WO2018117034A1 - Oxadiazole compound and plant disease control method - Google Patents

Abstract

Provided are a plant disease control method, said method comprising applying a compound represented by formula (I) to a plant or soil, and the compound. [In formula (I): G represents a thiophene ring, a furan ring, etc.; n represents 1, 2, 3 or 4; in the combination of L, X and R², L represents C(O), X represents a single bond, NR³ or an oxygen atom, and R² represents a C₁-C₆ alkyl group optionally having one or more substituents selected from group A, etc.; R¹ represents a C₁-C₆ alkyl group optionally having one or more substituents selected from group A, etc., or R¹ and R² may form, together with the carbon atom to which R¹ and R² are attached, a 3- to 7-membered cycloalkylene group, etc.; R³ represents a C₁-C₆ alkyl group optionally having one or more substituents selected from group A, etc.; and Z represents a C₃-C₆ cycloalkyl group, etc., or X and Z may form, together with L to which X and Z are attached, a 4- to 7-membered heterocycle, etc.]

Description

Oxadiazole compound and method for controlling plant diseases

The present invention relates to an oxadiazole compound and a method for controlling plant diseases.

Patent Document 1 describes an oxadiazole compound for pharmaceutical use.

International Publication No. 2013/066835

An object of the present invention is to provide an excellent control method for plant diseases.

As a result of studying to find an excellent method for controlling plant diseases, the present inventor has found that the compound represented by the following formula (I) has an excellent control effect against plant diseases.
That is, the present invention is as follows.
[1] Formula (I)

[Where,
G is a thiophene ring, furan ring, pyrrole ring, imidazole ring, oxazole ring, isoxazole ring, thiazole ring, isothiazole ring, oxadiazole ring, thiadiazole ring, pyrazole ring, pyridine ring, pyrazine ring, pyridazine ring, pyrimidine Ring or benzene ring {the thiophene ring, the furan ring, the pyrrole ring, the imidazole ring, the oxazole ring, the isoxazole ring, the thiazole ring, the isothiazole ring, the pyrazole ring, the pyridine ring, the pyrazine ring , The pyridazine ring, the pyrimidine ring and the benzene ring each may have one or more substituents selected from group D}
n represents 1, 2, 3 or 4;
when n is 2, 3 or 4, the plurality of R ¹ and the plurality of R ² are the same or different,
The combination of L, X and R ² is
L is C (O), X is a single bond, NR ³ or an oxygen atom, and R ² is a C1-C6 alkyl group optionally having one or more substituents selected from group A, group A C1-C6 alkoxy group optionally having one or more substituents selected from B, a phenyl group optionally having one or more substituents selected from Group D, one or more selected from Group D An optionally substituted 5-6 membered aromatic heterocyclic group, one or more substituents selected from group D, a C3-C6 cycloalkyl group, a hydrogen atom, a halogen atom or cyano A combination that is a group, or
L is S (O) ₂ , X is NR ³ or an oxygen atom, R ² is a C1-C6 alkyl group optionally having one or more substituents selected from group A, from group B A C1-C6 alkoxy group optionally having one or more substituents selected, a phenyl group optionally having one or more substituents selected from Group D, one or more substituents selected from Group D A combination of a 5- to 6-membered aromatic heterocyclic group optionally having one or more, a C3-C6 cycloalkyl group optionally having one or more substituents selected from Group D, a halogen atom or a cyano group Represent,
R ¹ is a C1-C6 alkyl group optionally having one or more substituents selected from group A, a C1-C6 alkoxy group optionally having one or more substituents selected from group B, A phenyl group optionally having one or more substituents selected from group D, a 5-6-membered aromatic heterocyclic group optionally having one or more substituents selected from group D, from group D Represents a C3-C6 cycloalkyl group optionally having one or more selected substituents, a hydrogen atom, a halogen atom or a cyano group,
R ¹ and R ^2, together with the carbon atoms to which they are attached, 3-7 membered cycloalkylene group, or 3-7-membered saturated heterocyclic ring (wherein 3-7 membered cycloalkylene group, and 3-7-membered saturated heterocyclic The ring may have one or more substituents selected from group D),
R ³ is a C1-C6 alkyl group optionally having one or more substituents selected from group A, a C3-C6 alkenyl group optionally having one or more substituents selected from group A, A C3-C6 alkynyl group optionally having one or more substituents selected from group A, a C1-C6 alkoxy group optionally having one or more halogen atoms, one or more substituents selected from group D A C3-C6 cycloalkyl group optionally having a group, a phenyl group optionally having one or more substituents selected from group D, and one or more substituents selected from group D May represent a 5-6 membered aromatic heterocyclic group or a hydrogen atom,
Z is a C3-C6 cycloalkyl group, a phenyl group, a 5-6 membered aromatic heterocyclic group, a 3-6 membered non-aromatic heterocyclic group (the C3-C6 cycloalkyl group, the phenyl group, the 5-6 And the 3-6-membered non-aromatic heterocyclic group may have one or more substituents selected from group D), CR ⁴ R ⁵ R ⁶ , NR ⁷ R Represents ⁸ or OR ⁹ or
X and Z together with L to which they are attached form a 4-7 membered heterocycle (the 4-7 membered heterocycle may have one or more substituents selected from group D) You may,
R ⁴ , R ⁵ and R ⁶ are the same or different and are a C1-C6 alkyl group optionally having one or more substituents selected from the group consisting of Group A and Group E, 1 selected from Group A A C3-C6 alkenyl group optionally having one or more substituents, a C3-C6 alkynyl group optionally having one or more substituents selected from group A, and one or more substituents selected from group B A C1-C6 alkoxy group which may have, a C3-C6 cycloalkyl group which may have one or more substituents selected from group D, and one or more substituents selected from group D An optionally substituted phenyl group, a 5-6 membered aromatic heterocyclic group optionally having one or more substituents selected from group D, a hydrogen atom, a halogen atom or a cyano group;
R ⁷ and R ⁸ are the same or different and are each a C1-C6 alkyl group optionally having one or more substituents selected from the group consisting of group A and group E; one or more substituents selected from group A A C3-C6 alkenyl group which may have a group, a C3-C6 alkynyl group which may have one or more substituents selected from group A, and a C1 which may have one or more halogen atoms -C6 alkoxy group, C3-C6 cycloalkyl group optionally having one or more substituents selected from group D, phenyl group optionally having one or more substituents selected from group D, group Represents a 5- or 6-membered aromatic heterocyclic group which may have one or more substituents selected from D or a hydrogen atom, or R ⁷ and R ⁸ together with the nitrogen atom to which they are bonded 3-8 membered heterocycle (the 3-8 membered heterocycle is group D It may form may also be) have one or more substituents selected,
R ⁹ may have one or more substituents selected from the group consisting of group A and group E, and may have one or more substituents selected from group A. C3-C6 alkenyl group, C3-C6 alkynyl group optionally having one or more substituents selected from group A, C3-C6 cyclo optionally having one or more substituents selected from group D An alkyl group, a phenyl group optionally having one or more substituents selected from group D, a 5-6-membered aromatic heterocyclic group optionally having one or more substituents selected from group D, or Represents a hydrogen atom.
Group A: a C1-C6 alkoxy group optionally having one or more halogen atoms, a C1-C6 alkylthio group optionally having one or more halogen atoms, one or more substituents selected from group C A C3-C6 cycloalkyl group which may have, a phenyl group which may have one or more substituents selected from group F, and one or more substituents selected from group F. A group consisting of a 5-6 membered aromatic heterocyclic group, a halogen atom, a nitro group and a cyano group.
Group B: C1-C6 alkylthio group optionally having one or more halogen atoms, phenyl group optionally having one or more substituents selected from Group F, one or more substituents selected from Group F A group consisting of a 5-6-membered aromatic heterocyclic group, a halogen atom, a nitro group and a cyano group, which may have a group;
Group C: Group consisting of halogen atom, nitro group and cyano group.
Group D: a C1-C6 alkyl group optionally having one or more substituents selected from group C, a C3-C6 cycloalkyl group optionally having one or more substituents selected from group C, C1-C6 alkoxy group which may have one or more halogen atoms, C3-C6 alkenyloxy group which may have one or more halogen atoms, C3 which may have one or more halogen atoms -C6 alkynyloxy group, C1-C6 alkylthio group optionally having one or more halogen atoms, C1-C6 alkylsulfonyloxy group optionally having one or more halogen atoms, halogen atom, cyano group, A group consisting of a nitro group, a hydroxy group and an amino group.
Group E: (C1-C6 alkyl) carbonylamino group optionally having one or more substituents selected from group C, or one or more substituents selected from group C (C1-C6) C6 alkyl) aminocarbonyl group, di (C1-C6 alkyl) aminocarbonyl group optionally having one or more substituents selected from group C, having one or more substituents selected from group C A C1-C6 alkylsulfonylamino group, a C1-C6 alkylaminosulfonyl group optionally having one or more substituents selected from group C, and one or more substituents selected from group C. A group consisting of a di (C1-C6 alkyl) aminosulfonyl group, a hydroxy group and an amino group.
Group F: a group consisting of a C1-C6 alkyl group optionally having one or more halogen atoms, a C1-C6 alkoxy group optionally having one or more halogen atoms, a halogen atom and a cyano group. ]
A method for controlling plant diseases by treating a plant or soil with a compound represented by formula (hereinafter referred to as the present compound).
[2] Formula (II)

[Where,
G ^X represents thiophene ring, furan ring, pyrrole ring, imidazole ring, oxazole ring, isoxazole ring, thiazole ring, isothiazole ring, oxadiazole ring, thiadiazole ring, pyrazole ring, pyridine ring, pyrazine ring, pyridazine ring, Pyrimidine ring or benzene ring {the thiophene ring, the furan ring, the pyrrole ring, the imidazole ring, the oxazole ring, the isoxazole ring, the thiazole ring, the isothiazole ring, the pyrazole ring, the pyridine ring, the pyrazine The ring, the pyridazine ring, the pyrimidine ring, and the benzene ring may have one or more substituents selected from the group D ^X },
m represents 1, 2, 3 or 4;
when m is 2, 3 or 4, a plurality of R ^1X and a plurality of R ^2X are the same or different, respectively,
The combination of L ^X, X ^X and R ^2X is
L ^X is C (O), X ^X is NR ^3X or an oxygen atom, R ^2X is a C1-C6 alkyl group optionally having one or more substituents selected from group A ^X , 1 or more substituents optionally may C1-C6 alkoxy group which may have a phenyl group which may have one or more substituents selected from the group D ^X selected from B ^X, is selected from the group D ^X A 5-6 membered aromatic heterocyclic group optionally having one or more substituents, a C3-C6 cycloalkyl group optionally having one or more substituents selected from the group D ^X , a hydrogen atom, A combination that is a halogen atom or a cyano group, or
L ^X is S (O) ₂ , X ^X is NR ^3X or an oxygen atom, and R ^2X may have one or more substituents selected from group A ^X , 1 or more substituents optionally may C1-C6 alkoxy group which may have a phenyl group which may have one or more substituents selected from the group D ^X selected from the group B ^X, selected from the group D ^X A 5- or 6-membered aromatic heterocyclic group optionally having one or more substituents, a C3-C6 cycloalkyl group optionally having one or more substituents selected from group D ^X , a halogen atom Or represents a combination that is a cyano group,
R ^1X is one or more substituents optionally may be C1-C6 alkyl group optionally having a one or more substituents may C1-C6 alkoxy which may have a selected from the group B ^X selected from the group A ^X group, one or more substituents phenyl group which may have a one or more substituents may be a 5-6 membered aromatic heterocyclic group selected from the group D ^X is selected from the group D ^X represents one or more substituents optionally may be C3-C6 cycloalkyl group having a hydrogen atom, a halogen atom or a cyano group selected from the group D ^X,
R ^1X and R ^2X , together with the carbon atom to which they are attached, represent a 3-7 membered cycloalkylene group or a 3-7 membered saturated heterocycle (the 3-7 membered cycloalkylene group and 3-7 membered saturated heterocycle). The ring may have one or more substituents selected from group D ^X ),
R ^3X is one or more substituents optionally may C1-C6 alkyl group which may have one or more substituents may C3-C6 alkenyl which may have a selected from the group A ^X selected from the group A ^X A group, a C3-C6 alkynyl group optionally having one or more substituents selected from group A ^X , a C1-C6 alkoxy group optionally having one or more halogen atoms, selected from group D ^X 1 or may C3-C6 have a substituent of the cycloalkyl group, one or more substituents phenyl group which may have a selected from the group D ^X, one or more substituents selected from the group D ^X A 6-membered aromatic heterocyclic group which may have a group or a hydrogen atom,
Z ^X represents C3-C6 cycloalkyl group, phenyl group, 6-membered aromatic heterocyclic group, 3-6-membered non-aromatic heterocyclic group, pyrazol-4-yl group, thienyl group, furyl group, imidazolyl group, oxazolyl Group, isoxazolyl group, thiazolyl group, isothiazolyl group, oxadiazolyl group, thiadiazolyl group (the C3-C6 cycloalkyl group, the phenyl group, the 6-membered aromatic heterocyclic group, the 3-6-membered non-aromatic heterocyclic group, The pyrazol-4-yl group, the thienyl group, the furyl group, the imidazolyl group, the oxazolyl group, the isoxazolyl group, the thiazolyl group, the isothiazolyl group, the oxadiazolyl group, and the thiadiazolyl group are selected from the group D ^X Or may represent one or more substituents), CR ^4X R ^5X R ^6X , NR ^7X R ^8X or OR ^9X , or
X ^X and Z ^X together with L ^{X to} which they are bonded have a 4-7 membered heterocycle (the 4-7 membered heterocycle may have one or more substituents selected from group D ^X Good)
R ^4X, R ^5X and R ^6X are identical or different phases, one or more substituents optionally may C1-C6 alkyl group which may have a selected from the group consisting of the group A ^X and the group E ^X, from the group A ^X C3-C6 alkenyl group optionally having one or more substituents selected, C3-C6 alkynyl group optionally having one or more substituents selected from group A ^X , selected from group B ^X 1 or more substituents optionally may C1-C6 alkoxy group which may have one or more substituents may be a C3-C6 cycloalkyl group selected from the group D ^X, 1 is selected from the group D ^X A phenyl group optionally having the above substituents, a 5-6 membered aromatic heterocyclic group optionally having one or more substituents selected from the group D ^X , a hydrogen atom, a halogen atom or a cyano group Represents
R ^7X and R ^8X are the same or different and are a C1-C6 alkyl group optionally having one or more substituents selected from the group consisting of group A ^X and group E ^X , 1 selected from group A ^X or more substituents may have a C3-C6 alkenyl group, one or more substituents optionally may C3-C6 alkynyl group which may have a selected from the group a ^X, have one or more halogen atoms it may also be C1-C6 alkoxy group, one or more substituents the have optionally may C3-C6 cycloalkyl group selected from the group D ^X, have one or more substituents selected from the group D ^X Or a phenyl group, a 5- or 6-membered aromatic heterocyclic group which may have one or more substituents selected from the group D ^X or a hydrogen atom, or R ^7X and R ^8X are Combined with the nitrogen atom to be bonded, a 3-8 membered heterocycle (the 3-8 membered Ring may form a good) have one or more substituents selected from the group D ^X,
R ^9X is one or more substituents optionally may C1-C3 alkyl group which may have a selected from the group consisting of the group E ^X and the group G ^X, have one or more substituents selected from the group A ^X An optionally substituted C3-C6 alkenyl group, a C3-C6 alkynyl group optionally having one or more substituents selected from group A ^X , and one or more substituents selected from group D ^X good C3-C6 cycloalkyl group optionally substituted with one or more substituents phenyl group which may have a one or more substituents selected from the group D ^X is selected from the group D ^X 5-6 Represents a membered aromatic heterocyclic group or a hydrogen atom.
Group A ^X : C1-C6 alkoxy group optionally having one or more halogen atoms, C1-C6 alkylthio group optionally having one or more halogen atoms, one or more substitutions selected from Group C ^X optionally may be C3-C6 cycloalkyl group having a group, one or more substituents phenyl group which may have a selected from the group F ^X, have one or more substituents selected from the group F ^X A group consisting of a 5-6 membered aromatic heterocyclic group, a halogen atom, a nitro group and a cyano group, which may be
Group B ^X: 1 or more halogen atoms optionally may C1-C6 alkylthio group which may have one or more substituents phenyl group which may have a selected from the group F ^X, 1 is selected from the group F ^X A group consisting of a 5-6 membered aromatic heterocyclic group, a halogen atom, a nitro group and a cyano group, which may have the above substituents.
Group C ^X: a halogen atom, the group consisting of a nitro group and a cyano group.
Group D ^X: 1 or more substituents optionally may C1-C6 alkyl group which may have one or more substituents may C3-C6 cycloalkyl which may have a selected from the group C ^X selected from the group C ^X An alkyl group, a C1-C6 alkoxy group optionally having one or more halogen atoms, a C3-C6 alkenyloxy group optionally having one or more halogen atoms, and having one or more halogen atoms. A C3-C6 alkynyloxy group, a C1-C6 alkylthio group optionally having one or more halogen atoms, a C1-C6 alkylsulfonyloxy group optionally having one or more halogen atoms, a halogen atom, A group consisting of a cyano group, a nitro group, a hydroxy group and an amino group.
Group E ^X : may have one or more substituents selected from group C ^X (C1-C6 alkyl) carbonylamino group, may have one or more substituents selected from group C ^X (C1-C6 alkyl) aminocarbonyl group, one or more may have a substituent di (C1-C6 alkyl) aminocarbonyl group, one or more substituents selected from the group C ^X selected from the group C ^X the a and may C1-C6 alkylsulfonylamino group, one or more may C1-C6 be substituted alkylaminosulfonyl group selected from the group C ^X, one or more selected from the group C ^X A group consisting of a di (C1-C6 alkyl) aminosulfonyl group, a hydroxy group and an amino group, which may have a substituent.
Group F ^X : A group consisting of a C1-C6 alkyl group optionally having one or more halogen atoms, a C1-C6 alkoxy group optionally having one or more halogen atoms, a halogen atom and a cyano group.
Group G ^X : C1-C6 alkoxy group optionally having one or more halogen atoms, C1-C6 alkylthio group optionally having one or more halogen atoms, one or more substitutions selected from Group C ^X optionally may be C3-C6 cycloalkyl group having a group, one or more substituents phenyl group which may have a selected from the group F ^X, have one or more substituents selected from the group F ^X A group consisting of a 5-membered aromatic heterocyclic group, a halogen atom, a nitro group, and a cyano group, which may be ]
(Hereinafter referred to as the present compound).
[3] G ^X is a benzene ring optionally having one or more substituents selected from the group consisting of a halogen atom and a C1-C6 alkyl group,
The combination of L ^X, X ^X and R ^2X is,
L ^X is C a (O), X ^X is a NR ^3X or an oxygen atom, R ^2X is C1-C6 alkyl group, or a combination of a hydrogen atom or halogen atom, or L ^X is S (O) ₂ , X ^X is NR ^3X , R ^2X is a combination of a C1-C6 alkyl group or a halogen atom,
R ^1X is a C1-C6 alkyl group, a hydrogen atom or a halogen atom,
R ^3X may have one or more substituents selected from group A ^X, and may have one or more substituents selected from group A ^X, C3-C6 alkynyl group, one or more halogen atoms optionally may C1-C6 alkoxy group which may have one or more substituents have may be C3-C6 cycloalkyl group selected from the group D ^X, selected from the group D ^X is one or more substituents phenyl group which may have a one or more 6-membered aromatic or substituted heterocyclic group or a hydrogen atom selected from the group D ^X to be,
Z ^X is 1 or more may C3-C6 have a substituent of the cycloalkyl group, one or more substituents phenyl group which may have a selected from the group D ^X selected from the group D ^X, A 6-membered aromatic heterocyclic group ^optionally having one or more substituents selected from the group D ^X , CR ^4X R ^5X R ^6X , NR ^7X R ^8X or OR ^9X , or
X ^X and Z ^X together with L ^{X to} which they are attached may have a 5-6 membered heterocycle (the 5-6 membered heterocycle may have one or more substituents selected from group D ^X Good) and
Z ^X -L ^X -X ^X- (CR ^1X R ^2X ) _m on G ^X is bonded to the meta or para position with respect to the oxadiazole ring,
R ^4X, R ^5X and R ^6X are the same or different phases, one or more substituents optionally may C1-C6 alkyl group which may have a selected from the group consisting of the group A ^X and the group E ^X, from the group A ^X C3-C6 alkynyl group optionally having one or more substituents selected, C1-C6 alkoxy group optionally having one or more substituents selected from group B ^X , selected from group D ^X 1 or may C3-C6 have a substituent of the cycloalkyl group, one or more substituents phenyl group which may have a selected from the group D ^X, one or more substituents selected from the group D ^X A 5-6 membered aromatic heterocyclic group optionally having a group, a hydrogen atom, a halogen atom or a cyano group,
R ^7X and R ^8X are the same or different and are a C1-C6 alkyl group optionally having one or more substituents selected from the group consisting of group A ^X and group E ^X , 1 selected from group A ^X A C3-C6 alkynyl group optionally having one or more substituents, a C1-C6 alkoxy group optionally having one or more halogen atoms, and one or more substituents selected from the group D ^X. An optionally substituted C3-C6 cycloalkyl group, a phenyl group optionally having one or more substituents selected from group D ^X , and an optionally substituted one or more substituents selected from group D ^X 5 A 6-membered aromatic heterocyclic group or a hydrogen atom, or R ^7X and R ^8X together with the nitrogen atom to which they are bonded (the 3-6-membered heterocyclic ring is have one or more substituents selected from the group D ^X forms also may), The compound according to 2].
[4] G ^X is a benzene ring optionally having one or more halogen atoms,
m is 1,
The combination of L ^X, X ^X and R ^2X is,
L ^X is C (O), X ^X is an oxygen atom, R ^2X is a combination of hydrogen atoms, or L ^X is S (O) ₂ , X ^X is NR ^3X , R ^2X Is a C1-C3 alkyl group,
R ^1X is a hydrogen atom,
R ^3X is a hydrogen atom,
Z ^X is CR ^4X R ^5X R ^6X or NR ^7X R ^8X ;
G ^X on the ^{Z X -L X -X X - (} CR 1X R 2X) m is attached at the para position relative to the oxadiazole ring,
R ^4X , R ^5X and R ^6X are the same or different and are a C1-C6 alkyl group or a hydrogen atom,
R ^7X and R ^8X are the same or different and have a C1-C6 alkyl group (the C1-C6 alkyl group has one or more substituents selected from the group consisting of a cyano group and a C1-C3 alkoxy group). Or the compound according to [2], which is a C3-C6 cycloalkyl group.
[5] A pest control agent containing the compound according to [2], [3] or [4] (hereinafter referred to as the present invention control agent).
[6] A method for controlling pests by treating a plant or soil with an effective amount of the compound according to [2], [3] or [4].
[7] Use of the compound according to [2], [3] or [4] for controlling pests.
[8] One or more selected from the group consisting of bactericidal active ingredients, insecticidal active ingredients, acaricidal active ingredients, nematicidal active ingredients and plant growth regulating ingredients, and [2], [3] or [4] A composition containing a compound.

According to the present invention, plant diseases can be controlled.

The substituents in this specification will be described.
In this specification, when a substituent has two or more halogen atoms, those halogen atoms may be the same or different from each other.
In the present specification, “may have one or more substituents selected from group X” (X is any one of A to F or a combination thereof, or any one of A ^X to G ^X or The expression “means a combination thereof”, when two or more substituents selected from group X are present, may be the same or different.
In the present specification, the expression “CY-CW” means that the number of carbon atoms is Y to W. For example, the notation “C1-C6” means 1 to 6 carbon atoms.

The halogen atom represents a fluorine atom, a chlorine atom, a bromine atom or an iodine atom.
Examples of the “alkyl group” include methyl group, ethyl group, propyl group, isopropyl group, 1,1-dimethylpropyl group, 1,2-dimethylpropyl group, 1-ethylpropyl group, butyl group, isobutyl group, tert- A butyl group, a pentyl group, and a hexyl group are mentioned.
Examples of the “alkenyl group” include a vinyl group, 1-propenyl group, 2-propenyl group, 1-methyl-1-propenyl group, 1-methyl-2-propenyl group, 1,2-dimethyl-1-propenyl group, Examples include 1,1-dimethyl-2-propenyl group, 1-ethyl-1-propenyl group, 1-ethyl-2-propenyl group, 3-butenyl group, 4-pentenyl group and 5-hexenyl group.
Examples of the “alkynyl group” include ethynyl group, 1-propynyl group, 2-propynyl group, 1-methyl-2-propynyl group, 1,1-dimethyl-2-propynyl group, 1-ethyl-2-propynyl group, Examples thereof include 2-butynyl group, 4-pentynyl group and 5-hexynyl group.
“5-6-membered aromatic heterocyclic group” means a 5-membered aromatic heterocyclic group or a 6-membered aromatic heterocyclic group, and the 5-membered aromatic heterocyclic group means a pyrrolyl group, a furyl group, a thienyl group, A pyrazolyl group, an imidazolyl group, a triazolyl group, a tetrazolyl group, an oxazolyl group, an isoxazolyl group, a thiazolyl group, an isothiazolyl group, an oxadiazolyl group, or a thiadiazolyl group. Or represents a pyrazinyl group.
“3-6-membered non-aromatic heterocyclic group” means oxirane group, oxacyclobutane group, tetrahydrofuran group, pyran group, dihydropyran group, aziridine group, azacyclobutane group, pyrrolidine group, piperidine group, oxazoline group, Represents an isoxazoline group, a thiazoline group, or an isothiazoline group;

The “cycloalkyl group” represents a cyclopropyl group, a cyclobutyl group, a cyclopentyl group, or a cyclohexyl group.
The “3-7 membered cycloalkylene group” represents any one of the structures shown below (ZAA1 to ZAA5) (● represents a bonding position).

Examples of the “3-7 membered saturated heterocyclic group” include an oxirane ring, oxetane ring, oxolane ring, oxane ring, oxepane ring, thiirane ring, thietane ring, thiolane ring, thiane ring, thiepan ring, 1,3-dioxolane ring. 1,3-dioxane ring, 1,3-dithiolane ring, and 1,3-dithiane ring.

“R ⁷ and R ⁸ together with the nitrogen atom to which they are attached form a 3-8 membered heterocycle” and “R ^7X and R ^8X are together with the nitrogen atom to which they are attached, 3- The “8-membered heterocycle” in the “form 8-membered heterocycle” represents any of the structures shown in the following (ZC1 to ZC21) (● represents the bonding position).

“X and Z together with L to which they are attached form a 4-7 membered heterocycle” and “X ^X and Z ^X together with L ^{X to} which they are attached are 4-7 membered heterocycles. The “4-7 membered heterocycle” in “form a ring” represents, for example, any one of the structures shown below (ZF1 to ZF22) (• represents a bonding position).

The compound of the present invention may have one or more stereoisomers. Stereoisomers include enantiomers, diastereomers, atropisomers and geometric isomers. The present invention includes each stereoisomer and any ratio of stereoisomer mixtures.

The compound of the present invention is mixed with an acid such as hydrochloric acid, sulfuric acid, nitric acid, phosphoric acid, acetic acid or benzoic acid, thereby adding an acid addition salt such as hydrochloride, sulfate, nitrate, phosphate, acetate or benzoate. May form.

Examples of the compound of the present invention include the following compounds.

[Aspect 1] In the compound of the present invention, G ^X is a benzene ring optionally having one or more fluorine atoms,
In the combination of L ^X , X ^X and R ^2X , L ^X is C (O), X ^X is NR ^3X or an oxygen atom, R ^2X is a C1-C6 alkyl group, hydrogen atom or halogen atom A combination, or a combination in which L ^X is S (O) ₂ , X ^X is NR ^3X , and R ^2X is a C1-C6 alkyl group or a halogen atom,
R ^1X is a C1-C6 alkyl group, a hydrogen atom or a halogen atom,
R ^3X may have one or more substituents selected from group A ^X, and may have one or more substituents selected from group A ^X, C3-C6 alkynyl group, one or more halogen atoms optionally may C1-C6 alkoxy group which may have one or more substituents have may be C3-C6 cycloalkyl group selected from the group D ^X, selected from the group D ^X A phenyl group or a hydrogen atom optionally having one or more substituents,
Z ^X is a C3-C6 cycloalkyl group, a phenyl group, a 6-membered aromatic heterocyclic group (the C3-C6 cycloalkyl group, the phenyl group, and the 6-membered aromatic heterocyclic group are selected from the group D ^X CR ^4X R ^5X R ^6X , NR ^7X R ^8X or OR ^9X , or X ^X and Z ^X together with L ^{X to} which they are attached. To form a 5-6 membered heterocycle (the 5-6 membered heterocycle may have one or more substituents selected from group D ^X ),
Z ^X -L ^X -X ^X- (CR ^1X R ^2X ) _m on G ^X is bonded to the para position with respect to the oxadiazole ring,
R ^4X, R ^5X and R ^6X are the same or different phases, one or more substituents optionally may C1-C6 alkyl group which may have a selected from the group consisting of the group A ^X and the group E ^X, from the group A ^X C3-C6 alkynyl group optionally having one or more substituents selected, C1-C6 alkoxy group optionally having one or more substituents selected from group B ^X , selected from group D ^X 1 or may C3-C6 have a substituent of the cycloalkyl group, one or more substituents phenyl group which may have a selected from the group D ^X, one or more substituents selected from the group D ^X A 5-6 membered aromatic heterocyclic group optionally having a group, a hydrogen atom, a halogen atom or a cyano group,
R ^7X and R ^8X are the same or different and are a C1-C6 alkyl group optionally having one or more substituents selected from the group consisting of group A ^X and group E ^X , 1 selected from group A ^X A C3-C6 alkynyl group optionally having one or more substituents, a C1-C6 alkoxy group optionally having one or more halogen atoms, and one or more substituents selected from the group D ^X. An optionally substituted C3-C6 cycloalkyl group, a phenyl group optionally having one or more substituents selected from group D ^X , and an optionally substituted one or more substituents selected from group D ^X 5 A 6-membered aromatic heterocyclic group or a hydrogen atom, or R ^7X and R ^8X together with the nitrogen atom to which they are bonded (the 3-6-membered heterocyclic ring is compounds that form may) have one or more substituents selected from the group D ^X
[Aspect 2] In aspect 1, G ^X is a benzene ring,
L ^X is S (O) ₂ , X ^X is NR ^3X , R ^2X is a C1-C6 alkyl group or a halogen atom,
Z ^X is a C3-C6 cycloalkyl group, CR ^4X R ^5X R ^6X or NR ^7X R ^8X which may have one or more substituents selected from group D ^X ;
R ^4X , R ^5X and R ^6X are the same or different and are each a C1-C6 alkyl group optionally having one or more substituents selected from the group consisting of group A ^X and group E ^X, from group D ^X A C3-C6 cycloalkyl group optionally having one or more selected substituents, a hydrogen atom or a halogen atom,
A compound in which R ^7X and R ^8X are the same or different and each is a C1-C6 alkyl group optionally having one or more substituents selected from the group consisting of Group A ^X and Group E ^X.
[Aspect 3] In Aspect 1, G ^X is a benzene ring,
L ^X is S (O) ₂ , X ^X is NR ^3X , R ^2X is a C1-C6 alkyl group or a halogen atom,
R ^3X is a C1-C6 alkyl group, a C3-C6 alkynyl group or a C3-C6 cycloalkyl group ^optionally having one or more halogen atoms,
Z ^X is a C3-C6 cycloalkyl group, CR ^4X R ^5X R ^6X or NR ^7X R ^8X ;
R ^4X , R ^5X and R ^6X are the same or different and each is a C1-C6 alkyl group, a C3-C6 cycloalkyl group, a hydrogen atom or a halogen atom which may have one or more halogen atoms,
A compound in which R ^7X and R ^8X are the same or different and are a C1-C6 alkyl group.
[Aspect 4] In the compound of the present invention, G ^X is a benzene ring optionally having one or more fluorine atoms,
L ^X is C (O), X ^X is an oxygen atom, R ^1X and R ^2X are the same or different and are a C1-C6 alkyl group, a hydrogen atom or a halogen atom,
m is 1, Z ^X is NR ^7X R ^8X ,
Z ^X -L ^X -X ^X- (CR ^1X R ^2X ) _m on G ^X is bonded to the meta or para position with respect to the oxadiazole ring,
R ^7X and R ^8X are the same or different and are a C1-C6 alkyl group optionally having one or more substituents selected from the group consisting of group A ^X and group E ^X , 1 selected from group A ^X A C3-C6 alkynyl group optionally having one or more substituents, a C1-C6 alkoxy group optionally having one or more halogen atoms, and one or more substituents selected from the group D ^X. An optionally substituted C3-C6 cycloalkyl group, a phenyl group optionally having one or more substituents selected from group D ^X , and an optionally substituted one or more substituents selected from group D ^X 5 A 6-membered aromatic heterocyclic group or a hydrogen atom, or R ^7X and R ^8X together with the nitrogen atom to which they are bonded (the 3-6-membered heterocyclic ring is compounds that form may) have one or more substituents selected from the group D ^X
[Aspect 5] In Aspect 4, G ^X is a benzene ring,
R ^1X and R ^2X are hydrogen atoms,
A compound in which Z ^X -L ^X -X ^X- (CR ^1X R ^2X ) _m is bonded to the para position relative to the oxadiazole ring on G ^X.
[Aspect 6] In Aspect 4, R ^1X is a hydrogen atom, R ^2X is a hydrogen atom or a methyl group,
R ^7X and R ^8X are the same or different and each may have one or more substituents selected from the group consisting of group A ^X and group E ^{X, a} C1-C6 alkyl group, a C3-C6 alkenyl group, C3 -C6 alkynyl group, C1-C6 alkoxy group, C3-C6 cycloalkyl group, phenyl group or a hydrogen atom, or R ^7X and R ^8X together with the nitrogen atom to which they are attached A compound that forms a membered heterocycle (the 5-6 membered heterocycle may have one or more substituents selected from group D ^X ).
[Aspect 7] In aspect 4, G ^X is a benzene ring,
R ^1X and R ^2X are hydrogen atoms,
Z ^X -L ^X -X ^X- (CR ^1X R ^2X ) _m on G ^X is bonded to the para position with respect to the oxadiazole ring,
R ^7X and R ^8X are the same or different and each may have one or more substituents selected from the group consisting of group A ^X and group E ^{X, a} C1-C6 alkyl group, a C3-C6 alkenyl group, C3 -C6 alkynyl group, C1-C6 alkoxy group, C3-C6 cycloalkyl group, phenyl group or a hydrogen atom, or R ^7X and R ^8X together with the nitrogen atom to which they are attached A compound that forms a membered heterocycle (the 5-6 membered heterocycle may have one or more substituents selected from group D ^X ).
[Aspect 8] In Aspect 4, R ^1X is a hydrogen atom, R ^2X is a hydrogen atom or a methyl group,
R ^7X and R ^8X are the same or different and each may have one or more substituents selected from the group consisting of a C1-C3 alkoxy group and a cyano group, a C1-C6 alkyl group, a C3-C6 cycloalkyl group Or a compound which is a hydrogen atom.
[Aspect 9] In Aspect 4, G ^X is a benzene ring,
R ^1X and R ^2X are hydrogen atoms,
Z ^X -L ^X -X ^X- (CR ^1X R ^2X ) _m on G ^X is bonded to the para position with respect to the oxadiazole ring,
R ^7X and R ^8X are the same or different and each may have one or more substituents selected from the group consisting of a C1-C3 alkoxy group and a cyano group, a C1-C6 alkyl group, a C3-C6 cycloalkyl group Or a compound which is a hydrogen atom.
[Aspect 10] In the compound of the present invention, G ^X is a benzene ring optionally having one or more fluorine atoms,
L ^X is C (O), X ^X is NR ^3X , R ^1X and R ^2X are the same or different and are a C1-C6 alkyl group, a hydrogen atom or a halogen atom, and m is 1 or 2 Yes,
R ^3X may have one or more substituents selected from group A ^X, and may have one or more substituents selected from group A ^X, C3-C6 alkynyl group, one or more halogen atoms optionally may C1-C6 alkoxy group which may have one or more substituents have may be C3-C6 cycloalkyl group selected from the group D ^X, selected from the group D ^X is one or more substituents phenyl group which may have a one or more 6-membered aromatic or substituted heterocyclic group or a hydrogen atom selected from the group D ^X to be,
Z ^X is CR ^4X R ^5X R ^6X , NR ^7X R ^8X or OR ^9X , or
X ^X and Z ^X together with L ^{X to} which they are attached may have a 5-6 membered heterocycle (the 5-6 membered heterocycle may have one or more substituents selected from group D ^X Good) and
Z ^X -L ^X -X ^X- (CR ^1X R ^2X ) _m on G ^X is bonded to the meta or para position with respect to the oxadiazole ring,
R ^4X, R ^5X and R ^6X are the same or different phases, one or more substituents optionally may C1-C6 alkyl group which may have a selected from the group consisting of the group A ^X and the group E ^X, from the group A ^X C3-C6 alkynyl group optionally having one or more substituents selected, C1-C6 alkoxy group optionally having one or more substituents selected from group B ^X , selected from group D ^X 1 or may C3-C6 have a substituent of the cycloalkyl group, one or more substituents phenyl group which may have a selected from the group D ^X, one or more substituents selected from the group D ^X A 5-6 membered aromatic heterocyclic group optionally having a group, a hydrogen atom, a halogen atom or a cyano group,
R ^7X and R ^8X are the same or different and are a C1-C6 alkyl group optionally having one or more substituents selected from the group consisting of group A ^X and group E ^X , 1 selected from group A ^X A C3-C6 alkynyl group optionally having one or more substituents, a C1-C6 alkoxy group optionally having one or more halogen atoms, and one or more substituents selected from the group D ^X. An optionally substituted C3-C6 cycloalkyl group, a phenyl group optionally having one or more substituents selected from group D ^X , and an optionally substituted one or more substituents selected from group D ^X 5 A 6-membered aromatic heterocyclic group or a hydrogen atom, or R ^7X and R ^8X together with the nitrogen atom to which they are bonded (the 3-6-membered heterocyclic ring is One or more substituents selected from the group D ^X may be formed),
R ^9X is 1 or more substituents optionally may C1-C3 alkyl group which may have a selected from the group consisting of the group E ^X and the group G ^X, have one or more substituents selected from the group A ^X An optionally substituted C3-C6 alkenyl group, a C3-C6 alkynyl group optionally having one or more substituents selected from group A ^X , and one or more substituents selected from group D ^X good C3-C6 cycloalkyl group optionally substituted with one or more substituents phenyl group which may have a one or more substituents selected from the group D ^X is selected from the group D ^X 5-6 A compound which is a membered aromatic heterocyclic group or a hydrogen atom.
[Aspect 11] In aspect 10, G ^X is a benzene ring,
A compound in which R ^1X and R ^2X are a hydrogen atom and m is 1.
[Aspect 12] In Aspect 10, R ^1X is a hydrogen atom, R ^2X is a hydrogen atom or a methyl group,
R ^3X is 1 or more substituents optionally may C1-C6 alkyl group which may have a selected from the group A ^X, C3-C6 alkynyl group, C1-C6 alkoxy group, C3-C6 cycloalkyl group, a phenyl group or A hydrogen atom,
R ^4X , R ^5X and R ^6X are the same or different and each may have one or more substituents selected from the group consisting of group A ^X and group E ^X, C1-C6 alkenyl group, C3-C6 alkenyl A group, a C3-C6 alkynyl group, a C1-C6 alkoxy group, a C3-C6 cycloalkyl group, a phenyl group, a hydrogen atom, a halogen atom or a cyano group,
R ^7X and R ^8X are the same or different and each may have one or more substituents selected from the group consisting of group A ^X and group E ^{X, a} C1-C6 alkyl group, a C3-C6 alkenyl group, C3 -C6 alkynyl group, C1-C6 alkoxy group, C3-C6 cycloalkyl group, phenyl group or a hydrogen atom, or R ^7X and R ^8X together with the nitrogen atom to which they are attached Forming a membered heterocycle (wherein the 5-6 membered heterocycle may have one or more substituents selected from group D ^X );
R ^9X may have one or more substituents selected from the group consisting of group E ^X and group G ^X, C1-C3 alkyl group, C3-C6 alkenyl group, C3-C6 alkynyl group, C3-C6 A compound which is a cycloalkyl group, a phenyl group or a hydrogen atom.
[Aspect 13] In Aspect 10, G ^X is a benzene ring,
R ^1X and R ^2X are hydrogen atoms, m is 1,
R ^3X is 1 or more substituents optionally may C1-C6 alkyl group which may have a selected from the group A ^X, C3-C6 alkynyl group, C1-C6 alkoxy group, C3-C6 cycloalkyl group, a phenyl group or A hydrogen atom,
Z ^X -L ^X -X ^X- (CR ^1X R ^2X ) _m on G ^X is bonded to the para position with respect to the oxadiazole ring,
R ^4X , R ^5X and R ^6X are the same or different and each may have one or more substituents selected from the group consisting of group A ^X and group E ^X, C1-C6 alkenyl group, C3-C6 alkenyl A group, a C3-C6 alkynyl group, a C1-C6 alkoxy group, a C3-C6 cycloalkyl group, a phenyl group, a hydrogen atom, a halogen atom or a cyano group,
R ^7X and R ^8X are the same or different and each may have one or more substituents selected from the group consisting of group A ^X and group E ^{X, a} C1-C6 alkyl group, a C3-C6 alkenyl group, C3 -C6 alkynyl group, C1-C6 alkoxy group, C3-C6 cycloalkyl group, phenyl group or a hydrogen atom, or R ^7X and R ^8X together with the nitrogen atom to which they are attached Forming a membered heterocycle (wherein the 5-6 membered heterocycle may have one or more substituents selected from group D ^X );
R ^9X may have one or more substituents selected from the group consisting of group E ^X and group G ^X, C1-C3 alkyl group, C3-C6 alkenyl group, C3-C6 alkynyl group, C3-C6 A compound which is a cycloalkyl group, a phenyl group or a hydrogen atom.
[Aspect 14] In Aspect 10, R ^1X is a hydrogen atom, R ^2X is a hydrogen atom or a methyl group, m is 1,
R ^3X is 1 or more substituents optionally C1-C6 may be alkyl groups having a selected from the group A ^X, a phenyl group or a hydrogen atom,
Z ^X is CR ^4X R ^5X R ^6X or OR ^9X , or X ^X and Z ^X are taken together with L ^{X to} which they are attached to form a 5-6 membered heterocycle (the 5-6 membered heterocycle forms may) have one or more substituents selected from the group D ^X,
Z ^X -L ^X -X ^X- (CR ^1X R ^2X ) _m on G ^X is bonded to the para position with respect to the oxadiazole ring,
R ^4X , R ^5X and R ^6X are the same or different and are a C1-C6 alkyl group, a C3-C6 cycloalkyl group, a phenyl group, a hydrogen atom or a halogen atom,
A compound wherein R ^9X is a C1-C3 alkyl group or a phenyl group optionally having one or more substituents selected from the group consisting of group G ^X.
[Aspect 15] In Aspect 10, G ^X is a benzene ring,
R ^1X and R ^2X are hydrogen atoms, m is 1,
R ^3X is 1 or more substituents optionally C1-C6 may be alkyl groups having a selected from the group A ^X, a phenyl group or a hydrogen atom,
Z ^X is CR ^4X R ^5X R ^6X or OR ^9X , or X ^X and Z ^X together with L ^{X to} which they are attached form a pyrrolidinone ring or piperidinone ring,
Z ^X -L ^X -X ^X- (CR ^1X R ^2X ) _m on G ^X is bonded to the para position with respect to the oxadiazole ring,
R ^4X , R ^5X and R ^6X are the same or different and are a C1-C6 alkyl group, a C3-C6 cycloalkyl group, a phenyl group, a hydrogen atom or a halogen atom,
A compound wherein R ^9X is a C1-C3 alkyl group or a phenyl group optionally having one or more substituents selected from the group consisting of group G ^X.
[Aspect 16] In the compound of the present invention, G ^X is a benzene ring optionally having one or more fluorine atoms,
L ^X is C (O), X ^X is NR ^3X or an oxygen atom, R ^1X is a hydrogen atom, R ^2X is a hydrogen atom or a methyl group, m is 1,
R ^3X is 1 or more substituents optionally C1-C6 may be alkyl groups having a selected from the group A ^X, a phenyl group or a hydrogen atom,
Z ^X is CR ^4X R ^5X R ^6X , NR ^7X R ^8X or OR ^9X , or X ^X and Z ^X together with L ^{X to} which they are attached are 5-6 membered heterocycles The 5-6 membered heterocyclic ring may have one or more substituents selected from group D ^X ),
Z ^X -L ^X -X ^X- (CR ^1X R ^2X ) _m on G ^X is bonded to the para position with respect to the oxadiazole ring,
R ^4X , R ^5X and R ^6X are the same or different and are a C1-C6 alkyl group, a C3-C6 cycloalkyl group, a phenyl group, a hydrogen atom or a halogen atom,
R ^7X and R ^8X are the same or different and each may have one or more substituents selected from the group consisting of a C1-C3 alkoxy group and a cyano group, a C1-C6 alkyl group, a C3-C6 cycloalkyl group Or a hydrogen atom,
A compound wherein R ^9X is a C1-C3 alkyl group or a phenyl group optionally having one or more substituents selected from the group consisting of group G ^X.
[Aspect 17] In Aspect 16, G ^X is a benzene ring,
R ^2X is a hydrogen atom,
R ^3X is a C1-C6 alkyl group optionally having one or more halogen atoms, a phenyl group, or a hydrogen atom,
Z ^X is CR ^4X R ^5X R ^6X , NR ^7X R ^8X, or OR ^9X , or X ^X and Z ^X together with L ^{X to} which they are attached, a pyrrolidinone ring or piperidinone ring Form the
A compound in which R ^9X is a C1-C3 alkyl group or a phenyl group.

Next, a method for producing this compound will be described.

This compound can be produced by the following production method and the like.

Manufacturing method A
This compound can be produced by reacting a compound represented by formula (A1) (hereinafter referred to as compound (A1)) with trifluoroacetic anhydride in the presence of a base.

[Wherein the symbols have the same meaning as described above. ]
The reaction is usually performed in a solvent. Examples of the solvent used in the reaction include hydrocarbons such as hexane, cyclohexane, toluene and xylene (hereinafter referred to as hydrocarbons), diethyl ether, tetrahydrofuran, 1,4-dioxane, ethylene glycol dimethyl ether, methyl tert- Ethers such as butyl ether and diisopropyl ether (hereinafter referred to as ethers), halogenated hydrocarbons such as chloroform, dichloromethane and chlorobenzene (hereinafter referred to as halogenated hydrocarbons), dimethylformamide (hereinafter referred to as DMF). ), Amides such as 1,3-dimethyl-2-imidazolidinone and N-methylpyrrolidone (hereinafter referred to as amides), esters such as methyl acetate and ethyl acetate (hereinafter referred to as esters), acetonitrile , Propionitrile, etc. Lil (hereinafter, referred to as nitriles.), Water and mixtures thereof.
Examples of the base used in the reaction include organic bases such as triethylamine, pyridine, 2,2′-bipyridine, diazabicycloundecene (hereinafter referred to as organic bases), carbonates such as sodium carbonate and potassium carbonate ( Hereinafter, it is referred to as carbonates.), And bicarbonates such as sodium bicarbonate and potassium bicarbonate (hereinafter referred to as bicarbonates).
For the reaction, trifluoroacetic anhydride is usually used in a proportion of 1 to 10 mol, and base is usually used in a proportion of 1 to 10 mol, relative to 1 mol of compound (A1).
The reaction temperature is usually in the range of −20 to 150 ° C. The reaction time is usually in the range of 0.1 to 120 hours.
After completion of the reaction, the compound can be isolated by mixing the reaction mixture with water and extracting with an organic solvent, and subjecting the organic layer to post-treatment operations such as drying and concentration.

Manufacturing method B
A compound represented by formula (2A2) (hereinafter referred to as compound (2A2)) is a compound represented by formula (2A1) (hereinafter referred to as compound (2A1)) and a compound represented by formula (M1) ( Hereinafter, it can be produced by reacting the compound (M1)) in the presence of a base.

