3085455A patent/CA3085455C/fr active Active
- 2018-12-14 EP EP18914956.0A patent/EP3723761A4/fr active Pending
- 2018-12-14 WO PCT/TR2018/050812 patent/WO2019203755A2/fr unknown
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN106138059A (zh) * | 2015-03-27 | 2016-11-23 | 天津汉瑞药业有限公司 | 一种稳定的利格列汀药物组合物 |
EP3156048A1 (fr) * | 2015-10-13 | 2017-04-19 | Galenicum Health S.L. | Composition pharmaceutique stable de linagliptine sous forme de comprimé à libération immédiate |
Also Published As
Publication number | Publication date |
---|---|
EP3723761A4 (fr) | 2021-06-30 |
EP3723761A2 (fr) | 2020-10-21 |
TR201720515A2 (tr) | 2019-07-22 |
WO2019203755A2 (fr) | 2019-10-24 |
CA3085455A1 (fr) | 2019-10-24 |
CA3085455C (fr) | 2022-08-16 |
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