[Wherein, X ¹ represents a leaving group such as a chlorine atom, a bromine atom, an iodine atom, a methanesulfonyloxy group, a trifluoromethanesulfonyloxy group, and other symbols have the same meaning as described above. ]
The reaction is usually performed in a solvent. Examples of the solvent used in the reaction include hydrocarbons, ethers, halogenated hydrocarbons, amides, esters, nitriles, methanol and ethanol and other alcohols (hereinafter referred to as alcohols), water, and these. A mixture etc. are mentioned.
Examples of the base used in the reaction include organic bases, carbonates, hydrogen carbonates, and metal hydrides such as sodium hydride, potassium hydride, and lithium hydride (hereinafter referred to as metal hydrides). It is done.
In the reaction, compound (M1) is usually used in a proportion of 1 to 10 mol and base is used in a proportion of 1 to 10 mol with respect to 1 mol of compound (2A1).
The reaction temperature is usually in the range of −20 to 150 ° C. The reaction time is usually in the range of 0.1 to 120 hours.
After completion of the reaction, the compound (2A2) can be isolated by performing post-treatment operations such as extraction of the reaction mixture with water and extraction with an organic solvent, and drying and concentration of the organic layer.
The compound (M1) is known or can be produced according to a known method.

Manufacturing method C
A compound represented by formula (2A3) (hereinafter referred to as compound (2A3)) is a compound represented by formula (A3) (hereinafter referred to as compound (A3)) and a compound represented by formula (M3) ( Hereinafter, it can be produced by reacting the compound (M3) in the presence of a base.

[Wherein, Z ¹ represents NR ⁷ R ⁸ or OR ⁹ , and other symbols have the same meaning as described above. ]
The reaction is usually performed in a solvent. Examples of the solvent used in the reaction include hydrocarbons, ethers, halogenated hydrocarbons, amides, esters, nitriles, water, and mixtures thereof.
When Z ¹ is NR ⁷ R ⁸ , the compound (M3) may be in the form of an acid addition salt. Examples of the acid addition salt of compound (M3) include hydrochloride and sulfate.
Examples of the base used in the reaction include organic bases, alkali metal hydroxides such as sodium hydroxide and potassium hydroxide (hereinafter referred to as alkali metal hydroxides), carbonates, and bicarbonates. It is done.
In the reaction, with respect to 1 mol of compound (A3), compound (M3) is usually used at a ratio of 1 to 10 mol, and base is used at a ratio of 1 to 10 mol.
The reaction temperature is usually in the range of −20 to 150 ° C. The reaction time is usually in the range of 0.1 to 120 hours.
After completion of the reaction, the compound (2A3) can be isolated by performing post-treatment operations such as mixing the reaction mixture with water, extracting with an organic solvent, and drying and concentrating the organic layer.
Compound (M3) is publicly known or can be produced according to a publicly known method.

Manufacturing method D
A compound represented by formula (2A4) (hereinafter referred to as compound (2A4)) is a compound represented by formula (A3-2) (hereinafter referred to as compound (A3-2)) and formula (M4). It can be produced by reacting the compound shown below (hereinafter referred to as compound (M4)) in the presence of a base or a Lewis acid.

[Wherein the symbols have the same meaning as described above. ]
The reaction is usually performed in a solvent. Examples of the solvent used in the reaction include hydrocarbons, ethers, halogenated hydrocarbons, amides, esters, nitriles, and mixtures thereof.
Examples of the base used in the reaction include organic bases, carbonates, bicarbonates, and metal hydrides.
Examples of the Lewis acid used in the reaction include aluminum (III) oxide.
In the reaction, compound (M4) is usually used in a proportion of 1 to 10 mol and base or Lewis acid is used in a proportion of 1 to 10 mol per 1 mol of compound (A3-2).
The reaction temperature is usually in the range of −20 to 150 ° C. The reaction time is usually in the range of 0.1 to 120 hours.
After completion of the reaction, the compound (2A4) can be isolated by performing post-treatment operations such as extraction of the reaction mixture with water and extraction with an organic solvent, and drying and concentration of the organic layer.
Compound (M4) is publicly known or can be produced according to a publicly known method.

Next, a method for producing the intermediate of this compound will be described.

Reference manufacturing method A
Compound (A1) can be produced by reacting a compound represented by formula (A2) with hydroxylamine.

[Wherein the symbols have the same meaning as described above. ]
The reaction can be carried out, for example, according to the method described in WO2009 / 081891.

Reference manufacturing method B
The compound represented by the formula (A2-2) is a compound represented by the formula (A2-3) (hereinafter referred to as the compound (A2-3)) and a compound represented by the formula (M2) (hereinafter referred to as the compound (M2 And) in the presence of a base.

[Wherein the symbols have the same meaning as described above. ]
The reaction can be carried out according to the method described in International Publication No. 2015/004282.
Compound (A2-3) is known or can be produced according to the method described in International Publication No. 2011/142356.
Compound (M2) is known or can be produced according to a known method.

Reference manufacturing method C
Compound (A3) can be produced by reacting compound (A3-2) with phosgene, diphosgene, or triphosgene in the presence of a base.

[Wherein the symbols have the same meaning as described above. ]
The reaction is usually performed in a solvent. Examples of the solvent used in the reaction include hydrocarbons, ethers, halogenated hydrocarbons, amides, esters, nitriles, water, and mixtures thereof.
Examples of the base used in the reaction include organic bases, alkali metal hydroxides, carbonates, and hydrogen carbonates.
In the reaction, with respect to 1 mol of compound (A3-2), phosgene is usually used at a ratio of 1 to 10 mol, and base is used at a ratio of 1 to 10 mol.
In the reaction, with respect to 1 mol of compound (A3-2), diphosgene is usually used at a ratio of 0.5 to 5 mol, and the base is used at a ratio of 1 to 10 mol.
In the reaction, with respect to 1 mol of compound (A3-2), triphosgene is usually used in a proportion of 0.3 to 3 mol, and the base is used in a proportion of 1 to 10 mol.
The reaction temperature is usually in the range of −20 to 150 ° C. The reaction time is usually in the range of 0.1 to 120 hours.
After completion of the reaction, the compound (A3) can be obtained by concentrating the reaction mixture. Moreover, you may use for the method as described in the manufacturing method C, without concentrating a reaction mixture.

Reference manufacturing method D
The compound (A3-2) is produced by reacting a compound represented by the formula (A3-3) (hereinafter referred to as the compound (A3-3)) and an acid in the presence of water or alcohols. be able to.

[Wherein the symbols have the same meaning as described above. ]
The reaction is usually carried out using water and / or alcohols as a solvent, but a solvent may be further added. Examples of such solvents include hydrocarbons, ethers, halogenated hydrocarbons, amides, esters, nitriles, and mixtures thereof.
Examples of the acid used in the reaction include hydrochloric acid, sulfuric acid, and paratoluenesulfonic acid.
In the reaction, the acid is usually used at a ratio of 1 to 1000 mol per 1 mol of the compound (A3-3).
The reaction temperature is usually in the range of −20 to 150 ° C. The reaction time is usually in the range of 0.1 to 120 hours.
After completion of the reaction, the compound (A3-2) can be isolated by performing post-treatment operations such as mixing of the reaction mixture with water and extraction with an organic solvent, and drying and concentration of the organic layer.

Reference manufacturing method E
Compound (A3-3) is produced by reacting a compound represented by formula (A1-2) (hereinafter referred to as Compound (A1-2)) with trifluoroacetic anhydride in the presence of a base. be able to.

[Wherein the symbols have the same meaning as described above. ]
The reaction can be carried out according to the method described in Production Method A.

Reference manufacturing method F
Compound (A1-2) can be produced by reacting a compound represented by formula (A2-4) (hereinafter referred to as compound (A2-4)) with hydroxylamine.

[Wherein the symbols have the same meaning as described above. ]
The reaction can be carried out, for example, according to the method described in WO2009 / 081891.

Reference manufacturing method G
Compound (A2-4) can be produced by reacting a compound represented by the formula (A2-5) (hereinafter referred to as compound (A2-5)) with chloromethyl methyl ether.

[Wherein the symbols have the same meaning as described above. ]
The reaction is described in, for example, J. Am. Chem. Soc. , 1977, 99, 1275.
Compound (A2-5) is publicly known or can be produced according to the method described in US Patent Application Publication No. 2007/270438.

Reference manufacturing method H
The compound represented by formula (A2-6) is a compound represented by formula (A4-1) (hereinafter referred to as compound (A4-1)) and a compound represented by formula (M5) (hereinafter referred to as compound (M5 And) in the presence of a base.

[Wherein the symbols have the same meaning as described above. ]
The reaction can be carried out according to the method described in Angew. Chem. Int. Ed., 2016, 55, 8452.
Compound (A4-1) is publicly known or can be produced according to the method described in International Publication No. 2011/142356.
Compound (M5) is publicly known or can be produced according to a publicly known method.

This compound is usually mixed with a solid carrier, liquid carrier, oil, and / or surfactant, etc., and if necessary, an adjuvant for formulation such as a sticking agent, a dispersing agent, a stabilizer and the like, It is formulated into granular wettable powder, flowable powder, granule, dry flowable liquid, emulsion, aqueous liquid, oil, smoke, aerosol, microcapsule and the like. These preparations contain the present compound in a weight ratio of usually 0.1 to 99%, preferably 0.2 to 90%.

The control agent of the present invention is usually prepared by mixing the compound of the present invention with a solid carrier, liquid carrier, oil, and / or surfactant, and if necessary, an auxiliary agent for formulation such as a fixing agent, a dispersant, a stabilizer and the like. Add, wettable powder, granular wettable powder, flowable powder, granule, dry flowable powder, emulsion, aqueous solution, oil, smoke, aerosol, microcapsule, poison bait, resin formulation, shampoo, It is formulated into paste-form preparations, foams, carbon dioxide preparations, tablets and the like. These preparations may be used after being processed into mosquito coils, electric mosquito mats, liquid mosquito traps, fumigants, fumigants, sheet preparations, spot-on agents, or oral treatments. These preparations contain the compound of the present invention in a weight ratio of usually 0.1 to 99%, preferably 0.2 to 90%.

Examples of the solid support include clays (for example, kaolin, diatomaceous earth, scissors clay, bentonite, acidic clay), dry silica, wet silica, talc, and other inorganic minerals (for example, sericite, quartz powder, sulfur powder, activated carbon). , Calcium carbonate) and the like.
Examples of the liquid carrier include water, alcohols, ketones (eg, acetone, methyl ethyl ketone, cyclohexanone), aromatic hydrocarbons (eg, benzene, toluene, xylene, ethylbenzene, methylnaphthalene), aliphatic hydrocarbons ( Examples thereof include n-hexane, kerosene), esters, nitriles, ethers, amides, and halogenated hydrocarbons.

Examples of the surfactant include alkyl sulfates, alkyl sulfonates, alkyl aryl sulfonates, alkyl aryl ethers and polyoxyethylene compounds thereof, polyoxyethylene glycol ethers, polyhydric alcohol esters, sugar alcohol derivatives. Is mentioned.

Examples of other formulation adjuvants include, for example, a fixing agent, a dispersant, and a stabilizer. Specifically, casein, gelatin, polysaccharides (for example, starch, arabic gum, cellulose derivatives, alginic acid), lignin derivatives, bentonite, Saccharides, synthetic water-soluble polymers (eg, polyvinyl alcohol, polyvinylpyrrolidone, polyacrylic acids), isopropyl acid phosphate, 2,6-di-tert-butyl-4-methylphenol, BHA (2-tert-butyl-4 -Mixtures of -methoxyphenol and 3-tert-butyl-4-methoxyphenol), vegetable oils, mineral oils, fatty acids or esters thereof.

In addition, the present compound may be used for controlling plant diseases by mixing with mineral oil, oil such as vegetable oil, or surfactant. The compound of the present invention may be used for controlling pests by mixing with oils such as mineral oil and vegetable oil, or surfactants. Oils that can be used in combination, or surfactants include Nimbus (registered trademark), Assist (registered trademark), Aureo (registered trademark), Iharol (registered trademark), Silwet L-77 (registered trademark), BreakThru ( (Registered trademark), Sundance II (registered trademark), Induce (registered trademark), Penetrator (registered trademark), AgriDex (registered trademark), Lutensol A8 (registered trademark), NP-7 (registered trademark), Triton (registered trademark), Nufilm (Registered trademark), Emulator NP7 (registered trademark), Emulad (registered trademark), TRITON X 45 (registered trademark), AGLAR 90 (registered trademark), AGROTIN (registered trademark), ARPON (registered trademark), EnSpray N (registered trademark) Mark), and BANOLE (registered trademark).

As a method of applying the present compound, the method is not particularly limited as long as the present compound can be applied. For example, seed treatment such as seed disinfection.
The method of applying the compound of the present invention is not particularly limited as long as the compound of the present invention can be applied. Treatment, seed treatment such as seed disinfection, treatment of harmful arthropods, and the like.

The application amount of the present compound or the present compound varies depending on weather conditions, formulation form, application time, application method, application location, target disease, target crop, etc. In the case of the treatment, the amount is usually 1 to 500 g, preferably 2 to 200 g per 1000 m ² . In the case of treating seeds, the amount of the present compound or the compound of the present invention is usually applied in the range of 0.001 to 100 g, preferably 0.01 to 50 g per 1 kg of seeds. Emulsions, wettable powders, suspensions and the like are usually diluted with water before use. In this case, the concentration of the present compound or the present compound after dilution is usually 0.0005 to 2% by weight, preferably 0. 0.005 to 2% by weight. Powders, granules and the like are usually applied as they are without dilution.

In addition, the present compound or the present compound can be used as a plant disease control agent in agricultural land such as fields, paddy fields, lawns, orchards. This compound or this invention compound can control the disease of the said agricultural land in the agricultural land etc. which grow the plant etc. which are mentioned below. Moreover, this invention compound can control the harmful arthropod of the said agricultural field.

Agricultural crops: corn, rice, wheat, barley, rye, oats, sorghum, cotton, soybean, peanuts, buckwheat, sugar beet, rapeseed, sunflower, sugarcane, tobacco, etc. Cucumber, pumpkin, zucchini, watermelon, melon, etc., cruciferous vegetables (radish, turnip, horseradish, coral rabi, cabbage, cabbage, mustard, broccoli, cauliflower, etc.), asteraceae vegetables ( Burdock, garlic, artichoke, lettuce, etc.), liliaceae vegetables (leek, onion, garlic, asparagus), celery vegetables (carrots, parsley, celery, American burdock etc.), red crustacean vegetables (spinach, chard, etc.), perilla Vegetables (Perilla, Mint, Basil) Etc.), strawberry, sweet potato, yam, taro, etc., flower bud, houseplant,
Fruit trees; pears (apples, pears, Japanese pears, quince, quince, etc.), nuclear fruits (peaches, plums, nectarines, ume, sweet cherry, apricots, prunes, etc.), citrus (satsuma mandarin, orange, lemon, lime, grapefruit) ), Nuts (chestnut, walnut, hazel, almond, pistachio, cashew nut, macadamia nut, etc.), berries (blueberry, cranberry, blackberry, raspberry, etc.), grape, oyster, olive, loquat, banana, coffee, Date palm, coconut palm, etc.
Trees other than fruit trees: Cha, mulberry, flowering trees, street trees (ash, birch, dogwood, eucalyptus, ginkgo, lilac, maple, oak, poplar, redwood, fu, sycamore, zelkova, black bean, peach tree, Tsuga, rat, pine, Spruce, yew) etc.

The above plants include genetically modified crops.

Examples of plant diseases that can be controlled by the present compound or the compound of the present invention include phytopathogenic fungi such as filamentous fungi and bacteria. Specific examples include, but are not limited to, the following: is not.

Rice blast (Magnaporthe grisea), sesame leaf blight (Cochliobolus miyabeanus), blight (Rhizoctonia solani), idiot seedling (Gibberella fujikuroi), yellow dwarf (Sclerophthora macrospora); wheat powdery mildew (Erysiphe) graminis), red mold (Fusarium graminearum, F. avenaceum, F. culmorum, Microdochium nivale), rust (Puccinia striiformis, P. graminis, P. recondita), red snow rot (Micronectriella nivale, M.majus), Snow rot microbe nuclei (Typhula sp.), Naked smut (Ustilago tritici), black scab (Tilletia caries, T. controversa), eye spot (Pseudocercosporella herpotrichoides), leaf blight (Septoria tritici), blight Diseases (Stagonospora nodorum), maculopathy (Pyrenophora tritici-repentis), Rhizoctonia solani, blight (Gaeumannomyces graminis); barley powdery mildew (Erysiphe graminis), red mold ( Fusarium gramine arum, F. avenaceum, F. culmorum, Microdochium nivale), rust disease (Puccinia striiformis, P.graminis, P.hordei), naked smut (Ustilago nuda), cloud disease (Rhynchosporium secalis), reticular disease (Pyrenophora teres) ), Spot disease (Cochliobolus sativus), leafy leaf disease (Pyrenophora graminea), lambaria disease (Ramularia collo-cygni), Rhizoctonia solani (Rhizoctonia solani); corn rust (Puccinia sorghi), southern rust Diseases (Puccinia polysora), soot rot (Setosphaeria turcica), tropical rust (Physopella zeae), sesame leaf blight (Cochliobolus heterostrophus), anthracnose (Colletotrichum graminicola), gray leaf spot disease (Cercospora zeae-maydis) , Brown spot disease (Kabatiella zeae), Phaeosfaeria reef spot disease (Phaeosphaeria maydis) diplodia disease (Stenocarpella maydis, Stenocarpella macrospora), Stokelot disease (Fusar) ium graminearum, Fusarium verticilioides, Colletotrichum graminicola), smut (Ustilago maydis); cotton anthracnose (Colletotrichum gossypii), mildew (Ramuraria areola), black spot (Alternaria macrospora, A. gossypii), Thielaviopsis Black root rot disease (Thielaviopsis basicola); Coffee rust (Hemileia vastatrix); Leaf spot disease (Cercospora coffeicola); Rapeseed sclerotia (Sclerotinia sclerotiorum); Black spot disease (Alternaria brassicae); lingam); sugarcane rust (Puccinia melanocephela, Puccinia kuehnii), smut (Ustilago scitaminea); sunflower rust (Puccinia helianthi), downy mildew (Plasmopara halstedii); citrus black spot (Diaporthe citri) Disease (Elsinoe fawcetti), fruit rot (Penicillium digitatum, P. italicum), plague (Phytophthora parasitica, Phytophthora citrophthora); apple monilinia (Monilinia) mali), rot (Valsa ceratosperma), powdery mildew (Podosphaera leucotricha), spotted leaf disease (Alternaria alternata apple pathotype), black star disease (Venturia inaequalis), anthracnose (Glomerella cingulata), brown spot disease (Diplocarpon mali) Botryosphaeria berengeriana, plague (Phytophtora cactorum); pear black spot (Venturia nashicola, V. pirina), black spot (Alternaria alternata Japanese pear pathotype), red star disease (Gymnosporangium haraeanum); Disease (Monilinia fructicola), black scab (Cladosporium carpophilum), phomopsis sp. (Phomopsis sp.); Grape black rot (Elsinoe ampelina), late rot (Glomerella cingulata), powdery mildew (Uncinula necator), rust (Phakopsora ampelopsidis), blacklot disease (Guignardia bidwellii), downy mildew (Plasmopara viticola); oyster anthracnose (Gloeosporium kaki), deciduous disease (Cercospora kaki, Mycosphaerella nawae) Colletotrichum lagenarium, powdery mildew (Sphaerotheca fuliginea), vine blight (Didymella bryoniae), brown spot (Corynespora cassiicola), vine split (Fusarium oxysporum), downy mildew (Pseudoperonospora cubensis) , Plague (Phytophthora sp.), Seedling blight (Pythium sp.); Tomato ring-rot (Alternaria solani), leaf mold (Cladosporium fulvum), subtilis (Pseudocercospora fuligena), plague (Phytophthora infestans), Powdery mildew (Leveillula taurica); eggplant brown spot (Phomopsis vexans), powdery mildew (Erysiphe cichoracearum); cruciferous vegetable black spot (Alternaria japonica), white spot (Cercosporella brassicae), clubroot (Plasmodiophora) brassicae), downy mildew (Peronospora parasitica); leek rust (Puccinia allii); soybean purpura (Cercospora kikuchii), black scab (Elsinoe glycines), black spot (Diaporthe phaseolorum var. sojae), Disease (Phakopsora pachyrhizi), brown ring disease (Corynespora cassiicola), anthrax (Colletotrithum glycines, C. truncatum), leaf rot (Rhizoctonia solani), brown leaf disease (Septoria glycines), spot disease (Cercospora sojina), fungus Nuclear disease (Sclerotinia sclerotiorum), powdery mildew (Microspaera diffusa), stem blight (Phytophthora sojae), downy mildew (Peronospora manshurica), sudden death (Fusarium virguliforme); bean sclerotia (Sclerotinia sclerotiorum), rust (Uromyces appendiculatus), horn spot disease (Phaeoisariopsis griseola), anthracnose (Colletotrichum lindemuthianum); groundnut black rot (Cercospora personata), brown spot disease (Cercospora arachidicola), silkworm disease (Sclerotium rolfsii); Erysiphe pisi; Potato summer plague (Alternaria solani), plague (Phytophthora infestans), scarlet rot (Phytophthora erythroseptica), powdery scab (Spongospora subterranea f. sp. subterranea), half body wilt disease (Verticillium albo-atrum, V. dahliae, V. nigrescens); Strawberry powdery mildew (Sphaerotheca humuli); Cha net rot (Exobasidium reticulatum), white spot disease (Elsinoe leucospila), Ring spot disease (Pestalotiopsis sp.), Anthracnose (Colletotrichum theae-sinensis); Tobacco red blight (Alternaria longipes), Anthracnose (Colletotrichum tabacum), Downy mildew (Peronospora tabacina), Plague (Phytophthora nicotianae); Sugar beet brown spot (Cercospora beticola), leaf rot (Thanatephorus cucumeris), root rot (Thanatephorus cucumeris), black root (Aphanomyces cochlioides); rose scab (Diplocarpon rosae), powdery mildew (Sphaerotheca pannosa) Chrysanthemum brown spot (Septoria chrysanthemi-indici), white rust (Puccinia horiana); onion white spot (Botrytis cinerea, B. byssoidea, B. squamosa), gray rot (Botrytis alli), small sclerotia Sexual rot (Botryt) is squamosa); various crops of gray mold (Botrytis cinerea), sclerotia (Sclerotinia sclerotiorum); radish black spot (Alternaria brassicicola); buckwheat dollar spot (Sclerotinia homoeocarpa), buckwheat brown patch disease and large Patch disease (Rhizoctonia solani); and banana sigatoka disease (Mycosphaerella fijiensis, Mycosphaerella musicola).
Seed disease or early growth of various crops caused by Aspergillus, Penicillium, Fusarium, Gibberella, Tricoderma, Thielaviopsis, Rhizopus, Mucor, Corticium, Phoma, Rhizoctonia, and Diplodia Disease. Viral diseases of various crops mediated by Polymyxa genus or Olpidium genus.
Rice seed blight (Burkholderia plantarii); Cucumber spotted bacterial disease (Pseudomonas syringae pv. Lachrymans); Eggplant blight (Ralstonia solanacearum); Citrus scab (Xanthomonas citri); carotovora) etc.

Examples of harmful arthropods that can be controlled by the compounds of the present invention include the following.
Hemiptera: Japanese brown planthopper (Laodelphax striatellus), Japanese brown planthopper (Nilaparvata lugens), white-tailed planthopper (Sogatella furcifera), corn planter (Peregrinus maidis), yellow-spotted plant (Javesella pellucida), black-tailed squid (Delphacidae); Nephotettix cincticeps, Nephotettix virescens, Nephotettix nigropictus, Recilia dorsalis, Eki ca ), Corn Leaf Hopper (Dalbulus maidis), Cofana spectra, etc., Cicadellidae; Mahanarva posticata, Mahanarva fimbriolata, etc., Cercopidae; Aphis fabae, soybean aphids (Aphis glycines), cotton aphids (Aphis gossypii), European apple aphids (Aphis pomi), snowy aphids (Aphis spiraecola), peach aphids (Myzus persicae), wheat arasi , Radish aphids (Brevicoryne brassicae), Rosy apple aphid (Dysaphis plantaginea), black radish aphids (Lipaphis erysimi), tulip beetle aphids (Macrosiphum euphorbiae), potato beetle aphids (Aulacorthum solani), aphids Aphids (Rhopalosiphum padi), corn aphids (Rhopalosiphum maidis), citrus aphids (Toxoptera citricida), peach beetle (Hyalopterus pruni), hyena aphids (Melanaphi) s sacchari), Tetraneura nigriabdominalis, Ceratovacuna lanigera, Eriosoma lanigerum, etc. (Aphididae); Leaf phylloxera (Phylloxera notabilis), Southern pecan leaf phylloxera (Phylloxera russellae) and other aphids (Phylloxeridae); ; Scotinophara lurida, Malayan rice black bug (Scotinophara coarctata), Nezara antennata, Eysarcoris aeneus, Eysarcoris ysori village Eysarcoris annamita, Hailyomorpha halys, Southern stink bug (Nezara viridula), Brown stink bug (Euschistus heros), Red banded stink bug (Piezodorus guildinii), Oebalchel pugnax Pentatomidae); Burrower brown bug (Scaptocoris castanea) and other hornworms (Cydnidae); ); Coleus punctiger, Leptoglossus australis, etc. (Coreidae); Blissus leucopterus) (Lygaeidae); Trigonotylus caelestialium, Stenotus rubrovittatus, Stenodema calcarata, ario des riode (Rygus) , Tobacco whitefly (Bemisia tabaci), Daleurodes citri, Aleurocanthus spiniferus, Aleurocanthus camelliae, Peleius eleyae, etc. (Abgrallaspis cyanophylli), Aonidiella aurantii, Nasimaru scale (Diaspidiotus perniciosus), Scarab scale (Pseudaulacaspis pentagona), Bamboo scale (Unaspis yanonensis), Diaspididae such as Unaspis citri; Coccidae such as Ceroplastes rubens; Icerya purchasi; Icerya purchasi; Icerya seychellarum Scales (Margarodidae); Phenacoccus solani, Phenacoccus solenopsis, Pteracoccus kraunhiae, Pseudococcus comstockicus, trichomec (Pseudococcus calceolariae), Pseudodococcus longispinus, Tattlemy Lee bug (Brevennia rehi), etc., Pseudococcidae; Diaphorina citri; ioza erytreae), Pepylthalidae (Cacopsylla pyrisuga), Pepylthiaceae (Psylliduch), Pear psylla (Cacopsylla pyricola) Corythucha marmorata), Stephanitis nashi, Stephanitis pyrioides, and other species; Cimex lectularius, such as Cimicidae;

Lepidoptera: Green moth (Chilo suppressalis), Darkheaded stem borer (Chilo polychrysus), White stem borer (Scirpophaga innotata), Itteno eel moth (Scirpophaga incertulas), Rupela albina medina, Hacasino maiga (Marasmia exigua), cotton moth (Notarcha derogata), yellow corn borer (Ostrinia furnacalis), European corn borer (Ostrinia nubilalis), yellow moth (Hellula undalis), monk black moth terrel Rice case worms (Nymphula depunctalis), Sugarcane borer (Diatraea saccharalis), etc. (Cambidae); tera litura, Spodoptera exigua, Mythimna separata, Mamestra brassicae, Sesamia inferens, Spodoptera mauritae, ranga pods Spodoptera exempta, Tamanayaga (Agrotis ipsilon), Tamanaginawaba (Autographa nigrisigna), Echinocera (Plusia festucae), Soybean looper (Chrysodeixis includens), Trichoplusia thisppa, Trichoplusia spp Genus (Heliothis spp.), Helicoverpa armigera, American tobacco moth (Helicoverpa zea), Helicobelpa genus (Helicoverpa spp.), Velvetbean caterpillar (Anticarsia gemmatalis), Cotton leafworm (Alabama argillacea), Hop Noctuidae such as borer (Hydraecia immanis); Pieridae such as Pieris rapae; Grapholita molesta, Grapholita dimorpha, M. azukivora), apple wolfberry (Adoxophyes orana fasciata), tea wolfberry (Adoxophyes honmai), chamonaki (Homona magnanima), midarekamonmonki (Archips fuscocupreanus), codialinga (Cydia pomonana ), Bean Shoot Borer (Epinotia aporema), Citrus fruit borer (Ecdytolopha aurantiana), etc. (Tortricidae); (Carposina sasakii), etc. (Carposinidae); Coffee Leaf miner (Leucoptera coffeella), peach leaf (Lyonetia clerkella), winged leaf (Lyonetia prunifoliella), etc. Lymantria spp.), Euproctis pseudoconspersa, Euproctis spp., Etc., Lymantriidae; Helcystogramma triannulella), cotton moth (Pectinophora gossypiella), potato moth (Phthorimaea operculella), Tuta absoluta, etc. (Gelechiidae); Castniidae; Cossidae such as Cossus ボ insularis; Geometridae such as Ascotis selenaria; Limacodidae such as Parasa lepida; Family (Stathmopodidae); Sphingidae such as Acherontia lachesis; Ssiidae such as Nokona feralis; Sesperidae such as Parnara guttata

Thysanoptera: Citrus thrips (Frankliniella occidentalis), Thrips palmiet (Sriptos etbisiton) ), Thripidae such as Echinothrips americanus; Phthaothripripae such as Haplothrips aculeatus.

Diptera: Drosophila (Delia platura), onion flies (Delia antiqua), etc., Anthomyiidae; Tomato leafhopper (Liriomyza sativae), bean leafworm (Liriomyza trifolii), leafhopper (Chromatomyia horticola) and other leafworms (Agromyzidae); ), Eggplant fly (Bactrocera latifrons), olive fruit fly (Bactrocera oleae), quinzland fruit fly (Bactrocera tryoni), CeratitisCcapitata, etc. (Tephritidae); Hydrellia philippina, Hydrellia sasakii, and other species (Ephydridae); Drosophila suzukii, etc .; ); Drosophila such as Clogmia punctalbipunctata; Bradysia difformis and other species, Sciaridae; ); Diopsis macrophthalma, etc. (Diopsidae); Crane fly (Tipula aino), Common cranefly (Tipula oleracea), European cranefly (Tipula paludosa), etc.

Coleoptera: Western corn rootworm (Diabrotica virgifera virgifera), Southern corn rootworm (Diabrotica undecimpunctata howardi), Northern corn rootworm (Diabrotica barberi), Mexican corn rootworm (Diabrotica virgifera zeae), Banded cue Diabrotica balteata), Cucurbit tle Beetle (Diabrotica speciosa), Bean leaf beetle (Cerotoma trifurcata), Bark beetle (Oulema melanopus), potato beetle (Aulacophora femoralis), Phyllotreta bb Cabe black flea beetle (Phyllotreta pusilla), Cabbage stem flea beetle (Psylliodes chrysocephala), Colorado potato beetle (Leptinotarsa decemlineata), Inedro beetle (Oulema oryzae), Grape colaspis (Colaspis brunnea) ), Corn flare beetle (Chaetocnema pulicaria), sweet potato beetle (Chaetocnema confinis), potato flare beetle (Epitrix cucumeris), rice beetle (Dicladispa armigera), southern corn leaf ), Chrysomelidae such as Epitrix hirtipennis; Seedcorn beetle (Stenolophus lecontei), Slender seedcorn beetle (Clivina impressifrons), etc. Carabidae; , Anomala albopilosa, Japanese beetle (Popillia japonica), Nagachakogane (Heptophylla picea), European Chafer (Rhizotrogus majalis), Black marsh (Tomarus gibbosus), Holotrichiall Haga crinita) and other genus Phyllophaga genus (Phyllophaga spp.), Diloboderus usabderus genus Diloboderus genus (Diloboderus spp.) and other scarab beetles (Scarabaeidae); Eusces Sphenophorus venatus), Southern Corn Billbug (Sphenophorus callosus), Soybean stalk weevil (Sternechus S subsignatus), Sugarcane weevil (Sphenophorus levis), Sabihyo weevil (Scepticus griseus) mis), Brazilian weevil (Zabrotes subfasciatus), pine beetle (Tomicus piniperda), Coffee Berry Borer (Hypothenemus hampei), Aracanthus mourei, etc. ); Tribolium castaneum, Tribolium confusum, etc .; Tenebrionidae; Epilachna vigintioctopunctata, etc .; Bostrychidae; Leopardidae (Ptinidae); Anoplophora malasiaca, Migdolus fryanus, etc. , Melanotus legatus, Anchastus spp., Connoderus spp., Ctenicera spp., Limonius spp., Aeolus spp., Etc. Elateridae; Staphylinidae such as Paederus fuscipes.

Orthoptera: Tosama locust (Locusta migratoria), Moroccan flying grasshopper (Dociostaurus maroccanus), Australian flying grasshopper (Chortoicetes terminifera), Red-spotted grasshopper (Nomadacris septemfasciata), Brown Locust ina Italian Locust (Calliptamus italicus), Differential grasshopper (Melanoplus differentialis), Two striped grasshopper (Melanoplus bivittatus), Migratory grasshopper (Melanoplus sanguinipes), Red-Legged grasshopper (Melanoula femurrubrum) gregaria), Yellow-winged locust (Gastrimargus musicus), Spur-throated locust (Austracris guttulosa), Cobainago (Oxya yezoensis), Red-tailed hawk (Oxya japonica), Grasshopper Locust (Patanga succincta), etc. rididae); Gryllotalpidae such as Gryllotalpa orientalis; Grylidae such as Acheta domestica; Gryllidae such as Teleogryllus emma;

Hymenoptera: bee (Athalia rosae), Japanese bee (Athalia japonica) and other bees (Tenthredinidae); Department (Formicidae) etc.

Cockroaches (Blattodea): German cockroaches (Blattellidae) such as the German cockroach (Blattella germanica); Family (Blattidae); Yamato termite (Reticulitermes speratus), Japanese termite (Coptotermes formosanus), American ant termite (Incisitermes orminor), Great white termite (Cryptotermes domesticus), Thai one termite (Odontotermes マ ant hunter) (Glyptotermes satsumensis), Nakajima Termites (Glyptotermes nakajimai), Caterpillars (Glyptotermes fuscus), Termites (Hodotermopsis sjostedti), Coptotermes guangzhouen sis), Amite Termites (Reticulitermes amamianus), Miyatake Termites (Reticulitermes miyatakei), Camellia Termites (Reticulitermes kanmonensis), Takashi Termites (Nasutitermes takasagoensis), Nitobe Termites (Pericapritermes sharimuestermitermes) Termitidae (Termitidae).

Hereinafter, the present invention will be described more specifically with reference to production examples, reference production examples, formulation examples and test examples, but the present invention is not limited to these examples.

Examples of production of the present compound and the present compound are shown below.

Production Example 1-1
At room temperature, 0.6 mL of trifluoroacetic anhydride was added to a mixture of 0.9 g of the intermediate (A1a1) described in Reference Production Example 1-1, 20 mL of DMF and 0.8 mL of pyridine, and the mixture was stirred at 90 ° C. for 6 hours. To the reaction solution, 20 mL of water was added at room temperature, and the mixture was extracted with ethyl acetate. The organic layer was washed with 2N hydrochloric acid, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 1: 1) to obtain 0.5 g of the present compound 1 shown below.

The present compound 1: ¹ H-NMR (CDCl ₃ ) δ: 8.15-8.11 (2H, m), 7.53-7.50 (2H, m), 4.76-4.72 (1H, m), 4.59 (1H, d), 2.86 -2.79 (1H, m), 2.76-2.69 (1H, m), 1.59 (3H, d), 1.24 (3H, t).

Production Example 2-1
To a mixture of 0.13 g of triphosgene and 10 mL of chloroform was added dropwise a mixture of 0.30 g of the intermediate (A3a2) described in Reference Production Example 3-2, 0.22 mL of diisopropylethylamine, and 10 mL of tetrahydrofuran, and the mixture was stirred at room temperature for 1 hour. did. To the resulting mixture, a mixture of N- (2-methoxyethyl) methylamine 0.21 mL, diisopropylethylamine 0.33 mL, and chloroform 10 mL was added dropwise and stirred overnight at room temperature. A saturated aqueous sodium hydrogen carbonate solution was added to the reaction solution, and the mixture was extracted with chloroform. The organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 1: 1) to obtain 0.23 g of the present compound 2 shown below.

Compound 2 of the present invention: ¹ H-NMR (CDCl ₃ ) δ: 8.11 (2H, d), 7.51 (2H, d), 5.20 (2H, s), 2.97 (6H, s).

Production Example 2-2
The compounds produced according to the method described in Production Example 2-1 and their physical properties are shown below.
Formula (a-1)

In which R ¹¹ and R ¹² are represented by the following:

Compound 3 of the present invention (R ¹¹ : CH ₃ , R ¹² : CH ₂ CH ₃ ):
¹ H-NMR (CDCl ₃ ) δ: 8.11 (2H, d), 7.51 (2H, d), 5.20 (2H, s), 3.36 (2H, q), 2.94 (3H, s), 1.14 (3H, t ).
Compound 4 of the present invention (R ¹¹ : CH ₃ , R ¹² : CH ₂ CH ₂ OCH ₃ ):
¹ H-NMR (CDCl ₃ ) δ: 8.11 (2H, d), 7.51 (2H, d), 5.21 (2H, s), 3.59-3.46 (4H, m), 3.40-3.31 (3H, m), 3.06 -2.99 (3H, m).
Compound 5 of the present invention (R ¹¹ : CH ₃ , R ¹² : CH ₂ CN):
¹ H-NMR (CDCl ₃ ) δ: 8.13 (2H, d), 7.52 (2H, d), 5.25 (2H, s), 4.37-4.16 (2H, m), 3.09 (3H, s).
Compound 6 of the present invention (R ¹¹ : CH ₃ , R ¹² : CH ₂ CH ₂ CN):
¹ H-NMR (CDCl ₃ ) δ: 8.13 (2H, d), 7.52 (2H, d), 5.22 (2H, s), 3.66-3.55 (2H, m), 3.14-3.02 (3H, m), 2.72 -2.52 (2H, m).
The present invention compounds _{^{7 (R 11: CH 3,}} R 12: c-Hex):
¹ H-NMR (CDCl ₃ ) δ: 8.11 (2H, d), 7.51 (2H, d), 5.21 (2H, s), 4.07-3.82 (1H, m), 2.83 (3H, s), 1.90-1.02 (10H, m).

Production Example 3-1
0.15 mL of acetyl chloride was added dropwise to a mixture of 0.25 g of the intermediate (A3a2) described in Reference Production Example 3-2 and 0.16 g of aluminum (III) oxide, and the mixture was stirred at room temperature for 1 hour. Ethyl acetate was added to the mixture and filtered. Saturated brine was added to the filtrate, and the mixture was extracted with ethyl acetate. The organic layer was dried over anhydrous magnesium sulfate and concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 1: 4) to obtain 0.25 g of the present compound 8 shown below.

Compound 8 of the present invention: ¹ H-NMR (CDCl ₃ ) δ: 8.12 (2H, d), 7.51 (2H, d), 5.18 (2H, s), 2.15 (3H, s).

Production Example 4-1
At room temperature, 0.95 mL of 50% aqueous hydroxylamine solution was added dropwise to a mixture of 1.4 g of the intermediate (A4a1) described in Reference Production Example 4-1, and 30 mL of ethanol, and the mixture was stirred at 80 ° C. for 2 hours. The mixture was concentrated under reduced pressure. To a mixture of the obtained residue and 50 mL of DMF, 1.1 mL of pyridine was added dropwise at room temperature, and subsequently 0.90 mL of trifluoroacetic anhydride was added dropwise, followed by stirring at 120 ° C. for 3 hours. Water was added to the reaction solution, and the mixture was extracted with ethyl acetate. The organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 1: 1) to obtain 1.4 g of the present compound 9 shown below.

Compound 9 of the present invention: ¹ H-NMR (CDCl ₃ ) δ: 8.09 (2H, d), 7.45 (2H, d), 5.09 (1H, s), 4.46-4.47 (2H, m), 3.73 (3H, s )

Production Example 4-2
The compounds produced according to the method described in Production Example 4-1, and their physical properties are shown below.
Formula (a-2)

Wherein Z ^X and R ^3X are:

Compound 10 of the present invention (Z ^X : OCH ₂ CH ₃ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.09 (2H, d), 7.45 (2H, d), 5.06 (1H, s), 4.46 (2H, d), 4.15-4.20 (2H, m), 1.25-1.29 (3H, m)
Compound 11 of the present invention (Z ^X : OCH (CH ₃ ) ₂ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.08 (2H, d), 7.44 (2H, d), 4.95-5.00 (1H, m), 4.44 (2H, d), 1.25 (6H, d)
Compound 12 of the present invention (Z ^X : OC (CH ₃ ) ₃ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.12 (2H, d), 7.45 (2H, d), 4.62 (2H, d), 1.55 (9H, s)
Compound 13 of the present invention (Z ^X : OCH ₂ Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.07-8.14 (4H, m), 7.32-7.47 (5H, m), 4.62-4.64 (2H, m), 4.47-4.48 (2H, m)
Compound 14 of the present invention (Z ^X : OCH ₂ CH ₂ OCH ₃ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.07 (2H, d), 7.43 (2H, d), 5.17 (1H, s), 4.45 (2H, d), 4.26-4.28 (2H, m), 3.58-3.61 (2H, m), 3.39 (3H, s)
Compound 15 of the present invention (Z ^X : CH ₃ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.09 (2H, d), 7.45 (2H, d), 5.84 (1H, s), 4.54 (2H, d), 2.09 (3H, s)
Compound 16 of the present invention (Z ^X : CH ₂ CH ₃ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.09 (2H, d), 7.44 (2H, d), 5.82 (1H, s), 4.55 (2H, d), 2.27-2.34 (2H, m), 1.20-1.24 (3H, m)
Compound 17 of the present invention (Z ^X : CH ₂ CH ₂ CH ₃ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.07 (2H, d), 7.42 (2H, d), 5.78 (1H, s), 4.52 (2H, d), 2.21-2.25 (2H, m), 1.68-1.76 (2H, m), 0.95-0.98 (3H, m)
Compound 18 of the present invention (Z ^X : CH ₂ CH ₂ CH ₂ CH ₃ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.06 (2H, d), 7.42 (2H, d), 5.78 (1H, s), 4.52 (2H, d), 2.23-2.27 (2H, m), 1.60-1.69 (2H, m), 1.32-1.39 (2H, m), 0.90-0.94 (3H, m)
Compound 19 of the present invention (Z ^X : CH ₂ CH ₂ CH ₂ CH ₂ CH ₃ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.07 (2H, d), 7.42 (2H, d), 5.79 (1H, s), 4.52 (2H, d), 2.22-2.26 (2H, m), 1.62-1.70 (2H, m), 1.29-1.33 (4H, m), 0.87-0.90 (3H, m)
Compound 20 of the present invention (Z ^X : CH ₂ CH ₂ CH ₂ CH ₂ CH ₂ CH ₃ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.08 (2H, d), 7.43 (2H, d), 5.80 (1H, s), 4.54 (2H, d), 2.26 (2H, t), 1.65-1.73 (2H , m), 1.26-1.36 (6H, m), 0.87-0.90 (3H, m)
Compound 21 of the present invention (Z ^X : CH ₂ CH ₂ CH ₂ CH ₂ CH ₂ CH ₂ CH ₃ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.08 (2H, d), 7.43 (2H, d), 5.80 (1H, s), 4.54 (2H, d), 2.26 (2H, t), 1.67-1.70 (2H , m), 1.26-1.36 (8H, m), 0.88 (3H, t)
Compound 22 of the present invention (Z ^X : CH (CH ₃ ) ₂ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.08 (2H, d), 7.43 (2H, d), 5.82 (1H, s), 4.53 (2H, d), 2.40-2.47 (1H, m), 1.22 (6H , d)
Compound 23 of the present invention (Z ^X : CH ₂ CH (CH ₃ ) ₂ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.08 (2H, d), 7.44 (2H, d), 5.77 (1H, s), 4.54 (2H, d), 2.11-2.21 (3H, m), 0.98 (6H , d)
Compound 24 of the present invention (Z ^X : C (CH ₃ ) ₃ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.08 (2H, d), 7.42 (2H, d), 6.02 (1H, s), 4.53 (2H, d), 1.26 (9H, s)
Compound 25 of the present invention (Z ^X : c-Pr, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.07 (2H, d), 7.43 (2H, d), 5.97 (1H, s), 4.54 (2H, d), 1.36-1.42 (1H, m), 1.01-1.05 (2H, m), 0.76-0.81 (2H, m)
Compound 26 of the present invention (Z ^X : c-Bu, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.08 (2H, d), 7.43 (2H, d), 5.71 (1H, s), 4.53 (2H, d), 3.03-3.11 (1H, m), 2.28-2.39 (2H, m), 2.14-2.23 (2H, m), 1.88-2.05 (2H, m)
Compound 27 of the present invention (Z ^X : c-Hex, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.06 (2H, d), 7.40 (2H, d), 5.80 (1H, s), 4.51 (2H, d), 2.10-2.18 (1H, m), 1.20-1.92 (10H, m)
Compound 28 of the present invention (Z ^X : Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.09 (2H, d), 7.82 (2H, s), 7.43-7.53 (5H, m), 6.48 (1H, s), 4.74 (2H, d)
Compound 29 of the present invention (Z ^X : CH ₂ Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.02 (2H, d), 7.27-7.36 (7H, m), 5.74 (1H, s), 4.48 (2H, d), 3.66 (2H, s)
Compound 30 of the present invention (Z ^X : CH ₂ CH ₂ Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.06 (2H, d), 7.24-7.35 (7H, m), 5.71 (1H, s), 4.51 (2H, d), 3.04-3.08 (2H, m), 2.59 -2.62 (2H, m)
Compound 31 of the present invention (Z ^X : CF ₃ , R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.15 (2H, d), 7.47 (2H, d), 6.63 (1H, s), 4.64 (2H, d)
Compound 33 of the present invention (Z ^X : OCH ₂ CH ₃ , R ^3X : CH ₃ )
¹ H-NMR (CDCl ₃ ) δ: 8.09 (2H, d), 7.41 (2H, d), 4.55 (2H, s), 4.18-4.23 (2H, m), 2.88 (3H, s), 1.22-1.31 (3H, m)
Compound 34 of the present invention (Z ^X : OCH ₂ CH ₃ , R ^3X : CH ₂ CH ₃ )
¹ H-NMR (CDCl ₃ ) δ: 8.06 (2H, d), 7.38 (2H, d), 4.53 (2H, s), 4.15-4.21 (2H, m), 3.24-3.36 (2H, m), 1.20 -1.29 (3H, m), 1.05-1.13 (3H, m)
Compound 35 of the present invention (Z ^X : OCH (CH ₃ ) ₂ , R ^3X : CH ₃ )
¹ H-NMR (CDCl ₃ ) δ: 8.07 (2H, d), 7.36 (2H, d), 4.93-5.03 (1H, m), 4.51-4.53 (2H, m), 2.91 (3H, s), 1.24 -1.26 (6H, m)
Compound 36 of the present invention (Z ^X : OCH (CH ₃ ) ₂ , R ^3X : CH ₂ CH ₃ )
¹ H-NMR (CDCl ₃ ) δ: 8.06 (2H, d), 7.39 (2H, d), 4.92-5.01 (1H, m), 4.51 (2H, s), 3.21-3.35 (2H, m), 1.03 -1.32 (9H, m)
Compound 37 of the present invention (Z ^X : CH ₂ CH ₃ , R ^3X : CH ₃ )
¹ H-NMR (CDCl ₃ ) δ: 8.08 (2H, d), 7.39 (2H, d), 4.67 (2H, d), 2.97 (3H, s), 2.41-2.47 (2H, m), 1.20-1.23 (3H, m)
Compound 38 of the present invention (Z ^X : CH ₂ CH ₃ , R ^3X : CH ₂ CH ₃ )
¹ H-NMR (CDCl ₃ ) δ: 8.04 (2H, d), 7.37 (2H, d), 4.65 (2H, s), 3.28-3.33 (2H, m), 2.41-2.47 (2H, m), 1.19 -1.23 (3H, m), 1.13-1.16 (3H, m)
Compound 39 of the present invention (Z ^X : CH ₂ CH (CH ₃ ) ₂ , R ^3X : CH ₃ )
¹ H-NMR (CDCl ₃ ) δ: 8.06 (2H, d), 7.38 (2H, d), 4.66 (2H, s), 2.96 (3H, s), 2.16-2.29 (3H, m), 1.00 (6H , d)
Compound 40 of the present invention (Z ^X : OCH ₂ CH ₃ , R ^3X : Ph)
¹ H-NMR (CDCl ₃ ) δ: 8.03 (2H, d), 7.38 (2H, d), 7.10-7.31 (5H, m), 4.91 (2H, s), 4.16-4.21 (2H, m), 1.18 -1.21 (3H, m)
Compound 46 of the present invention (Z ^X : CHCH ₂ (CH ₃ ) ₂ , R ^3X : OCH ₃ )
¹ H-NMR (CDCl ₃ ) δ: 8.07 (2H, d), 7.47 (2H, d), 4.85 (2H, s), 3.66 (3H, s), 2.36 (2H, d), 2.15-2.25 (1H , m), 0.96 (6H, d)
Compound 41 of the present invention (Z ^X : OCH ₂ CH ₃ , R ^3X : CH ₂ Ph)
¹ H-NMR (CDCl ₃ ) δ: 8.07 (2H, d), 7.17-7.39 (7H, m), 4.44-4.51 (4H, m), 4.25-4.28 (2H, m), 1.28-1.36 (3H, m)
Compound 42 of the present invention (Z ^X : CH ₂ CH ₃ , R ^3X : Ph)
¹ H-NMR (CDCl ₃ ) δ: 8.00 (2H, d), 7.30-7.36 (5H, m), 6.97-6.99 (2H, m), 4.94 (2H, s), 2.07-2.12 (2H, m) , 1.08-1.10 (3H, m)

Production Example 4-3
The compounds produced according to the method described in Production Example 4-1, and their physical properties are shown below.

Compound 43 of the present invention: ¹ H-NMR (CDCl ₃ ) δ: 8.10 (2H, d), 7.41 (2H, d), 4.54 (2H, s), 3.30-3.33 (2H, m), 2.47-2.51 (2H , m), 2.01-2.09 (2H, m)

Compound 44 of the present invention: ¹ H-NMR (CDCl ₃ ) δ: 8.06 (2H, dd), 7.38-7.40 (2H, m), 4.66 (2H, s), 3.21-3.24 (2H, m), 2.49 (2H , t), 1.76-1.85 (4H, m)

Compound 45 of the present invention: ¹ H-NMR (CDCl ₃ ) δ: 7.66 (2H, d), 7.35 (2H, d), 4.42 (2H, s), 2.98 (2H, s), 1.32 (6H, s)

Production Example 5-1
To a mixture of 0.3 g of the present compound 2 and 10 mL of tetrahydrofuran at room temperature was added 0.07 g of sodium hydride (oily, 60%). To the mixture was added 0.09 mL of methyl iodide, and the mixture was stirred at 40 ° C. for 3 hours. Water was added to the obtained mixture, and the mixture was extracted with ethyl acetate. The organic layer was washed with saturated brine, and the organic layer was dried over anhydrous magnesium sulfate and concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 1: 1) to obtain 0.1 g of the present compound 32 shown below.

Compound 32 of the present invention: ¹ H-NMR (CDCl ₃ ) δ: 7.43 (2H, d), 7.31 (2H, d), 4.47-4.51 (2H, m), 4.03 (3H, s), 3.73 (3H, s )

Production Example 6-1
At room temperature, a mixture of 0.2 g of 4- [5- (trifluoromethyl) -1,2,4-oxadiazol-3-yl] benzenemethanamine hydrochloride and 10 mL of tetrahydrofuran was added with 0.26 mL and 2- Chlorobenzoyl chloride (0.11 mL) was sequentially added, and the mixture was stirred at room temperature for 1 hour. The mixture was filtered and the filtrate was concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 1: 1) to obtain 0.15 g of the present compound 47 shown below.

Compound 47 of the present invention: ¹ H-NMR (CDCl ₃ ) δ: 8.11 (2H, d), 7.81-7.81 (1H, m), 7.68-7.70 (1H, m), 7.50-7.52 (3H, m), 7.38 -7.42 (1H, m), 6.46 (1H, s), 4.73-4.74 (2H, m)

Production Example 6-2
The compounds produced according to the method described in Production Example 6-1 and their physical properties are shown below.
Formula (a-3)

Wherein Z ^X and R ^3X are:

Compound 48 of the present invention (Z ^X : 3-Cl—Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.13 (2H, d), 7.74-7.77 (1H, m), 7.57 (2H, d), 7.35-7.46 (3H, m), 6.64 (1H, s), 4.78 (2H, d)
Compound 49 of the present invention (Z ^X : 4-Cl-Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.11 (2H, d), 7.76 (2H, d), 7.51 (2H, d), 7.44 (2H, d), 6.45 (1H, s), 4.74 (2H, d )
Compound 50 of the present invention (Z ^X : 2-OMe-Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.26-8.34 (2H, m), 8.10 (2H, d), 7.48-7.54 (3H, m), 7.11-7.14 (1H, m), 7.01 (1H, d) , 4.78 (2H, d), 3.97 (3H, s)
Compound 51 of the present invention (Z ^X : 3-OMe-Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.11 (2H, d), 7.51 (2H, d), 7.31-7.41 (3H, m), 7.05-7.07 (1H, m), 6.49 (1H, s), 4.74 (2H, d), 3.86 (3H, s)
Compound 52 of the present invention (Z ^X : 4-OMe-Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.10 (2H, d), 7.79 (2H, d), 7.52 (2H, d), 6.95 (2H, d), 6.41 (1H, s), 4.74 (2H, d ), 3.86 (3H, s)
Compound 53 of the present invention (Z ^X : 2-CF ₃ -Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.12 (2H, d), 7.72-7.73 (1H, m), 7.52-7.64 (5H, m), 6.13 (1H, s), 4.73 (2H, d)
Compound 54 of the present invention (Z ^X : 3-CF ₃ -Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.12 (2H, d), 8.08 (1H, s), 8.00-8.02 (1H, m), 7.79-7.81 (1H, m), 7.59-7.63 (1H, m) , 7.53 (2H, d), 6.54 (1H, s), 4.77 (2H, d)
Compound 55 of the present invention (Z ^X : 4-CF ₃ -Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.12 (2H, d), 7.93 (2H, d), 7.73 (2H, d), 7.52 (2H, d), 6.52 (1H, s), 4.76 (2H, d )
Compound 56 of the present invention (Z ^X : 2-F-Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.10-8.18 (3H, m), 7.48-7.54 (3H, m), 7.28-7.32 (1H, m), 7.12-7.20 (2H, m), 4.78 (2H, d)
Compound 57 of the present invention (Z ^X : 3-F-Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.11 (2H, d), 7.40-7.58 (5H, m), 7.21-7.26 (1H, m), 6.47 (1H, s), 4.74 (2H, d)
Compound 58 of the present invention (Z ^X : 4-F-Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.11 (2H, d), 7.82-7.85 (2H, m), 7.52 (2H, d), 7.12-7.16 (2H, m), 6.43 (1H, s), 4.74 (2H, d)
Compound 59 of the present invention (Z ^X : 2-Me-Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.12 (2H, d), 7.53 (2H, d), 7.20-7.42 (4H, m), 6.14 (1H, s), 4.72 (2H, d), 2.48 (3H , s)
Compound 60 of the present invention (Z ^X : 3-Me-Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.11 (2H, d), 7.65-7.65 (1H, m), 7.58-7.60 (1H, m), 7.52 (2H, d), 7.34-7.35 (2H, m) , 6.47 (1H, s), 4.75 (2H, d), 2.41 (3H, s)
Compound 61 of the present invention (Z ^X : 4-Me-Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.10 (2H, d), 7.72 (2H, d), 7.51 (2H, d), 7.26 (2H, d), 6.47 (1H, s), 4.74 (2H, d ), 2.41 (3H, s)
Compound 62 of the present invention (Z ^X : 4-C (CH ₃ ) ₃ —Ph, R ^3X : H):
¹ H-NMR (CDCl ₃ ) δ: 8.10 (2H, d), 7.76 (2H, d), 7.46-7.52 (4H, m), 6.47 (1H, s), 4.75 (2H, d), 1.34 (9H , s)

Production Example 6-3
The compounds produced according to the method described in Production Example 6-1 and their physical properties are shown below.

Compound 63 of the present invention: ¹ H-NMR (CDCl ₃ ) δ: 8.10 (2H, d), 7.98 (1H, s), 7.49 (2H, d), 6.68-6.95 (2H, m), 4.70 (2H, d ), 3.94 (3H, s)

Compound 64 of the present invention: ¹ H-NMR (CDCl ₃ ) δ: 8.17-8.18 (1H, m), 8.10 (2H, d), 7.61-7.63 (1H, m), 7.48 (2H, d), 6.58-6.61 (1H, m), 6.35-6.35 (3H, m), 4.67-4.69 (2H, m)

Production Example 7-1
At room temperature, 0.50 mL of 50% aqueous hydroxylamine solution was added dropwise to a mixture of 0.47 g of the intermediate (A7a1) described in Reference Production Example 7-1 and 5 mL of isopropyl alcohol, and the mixture was stirred at 80 ° C. for 5 hours. The mixture was concentrated under reduced pressure. At room temperature, 0.53 mL of pyridine was added dropwise to a mixture of the obtained residue and 5 mL of DMF, and then 0.34 mL of trifluoroacetic anhydride was added dropwise, followed by stirring at 80 ° C. for 6 hours. Water was added to the reaction solution, and the mixture was extracted with ethyl acetate. The organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 1: 1) to obtain 0.32 g of the present compound 1 shown below.

This compound 1: ¹ H-NMR (CDCl ₃ ) δ: 8.08 (2H, d), 7.42 (2H, d), 3.80 (2H, s), 3.04 (3H, s), 3.00 (3H, s).

Next, reference production examples of the above-mentioned present compound and production intermediates of the present compound are shown.

Reference production example 1-1
A mixture of 0.8 g of intermediate (A2a1), 20 mL of ethanol and 0.9 mL of 50% aqueous hydroxylamine was stirred for 7 hours under reflux. The mixture was concentrated under reduced pressure to obtain 0.9 g of intermediate (A1a1) shown below.

Intermediate (A1a1): ¹ H-NMR (DMSO-D ₆ ) δ: 9.59 (1H, s), 7.64-7.62 (2H, m), 7.38-7.36 (2H, m), 5.77 (2H, s), 4.48-4.44 (1H, m), 2.85-2.76 (1H, m), 2.70-2.61 (1H, m), 1.39 (3H, d), 1.06 (3H, t).

Reference production example 1-2
The compounds produced according to the method described in Reference Production Example 1-1 and their physical properties are shown below.

Intermediate (A1a2): ¹ H-NMR (CDCl ₃ ) δ: 7.62 (2H, d), 7.40 (2H, d), 4.87 (2H, br s), 4.72 (2H, s), 4.62 (2H, s ), 3.42 (3H, s).

Reference Production Example 2-1
At room temperature, 0.4 mL of ethanesulfonyl chloride and 0.7 mL of triethylamine were sequentially added to a mixture of 0.5 g of 4- (1-aminoethyl) benzonitrile and 10 mL of tetrahydrofuran, and the mixture was stirred for 10 hours. 20 mL of water was added to the reaction solution, and the mixture was extracted with ethyl acetate. The organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure to obtain 1.1 g of intermediate (A2a1) shown below.

Intermediate ^{(A2a1): 1 H-NMR} (CDCl 3) δ: 7.69-7.67 (2H, m), 7.49-7.46 (2H, m), 4.75-4.68 (1H, m), 4.55 (1H, br s) , 2.89-2.80 (1H, m), 2.79-2.70 (1H, m), 1.55 (3H, d), 1.26 (3H, t).

Reference Production Example 3-1
To a mixture of 0.50 g of intermediate (A1a2), 5 mL of DMF and 0.57 mL of pyridine, 0.35 mL of trifluoroacetic anhydride was added at room temperature, and the mixture was stirred at 80 ° C. for 3 hours. 20 mL of water was added to the reaction solution at room temperature, and the mixture was extracted with ethyl acetate. The organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 1: 4) to obtain 0.35 g of an intermediate (A3a1) shown below.

Intermediate (A3a1): ¹ H-NMR (CDCl ₃ ) δ: 8.11 (2H, d), 7.52 (2H, d), 4.75 (2H, s), 4.68 (2H, s), 3.43 (3H, s) .

Reference Production Example 3-2
A mixture of 0.2 g of the intermediate (A3a1), 2 mL of methanol and 1.0 mL of 6N hydrochloric acid was stirred at 40 ° C. for 5 hours. Saturated aqueous sodium hydrogen carbonate was added to the reaction mixture, and the mixture was extracted with ethyl acetate. The organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 2: 3) to obtain 0.14 g of an intermediate (A3a2) shown below.

Intermediate (A3a2): ¹ H-NMR (CDCl ₃ ) δ: 8.12 (2H, d), 7.54 (2H, d), 4.81 (2H, d), 1.83 (1H, t).

Reference Production Example 4-1
At room temperature, 0.70 mL of methyl chloroformate and 1.6 mL of triethylamine were sequentially added to a mixture of 1.0 g of 4-cyanobenzylamine and 50 mL of tetrahydrofuran, and the mixture was stirred for 4 hours. The mixture was filtered and the filtrate was concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 2: 1) to obtain 1.4 g of an intermediate (A4a1) shown below.

Intermediate (A4a1): ¹ H-NMR (CDCl ₃ ) δ: 7.63 (2H, d), 7.40 (2H, d), 5.11 (1H, s), 4.40-4.48 (2H, m), 3.72 (3H, s)

Reference production example 4-2
The compounds produced according to the method described in Reference Production Example 4-1 and their physical properties are shown below.

Intermediate (A4a2): ¹ H-NMR (CDCl ₃ ) δ: 7.63 (2H, d), 7.40 (2H, d), 5.06 (1H, s), 4.43 (2H, d), 4.14-4.19 (2H, m), 1.25-1.28 (3H, m)

Reference Production Example 5-1
At room temperature, 1.8 mL of potassium tert-butoxide (1.0 M, tetrahydrofuran solution) was added to a mixture of 0.30 g of intermediate (A4a2) and 10 mL of tetrahydrofuran. To the mixture, 0.11 mL of methyl iodide was added and stirred at room temperature for 4 hours. 20 mL of water was added to the reaction solution, and the mixture was extracted with ethyl acetate. The organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 1: 1) to obtain 0.30 g of an intermediate (A5a1) shown below.

Intermediate (A5a1): ¹ H-NMR (CDCl ₃ ) δ: 7.60 (2H, d), 7.32 (2H, d), 4.62 (2H, s), 2.94-2.93 (3H, m), 2.38-2.44 ( 2H, m), 1.16-1.20 (3H, m)

Reference production example 5-2
At room temperature, 3.6 mL of potassium tert-butoxide (1.0 M, tetrahydrofuran solution) was added to a mixture of 0.50 g of phenylurethane and 15 mL of tetrahydrofuran. To the mixture, 0.58 g of 4-cyanobenzyl bromide was added and stirred at room temperature for 2 hours. Water was added to the reaction solution, and the mixture was extracted with ethyl acetate. The organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 1: 1) to obtain 0.84 g of an intermediate (A5a2) shown below.

Intermediate (A5a2): ¹ H-NMR (CDCl ₃ ) δ: 7.58 (2H, d), 7.08-7.35 (7H, m), 4.88 (2H, s), 4.14-4.19 (2H, m), 1.17- 1.20 (3H, m)

Reference production example 5-3
At room temperature, 0.23 mL of isovaleryl chloride and 0.39 mL of triethylamine were sequentially added to a mixture of 0.30 g of 4- (methoxyamino) methylbenzonitrile and 10 mL of tetrahydrofuran, and the mixture was stirred for 1 hour. The mixture was filtered and the filtrate was concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 2: 1) to obtain 0.45 g of an intermediate (A5a3) shown below.

Intermediate (A5a3): ¹ H-NMR (CDCl ₃ ) δ: 7.62 (2H, d), 7.42 (2H, d), 4.82 (2H, s), 3.66 (3H, s), 2.32-2.33 (2H, m), 2.08-2.25 (1H, m), 1.01 (9H, d)

Reference Production Example 6-1
At room temperature, 0.13 g of sodium hydride (oily, 60%) was added to a mixture of 0.57 g of 3-chloro-N-[(4-cyanophenyl) methyl] -2,2-dimethylpropanamide and 15 mL of tetrahydrofuran, Stir for 2 hours. 10 mL of water was added to the mixture, and the mixture was extracted with ethyl acetate. The organic layer was washed with saturated brine, dried over anhydrous magnesium sulfate, and concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 1: 1) to obtain 0.48 g of an intermediate (A6a1) shown below.

Intermediate (A6a1): ¹ H-NMR (CDCl ₃ ) δ: 7.66 (2H, d), 7.35 (2H, d), 4.42 (2H, s), 2.98 (2H, s), 1.32 (6H, s)

Reference Production Example 7-1
At room temperature, 0.50 mL of thionyl chloride was added to a mixture of 1.0 g of 4-cyanophenylacetic acid and 10 mL of toluene, and the mixture was stirred at 110 ° C. for 1 hour. The mixture was concentrated under reduced pressure, 4 mL of DMF, 6.4 mL of dimethylamine (2M, tetrahydrofuran solution) and 2.1 mL of triethylamine were sequentially added, and the mixture was stirred at room temperature for 2 hours. Water was added to the obtained mixture, and the mixture was extracted with ethyl acetate. The organic layer was washed with saturated brine, and the organic layer was dried over anhydrous magnesium sulfate and concentrated under reduced pressure. The obtained residue was subjected to silica gel column chromatography (ethyl acetate: hexane = 3: 7) to obtain 0.47 g of an intermediate (A7a1) shown below.

Intermediate (A7a1): ¹ H-NMR (CDCl ₃ ) δ: 7.62 (2H, d), 7.37 (2H, d), 3.76 (2H, s), 3.04 (3H, s), 2.98 (3H, s) .

In the present specification, Me represents a methyl group, Et represents an ethyl group, Pr represents a propyl group, i-Pr represents an isopropyl group, c-Pr represents a cyclopropyl group, and Bu represents a butyl group. I-Bu represents an isobutyl group, t-Bu represents a tert-butyl group, c-Bu represents a cyclobutyl group, Pen represents a pentyl group, c-Pen represents a cyclopentyl group, Hex represents hexyl C-Hex represents a cyclohexyl group, OCH ₂ CH═CH ₂ represents an allyloxy group, OCH ₂ C≡CH represents a propargyloxy group, Ph represents a phenyl group, and Bn represents a benzyl group. , 2-Py represents a 2-pyridyl group, 3-Py represents a 3-pyridyl group, 4-Py represents a 4-pyridyl group, Pyr represents a 1-pyrrolidinyl group, and Pip represents - represents a piperidyl group, Mor represents a morpholin-4-yl group.

Formula (III)

In which the combination of R ²¹ , R ²² , R ²³ , R ²⁴ , R ²⁵ and R ²⁶ is a combination described in any of substituent numbers RA1 to RA11232 shown below (Hereinafter, the compounds of the substituent numbers RA1 to RA11232 are represented as the present compounds RA1 to RA11232, and the present compounds RA1 to RA11232 are collectively referred to as the present compound RA) can be obtained according to the method described in the above production method. it can.
The substituent numbers RA1 to RA11232 represent a combination of R ²¹ , R ²² , R ²³ , R ²⁴ , R ²⁵ and R ^{26 in} the compound represented by the formula (III). [Substituent number: R ²¹ , R ²² , R ²³ , R ²⁴ , R ²⁵ , R ²⁶ ]
For example, the substituent number RA4 represents a combination in which R ²¹ , R ²² , R ²⁴ and R ²⁵ are hydrogen atoms, R ²³ is a methyl group, and R ²⁶ is an isopropyl group.

For example, the present compound RA4 means a compound having a substituent number of RA4 in the compound represented by the formula (III), and R ²¹ , R ²² , R ²⁴ and R in the compound represented by the formula (III). ^In the following compounds, ²⁵ represents a hydrogen atom, R ²³ represents a methyl group, and R ²⁶ represents an isopropyl group.

[Substituent number; R ²¹ , R ²² , R ²³ , R ²⁴ , R ²⁵ , R ²⁶ ]: [RA1; H, H, Me, H, H, Me], [RA2; H, H, Me, H , H, Et], [RA3; H, H, Me, H, H, Pr], [RA4; H, H, Me, H, H, i-Pr], [RA5; H, H, Me, H , H, c-Pr], [RA6; H, H, Me, H, H, Bu], [RA7; H, H, Me, H, H, i-Bu], [RA8; H, H, Me , H, H, t-Bu], [RA9; H, H, Me, H, H, c-PrCH ₂ ], [RA10; H, H, Me, H, H, Ph], [RA11; H, H, Me, H, H, Bn], [RA12; H, H, Me, H, H, CF ₃ ], [RA13; H, H, Me, H, H, CF ₃ CH ₂ ], [RA14; H, H, Me, H, H, CF ₃ CF ₂ ], [RA15; H, H, Me, H, H, CF ₂ H], [RA16; H, H, Me, H, H, CF ₂ HCH ₂ ], [RA17; H, H, Me, Me, H, Me], [RA18; H, H, Me, Me, H, Et], [RA19; H, H, Me, Me, H, Pr] , [RA20; H, H, Me, Me, H, i-Pr], [RA21; H, H, Me, Me, H, c-Pr], [RA22; H, H, Me, Me, H, Bu], [RA23; H, H, Me, Me, H, i-Bu], [RA24; H, H, Me, Me, H, t-Bu], [RA25; H, H, Me, Me, H, c-PrCH ₂ ], [RA26; H, H, Me, Me, H, Ph], [RA27; H, H, Me, Me, H, Bn], [RA28; H, H, Me, Me , H, CF ₃ ], [RA29; H, H, Me, Me, H, CF ₃ CH ₂ ], [RA30; H, H, Me, Me, H, CF ₃ CF ₂ ], [RA31; H, H, Me, Me, H, CF ₂ H], [RA32; H, H, Me, Me, H, CF ₂ HCH ₂ ], [RA33; H, H, Me, Et, H, Me], [RA34 ; H, H, Me, Et, H, Et], [RA35; H, H, Me, Et, H, Pr], [RA36; H, H, Me, Et, H, i-Pr], [RA37 ; H, H, Me, Et, H, c-Pr], [RA38; H, H, Me, Et, H, Bu], [RA39; H, H, Me, Et, H, i-Bu], [RA40; H, H, Me, Et, H, t-Bu], [RA41; H, H, Me, Et, H, c-PrCH ₂ ], [RA42; H, H, Me, Et, H, Ph], [RA43; H, H , Me, Et, H, Bn], [RA44; H, H, Me, Et, H, CF ₃ ], [RA45; H, H, Me, Et, H, CF ₃ CH ₂ ], [RA46; H , H, Me, Et, H, CF ₃ CF ₂ ], [RA47; H, H, Me, Et, H, CF ₂ H], [RA48; H, H, Me, Et, H, CF ₂ HCH ₂ ], [RA49; H, H, Me, F, H, Me], [RA50; H, H, Me, F, H, Et], [RA51; H, H, Me, F, H, Pr], [RA52; H, H, Me, F, H, i-Pr], [RA53; H, H, Me, F, H, c-Pr], [RA54; H, H, Me, F, H, Bu ], [RA55; H, H, Me, F, H, i-Bu], [RA56; H, H, Me, F, H, t-Bu], [RA57; H, H, Me, F, H , c-PrCH ₂ ], [RA58; H, H, Me, F, H, Ph], [RA59; H, H, Me, F, H, Bn], [RA60; H, H, Me, F, H, CF ₃ ], [RA61; H, H, Me, F, H, CF ₃ CH ₂ ], [RA62; H, H, Me, F, H, CF ₃ CF ₂ ], [RA63; H, H , Me, F, H, CF ₂ H], [RA64; H, H, Me, F, H, CF ₂ HCH ₂ ], [RA65; H, H, Me, Cl, H, Me], [RA66; H, H, Me, Cl, H, Et], [RA67; H, H, Me, Cl, H, Pr], [RA68; H, H, Me, Cl, H, i-Pr], [RA69; H, H, Me, Cl, H, c-Pr], [RA70; H, H, Me, Cl, H, Bu], [RA71; H, H, Me, Cl, H, i-Bu], [ RA72; H, H, Me, Cl, H, t-Bu], [RA73; H, H, Me, Cl, H, c-PrCH ₂ ], [RA74; H, H, Me, Cl, H, Ph ], [RA75; H, H, Me, Cl, H, Bn], [RA76; H, H, Me, Cl, H, CF ₃ ], [RA77; H, H, Me, Cl, H, CF ₃ CH ₂ ], [RA78; H, H, Me, Cl, H, CF ₃ CF ₂ ], [RA79; H, H, Me, Cl, H, CF ₂ H], [RA80; H, H, Me, Cl, H, CF ₂ HCH ₂ ], [RA81; H, H, Et, H, H, Me], [RA82; H, H, Et, H, H, Et], [RA83; H, H, Et, H, H, Pr ], [RA84; H, H, Et, H, H, i-Pr], [RA85; H, H, Et, H, H, c-Pr], [RA86; H, H, Et, H, H , Bu], [RA87; H, H, Et, H, H, i-Bu], [RA88; H, H, Et, H, H, t-Bu], [RA89; H, H, Et, H , H, c-PrCH ₂ ], [RA90; H, H, Et, H, H, Ph], [RA91; H, H, Et, H, H, Bn], [RA92; H, H, Et, H, H, CF ₃ ], [RA93; H, H, Et, H, H, CF ₃ CH ₂ ], [RA94; H, H, Et, H, H, CF ₃ CF ₂ ], [RA95; H , H, Et, H, H, CF ₂ H], [RA96; H, H, Et, H, H, CF ₂ HCH ₂ ], [RA97; H, H, Et, F, H, Me], [ RA98; H, H, Et, F, H, Et], [RA99; H, H, Et, F, H, Pr], [RA100; H, H, Et, F, H, i-Pr], [ RA101; H, H, Et, F, H, c-Pr], [RA102; H, H, Et, F, H, Bu], [RA103; H, H, Et, F, H, i-Bu] , [RA104; H, H, Et, F, H, t-Bu], [RA105; H, H, Et, F, H, c-PrCH ₂ ], [RA106; H, H, Et, F, H , Ph], [RA107; H, H, Et, F, H, Bn], [RA108; H, H, Et, F, H, CF ₃ ], [RA109; H, H, Et, F, H, CF ₃ CH ₂ ], [RA110; H, H, Et, F, H, CF ₃ CF ₂ ], [RA111; H, H, Et, F, H, CF ₂ H], [RA112; H, H, Et, F, H, CF ₂ HCH ₂ ], [RA113; H, H, Et, Cl, H, Me], [RA114; H, H, Et, Cl, H, Et], [RA115; H, H , Et, Cl, H, Pr], [RA116; H, H, Et, Cl, H, i-Pr], [RA117; H, H, Et, Cl, H, c-Pr], [RA118; H , H, Et, Cl, H, Bu], [RA119; H, H, Et, Cl, H, i-Bu], [RA120; H, H, Et, Cl, H, t-Bu], [RA121 ; H, H, Et, Cl, H, c- PrCH ₂ ], [RA122; H, H, Et, Cl, H, Ph], [RA123; H, H, Et, Cl, H, Bn], [RA124; H, H, Et, Cl, H, CF ₃ ], [RA125; H, H, Et, Cl, H, CF ₃ CH ₂ ], [RA126; H, H, Et, Cl, H, CF ₃ CF ₂ ], [RA127; H, H, Et, Cl, H, CF ₂ H], [RA128; H, H, Et, Cl, H, CF ₂ HCH ₂ ], [RA129; H, H, F, H, H, Me], [RA130; H, H , F, H, H, Et], [RA131; H, H, F, H, H, Pr], [RA132; H, H, F, H, H, i-Pr], [RA133; H, H , F, H, H, c-Pr], [RA134; H, H, F, H, H, Bu], [RA135; H, H, F, H, H, i-Bu], [RA136; H , H, F, H, H, t-Bu], [RA137; H, H, F, H, H, c-PrCH ₂ ], [RA138; H, H, F, H, H, Ph], [ RA139; H, H, F, H, H, Bn], [RA140; H, H, F, H, H, CF ₃ ], [RA141; H, H, F, H, H, CF ₃ CH ₂ ] , [RA142; H, H, F, H, H, CF ₃ CF ₂ ], [RA143; H, H, F, H, H, CF ₂ H], [RA144; H, H, F, H, H , CF ₂ HCH ₂ ], [RA145; H, H, F, F, H, Me], [RA146; H, H, F, F, H, Et], [RA147; H, H, F, F, H, Pr], [RA148; H, H, F, F, H, i-Pr], [RA149; H, H, F, F, H, c-Pr], [RA150; H, H, F, F, H, Bu], [RA151; H, H, F, F, H, i-Bu], [RA152; H, H, F, F, H, t-Bu], [RA153; H, H, F, F, H, c-PrCH ₂ ], [RA154; H, H, F, F, H, Ph], [RA155; H, H, F, F, H, Bn], [RA156; H, H , F, F, H, CF ₃ ], [RA157; H, H, F, F, H, CF ₃ CH ₂ ], [RA158; H, H, F, F, H, CF ₃ CF ₂ ], [ RA159; H, H, F, F, H, CF ₂ H], [RA160; H, H, F, F, H, CF ₂ HCH ₂ ], [RA161; H, H, F, Cl, H, Me ], [RA162; H, H , F, Cl, H, Et], [RA163; H, H, F, Cl, H, Pr], [RA164; H, H, F, Cl, H, i-Pr], [RA165; H, H , F, Cl, H, c-Pr], [RA166; H, H, F, Cl, H, Bu], [RA167; H, H, F, Cl, H, i-Bu], [RA168; H , H, F, Cl, H, t-Bu], [RA169; H, H, F, Cl, H, c-PrCH ₂ ], [RA170; H, H, F, Cl, H, Ph], [ RA171; H, H, F, Cl, H, Bn], [RA172; H, H, F, Cl, H, CF ₃ ], [RA173; H, H, F, Cl, H, CF ₃ CH ₂ ] , [RA174; H, H, F, Cl, H, CF ₃ CF ₂ ], [RA175; H, H, F, Cl, H, CF ₂ H], [RA176; H, H, F, Cl, H , CF ₂ HCH ₂ ], [RA177; H, H, Cl, H, H, Me], [RA178; H, H, Cl, H, H, Et], [RA179; H, H, Cl, H, H, Pr], [RA180; H, H, Cl, H, H, i-Pr], [RA181; H, H, Cl, H, H, c-Pr], [RA182; H, H, Cl, H, H, Bu], [RA183; H, H, Cl, H, H, i-Bu], [RA184; H, H, Cl, H, H, t-Bu], [RA185; H, H, Cl, H, H, c-PrCH ₂ ], [RA186; H, H, Cl, H, H, Ph], [RA187; H, H, Cl, H, H, Bn], [RA188; H, H , Cl, H, H, CF ₃ ], [RA189; H, H, Cl, H, H, CF ₃ CH ₂ ], [RA190; H, H, Cl, H, H, CF ₃ CF ₂ ], [ RA191; H, H, Cl, H, H, CF ₂ H], [RA192; H, H, Cl, H, H, CF ₂ HCH ₂ ], [RA193; H, H, Cl, Cl, H, Me ], [RA194; H, H, Cl, Cl, H, Et], [RA195; H, H, Cl, Cl, H, Pr], [RA196; H, H, Cl, Cl, H, i-Pr ], [RA197; H, H, Cl, Cl, H, c-Pr], [RA198; H, H, Cl, Cl, H, Bu], [RA199; H, H, Cl, Cl, H, i -Bu], [RA200; H, H, Cl, Cl, H, t-Bu],

[RA201; H, H, Cl, Cl, H, c-PrCH ₂ ], [RA202; H, H, Cl, Cl, H, Ph], [RA203; H, H, Cl, Cl, H, Bn] , [RA204; H, H, Cl, Cl, H, CF ₃ ], [RA205; H, H, Cl, Cl, H, CF ₃ CH ₂ ], [RA206; H, H, Cl, Cl, H, CF ₃ CF ₂ ], [RA207; H, H, Cl, Cl, H, CF ₂ H], [RA208; H, H, Cl, Cl, H, CF ₂ HCH ₂ ], [RA209; H, H, Me, H, Me, Me], [RA210; H, H, Me, H, Me, Et], [RA211; H, H, Me, H, Me, Pr], [RA212; H, H, Me, H, Me, i-Pr], [RA213; H, H, Me, H, Me, c-Pr], [RA214; H, H, Me, H, Me, Bu], [RA215; H, H, Me, H, Me, i-Bu], [RA216; H, H, Me, H, Me, t-Bu], [RA217; H, H, Me, H, Me, c-PrCH ₂ ], [RA218 ; H, H, Me, H, Me, Ph], [RA219; H, H, Me, H, Me, Bn], [RA220; H, H, Me, H, Me, CF ₃ ], [RA221; H, H, Me, H, Me, CF ₃ CH ₂ ], [RA222; H, H, Me, H, Me, CF ₃ CF ₂ ], [RA223; H, H, Me, H, Me, CF ₂ H], [RA224; H, H, Me, H, Me, CF ₂ HCH ₂ ], [RA225; H, H, Me, Me, Me, Me], [RA226; H, H, Me, Me, Me , Et], [RA227; H, H, Me, Me, Me, Pr], [RA228; H, H, Me, Me, Me, i-Pr], [RA229; H, H, Me, Me, Me , c-Pr], [RA230; H, H, Me, Me, Me, Bu], [RA231; H, H, Me, Me, Me, i-Bu], [RA232; H, H, Me, Me , Me, t-Bu], [RA233; H, H, Me, Me, Me, c-PrCH ₂ ], [RA234; H, H, Me, Me, Me, Ph], [RA235; H, H, Me, Me, Me, Bn], [RA236; H, H, Me, Me, Me, CF ₃ ], [RA237; H, H, Me, Me, Me, CF ₃ CH ₂ ], [RA238; H, H, Me, Me, Me, CF ₃ CF ₂ ], [RA239; H, H, Me, Me, Me, CF ₂ H], [RA240; H, H, Me, Me, Me, CF ₂ HCH ₂ ], [RA241; H, H, Me, Et, Me, Me], [RA242; H, H, Me, Et, Me, Et], [RA243; H, H, Me, Et, Me, Pr], [RA244; H, H, Me, Et, Me, i-Pr], [RA245; H, H, Me, Et, Me, c-Pr], [RA246; H, H, Me, Et, Me, Bu], [RA247; H, H, Me, Et, Me, i-Bu], [RA248; H, H, Me, Et, Me, t-Bu], [RA249; H, H, Me, Et, Me, c-PrCH ₂ ], [RA250; H , H, Me, Et, Me, Ph], [RA251; H, H, Me, Et, Me, Bn], [RA252; H, H, Me, Et, Me, CF ₃ ], [RA253; H, H, Me, Et, Me, CF ₃ CH ₂ ], [RA254; H, H, Me, Et, Me, CF ₃ CF ₂ ], [RA255; H, H, Me, Et, Me, CF ₂ H] , [RA256; H, H, Me, Et, Me, CF ₂ HCH ₂ ], [RA257; H, H, Me, F, Me, Me], [RA258; H, H, Me, F, Me, Et ], [RA259; H, H, Me, F, Me, Pr], [RA260; H, H, Me, F, Me, i-Pr], [RA261; H, H, Me, F, Me, c -Pr], [RA262; H, H, Me, F, Me, Bu], [RA263; H, H, Me, F, Me, i-Bu], [RA264; H, H, Me, F, Me , t-Bu], [RA265; H, H, Me, F, Me, c-PrCH ₂ ], [RA266; H, H, Me, F, Me, Ph], [RA267; H, H, Me, F, Me, Bn], [RA268; H, H, Me, F, Me, CF ₃ ], [RA269; H, H, Me, F, Me, CF ₃ CH ₂ ], [RA270; H, H, Me, F, Me, CF ₃ CF ₂ ], [RA271; H, H, Me, F, Me, CF ₂ H], [RA272; H, H, Me, F, Me, CF ₂ HCH ₂ ], [ RA273; H, H, Me, Cl, Me, Me], [RA274; H, H, Me, Cl, Me, Et], [RA275; H, H, Me, Cl, Me, Pr], [RA276; H, H, Me , Cl, Me, i-Pr], [RA277; H, H, Me, Cl, Me, c-Pr], [RA278; H, H, Me, Cl, Me, Bu], [RA279; H, H , Me, Cl, Me, i-Bu], [RA280; H, H, Me, Cl, Me, t-Bu], [RA281; H, H, Me, Cl, Me, c-PrCH ₂ ], [ RA282; H, H, Me, Cl, Me, Ph], [RA283; H, H, Me, Cl, Me, Bn], [RA284; H, H, Me, Cl, Me, CF ₃ ], [RA285 ; H, H, Me, Cl, Me, CF ₃ CH ₂ ], [RA286; H, H, Me, Cl, Me, CF ₃ CF ₂ ], [RA287; H, H, Me, Cl, Me, CF ₂ H], [RA288; H, H, Me, Cl, Me, CF ₂ HCH ₂ ], [RA289; H, H, Et, H, Me, Me], [RA290; H, H, Et, H, Me, Et], [RA291; H, H, Et, H, Me, Pr], [RA292; H, H, Et, H, Me, i-Pr], [RA293; H, H, Et, H, Me, c-Pr], [RA294; H, H, Et, H, Me, Bu], [RA295; H, H, Et, H, Me, i-Bu], [RA296; H, H, Et, H, Me, t-Bu], [RA297; H, H, Et, H, Me, c-PrCH ₂ ], [RA298; H, H, Et, H, Me, Ph], [RA299; H, H , Et, H, Me, Bn], [RA300; H, H, Et, H, Me, CF ₃ ], [RA301; H, H, Et, H, Me, CF ₃ CH ₂ ], [RA302; H , H, Et, H, Me, CF ₃ CF ₂ ], [RA303; H, H, Et, H, Me, CF ₂ H], [RA304; H, H, Et, H, Me, CF ₂ HCH ₂ ], [RA305; H, H, Et, F, Me, Me], [RA306; H, H, Et, F, Me, Et], [RA307; H, H, Et, F, Me, Pr], [RA308; H, H, Et, F, Me, i-Pr], [RA309; H, H, Et, F, Me, c-Pr], [RA310; H, H, Et, F, Me, Bu ], [RA311; H, H, Et, F, Me, i-Bu], [RA312; H, H, Et, F, Me, t-Bu], [RA313; H, H, Et, F, Me , c-PrCH ₂ ], [RA314; H, H, Et, F, M e, Ph], [RA315; H, H, Et, F, Me, Bn], [RA316; H, H, Et, F, Me, CF ₃ ], [RA317; H, H, Et, F, Me , CF ₃ CH ₂ ], [RA318; H, H, Et, F, Me, CF ₃ CF ₂ ], [RA319; H, H, Et, F, Me, CF ₂ H], [RA320; H, H , Et, F, Me, CF ₂ HCH ₂ ], [RA321; H, H, Et, Cl, Me, Me], [RA322; H, H, Et, Cl, Me, Et], [RA323; H, H, Et, Cl, Me, Pr], [RA324; H, H, Et, Cl, Me, i-Pr], [RA325; H, H, Et, Cl, Me, c-Pr], [RA326; H, H, Et, Cl, Me, Bu], [RA327; H, H, Et, Cl, Me, i-Bu], [RA328; H, H, Et, Cl, Me, t-Bu], [ RA329; H, H, Et, Cl, Me, c-PrCH ₂ ], [RA330; H, H, Et, Cl, Me, Ph], [RA331; H, H, Et, Cl, Me, Bn], [RA332; H, H, Et, Cl, Me, CF ₃ ], [RA333; H, H, Et, Cl, Me, CF ₃ CH ₂ ], [RA334; H, H, Et, Cl, Me, CF ₃ CF ₂ ], [RA335; H, H, Et, Cl, Me, CF ₂ H], [RA336; H, H, Et, Cl, Me, CF ₂ HCH ₂ ], [RA337; H, H, F , H, Me, Me], [RA338; H, H, F, H, Me, Et], [RA339; H, H, F, H, Me, Pr], [RA340; H, H, F, H , Me, i-Pr], [RA341; H, H, F, H, Me, c-Pr], [RA342; H, H, F, H, Me, Bu], [RA343; H, H, F , H, Me, i-Bu], [RA344; H, H, F, H, Me, t-Bu], [RA345; H, H, F, H, Me, c-PrCH ₂ ], [RA346; H, H, F, H, Me, Ph], [RA347; H, H, F, H, Me, Bn], [RA348; H, H, F, H, Me, CF ₃ ], [RA349; H , H, F, H, Me, CF ₃ CH ₂ ], [RA350; H, H, F, H, Me, CF ₃ CF ₂ ], [RA351; H, H, F, H, Me, CF ₂ H ], [RA352; H, H, F, H, Me, CF ₂ HC H ₂ ], [RA353; H, H, F, F, Me, Me], [RA354; H, H, F, F, Me, Et], [RA355; H, H, F, F, Me, Pr ], [RA356; H, H, F, F, Me, i-Pr], [RA357; H, H, F, F, Me, c-Pr], [RA358; H, H, F, F, Me , Bu], [RA359; H, H, F, F, Me, i-Bu], [RA360; H, H, F, F, Me, t-Bu], [RA361; H, H, F, F , Me, c-PrCH ₂ ], [RA362; H, H, F, F, Me, Ph], [RA363; H, H, F, F, Me, Bn], [RA364; H, H, F, F, Me, CF ₃ ], [RA365; H, H, F, F, Me, CF ₃ CH ₂ ], [RA366; H, H, F, F, Me, CF ₃ CF ₂ ], [RA367; H , H, F, F, Me, CF ₂ H], [RA368; H, H, F, F, Me, CF ₂ HCH ₂ ], [RA369; H, H, F, Cl, Me, Me], [ RA370; H, H, F, Cl, Me, Et], [RA371; H, H, F, Cl, Me, Pr], [RA372; H, H, F, Cl, Me, i-Pr], [ RA373; H, H, F, Cl, Me, c-Pr], [RA374; H, H, F, Cl, Me, Bu], [RA375; H, H, F, Cl, Me, i-Bu] , [RA376; H, H, F, Cl, Me, t-Bu], [RA377; H, H, F, Cl, Me, c-PrCH ₂ ], [RA378; H, H, F, Cl, Me , Ph], [RA379; H, H, F, Cl, Me, Bn], [RA380; H, H, F, Cl, Me, CF ₃ ], [RA381; H, H, F, Cl, Me, CF ₃ CH ₂ ], [RA382; H, H, F, Cl, Me, CF ₃ CF ₂ ], [RA383; H, H, F, Cl, Me, CF ₂ H], [RA384; H, H, F, Cl, Me, CF ₂ HCH ₂ ], [RA385; H, H, Cl, H, Me, Me], [RA386; H, H, Cl, H, Me, Et], [RA387; H, H , Cl, H, Me, Pr], [RA388; H, H, Cl, H, Me, i-Pr], [RA389; H, H, Cl, H, Me, c-Pr], [RA390; H , H, Cl, H, Me, Bu], [RA391; H, H, Cl, H, Me, i-Bu], [RA392; H, H, Cl , H, Me, t-Bu], [RA393; H, H, Cl, H, Me, c-PrCH ₂ ], [RA394; H, H, Cl, H, Me, Ph], [RA395; H, H, Cl, H, Me, Bn], [RA396; H, H, Cl, H, Me, CF ₃ ], [RA397; H, H, Cl, H, Me, CF ₃ CH ₂ ], [RA398; H, H, Cl, H, Me, CF ₃ CF ₂ ], [RA399; H, H, Cl, H, Me, CF ₂ H], [RA400; H, H, Cl, H, Me, CF ₂ HCH ₂ ],

[RA401; H, H, Cl, Cl, Me, Me], [RA402; H, H, Cl, Cl, Me, Et], [RA403; H, H, Cl, Cl, Me, Pr], [RA404 ; H, H, Cl, Cl, Me, i-Pr], [RA405; H, H, Cl, Cl, Me, c-Pr], [RA406; H, H, Cl, Cl, Me, Bu], [RA407; H, H, Cl, Cl, Me, i-Bu], [RA408; H, H, Cl, Cl, Me, t-Bu], [RA409; H, H, Cl, Cl, Me, c -PrCH ₂ ], [RA410; H, H, Cl, Cl, Me, Ph], [RA411; H, H, Cl, Cl, Me, Bn], [RA412; H, H, Cl, Cl, Me, CF ₃ ], [RA413; H, H, Cl, Cl, Me, CF ₃ CH ₂ ], [RA414; H, H, Cl, Cl, Me, CF ₃ CF ₂ ], [RA415; H, H, Cl , Cl, Me, CF ₂ H], [RA416; H, H, Cl, Cl, Me, CF ₂ HCH ₂ ], [RA417; H, H, Me, H, Et, Me], [RA418; H, H, Me, H, Et, Et], [RA419; H, H, Me, H, Et, Pr], [RA420; H, H, Me, H, Et, i-Pr], [RA421; H, H, Me, H, Et, c-Pr], [RA422; H, H, Me, H, Et, Bu], [RA423; H, H, Me, H, Et, i-Bu], [RA424; H, H, Me, H, Et, t-Bu], [RA425; H, H, Me, H, Et, c-PrCH ₂ ], [RA426; H, H, Me, H, Et, Ph], [RA427; H, H, Me, H, Et, Bn], [RA428; H, H, Me, H, Et, CF ₃ ], [RA429; H, H, Me, H, Et, CF ₃ CH ₂ ], [RA430; H, H, Me, H, Et, CF ₃ CF ₂ ], [RA431; H, H, Me, H, Et, CF ₂ H], [RA432; H, H, Me, H, Et, CF ₂ HCH ₂ ], [RA433; H, H, Me, Me, Et, Me], [RA434; H, H, Me, Me, Et, Et], [RA435; H, H, Me, Me , Et, Pr], [RA436; H, H, Me, Me, Et, i-Pr], [RA437; H, H, Me, Me, Et, c-Pr], [RA438; H, H, Me , Me, Et, Bu], [RA439 ; H, H, Me, Me, Et, i-Bu], [RA440; H, H, Me, Me, Et, t-Bu], [RA441; H, H, Me, Me, Et, c-PrCH ₂ ], [RA442; H, H, Me, Me, Et, Ph], [RA443; H, H, Me, Me, Et, Bn], [RA444; H, H, Me, Me, Et, CF ₃ ], [RA445; H, H, Me, Me, Et, CF ₃ CH ₂ ], [RA446; H, H, Me, Me, Et, CF ₃ CF ₂ ], [RA447; H, H, Me, Me , Et, CF ₂ H], [RA448; H, H, Me, Me, Et, CF ₂ HCH ₂ ], [RA449; H, H, Me, Et, Et, Me], [RA450; H, H, Me, Et, Et, Et], [RA451; H, H, Me, Et, Et, Pr], [RA452; H, H, Me, Et, Et, i-Pr], [RA453; H, H, Me, Et, Et, c-Pr], [RA454; H, H, Me, Et, Et, Bu], [RA455; H, H, Me, Et, Et, i-Bu], [RA456; H, H, Me, Et, Et, t-Bu], [RA457; H, H, Me, Et, Et, c-PrCH ₂ ], [RA458; H, H, Me, Et, Et, Ph], [RA459 ; H, H, Me, Et, Et, Bn], [RA460; H, H, Me, Et, Et, CF ₃ ], [RA461; H, H, Me, Et, Et, CF ₃ CH ₂ ], [RA462; H, H, Me, Et, Et, CF ₃ CF ₂ ], [RA463; H, H, Me, Et, Et, CF ₂ H], [RA464; H, H, Me, Et, Et, CF ₂ HCH ₂ ], [RA465; H, H, Me, F, Et, Me], [RA466; H, H, Me, F, Et, Et], [RA467; H, H, Me, F, Et , Pr], [RA468; H, H, Me, F, Et, i-Pr], [RA469; H, H, Me, F, Et, c-Pr], [RA470; H, H, Me, F , Et, Bu], [RA471; H, H, Me, F, Et, i-Bu], [RA472; H, H, Me, F, Et, t-Bu], [RA473; H, H, Me , F, Et, c-PrCH ₂ ], [RA474; H, H, Me, F, Et, Ph], [RA475; H, H, Me, F, Et, Bn], [RA476; H, H, Me, F, Et, CF ₃ ], [RA477; H, H, Me, F, Et, CF ₃ CH ₂ ], [RA478; H, H, Me, F, Et, CF ₃ CF ₂ ], [RA479; H, H, Me, F , Et, CF ₂ H], [RA480; H, H, Me, F, Et, CF ₂ HCH ₂ ], [RA481; H, H, Me, Cl, Et, Me], [RA482; H, H, Me, Cl, Et, Et], [RA483; H, H, Me, Cl, Et, Pr], [RA484; H, H, Me, Cl, Et, i-Pr], [RA485; H, H, Me, Cl, Et, c-Pr], [RA486; H, H, Me, Cl, Et, Bu], [RA487; H, H, Me, Cl, Et, i-Bu], [RA488; H, H, Me, Cl, Et, t-Bu], [RA489; H, H, Me, Cl, Et, c-PrCH ₂ ], [RA490; H, H, Me, Cl, Et, Ph], [RA491 ; H, H, Me, Cl, Et, Bn], [RA492; H, H, Me, Cl, Et, CF ₃ ], [RA493; H, H, Me, Cl, Et, CF ₃ CH ₂ ], [RA494; H, H, Me, Cl, Et, CF ₃ CF ₂ ], [RA495; H, H, Me, Cl, Et, CF ₂ H], [RA496; H, H, Me, Cl, Et, CF ₂ HCH ₂ ], [RA497; H, H, Et, H, Et, Me], [RA498; H, H, Et, H, Et, Et], [RA499; H, H, Et, H, Et , Pr], [RA500; H, H, Et, H, Et, i-Pr], [RA501; H, H, Et, H, Et, c-Pr], [RA502; H, H, Et, H , Et, Bu], [RA503; H, H, Et, H, Et, i-Bu], [RA504; H, H, Et, H, Et, t-Bu], [RA505; H, H, Et , H, Et, c-PrCH ₂ ], [RA506; H, H, Et, H, Et, Ph], [RA507; H, H, Et, H, Et, Bn], [RA508; H, H, Et, H, Et, CF ₃ ], [RA509; H, H, Et, H, Et, CF ₃ CH ₂ ], [RA510; H, H, Et, H, Et, CF ₃ CF ₂ ], [RA511 ; H, H, Et, H, Et, CF ₂ H], [RA512; H, H, Et, H, Et, CF ₂ HCH ₂ ], [RA513; H, H, Et, F, Et, Me] , [RA514; H , H, Et, F, Et, Et], [RA515; H, H, Et, F, Et, Pr], [RA516; H, H, Et, F, Et, i-Pr], [RA517; H , H, Et, F, Et, c-Pr], [RA518; H, H, Et, F, Et, Bu], [RA519; H, H, Et, F, Et, i-Bu], [RA520 ; H, H, Et, F, Et, t-Bu], [RA521; H, H, Et, F, Et, c-PrCH ₂ ], [RA522; H, H, Et, F, Et, Ph] , [RA523; H, H, Et, F, Et, Bn], [RA524; H, H, Et, F, Et, CF ₃ ], [RA525; H, H, Et, F, Et, CF ₃ CH ₂ ], [RA526; H, H, Et, F, Et, CF ₃ CF ₂ ], [RA527; H, H, Et, F, Et, CF ₂ H], [RA528; H, H, Et, F , Et, CF ₂ HCH ₂ ], [RA529; H, H, Et, Cl, Et, Me], [RA530; H, H, Et, Cl, Et, Et], [RA531; H, H, Et, Cl, Et, Pr], [RA532; H, H, Et, Cl, Et, i-Pr], [RA533; H, H, Et, Cl, Et, c-Pr], [RA534; H, H, Et, Cl, Et, Bu], [RA535; H, H, Et, Cl, Et, i-Bu], [RA536; H, H, Et, Cl, Et, t-Bu], [RA537; H, H, Et, Cl, Et, c-PrCH ₂ ], [RA538; H, H, Et, Cl, Et, Ph], [RA539; H, H, Et, Cl, Et, Bn], [RA540; H , H, Et, Cl, Et, CF ₃ ], [RA541; H, H, Et, Cl, Et, CF ₃ CH ₂ ], [RA542; H, H, Et, Cl, Et, CF ₃ CF ₂ ] , [RA543; H, H, Et, Cl, Et, CF ₂ H], [RA544; H, H, Et, Cl, Et, CF ₂ HCH ₂ ], [RA545; H, H, F, H, Et , Me], [RA546; H, H, F, H, Et, Et], [RA547; H, H, F, H, Et, Pr], [RA548; H, H, F, H, Et, i -Pr], [RA549; H, H, F, H, Et, c-Pr], [RA550; H, H, F, H, Et, Bu], [RA551; H, H, F, H, Et , i-Bu], [RA552; H, H, F, H, Et, t-Bu], [ RA553; H, H, F, H, Et, c-PrCH ₂ ], [RA554; H, H, F, H, Et, Ph], [RA555; H, H, F, H, Et, Bn], [RA556; H, H, F, H, Et, CF ₃ ], [RA557; H, H, F, H, Et, CF ₃ CH ₂ ], [RA558; H, H, F, H, Et, CF ₃ CF ₂ ], [RA559; H, H, F, H, Et, CF ₂ H], [RA560; H, H, F, H, Et, CF ₂ HCH ₂ ], [RA561; H, H, F , F, Et, Me], [RA562; H, H, F, F, Et, Et], [RA563; H, H, F, F, Et, Pr], [RA564; H, H, F, F , Et, i-Pr], [RA565; H, H, F, F, Et, c-Pr], [RA566; H, H, F, F, Et, Bu], [RA567; H, H, F , F, Et, i-Bu], [RA568; H, H, F, F, Et, t-Bu], [RA569; H, H, F, F, Et, c-PrCH ₂ ], [RA570; H, H, F, F, Et, Ph], [RA571; H, H, F, F, Et, Bn], [RA572; H, H, F, F, Et, CF ₃ ], [RA573; H , H, F, F, Et, CF ₃ CH ₂ ], [RA574; H, H, F, F, Et, CF ₃ CF ₂ ], [RA575; H, H, F, F, Et, CF ₂ H ], [RA576; H, H, F, F, Et, CF ₂ HCH ₂ ], [RA577; H, H, F, Cl, Et, Me], [RA578; H, H, F, Cl, Et, Et], [RA579; H, H, F, Cl, Et, Pr], [RA580; H, H, F, Cl, Et, i-Pr], [RA581; H, H, F, Cl, Et, c-Pr], [RA582; H, H, F, Cl, Et, Bu], [RA583; H, H, F, Cl, Et, i-Bu], [RA584; H, H, F, Cl, Et, t-Bu], [RA585; H, H, F, Cl, Et, c-PrCH ₂ ], [RA586; H, H, F, Cl, Et, Ph], [RA587; H, H, F , Cl, Et, Bn], [RA588; H, H, F, Cl, Et, CF ₃ ], [RA589; H, H, F, Cl, Et, CF ₃ CH ₂ ], [RA590; H, H , F, Cl, Et, CF ₃ CF ₂ ], [RA591; H, H, F, Cl, Et, CF ₂ H], [RA5 92; H, H, F, Cl, Et, CF ₂ HCH ₂ ], [RA593; H, H, Cl, H, Et, Me], [RA594; H, H, Cl, H, Et, Et], [RA595; H, H, Cl, H, Et, Pr], [RA596; H, H, Cl, H, Et, i-Pr], [RA597; H, H, Cl, H, Et, c-Pr ], [RA598; H, H, Cl, H, Et, Bu], [RA599; H, H, Cl, H, Et, i-Bu], [RA600; H, H, Cl, H, Et, t -Bu],

[RA601; H, H, Cl, H, Et, c-PrCH ₂ ], [RA602; H, H, Cl, H, Et, Ph], [RA603; H, H, Cl, H, Et, Bn] , [RA604; H, H, Cl, H, Et, CF ₃ ], [RA605; H, H, Cl, H, Et, CF ₃ CH ₂ ], [RA606; H, H, Cl, H, Et, CF ₃ CF ₂ ], [RA607; H, H, Cl, H, Et, CF ₂ H], [RA608; H, H, Cl, H, Et, CF ₂ HCH ₂ ], [RA609; H, H, Cl, Cl, Et, Me], [RA610; H, H, Cl, Cl, Et, Et], [RA611; H, H, Cl, Cl, Et, Pr], [RA612; H, H, Cl, Cl, Et, i-Pr], [RA613; H, H, Cl, Cl, Et, c-Pr], [RA614; H, H, Cl, Cl, Et, Bu], [RA615; H, H, Cl, Cl, Et, i-Bu], [RA616; H, H, Cl, Cl, Et, t-Bu], [RA617; H, H, Cl, Cl, Et, c-PrCH ₂ ], [RA618 ; H, H, Cl, Cl, Et, Ph], [RA619; H, H, Cl, Cl, Et, Bn], [RA620; H, H, Cl, Cl, Et, CF ₃ ], [RA621; H, H, Cl, Cl, Et, CF ₃ CH ₂ ], [RA622; H, H, Cl, Cl, Et, CF ₃ CF ₂ ], [RA623; H, H, Cl, Cl, Et, CF ₂ H], [RA624; H, H, Cl, Cl, Et, CF ₂ HCH ₂ ], [RA625; H, H, Me, H, Pr, Me], [RA626; H, H, Me, H, Pr , Et], [RA627; H, H, Me, H, Pr, Pr], [RA628; H, H, Me, H, Pr, i-Pr], [RA629; H, H, Me, H, Pr , c-Pr], [RA630; H, H, Me, H, Pr, Bu], [RA631; H, H, Me, H, Pr, i-Bu], [RA632; H, H, Me, H , Pr, t-Bu], [RA633; H, H, Me, H, Pr, c-PrCH ₂ ], [RA634; H, H, Me, H, Pr, Ph], [RA635; H, H, Me, H, Pr, Bn], [RA636; H, H, Me, H, Pr, CF ₃ ], [RA637; H, H, Me, H, Pr, CF ₃ CH ₂ ], [RA638; H, H, Me, H, Pr, CF ₃ CF ₂ ], [RA639; H, H, Me, H, Pr, CF ₂ H], [RA640; H, H, Me, H, Pr, CF ₂ HCH ₂ ], [RA641; H, H, Me , Me, Pr, Me], [RA642; H, H, Me, Me, Pr, Et], [RA643; H, H, Me, Me, Pr, Pr], [RA644; H, H, Me, Me , Pr, i-Pr], [RA645; H, H, Me, Me, Pr, c-Pr], [RA646; H, H, Me, Me, Pr, Bu], [RA647; H, H, Me , Me, Pr, i-Bu], [RA648; H, H, Me, Me, Pr, t-Bu], [RA649; H, H, Me, Me, Pr, c-PrCH ₂ ], [RA650; H, H, Me, Me, Pr, Ph], [RA651; H, H, Me, Me, Pr, Bn], [RA652; H, H, Me, Me, Pr, CF ₃ ], [RA653; H , H, Me, Me, Pr, CF ₃ CH ₂ ], [RA654; H, H, Me, Me, Pr, CF ₃ CF ₂ ], [RA655; H, H, Me, Me, Pr, CF ₂ H ], [RA656; H, H, Me, Me, Pr, CF ₂ HCH ₂ ], [RA657; H, H, Me, Et, Pr, Me], [RA658; H, H, Me, Et, Pr, Et], [RA659; H, H, Me, Et, Pr, Pr], [RA660; H, H, Me, Et, Pr, i-Pr], [RA661; H, H, Me, Et, Pr, c-Pr], [RA662; H, H, Me, Et, Pr, Bu], [RA663; H, H, Me, Et, Pr, i-Bu], [RA664; H, H, Me, Et, Pr, t-Bu], [RA665; H, H, Me, Et, Pr, c-PrCH ₂ ], [RA666; H, H, Me, Et, Pr, Ph], [RA667; H, H, Me , Et, Pr, Bn], [RA668; H, H, Me, Et, Pr, CF ₃ ], [RA669; H, H, Me, Et, Pr, CF ₃ CH ₂ ], [RA670; H, H , Me, Et, Pr, CF ₃ CF ₂ ], [RA671; H, H, Me, Et, Pr, CF ₂ H], [RA672; H, H, Me, Et, Pr, CF ₂ HCH ₂ ], [RA673; H, H, Me, F, Pr, Me], [RA674; H, H, Me, F, Pr, Et], [RA675; H, H, Me, F, Pr, Pr], [RA676; H, H, Me, F, Pr, i-Pr], [RA677; H, H, Me, F, Pr, c-Pr], [RA678; H, H, Me, F, Pr, Bu ], [RA679; H, H, Me, F, Pr, i-Bu], [RA680; H, H, Me, F, Pr, t-Bu], [RA681; H, H, Me, F, Pr , c-PrCH ₂ ], [RA682; H, H, Me, F, Pr, Ph], [RA683; H, H, Me, F, Pr, Bn], [RA684; H, H, Me, F, Pr, CF ₃ ], [RA685; H, H, Me, F, Pr, CF ₃ CH ₂ ], [RA686; H, H, Me, F, Pr, CF ₃ CF ₂ ], [RA687; H, H , Me, F, Pr, CF ₂ H], [RA688; H, H, Me, F, Pr, CF ₂ HCH ₂ ], [RA689; H, H, Me, Cl, Pr, Me], [RA690; H, H, Me, Cl, Pr, Et], [RA691; H, H, Me, Cl, Pr, Pr], [RA692; H, H, Me, Cl, Pr, i-Pr], [RA693; H, H, Me, Cl, Pr, c-Pr], [RA694; H, H, Me, Cl, Pr, Bu], [RA695; H, H, Me, Cl, Pr, i-Bu], [ RA696; H, H, Me, Cl, Pr, t-Bu], [RA697; H, H, Me, Cl, Pr, c-PrCH ₂ ], [RA698; H, H, Me, Cl, Pr, Ph ], [RA699; H, H, Me, Cl, Pr, Bn], [RA700; H, H, Me, Cl, Pr, CF ₃ ], [RA701; H, H, Me, Cl, Pr, CF ₃ CH ₂ ], [RA702; H, H, Me, Cl, Pr, CF ₃ CF ₂ ], [RA703; H, H, Me, Cl, Pr, CF ₂ H], [RA704; H, H, Me, Cl, Pr, CF ₂ HCH ₂ ], [RA705; H, H, Et, H, Pr, Me], [RA706; H, H, Et, H, Pr, Et], [RA707; H, H, Et , H, Pr, Pr], [RA708; H, H, Et, H, Pr, i-Pr], [RA709; H, H, Et, H, Pr, c-Pr], [RA710; H, H , Et, H, Pr, Bu], [RA711; H, H, Et, H, Pr, i-Bu], [RA712; H, H, Et, H, Pr, t-Bu], [RA713; H , H, Et, H, Pr, c-PrCH ₂ ], [ RA714; H, H, Et, H, Pr, Ph], [RA715; H, H, Et, H, Pr, Bn], [RA716; H, H, Et, H, Pr, CF ₃ ], [RA717 ; H, H, Et, H, Pr, CF ₃ CH ₂ ], [RA718; H, H, Et, H, Pr, CF ₃ CF ₂ ], [RA719; H, H, Et, H, Pr, CF ₂ H], [RA720; H, H, Et, H, Pr, CF ₂ HCH ₂ ], [RA721; H, H, Et, F, Pr, Me], [RA722; H, H, Et, F, Pr, Et], [RA723; H, H, Et, F, Pr, Pr], [RA724; H, H, Et, F, Pr, i-Pr], [RA725; H, H, Et, F, Pr, c-Pr], [RA726; H, H, Et, F, Pr, Bu], [RA727; H, H, Et, F, Pr, i-Bu], [RA728; H, H, Et, F, Pr, t-Bu], [RA729; H, H, Et, F, Pr, c-PrCH ₂ ], [RA730; H, H, Et, F, Pr, Ph], [RA731; H, H , Et, F, Pr, Bn], [RA732; H, H, Et, F, Pr, CF ₃ ], [RA733; H, H, Et, F, Pr, CF ₃ CH ₂ ], [RA734; H , H, Et, F, Pr, CF ₃ CF ₂ ], [RA735; H, H, Et, F, Pr, CF ₂ H], [RA736; H, H, Et, F, Pr, CF ₂ HCH ₂ ], [RA737; H, H, Et, Cl, Pr, Me], [RA738; H, H, Et, Cl, Pr, Et], [RA739; H, H, Et, Cl, Pr, Pr], [RA740; H, H, Et, Cl, Pr, i-Pr], [RA741; H, H, Et, Cl, Pr, c-Pr], [RA742; H, H, Et, Cl, Pr, Bu ], [RA743; H, H, Et, Cl, Pr, i-Bu], [RA744; H, H, Et, Cl, Pr, t-Bu], [RA745; H, H, Et, Cl, Pr , c-PrCH ₂ ], [RA746; H, H, Et, Cl, Pr, Ph], [RA747; H, H, Et, Cl, Pr, Bn], [RA748; H, H, Et, Cl, Pr, CF ₃ ], [RA749; H, H, Et, Cl, Pr, CF ₃ CH ₂ ], [RA750; H, H, Et, Cl, Pr, CF ₃ CF ₂ ], [RA751; H, H , Et, Cl, Pr, CF ₂ H], [RA752; H, H, Et, Cl, Pr, CF ₂ HCH ₂ ], [RA753; H, H, F, H, Pr, Me], [RA754; H, H, F, H, Pr, Et], [RA755; H, H, F, H, Pr, Pr], [RA756; H, H, F, H, Pr, i-Pr], [RA757; H, H, F, H, Pr, c-Pr], [RA758; H, H, F, H, Pr, Bu], [RA759; H, H, F, H, Pr, i-Bu], [RA760; H, H, F, H, Pr, t-Bu], [RA761; H, H, F, H, Pr, c-PrCH ₂ ], [RA762; H, H, F, H, Pr, Ph], [RA763; H, H , F, H, Pr, Bn], [RA764; H, H, F, H, Pr, CF ₃ ], [RA765; H, H, F, H, Pr, CF ₃ CH ₂ ], [RA766; H , H, F, H, Pr, CF ₃ CF ₂ ], [RA767; H, H, F, H, Pr, CF ₂ H], [RA768; H, H, F, H, Pr, CF ₂ HCH ₂ ], [RA769; H, H, F, F, Pr, Me], [RA770; H, H, F, F, Pr, Et], [RA771; H, H, F, F, Pr, Pr], [RA772; H, H, F, F, Pr, i-Pr], [RA773; H, H, F, F, Pr, c-Pr], [RA774; H, H, F, F, Pr, Bu ], [RA775; H, H, F, F, Pr, i-Bu], [RA776; H, H, F, F, Pr, t-Bu], [RA777; H, H, F, F, Pr , c-PrCH ₂ ], [RA778; H, H, F, F, Pr, Ph], [RA779; H, H, F, F, Pr, Bn], [RA780; H, H, F, F, Pr, CF ₃ ], [RA781; H, H, F, F, Pr, CF ₃ CH ₂ ], [RA782; H, H, F, F, Pr, CF ₃ CF ₂ ], [RA783; H, H , F, F, Pr, CF ₂ H], [RA784; H, H, F, F, Pr, CF ₂ HCH ₂ ], [RA785; H, H, F, Cl, Pr, Me], [RA786; H, H, F, Cl, Pr, Et], [RA787; H, H, F, Cl, Pr, Pr], [RA788; H, H, F, Cl, Pr, i-Pr], [RA789; H, H, F, Cl, Pr, c-Pr], [RA790; H, H, F, Cl, Pr, Bu], [RA791; H, H, F, Cl, Pr, iB u], [RA792; H, H, F, Cl, Pr, t-Bu], [RA793; H, H, F, Cl, Pr, c-PrCH ₂ ], [RA794; H, H, F, Cl , Pr, Ph], [RA795; H, H, F, Cl, Pr, Bn], [RA796; H, H, F, Cl, Pr, CF ₃ ], [RA797; H, H, F, Cl, Pr, CF ₃ CH ₂ ], [RA798; H, H, F, Cl, Pr, CF ₃ CF ₂ ], [RA799; H, H, F, Cl, Pr, CF ₂ H], [RA800; H, H, F, Cl, Pr, CF ₂ HCH ₂ ],

[RA801; H, H, Cl, H, Pr, Me], [RA802; H, H, Cl, H, Pr, Et], [RA803; H, H, Cl, H, Pr, Pr], [RA804 ; H, H, Cl, H, Pr, i-Pr], [RA805; H, H, Cl, H, Pr, c-Pr], [RA806; H, H, Cl, H, Pr, Bu], [RA807; H, H, Cl, H, Pr, i-Bu], [RA808; H, H, Cl, H, Pr, t-Bu], [RA809; H, H, Cl, H, Pr, c -PrCH ₂ ], [RA810; H, H, Cl, H, Pr, Ph], [RA811; H, H, Cl, H, Pr, Bn], [RA812; H, H, Cl, H, Pr, CF ₃ ], [RA813; H, H, Cl, H, Pr, CF ₃ CH ₂ ], [RA814; H, H, Cl, H, Pr, CF ₃ CF ₂ ], [RA815; H, H, Cl , H, Pr, CF ₂ H], [RA816; H, H, Cl, H, Pr, CF ₂ HCH ₂ ], [RA817; H, H, Cl, Cl, Pr, Me], [RA818; H, H, Cl, Cl, Pr, Et], [RA819; H, H, Cl, Cl, Pr, Pr], [RA820; H, H, Cl, Cl, Pr, i-Pr], [RA821; H, H, Cl, Cl, Pr, c-Pr], [RA822; H, H, Cl, Cl, Pr, Bu], [RA823; H, H, Cl, Cl, Pr, i-Bu], [RA824; H, H, Cl, Cl, Pr, t-Bu], [RA825; H, H, Cl, Cl, Pr, c-PrCH ₂ ], [RA826; H, H, Cl, Cl, Pr, Ph], [RA827; H, H, Cl, Cl, Pr, Bn], [RA828; H, H, Cl, Cl, Pr, CF ₃ ], [RA829; H, H, Cl, Cl, Pr, CF ₃ CH ₂ ], [RA830; H, H, Cl, Cl, Pr, CF ₃ CF ₂ ], [RA831; H, H, Cl, Cl, Pr, CF ₂ H], [RA832; H, H, Cl, Cl, Pr, CF ₂ HCH ₂ ], [RA833; H, H, Me, H, Bu, Me], [RA834; H, H, Me, H, Bu, Et], [RA835; H, H, Me, H , Bu, Pr], [RA836; H, H, Me, H, Bu, i-Pr], [RA837; H, H, Me, H, Bu, c-Pr], [RA838; H, H, Me , H, Bu, Bu], [RA839; H, H, M e, H, Bu, i-Bu], [RA840; H, H, Me, H, Bu, t-Bu], [RA841; H, H, Me, H, Bu, c-PrCH ₂ ], [RA842 ; H, H, Me, H, Bu, Ph], [RA843; H, H, Me, H, Bu, Bn], [RA844; H, H, Me, H, Bu, CF ₃ ], [RA845; H, H, Me, H, Bu, CF ₃ CH ₂ ], [RA846; H, H, Me, H, Bu, CF ₃ CF ₂ ], [RA847; H, H, Me, H, Bu, CF ₂ H], [RA848; H, H, Me, H, Bu, CF ₂ HCH ₂ ], [RA849; H, H, Me, Me, Bu, Me], [RA850; H, H, Me, Me, Bu , Et], [RA851; H, H, Me, Me, Bu, Pr], [RA852; H, H, Me, Me, Bu, i-Pr], [RA853; H, H, Me, Me, Bu , c-Pr], [RA854; H, H, Me, Me, Bu, Bu], [RA855; H, H, Me, Me, Bu, i-Bu], [RA856; H, H, Me, Me , Bu, t-Bu], [RA857; H, H, Me, Me, Bu, c-PrCH ₂ ], [RA858; H, H, Me, Me, Bu, Ph], [RA859; H, H, Me, Me, Bu, Bn], [RA860; H, H, Me, Me, Bu, CF ₃ ], [RA861; H, H, Me, Me, Bu, CF ₃ CH ₂ ], [RA862; H, H, Me, Me, Bu, CF ₃ CF ₂ ], [RA863; H, H, Me, Me, Bu, CF ₂ H], [RA864; H, H, Me, Me, Bu, CF ₂ HCH ₂ ] , [RA865; H, H, Me, Et, Bu, Me], [RA866; H, H, Me, Et, Bu, Et], [RA867; H, H, Me, Et, Bu, Pr], [ RA868; H, H, Me, Et, Bu, i-Pr], [RA869; H, H, Me, Et, Bu, c-Pr], [RA870; H, H, Me, Et, Bu, Bu] , [RA871; H, H, Me, Et, Bu, i-Bu], [RA872; H, H, Me, Et, Bu, t-Bu], [RA873; H, H, Me, Et, Bu, c-PrCH ₂ ], [RA874; H, H, Me, Et, Bu, Ph], [RA875; H, H, Me, Et, Bu, Bn], [RA876; H, H, Me, Et, Bu , CF ₃ ], [R A877; H, H, Me, Et, Bu, CF ₃ CH ₂ ], [RA878; H, H, Me, Et, Bu, CF ₃ CF ₂ ], [RA879; H, H, Me, Et, Bu, CF ₂ H], [RA880; H, H, Me, Et, Bu, CF ₂ HCH ₂ ], [RA881; H, H, Me, F, Bu, Me], [RA882; H, H, Me, F , Bu, Et], [RA883; H, H, Me, F, Bu, Pr], [RA884; H, H, Me, F, Bu, i-Pr], [RA885; H, H, Me, F , Bu, c-Pr], [RA886; H, H, Me, F, Bu, Bu], [RA887; H, H, Me, F, Bu, i-Bu], [RA888; H, H, Me , F, Bu, t-Bu], [RA889; H, H, Me, F, Bu, c-PrCH ₂ ], [RA890; H, H, Me, F, Bu, Ph], [RA891; H, H, Me, F, Bu, Bn], [RA892; H, H, Me, F, Bu, CF ₃ ], [RA893; H, H, Me, F, Bu, CF ₃ CH ₂ ], [RA894; H, H, Me, F, Bu, CF ₃ CF ₂ ], [RA895; H, H, Me, F, Bu, CF ₂ H], [RA896; H, H, Me, F, Bu, CF ₂ HCH ₂ ], [RA897; H, H, Me, Cl, Bu, Me], [RA898; H, H, Me, Cl, Bu, Et], [RA899; H, H, Me, Cl, Bu, Pr] , [RA900; H, H, Me, Cl, Bu, i-Pr], [RA901; H, H, Me, Cl, Bu, c-Pr], [RA902; H, H, Me, Cl, Bu, Bu], [RA903; H, H, Me, Cl, Bu, i-Bu], [RA904; H, H, Me, Cl, Bu, t-Bu], [RA905; H, H, Me, Cl, Bu, c-PrCH ₂ ], [RA906; H, H, Me, Cl, Bu, Ph], [RA907; H, H, Me, Cl, Bu, Bn], [RA908; H, H, Me, Cl , Bu, CF ₃ ], [RA909; H, H, Me, Cl, Bu, CF ₃ CH ₂ ], [RA910; H, H, Me, Cl, Bu, CF ₃ CF ₂ ], [RA911; H, H, Me, Cl, Bu, CF ₂ H], [RA912; H, H, Me, Cl, Bu, CF ₂ HCH ₂ ], [RA913; H, H, Et, H, Bu, Me], [RA914 ; H , H, Et, H, Bu, Et], [RA915; H, H, Et, H, Bu, Pr], [RA916; H, H, Et, H, Bu, i-Pr], [RA917; H , H, Et, H, Bu, c-Pr], [RA918; H, H, Et, H, Bu, Bu], [RA919; H, H, Et, H, Bu, i-Bu], [RA920 ; H, H, Et, H, Bu, t-Bu], [RA921; H, H, Et, H, Bu, c-PrCH ₂ ], [RA922; H, H, Et, H, Bu, Ph] , [RA923; H, H, Et, H, Bu, Bn], [RA924; H, H, Et, H, Bu, CF ₃ ], [RA925; H, H, Et, H, Bu, CF ₃ CH ₂ ], [RA926; H, H, Et, H, Bu, CF ₃ CF ₂ ], [RA927; H, H, Et, H, Bu, CF ₂ H], [RA928; H, H, Et, H , Bu, CF ₂ HCH ₂ ], [RA929; H, H, Et, F, Bu, Me], [RA930; H, H, Et, F, Bu, Et], [RA931; H, H, Et, F, Bu, Pr], [RA932; H, H, Et, F, Bu, i-Pr], [RA933; H, H, Et, F, Bu, c-Pr], [RA934; H, H, Et, F, Bu, Bu], [RA935; H, H, Et, F, Bu, i-Bu], [RA936; H, H, Et, F, Bu, t-Bu], [RA937; H, H, Et, F, Bu, c-PrCH ₂ ], [RA938; H, H, Et, F, Bu, Ph], [RA939; H, H, Et, F, Bu, Bn], [RA940; H , H, Et, F, Bu, CF ₃ ], [RA941; H, H, Et, F, Bu, CF ₃ CH ₂ ], [RA942; H, H, Et, F, Bu, CF ₃ CF ₂ ] , [RA943; H, H, Et, F, Bu, CF ₂ H], [RA944; H, H, Et, F, Bu, CF ₂ HCH ₂ ], [RA945; H, H, Et, Cl, Bu , Me], [RA946; H, H, Et, Cl, Bu, Et], [RA947; H, H, Et, Cl, Bu, Pr], [RA948; H, H, Et, Cl, Bu, i -Pr], [RA949; H, H, Et, Cl, Bu, c-Pr], [RA950; H, H, Et, Cl, Bu, Bu], [RA951; H, H, Et, Cl, Bu , i-Bu], [RA952; H, H, Et, Cl, Bu, t-Bu], [ RA953; H, H, Et, Cl, Bu, c-PrCH ₂ ], [RA954; H, H, Et, Cl, Bu, Ph], [RA955; H, H, Et, Cl, Bu, Bn], [RA956; H, H, Et, Cl, Bu, CF ₃ ], [RA957; H, H, Et, Cl, Bu, CF ₃ CH ₂ ], [RA958; H, H, Et, Cl, Bu, CF ₃ CF ₂ ], [RA959; H, H, Et, Cl, Bu, CF ₂ H], [RA960; H, H, Et, Cl, Bu, CF ₂ HCH ₂ ], [RA961; H, H, F , H, Bu, Me], [RA962; H, H, F, H, Bu, Et], [RA963; H, H, F, H, Bu, Pr], [RA964; H, H, F, H , Bu, i-Pr], [RA965; H, H, F, H, Bu, c-Pr], [RA966; H, H, F, H, Bu, Bu], [RA967; H, H, F , H, Bu, i-Bu], [RA968; H, H, F, H, Bu, t-Bu], [RA969; H, H, F, H, Bu, c-PrCH ₂ ], [RA970; H, H, F, H, Bu, Ph], [RA971; H, H, F, H, Bu, Bn], [RA972; H, H, F, H, Bu, CF ₃ ], [RA973; H , H, F, H, Bu, CF ₃ CH ₂ ], [RA974; H, H, F, H, Bu, CF ₃ CF ₂ ], [RA975; H, H, F, H, Bu, CF ₂ H ], [RA976; H, H, F, H, Bu, CF ₂ HCH ₂ ], [RA977; H, H, F, F, Bu, Me], [RA978; H, H, F, F, Bu, Et], [RA979; H, H, F, F, Bu, Pr], [RA980; H, H, F, F, Bu, i-Pr], [RA981; H, H, F, F, Bu, c-Pr], [RA982; H, H, F, F, Bu, Bu], [RA983; H, H, F, F, Bu, i-Bu], [RA984; H, H, F, F, Bu, t-Bu], [RA985; H, H, F, F, Bu, c-PrCH ₂ ], [RA986; H, H, F, F, Bu, Ph], [RA987; H, H, F , F, Bu, Bn], [RA988; H, H, F, F, Bu, CF ₃ ], [RA989; H, H, F, F, Bu, CF ₃ CH ₂ ], [RA990; H, H , F, F, Bu, CF ₃ CF ₂ ], [RA991; H, H, F, F, Bu, CF ₂ H], [RA 992, H, H, F, F, Bu, CF ₂ HCH ₂ ], [RA993; H, H, F, Cl, Bu, Me], [RA994; H, H, F, Cl, Bu, Et], [RA995; H, H, F, Cl, Bu, Pr], [RA996; H, H, F, Cl, Bu, i-Pr], [RA997; H, H, F, Cl, Bu, c-Pr ], [RA998; H, H, F, Cl, Bu, Bu], [RA999; H, H, F, Cl, Bu, i-Bu], [RA1000; H, H, F, Cl, Bu, t -Bu],

[RA1001; H, H, F, Cl, Bu, c-PrCH ₂ ], [RA1002; H, H, F, Cl, Bu, Ph], [RA1003; H, H, F, Cl, Bu, Bn] , [RA1004; H, H, F, Cl, Bu, CF ₃ ], [RA1005; H, H, F, Cl, Bu, CF ₃ CH ₂ ], [RA1006; H, H, F, Cl, Bu, CF ₃ CF ₂ ], [RA1007; H, H, F, Cl, Bu, CF ₂ H], [RA1008; H, H, F, Cl, Bu, CF ₂ HCH ₂ ], [RA1009; H, H, Cl, H, Bu, Me], [RA1010; H, H, Cl, H, Bu, Et], [RA1011; H, H, Cl, H, Bu, Pr], [RA1012; H, H, Cl, H, Bu, i-Pr], [RA1013; H, H, Cl, H, Bu, c-Pr], [RA1014; H, H, Cl, H, Bu, Bu], [RA1015; H, H, Cl, H, Bu, i-Bu], [RA1016; H, H, Cl, H, Bu, t-Bu], [RA1017; H, H, Cl, H, Bu, c-PrCH ₂ ], [RA1018 ; H, H, Cl, H, Bu, Ph], [RA1019; H, H, Cl, H, Bu, Bn], [RA1020; H, H, Cl, H, Bu, CF ₃ ], [RA1021; H, H, Cl, H, Bu, CF ₃ CH ₂ ], [RA1022; H, H, Cl, H, Bu, CF ₃ CF ₂ ], [RA1023; H, H, Cl, H, Bu, CF ₂ H], [RA1024; H, H, Cl, H, Bu, CF ₂ HCH ₂ ], [RA1025; H, H, Cl, Cl, Bu, Me], [RA1026; H, H, Cl, Cl, Bu , Et], [RA1027; H, H, Cl, Cl, Bu, Pr], [RA1028; H, H, Cl, Cl, Bu, i-Pr], [RA1029; H, H, Cl, Cl, Bu , c-Pr], [RA1030; H, H, Cl, Cl, Bu, Bu], [RA1031; H, H, Cl, Cl, Bu, i-Bu], [RA1032; H, H, Cl, Cl , Bu, t-Bu], [RA1033; H, H, Cl, Cl, Bu, c-PrCH ₂ ], [RA1034; H, H, Cl, Cl, Bu, Ph], [RA1035; H, H, Cl, Cl, Bu, Bn], [RA1036; H, H, Cl, Cl, Bu, CF ₃ ], [RA1037; H, H, Cl, Cl, Bu , CF ₃ CH ₂ ], [RA1038; H, H, Cl, Cl, Bu, CF ₃ CF ₂ ], [RA1039; H, H, Cl, Cl, Bu, CF ₂ H], [RA1040; H, H , Cl, Cl, Bu, CF ₂ HCH ₂ ], [RA1041; H, H, Me, H, i-Pr, Me], [RA1042; H, H, Me, H, i-Pr, Et], [ RA1043; H, H, Me, H, i-Pr, Pr], [RA1044; H, H, Me, H, i-Pr, i-Pr], [RA1045; H, H, Me, H, i- Pr, c-Pr], [RA1046; H, H, Me, H, i-Pr, Bu], [RA1047; H, H, Me, H, i-Pr, i-Bu], [RA1048; H, H, Me, H, i-Pr, t-Bu], [RA1049; H, H, Me, H, i-Pr, c-PrCH ₂ ], [RA1050; H, H, Me, H, i-Pr , Ph], [RA1051; H, H, Me, H, i-Pr, Bn], [RA1052; H, H, Me, H, i-Pr, CF ₃ ], [RA1053; H, H, Me, H, i-Pr, CF ₃ CH ₂ ], [RA1054; H, H, Me, H, i-Pr, CF ₃ CF ₂ ], [RA1055; H, H, Me, H, i-Pr, CF ₂ H], [RA1056; H, H, Me, H, i-Pr, CF ₂ HCH ₂ ], [RA1057; H, H, Me, Me, i-Pr, Me], [RA1058; H, H, Me , Me, i-Pr, Et], [RA1059; H, H, Me, Me, i-Pr, Pr], [RA1060; H, H, Me, Me, i-Pr, i-Pr], [RA1061 ; H, H, Me, Me, i-Pr, c-Pr], [RA1062; H, H, Me, Me, i-Pr, Bu], [RA1063; H, H, Me, Me, i-Pr , i-Bu], [RA1064; H, H, Me, Me, i-Pr, t-Bu], [RA1065; H, H, Me, Me, i-Pr, c-PrCH ₂ ], [RA1066; H, H, Me, Me, i-Pr, Ph], [RA1067; H, H, Me, Me, i-Pr, Bn], [RA1068; H, H, Me, Me, i-Pr, CF ₃ ], [RA1069; H, H, Me, Me, i-Pr, CF ₃ CH ₂ ], [RA1070; H, H, Me, Me, i-Pr, CF ₃ CF ₂ ], [RA1071; H, H , Me, M e, i-Pr, CF ₂ H], [RA1072; H, H, Me, Me, i-Pr, CF ₂ HCH ₂ ], [RA1073; H, H, Me, Et, i-Pr, Me], [RA1074; H, H, Me, Et, i-Pr, Et], [RA1075; H, H, Me, Et, i-Pr, Pr], [RA1076; H, H, Me, Et, i-Pr , i-Pr], [RA1077; H, H, Me, Et, i-Pr, c-Pr], [RA1078; H, H, Me, Et, i-Pr, Bu], [RA1079; H, H , Me, Et, i-Pr, i-Bu], [RA1080; H, H, Me, Et, i-Pr, t-Bu], [RA1081; H, H, Me, Et, i-Pr, c -PrCH ₂ ], [RA1082; H, H, Me, Et, i-Pr, Ph], [RA1083; H, H, Me, Et, i-Pr, Bn], [RA1084; H, H, Me, Et, i-Pr, CF ₃ ], [RA1085; H, H, Me, Et, i-Pr, CF ₃ CH ₂ ], [RA1086; H, H, Me, Et, i-Pr, CF ₃ CF ₂ ], [RA1087; H, H, Me, Et, i-Pr, CF ₂ H], [RA1088; H, H, Me, Et, i-Pr, CF ₂ HCH ₂ ], [RA1089; H, H, Me, F, i-Pr, Me], [RA1090; H, H, Me, F, i-Pr, Et], [RA1091; H, H, Me, F, i-Pr, Pr], [RA1092; H, H, Me, F, i-Pr, i-Pr], [RA1093; H, H, Me, F, i-Pr, c-Pr], [RA1094; H, H, Me, F, i- Pr, Bu], [RA1095; H, H, Me, F, i-Pr, i-Bu], [RA1096; H, H, Me, F, i-Pr, t-Bu], [RA1097; H, H, Me, F, i-Pr, c-PrCH ₂ ], [RA1098; H, H, Me, F, i-Pr, Ph], [RA1099; H, H, Me, F, i-Pr, Bn ], [RA1100; H, H, Me, F, i-Pr, CF ₃ ], [RA1101; H, H, Me, F, i-Pr, CF ₃ CH ₂ ], [RA1102; H, H, Me , F, i-Pr, CF ₃ CF ₂ ], [RA1103; H, H, Me, F, i-Pr, CF ₂ H], [RA1104; H, H, Me, F, i-Pr, CF ₂ HCH ₂ ], [RA1105 ; H, H, Me, Cl, i-Pr, Me], [RA1106; H, H, Me, Cl, i-Pr, Et], [RA1107; H, H, Me, Cl, i-Pr, Pr ], [RA1108; H, H, Me, Cl, i-Pr, i-Pr], [RA1109; H, H, Me, Cl, i-Pr, c-Pr], [RA1110; H, H, Me , Cl, i-Pr, Bu], [RA1111; H, H, Me, Cl, i-Pr, i-Bu], [RA1112; H, H, Me, Cl, i-Pr, t-Bu], [RA1113; H, H, Me, Cl, i-Pr, c-PrCH ₂ ], [RA1114; H, H, Me, Cl, i-Pr, Ph], [RA1115; H, H, Me, Cl, i-Pr, Bn], [RA1116; H, H, Me, Cl, i-Pr, CF ₃ ], [RA1117; H, H, Me, Cl, i-Pr, CF ₃ CH ₂ ], [RA1118; H, H, Me, Cl, i-Pr, CF ₃ CF ₂ ], [RA1119; H, H, Me, Cl, i-Pr, CF ₂ H], [RA1120; H, H, Me, Cl, i -Pr, CF ₂ HCH ₂ ], [RA1121; H, H, Et, H, i-Pr, Me], [RA1122; H, H, Et, H, i-Pr, Et], [RA1123; H, H, Et, H, i-Pr, Pr], [RA1124; H, H, Et, H, i-Pr, i-Pr], [RA1125; H, H, Et, H, i-Pr, c- Pr], [RA1126; H, H, Et, H, i-Pr, Bu], [RA1127; H, H, Et, H, i-Pr, i-Bu], [RA1128; H, H, Et, H, i-Pr, t-Bu], [RA1129; H, H, Et, H, i-Pr, c-PrCH ₂ ], [RA1130; H, H, Et, H, i-Pr, Ph], [RA1131; H, H, Et, H, i-Pr, Bn], [RA1132; H, H, Et, H, i-Pr, CF ₃ ], [RA1133; H, H, Et, H, i- Pr, CF ₃ CH ₂ ], [RA1134; H, H, Et, H, i-Pr, CF ₃ CF ₂ ], [RA1135; H, H, Et, H, i-Pr, CF ₂ H], [ RA1136; H, H, Et, H, i-Pr, CF ₂ HCH ₂ ], [RA1137; H, H, Et, F, i-Pr, Me], [RA1138; H, H, Et, F, i -Pr, Et], [RA1139; H, H, E t, F, i-Pr, Pr], [RA1140; H, H, Et, F, i-Pr, i-Pr], [RA1141; H, H, Et, F, i-Pr, c-Pr] , [RA1142; H, H, Et, F, i-Pr, Bu], [RA1143; H, H, Et, F, i-Pr, i-Bu], [RA1144; H, H, Et, F, i-Pr, t-Bu], [RA1145; H, H, Et, F, i-Pr, c-PrCH ₂ ], [RA1146; H, H, Et, F, i-Pr, Ph], [RA1147 ; H, H, Et, F, i-Pr, Bn], [RA1148; H, H, Et, F, i-Pr, CF ₃ ], [RA1149; H, H, Et, F, i-Pr, CF ₃ CH ₂ ], [RA1150; H, H, Et, F, i-Pr, CF ₃ CF ₂ ], [RA1151; H, H, Et, F, i-Pr, CF ₂ H], [RA1152; H, H, Et, F, i-Pr, CF ₂ HCH ₂ ], [RA1153; H, H, Et, Cl, i-Pr, Me], [RA1154; H, H, Et, Cl, i-Pr , Et], [RA1155; H, H, Et, Cl, i-Pr, Pr], [RA1156; H, H, Et, Cl, i-Pr, i-Pr], [RA1157; H, H, Et , Cl, i-Pr, c-Pr], [RA1158; H, H, Et, Cl, i-Pr, Bu], [RA1159; H, H, Et, Cl, i-Pr, i-Bu], [RA1160; H, H, Et, Cl, i-Pr, t-Bu], [RA1161; H, H, Et, Cl, i-Pr, c-PrCH ₂ ], [RA1162; H, H, Et, Cl, i-Pr, Ph], [RA1163; H, H, Et, Cl, i-Pr, Bn], [RA1164; H, H, Et, Cl, i-Pr, CF ₃ ], [RA1165; H , H, Et, Cl, i-Pr, CF ₃ CH ₂ ], [RA1166; H, H, Et, Cl, i-Pr, CF ₃ CF ₂ ], [RA1167; H, H, Et, Cl, i -Pr, CF ₂ H], [RA1168; H, H, Et, Cl, i-Pr, CF ₂ HCH ₂ ], [RA1169; H, H, F, H, i-Pr, Me], [RA1170; H, H, F, H, i-Pr, Et], [RA1171; H, H, F, H, i-Pr, Pr], [RA1172; H, H, F, H, i-Pr, i- Pr], [RA1173; H, H, F, H, i-Pr, c-Pr], [RA1174; H, H, F, H, i-Pr, Bu], [RA1175; H, H, F, H, i-Pr, i-Bu], [RA1176; H, H, F, H, i-Pr, t-Bu], [RA1177; H, H, F, H, i-Pr, c-PrCH ₂ ], [RA1178; H, H, F, H, i-Pr, Ph ], [RA1179; H, H, F, H, i-Pr, Bn], [RA1180; H, H, F, H, i-Pr, CF ₃ ], [RA1181; H, H, F, H, i-Pr, CF ₃ CH ₂ ], [RA1182; H, H, F, H, i-Pr, CF ₃ CF ₂ ], [RA1183; H, H, F, H, i-Pr, CF ₂ H] , [RA1184; H, H, F, H, i-Pr, CF ₂ HCH ₂ ], [RA1185; H, H, F, F, i-Pr, Me], [RA1186; H, H, F, F , i-Pr, Et], [RA1187; H, H, F, F, i-Pr, Pr], [RA1188; H, H, F, F, i-Pr, i-Pr], [RA1189; H , H, F, F, i-Pr, c-Pr], [RA1190; H, H, F, F, i-Pr, Bu], [RA1191; H, H, F, F, i-Pr, i -Bu], [RA1192; H, H, F, F, i-Pr, t-Bu], [RA1193; H, H, F, F, i-Pr, c-PrCH ₂ ], [RA1194; H, H, F, F, i-Pr, Ph], [RA1195; H, H, F, F, i-Pr, Bn], [RA1196; H, H, F, F, i-Pr, CF ₃ ], [RA1197; H, H, F, F, i-Pr, CF ₃ CH ₂ ], [RA1198; H, H, F, F, i-Pr, CF ₃ CF ₂ ], [RA1199; H, H, F , F, i-Pr, CF ₂ H], [RA1200; H, H, F, F, i-Pr, CF ₂ HCH ₂ ],

[RA1201; H, H, F, Cl, i-Pr, Me], [RA1202; H, H, F, Cl, i-Pr, Et], [RA1203; H, H, F, Cl, i-Pr , Pr], [RA1204; H, H, F, Cl, i-Pr, i-Pr], [RA1205; H, H, F, Cl, i-Pr, c-Pr], [RA1206; H, H , F, Cl, i-Pr, Bu], [RA1207; H, H, F, Cl, i-Pr, i-Bu], [RA1208; H, H, F, Cl, i-Pr, t-Bu ], [RA1209; H, H, F, Cl, i-Pr, c-PrCH ₂ ], [RA1210; H, H, F, Cl, i-Pr, Ph], [RA1211; H, H, F, Cl, i-Pr, Bn], [RA1212; H, H, F, Cl, i-Pr, CF ₃ ], [RA1213; H, H, F, Cl, i-Pr, CF ₃ CH ₂ ], [ RA1214; H, H, F, Cl, i-Pr, CF ₃ CF ₂ ], [RA1215; H, H, F, Cl, i-Pr, CF ₂ H], [RA1216; H, H, F, Cl , i-Pr, CF ₂ HCH ₂ ], [RA1217; H, H, Cl, H, i-Pr, Me], [RA1218; H, H, Cl, H, i-Pr, Et], [RA1219; H, H, Cl, H, i-Pr, Pr], [RA1220; H, H, Cl, H, i-Pr, i-Pr], [RA1221; H, H, Cl, H, i-Pr, c-Pr], [RA1222; H, H, Cl, H, i-Pr, Bu], [RA1223; H, H, Cl, H, i-Pr, i-Bu], [RA1224; H, H, Cl, H, i-Pr, t-Bu], [RA1225; H, H, Cl, H, i-Pr, c-PrCH ₂ ], [RA1226; H, H, Cl, H, i-Pr, Ph ], [RA1227; H, H, Cl, H, i-Pr, Bn], [RA1228; H, H, Cl, H, i-Pr, CF ₃ ], [RA1229; H, H, Cl, H, i-Pr, CF ₃ CH ₂ ], [RA1230; H, H, Cl, H, i-Pr, CF ₃ CF ₂ ], [RA1231; H, H, Cl, H, i-Pr, CF ₂ H] , [RA1232; H, H, Cl, H, i-Pr, CF ₂ HCH ₂ ], [RA1233; H, H, Cl, Cl, i-Pr, Me], [RA1234; H, H, Cl, Cl , i-Pr, Et], [RA1235; H, H, Cl, Cl, i- Pr, Pr], [RA1236; H, H, Cl, Cl, i-Pr, i-Pr], [RA1237; H, H, Cl, Cl, i-Pr, c-Pr], [RA1238; H, H, Cl, Cl, i-Pr, Bu], [RA1239; H, H, Cl, Cl, i-Pr, i-Bu], [RA1240; H, H, Cl, Cl, i-Pr, t- Bu], [RA1241; H, H, Cl, Cl, i-Pr, c-PrCH ₂ ], [RA1242; H, H, Cl, Cl, i-Pr, Ph], [RA1243; H, H, Cl , Cl, i-Pr, Bn], [RA1244; H, H, Cl, Cl, i-Pr, CF ₃ ], [RA1245; H, H, Cl, Cl, i-Pr, CF ₃ CH ₂ ], [RA1246; H, H, Cl, Cl, i-Pr, CF ₃ CF ₂ ], [RA1247; H, H, Cl, Cl, i-Pr, CF ₂ H], [RA1248; H, H, Cl, Cl, i-Pr, CF ₂ HCH ₂ ], [RA1249; H, H, Me, H, c-Pr, Me], [RA1250; H, H, Me, H, c-Pr, Et], [RA1251 ; H, H, Me, H, c-Pr, Pr], [RA1252; H, H, Me, H, c-Pr, i-Pr], [RA1253; H, H, Me, H, c-Pr , c-Pr], [RA1254; H, H, Me, H, c-Pr, Bu], [RA1255; H, H, Me, H, c-Pr, i-Bu], [RA1256; H, H , Me, H, c-Pr, t-Bu], [RA1257; H, H, Me, H, c-Pr, c-PrCH ₂ ], [RA1258; H, H, Me, H, c-Pr, Ph], [RA1259; H, H, Me, H, c-Pr, Bn], [RA1260; H, H, Me, H, c-Pr, CF ₃ ], [RA1261; H, H, Me, H , c-Pr, CF ₃ CH ₂ ], [RA1262; H, H, Me, H, c-Pr, CF ₃ CF ₂ ], [RA1263; H, H, Me, H, c-Pr, CF ₂ H ], [RA1264; H, H, Me, H, c-Pr, CF ₂ HCH ₂ ], [RA1265; H, H, Me, Me, c-Pr, Me], [RA1266; H, H, Me, Me, c-Pr, Et], [RA1267; H, H, Me, Me, c-Pr, Pr], [RA1268; H, H, Me, Me, c-Pr, i-Pr], [RA1269; H, H, Me, Me, c-Pr , c-Pr], [RA1270; H, H, Me, Me, c-Pr, Bu], [RA1271; H, H, Me, Me, c-Pr, i-Bu], [RA1272; H, H , Me, Me, c-Pr, t-Bu], [RA1273; H, H, Me, Me, c-Pr, c-PrCH ₂ ], [RA1274; H, H, Me, Me, c-Pr, Ph], [RA1275; H, H, Me, Me, c-Pr, Bn], [RA1276; H, H, Me, Me, c-Pr, CF ₃ ], [RA1277; H, H, Me, Me , c-Pr, CF ₃ CH ₂ ], [RA1278; H, H, Me, Me, c-Pr, CF ₃ CF ₂ ], [RA1279; H, H, Me, Me, c-Pr, CF ₂ H ], [RA1280; H, H, Me, Me, c-Pr, CF ₂ HCH ₂ ], [RA1281; H, H, Me, Et, c-Pr, Me], [RA1282; H, H, Me, Et, c-Pr, Et], [RA1283; H, H, Me, Et, c-Pr, Pr], [RA1284; H, H, Me, Et, c-Pr, i-Pr], [RA1285; H, H, Me, Et, c-Pr, c-Pr], [RA1286; H, H, Me, Et, c-Pr, Bu], [RA1287; H, H, Me, Et, c-Pr, i-Bu], [RA1288; H, H, Me, Et, c-Pr, t-Bu], [RA1289; H, H, Me, Et, c-Pr, c-PrCH ₂ ], [RA1290; H , H, Me, Et, c-Pr, Ph], [RA1291; H, H, Me, Et, c-Pr, Bn], [RA1292; H, H, Me, Et, c-Pr, CF ₃ ] , [RA1293; H, H, Me, Et, c-Pr, CF ₃ CH ₂ ], [RA1294; H, H, Me, Et, c-Pr, CF ₃ CF ₂ ], [RA1295; H, H, Me, Et, c-Pr, CF ₂ H], [RA1296; H, H, Me, Et, c-Pr, CF ₂ HCH ₂ ], [RA1297; H, H, Me, F, c-Pr, Me ], [RA1298; H, H, Me, F, c-Pr, Et], [RA1299; H, H, Me, F, c-Pr, Pr], [RA1300; H, H, Me, F, c -Pr, i-Pr], [RA1301; H, H, Me, F, c-Pr, c-Pr], [RA1302; H, H, Me, F, c-Pr, Bu], [RA1303; H , H, Me , F, c-Pr, i-Bu], [RA1304; H, H, Me, F, c-Pr, t-Bu], [RA1305; H, H, Me, F, c-Pr, c-PrCH ₂ ], [RA1306; H, H, Me, F, c-Pr, Ph], [RA1307; H, H, Me, F, c-Pr, Bn], [RA1308; H, H, Me, F, c-Pr, CF ₃ ], [RA1309; H, H, Me, F, c-Pr, CF ₃ CH ₂ ], [RA1310; H, H, Me, F, c-Pr, CF ₃ CF ₂ ], [RA1311; H, H, Me, F, c-Pr, CF ₂ H], [RA1312; H, H, Me, F, c-Pr, CF ₂ HCH ₂ ], [RA1313; H, H, Me, Cl, c-Pr, Me], [RA1314; H, H, Me, Cl, c-Pr, Et], [RA1315; H, H, Me, Cl, c-Pr, Pr], [RA1316; H, H, Me, Cl, c-Pr, i-Pr], [RA1317; H, H, Me, Cl, c-Pr, c-Pr], [RA1318; H, H, Me, Cl, c-Pr, Bu], [RA1319; H, H, Me, Cl, c-Pr, i-Bu], [RA1320; H, H, Me, Cl, c-Pr, t-Bu], [RA1321; H, H, Me, Cl, c-Pr, c-PrCH ₂ ], [RA1322; H, H, Me, Cl, c-Pr, Ph], [RA1323; H, H, Me, Cl, c-Pr, Bn], [RA1324; H, H, Me, Cl, c-Pr, CF ₃ ], [RA1325; H, H, Me, Cl, c-Pr, CF ₃ CH ₂ ], [RA1326; H, H, Me, Cl , c-Pr, CF ₃ CF ₂ ], [RA1327; H, H, Me, Cl, c-Pr, CF ₂ H], [RA1328; H, H, Me, Cl, c-Pr, CF ₂ HCH ₂ ], [RA1329; H, H, Et, H, c-Pr, Me], [RA1330; H, H, Et, H, c-Pr, Et], [RA1331; H, H, Et, H, c -Pr, Pr], [RA1332; H, H, Et, H, c-Pr, i-Pr], [RA1333; H, H, Et, H, c-Pr, c-Pr], [RA1334; H , H, Et, H, c-Pr, Bu], [RA1335; H, H, Et, H, c-Pr, i-Bu], [RA1336; H, H, Et, H, c-Pr, t -Bu], [RA1337; H, H, Et, H , c-Pr, c-PrCH 2], [RA1338; H, H, Et, H, c-Pr, Ph], [RA1339; H, H, Et, H, c-Pr, Bn], [RA1340; H, H, Et, H, c-Pr, CF ₃ ], [RA1341; H, H, Et, H, c-Pr, CF ₃ CH ₂ ], [RA1342; H, H, Et, H, c- Pr, CF ₃ CF ₂ ], [RA1343; H, H, Et, H, c-Pr, CF ₂ H], [RA1344; H, H, Et, H, c-Pr, CF ₂ HCH ₂ ], [ RA1345; H, H, Et, F, c-Pr, Me], [RA1346; H, H, Et, F, c-Pr, Et], [RA1347; H, H, Et, F, c-Pr, Pr], [RA1348; H, H, Et, F, c-Pr, i-Pr], [RA1349; H, H, Et, F, c-Pr, c-Pr], [RA1350; H, H, Et, F, c-Pr, Bu], [RA1351; H, H, Et, F, c-Pr, i-Bu], [RA1352; H, H, Et, F, c-Pr, t-Bu] , [RA1353; H, H, Et, F, c-Pr, c-PrCH ₂ ], [RA1354; H, H, Et, F, c-Pr, Ph], [RA1355; H, H, Et, F , c-Pr, Bn], [RA1356; H, H, Et, F, c-Pr, CF ₃ ], [RA1357; H, H, Et, F, c-Pr, CF ₃ CH ₂ ], [RA1358 ; H, H, Et, F, c-Pr, CF ₃ CF ₂ ], [RA1359; H, H, Et, F, c-Pr, CF ₂ H], [RA1360; H, H, Et, F, c-Pr, CF ₂ HCH ₂ ], [RA1361; H, H, Et, Cl, c-Pr, Me], [RA1362; H, H, Et, Cl, c-Pr, Et], [RA1363; H , H, Et, Cl, c-Pr, Pr], [RA1364; H, H, Et, Cl, c-Pr, i-Pr], [RA1365; H, H, Et, Cl, c-Pr, c -Pr], [RA1366; H, H, Et, Cl, c-Pr, Bu], [RA1367; H, H, Et, Cl, c-Pr, i-Bu], [RA1368; H, H, Et , Cl, c-Pr, t-Bu], [RA1369; H, H, Et, Cl, c-Pr, c-PrCH ₂ ], [RA1370; H, H, Et, Cl, c-Pr, Ph] , [RA1371; H, H, Et, Cl, cP r, Bn], [RA1372; H, H, Et, Cl, c-Pr, CF ₃ ], [RA1373; H, H, Et, Cl, c-Pr, CF ₃ CH ₂ ], [RA1374; H, H, Et, Cl, c-Pr, CF ₃ CF ₂ ], [RA1375; H, H, Et, Cl, c-Pr, CF ₂ H], [RA1376; H, H, Et, Cl, c-Pr , CF ₂ HCH ₂ ], [RA1377; H, H, F, H, c-Pr, Me], [RA1378; H, H, F, H, c-Pr, Et], [RA1379; H, H, F, H, c-Pr, Pr], [RA1380; H, H, F, H, c-Pr, i-Pr], [RA1381; H, H, F, H, c-Pr, c-Pr] , [RA1382; H, H, F, H, c-Pr, Bu], [RA1383; H, H, F, H, c-Pr, i-Bu], [RA1384; H, H, F, H, c-Pr, t-Bu], [RA1385; H, H, F, H, c-Pr, c-PrCH ₂ ], [RA1386; H, H, F, H, c-Pr, Ph], [RA1387 ; H, H, F, H, c-Pr, Bn], [RA1388; H, H, F, H, c-Pr, CF ₃ ], [RA1389; H, H, F, H, c-Pr, CF ₃ CH ₂ ], [RA1390; H, H, F, H, c-Pr, CF ₃ CF ₂ ], [RA1391; H, H, F, H, c-Pr, CF ₂ H], [RA1392; H, H, F, H, c-Pr, CF ₂ HCH ₂ ], [RA1393; H, H, F, F, c-Pr, Me], [RA1394; H, H, F, F, c-Pr , Et], [RA1395; H, H, F, F, c-Pr, Pr], [RA1396; H, H, F, F, c-Pr, i-Pr], [RA1397; H, H, F , F, c-Pr, c-Pr], [RA1398; H, H, F, F, c-Pr, Bu], [RA1399; H, H, F, F, c-Pr, i-Bu], [RA1400; H, H, F, F, c-Pr, t-Bu],

[RA1401; H, H, F, F, c-Pr, c-PrCH ₂ ], [RA1402; H, H, F, F, c-Pr, Ph], [RA1403; H, H, F, F, c-Pr, Bn], [RA1404; H, H, F, F, c-Pr, CF ₃ ], [RA1405; H, H, F, F, c-Pr, CF ₃ CH ₂ ], [RA1406; H, H, F, F, c-Pr, CF ₃ CF ₂ ], [RA1407; H, H, F, F, c-Pr, CF ₂ H], [RA1408; H, H, F, F, c -Pr, CF ₂ HCH ₂ ], [RA1409; H, H, F, Cl, c-Pr, Me], [RA1410; H, H, F, Cl, c-Pr, Et], [RA1411; H, H, F, Cl, c-Pr, Pr], [RA1412; H, H, F, Cl, c-Pr, i-Pr], [RA1413; H, H, F, Cl, c-Pr, c- Pr], [RA1414; H, H, F, Cl, c-Pr, Bu], [RA1415; H, H, F, Cl, c-Pr, i-Bu], [RA1416; H, H, F, Cl, c-Pr, t-Bu], [RA1417; H, H, F, Cl, c-Pr, c-PrCH ₂ ], [RA1418; H, H, F, Cl, c-Pr, Ph], [RA1419; H, H, F, Cl, c-Pr, Bn], [RA1420; H, H, F, Cl, c-Pr, CF ₃ ], [RA1421; H, H, F, Cl, c- Pr, CF ₃ CH ₂ ], [RA1422; H, H, F, Cl, c-Pr, CF ₃ CF ₂ ], [RA1423; H, H, F, Cl, c-Pr, CF ₂ H], [ RA1424; H, H, F, Cl, c-Pr, CF ₂ HCH ₂ ], [RA1425; H, H, Cl, H, c-Pr, Me], [RA1426; H, H, Cl, H, c -Pr, Et], [RA1427; H, H, Cl, H, c-Pr, Pr], [RA1428; H, H, Cl, H, c-Pr, i-Pr], [RA1429; H, H , Cl, H, c-Pr, c-Pr], [RA1430; H, H, Cl, H, c-Pr, Bu], [RA1431; H, H, Cl, H, c-Pr, i-Bu ], [RA1432; H, H, Cl, H, c-Pr, t-Bu], [RA1433; H, H, Cl, H, c-Pr, c-PrCH ₂ ], [RA1434; H, H, Cl, H, c-Pr, Ph], [RA1435; H, H, Cl, H, c-Pr, B n], [RA1436; H, H, Cl, H, c-Pr, CF ₃ ], [RA1437; H, H, Cl, H, c-Pr, CF ₃ CH ₂ ], [RA1438; H, H, Cl, H, c-Pr, CF ₃ CF ₂ ], [RA1439; H, H, Cl, H, c-Pr, CF ₂ H], [RA1440; H, H, Cl, H, c-Pr, CF ₂ HCH ₂ ], [RA1441; H, H, Cl, Cl, c-Pr, Me], [RA1442; H, H, Cl, Cl, c-Pr, Et], [RA1443; H, H, Cl, Cl, c-Pr, Pr], [RA1444; H, H, Cl, Cl, c-Pr, i-Pr], [RA1445; H, H, Cl, Cl, c-Pr, c-Pr], [ RA1446; H, H, Cl, Cl, c-Pr, Bu], [RA1447; H, H, Cl, Cl, c-Pr, i-Bu], [RA1448; H, H, Cl, Cl, c- Pr, t-Bu], [RA1449; H, H, Cl, Cl, c-Pr, c-PrCH ₂ ], [RA1450; H, H, Cl, Cl, c-Pr, Ph], [RA1451; H , H, Cl, Cl, c-Pr, Bn], [RA1452; H, H, Cl, Cl, c-Pr, CF ₃ ], [RA1453; H, H, Cl, Cl, c-Pr, CF ₃ CH ₂ ], [RA1454; H, H, Cl, Cl, c-Pr, CF ₃ CF ₂ ], [RA1455; H, H, Cl, Cl, c-Pr, CF ₂ H], [RA1456; H, H, Cl, Cl, c-Pr, CF ₂ HCH ₂ ], [RA1457; H, H, Me, H, i-Bu, Me], [RA1458; H, H, Me, H, i-Bu, Et ], [RA1459; H, H, Me, H, i-Bu, Pr], [RA1460; H, H, Me, H, i-Bu, i-Pr], [RA1461; H, H, Me, H , i-Bu, c-Pr], [RA1462; H, H, Me, H, i-Bu, Bu], [RA1463; H, H, Me, H, i-Bu, i-Bu], [RA1464 ; H, H, Me, H, i-Bu, t-Bu], [RA1465; H, H, Me, H, i-Bu, c-PrCH ₂ ], [RA1466; H, H, Me, H, i-Bu, Ph], [RA1467; H, H, Me, H, i-Bu, Bn], [RA1468; H, H, Me, H, i-Bu, CF ₃ ], [RA1469; H, H , Me, H, i-Bu, CF ₃ CH ₂ ], [RA1470; H, H, Me, H, i-Bu, CF ₃ CF ₂ ], [RA1471; H, H, Me, H, i-Bu, CF ₂ H], [RA1472; H, H, Me, H, i-Bu, CF ₂ HCH ₂ ], [RA1473; H, H, Me, Me, i-Bu, Me], [RA1474; H, H, Me, Me, i-Bu, Et ], [RA1475; H, H, Me, Me, i-Bu, Pr], [RA1476; H, H, Me, Me, i-Bu, i-Pr], [RA1477; H, H, Me, Me , i-Bu, c-Pr], [RA1478; H, H, Me, Me, i-Bu, Bu], [RA1479; H, H, Me, Me, i-Bu, i-Bu], [RA1480 ; H, H, Me, Me, i-Bu, t-Bu], [RA1481; H, H, Me, Me, i-Bu, c-PrCH ₂ ], [RA1482; H, H, Me, Me, i-Bu, Ph], [RA1483; H, H, Me, Me, i-Bu, Bn], [RA1484; H, H, Me, Me, i-Bu, CF ₃ ], [RA1485; H, H , Me, Me, i-Bu, CF ₃ CH ₂ ], [RA1486; H, H, Me, Me, i-Bu, CF ₃ CF ₂ ], [RA1487; H, H, Me, Me, i-Bu , CF ₂ H], [RA1488; H, H, Me, Me, i-Bu, CF ₂ HCH ₂ ], [RA1489; H, H, Me, Et, i-Bu, Me], [RA1490; H, H, Me, Et, i-Bu, Et], [RA1491; H, H, Me, Et, i-Bu, Pr], [RA1492; H, H, Me, Et, i-Bu, i-Pr] , [RA1493; H, H, Me, Et, i-Bu, c-Pr], [RA1494; H, H, Me, Et, i-Bu, Bu], [RA1495; H, H, Me, Et, i-Bu, i-Bu], [RA1496; H, H, Me, Et, i-Bu, t-Bu], [RA1497; H, H, Me, Et, i-Bu, c-PrCH ₂ ], [RA1498; H, H, Me, Et, i-Bu, Ph], [RA1499; H, H, Me, Et, i-Bu, Bn], [RA1500; H, H, Me, Et, i-Bu , CF ₃ ], [RA1501; H, H, Me, Et, i-Bu, CF ₃ CH ₂ ], [RA1502; H, H, Me, Et, i-Bu, CF ₃ CF ₂ ], [R A1503; H, H, Me, Et, i-Bu, CF ₂ H], [RA1504; H, H, Me, Et, i-Bu, CF ₂ HCH ₂ ], [RA1505; H, H, Me, F , i-Bu, Me], [RA1506; H, H, Me, F, i-Bu, Et], [RA1507; H, H, Me, F, i-Bu, Pr], [RA1508; H, H , Me, F, i-Bu, i-Pr], [RA1509; H, H, Me, F, i-Bu, c-Pr], [RA1510; H, H, Me, F, i-Bu, Bu ], [RA1511; H, H, Me, F, i-Bu, i-Bu], [RA1512; H, H, Me, F, i-Bu, t-Bu], [RA1513; H, H, Me , F, i-Bu, c-PrCH ₂ ], [RA1514; H, H, Me, F, i-Bu, Ph], [RA1515; H, H, Me, F, i-Bu, Bn], [ RA1516; H, H, Me, F, i-Bu, CF ₃ ], [RA1517; H, H, Me, F, i-Bu, CF ₃ CH ₂ ], [RA1518; H, H, Me, F, i-Bu, CF ₃ CF ₂ ], [RA1519; H, H, Me, F, i-Bu, CF ₂ H], [RA1520; H, H, Me, F, i-Bu, CF ₂ HCH ₂ ] , [RA1521; H, H, Me, Cl, i-Bu, Me], [RA1522; H, H, Me, Cl, i-Bu, Et], [RA1523; H, H, Me, Cl, i- Bu, Pr], [RA1524; H, H, Me, Cl, i-Bu, i-Pr], [RA1525; H, H, Me, Cl, i-Bu, c-Pr], [RA1526; H, H, Me, Cl, i-Bu, Bu], [RA1527; H, H, Me, Cl, i-Bu, i-Bu], [RA1528; H, H, Me, Cl, i-Bu, t- Bu], [RA1529; H, H, Me, Cl, i-Bu, c-PrCH ₂ ], [RA1530; H, H, Me, Cl, i-Bu, Ph], [RA1531; H, H, Me , Cl, i-Bu, Bn], [RA1532; H, H, Me, Cl, i-Bu, CF ₃ ], [RA1533; H, H, Me, Cl, i-Bu, CF ₃ CH ₂ ], [RA1534; H, H, Me, Cl, i-Bu, CF ₃ CF ₂ ], [RA1535; H, H, Me, Cl, i-Bu, CF ₂ H], [RA1536; H, H, Me, Cl, i-Bu, CF ₂ H CH ₂ ], [RA1537; H, H, Et, H, i-Bu, Me], [RA1538; H, H, Et, H, i-Bu, Et], [RA1539; H, H, Et, H , i-Bu, Pr], [RA1540; H, H, Et, H, i-Bu, i-Pr], [RA1541; H, H, Et, H, i-Bu, c-Pr], [RA1542 ; H, H, Et, H, i-Bu, Bu], [RA1543; H, H, Et, H, i-Bu, i-Bu], [RA1544; H, H, Et, H, i-Bu , t-Bu], [RA1545; H, H, Et, H, i-Bu, c-PrCH ₂ ], [RA1546; H, H, Et, H, i-Bu, Ph], [RA1547; H, H, Et, H, i-Bu, Bn], [RA1548; H, H, Et, H, i-Bu, CF ₃ ], [RA1549; H, H, Et, H, i-Bu, CF ₃ CH ₂ ], [RA1550; H, H, Et, H, i-Bu, CF ₃ CF ₂ ], [RA1551; H, H, Et, H, i-Bu, CF ₂ H], [RA1552; H, H , Et, H, i-Bu, CF ₂ HCH ₂ ], [RA1553; H, H, Et, F, i-Bu, Me], [RA1554; H, H, Et, F, i-Bu, Et] , [RA1555; H, H, Et, F, i-Bu, Pr], [RA1556; H, H, Et, F, i-Bu, i-Pr], [RA1557; H, H, Et, F, i-Bu, c-Pr], [RA1558; H, H, Et, F, i-Bu, Bu], [RA1559; H, H, Et, F, i-Bu, i-Bu], [RA1560; H, H, Et, F, i-Bu, t-Bu], [RA1561; H, H, Et, F, i-Bu, c-PrCH ₂ ], [RA1562; H, H, Et, F, i -Bu, Ph], [RA1563; H, H, Et, F, i-Bu, Bn], [RA1564; H, H, Et, F, i-Bu, CF ₃ ], [RA1565; H, H, Et, F, i-Bu, CF ₃ CH ₂ ], [RA1566; H, H, Et, F, i-Bu, CF ₃ CF ₂ ], [RA1567; H, H, Et, F, i-Bu, CF ₂ H], [RA1568; H, H, Et, F, i-Bu, CF ₂ HCH ₂ ], [RA1569; H, H, Et, Cl, i-Bu, Me], [RA1570; H, H , Et, Cl, i-Bu, Et], [RA1571; H, H, E t, Cl, i-Bu, Pr], [RA1572; H, H, Et, Cl, i-Bu, i-Pr], [RA1573; H, H, Et, Cl, i-Bu, c-Pr] , [RA1574; H, H, Et, Cl, i-Bu, Bu], [RA1575; H, H, Et, Cl, i-Bu, i-Bu], [RA1576; H, H, Et, Cl, i-Bu, t-Bu], [RA1577; H, H, Et, Cl, i-Bu, c-PrCH ₂ ], [RA1578; H, H, Et, Cl, i-Bu, Ph], [RA1579 ; H, H, Et, Cl, i-Bu, Bn], [RA1580; H, H, Et, Cl, i-Bu, CF ₃ ], [RA1581; H, H, Et, Cl, i-Bu, CF ₃ CH ₂ ], [RA1582; H, H, Et, Cl, i-Bu, CF ₃ CF ₂ ], [RA1583; H, H, Et, Cl, i-Bu, CF ₂ H], [RA1584; H, H, Et, Cl, i-Bu, CF ₂ HCH ₂ ], [RA1585; H, H, F, H, i-Bu, Me], [RA1586; H, H, F, H, i-Bu , Et], [RA1587; H, H, F, H, i-Bu, Pr], [RA1588; H, H, F, H, i-Bu, i-Pr], [RA1589; H, H, F , H, i-Bu, c-Pr], [RA1590; H, H, F, H, i-Bu, Bu], [RA1591; H, H, F, H, i-Bu, i-Bu], [RA1592; H, H, F, H, i-Bu, t-Bu], [RA1593; H, H, F, H, i-Bu, c-PrCH ₂ ], [RA1594; H, H, F, H, i-Bu, Ph], [RA1595; H, H, F, H, i-Bu, Bn], [RA1596; H, H, F, H, i-Bu, CF ₃ ], [RA1597; H , H, F, H, i-Bu, CF ₃ CH ₂ ], [RA1598; H, H, F, H, i-Bu, CF ₃ CF ₂ ], [RA1599; H, H, F, H, i -Bu, CF ₂ H], [RA1600; H, H, F, H, i-Bu, CF ₂ HCH ₂ ],

[RA1601; H, H, F, F, i-Bu, Me], [RA1602; H, H, F, F, i-Bu, Et], [RA1603; H, H, F, F, i-Bu , Pr], [RA1604; H, H, F, F, i-Bu, i-Pr], [RA1605; H, H, F, F, i-Bu, c-Pr], [RA1606; H, H , F, F, i-Bu, Bu], [RA1607; H, H, F, F, i-Bu, i-Bu], [RA1608; H, H, F, F, i-Bu, t-Bu ], [RA1609; H, H, F, F, i-Bu, c-PrCH ₂ ], [RA1610; H, H, F, F, i-Bu, Ph], [RA1611; H, H, F, F, i-Bu, Bn], [RA1612; H, H, F, F, i-Bu, CF ₃ ], [RA1613; H, H, F, F, i-Bu, CF ₃ CH ₂ ], [ RA1614; H, H, F, F, i-Bu, CF ₃ CF ₂ ], [RA1615; H, H, F, F, i-Bu, CF ₂ H], [RA1616; H, H, F, F , i-Bu, CF ₂ HCH ₂ ], [RA1617; H, H, F, Cl, i-Bu, Me], [RA1618; H, H, F, Cl, i-Bu, Et], [RA1619; H, H, F, Cl, i-Bu, Pr], [RA1620; H, H, F, Cl, i-Bu, i-Pr], [RA1621; H, H, F, Cl, i-Bu, c-Pr], [RA1622; H, H, F, Cl, i-Bu, Bu], [RA1623; H, H, F, Cl, i-Bu, i-Bu], [RA1624; H, H, F, Cl, i-Bu, t-Bu], [RA1625; H, H, F, Cl, i-Bu, c-PrCH ₂ ], [RA1626; H, H, F, Cl, i-Bu, Ph ], [RA1627; H, H, F, Cl, i-Bu, Bn], [RA1628; H, H, F, Cl, i-Bu, CF ₃ ], [RA1629; H, H, F, Cl, i-Bu, CF ₃ CH ₂ ], [RA1630; H, H, F, Cl, i-Bu, CF ₃ CF ₂ ], [RA1631; H, H, F, Cl, i-Bu, CF ₂ H] , [RA1632; H, H, F, Cl, i-Bu, CF ₂ HCH ₂ ], [RA1633; H, H, Cl, H, i-Bu, Me], [RA1634; H, H, Cl, H , i-Bu, Et], [RA1635; H, H, Cl, H, i-Bu, Pr], [RA1636; H, H, Cl, H, i-Bu, i-Pr], [RA1637; H, H, Cl, H, i-Bu, c-Pr], [RA1638; H, H, Cl, H, i-Bu, Bu] , [RA1639; H, H, Cl, H, i-Bu, i-Bu], [RA1640; H, H, Cl, H, i-Bu, t-Bu], [RA1641; H, H, Cl, H, i-Bu, c-PrCH ₂ ], [RA1642; H, H, Cl, H, i-Bu, Ph], [RA1643; H, H, Cl, H, i-Bu, Bn], [RA1644 ; H, H, Cl, H, i-Bu, CF ₃ ], [RA1645; H, H, Cl, H, i-Bu, CF ₃ CH ₂ ], [RA1646; H, H, Cl, H, i -Bu, CF ₃ CF ₂ ], [RA1647; H, H, Cl, H, i-Bu, CF ₂ H], [RA1648; H, H, Cl, H, i-Bu, CF ₂ HCH ₂ ], [RA1649; H, H, Cl, Cl, i-Bu, Me], [RA1650; H, H, Cl, Cl, i-Bu, Et], [RA1651; H, H, Cl, Cl, i-Bu , Pr], [RA1652; H, H, Cl, Cl, i-Bu, i-Pr], [RA1653; H, H, Cl, Cl, i-Bu, c-Pr], [RA1654; H, H , Cl, Cl, i-Bu, Bu], [RA1655; H, H, Cl, Cl, i-Bu, i-Bu], [RA1656; H, H, Cl, Cl, i-Bu, t-Bu ], [RA1657; H, H, Cl, Cl, i-Bu, c-PrCH ₂ ], [RA1658; H, H, Cl, Cl, i-Bu, Ph], [RA1659; H, H, Cl, Cl, i-Bu, Bn], [RA1660; H, H, Cl, Cl, i-Bu, CF ₃ ], [RA1661; H, H, Cl, Cl, i-Bu, CF ₃ CH ₂ ], [ RA1662; H, H, Cl, Cl, i-Bu, CF ₃ CF ₂ ], [RA1663; H, H, Cl, Cl, i-Bu, CF ₂ H], [RA1664; H, H, Cl, Cl , i-Bu, CF ₂ HCH ₂ ], [RA1665; H, H, Me, H, t-Bu, Me], [RA1666; H, H, Me, H, t-Bu, Et], [RA1667; H, H, Me, H, t-Bu, Pr], [RA1668; H, H, Me, H, t-Bu, i-Pr], [RA1669; H, H, Me, H, t-Bu, c-Pr], [RA1670; H, H, Me , H, t-Bu, Bu], [RA1671; H, H, Me, H, t-Bu, i-Bu], [RA1672; H, H, Me, H, t-Bu, t-Bu], [RA1673; H, H, Me, H, t-Bu, c-PrCH ₂ ], [RA1674; H, H, Me, H, t-Bu, Ph], [RA1675; H, H, Me, H, t-Bu, Bn], [RA1676; H, H, Me, H, t-Bu, CF ₃ ], [RA1677; H, H, Me, H, t-Bu, CF ₃ CH ₂ ], [RA1678; H, H, Me, H, t-Bu, CF ₃ CF ₂ ], [RA1679; H, H, Me, H, t-Bu, CF ₂ H], [RA1680; H, H, Me, H, t -Bu, CF ₂ HCH ₂ ], [RA1681; H, H, Me, Me, t-Bu, Me], [RA1682; H, H, Me, Me, t-Bu, Et], [RA1683; H, H, Me, Me, t-Bu, Pr], [RA1684; H, H, Me, Me, t-Bu, i-Pr], [RA1685; H, H, Me, Me, t-Bu, c- Pr], [RA1686; H, H, Me, Me, t-Bu, Bu], [RA1687; H, H, Me, Me, t-Bu, i-Bu], [RA1688; H, H, Me, Me, t-Bu, t-Bu], [RA1689; H, H, Me, Me, t-Bu, c-PrCH ₂ ], [RA1690; H, H, Me, Me, t-Bu, Ph], [RA1691; H, H, Me, Me, t-Bu, Bn], [RA1692; H, H, Me, Me, t-Bu, CF ₃ ], [RA1693; H, H, Me, Me, t- Bu, CF ₃ CH ₂ ], [RA1694; H, H, Me, Me, t-Bu, CF ₃ CF ₂ ], [RA1695; H, H, Me, Me, t-Bu, CF ₂ H], [ RA1696; H, H, Me, Me, t-Bu, CF ₂ HCH ₂ ], [RA1697; H, H, Me, Et, t-Bu, Me], [RA1698; H, H, Me, Et, t -Bu, Et], [RA1699; H, H, Me, Et, t-Bu, Pr], [RA1700; H, H, Me, Et, t-Bu, i-Pr], [RA1701; H, H , Me, Et, t-Bu, c-Pr], [RA1702; H, H, Me, Et, t-Bu, Bu], [RA1703; H, H, Me, Et, t-Bu, i-Bu ], [RA1704; H, H , Me, Et, t-Bu, t-Bu], [RA1705; H, H, Me, Et, t-Bu, c-PrCH ₂ ], [RA1706; H, H, Me, Et, t-Bu, Ph], [RA1707; H, H, Me, Et, t-Bu, Bn], [RA1708; H, H, Me, Et, t-Bu, CF ₃ ], [RA1709; H, H, Me, Et , t-Bu, CF ₃ CH ₂ ], [RA1710; H, H, Me, Et, t-Bu, CF ₃ CF ₂ ], [RA1711; H, H, Me, Et, t-Bu, CF ₂ H ], [RA1712; H, H, Me, Et, t-Bu, CF ₂ HCH ₂ ], [RA1713; H, H, Me, F, t-Bu, Me], [RA1714; H, H, Me, F, t-Bu, Et], [RA1715; H, H, Me, F, t-Bu, Pr], [RA1716; H, H, Me, F, t-Bu, i-Pr], [RA1717; H, H, Me, F, t-Bu, c-Pr], [RA1718; H, H, Me, F, t-Bu, Bu], [RA1719; H, H, Me, F, t-Bu, i-Bu], [RA1720; H, H, Me, F, t-Bu, t-Bu], [RA1721; H, H, Me, F, t-Bu, c-PrCH ₂ ], [RA1722; H , H, Me, F, t-Bu, Ph], [RA1723; H, H, Me, F, t-Bu, Bn], [RA1724; H, H, Me, F, t-Bu, CF ₃ ] , [RA1725; H, H, Me, F, t-Bu, CF ₃ CH ₂ ], [RA1726; H, H, Me, F, t-Bu, CF ₃ CF ₂ ], [RA1727; H, H, Me, F, t-Bu, CF ₂ H], [RA1728; H, H, Me, F, t-Bu, CF ₂ HCH ₂ ], [RA1729; H, H, Me, Cl, t-Bu, Me ], [RA1730; H, H, Me, Cl, t-Bu, Et], [RA1731; H, H, Me, Cl, t-Bu, Pr], [RA1732; H, H, Me, Cl, t -Bu, i-Pr], [RA1733; H, H, Me, Cl, t-Bu, c-Pr], [RA1734; H, H, Me, Cl, t-Bu, Bu], [RA1735; H , H, Me, Cl, t-Bu, i-Bu], [RA1736; H, H, Me, Cl, t-Bu, t-Bu], [RA1737; H, H, Me, Cl, t-Bu , c-PrCH ₂ ], [RA173 8; H, H, Me, Cl, t-Bu, Ph], [RA1739; H, H, Me, Cl, t-Bu, Bn], [RA1740; H, H, Me, Cl, t-Bu, CF ₃ ], [RA1741; H, H, Me, Cl, t-Bu, CF ₃ CH ₂ ], [RA1742; H, H, Me, Cl, t-Bu, CF ₃ CF ₂ ], [RA1743; H , H, Me, Cl, t-Bu, CF ₂ H], [RA1744; H, H, Me, Cl, t-Bu, CF ₂ HCH ₂ ], [RA1745; H, H, Et, H, t- Bu, Me], [RA1746; H, H, Et, H, t-Bu, Et], [RA1747; H, H, Et, H, t-Bu, Pr], [RA1748; H, H, Et, H, t-Bu, i-Pr], [RA1749; H, H, Et, H, t-Bu, c-Pr], [RA1750; H, H, Et, H, t-Bu, Bu], [ RA1751; H, H, Et, H, t-Bu, i-Bu], [RA1752; H, H, Et, H, t-Bu, t-Bu], [RA1753; H, H, Et, H, t-Bu, c-PrCH ₂ ], [RA1754; H, H, Et, H, t-Bu, Ph], [RA1755; H, H, Et, H, t-Bu, Bn], [RA1756; H , H, Et, H, t-Bu, CF ₃ ], [RA1757; H, H, Et, H, t-Bu, CF ₃ CH ₂ ], [RA1758; H, H, Et, H, t-Bu , CF ₃ CF ₂ ], [RA1759; H, H, Et, H, t-Bu, CF ₂ H], [RA1760; H, H, Et, H, t-Bu, CF ₂ HCH ₂ ], [RA1761 ; H, H, Et, F, t-Bu, Me], [RA1762; H, H, Et, F, t-Bu, Et], [RA1763; H, H, Et, F, t-Bu, Pr ], [RA1764; H, H, Et, F, t-Bu, i-Pr], [RA1765; H, H, Et, F, t-Bu, c-Pr], [RA1766; H, H, Et , F, t-Bu, Bu], [RA1767; H, H, Et, F, t-Bu, i-Bu], [RA1768; H, H, Et, F, t-Bu, t-Bu], [RA1769; H, H, Et, F, t-Bu, c-PrCH ₂ ], [RA1770; H, H, Et, F, t-Bu, Ph], [RA1771; H, H, Et, F, t-Bu, Bn], [RA1772; H, H, Et, F, t-Bu , CF ₃ ], [RA1773; H, H, Et, F, t-Bu, CF ₃ CH ₂ ], [RA1774; H, H, Et, F, t-Bu, CF ₃ CF ₂ ], [RA1775; H, H, Et, F, t-Bu, CF ₂ H], [RA1776; H, H, Et, F, t-Bu, CF ₂ HCH ₂ ], [RA1777; H, H, Et, Cl, t -Bu, Me], [RA1778; H, H, Et, Cl, t-Bu, Et], [RA1779; H, H, Et, Cl, t-Bu, Pr], [RA1780; H, H, Et , Cl, t-Bu, i-Pr], [RA1781; H, H, Et, Cl, t-Bu, c-Pr], [RA1782; H, H, Et, Cl, t-Bu, Bu], [RA1783; H, H, Et, Cl, t-Bu, i-Bu], [RA1784; H, H, Et, Cl, t-Bu, t-Bu], [RA1785; H, H, Et, Cl , t-Bu, c-PrCH ₂ ], [RA1786; H, H, Et, Cl, t-Bu, Ph], [RA1787; H, H, Et, Cl, t-Bu, Bn], [RA1788; H, H, Et, Cl, t-Bu, CF ₃ ], [RA1789; H, H, Et, Cl, t-Bu, CF ₃ CH ₂ ], [RA1790; H, H, Et, Cl, t- Bu, CF ₃ CF ₂ ], [RA1791; H, H, Et, Cl, t-Bu, CF ₂ H], [RA1792; H, H, Et, Cl, t-Bu, CF ₂ HCH ₂ ], [ RA1793; H, H, F, H, t-Bu, Me], [RA1794; H, H, F, H, t-Bu, Et], [RA1795; H, H, F, H, t-Bu, Pr], [RA1796; H, H, F, H, t-Bu, i-Pr], [RA1797; H, H, F, H, t-Bu, c-Pr], [RA1798; H, H, F, H, t-Bu, Bu], [RA1799; H, H, F, H, t-Bu, i-Bu], [RA1800; H, H, F, H, t-Bu, t-Bu] ,

[RA1801; H, H, F, H, t-Bu, c-PrCH ₂ ], [RA1802; H, H, F, H, t-Bu, Ph], [RA1803; H, H, F, H, t-Bu, Bn], [RA1804; H, H, F, H, t-Bu, CF ₃ ], [RA1805; H, H, F, H, t-Bu, CF ₃ CH ₂ ], [RA1806; H, H, F, H, t-Bu, CF ₃ CF ₂ ], [RA1807; H, H, F, H, t-Bu, CF ₂ H], [RA1808; H, H, F, H, t -Bu, CF ₂ HCH ₂ ], [RA1809; H, H, F, F, t-Bu, Me], [RA1810; H, H, F, F, t-Bu, Et], [RA1811; H, H, F, F, t-Bu, Pr], [RA1812; H, H, F, F, t-Bu, i-Pr], [RA1813; H, H, F, F, t-Bu, c- Pr], [RA1814; H, H, F, F, t-Bu, Bu], [RA1815; H, H, F, F, t-Bu, i-Bu], [RA1816; H, H, F, F, t-Bu, t-Bu], [RA1817; H, H, F, F, t-Bu, c-PrCH ₂ ], [RA1818; H, H, F, F, t-Bu, Ph], [RA1819; H, H, F, F, t-Bu, Bn], [RA1820; H, H, F, F, t-Bu, CF ₃ ], [RA1821; H, H, F, F, t- Bu, CF ₃ CH ₂ ], [RA1822; H, H, F, F, t-Bu, CF ₃ CF ₂ ], [RA1823; H, H, F, F, t-Bu, CF ₂ H], [ RA1824; H, H, F, F, t-Bu, CF ₂ HCH ₂ ], [RA1825; H, H, F, Cl, t-Bu, Me], [RA1826; H, H, F, Cl, t -Bu, Et], [RA1827; H, H, F, Cl, t-Bu, Pr], [RA1828; H, H, F, Cl, t-Bu, i-Pr], [RA1829; H, H , F, Cl, t-Bu, c-Pr], [RA1830; H, H, F, Cl, t-Bu, Bu], [RA1831; H, H, F, Cl, t-Bu, i-Bu ], [RA1832; H, H, F, Cl, t-Bu, t-Bu], [RA1833; H, H, F, Cl, t-Bu, c-PrCH ₂ ], [RA1834; H, H, F, Cl, t-Bu, Ph], [RA1835; H, H, F, Cl, t-Bu, Bn], [RA1836; H, H, F , Cl, t-Bu, CF ₃ ], [RA1837; H, H, F, Cl, t-Bu, CF ₃ CH ₂ ], [RA1838; H, H, F, Cl, t-Bu, CF ₃ CF ₂ ], [RA1839; H, H, F, Cl, t-Bu, CF ₂ H], [RA1840; H, H, F, Cl, t-Bu, CF ₂ HCH ₂ ], [RA1841; H, H , Cl, H, t-Bu, Me], [RA1842; H, H, Cl, H, t-Bu, Et], [RA1843; H, H, Cl, H, t-Bu, Pr], [RA1844 ; H, H, Cl, H, t-Bu, i-Pr], [RA1845; H, H, Cl, H, t-Bu, c-Pr], [RA1846; H, H, Cl, H, t -Bu, Bu], [RA1847; H, H, Cl, H, t-Bu, i-Bu], [RA1848; H, H, Cl, H, t-Bu, t-Bu], [RA1849; H , H, Cl, H, t-Bu, c-PrCH ₂ ], [RA1850; H, H, Cl, H, t-Bu, Ph], [RA1851; H, H, Cl, H, t-Bu, Bn], [RA1852; H, H, Cl, H, t-Bu, CF ₃ ], [RA1853; H, H, Cl, H, t-Bu, CF ₃ CH ₂ ], [RA1854; H, H, Cl, H, t-Bu, CF ₃ CF ₂ ], [RA1855; H, H, Cl, H, t-Bu, CF ₂ H], [RA1856; H, H, Cl, H, t-Bu, CF ₂ HCH ₂ ], [RA1857; H, H, Cl, Cl, t-Bu, Me], [RA1858; H, H, Cl, Cl, t-Bu, Et], [RA1859; H, H, Cl, Cl, t-Bu, Pr], [RA1860; H, H, Cl, Cl, t-Bu, i-Pr], [RA1861; H, H, Cl, Cl, t-Bu, c-Pr], [ RA1862; H, H, Cl, Cl, t-Bu, Bu], [RA1863; H, H, Cl, Cl, t-Bu, i-Bu], [RA1864; H, H, Cl, Cl, t- Bu, t-Bu], [RA1865; H, H, Cl, Cl, t-Bu, c-PrCH ₂ ], [RA1866; H, H, Cl, Cl, t-Bu, Ph], [RA1867; H , H, Cl, Cl, t-Bu, Bn], [RA1868; H, H, Cl, Cl, t-Bu, CF ₃ ], [RA1869; H, H, Cl, Cl, t-Bu, CF ₃ CH ₂ ], [RA1870; H, H , Cl, Cl, t-Bu, CF ₃ CF ₂ ], [RA1871; H, H, Cl, Cl, t-Bu, CF ₂ H], [RA1872; H, H, Cl, Cl, t-Bu, CF ₂ HCH ₂ ], [RA1873; H, H, Me, H, CF ₂ H, Me], [RA1874; H, H, Me, H, CF ₂ H, Et], [RA1875; H, H, Me , H, CF ₂ H, Pr], [RA1876; H, H, Me, H, CF ₂ H, i-Pr], [RA1877; H, H, Me, H, CF ₂ H, c-Pr], [RA1878; H, H, Me, H, CF ₂ H, Bu], [RA1879; H, H, Me, H, CF ₂ H, i-Bu], [RA1880; H, H, Me, H, CF ₂ H, t-Bu], [RA1881; H, H, Me, H, CF ₂ H, c-PrCH ₂ ], [RA1882; H, H, Me, H, CF ₂ H, Ph], [RA1883; H, H, Me, H, CF ₂ H, Bn], [RA1884; H, H, Me, H, CF ₂ H, CF ₃ ], [RA1885; H, H, Me, H, CF ₂ H, CF ₃ CH ₂ ], [RA1886; H, H, Me, H, CF ₂ H, CF ₃ CF ₂ ], [RA1887; H, H, Me, H, CF ₂ H, CF ₂ H], [RA1888; H , H, Me, H, CF ₂ H, CF ₂ HCH ₂ ], [RA1889; H, H, Me, Me, CF ₂ H, Me], [RA1890; H, H, Me, Me, CF ₂ H, Et], [RA1891; H, H, Me, Me, CF ₂ H, Pr], [RA1892; H, H, Me, Me, CF ₂ H, i-Pr], [RA1893; H, H, Me, Me, CF ₂ H, c-Pr], [RA1894; H, H, Me, Me, CF ₂ H, Bu], [RA1895; H, H, Me, Me, CF ₂ H, i-Bu], [ RA1896; H, H, Me, Me, CF ₂ H, t-Bu], [RA1897; H, H, Me, Me, CF ₂ H, c-PrCH ₂ ], [RA1898; H, H, Me, Me , CF ₂ H, Ph], [RA1899; H, H, Me, Me, CF ₂ H, Bn], [RA1900; H, H, Me, Me, CF ₂ H, CF ₃ ], [RA1901; H, H, Me, Me, CF ₂ H, CF ₃ CH ₂ ], [RA1902; H, H , Me, Me, CF ₂ H, CF ₃ CF ₂ ], [RA1903; H, H, Me, Me, CF ₂ H, CF ₂ H], [RA1904; H, H, Me, Me, CF ₂ H, CF ₂ HCH ₂ ], [RA1905; H, H, Me, Et, CF ₂ H, Me], [RA1906; H, H, Me, Et, CF ₂ H, Et], [RA1907; H, H, Me , Et, CF ₂ H, Pr], [RA1908; H, H, Me, Et, CF ₂ H, i-Pr], [RA1909; H, H, Me, Et, CF ₂ H, c-Pr], [RA1910; H, H, Me, Et, CF ₂ H, Bu], [RA1911; H, H, Me, Et, CF ₂ H, i-Bu], [RA1912; H, H, Me, Et, CF ₂ H, t-Bu], [RA1913; H, H, Me, Et, CF ₂ H, c-PrCH ₂ ], [RA1914; H, H, Me, Et, CF ₂ H, Ph], [RA1915; H, H, Me, Et, CF ₂ H, Bn], [RA1916; H, H, Me, Et, CF ₂ H, CF ₃ ], [RA1917; H, H, Me, Et, CF ₂ H, CF ₃ CH ₂ ], [RA1918; H, H, Me, Et, CF ₂ H, CF ₃ CF ₂ ], [RA1919; H, H, Me, Et, CF ₂ H, CF ₂ H], [RA1920; H , H, Me, Et, CF ₂ H, CF ₂ HCH ₂ ], [RA1921; H, H, Me, F, CF ₂ H, Me], [RA1922; H, H, Me, F, CF ₂ H, Et], [RA1923; H, H, Me, F, CF ₂ H, Pr], [RA1924; H, H, Me, F, CF ₂ H, i-Pr], [RA1925; H, H, Me, F, CF ₂ H, c-Pr], [RA1926; H, H, Me, F, CF ₂ H, Bu], [RA1927; H, H, Me, F, CF ₂ H, i-Bu], [ RA1928; H, H, Me, F, CF ₂ H, t-Bu], [RA1929; H, H, Me, F, CF ₂ H, c-PrCH ₂ ], [RA1930; H, H, Me, F , CF ₂ H, Ph], [RA1931; H, H, Me, F, CF ₂ H, Bn], [RA1932; H, H, Me, F, CF ₂ H, CF ₃ ], [RA1933; H, H, Me, F, CF ₂ H, CF ₃ CH ₂ ], [R A1934; H, H, Me, F, CF ₂ H, CF ₃ CF ₂ ], [RA1935; H, H, Me, F, CF ₂ H, CF ₂ H], [RA1936; H, H, Me, F , CF ₂ H, CF ₂ HCH ₂ ], [RA1937; H, H, Me, Cl, CF ₂ H, Me], [RA1938; H, H, Me, Cl, CF ₂ H, Et], [RA1939; H, H, Me, Cl, CF ₂ H, Pr], [RA1940; H, H, Me, Cl, CF ₂ H, i-Pr], [RA1941; H, H, Me, Cl, CF ₂ H, c-Pr], [RA1942; H, H, Me, Cl, CF ₂ H, Bu], [RA1943; H, H, Me, Cl, CF ₂ H, i-Bu], [RA1944; H, H, Me, Cl, CF ₂ H, t-Bu], [RA1945; H, H, Me, Cl, CF ₂ H, c-PrCH ₂ ], [RA1946; H, H, Me, Cl, CF ₂ H, Ph ], [RA1947; H, H, Me, Cl, CF ₂ H, Bn], [RA1948; H, H, Me, Cl, CF ₂ H, CF ₃ ], [RA1949; H, H, Me, Cl, CF ₂ H, CF ₃ CH ₂ ], [RA1950; H, H, Me, Cl, CF ₂ H, CF ₃ CF ₂ ], [RA1951; H, H, Me, Cl, CF ₂ H, CF ₂ H] , [RA1952; H, H, Me, Cl, CF ₂ H, CF ₂ HCH ₂ ], [RA1953; H, H, Et, H, CF ₂ H, Me], [RA1954; H, H, Et, H , CF ₂ H, Et], [RA1955; H, H, Et, H, CF ₂ H, Pr], [RA1956; H, H, Et, H, CF ₂ H, i-Pr], [RA1957; H , H, Et, H, CF ₂ H, c-Pr], [RA1958; H, H, Et, H, CF ₂ H, Bu], [RA1959; H, H, Et, H, CF ₂ H, i -Bu], [RA1960; H, H, Et, H, CF ₂ H, t-Bu], [RA1961; H, H, Et, H, CF ₂ H, c-PrCH ₂ ], [RA1962; H, H, Et, H, CF ₂ H, Ph], [RA1963; H, H, Et, H, CF ₂ H, Bn], [RA1964; H, H, Et, H, CF ₂ H, CF ₃ ], [RA1965; H, H, Et, H, CF ₂ H, CF ₃ CH ₂ ], [RA1966; H, H, Et, H, CF ₂ H, CF ₃ CF ₂ ], [RA1967; H, H, Et, H, CF ₂ H, CF ₂ H], [RA1968; H, H , Et, H, CF ₂ H, CF ₂ HCH ₂ ], [RA1969; H, H, Et, F, CF ₂ H, Me], [RA1970; H, H, Et, F, CF ₂ H, Et] , [RA1971; H, H, Et, F, CF ₂ H, Pr], [RA1972; H, H, Et, F, CF ₂ H, i-Pr], [RA1973; H, H, Et, F, CF ₂ H, c-Pr], [RA1974; H, H, Et, F, CF ₂ H, Bu], [RA1975; H, H, Et, F, CF ₂ H, i-Bu], [RA1976; H, H, Et, F, CF ₂ H, t-Bu], [RA1977; H, H, Et, F, CF ₂ H, c-PrCH ₂ ], [RA1978; H, H, Et, F, CF ₂ H, Ph], [RA1979; H, H, Et, F, CF ₂ H, Bn], [RA1980; H, H, Et, F, CF ₂ H, CF ₃ ], [RA1981; H, H, Et, F, CF ₂ H, CF ₃ CH ₂ ], [RA1982; H, H, Et, F, CF ₂ H, CF ₃ CF ₂ ], [RA1983; H, H, Et, F, CF ₂ H, CF ₂ H], [RA1984; H, H, Et, F, CF ₂ H, CF ₂ HCH ₂ ], [RA1985; H, H, Et, Cl, CF ₂ H, Me], [RA1986; H, H , Et, Cl, CF ₂ H, Et], [RA1987; H, H, Et, Cl, CF ₂ H, Pr], [RA1988; H, H, Et, Cl, CF ₂ H, i-Pr], [RA1989; H, H, Et, Cl, CF ₂ H, c-Pr], [RA1990; H, H, Et, Cl, CF ₂ H, Bu], [RA1991; H, H, Et, Cl, CF ₂ H, i-Bu], [RA1992; H, H, Et, Cl, CF ₂ H, t-Bu], [RA1993; H, H, Et, Cl, CF ₂ H, c-PrCH ₂ ], [ RA1994; H, H, Et, Cl, CF 2 H, Ph], [RA1995; H, H, Et, Cl, CF 2 H, Bn], [RA1996; H, H, Et, Cl, CF 2 H, CF ₃ ], [RA1997; H, H, Et, Cl, CF ₂ H, CF ₃ CH ₂ ], [RA1998; H, H, Et, Cl, CF ₂ H, CF ₃ CF ₂ ], [RA1999; H, H, Et, Cl, CF ₂ H, CF ₂ H], [RA2000; H, H, Et, Cl, CF ₂ H, CF ₂ HCH ₂ ],

[RA2001; H, H, F, H, CF ₂ H, Me], [RA2002; H, H, F, H, CF ₂ H, Et], [RA2003; H, H, F, H, CF ₂ H , Pr], [RA2004; H, H, F, H, CF ₂ H, i-Pr], [RA2005; H, H, F, H, CF ₂ H, c-Pr], [RA2006; H, H , F, H, CF ₂ H, Bu], [RA2007; H, H, F, H, CF ₂ H, i-Bu], [RA2008; H, H, F, H, CF ₂ H, t-Bu ], [RA2009; H, H, F, H, CF ₂ H, c-PrCH ₂ ], [RA2010; H, H, F, H, CF ₂ H, Ph], [RA2011; H, H, F, H, CF ₂ H, Bn], [RA2012; H, H, F, H, CF ₂ H, CF ₃ ], [RA2013; H, H, F, H, CF ₂ H, CF ₃ CH ₂ ], [ RA2014; H, H, F, H, CF ₂ H, CF ₃ CF ₂ ], [RA2015; H, H, F, H, CF ₂ H, CF ₂ H], [RA2016; H, H, F, H , CF ₂ H, CF ₂ HCH ₂ ], [RA2017; H, H, F, F, CF ₂ H, Me], [RA2018; H, H, F, F, CF ₂ H, Et], [RA2019; H, H, F, F, CF ₂ H, Pr], [RA2020; H, H, F, F, CF ₂ H, i-Pr], [RA2021; H, H, F, F, CF ₂ H, c-Pr], [RA2022; H, H, F, F, CF ₂ H, Bu], [RA2023; H, H, F, F, CF ₂ H, i-Bu], [RA2024; H, H, F, F, CF ₂ H, t-Bu], [RA2025; H, H, F, F, CF ₂ H, c-PrCH ₂ ], [RA2026; H, H, F, F, CF ₂ H, Ph ], [RA2027; H, H, F, F, CF ₂ H, Bn], [RA2028; H, H, F, F, CF ₂ H, CF ₃ ], [RA2029; H, H, F, F, CF ₂ H, CF ₃ CH ₂ ], [RA2030; H, H, F, F, CF ₂ H, CF ₃ CF ₂ ], [RA2031; H, H, F, F, CF ₂ H, CF ₂ H] , [RA2032; H, H, F, F, CF ₂ H, CF ₂ HCH ₂ ], [RA2033; H, H, F, Cl, CF ₂ H, Me], [RA2034; H, H, F, Cl, CF ₂ H, Et], [RA2035; H, H, F, Cl, CF ₂ H, Pr], [RA2036; H, H, F, Cl, CF ₂ H, i-Pr], [RA2037; H, H, F, Cl, CF ₂ H, c-Pr], [RA2038; H, H, F, Cl, CF ₂ H, Bu], [RA2039; H, H, F, Cl, CF ₂ H, i-Bu], [RA2040; H, H, F, Cl, CF ₂ H, t-Bu], [RA2041; H, H, F, Cl, CF ₂ H, c-PrCH ₂ ], [RA2042; H , H, F, Cl, CF ₂ H, Ph], [RA2043; H, H, F, Cl, CF ₂ H, Bn], [RA2044; H, H, F, Cl, CF ₂ H, CF ₃ ] , [RA2045; H, H, F, Cl, CF ₂ H, CF ₃ CH ₂ ], [RA2046; H, H, F, Cl, CF ₂ H, CF ₃ CF ₂ ], [RA2047; H, H, F, Cl, CF ₂ H, CF ₂ H], [RA2048; H, H, F, Cl, CF ₂ H, CF ₂ HCH ₂ ], [RA2049; H, H, Cl, H, CF ₂ H, Me ], [RA2050; H, H, Cl, H, CF ₂ H, Et], [RA2051; H, H, Cl, H, CF ₂ H, Pr], [RA2052; H, H, Cl, H, CF ₂ H, i-Pr], [RA2053; H, H, Cl, H, CF ₂ H, c-Pr], [RA2054; H, H, Cl, H, CF ₂ H, Bu], [RA2055; H , H, Cl, H, CF ₂ H, i-Bu], [RA2056; H, H, Cl, H, CF ₂ H, t-Bu], [RA2057; H, H, Cl, H, CF ₂ H , c-PrCH ₂ ], [RA2058; H, H, Cl, H, CF ₂ H, Ph], [RA2059; H, H, Cl, H, CF ₂ H, Bn], [RA2060; H, H, Cl, H, CF ₂ H, CF ₃ ], [RA2061; H, H, Cl, H, CF ₂ H, CF ₃ CH ₂ ], [RA2062; H, H, Cl, H, CF ₂ H, CF ₃ CF ₂ ], [RA2063; H, H, Cl, H, CF ₂ H, CF ₂ H], [RA2064; H, H, Cl, H, CF ₂ H, CF ₂ HCH ₂ ], [RA2065; H, H, Cl, Cl, CF ₂ H, Me], [RA2066; H, H, Cl, Cl, CF ₂ H, Et], [RA2067; H, H, Cl, Cl, CF 2 H, Pr], [RA2068; H, H, Cl, Cl, CF 2 H, i-Pr], [RA2069; H, H, Cl, Cl, CF ₂ H, c-Pr], [RA2070; H, H, Cl, Cl, CF ₂ H, Bu], [RA2071; H, H, Cl, Cl, CF ₂ H, i-Bu] , [RA2072; H, H, Cl, Cl, CF ₂ H, t-Bu], [RA2073; H, H, Cl, Cl, CF ₂ H, c-PrCH ₂ ], [RA2074; H, H, Cl , Cl, CF ₂ H, Ph], [RA2075; H, H, Cl, Cl, CF ₂ H, Bn], [RA2076; H, H, Cl, Cl, CF ₂ H, CF ₃ ], [RA2077; H, H, Cl, Cl, CF ₂ H, CF ₃ CH ₂ ], [RA2078; H, H, Cl, Cl, CF ₂ H, CF ₃ CF ₂ ], [RA2079; H, H, Cl, Cl, CF ₂ H, CF ₂ H], [RA2080; H, H, Cl, Cl, CF ₂ H, CF ₂ HCH ₂ ], [RA2081; H, H, Me, H, CF ₃ , Me], [RA2082; H, H, Me, H, CF ₃ , Et], [RA2083; H, H, Me, H, CF ₃ , Pr], [RA2084; H, H, Me, H, CF ₃ , i-Pr], [RA2085; H, H, Me, H, CF ₃ , c-Pr], [RA2086; H, H, Me, H, CF ₃ , Bu], [RA2087; H, H, Me, H, CF ₃ , i-Bu], [RA2088; H, H, Me, H, CF ₃ , t-Bu], [RA2089; H, H, Me, H, CF ₃ , c-PrCH ₂ ], [RA2090; H, H , Me, H, CF ₃ , Ph], [RA2091; H, H, Me, H, CF ₃ , Bn], [RA2092; H, H, Me, H, CF ₃ , CF ₃ ], [RA2093; H , H, Me, H, CF ₃ , CF ₃ CH ₂ ], [RA2094; H, H, Me, H, CF ₃ , CF ₃ CF ₂ ], [RA2095; H, H, Me, H, CF ₃ , CF ₂ H], [RA2096; H, H, Me, H, CF ₃ , CF ₂ HCH ₂ ], [RA2097; H, H, Me, Me, CF ₃ , Me], [RA2098; H, H, Me , Me, CF ₃ , Et], [RA209 9; H, H, Me, Me, CF ₃ , Pr], [RA2100; H, H, Me, Me, CF ₃ , i-Pr], [RA2101; H, H, Me, Me, CF ₃ , c -Pr], [RA2102; H, H, Me, Me, CF ₃ , Bu], [RA2103; H, H, Me, Me, CF ₃ , i-Bu], [RA2104; H, H, Me, Me , CF ₃ , t-Bu], [RA2105; H, H, Me, Me, CF ₃ , c-PrCH ₂ ], [RA2106; H, H, Me, Me, CF ₃ , Ph], [RA2107; H , H, Me, Me, CF ₃ , Bn], [RA2108; H, H, Me, Me, CF ₃ , CF ₃ ], [RA2109; H, H, Me, Me, CF ₃ , CF ₃ CH ₂ ] , [RA2110; H, H, Me, Me, CF ₃ , CF ₃ CF ₂ ], [RA2111; H, H, Me, Me, CF ₃ , CF ₂ H], [RA2112; H, H, Me, Me , CF ₃ , CF ₂ HCH ₂ ], [RA2113; H, H, Me, Et, CF ₃ , Me], [RA2114; H, H, Me, Et, CF ₃ , Et], [RA2115; H, H , Me, Et, CF ₃ , Pr], [RA2116; H, H, Me, Et, CF ₃ , i-Pr], [RA2117; H, H, Me, Et, CF ₃ , c-Pr], [ RA2118; H, H, Me, Et, CF ₃ , Bu], [RA2119; H, H, Me, Et, CF ₃ , i-Bu], [RA2120; H, H, Me, Et, CF ₃ , t -Bu], [RA2121; H, H, Me, Et, CF ₃ , c-PrCH ₂ ], [RA2122; H, H, Me, Et, CF ₃ , Ph], [RA2123; H, H, Me, Et, CF ₃ , Bn], [RA2124; H, H, Me, Et, CF ₃ , CF ₃ ], [RA2125; H, H, Me, Et, CF ₃ , CF ₃ CH ₂ ], [RA2126; H , H, Me, Et, CF ₃ , CF ₃ CF ₂ ], [RA2127; H, H, Me, Et, CF ₃ , CF ₂ H], [RA2128; H, H, Me, Et, CF ₃ , CF ₂ HCH ₂ ], [RA2129; H, H, Me, F, CF ₃ , Me], [RA2130; H, H, Me, F, CF ₃ , Et], [RA2131; H, H, Me, F, C F ₃ , Pr], [RA2132; H, H, Me, F, CF ₃ , i-Pr], [RA2133; H, H, Me, F, CF ₃ , c-Pr], [RA2134; H, H , Me, F, CF ₃ , Bu], [RA2135; H, H, Me, F, CF ₃ , i-Bu], [RA2136; H, H, Me, F, CF ₃ , t-Bu], [ RA2137; H, H, Me, F, CF ₃ , c-PrCH ₂ ], [RA2138; H, H, Me, F, CF ₃ , Ph], [RA2139; H, H, Me, F, CF ₃ , Bn], [RA2140; H, H, Me, F, CF ₃ , CF ₃ ], [RA2141; H, H, Me, F, CF ₃ , CF ₃ CH ₂ ], [RA2142; H, H, Me, F, CF ₃ , CF ₃ CF ₂ ], [RA2143; H, H, Me, F, CF ₃ , CF ₂ H], [RA2144; H, H, Me, F, CF ₃ , CF ₂ HCH ₂ ], [RA2145; H, H, Me, Cl, CF ₃ , Me], [RA2146; H, H, Me, Cl, CF ₃ , Et], [RA2147; H, H, Me, Cl, CF ₃ , Pr] , [RA2148; H, H, Me, Cl, CF ₃ , i-Pr], [RA2149; H, H, Me, Cl, CF ₃ , c-Pr], [RA2150; H, H, Me, Cl, CF ₃ , Bu], [RA2151; H, H, Me, Cl, CF ₃ , i-Bu], [RA2152; H, H, Me, Cl, CF ₃ , t-Bu], [RA2153; H, H , Me, Cl, CF ₃ , c-PrCH ₂ ], [RA2154; H, H, Me, Cl, CF ₃ , Ph], [RA2155; H, H, Me, Cl, CF ₃ , Bn], [RA2156 ; H, H, Me, Cl, CF ₃ , CF ₃ ], [RA2157; H, H, Me, Cl, CF ₃ , CF ₃ CH ₂ ], [RA2158; H, H, Me, Cl, CF ₃ , CF ₃ CF ₂ ], [RA2159; H, H, Me, Cl, CF ₃ , CF ₂ H], [RA2160; H, H, Me, Cl, CF ₃ , CF ₂ HCH ₂ ], [RA2161; H, H, Et, H, CF ₃ , Me], [RA2162; H, H, Et, H, CF ₃ , Et], [RA2163; H, H, Et, H, CF ₃ , Pr], [RA2164; H , H, Et, H, CF ₃ , i-Pr], [RA2165; H, H, Et, H, CF ₃ , c-Pr], [RA2166; H, H, Et, H, CF ₃ , Bu], [RA2167; H, H , Et, H, CF ₃ , i-Bu], [RA2168; H, H, Et, H, CF ₃ , t-Bu], [RA2169; H, H, Et, H, CF ₃ , c-PrCH ₂ ], [RA2170; H, H, Et, H, CF ₃ , Ph], [RA2171; H, H, Et, H, CF ₃ , Bn], [RA2172; H, H, Et, H, CF ₃ , CF ₃ ], [RA2173; H, H, Et, H, CF ₃ , CF ₃ CH ₂ ], [RA2174; H, H, Et, H, CF ₃ , CF ₃ CF ₂ ], [RA2175; H, H , Et, H, CF ₃ , CF ₂ H], [RA2176; H, H, Et, H, CF ₃ , CF ₂ HCH ₂ ], [RA2177; H, H, Et, F, CF ₃ , Me], [RA2178; H, H, Et, F, CF ₃ , Et], [RA2179; H, H, Et, F, CF ₃ , Pr], [RA2180; H, H, Et, F, CF ₃ , i- Pr], [RA2181; H, H, Et, F, CF ₃ , c-Pr], [RA2182; H, H, Et, F, CF ₃ , Bu], [RA2183; H, H, Et, F, CF ₃ , i-Bu], [RA2184; H, H, Et, F, CF ₃ , t-Bu], [RA2185; H, H, Et, F, CF ₃ , c-PrCH ₂ ], [RA2186; H, H, Et, F, CF ₃ , Ph], [RA2187; H, H, Et, F, CF ₃ , Bn], [RA2188; H, H, Et, F, CF ₃ , CF ₃ ], [ RA2189; H, H, Et, F, CF ₃ , CF ₃ CH ₂ ], [RA2190; H, H, Et, F, CF ₃ , CF ₃ CF ₂ ], [RA2191; H, H, Et, F, CF ₃ , CF ₂ H], [RA2192; H, H, Et, F, CF ₃ , CF ₂ HCH ₂ ], [RA2193; H, H, Et, Cl, CF ₃ , Me], [RA2194; H, H, Et, Cl, CF ₃ , Et], [RA2195; H, H, Et, Cl, CF ₃ , Pr], [RA2196; H, H, Et, Cl, CF ₃ , i-Pr], [RA2197 ; H, H, Et, Cl, CF ₃ , c- Pr], [RA2198; H, H, Et, Cl, CF ₃ , Bu], [RA2199; H, H, Et, Cl, CF ₃ , i-Bu], [RA2200; H, H, Et, Cl, CF ₃ , t-Bu],

[RA2201; H, H, Et, Cl, CF ₃ , c-PrCH ₂ ], [RA2202; H, H, Et, Cl, CF ₃ , Ph], [RA2203; H, H, Et, Cl, CF ₃ , Bn], [RA2204; H, H, Et, Cl, CF ₃ , CF ₃ ], [RA2205; H, H, Et, Cl, CF ₃ , CF ₃ CH ₂ ], [RA2206; H, H, Et , Cl, CF ₃ , CF ₃ CF ₂ ], [RA2207; H, H, Et, Cl, CF ₃ , CF ₂ H], [RA2208; H, H, Et, Cl, CF ₃ , CF ₂ HCH ₂ ] , [RA2209; H, H, F, H, CF ₃ , Me], [RA2210; H, H, F, H, CF ₃ , Et], [RA2211; H, H, F, H, CF ₃ , Pr ], [RA2212; H, H, F, H, CF ₃ , i-Pr], [RA2213; H, H, F, H, CF ₃ , c-Pr], [RA2214; H, H, F, H , CF ₃ , Bu], [RA2215; H, H, F, H, CF ₃ , i-Bu], [RA2216; H, H, F, H, CF ₃ , t-Bu], [RA2217; H, H, F, H, CF ₃ , c-PrCH ₂ ], [RA2218; H, H, F, H, CF ₃ , Ph], [RA2219; H, H, F, H, CF ₃ , Bn], [ RA2220; H, H, F, H, CF ₃ , CF ₃ ], [RA2221; H, H, F, H, CF ₃ , CF ₃ CH ₂ ], [RA2222; H, H, F, H, CF ₃ , CF ₃ CF ₂ ], [RA2223; H, H, F, H, CF ₃ , CF ₂ H], [RA2224; H, H, F, H, CF ₃ , CF ₂ HCH ₂ ], [RA2225; H , H, F, F, CF ₃ , Me], [RA2226; H, H, F, F, CF ₃ , Et], [RA2227; H, H, F, F, CF ₃ , Pr], [RA2228; H, H, F, F, CF ₃ , i-Pr], [RA2229; H, H, F, F, CF ₃ , c-Pr], [RA2230; H, H, F, F, CF ₃ , Bu ], [RA2231; H, H, F, F, CF ₃ , i-Bu], [RA2232; H, H, F, F, CF ₃ , t-Bu], [RA2233; H, H, F, F , CF ₃ , c-PrCH ₂ ], [RA2234; H, H, F, F, CF ₃ , Ph] , [RA2235; H, H, F, F, CF ₃ , Bn], [RA2236; H, H, F, F, CF ₃ , CF ₃ ], [RA2237; H, H, F, F, CF ₃ , CF ₃ CH ₂ ], [RA2238; H, H, F, F, CF ₃ , CF ₃ CF ₂ ], [RA2239; H, H, F, F, CF ₃ , CF ₂ H], [RA2240; H, H, F, F, CF ₃ , CF ₂ HCH ₂ ], [RA2241; H, H, F, Cl, CF ₃ , Me], [RA2242; H, H, F, Cl, CF ₃ , Et], [ RA2243; H, H, F, Cl, CF ₃ , Pr], [RA2244; H, H, F, Cl, CF ₃ , i-Pr], [RA2245; H, H, F, Cl, CF ₃ , c -Pr], [RA2246; H, H, F, Cl, CF ₃ , Bu], [RA2247; H, H, F, Cl, CF ₃ , i-Bu], [RA2248; H, H, F, Cl , CF ₃ , t-Bu], [RA2249; H, H, F, Cl, CF ₃ , c-PrCH ₂ ], [RA2250; H, H, F, Cl, CF ₃ , Ph], [RA2251; H , H, F, Cl, CF ₃ , Bn], [RA2252; H, H, F, Cl, CF ₃ , CF ₃ ], [RA2253; H, H, F, Cl, CF ₃ , CF ₃ CH ₂ ] , [RA2254; H, H, F, Cl, CF ₃ , CF ₃ CF ₂ ], [RA2255; H, H, F, Cl, CF ₃ , CF ₂ H], [RA2256; H, H, F, Cl , CF ₃ , CF ₂ HCH ₂ ], [RA2257; H, H, Cl, H, CF ₃ , Me], [RA2258; H, H, Cl, H, CF ₃ , Et], [RA2259; H, H , Cl, H, CF ₃ , Pr], [RA2260; H, H, Cl, H, CF ₃ , i-Pr], [RA2261; H, H, Cl, H, CF ₃ , c-Pr], [ RA2262; H, H, Cl, H, CF ₃ , Bu], [RA2263; H, H, Cl, H, CF ₃ , i-Bu], [RA2264; H, H, Cl, H, CF ₃ , t -Bu], [RA2265; H, H, Cl, H, CF ₃ , c-PrCH ₂ ], [RA2266; H, H, Cl, H, CF ₃ , Ph], [RA2267; H, H, Cl, H, CF ₃ , Bn], [RA2268; H, H, Cl, H, CF ₃ , CF ₃ ], [RA2269; H, H, Cl, H, CF ₃ , CF ₃ CH ₂ ], [RA2270; H, H, Cl, H, CF ₃ , CF ₃ CF ₂ ], [RA2271; H , H, Cl, H, CF ₃ , CF ₂ H], [RA2272; H, H, Cl, H, CF ₃ , CF ₂ HCH ₂ ], [RA2273; H, H, Cl, Cl, CF ₃ , Me ], [RA2274; H, H, Cl, Cl, CF ₃ , Et], [RA2275; H, H, Cl, Cl, CF ₃ , Pr], [RA2276; H, H, Cl, Cl, CF ₃ , i-Pr], [RA2277; H, H, Cl, Cl, CF ₃ , c-Pr], [RA2278; H, H, Cl, Cl, CF ₃ , Bu], [RA2279; H, H, Cl, Cl, CF ₃ , i-Bu], [RA2280; H, H, Cl, Cl, CF ₃ , t-Bu], [RA2281; H, H, Cl, Cl, CF ₃ , c-PrCH ₂ ], [ RA2282; H, H, Cl, Cl, CF 3, Ph], [RA2283; H, H, Cl, Cl, CF 3, Bn], [RA2284; H, H, Cl, Cl, CF 3, CF 3] , [RA2285; H, H, Cl, Cl, CF ₃ , CF ₃ CH ₂ ], [RA2286; H, H, Cl, Cl, CF ₃ , CF ₃ CF ₂ ], [RA2287; H, H, Cl, Cl, CF ₃ , CF ₂ H], [RA2288; H, H, Cl, Cl, CF ₃ , CF ₂ HCH ₂ ], [RA2289; H, H, Me, H, CF ₂ HCH ₂ , Me], [ RA2290; H, H, Me, H, CF ₂ HCH ₂ , Et], [RA2291; H, H, Me, H, CF ₂ HCH ₂ , Pr], [RA2292; H, H, Me, H, CF _{2 HCH 2, i-Pr],} [RA2293; H, H, Me, H, CF 2 HCH 2, c-Pr], [RA2294; H, H, Me, H, CF 2 HCH 2, Bu], [RA2295 ; H, H, Me, H, CF ₂ HCH ₂ , i-Bu], [RA2296; H, H, Me, H, CF ₂ HCH ₂ , t-Bu], [RA2297; H, H, Me, H , CF ₂ HCH ₂ , c-PrCH ₂ ], [RA2298; H, H, Me, H, CF ₂ HCH ₂ , Ph], [RA2299; H, H, M e, H, CF ₂ HCH ₂ , Bn], [RA2300; H, H, Me, H, CF ₂ HCH ₂ , CF ₃ ], [RA2301; H, H, Me, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA2302; H, H, Me, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA2303; H, H, Me, H, CF ₂ HCH ₂ , CF ₂ H], [RA2304; H, H, Me, H, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA2305; H, H, Me, Me, CF ₂ HCH ₂ , Me], [RA2306; H, H, Me, Me, CF ₂ HCH ₂ , Et], [RA2307; H, H, Me, Me, CF ₂ HCH ₂ , Pr], [RA2308; H, H, Me, Me, CF ₂ HCH ₂ , i-Pr], [RA2309; H, H, Me, Me, CF ₂ HCH ₂ , c-Pr], [RA2310; H, H, Me, Me, CF ₂ HCH ₂ , Bu], [RA2311; H, H, Me, Me, CF ₂ HCH ₂ , i-Bu], [RA2312; H, H, Me, Me, CF ₂ HCH ₂ , t-Bu], [RA2313; H, H, Me, Me, CF ₂ HCH ₂ , c-PrCH ₂ ] , [RA2314; H, H, Me, Me, CF ₂ HCH ₂ , Ph], [RA2315; H, H, Me, Me, CF ₂ HCH ₂ , Bn], [RA2316; H, H, Me, Me, CF ₂ HCH ₂ , CF ₃ ], [RA2317; H, H, Me, Me, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA2318; H, H, Me, Me, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA2319; H, H, Me, Me, CF ₂ HCH ₂ , CF ₂ H], [RA2320; H, H, Me, Me, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA2321; H , H, Me, Et, CF ₂ HCH ₂ , Me], [RA2322; H, H, Me, Et, CF ₂ HCH ₂ , Et], [RA2323; H, H, Me, Et, CF ₂ HCH ₂ , Pr], [RA2324; H, H, Me, Et, CF ₂ HCH ₂ , i-Pr], [RA2325; H, H, Me, Et, CF ₂ HCH ₂ , c-Pr], [RA2326; H, H, Me, Et, CF ₂ HCH ₂ , Bu], [RA2327; H, H, Me, Et, CF ₂ HCH ₂ , i-Bu], [RA2328; H, H, Me, Et, CF ₂ HCH ₂ , t-Bu], [RA2329; H, H, Me, Et, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA2330; H, H, Me, Et, CF ₂ HCH ₂ , Ph], [RA2331; H, H, Me, Et, CF ₂ HCH ₂ , Bn], [RA2332; H, H, Me, Et, CF ₂ HCH ₂ , CF ₃ ], [RA2333; H, H, Me, Et, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA2334; H, H, Me, Et, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA2335; H, H, Me, Et, CF ₂ HCH ₂ , CF ₂ H], [RA2336; H, H, Me, Et, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA2337; H, H, Me, F, CF ₂ HCH ₂ , Me], [RA2338; H, H, Me, F, CF ₂ HCH ₂ , Et], [RA2339; H, H, Me, F, CF ₂ HCH ₂ , Pr], [RA 2340; H, H, Me, F, CF ₂ HCH ₂ , i-Pr], [RA2341; H, H, Me, F, CF ₂ HCH ₂ , c-Pr], [RA2342; H, H, Me, F, CF ₂ HCH ₂ , Bu], [RA2343; H, H, Me, F, CF ₂ HCH ₂ , i-Bu], [RA2344; H, H, Me, F, CF ₂ HCH ₂ , t-Bu], [RA2345; H, H, Me, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [ RA2346; H, H, Me, F, CF ₂ HCH ₂ , Ph], [RA2347; H, H, Me, F, CF ₂ HCH ₂ , Bn], [RA2348; H, H, Me, F, CF ₂ HCH ₂ , CF ₃ ], [RA2349; H, H, Me, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA2350; H, H, Me, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ] , [RA2351; H, H, Me, F, CF ₂ HCH ₂ , CF ₂ H], [RA2352; H, H, Me, F, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA2353; H, H , Me, Cl, CF ₂ HCH _{2, Me], [RA2354;} H, H, Me, Cl, CF 2 HCH 2, Et], [RA2355; H, H, Me, Cl, CF 2 HCH 2, Pr], [RA2356; H, H, Me, Cl, CF ₂ HCH ₂ , i-Pr], [RA2357; H, H, Me, Cl, CF ₂ HCH ₂ , c-Pr], [RA2358; H, H, Me, Cl, CF ₂ HCH ₂ , Bu], [RA2359; H, H, Me, Cl, CF ₂ HCH ₂ , i-Bu], [RA2360; H, H, Me, Cl, CF ₂ HCH ₂ , t-Bu], [RA2361; H , H, Me, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA2362; H, H, Me, Cl, CF ₂ HCH ₂ , Ph], [RA2363; H, H, Me, Cl, CF ₂ HCH ₂ , Bn], [RA2364; H, H, Me, Cl, CF ₂ HCH ₂ , CF ₃ ], [RA2365; H, H, Me, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA2366 ; H, H, Me, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA2367; H, H, Me, Cl, CF ₂ HCH ₂ , CF ₂ H], [RA2368; H, H, Me, Cl, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA2369; H, H, Et, H, CF ₂ HCH ₂ , Me], [RA2370; H, H, Et, H, CF ₂ HCH ₂ , Et] , [RA2371; H, H, Et, H, CF ₂ HCH ₂ , Pr], [RA2372; H, H, Et, H, CF ₂ HCH ₂ , i-Pr], [RA2373; H, H, Et, H, CF ₂ HCH ₂ , c-Pr], [RA2374; H, H, Et, H, CF ₂ HCH ₂ , Bu], [RA2375; H, H, Et, H, CF ₂ HCH ₂ , i-Bu ], [RA2376; H, H, Et, H, CF ₂ HCH ₂ , t-Bu], [RA2377; H, H, Et, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA2378; H, H, Et, H, CF ₂ HCH ₂ , Ph], [RA2379; H, H, Et, H, CF ₂ HCH ₂ , Bn], [RA2380; H, H, Et, H, CF ₂ HCH ₂ , CF ₃ ], [RA2381; H, H, Et, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA2382; H, H, Et, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA2383; H, H, Et, H, CF ₂ HCH ₂ , CF ₂ H ], [RA2384; H, H, Et, H, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA2385; H, H, Et, F, CF ₂ HCH ₂ , Me], [RA2386; H, H, Et, F, CF ₂ HCH ₂ , Et], [RA2387; H, H, Et, F, CF ₂ HCH ₂ , Pr], [RA2388; H, H, Et, F, CF ₂ HCH ₂ , i-Pr ], [RA2389; H, H, Et, F, CF ₂ HCH ₂ , c-Pr], [RA2390; H, H, Et, F, CF ₂ HCH ₂ , Bu], [RA2391; H, H, Et , F, CF ₂ HCH ₂ , i-Bu], [RA2392; H, H, Et, F, CF ₂ HCH ₂ , t-Bu], [RA2393; H, H, Et, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA2394; H, H, Et, F, CF ₂ HCH ₂ , Ph], [RA2395; H, H, Et, F, CF ₂ HCH ₂ , Bn], [RA2396; H, H , Et, F, CF
₂ HCH ₂ , CF ₃ ], [RA2397; H, H, Et, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA2398; H, H, Et, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA2399; H, H, Et, F, CF ₂ HCH ₂ , CF ₂ H], [RA2400; H, H, Et, F, CF ₂ HCH ₂ , CF ₂ HCH ₂ ],

[RA2401; H, H, Et, Cl, CF ₂ HCH ₂ , Me], [RA2402; H, H, Et, Cl, CF ₂ HCH ₂ , Et], [RA2403; H, H, Et, Cl, CF ₂ HCH ₂ , Pr], [RA2404; H, H, Et, Cl, CF ₂ HCH ₂ , i-Pr], [RA2405; H, H, Et, Cl, CF ₂ HCH ₂ , c-Pr], [ RA2406; H, H, Et, Cl, CF ₂ HCH ₂ , Bu], [RA2407; H, H, Et, Cl, CF ₂ HCH ₂ , i-Bu], [RA2408; H, H, Et, Cl, CF ₂ HCH ₂ , t-Bu], [RA2409; H, H, Et, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA2410; H, H, Et, Cl, CF ₂ HCH ₂ , Ph] , [RA2411; H, H, Et, Cl, CF ₂ HCH ₂ , Bn], [RA2412; H, H, Et, Cl, CF ₂ HCH ₂ , CF ₃ ], [RA2413; H, H, Et, Cl , CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA2414; H, H, Et, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA2415; H, H, Et, Cl, CF ₂ HCH ₂ , CF ₂ H], [RA2416; H, H, Et, Cl, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA2417; H, H, F, H, CF ₂ HCH ₂ , Me], [RA2418; H , H, F, H, CF ₂ HCH ₂ , Et], [RA2419; H, H, F, H, CF ₂ HCH ₂ , Pr], [RA2420; H, H, F, H, CF ₂ HCH ₂ , i-Pr], [RA2421; H, H, F, H, CF ₂ HCH ₂ , c-Pr], [RA2422; H, H, F, H, CF ₂ HCH ₂ , Bu], [RA2423; H, H, F, H, CF ₂ HCH ₂ , i-Bu], [RA2424; H, H, F, H, CF ₂ HCH ₂ , t-Bu], [RA2425; H, H, F, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA2426; H, H, F, H, CF ₂ HCH ₂ , Ph], [RA2427; H, H, F, H, CF ₂ HCH ₂ , Bn], [RA2428; H, H, F, H, CF ₂ HCH ₂ , CF ₃ ], [RA2429 ; H, H, F, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA2430; H, H, F, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA2431; H, H, F , H, CF ₂ HCH ₂ , CF ₂ H], [RA2432; H, H, F, H, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA2433; H, H, F, F, CF ₂ HCH ₂ , Me], [RA2434; H, H, F, F, CF ₂ HCH ₂ , Et], [RA2435; H, H, F, F, CF ₂ HCH ₂ , Pr], [RA2436; H, H, F , F, CF ₂ HCH ₂ , i-Pr], [RA2437; H, H, F, F, CF ₂ HCH ₂ , c-Pr], [RA2438; H, H, F, F, CF ₂ HCH ₂ , Bu], [RA2439; H, H, F, F, CF ₂ HCH ₂ , i-Bu], [RA2440; H, H, F, F, CF ₂ HCH ₂ , t-Bu], [RA2441; H, H, F, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA2442; H, H, F, F, CF ₂ HCH ₂ , Ph], [RA2443; H, H, F, F, CF ₂ HCH _{2, Bn], [RA2444;} H, H, F, F, CF 2 HCH 2, CF 3], [RA2445; H, H, F, F, CF 2 HCH 2, CF 3 CH 2], [RA2446; H, H, F, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA2447; H, H, F, F, CF ₂ HCH ₂ , CF ₂ H], [RA2448; H, H, F, F , CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA2449; H, H, F, Cl, CF ₂ HCH ₂ , Me], [RA2450; H, H, F, Cl, CF ₂ HCH ₂ , Et], [RA2451; H, H, F, Cl, CF ₂ HCH ₂ , Pr], [RA2452; H, H, F, Cl, CF ₂ HCH ₂ , i-Pr], [RA2453; H, H, F, Cl , CF ₂ HCH ₂ , c-Pr], [RA2454; H, H, F, Cl, CF ₂ HCH ₂ , Bu], [RA2455; H, H, F, Cl, CF ₂ HCH ₂ , i-Bu] , [RA2456; H, H, F, Cl, CF ₂ HCH ₂ , t-Bu], [RA2457; H, H, F, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA2458; H, H, F, Cl, CF ₂ HCH ₂ , Ph], [RA2459; H, H, F, Cl, CF ₂ HCH ₂ , Bn], [RA2460 ; H, H, F, Cl, CF ₂ HCH ₂ , CF ₃ ], [RA2461; H, H, F, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA2462; H, H, F, Cl , CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA2463; H, H, F, Cl, CF ₂ HCH ₂ , CF ₂ H], [RA2464; H, H, F, Cl, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA2465; H, H, Cl, H, CF ₂ HCH ₂ , Me], [RA2466; H, H, Cl, H, CF ₂ HCH ₂ , Et], [RA2467; H, H, Cl, H, CF ₂ HCH ₂ , Pr], [RA2468; H, H, Cl, H, CF ₂ HCH ₂ , i-Pr], [RA2469; H, H, Cl, H, CF ₂ HCH ₂ , c -Pr], [RA2470; H, H, Cl, H, CF ₂ HCH ₂ , Bu], [RA2471; H, H, Cl, H, CF ₂ HCH ₂ , i-Bu], [RA2472; H, H , Cl, H, CF ₂ HCH ₂ , t-Bu], [RA2473; H, H, Cl, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA2474; H, H, Cl, H, CF _{2 HCH 2, Ph], [RA2475} ; H, H, Cl, H, CF 2 HCH 2, Bn], [RA2476; H, H, Cl, H, CF 2 HCH 2, CF 3], [RA2477; H, H, Cl, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA2478; H, H, Cl, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA2479; H, H, Cl, H, CF ₂ HCH ₂ , CF ₂ H], [RA2480; H, H, Cl, H, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA2481; H, H, Cl, Cl, CF ₂ HCH ₂ , Me] , [RA2482; H, H, Cl, Cl, CF ₂ HCH ₂ , Et], [RA2483; H, H, Cl, Cl, CF ₂ HCH ₂ , Pr], [RA2484; H, H, Cl, Cl, CF ₂ HCH ₂ , i-Pr], [RA 2485; H, H, Cl, Cl, CF ₂ HCH ₂ , c-Pr], [RA2486; H, H, Cl, Cl, CF ₂ HCH ₂ , Bu], [RA2487; H, H, Cl, Cl, CF ₂ HCH ₂ , i-Bu], [RA2488; H, H, Cl, Cl, CF ₂ HCH ₂ , t-Bu], [RA2489; H, H, Cl, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA2490; H, H, Cl, Cl, CF ₂ HCH ₂ , Ph], [RA2491; H, H, Cl, Cl, CF ₂ HCH ₂ , Bn], [RA2492; H, H, Cl, Cl, CF ₂ HCH ₂ , CF ₃ ], [RA2493; H, H, Cl, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA2494; H, H, Cl, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA2495; H, H, Cl, Cl, CF ₂ HCH ₂ , CF ₂ H], [RA2496; H, H, Cl, Cl, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA2497 ; H, H, Me, H, CF ₃ CH ₂ , Me], [RA2498; H, H, Me, H, CF ₃ CH ₂ , Et], [RA2499; H, H, Me, H, CF ₃ CH ₂ , Pr], [RA2500; H, H, Me, H, CF ₃ CH ₂ , i-Pr], [RA2501; H, H, Me, H, CF ₃ CH ₂ , c-Pr], [RA2502; H, H, Me, H, CF ₃ CH ₂ , Bu], [RA2503; H, H, Me, H, CF ₃ CH ₂ , i-Bu], [RA2504; H, H, Me, H, CF ₃ CH ₂ , t-Bu], [RA2505; H, H, Me, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RA2506; H, H, Me, H, CF ₃ CH ₂ , Ph], [ RA2507; H, H, Me, H, CF ₃ CH ₂ , Bn], [RA2508; H, H, Me, H, CF ₃ CH ₂ , CF ₃ ], [RA2509; H, H, Me, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA2510; H, H, Me, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA2511; H, H, Me, H, CF ₃ CH ₂ , CF ₂ H], [RA2512; H, H, Me, H, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA2513; H, H, Me, Me, CF ₃ CH ₂ , Me], [RA2514; H, H, Me, Me, CF ₃ CH ₂ , Et], [RA2515; H, H, Me , Me, CF ₃ CH ₂ , Pr], [RA2516; H, H, Me, Me, CF ₃ CH ₂ , i-Pr], [RA2517; H, H, Me, Me, CF ₃ CH ₂ , c- Pr], [RA2518; H, H, Me, Me, CF ₃ CH ₂ , Bu], [RA2519; H, H, Me, Me, CF ₃ CH ₂ , i-Bu], [RA2520; H, H, Me, Me, CF ₃ CH ₂ , t-Bu], [RA2521; H, H, Me, Me, CF ₃ CH ₂ , c-PrCH ₂ ], [RA2522; H, H, Me, Me, CF ₃ CH ₂ , Ph], [RA2523; H, H, Me, Me, CF ₃ CH ₂ , Bn], [RA2524; H, H, Me, Me, CF ₃ CH ₂ , CF ₃ ], [RA2525; H, H , Me, Me, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA2526; H, H, Me, Me, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA2527; H, H, Me, Me, CF ₃ CH ₂ , CF ₂ H], [RA2528; H, H, Me, Me, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA2529; H, H, Me, Et, CF ₃ CH ₂ , Me], [RA2530; H, H, Me, Et, CF ₃ CH ₂ , Et], [RA2531; H, H, Me, Et, CF ₃ CH ₂ , Pr], [RA2532; H, H, Me, Et, CF ₃ CH ₂ , i-Pr], [RA2533; H, H, Me, Et, CF ₃ CH ₂ , c-Pr], [RA2534; H, H, Me, Et, CF ₃ CH ₂ , Bu], [ RA2535; H, H, Me, Et, CF ₃ CH ₂ , i-Bu], [RA2536; H, H, Me, Et, CF ₃ CH ₂ , t-Bu], [RA2537; H, H, Me, Et, CF ₃ CH ₂ , c-PrCH ₂ ], [RA2538; H, H, Me, Et, CF ₃ CH ₂ , Ph], [RA2539; H, H, Me, Et, CF ₃ CH ₂ , Bn] , [RA2540; H, H, Me, Et, CF ₃ CH ₂ , CF ₃ ], [R A2541; H, H, Me, Et, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA2542; H, H, Me, Et, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA2543; H, H, Me, Et, CF ₃ CH ₂ , CF ₂ H], [RA2544; H, H, Me, Et, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA2545; H, H, Me, F, CF ₃ CH ₂ , Me], [RA2546; H, H, Me, F, CF ₃ CH ₂ , Et], [RA2547; H, H, Me, F, CF ₃ CH ₂ , Pr], [RA2548; H, H, Me, F, CF ₃ CH ₂ , i-Pr], [RA2549; H, H, Me, F, CF ₃ CH ₂ , c-Pr], [RA2550; H, H, Me, F, CF ₃ CH ₂ , Bu], [RA2551; H, H, Me, F, CF ₃ CH ₂ , i-Bu], [RA2552; H, H, Me, F, CF ₃ CH ₂ , t-Bu], [RA2553; H , H, Me, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RA2554; H, H, Me, F, CF ₃ CH ₂ , Ph], [RA2555; H, H, Me, F, CF ₃ CH ₂ , Bn], [RA2556; H, H, Me, F, CF ₃ CH ₂ , CF ₃ ], [RA2557; H, H, Me, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA2558 ; H, H, Me, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA2559; H, H, Me, F, CF ₃ CH ₂ , CF ₂ H], [RA2560; H, H, Me, F, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA2561; H, H, Me, Cl, CF ₃ CH ₂ , Me], [RA2562; H, H, Me, Cl, CF ₃ CH ₂ , Et] , [RA2563; H, H, Me, Cl, CF ₃ CH ₂ , Pr], [RA2564; H, H, Me, Cl, CF ₃ CH ₂ , i-Pr], [RA2565; H, H, Me, Cl, CF ₃ CH ₂ , c-Pr], [RA2566; H, H, Me, Cl, CF ₃ CH ₂ , Bu], [RA2567; H, H, Me, Cl, CF ₃ CH ₂ , i-Bu ], [RA2568; H, H, Me, Cl, CF ₃ CH ₂ , t-Bu], [RA2569; H, H, Me, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RA2570; H, H, Me, Cl, CF ₃ CH ₂ , Ph], [RA2571; H, H, Me, Cl, CF ₃ CH ₂ , Bn], [RA2572; H, H, Me, Cl, CF ₃ CH ₂ , CF ₃ ], [RA2573; H, H, Me, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA2574; H, H, Me, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA2575; H, H, Me, Cl, CF _{3
CH 2, CF 2 H],} [RA2576; H, H, Me, Cl, CF 3 CH 2, CF 2 HCH 2], [RA2577; H, H, Et, H, CF 3 CH 2, Me], [ RA2578; H, H, Et, H, CF ₃ CH ₂ , Et], [RA2579; H, H, Et, H, CF ₃ CH ₂ , Pr], [RA2580; H, H, Et, H, CF _{3 CH 2, i-Pr],} [RA2581; H, H, Et, H, CF 3 CH 2, c-Pr], [RA2582; H, H, Et, H, CF 3 CH 2, Bu], [RA2583 ; H, H, Et, H, CF ₃ CH ₂ , i-Bu], [RA2584; H, H, Et, H, CF ₃ CH ₂ , t-Bu], [RA2585; H, H, Et, H , CF ₃ CH ₂ , c-PrCH ₂ ], [RA2586; H, H, Et, H, CF ₃ CH ₂ , Ph], [RA2587; H, H, Et, H, CF ₃ CH ₂ , Bn], [RA2588; H, H, Et, H, CF ₃ CH ₂ , CF ₃ ], [RA2589; H, H, Et, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA2590; H, H, Et , H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA2591; H, H, Et, H, CF ₃ CH ₂ , CF ₂ H], [RA2592; H, H, Et, H, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA2593; H, H, Et, F, CF ₃ CH ₂ , Me], [RA2594; H, H, Et, F, CF ₃ CH ₂ , Et], [RA2595; H, H, Et, F, CF ₃ CH ₂ , Pr], [RA2596; H, H, Et, F, CF ₃ CH ₂ , i-Pr], [RA2597; H, H, Et, F, CF ₃ CH ₂ , c-Pr], [RA2598; H, H, Et, F, CF ₃ CH ₂ , Bu], [RA2599; H, H, Et, F, CF ₃ CH ₂ , i-Bu], [RA2600; H , H, Et, F, CF ₃ CH ₂ , t-Bu],

[RA2601; H, H, Et, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RA2602; H, H, Et, F, CF ₃ CH ₂ , Ph], [RA2603; H, H, Et, F, CF ₃ CH ₂ , Bn], [RA2604; H, H, Et, F, CF ₃ CH ₂ , CF ₃ ], [RA2605; H, H, Et, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA2606; H, H, Et, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA2607; H, H, Et, F, CF ₃ CH ₂ , CF ₂ H], [RA2608; H, H, Et, F, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA2609; H, H, Et, Cl, CF ₃ CH ₂ , Me], [RA2610; H, H, Et, Cl, CF ₃ CH ₂ , Et], [RA2611; H, H, Et, Cl, CF ₃ CH ₂ , Pr], [RA2612; H, H, Et, Cl, CF ₃ CH ₂ , i-Pr], [RA2613; H, H, Et, Cl, CF ₃ CH ₂ , c-Pr], [RA2614; H, H, Et, Cl, CF ₃ CH ₂ , Bu], [RA2615; H, H, Et, Cl, CF ₃ CH ₂ , i-Bu], [RA2616; H, H, Et, Cl, CF ₃ CH ₂ , t-Bu], [RA2617; H, H, Et, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [ RA2618; H, H, Et, Cl, CF ₃ CH ₂ , Ph], [RA2619; H, H, Et, Cl, CF ₃ CH ₂ , Bn], [RA2620; H, H, Et, Cl, CF ₃ CH ₂ , CF ₃ ], [RA2621; H, H, Et, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA2622; H, H, Et, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ] , [RA2623; H, H, Et, Cl, CF ₃ CH ₂ , CF ₂ H], [RA2624; H, H, Et, Cl, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA2625; H, H , F, H, CF ₃ CH ₂ , Me], [RA2626; H, H, F, H, CF ₃ CH ₂ , Et], [RA2627; H, H, F, H, CF ₃ CH ₂ , Pr] , [RA2628; H, H, F, H, CF ₃ CH ₂ , i-Pr], [RA2 629; H, H, F, H, CF ₃ CH ₂ , c-Pr], [RA2630; H, H, F, H, CF ₃ CH ₂ , Bu], [RA2631; H, H, F, H, CF ₃ CH ₂ , i-Bu], [RA2632; H, H, F, H, CF ₃ CH ₂ , t-Bu], [RA2633; H, H, F, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RA2634; H, H, F, H, CF ₃ CH ₂ , Ph], [RA2635; H, H, F, H, CF ₃ CH ₂ , Bn], [RA2636; H, H, F, H, CF ₃ CH ₂ , CF ₃ ], [RA2637; H, H, F, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA2638; H, H, F, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA2639; H, H, F, H, CF ₃ CH ₂ , CF ₂ H], [RA2640; H, H, F, H, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA2641 ; H, H, F, F, CF ₃ CH ₂ , Me], [RA2642; H, H, F, F, CF ₃ CH ₂ , Et], [RA2643; H, H, F, F, CF ₃ CH ₂ , Pr], [RA2644; H, H, F, F, CF ₃ CH ₂ , i-Pr], [RA2645; H, H, F, F, CF ₃ CH ₂ , c-Pr], [RA2646; H, H, F, F, CF ₃ CH ₂ , Bu], [RA2647; H, H, F, F, CF ₃ CH ₂ , i-Bu], [RA2648; H, H, F, F, CF _{3 CH 2, t-Bu],} [RA2649; H, H, F, F, CF 3 CH 2, c-PrCH 2], [RA2650; H, H, F, F, CF 3 CH 2, Ph], [ RA2651; H, H, F, F, CF ₃ CH ₂ , Bn], [RA2652; H, H, F, F, CF ₃ CH ₂ , CF ₃ ], [RA2653; H, H, F, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA2654; H, H, F, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA2655; H, H, F, F, CF ₃ CH ₂ , CF ₂ H], [RA2656; H, H, F, F, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA2657; H, H, F, Cl, CF ₃ CH ₂ , Me], [RA2658; H, H , F, Cl, CF ₃ CH ₂ , Et], [RA2659; H, H, F, Cl, CF ₃ CH ₂ , Pr], [RA2660; H, H, F, Cl, CF ₃ CH ₂ , i-Pr ], [RA2661; H, H, F, Cl, CF ₃ CH ₂ , c-Pr], [RA2662; H, H, F, Cl, CF ₃ CH ₂ , Bu], [RA2663; H, H, F , Cl, CF ₃ CH ₂ , i-Bu], [RA2664; H, H, F, Cl, CF ₃ CH ₂ , t-Bu], [RA2665; H, H, F, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RA2666; H, H, F, Cl, CF ₃ CH ₂ , Ph], [RA2667; H, H, F, Cl, CF ₃ CH ₂ , Bn], [RA2668; H, H , F, Cl, CF ₃ CH ₂ , CF ₃ ], [RA2669; H, H, F, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA2670; H, H, F, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA2671; H, H, F, Cl, CF ₃ CH ₂ , CF ₂ H], [RA2672; H, H, F, Cl, CF ₃ CH ₂ , CF ₂ HCH ₂ ] , [RA2673; H, H, Cl, H, CF ₃ CH ₂ , Me], [RA2674; H, H, Cl, H, CF ₃ CH ₂ , Et], [RA2675; H, H, Cl, H, CF ₃ CH ₂ , Pr], [RA2676; H, H, Cl, H, CF ₃ CH ₂ , i-Pr], [RA2677; H, H, Cl, H, CF ₃ CH ₂ , c-Pr], [RA2678; H, H, Cl, H, CF ₃ CH ₂ , Bu], [RA2679; H, H, Cl, H, CF ₃ CH ₂ , i-Bu], [RA2680; H, H, Cl, H , CF ₃ CH ₂ , t-Bu], [RA2681; H, H, Cl, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RA2682; H, H, Cl, H, CF ₃ CH ₂ , Ph ], [RA2683; H, H, Cl, H, CF ₃ CH ₂ , Bn], [RA2684; H, H, Cl, H, CF ₃ CH ₂ , CF ₃ ], [RA2685; H, H, Cl, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA2686; H, H, Cl, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA 2687; H, H, Cl, H, CF ₃ CH ₂ , CF ₂ H], [RA2688; H, H, Cl, H, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA2689; H, H, Cl , Cl, CF ₃ CH ₂ , Me], [RA2690; H, H, Cl, Cl, CF ₃ CH ₂ , Et], [RA2691; H, H, Cl, Cl, CF ₃ CH ₂ , Pr], [ RA2692; H, H, Cl, Cl, CF ₃ CH ₂ , i-Pr], [RA2693; H, H, Cl, Cl, CF ₃ CH ₂ , c-Pr], [RA2694; H, H, Cl, Cl, CF ₃ CH ₂ , Bu], [RA2695; H, H, Cl, Cl, CF ₃ CH ₂ , i-Bu], [RA2696; H, H, Cl, Cl, CF ₃ CH ₂ , t-Bu ], [RA2697; H, H, Cl, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RA2698; H, H, Cl, Cl, CF ₃ CH ₂ , Ph], [RA2699; H, H, Cl, Cl, CF ₃ CH ₂ , Bn], [RA2700; H, H, Cl, Cl, CF ₃ CH ₂ , CF ₃ ], [RA2701; H, H, Cl, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA2702; H, H, Cl, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA2703; H, H, Cl, Cl, CF ₃ CH ₂ , CF ₂ H], [RA2704; H, H, Cl, Cl, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA2705; H, H, Me, H, HCCCH ₂ , Me], [RA2706; H, H, Me, H, HCCCH ₂ , Et], [RA2707; H, H, Me, H, HCCCH ₂ , Pr], [RA2708; H, H, Me, H, HCCCH ₂ , i-Pr], [RA2709; H, H, Me, H, HCCCH ₂ , c-Pr], [RA2710; H, H, Me, H, HCCCH ₂ , Bu], [RA2711; H, H, Me, H, HCCCH ₂ , i-Bu], [RA2712; H, H , Me, H, HCCCH ₂ , t-Bu], [RA2713; H, H, Me, H, HCCCH ₂ , c-PrCH ₂ ], [RA2714; H, H, Me, H, HCCCH ₂ , Ph], [RA2715; H, H, Me, H, HCCCH ₂ , Bn], [RA271 6; H, H, Me, H, HCCCH ₂ , CF ₃ ], [RA2717; H, H, Me, H, HCCCH ₂ , CF ₃ CH ₂ ], [RA2718; H, H, Me, H, HCCCH ₂ , CF ₃ CF ₂ ], [RA2719; H, H, Me, H, HCCCH ₂ , CF ₂ H], [RA2720; H, H, Me, H, HCCCH ₂ , CF ₂ HCH ₂ ], [RA2721; H , H, Me, Me, HCCCH ₂ , Me], [RA2722; H, H, Me, Me, HCCCH ₂ , Et], [RA2723; H, H, Me, Me, HCCCH ₂ , Pr], [RA2724; H, H, Me, Me, HCCCH ₂ , i-Pr], [RA2725; H, H, Me, Me, HCCCH ₂ , c-Pr], [RA2726; H, H, Me, Me, HCCCH ₂ , Bu ], [RA2727; H, H, Me, Me, HCCCH ₂ , i-Bu], [RA2728; H, H, Me, Me, HCCCH ₂ , t-Bu], [RA2729; H, H, Me, Me , HCCCH ₂ , c-PrCH ₂ ], [RA2730; H, H, Me, Me, HCCCH ₂ , Ph], [RA2731; H, H, Me, Me, HCCCH ₂ , Bn], [RA2732; H, H , Me, Me, HCCCH ₂ , CF ₃ ], [RA2733; H, H, Me, Me, HCCCH ₂ , CF ₃ CH ₂ ], [RA2734; H, H, Me, Me, HCCCH ₂ , CF ₃ CF ₂ ], [RA2735; H, H, Me, Me, HCCCH ₂ , CF ₂ H], [RA2736; H, H, Me, Me, HCCCH ₂ , CF ₂ HCH ₂ ], [RA2737; H, H, Me, Et, HCCCH ₂ , Me], [RA2738; H, H, Me, Et, HCCCH ₂ , Et], [RA2739; H, H, Me, Et, HCCCH ₂ , Pr], [RA2740; H, H, Me _{, Et, HCCCH 2, i-} Pr], [RA2741; H, H, Me, Et, HCCCH 2, c-Pr], [RA2742; H, H, Me, Et, HCCCH 2, Bu], [RA2743; H, H, Me, Et, HCCCH ₂ , i-Bu], [RA2744; H, H, Me, Et, HCCCH ₂ , t-Bu], [RA2745; H, H, Me, Et, HCCCH ₂ , c-PrCH ₂ ], [RA2746; H, H, Me, Et, HCCCH ₂ , Ph], [RA2747; H, H, Me, Et, HCCCH ₂ , Bn], [RA2748; H, H, Me, Et, HCCCH ₂ , CF ₃ ], [RA2749; H, H, Me, Et, HCCCH ₂ , CF ₃ CH ₂ ], [RA2750; H, H, Me, Et, HCCCH ₂ , CF ₃ CF ₂ ], [ RA2751; H, H, Me, Et, HCCCH ₂ , CF ₂ H], [RA2752; H, H, Me, Et, HCCCH ₂ , CF ₂ HCH ₂ ], [RA2753; H, H, Me, F, HCCCH ₂ , Me], [RA2754; H, H, Me, F, HCCCH ₂ , Et], [RA2755; H, H, Me, F, HCCCH ₂ , Pr], [RA2756; H, H, Me, F, HCCCH ₂ , i-Pr], [RA2757; H, H, Me, F, HCCCH ₂ , c-Pr], [RA2758; H, H, Me, F, HCCCH ₂ , Bu], [RA2759; H, H , Me, F, HCCCH ₂ , i-Bu], [RA2760; H, H, Me, F, HCCCH ₂ , t-Bu], [RA2761; H, H, Me, F, HCCCH ₂ , c-PrCH ₂ ], [RA2762; H, H, Me, F, HCCCH ₂ , Ph], [RA2763; H, H, Me, F, HCCCH ₂ , Bn], [RA2764; H, H, Me, F, HCCCH ₂ , CF ₃ ], [RA2765; H, H, Me, F, HCCCH ₂ , CF ₃ CH ₂ ], [RA2766; H, H, Me, F, HCCCH ₂ , CF ₃ CF ₂ ], [RA2767; H, H , Me, F, HCCCH ₂ , CF ₂ H], [RA2768; H, H, Me, F, HCCCH ₂ , CF ₂ HCH ₂ ], [RA2769; H, H, Me, Cl, HCCCH ₂ , Me], [RA2770; H, H, Me, Cl, HCCCH ₂ , Et], [RA2771; H, H, Me, Cl, HCCCH ₂ , Pr], [RA2772; H, H, Me, Cl, HCCCH ₂ , i- Pr], [RA2773; H, H, Me, Cl, HCCCH ₂ , c-Pr], [RA2774; H, H, Me, Cl, HCCCH ₂ , Bu], [RA2775; H, H, Me, Cl, HCC _{CH 2, i-Bu],} [RA2776; H, H, Me, Cl, HCCCH 2, t-Bu], [RA2777; H, H, Me, Cl, HCCCH 2, c-PrCH 2], [RA2778; H, H, Me, Cl, HCCCH ₂ , Ph], [RA2779; H, H, Me, Cl, HCCCH ₂ , Bn], [RA2780; H, H, Me, Cl, HCCCH ₂ , CF ₃ ], [ RA2781; H, H, Me, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RA2782; H, H, Me, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RA2783; H, H, Me, Cl, HCCCH ₂ , CF ₂ H], [RA2784; H, H, Me, Cl, HCCCH ₂ , CF ₂ HCH ₂ ], [RA2785; H, H, Et, H, HCCCH ₂ , Me], [RA2786; H, H, Et, H, HCCCH ₂ , Et], [RA2787; H, H, Et, H, HCCCH ₂ , Pr], [RA2788; H, H, Et, H, HCCCH ₂ , i-Pr], [RA2789 ; H, H, Et, H, HCCCH ₂ , c-Pr], [RA2790; H, H, Et, H, HCCCH ₂ , Bu], [RA2791; H, H, Et, H, HCCCH ₂ , i- Bu], [RA2792; H, H, Et, H, HCCCH ₂ , t-Bu], [RA2793; H, H, Et, H, HCCCH
₂ , c-PrCH ₂ ], [RA2794; H, H, Et, H, HCCCH ₂ , Ph], [RA2795; H, H, Et, H, HCCCH ₂ , Bn], [RA2796; H, H, Et , H, HCCCH ₂ , CF ₃ ], [RA2797; H, H, Et, H, HCCCH ₂ , CF ₃ CH ₂ ], [RA2798; H, H, Et, H, HCCCH ₂ , CF ₃ CF ₂ ], [RA2799; H, H, Et, H, HCCCH ₂ , CF ₂ H], [RA2800; H, H, Et, H, HCCCH ₂ , CF ₂ HCH ₂ ],

[RA2801; H, H, Et, F, HCCCH ₂ , Me], [RA2802; H, H, Et, F, HCCCH ₂ , Et], [RA2803; H, H, Et, F, HCCCH ₂ , Pr] , [RA2804; H, H, Et, F, HCCCH ₂ , i-Pr], [RA2805; H, H, Et, F, HCCCH ₂ , c-Pr], [RA2806; H, H, Et, F, HCCCH ₂ , Bu], [RA2807; H, H, Et, F, HCCCH ₂ , i-Bu], [RA2808; H, H, Et, F, HCCCH ₂ , t-Bu], [RA2809; H, H , Et, F, HCCCH ₂ , c-PrCH ₂ ], [RA2810; H, H, Et, F, HCCCH ₂ , Ph], [RA2811; H, H, Et, F, HCCCH ₂ , Bn], [RA2812 ; H, H, Et, F, HCCCH ₂ , CF ₃ ], [RA2813; H, H, Et, F, HCCCH ₂ , CF ₃ CH ₂ ], [RA2814; H, H, Et, F, HCCCH ₂ , CF ₃ CF ₂ ], [RA2815; H, H, Et, F, HCCCH ₂ , CF ₂ H], [RA2816; H, H, Et, F, HCCCH ₂ , CF ₂ HCH ₂ ], [RA2817; H, _{H, Et, Cl, HCCCH 2} , Me], [RA2818; H, H, Et, Cl, HCCCH 2, Et], [RA2819; H, H, Et, Cl, HCCCH 2, Pr], [RA2820; H , H, Et, Cl, HCCCH ₂ , i-Pr], [RA2821; H, H, Et, Cl, HCCCH ₂ , c-Pr], [RA2822; H, H, Et, Cl, HCCCH ₂ , Bu] , [RA2823; H, H, Et, Cl, HCCCH ₂ , i-Bu], [RA2824; H, H, Et, Cl, HCCCH ₂ , t-Bu], [RA2825; H, H, Et, Cl, HCCCH ₂ , c-PrCH ₂ ], [RA2826; H, H, Et, Cl, HCCCH ₂ , Ph], [RA2827; H, H, Et, Cl, HCCCH ₂ , Bn], [RA2828; H, H, Et, Cl, HCCCH ₂ , CF ₃ ], [RA2829; H, H, Et, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RA2830; H, H, Et, Cl, HCCCH ₂ , CF ₃ CF ₂ ] , [RA28 31; H, H, Et, Cl, HCCCH ₂ , CF ₂ H], [RA2832; H, H, Et, Cl, HCCCH ₂ , CF ₂ HCH ₂ ], [RA2833; H, H, F, H, HCCCH ₂ , Me], [RA2834; H, H, F, H, HCCCH ₂ , Et], [RA2835; H, H, F, H, HCCCH ₂ , Pr], [RA2836; H, H, F, H, HCCCH ₂ , i-Pr], [RA2837; H, H, F, H, HCCCH ₂ , c-Pr], [RA2838; H, H, F, H, HCCCH ₂ , Bu], [RA2839; H, H , F, H, HCCCH ₂ , i-Bu], [RA2840; H, H, F, H, HCCCH ₂ , t-Bu], [RA2841; H, H, F, H, HCCCH ₂ , c-PrCH ₂ ], [RA2842; H, H, F, H, HCCCH ₂ , Ph], [RA2843; H, H, F, H, HCCCH ₂ , Bn], [RA2844; H, H, F, H, HCCCH ₂ , CF ₃ ], [RA2845; H, H, F, H, HCCCH ₂ , CF ₃ CH ₂ ], [RA2846; H, H, F, H, HCCCH ₂ , CF ₃ CF ₂ ], [RA2847; H, H , F, H, HCCCH ₂ , CF ₂ H], [RA2848; H, H, F, H, HCCCH ₂ , CF ₂ HCH ₂ ], [RA2849; H, H, F, F, HCCCH ₂ , Me], [RA2850; H, H, F, F, HCCCH ₂ , Et], [RA2851; H, H, F, F, HCCCH ₂ , Pr], [RA2852; H, H, F, F, HCCCH ₂ , i- Pr], [RA2853; H, H, F, F, HCCCH ₂ , c-Pr], [RA2854; H, H, F, F, HCCCH ₂ , Bu], [RA2855; H, H, F, F, HCCCH ₂ , i-Bu], [RA2856; H, H, F, F, HCCCH ₂ , t-Bu], [RA2857; H, H, F, F, HCCCH ₂ , c-PrCH ₂ ], [RA2858; H, H, F, F, HCCCH ₂ , Ph], [RA2859; H, H, F, F, HCCCH ₂ , Bn], [RA2860; H, H, F, F, HCCCH ₂ , CF ₃ ], [ RA2861; H, H, F, F, HCCCH ₂ , CF ₃ CH ₂ ], [RA2862; H, H, F, F, HCCCH ₂ , CF ₃ CF ₂ ], [RA2863; H, H, F, F, HCCCH ₂ , CF ₂ H], [RA2864; H, H, F, F, HCCCH ₂ , CF ₂ HCH ₂ ], [RA2865 ; H, H, F, Cl, HCCCH ₂ , Me], [RA2866; H, H, F, Cl, HCCCH ₂ , Et], [RA2867; H, H, F, Cl, HCCCH ₂ , Pr], [ RA2868; H, H, F, Cl, HCCCH ₂ , i-Pr], [RA2869; H, H, F, Cl, HCCCH ₂ , c-Pr], [RA2870; H, H, F, Cl, HCCCH ₂ , Bu], [RA2871; H, H, F, Cl, HCCCH ₂ , i-Bu], [RA2872; H, H, F, Cl, HCCCH ₂ , t-Bu], [RA2873; H, H, F , Cl, HCCCH ₂ , c-PrCH ₂ ], [RA2874; H, H, F, Cl, HCCCH ₂ , Ph], [RA2875; H, H, F, Cl, HCCCH ₂ , Bn], [RA2876; H , H, F, Cl, HCCCH ₂ , CF ₃ ], [RA2877; H, H, F, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RA2878; H, H, F, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RA2879; H, H, F, Cl, HCCCH ₂ , CF ₂ H], [RA2880; H, H, F, Cl, HCCCH ₂ , CF ₂ HCH ₂ ], [RA2881; H, H, Cl, H, HCCCH ₂ , Me], [RA2882; H, H, Cl, H, HCCCH ₂ , Et], [RA2883; H, H, Cl, H, HCCCH ₂ , Pr], [RA2884; H, H , Cl, H, HCCCH ₂ , i-Pr], [RA2885; H, H, Cl, H, HCCCH ₂ , c-Pr], [RA2886; H, H, Cl, H, HCCCH ₂ , Bu], [ RA2887; H, H, Cl, H, HCCCH ₂ , i-Bu], [RA2888; H, H, Cl, H, HCCCH ₂ , t-Bu], [RA2889; H, H, Cl, H, HCCCH ₂ , c-PrCH ₂ ], [RA2890; H, H, Cl, H, HCCCH ₂ , Ph], [RA2891; H, H, Cl, H, HCCCH ₂ , Bn], [RA2892; H, H, Cl, H, HCCCH ₂ , CF ₃ ], [RA 2893; H, H, Cl, H, HCCCH ₂ , CF ₃ CH ₂ ], [RA2894; H, H, Cl, H, HCCCH ₂ , CF ₃ CF ₂ ], [RA2895; H, H, Cl, H, HCCCH ₂ , CF ₂ H], [RA2896; H, H, Cl, H, HCCCH ₂ , CF ₂ HCH ₂ ], [RA2897; H, H, Cl, Cl, HCCCH ₂ , Me], [RA2898; H, H, Cl, Cl, HCCCH ₂ , Et], [RA2899; H, H, Cl, Cl, HCCCH ₂ , Pr], [RA2900; H, H, Cl, Cl, HCCCH ₂ , i-Pr], [RA2901 ; H, H, Cl, Cl, HCCCH ₂ , c-Pr], [RA2902; H, H, Cl, Cl, HCCCH ₂ , Bu], [RA2903; H, H, Cl, Cl, HCCCH ₂ , i- Bu], [RA2904; H, H, Cl, Cl, HCCCH ₂ , t-Bu], [RA2905; H, H, Cl, Cl, HCCCH ₂ , c-PrCH ₂ ], [RA2906; H, H, Cl , Cl, HCCCH ₂ , Ph], [RA2907; H, H, Cl, Cl, HCCCH ₂ , Bn], [RA2908; H, H, Cl, Cl, HCCCH ₂ , CF ₃ ], [RA2909; H, H , Cl, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RA2910; H, H, Cl, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RA2911; H, H, Cl, Cl, HCCCH ₂ , CF ₂ H], [RA2912; H, H, Cl, Cl, HCCCH ₂ , CF ₂ HCH ₂ ], [RA2913; H, H, Me, H, CH ₃ CCCH ₂ , Me], [RA2914; H, H, Me , H, CH ₃ CCCH ₂ , Et], [RA2915; H, H, Me, H, CH ₃ CCCH ₂ , Pr], [RA2916; H, H, Me, H, CH ₃ CCCH ₂ , i-Pr] , [RA2917; H, H, Me, H, CH ₃ CCCH ₂ , c-Pr], [RA2918; H, H, Me, H, CH ₃ CCCH ₂ , Bu], [RA2919; H, H, Me, H, CH ₃ CCCH ₂ , i-Bu], [RA2920; H, H, Me, H, CH ₃ CCCH ₂ , t-Bu], [RA2921; H, H, Me, H, CH ₃ CCCH ₂ , c -PrCH ₂ ], [RA2922; H, H, Me, H, CH ₃ CCCH ₂ , Ph], [RA2923; H, H, Me, H, CH ₃ CCCH ₂ , Bn], [RA2924; H, H, Me, H, CH ₃ CCCH ₂ , CF ₃ ], [RA2925; H, H, Me, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA2926; H, H, Me, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA2927; H, H, Me, H, CH ₃ CCCH ₂ , CF ₂ H], [RA2928; H, H, Me, H, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA2929; H, H, Me, Me, CH ₃ CCCH ₂ , Me], [RA2930; H, H, Me, Me, CH ₃ CCCH ₂ , Et], [RA2931; H, H, Me, Me, CH ₃ CCCH ₂ , Pr], [RA2932; H, H, Me, Me, CH ₃ CCCH ₂ , i-Pr], [RA2933; H, H, Me, Me, CH ₃ CCCH ₂ , c-Pr], [ RA2934; H, H, Me, Me, CH ₃ CCCH ₂ , Bu], [RA2935; H, H, Me, Me, CH ₃ CCCH ₂ , i-Bu], [RA2936; H, H, Me, Me, CH ₃ CCCH ₂ , t-Bu], [RA2937; H, H, Me, Me, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA2938; H, H, Me, Me, CH ₃ CCCH ₂ , Ph] , [RA2939; H, H, Me, Me, CH ₃ CCCH ₂ , Bn], [RA2940; H, H, Me, Me, CH ₃ CCCH ₂ , CF ₃ ], [RA2941; H, H, Me, Me , CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA2942; H, H, Me, Me, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA2943; H, H, Me, Me, CH ₃ CCCH ₂ , CF ₂ H], [RA2944; H, H, Me, Me, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA2945; H, H, Me, Et, CH ₃ CCCH ₂ , Me], [RA2946; H , H, Me, Et, CH ₃ CCCH ₂ , Et], [RA2947; H, H, Me, Et, CH ₃ CCCH ₂ , Pr], [RA2948; H, H, Me, Et, CH ₃ CCCH ₂ , i-Pr], [RA2949; H, H, Me, Et, CH ₃ CCCH ₂ , c-Pr], [RA2950; H, H, Me, Et, CH ₃ CCCH ₂ , Bu], [RA2951; H, H, Me, Et, CH ₃ CCCH ₂ , i-Bu], [RA2952; H, H, Me, Et, CH ₃ CCCH ₂ , t-Bu], [RA2953; H, H, Me, Et, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA2954; H, H, Me, Et, CH ₃ CCCH ₂ , Ph], [RA2955; H, H, Me, Et, CH ₃ CCCH ₂ , Bn], [RA2956; H, H, Me, Et, CH ₃ CCCH ₂ , CF ₃ ], [RA2957; H, H, Me, Et, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA2958; H, H, Me, Et, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA2959; H, H, Me, Et, CH ₃ CCCH ₂ , CF ₂ H], [RA2960; H, H, Me, Et, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA2961; H, H, Me, F, CH ₃ CCCH ₂ , Me], [RA2962; H, H, Me, F, CH ₃ CCCH ₂ , Et], [RA2963; H, H, Me, F, CH ₃ CCCH ₂ , Pr], [RA2964; H, H, Me, F, CH ₃ CCCH ₂ , i-Pr], [RA2965; H, H, Me, F, CH ₃ CCCH ₂ , c-Pr], [RA2966; H, H, Me, F, CH ₃ CCCH ₂ , Bu], [RA2967; H, H, Me, F, CH ₃ CCCH ₂ , i-Bu], [RA2968; H, H, Me, F, CH ₃ CCCH ₂ , t-Bu], [RA2969; H, H, Me, F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [ RA2970; H, H, Me, F, CH ₃ CCCH ₂ , Ph], [RA2971; H, H, Me, F, CH ₃ CCCH ₂ , Bn], [RA2972; H, H, Me, F, CH ₃ CCCH ₂ , CF ₃ ], [RA2973; H, H, Me, F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA2974; H, H, Me, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA2975; H, H, Me, F, CH ₃ CCCH ₂ , CF ₂ H], [RA2976; H, H, Me, F, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA2977; H , H, Me, Cl, CH ₃ CCCH ₂ , Me], [RA2978; H, H, Me, Cl, CH ₃ CCCH ₂ , Et], [RA2979; H, H, Me, Cl, CH ₃ CCCH ₂ , Pr], [RA2980; H, H, Me, Cl, CH ₃ CCCH ₂ , i-Pr], [RA2981; H, H, Me, Cl, CH ₃ CCCH ₂ , c-Pr], [RA2982; H, H, Me, Cl, CH ₃ CCCH ₂ , Bu], [RA2983; H, H, Me, Cl, CH ₃ CCCH ₂ , i-Bu], [RA2984; H, H, Me, Cl, CH ₃ CCCH ₂ , t-Bu], [RA2985; H, H, Me, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA2986; H, H, Me, Cl, CH ₃ CCCH ₂ , Ph], [RA2987; H, H, Me, Cl, CH ₃ CCCH ₂ , Bn], [RA2988; H, H, Me, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RA2989; H, H, Me, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA2990; H, H, Me, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA2991; H, H, Me, Cl, CH ₃ CCCH ₂ , CF ₂ H] , [RA2992; H, H, Me, Cl, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA2993; H, H, Et, H, CH ₃ CCCH ₂ , Me], [RA2994; H, H, Et , H, CH ₃ CCCH ₂ , Et], [RA2995; H, H, Et, H, CH ₃
CCCH ₂ , Pr], [RA2996; H, H, Et, H, CH ₃ CCCH ₂ , i-Pr], [RA2997; H, H, Et, H, CH ₃ CCCH ₂ , c-Pr], [RA2998 ; H, H, Et, H, CH ₃ CCCH ₂ , Bu], [RA2999; H, H, Et, H, CH ₃ CCCH ₂ , i-Bu], [RA3000; H, H, Et, H, CH ₃ CCCH ₂ , t-Bu],

[RA3001; H, H, Et, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA3002; H, H, Et, H, CH ₃ CCCH ₂ , Ph], [RA3003; H, H, Et, H, CH ₃ CCCH ₂ , Bn], [RA3004; H, H, Et, H, CH ₃ CCCH ₂ , CF ₃ ], [RA3005; H, H, Et, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA3006; H, H, Et, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA3007; H, H, Et, H, CH ₃ CCCH ₂ , CF ₂ H], [RA3008; H, H, Et, H, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA3009; H, H, Et, F, CH ₃ CCCH ₂ , Me], [RA3010; H, H, Et, F, CH ₃ CCCH ₂ , Et], [RA3011; H, H, Et, F, CH ₃ CCCH ₂ , Pr], [RA3012; H, H, Et, F, CH ₃ CCCH ₂ , i-Pr], [RA3013; H, H, Et, F, CH ₃ CCCH ₂ , c-Pr], [RA3014; H, H, Et, F, CH ₃ CCCH ₂ , Bu], [RA3015; H, H, Et, F, CH ₃ CCCH ₂ , i-Bu], [RA3016; H, H, Et, F, CH ₃ CCCH ₂ , t-Bu], [RA3017; H, H, Et, F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [ RA3018; H, H, Et, F, CH ₃ CCCH ₂ , Ph], [RA3019; H, H, Et, F, CH ₃ CCCH ₂ , Bn], [RA3020; H, H, Et, F, CH ₃ CCCH ₂ , CF ₃ ], [RA3021; H, H, Et, F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA3022; H, H, Et, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ] , [RA3023; H, H, Et, F, CH ₃ CCCH ₂ , CF ₂ H], [RA3024; H, H, Et, F, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA3025; H, H , Et, Cl, CH ₃ CCCH ₂ , Me], [RA3026; H, H, Et, Cl, CH ₃ CCCH ₂ , Et], [RA3027; H, H, Et, Cl, CH ₃ CCCH ₂ , Pr], [RA3028; H, H, Et, Cl, CH ₃ CCCH ₂ , i-Pr], [RA3029; H, H, Et, Cl, CH ₃ CCCH ₂ , c-Pr], [RA3030; H, H, Et, Cl, CH ₃ CCCH ₂ , Bu], [RA3031; H, H, Et, Cl, CH ₃ CCCH ₂ , i-Bu], [RA3032; H, H, Et, Cl, CH ₃ CCCH ₂ , t-Bu], [RA3033; H, H, Et, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA3034; H, H, Et, Cl, CH ₃ CCCH ₂ , Ph], [ RA3035; H, H, Et, Cl, CH ₃ CCCH ₂ , Bn], [RA3036; H, H, Et, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RA3037; H, H, Et, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA3038; H, H, Et, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA3039; H, H, Et, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RA3040; H, H, Et, Cl, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA3041; H, H, F, H, CH ₃ CCCH ₂ , Me], [RA3042; H, H , F, H, CH ₃ CCCH ₂ , Et], [RA3043; H, H, F, H, CH ₃ CCCH ₂ , Pr], [RA3044; H, H, F, H, CH ₃ CCCH ₂ , i- Pr], [RA3045; H, H, F, H, CH ₃ CCCH ₂ , c-Pr], [RA3046; H, H, F, H, CH ₃ CCCH ₂ , Bu], [RA3047; H, H, F, H, CH ₃ CCCH ₂ , i-Bu], [RA3048; H, H, F, H, CH ₃ CCCH ₂ , t-Bu], [RA3049; H, H, F, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA3050; H, H, F, H, CH ₃ CCCH ₂ , Ph], [RA3051; H, H, F, H, CH ₃ CCCH ₂ , Bn], [RA3052; H, H, F, H, CH ₃ CCCH ₂ , CF ₃ ], [RA3053; H, H, F, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA3054; H, H, F, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA3055; H, H, F, H, CH ₃ CCCH ₂ , CF ₂ H], [RA3056; H, H, F, H, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA3057; H , H, F, F, CH ₃ CCCH ₂ , Me], [RA3058; H, H, F, F, CH ₃ CCCH ₂ , Et], [RA3059; H, H, F, F, CH ₃ CCCH ₂ , Pr], [RA3060; H, H, F, F, CH ₃ CCCH ₂ , i-Pr], [RA3061; H, H, F, F, CH ₃ CCCH ₂ , c-Pr], [RA3062; H, H, F, F, CH ₃ CCCH ₂ , Bu], [RA3063; H, H, F, F, CH ₃ CCCH ₂ , i-Bu], [RA3064; H, H, F, F, CH ₃ CCCH ₂ , t-Bu], [RA3065; H, H, F, F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA3066; H, H, F, F, CH ₃ CCCH ₂ , Ph], [RA3067; H, H, F, F, CH ₃ CCCH ₂ , Bn], [RA3068; H, H, F, F, CH ₃ CCCH ₂ , CF ₃ ], [RA3069; H, H, F, F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA3070; H, H, F, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA3071; H, H, F, F, CH ₃ CCCH ₂ , CF ₂ H] , [RA3072; H, H, F, F, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA3073; H, H, F, Cl, CH ₃ CCCH ₂ , Me], [RA3074; H, H, F , Cl, CH ₃ CCCH ₂ , Et], [RA3075; H, H, F, Cl, CH ₃ CCCH ₂ , Pr], [RA3076; H, H, F, Cl, CH ₃ CCCH ₂ , i-Pr] , [RA3077; H, H, F, Cl, CH ₃ CCCH ₂ , c-Pr], [RA3078; H, H, F, Cl, CH ₃ CCCH ₂ , Bu], [RA3079; H, H, F, Cl, CH ₃ CCCH ₂ , i-Bu], [RA3080; H, H, F, Cl, CH ₃ CCCH ₂ , t-Bu], [RA3081; H, H, F, Cl, CH ₃ CCCH ₂ , c -PrCH ₂ ], [RA3082; H, H, F, Cl, CH ₃ CCCH ₂ , Ph], [RA3083; H, H, F, Cl, CH ₃ CCCH ₂ , Bn], [RA3084; H, H, F, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RA3085; H , H, F, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA3086; H, H, F, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA3087; H, H, F, Cl , CH ₃ CCCH ₂ , CF ₂ H], [RA3088; H, H, F, Cl, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA3089; H, H, Cl, H, CH ₃ CCCH ₂ , Me ], [RA3090; H, H, Cl, H, CH ₃ CCCH ₂ , Et], [RA3091; H, H, Cl, H, CH ₃ CCCH ₂ , Pr], [RA3092; H, H, Cl, H , CH ₃ CCCH ₂ , i-Pr], [RA3093; H, H, Cl, H, CH ₃ CCCH ₂ , c-Pr], [RA3094; H, H, Cl, H, CH ₃ CCCH ₂ , Bu] , [RA3095; H, H, Cl, H, CH ₃ CCCH ₂ , i-Bu], [RA3096; H, H, Cl, H, CH ₃ CCCH ₂ , t-Bu], [RA3097; H, H, Cl, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA3098; H, H, Cl, H, CH ₃ CCCH ₂ , Ph], [RA3099; H, H, Cl, H, CH ₃ CCCH ₂ , Bn], [RA3100; H, H, Cl, H, CH ₃ CCCH ₂ , CF ₃ ], [RA3101; H, H, Cl, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA3102; H, H, Cl, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA3103; H, H, Cl, H, CH ₃ CCCH ₂ , CF ₂ H], [RA3104; H, H, Cl, H, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA3105; H, H, Cl, Cl, CH ₃ CCCH ₂ , Me], [RA3106; H, H, Cl, Cl, CH ₃ CCCH ₂ , Et], [RA3107 ; H, H, Cl, Cl, CH ₃ CCCH ₂ , Pr], [RA3108; H, H, Cl, Cl, CH ₃ CCCH ₂ , i-Pr], [RA3109; H, H, Cl, Cl , CH ₃ CCCH ₂ , c-Pr], [RA3110; H, H, Cl, Cl, CH ₃ CCCH ₂ , Bu], [RA3111; H, H, Cl, Cl, CH ₃ CCCH ₂ , i-Bu] , [RA3112; H, H, Cl, Cl, CH ₃ CCCH ₂ , t-Bu], [RA3113; H, H, Cl, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA3114; H, H , Cl, Cl, CH ₃ CCCH ₂ , Ph], [RA3115; H, H, Cl, Cl, CH ₃ CCCH ₂ , Bn], [RA3116; H, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RA3117; H, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA3118; H, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA3119; H , H, Cl, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RA3120; H, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA3121; H, H, Me, H, c-PrCH ₂ , Me], [RA3122; H, H, Me, H, c-PrCH ₂ , Et], [RA3123; H, H, Me, H, c-PrCH ₂ , Pr], [RA3124; H , H, Me, H, c-PrCH ₂ , i-Pr], [RA3125; H, H, Me, H, c-PrCH ₂ , c-Pr], [RA3126; H, H, Me, H, c -PrCH ₂ , Bu], [RA3127; H, H, Me, H, c-PrCH ₂ , i-Bu], [RA3128; H, H, Me, H, c-PrCH ₂ , t-Bu], [ RA3129; H, H, Me, H, c-PrCH ₂ , c-PrCH ₂ ], [RA3130; H, H, Me, H, c-PrCH ₂ , Ph], [RA3131; H, H, Me, H , c-PrCH ₂ , Bn], [RA3132; H, H, Me, H, c-PrCH ₂ , CF ₃ ], [RA3133; H, H, Me, H, c-PrCH ₂ , CF ₃ CH ₂ ] , [RA3134; H, H, Me, H, c-PrCH ₂ , CF ₃ CF ₂ ], [RA3135; H, H, Me, H, c-PrCH ₂ , CF ₂ H], [RA3136; H, H , Me, H, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA3137; H , H, Me, Me, c-PrCH ₂ , Me], [RA3138; H, H, Me, Me, c-PrCH ₂ , Et], [RA3139; H, H, Me, Me, c-PrCH ₂ , Pr], [RA3140; H, H, Me, Me, c-PrCH ₂ , i-Pr], [RA3141; H, H, Me, Me, c-PrCH ₂ , c-Pr], [RA3142; H, H, Me, Me, c-PrCH ₂ , Bu], [RA3143; H, H, Me, Me, c-PrCH ₂ , i-Bu], [RA3144; H, H, Me, Me, c-PrCH ₂ , t-Bu], [RA3145; H, H, Me, Me, c-PrCH ₂ , c-PrCH ₂ ], [RA3146; H, H, Me, Me, c-PrCH ₂ , Ph], [RA3147; H, H, Me, Me, c-PrCH ₂ , Bn], [RA3148; H, H, Me, Me, c-PrCH ₂ , CF ₃ ], [RA3149; H, H, Me, Me, c-PrCH ₂ , CF ₃ CH ₂ ], [RA3150; H, H, Me, Me, c-PrCH ₂ , CF ₃ CF ₂ ], [RA3151; H, H, Me, Me, c-PrCH ₂ , CF ₂ H] , [RA3152; H, H, Me, Me, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA3153; H, H, Me, Et, c-PrCH ₂ , Me], [RA3154; H, H, Me , Et, c-PrCH ₂ , Et], [RA3155; H, H, Me, Et, c-PrCH ₂ , Pr], [RA3156; H, H, Me, Et, c-PrCH ₂ , i-Pr] , [RA3157; H, H, Me, Et, c-PrCH ₂ , c-Pr], [RA3158; H, H, Me, Et, c-PrCH ₂ , Bu], [RA3159; H, H, Me, Et, c-PrCH ₂ , i-Bu], [RA3160; H, H, Me, Et, c-PrCH ₂ , t-Bu], [RA3161; H, H, Me, Et, c-PrCH ₂ , c -PrCH ₂ ], [RA3162; H, H, Me, Et, c-PrCH ₂ , Ph], [RA3163; H, H, Me, Et, c-PrCH ₂ , Bn], [RA3164; H, H, Me, Et, c-PrCH ₂ , CF ₃ ], [RA3165; H, H, Me, Et, c-PrCH ₂ , CF ₃ CH ₂ ], [RA3166; H, H, Me, Et, c-PrCH ₂ , CF ₃ CF ₂ ], [RA3167; H, H, Me, Et, c-PrCH ₂ , CF ₂ H], [RA3168; H, H, Me, Et , c-PrCH ₂ , CF ₂ HCH ₂ ], [RA3169; H, H, Me, F, c-PrCH ₂ , Me], [RA3170; H, H, Me, F, c-PrCH ₂ , Et], [RA3171; H, H, Me, F, c-PrCH ₂ , Pr], [RA3172; H, H, Me, F, c-PrCH ₂ , i-Pr], [RA3173; H, H, Me, F , c-PrCH ₂ , c-Pr], [RA3174; H, H, Me, F, c-PrCH ₂ , Bu], [RA3175; H, H, Me, F, c-PrCH ₂ , i-Bu] , [RA3176; H, H, Me, F, c-PrCH ₂ , t-Bu], [RA3177; H, H, Me, F, c-PrCH ₂ , c-PrCH ₂ ], [RA3178; H, H , Me, F, c-PrCH ₂ , Ph], [RA3179; H, H, Me, F, c-PrCH ₂ , Bn], [RA3180; H, H, Me, F, c-PrCH ₂ , CF ₃ ], [RA3181; H, H, Me, F, c-PrCH ₂ , CF ₃ CH ₂ ], [RA3182; H, H, Me, F, c-PrCH ₂ , CF ₃ CF ₂ ], [
RA3183; H, H, Me, F, c-PrCH ₂ , CF ₂ H], [RA3184; H, H, Me, F, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA3185; H, H, Me , Cl, c-PrCH ₂ , Me], [RA3186; H, H, Me, Cl, c-PrCH ₂ , Et], [RA3187; H, H, Me, Cl, c-PrCH ₂ , Pr], [ RA3188; H, H, Me, Cl, c-PrCH 2, i-Pr], [RA3189; H, H, Me, Cl, c-PrCH 2, c-Pr], [RA3190; H, H, Me, Cl, c-PrCH ₂ , Bu], [RA3191; H, H, Me, Cl, c-PrCH ₂ , i-Bu], [RA3192; H, H, Me, Cl, c-PrCH ₂ , t-Bu ], [RA3193; H, H, Me, Cl, c-PrCH ₂ , c-PrCH ₂ ], [RA3194; H, H, Me, Cl, c-PrCH ₂ , Ph], [RA3195; H, H, Me, Cl, c-PrCH ₂ , Bn], [RA3196; H, H, Me, Cl, c-PrCH ₂ , CF ₃ ], [RA3197; H, H, Me, Cl, c-PrCH ₂ , CF ₃ CH ₂ ], [RA3198; H, H, Me, Cl, c-PrCH ₂ , CF ₃ CF ₂ ], [RA3199; H, H, Me, Cl, c-PrCH ₂ , CF ₂ H], [RA3200; H, H, Me, Cl, c-PrCH ₂ , CF ₂ HCH ₂ ],

[RA3201; H, H, Et, H, c-PrCH ₂ , Me], [RA3202; H, H, Et, H, c-PrCH ₂ , Et], [RA3203; H, H, Et, H, c -PrCH ₂ , Pr], [RA3204; H, H, Et, H, c-PrCH ₂ , i-Pr], [RA3205; H, H, Et, H, c-PrCH ₂ , c-Pr], [ RA3206; H, H, Et, H, c-PrCH ₂ , Bu], [RA3207; H, H, Et, H, c-PrCH ₂ , i-Bu], [RA3208; H, H, Et, H, c-PrCH ₂ , t-Bu], [RA3209; H, H, Et, H, c-PrCH ₂ , c-PrCH ₂ ], [RA3210; H, H, Et, H, c-PrCH ₂ , Ph] , [RA3211; H, H, Et, H, c-PrCH ₂ , Bn], [RA3212; H, H, Et, H, c-PrCH ₂ , CF ₃ ], [RA3213; H, H, Et, H , c-PrCH ₂ , CF ₃ CH ₂ ], [RA3214; H, H, Et, H, c-PrCH ₂ , CF ₃ CF ₂ ], [RA3215; H, H, Et, H, c-PrCH ₂ , CF ₂ H], [RA3216; H, H, Et, H, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA3217; H, H, Et, F, c-PrCH ₂ , Me], [RA3218; H , H, Et, F, c-PrCH ₂ , Et], [RA3219; H, H, Et, F, c-PrCH ₂ , Pr], [RA3220; H, H, Et, F, c-PrCH ₂ , i-Pr], [RA3221; H, H, Et, F, c-PrCH ₂ , c-Pr], [RA3222; H, H, Et, F, c-PrCH ₂ , Bu], [RA3223; H, H, Et, F, c-PrCH ₂ , i-Bu], [RA3224; H, H, Et, F, c-PrCH ₂ , t-Bu], [RA3225; H, H, Et, F, c- _{PrCH 2, c-PrCH 2]} , [RA3226; H, H, Et, F, c-PrCH 2, Ph], [RA3227; H, H, Et, F, c-PrCH 2, Bn], [RA3228; H, H, Et, F, c-PrCH ₂ , CF ₃ ], [RA3229; H, H, Et, F, c-PrCH ₂ , CF ₃ CH ₂ ], [RA3230; H, H, Et, F, c-PrCH ₂ , C F ₃ CF ₂ ], [RA3231; H, H, Et, F, c-PrCH ₂ , CF ₂ H], [RA3232; H, H, Et, F, c-PrCH ₂ , CF ₂ HCH ₂ ], [ RA3233; H, H, Et, Cl, c-PrCH ₂ , Me], [RA3234; H, H, Et, Cl, c-PrCH ₂ , Et], [RA3235; H, H, Et, Cl, c- _{PrCH 2, Pr], [RA3236} ; H, H, Et, Cl, c-PrCH 2, i-Pr], [RA3237; H, H, Et, Cl, c-PrCH 2, c-Pr], [RA3238 ; H, H, Et, Cl, c-PrCH ₂ , Bu], [RA3239; H, H, Et, Cl, c-PrCH ₂ , i-Bu], [RA3240; H, H, Et, Cl, c -PrCH ₂ , t-Bu], [RA3241; H, H, Et, Cl, c-PrCH ₂ , c-PrCH ₂ ], [RA3242; H, H, Et, Cl, c-PrCH ₂ , Ph], [RA3243; H, H, Et, Cl, c-PrCH ₂ , Bn], [RA3244; H, H, Et, Cl, c-PrCH ₂ , CF ₃ ], [RA3245; H, H, Et, Cl, c-PrCH ₂ , CF ₃ CH ₂ ], [RA3246; H, H, Et, Cl, c-PrCH ₂ , CF ₃ CF ₂ ], [RA3247; H, H, Et, Cl, c-PrCH ₂ , CF ₂ H], [RA3248; H, H, Et, Cl, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA3249; H, H, F, H, c-PrCH ₂ , Me], [RA3250; H, H, F, H, c-PrCH ₂ , Et], [RA3251; H, H, F, H, c-PrCH ₂ , Pr], [RA3252; H, H, F, H, c-PrCH ₂ , i -Pr], [RA3253; H, H, F, H, c-PrCH ₂ , c-Pr], [RA3254; H, H, F, H, c-PrCH ₂ , Bu], [RA3255; H, H , F, H, c-PrCH ₂ , i-Bu], [RA3256; H, H, F, H, c-PrCH ₂ , t-Bu], [RA3257; H, H, F, H, c-PrCH ₂ , c-PrCH ₂ ], [RA3258; H, H, F, H, c-PrCH ₂ , Ph], [RA3259; H, H, F, H, c-PrCH ₂ , Bn], [RA3260; H , H, F, H, c-PrCH ₂ , CF ₃ ], [RA3261; H, H, F, H, c-PrCH ₂ , CF ₃ CH ₂ ], [RA3262; H, H, F, H, c- PrCH ₂ , CF ₃ CF ₂ ], [RA3263; H, H, F, H, c-PrCH ₂ , CF ₂ H], [RA3264; H, H, F, H, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA3265; H, H, F, F, c-PrCH ₂ , Me], [RA3266; H, H, F, F, c-PrCH ₂ , Et], [RA3267; H, H, F, F , c-PrCH ₂ , Pr], [RA3268; H, H, F, F, c-PrCH ₂ , i-Pr], [RA3269; H, H, F, F, c-PrCH ₂ , c-Pr] , [RA3270; H, H, F, F, c-PrCH ₂ , Bu], [RA3271; H, H, F, F, c-PrCH ₂ , i-Bu], [RA3272; H, H, F, F, c-PrCH ₂ , t-Bu], [RA3273; H, H, F, F, c-PrCH ₂ , c-PrCH ₂ ], [RA3274; H, H, F, F, c-PrCH ₂ , Ph], [RA3275; H, H, F, F, c-PrCH ₂ , Bn], [RA3276; H, H, F, F, c-PrCH ₂ , CF ₃ ], [RA3277; H, H, F , F, c-PrCH ₂ , CF ₃ CH ₂ ], [RA3278; H, H, F, F, c-PrCH ₂ , CF ₃ CF ₂ ], [RA3279; H, H, F, F, c-PrCH ₂ , CF ₂ H], [RA3280; H, H, F, F, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA3281; H, H, F, Cl, c-PrCH ₂ , Me], [RA3282 ; H, H, F, Cl, c-PrCH ₂ , Et], [RA3283; H, H, F, Cl, c-PrCH ₂ , Pr], [RA3284; H, H, F, Cl, c-PrCH _{2, i-Pr], [} RA3285; H, H, F, Cl, c-PrCH 2, c-Pr], [RA3286; H, H, F, Cl, c-PrCH 2, Bu], [RA3287; H, H, F, Cl, c-PrCH ₂ , i-Bu], [RA3288; H, H, F, Cl, c-PrCH ₂ , t-Bu], [RA3289; H, H, F, Cl, c-PrCH ₂ , c-PrCH ₂ ], [RA3290 ; H, H, F, Cl, c-PrCH ₂ , Ph], [RA3291; H, H, F, Cl, c-PrCH ₂ , Bn], [RA3292; H, H, F, Cl, c-PrCH ₂ , CF ₃ ], [RA3293; H, H, F, Cl, c-PrCH ₂ , CF ₃ CH ₂ ], [RA3294; H, H, F, Cl, c-PrCH ₂ , CF ₃ CF ₂ ], [RA3295; H, H, F, Cl, c-PrCH ₂ , CF ₂ H], [RA3296; H, H, F, Cl, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA3297; H, H, Cl, H, c-PrCH ₂ , Me], [RA3298; H, H, Cl, H, c-PrCH ₂ , Et], [RA3299; H, H, Cl, H, c-PrCH ₂ , Pr], [RA3300; H, H, Cl, H, c-PrCH ₂ , i-Pr], [RA3301; H, H, Cl, H, c-PrCH ₂ , c-Pr], [RA3302; H, H, Cl , H, c-PrCH ₂ , Bu], [RA3303; H, H, Cl, H, c-PrCH ₂ , i-Bu], [RA3304; H, H, Cl, H, c-PrCH ₂ , t- Bu], [RA3305; H, H, Cl, H, c-PrCH ₂ , c-PrCH ₂ ], [RA3306; H, H, Cl, H, c-PrCH ₂ , Ph], [RA3307; H, H , Cl, H, c-PrCH ₂ , Bn], [RA3308; H, H, Cl, H, c-PrCH ₂ , CF ₃ ], [RA3309; H, H, Cl, H, c-PrCH ₂ , CF ₃ CH ₂ ], [RA3310; H, H, Cl, H, c-PrCH ₂ , CF ₃ CF ₂ ], [RA3311; H, H, Cl, H, c-PrCH ₂ , CF ₂ H], [RA3312 ; H, H, Cl, H, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA3313; H, H, Cl, Cl, c-PrCH ₂ , Me], [RA3314; H, H, Cl, Cl, c-PrCH ₂ , Et], [RA3315; H, H, Cl, Cl, c-PrCH ₂ , Pr], [RA3316; H, H, Cl, Cl, c-PrCH ₂ , i-Pr], [RA3317 ; H, H, Cl, Cl, c-PrCH ₂ , c-Pr], [RA3318; H, H, Cl, Cl, c-PrCH ₂ , Bu], [RA3319; H, H, Cl, Cl, c -PrCH ₂ , i-Bu], [RA3320; H, H, Cl, Cl, c-PrCH ₂ , t-Bu], [RA3321; H, H, Cl, Cl, c-PrCH ₂ , c-PrCH ₂ ], [RA3322; H, H, Cl, Cl, c-PrCH ₂ , Ph], [RA3323; H, H, Cl, Cl, c-PrCH ₂ , Bn], [RA3324; H, H, Cl, Cl , c-PrCH ₂ , CF ₃ ], [RA3325; H, H, Cl, Cl, c-PrCH ₂ , CF ₃ CH ₂ ], [RA3326; H, H, Cl, Cl, c-PrCH ₂ , CF ₃ CF ₂ ], [RA3327; H, H, Cl, Cl, c-PrCH ₂ , CF ₂ H], [RA3328; H, H, Cl, Cl, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA3329; H, H, Me, H, Bn, Me], [RA3330; H, H, Me, H, Bn, Et], [RA3331; H, H, Me, H, Bn, Pr], [RA3332; H, H, Me, H, Bn, i-Pr], [RA3333; H, H, Me, H, Bn, c-Pr], [RA3334; H, H, Me, H, Bn, Bu], [RA3335; H, H, Me, H, Bn, i-Bu], [RA3336; H, H, Me, H, Bn, t-Bu], [RA3337; H, H, Me, H, Bn, c-PrCH ₂ ], [RA3338; H, H, Me, H, Bn, Ph], [RA3339; H, H, Me, H, Bn, Bn], [RA3340; H, H, Me, H, Bn, CF ₃ ] , [RA3341; H, H, Me, H, Bn, CF ₃ CH ₂ ], [RA3342; H, H, Me, H, Bn, CF ₃ CF ₂ ], [RA3343; H, H, Me, H, Bn, CF ₂ H], [RA3344; H, H, Me, H, Bn, CF ₂ HCH ₂ ], [RA3345; H, H, Me, Me, Bn, Me], [RA3346; H, H, Me , Me, Bn, Et], [RA3347; H, H, Me, Me, Bn, Pr], [RA3348; H, H, Me, Me, Bn, i-Pr], [RA3349; H, H, Me , Me, Bn, c-Pr], [RA3350; H, H, Me, Me, Bn, Bu], [RA3351; H, H, Me, Me, Bn, i-Bu], [RA3352; H, H , Me, Me, Bn, t-Bu], [RA3353; H, H, Me, Me , Bn, c-PrCH ₂ ], [RA3354; H, H, Me, Me, Bn, Ph], [RA3355; H, H, Me, Me, Bn, Bn], [RA3356; H, H, Me, Me, Bn, CF ₃ ], [RA3357; H, H, Me, Me, Bn, CF ₃ CH ₂ ], [RA3358; H, H, Me, Me, Bn, CF ₃ CF ₂ ], [RA3359; H , H, Me, Me, Bn, CF ₂ H], [RA3360; H, H, Me, Me, Bn, CF ₂ HCH ₂ ], [RA3361; H, H, Me, Et, Bn, Me], [ RA3362; H, H, Me, Et, Bn, Et], [RA3363; H, H, Me, Et, Bn, Pr], [RA3364; H, H, Me, Et, Bn, i-Pr], [ RA3365; H, H, Me, Et, Bn, c-Pr], [RA3366; H, H, Me, Et, Bn, Bu], [RA3367; H, H, Me, Et, Bn, i-Bu] , [RA3368; H, H, Me, Et, Bn, t-Bu], [RA3369; H, H, Me, Et, Bn, c-PrCH ₂ ], [RA3370; H, H, Me, Et, Bn , Ph], [RA3371; H, H, Me, Et, Bn, Bn], [RA3372; H, H, Me, Et, Bn, CF ₃ ], [RA3373; H, H, Me, Et, Bn, CF ₃ CH ₂ ], [RA3374; H, H, Me, Et, Bn, CF ₃ CF ₂ ], [RA3375; H, H, Me, Et, Bn, CF ₂ H], [RA3376; H, H, Me, Et, Bn, CF ₂ HCH ₂ ], [RA3377; H, H, Me, F, Bn, Me], [RA3378; H, H, Me, F, Bn, Et], [RA3379; H, H , Me, F, Bn, Pr], [RA3380; H, H, Me, F, Bn, i-Pr], [RA3381; H, H, Me, F, Bn, c-Pr], [RA3382; H , H, Me, F, Bn, Bu], [RA3383; H, H, Me, F, Bn, i-Bu], [RA3384; H, H, Me, F, Bn, t-Bu], [RA3385 ; H, H, Me, F, Bn, c-PrCH ₂ ], [RA3386; H, H, Me, F, Bn, Ph], [RA3387; H, H, Me, F, Bn, Bn], [ RA3388; H, H, Me, F, Bn, CF ₃ ], [RA3389; H, H, Me, F, Bn, CF ₃ CH ₂ ], [RA3390; H, H, Me, F, Bn, CF ₃ CF ₂ ], [RA3391; H, H, Me, F, Bn, CF ₂ H], [RA3392; H, H, Me, F, Bn, CF ₂ HCH ₂ ], [RA3393; H, H, Me, Cl, Bn, Me], [RA3394; H, H, Me, Cl, Bn, Et], [RA3395; H, H, Me , Cl, Bn, Pr], [RA3396; H, H, Me, Cl, Bn, i-Pr], [RA3397; H, H, Me, Cl, Bn, c-Pr], [RA3398; H, H , Me, Cl, Bn, Bu], [RA3399; H, H, Me, Cl, Bn, i-Bu], [RA3400; H, H, Me, Cl, Bn, t-Bu],

[RA3401; H, H, Me, Cl, Bn, c-PrCH ₂ ], [RA3402; H, H, Me, Cl, Bn, Ph], [RA3403; H, H, Me, Cl, Bn, Bn] , [RA3404; H, H, Me, Cl, Bn, CF ₃ ], [RA3405; H, H, Me, Cl, Bn, CF ₃ CH ₂ ], [RA3406; H, H, Me, Cl, Bn, CF ₃ CF ₂ ], [RA3407; H, H, Me, Cl, Bn, CF ₂ H], [RA3408; H, H, Me, Cl, Bn, CF ₂ HCH ₂ ], [RA3409; H, H, Et, H, Bn, Me], [RA3410; H, H, Et, H, Bn, Et], [RA3411; H, H, Et, H, Bn, Pr], [RA3412; H, H, Et, H, Bn, i-Pr], [RA3413; H, H, Et, H, Bn, c-Pr], [RA3414; H, H, Et, H, Bn, Bu], [RA3415; H, H, Et, H, Bn, i-Bu], [RA3416; H, H, Et, H, Bn, t-Bu], [RA3417; H, H, Et, H, Bn, c-PrCH ₂ ], [RA3418 ; H, H, Et, H, Bn, Ph], [RA3419; H, H, Et, H, Bn, Bn], [RA3420; H, H, Et, H, Bn, CF ₃ ], [RA3421; H, H, Et, H, Bn, CF ₃ CH ₂ ], [RA3422; H, H, Et, H, Bn, CF ₃ CF ₂ ], [RA3423; H, H, Et, H, Bn, CF ₂ H], [RA3424; H, H, Et, H, Bn, CF ₂ HCH ₂ ], [RA3425; H, H, Et, F, Bn, Me], [RA3426; H, H, Et, F, Bn , Et], [RA3427; H, H, Et, F, Bn, Pr], [RA3428; H, H, Et, F, Bn, i-Pr], [RA3429; H, H, Et, F, Bn , c-Pr], [RA3430; H, H, Et, F, Bn, Bu], [RA3431; H, H, Et, F, Bn, i-Bu], [RA3432; H, H, Et, F , Bn, t-Bu], [RA3433; H, H, Et, F, Bn, c-PrCH ₂ ], [RA3434; H, H, Et, F, Bn, Ph], [RA3435; H, H, Et, F, Bn, Bn], [RA3436; H, H, Et, F, Bn, CF ₃ ], [RA3437; H, H, Et, F, Bn, CF ₃ CH ₂ ], [RA3438; H, H, Et, F, Bn, CF ₃ CF ₂ ], [RA3439; H, H, Et, F, Bn, CF ₂ H], [RA3440; H, H, Et, F, Bn, CF ₂ HCH ₂ ], [RA3441; H, H, Et, Cl, Bn, Me], [RA3442; H, H, Et, Cl, Bn, Et], [RA3443; H, H, Et , Cl, Bn, Pr], [RA3444; H, H, Et, Cl, Bn, i-Pr], [RA3445; H, H, Et, Cl, Bn, c-Pr], [RA3446; H, H , Et, Cl, Bn, Bu], [RA3447; H, H, Et, Cl, Bn, i-Bu], [RA3448; H, H, Et, Cl, Bn, t-Bu], [RA3449; H , H, Et, Cl, Bn, c-PrCH ₂ ], [RA3450; H, H, Et, Cl, Bn, Ph], [RA3451; H, H, Et, Cl, Bn, Bn], [RA3452; H, H, Et, Cl, Bn, CF ₃ ], [RA3453; H, H, Et, Cl, Bn, CF ₃ CH ₂ ], [RA3454; H, H, Et, Cl, Bn, CF ₃ CF ₂ ], [RA3455; H, H, Et, Cl, Bn, CF ₂ H], [RA3456; H, H, Et, Cl, Bn, CF ₂ HCH ₂ ], [RA3457; H, H, F, H, Bn, Me], [RA3458; H, H, F, H, Bn, Et], [RA3459; H, H, F, H, Bn, Pr], [RA3460; H, H, F, H, Bn, i-Pr], [RA3461; H, H, F, H, Bn, c-Pr], [RA3462; H, H, F, H, Bn, Bu], [RA3463; H, H, F, H, Bn, i-Bu], [RA3464; H, H, F, H, Bn, t-Bu], [RA3465; H, H, F, H, Bn, c-PrCH ₂ ], [RA3466; H, H , F, H, Bn, Ph], [RA3467; H, H, F, H, Bn, Bn], [RA3468; H, H, F, H, Bn, CF ₃ ], [RA3469; H, H, F, H, Bn, CF ₃ CH ₂ ], [RA3470; H, H, F, H, Bn, CF ₃ CF ₂ ], [RA3471; H, H, F, H, Bn, CF ₂ H], [ RA3472; H, H, F, H, Bn, CF ₂ HCH ₂ ], [RA3473; H, H, F, F, Bn, Me], [RA3474; H, H, F, F, Bn, Et], [RA3475; H, H, F, F, Bn, Pr], [RA3476; H, H, F, F, Bn, i-Pr], [RA3477; H, H, F, F, Bn, c-Pr], [RA3478; H, H, F, F, Bn, Bu], [RA3479; H, H, F, F, Bn, i-Bu], [RA3480; H, H, F, F, Bn, t-Bu], [RA3481; H, H, F, F, Bn, c-PrCH ₂ ], [RA3482; H, H, F, F, Bn, Ph], [RA3483; H , H, F, F, Bn, Bn], [RA3484; H, H, F, F, Bn, CF ₃ ], [RA3485; H, H, F, F, Bn, CF ₃ CH ₂ ], [RA3486 ; H, H, F, F, Bn, CF ₃ CF ₂ ], [RA3487; H, H, F, F, Bn, CF ₂ H], [RA3488; H, H, F, F, Bn, CF ₂ HCH ₂ ], [RA3489; H, H, F, Cl, Bn, Me], [RA3490; H, H, F, Cl, Bn, Et], [RA3491; H, H, F, Cl, Bn, Pr ], [RA3492; H, H, F, Cl, Bn, i-Pr], [RA3493; H, H, F, Cl, Bn, c-Pr], [RA3494; H, H, F, Cl, Bn , Bu], [RA3495; H, H, F, Cl, Bn, i-Bu], [RA3496; H, H, F, Cl, Bn, t-Bu], [RA3497; H, H, F, Cl , Bn, c-PrCH ₂ ], [RA3498; H, H, F, Cl, Bn, Ph], [RA3499; H, H, F, Cl, Bn, Bn], [RA3500; H, H, F, Cl, Bn, CF ₃ ], [RA3501; H, H, F, Cl, Bn, CF ₃ CH ₂ ], [RA3502; H, H, F, Cl, Bn, CF ₃ CF ₂ ], [RA3503; H , H, F, Cl, Bn, CF ₂ H], [RA3504; H, H, F, Cl, Bn, CF ₂ HCH ₂ ], [RA3505; H, H, Cl, H, Bn, Me], [ RA3506; H, H, Cl, H, Bn, Et], [RA3507; H, H, Cl, H, Bn, Pr], [RA3508; H, H, Cl, H, Bn, i-Pr], [ RA3509; H, H, Cl, H, Bn, c-Pr], [RA3510; H, H, Cl, H, Bn, Bu], [RA3511; H, H, Cl, H, Bn, i-Bu] , [RA3512; H, H, Cl, H, Bn, t-Bu], [RA3513; H, H, Cl, H, Bn, c-PrCH ₂ ], [RA3514; H, H, Cl, H, Bn, Ph], [RA3515; H, H, Cl , H, Bn, Bn], [RA3516; H, H, Cl, H, Bn, CF ₃ ], [RA3517; H, H, Cl, H, Bn, CF ₃ CH ₂ ], [RA3518; H, H , Cl, H, Bn, CF ₃ CF ₂ ], [RA3519; H, H, Cl, H, Bn, CF ₂ H], [RA3520; H, H, Cl, H, Bn, CF ₂ HCH ₂ ], [RA3521; H, H, Cl, Cl, Bn, Me], [RA3522; H, H, Cl, Cl, Bn, Et], [RA3523; H, H, Cl, Cl, Bn, Pr], [RA3524 ; H, H, Cl, Cl, Bn, i-Pr], [RA3525; H, H, Cl, Cl, Bn, c-Pr], [RA3526; H, H, Cl, Cl, Bn, Bu], [RA3527; H, H, Cl, Cl, Bn, i-Bu], [RA3528; H, H, Cl, Cl, Bn, t-Bu], [RA3529; H, H, Cl, Cl, Bn, c -PrCH ₂ ], [RA3530; H, H, Cl, Cl, Bn, Ph], [RA3531; H, H, Cl, Cl, Bn, Bn], [RA3532; H, H, Cl, Cl, Bn, CF ₃ ], [RA3533; H, H, Cl, Cl, Bn, CF ₃ CH ₂ ], [RA3534; H, H, Cl, Cl, Bn, CF ₃ CF ₂ ], [RA3535; H, H, Cl , Cl, Bn, CF ₂ H], [RA3536; H, H, Cl, Cl, Bn, CF ₂ HCH ₂ ], [RA3537; H, H, Me, H, Ph, Me], [RA3538; H, H, Me, H, Ph, Et], [RA3539; H, H, Me, H, Ph, Pr], [RA3540; H, H, Me, H, Ph, i-Pr], [RA3541; H, H, Me, H, Ph, c-Pr], [RA3542; H, H, Me, H, Ph, Bu], [RA3543; H, H, Me, H, Ph, i-Bu], [RA3544; H, H, Me, H, Ph, t-Bu], [RA3545; H, H, Me, H, Ph, c-PrCH ₂ ], [RA3546; H, H, Me, H, Ph, Ph], [RA3547; H, H, Me, H, Ph, Bn], [RA3548; H, H, Me, H, Ph, CF ₃ ], [RA3549 ; H, H, Me, H, Ph, CF ₃ CH ₂ ], [RA3550; H, H, Me, H, Ph, CF ₃ CF ₂ ], [RA3551; H, H, Me, H, Ph, CF ₂ H], [RA3552; H, H, Me, H, Ph, CF ₂ HCH ₂ ], [RA3553; H, H, Me, Me, Ph, Me], [RA3554; H, H, Me, Me, Ph, Et], [RA3555; H, H, Me, Me, Ph, Pr], [RA3556; H, H, Me, Me, Ph, i-Pr], [RA3557; H, H, Me, Me, Ph, c-Pr], [RA3558; H, H, Me, Me, Ph, Bu], [RA3559; H, H, Me, Me, Ph, i-Bu], [RA3560; H, H, Me, Me, Ph, t-Bu], [RA3561; H, H, Me, Me, Ph, c-PrCH ₂ ], [RA3562; H, H, Me, Me, Ph, Ph], [RA3563; H, H , Me, Me, Ph, Bn], [RA3564; H, H, Me, Me, Ph, CF ₃ ], [RA3565; H, H, Me, Me, Ph, CF ₃ CH ₂ ], [RA3566; H , H, Me, Me, Ph, CF ₃ CF ₂ ], [RA3567; H, H, Me, Me, Ph, CF ₂ H], [RA3568; H, H, Me, Me, Ph, CF ₂ HCH ₂ ], [RA3569; H, H, Me, Et, Ph, Me], [RA3570; H, H, Me, Et, Ph, Et], [RA3571; H, H, Me, Et, Ph, Pr], [RA3572; H, H, Me, Et, Ph, i-Pr], [RA3573; H, H, Me, Et, Ph, c-Pr], [RA3574; H, H, Me, Et, Ph, Bu ], [RA3575; H, H, Me, Et, Ph, i-Bu], [RA3576; H, H, Me, Et, Ph, t-Bu], [RA3577; H, H, Me, Et, Ph , c-PrCH ₂ ], [RA3578; H, H, Me, Et, Ph, Ph], [RA3579; H, H, Me, Et, Ph, Bn], [RA3580; H, H, Me, Et, Ph, CF ₃ ], [RA3581; H, H, Me, Et, Ph, CF ₃ CH ₂ ], [RA3582; H, H, Me, Et, Ph, CF ₃ CF ₂ ], [RA3583; H, H , Me, Et, Ph, CF ₂ H], [RA3584; H, H, Me, Et, Ph, C F ₂ HCH ₂ ], [RA3585; H, H, Me, F, Ph, Me], [RA3586; H, H, Me, F, Ph, Et], [RA3587; H, H, Me, F, Ph , Pr], [RA3588; H, H, Me, F, Ph, i-Pr], [RA3589; H, H, Me, F, Ph, c-Pr], [RA3590; H, H, Me, F , Ph, Bu], [RA3591; H, H, Me, F, Ph, i-Bu], [RA3592; H, H, Me, F, Ph, t-Bu], [RA3593; H, H, Me , F, Ph, c-PrCH ₂ ], [RA3594; H, H, Me, F, Ph, Ph], [RA3595; H, H, Me, F, Ph, Bn], [RA3596; H, H, Me, F, Ph, CF ₃ ], [RA3597; H, H, Me, F, Ph, CF ₃ CH ₂ ], [RA3598; H, H, Me, F, Ph, CF ₃ CF ₂ ], [RA3599 ; H, H, Me, F, Ph, CF ₂ H], [RA3600; H, H, Me, F, Ph, CF ₂ HCH ₂ ],

[RA3601; H, H, Me, Cl, Ph, Me], [RA3602; H, H, Me, Cl, Ph, Et], [RA3603; H, H, Me, Cl, Ph, Pr], [RA3604 ; H, H, Me, Cl, Ph, i-Pr], [RA3605; H, H, Me, Cl, Ph, c-Pr], [RA3606; H, H, Me, Cl, Ph, Bu], [RA3607; H, H, Me, Cl, Ph, i-Bu], [RA3608; H, H, Me, Cl, Ph, t-Bu], [RA3609; H, H, Me, Cl, Ph, c -PrCH ₂ ], [RA3610; H, H, Me, Cl, Ph, Ph], [RA3611; H, H, Me, Cl, Ph, Bn], [RA3612; H, H, Me, Cl, Ph, CF ₃ ], [RA3613; H, H, Me, Cl, Ph, CF ₃ CH ₂ ], [RA3614; H, H, Me, Cl, Ph, CF ₃ CF ₂ ], [RA3615; H, H, Me , Cl, Ph, CF ₂ H], [RA3616; H, H, Me, Cl, Ph, CF ₂ HCH ₂ ], [RA3617; H, H, Et, H, Ph, Me], [RA3618; H, H, Et, H, Ph, Et], [RA3619; H, H, Et, H, Ph, Pr], [RA3620; H, H, Et, H, Ph, i-Pr], [RA3621; H, H, Et, H, Ph, c-Pr], [RA3622; H, H, Et, H, Ph, Bu], [RA3623; H, H, Et, H, Ph, i-Bu], [RA3624; H, H, Et, H, Ph, t-Bu], [RA3625; H, H, Et, H, Ph, c-PrCH ₂ ], [RA3626; H, H, Et, H, Ph, Ph], [RA3627; H, H, Et, H, Ph, Bn], [RA3628; H, H, Et, H, Ph, CF ₃ ], [RA3629; H, H, Et, H, Ph, CF ₃ CH ₂ ], [RA3630; H, H, Et, H, Ph, CF ₃ CF ₂ ], [RA3631; H, H, Et, H, Ph, CF ₂ H], [RA3632; H, H, Et, H, Ph, CF ₂ HCH ₂ ], [RA3633; H, H, Et, F, Ph, Me], [RA3634; H, H, Et, F, Ph, Et], [RA3635; H, H, Et, F , Ph, Pr], [RA3636; H, H, Et, F, Ph, i-Pr], [RA3637; H, H, Et, F, Ph, c-Pr ], [RA3638; H, H, Et, F, Ph, Bu], [RA3639; H, H, Et, F, Ph, i-Bu], [RA3640; H, H, Et, F, Ph, t -Bu], [RA3641; H, H, Et, F, Ph, c-PrCH ₂ ], [RA3642; H, H, Et, F, Ph, Ph], [RA3643; H, H, Et, F, Ph, Bn], [RA3644; H, H, Et, F, Ph, CF ₃ ], [RA3645; H, H, Et, F, Ph, CF ₃ CH ₂ ], [RA3646; H, H, Et, F, Ph, CF ₃ CF ₂ ], [RA3647; H, H, Et, F, Ph, CF ₂ H], [RA3648; H, H, Et, F, Ph, CF ₂ HCH ₂ ], [RA3649; H, H, Et, Cl, Ph, Me], [RA3650; H, H, Et, Cl, Ph, Et], [RA3651; H, H, Et, Cl, Ph, Pr], [RA3652; H, H, Et, Cl, Ph, i-Pr], [RA3653; H, H, Et, Cl, Ph, c-Pr], [RA3654; H, H, Et, Cl, Ph, Bu], [RA3655; H, H, Et, Cl, Ph, i-Bu], [RA3656; H, H, Et, Cl, Ph, t-Bu], [RA3657; H, H, Et, Cl, Ph, c-PrCH ₂ ], [RA3658; H, H, Et, Cl, Ph, Ph], [RA3659; H, H, Et, Cl, Ph, Bn], [RA3660; H, H, Et, Cl, Ph, CF ₃ ] , [RA3661; H, H, Et, Cl, Ph, CF ₃ CH ₂ ], [RA3662; H, H, Et, Cl, Ph, CF ₃ CF ₂ ], [RA3663; H, H, Et, Cl, Ph, CF ₂ H], [RA3664; H, H, Et, Cl, Ph, CF ₂ HCH ₂ ], [RA3665; H, H, F, H, Ph, Me], [RA3666; H, H, F , H, Ph, Et], [RA3667; H, H, F, H, Ph, Pr], [RA3668; H, H, F, H, Ph, i-Pr], [RA3669; H, H, F , H, Ph, c-Pr], [RA3670; H, H, F, H, Ph, Bu], [RA3671; H, H, F, H, Ph, i-Bu], [RA3672; H, H , F, H, Ph, t-Bu], [RA3673; H, H, F, H, Ph, c-PrCH ₂ ], [RA3674; H, H, F, H, Ph, Ph] , [RA3675; H, H, F, H, Ph, Bn], [RA3676; H, H, F, H, Ph, CF ₃ ], [RA3677; H, H, F, H, Ph, CF ₃ CH ₂ ], [RA3678; H, H, F, H, Ph, CF ₃ CF ₂ ], [RA3679; H, H, F, H, Ph, CF ₂ H], [RA3680; H, H, F, H , Ph, CF ₂ HCH ₂ ], [RA3681; H, H, F, F, Ph, Me], [RA3682; H, H, F, F, Ph, Et], [RA3683; H, H, F, F, Ph, Pr], [RA3684; H, H, F, F, Ph, i-Pr], [RA3685; H, H, F, F, Ph, c-Pr], [RA3686; H, H, F, F, Ph, Bu], [RA3687; H, H, F, F, Ph, i-Bu], [RA3688; H, H, F, F, Ph, t-Bu], [RA3689; H, H, F, F, Ph, c-PrCH ₂ ], [RA3690; H, H, F, F, Ph, Ph], [RA3691; H, H, F, F, Ph, Bn], [RA3692; H , H, F, F, Ph, CF ₃ ], [RA3693; H, H, F, F, Ph, CF ₃ CH ₂ ], [RA3694; H, H, F, F, Ph, CF ₃ CF ₂ ] , [RA3695; H, H, F, F, Ph, CF ₂ H], [RA3696; H, H, F, F, Ph, CF ₂ HCH ₂ ], [RA3697; H, H, F, Cl, Ph , Me], [RA3698; H, H, F, Cl, Ph, Et], [RA3699; H, H, F, Cl, Ph, Pr], [RA3700; H, H, F, Cl, Ph, i -Pr], [RA3701; H, H, F, Cl, Ph, c-Pr], [RA3702; H, H, F, Cl, Ph, Bu], [RA3703; H, H, F, Cl, Ph , i-Bu], [RA3704; H, H, F, Cl, Ph, t-Bu], [RA3705; H, H, F, Cl, Ph, c-PrCH ₂ ], [RA3706; H, H, F, Cl, Ph, Ph], [RA3707; H, H, F, Cl, Ph, Bn], [RA3708; H, H, F, Cl, Ph, CF ₃ ], [RA3709; H, H, F , Cl, Ph, CF ₃ CH ₂ ], [RA3710; H, H, F, Cl, Ph, CF ₃ CF ₂ ], [RA3711; H, H, F, Cl, Ph, CF ₂ H], [RA3712 ; H, H, F, Cl , Ph, CF ₂ HCH ₂ ], [RA3713; H, H, Cl, H, Ph, Me], [RA3714; H, H, Cl, H, Ph, Et], [RA3715; H, H, Cl, H, Ph, Pr], [RA3716; H, H, Cl, H, Ph, i-Pr], [RA3717; H, H, Cl, H, Ph, c-Pr], [RA3718; H, H, Cl, H, Ph, Bu], [RA3719; H, H, Cl, H, Ph, i-Bu], [RA3720; H, H, Cl, H, Ph, t-Bu], [RA3721; H, H, Cl, H, Ph, c-PrCH ₂ ], [RA3722; H, H, Cl, H, Ph, Ph], [RA3723; H, H, Cl, H, Ph, Bn], [RA3724; H , H, Cl, H, Ph, CF ₃ ], [RA3725; H, H, Cl, H, Ph, CF ₃ CH ₂ ], [RA3726; H, H, Cl, H, Ph, CF ₃ CF ₂ ] , [RA3727; H, H, Cl, H, Ph, CF ₂ H], [RA3728; H, H, Cl, H, Ph, CF ₂ HCH ₂ ], [RA3729; H, H, Cl, Cl, Ph , Me], [RA3730; H, H, Cl, Cl, Ph, Et], [RA3731; H, H, Cl, Cl, Ph, Pr], [RA3732; H, H, Cl, Cl, Ph, i -Pr], [RA3733; H, H, Cl, Cl, Ph, c-Pr], [RA3734; H, H, Cl, Cl, Ph, Bu], [RA3735; H, H, Cl, Cl, Ph , i-Bu], [RA3736; H, H, Cl, Cl, Ph, t-Bu], [RA3737; H, H, Cl, Cl, Ph, c-PrCH ₂ ], [RA3738; H, H, Cl, Cl, Ph, Ph], [RA3739; H, H, Cl, Cl, Ph, Bn], [RA3740; H, H, Cl, Cl, Ph, CF ₃ ], [RA3741; H, H, Cl , Cl, Ph, CF ₃ CH ₂ ], [RA3742; H, H, Cl, Cl, Ph, CF ₃ CF ₂ ], [RA3743; H, H, Cl, Cl, Ph, CF ₂ H], [RA3744 ; H, H, Cl, Cl, Ph, CF ₂ HCH ₂ ], [RA3745; F, H, Me, H, H, Me], [RA3746; F, H, Me, H, H, Et], [ RA3747; F, H, Me, H, H, Pr], [RA3748; F, H, Me, H, H, i-Pr], [RA3749; F, H , Me, H, H, c-Pr], [RA3750; F, H, Me, H, H, Bu], [RA3751; F, H, Me, H, H, i-Bu], [RA3752; F , H, Me, H, H, t-Bu], [RA3753; F, H, Me, H, H, c-PrCH ₂ ], [RA3754; F, H, Me, H, H, Ph], [ RA3755; F, H, Me, H, H, Bn], [RA3756; F, H, Me, H, H, CF ₃ ], [RA3757; F, H, Me, H, H, CF ₃ CH ₂ ] , [RA3758; F, H, Me, H, H, CF ₃ CF ₂ ], [RA3759; F, H, Me, H, H, CF ₂ H], [RA3760; F, H, Me, H, H , CF ₂ HCH ₂ ], [RA3761; F, H, Me, Me, H, Me], [RA3762; F, H, Me, Me, H, Et], [RA3763; F, H, Me, Me, H, Pr], [RA3764; F, H, Me, Me, H, i-Pr], [RA3765; F, H, Me, Me, H, c-Pr], [RA3766; F, H, Me, Me, H, Bu], [RA3767; F, H, Me, Me, H, i-Bu], [RA3768; F, H, Me, Me, H, t-Bu], [RA3769; F, H, Me, Me, H, c-PrCH ₂ ], [RA3770; F, H, Me, Me, H, Ph], [RA3771; F, H, Me, Me, H, Bn], [RA3772; F, H , Me, Me, H, CF ₃ ], [RA3773; F, H, Me, Me, H, CF ₃ CH ₂ ], [RA3774; F, H, Me, Me, H, CF ₃ CF ₂ ], [ RA3775; F, H, Me, Me, H, CF ₂ H], [RA3776; F, H, Me, Me, H, CF ₂ HCH ₂ ], [RA3777; F, H, Me, Et, H, Me ], [RA3778; F, H, Me, Et, H, Et], [RA3779; F, H, Me, Et, H, Pr], [RA3780; F, H, Me, Et, H, i-Pr ], [RA3781; F, H, Me, Et, H, c-Pr], [RA3782; F, H, Me, Et, H, Bu], [RA3783; F, H, Me, Et, H, i -Bu], [RA3784; F, H, Me, Et, H, t-Bu], [RA3785; F, H, Me, Et, H, c-PrCH ₂ ], [RA3786; F, H, Me, Et, H, Ph], [RA3 787; F, H, Me, Et, H, Bn], [RA3788; F, H, Me, Et, H, CF ₃ ], [RA3789; F, H, Me, Et, H, CF ₃ CH ₂ ] , [RA3790; F, H, Me, Et, H, CF ₃ CF ₂ ], [RA3791; F, H, Me, Et, H, CF ₂ H], [RA3792; F, H, Me, Et, H , CF ₂ HCH ₂ ], [RA3793; F, H, Me, F, H, Me], [RA3794; F, H, Me, F, H, Et], [RA3795; F, H, Me, F, H, Pr], [RA3796; F, H, Me, F, H, i-Pr], [RA3797; F, H, Me, F, H, c-Pr], [RA3798; F, H, Me, F, H, Bu], [RA3799; F, H, Me, F, H, i-Bu], [RA3800; F, H, Me, F, H, t-Bu],

[RA3801; F, H, Me, F, H, c-PrCH ₂ ], [RA3802; F, H, Me, F, H, Ph], [RA3803; F, H, Me, F, H, Bn] , [RA3804; F, H, Me, F, H, CF ₃ ], [RA3805; F, H, Me, F, H, CF ₃ CH ₂ ], [RA3806; F, H, Me, F, H, CF ₃ CF ₂ ], [RA3807; F, H, Me, F, H, CF ₂ H], [RA3808; F, H, Me, F, H, CF ₂ HCH ₂ ], [RA3809; F, H, Me, Cl, H, Me], [RA3810; F, H, Me, Cl, H, Et], [RA3811; F, H, Me, Cl, H, Pr], [RA3812; F, H, Me, Cl, H, i-Pr], [RA3813; F, H, Me, Cl, H, c-Pr], [RA3814; F, H, Me, Cl, H, Bu], [RA3815; F, H, Me, Cl, H, i-Bu], [RA3816; F, H, Me, Cl, H, t-Bu], [RA3817; F, H, Me, Cl, H, c-PrCH ₂ ], [RA3818 ; F, H, Me, Cl, H, Ph], [RA3819; F, H, Me, Cl, H, Bn], [RA3820; F, H, Me, Cl, H, CF ₃ ], [RA3821; F, H, Me, Cl, H, CF ₃ CH ₂ ], [RA3822; F, H, Me, Cl, H, CF ₃ CF ₂ ], [RA3823; F, H, Me, Cl, H, CF ₂ H], [RA3824; F, H, Me, Cl, H, CF ₂ HCH ₂ ], [RA3825; F, H, Et, H, H, Me], [RA3826; F, H, Et, H, H , Et], [RA3827; F, H, Et, H, H, Pr], [RA3828; F, H, Et, H, H, i-Pr], [RA3829; F, H, Et, H, H , c-Pr], [RA3830; F, H, Et, H, H, Bu], [RA3831; F, H, Et, H, H, i-Bu], [RA3832; F, H, Et, H , H, t-Bu], [RA3833; F, H, Et, H, H, c-PrCH ₂ ], [RA3834; F, H, Et, H, H, Ph], [RA3835; F, H, Et, H, H, Bn], [RA3836; F, H, Et, H, H, CF ₃ ], [RA3837; F, H, Et, H, H, CF ₃ CH ₂ ], [RA3838; F, H, Et, H, H, CF ₃ CF ₂ ], [RA3839; F, H, Et, H, H, CF ₂ H], [RA3840; F, H, Et, H, H, CF ₂ HCH ₂ ], [RA3841; F, H, Et , F, H, Me], [RA3842; F, H, Et, F, H, Et], [RA3843; F, H, Et, F, H, Pr], [RA3844; F, H, Et, F , H, i-Pr], [RA3845; F, H, Et, F, H, c-Pr], [RA3846; F, H, Et, F, H, Bu], [RA3847; F, H, Et , F, H, i-Bu], [RA3848; F, H, Et, F, H, t-Bu], [RA3849; F, H, Et, F, H, c-PrCH ₂ ], [RA3850; F, H, Et, F, H, Ph], [RA3851; F, H, Et, F, H, Bn], [RA3852; F, H, Et, F, H, CF ₃ ], [RA3853; F , H, Et, F, H, CF ₃ CH ₂ ], [RA3854; F, H, Et, F, H, CF ₃ CF ₂ ], [RA3855; F, H, Et, F, H, CF ₂ H ], [RA3856; F, H, Et, F, H, CF ₂ HCH ₂ ], [RA3857; F, H, Et, Cl, H, Me], [RA3858; F, H, Et, Cl, H, Et], [RA3859; F, H, Et, Cl, H, Pr], [RA3860; F, H, Et, Cl, H, i-Pr], [RA3861; F, H, Et, Cl, H, c-Pr], [RA3862; F, H, Et, Cl, H, Bu], [RA3863; F, H, Et, Cl, H, i-Bu], [RA3864; F, H, Et, Cl, H, t-Bu], [RA3865; F, H, Et, Cl, H, c-PrCH ₂ ], [RA3866; F, H, Et, Cl, H, Ph], [RA3867; F, H, Et , Cl, H, Bn], [RA3868; F, H, Et, Cl, H, CF ₃ ], [RA3869; F, H, Et, Cl, H, CF ₃ CH ₂ ], [RA3870; F, H , Et, Cl, H, CF ₃ CF ₂ ], [RA3871; F, H, Et, Cl, H, CF ₂ H], [RA3872; F, H, Et, Cl, H, CF ₂ HCH ₂ ], [RA3873; F, H, F, H, H, Me], [RA3874; F, H, F, H, H, Et], [RA3875; F, H, F, H, H, Pr], [RA3876 ; F, H, F, H, H, i -Pr], [RA3877; F, H, F, H, H, c-Pr], [RA3878; F, H, F, H, H, Bu], [RA3879; F, H, F, H, H , i-Bu], [RA3880; F, H, F, H, H, t-Bu], [RA3881; F, H, F, H, H, c-PrCH ₂ ], [RA3882; F, H, F, H, H, Ph], [RA3883; F, H, F, H, H, Bn], [RA3884; F, H, F, H, H, CF ₃ ], [RA3885; F, H, F , H, H, CF ₃ CH ₂ ], [RA3886; F, H, F, H, H, CF ₃ CF ₂ ], [RA3887; F, H, F, H, H, CF ₂ H], [RA3888 ; F, H, F, H, H, CF ₂ HCH ₂ ], [RA3889; F, H, F, F, H, Me], [RA3890; F, H, F, F, H, Et], [ RA3891; F, H, F, F, H, Pr], [RA3892; F, H, F, F, H, i-Pr], [RA3893; F, H, F, F, H, c-Pr] , [RA3894; F, H, F, F, H, Bu], [RA3895; F, H, F, F, H, i-Bu], [RA3896; F, H, F, F, H, t- Bu], [RA3897; F, H, F, F, H, c-PrCH ₂ ], [RA3898; F, H, F, F, H, Ph], [RA3899; F, H, F, F, H , Bn], [RA3900; F, H, F, F, H, CF ₃ ], [RA3901; F, H, F, F, H, CF ₃ CH ₂ ], [RA3902; F, H, F, F , H, CF ₃ CF ₂ ], [RA3903; F, H, F, F, H, CF ₂ H], [RA3904; F, H, F, F, H, CF ₂ HCH ₂ ], [RA3905; F , H, F, Cl, H, Me], [RA3906; F, H, F, Cl, H, Et], [RA3907; F, H, F, Cl, H, Pr], [RA3908; F, H , F, Cl, H, i-Pr], [RA3909; F, H, F, Cl, H, c-Pr], [RA3910; F, H, F, Cl, H, Bu], [RA3911; F , H, F, Cl, H, i-Bu], [RA3912; F, H, F, Cl, H, t-Bu], [RA3913; F, H, F, Cl, H, c-PrCH ₂ ] , [RA3914; F, H, F, Cl, H, Ph], [RA3915; F, H, F, Cl, H, Bn], [RA3916; F, H, F, Cl, H, CF ₃ ], [RA3917; F, H, F, Cl, H, CF ₃ CH ₂ ], [RA3918; F, H, F, Cl, H, CF ₃ CF ₂ ], [RA3919; F, H, F , Cl, H, CF ₂ H], [RA3920; F, H, F, Cl, H, CF ₂ HCH ₂ ], [RA3921; F, H, Cl, H, H, Me], [RA3922; F, H, Cl, H, H, Et], [RA3923; F, H, Cl, H, H, Pr], [RA3924; F, H, Cl, H, H, i-Pr], [RA3925; F, H, Cl, H, H, c-Pr], [RA3926; F, H, Cl, H, H, Bu], [RA3927; F, H, Cl, H, H, i-Bu], [RA3928; F, H, Cl, H, H, t-Bu], [RA3929; F, H, Cl, H, H, c-PrCH ₂ ], [RA3930; F, H, Cl, H, H, Ph], [RA3931; F, H, Cl, H, H, Bn], [RA3932; F, H, Cl, H, H, CF ₃ ], [RA3933; F, H, Cl, H, H, CF ₃ CH ₂ ], [RA3934; F, H, Cl, H, H, CF ₃ CF ₂ ], [RA3935; F, H, Cl, H, H, CF ₂ H], [RA3936; F, H, Cl, H, H, CF ₂ HCH ₂ ], [RA3937; F, H, Cl, Cl, H, Me], [RA3938; F, H, Cl, Cl, H, Et], [RA3939; F, H, Cl, Cl , H, Pr], [RA3940; F, H, Cl, Cl, H, i-Pr], [RA3941; F, H, Cl, Cl, H, c-Pr], [RA3942; F, H, Cl , Cl, H, Bu], [RA3943; F, H, Cl, Cl, H, i-Bu], [RA3944; F, H, Cl, Cl, H, t-Bu], [RA3945; F, H , Cl, Cl, H, c-PrCH ₂ ], [RA3946; F, H, Cl, Cl, H, Ph], [RA3947; F, H, Cl, Cl, H, Bn], [RA3948; F, H, Cl, Cl, H, CF ₃ ], [RA3949; F, H, Cl, Cl, H, CF ₃ CH ₂ ], [RA3950; F, H, Cl, Cl, H, CF ₃ CF ₂ ], [RA3951; F, H, Cl, Cl, H, CF ₂ H], [RA3952; F, H, Cl, Cl, H, CF ₂ HCH ₂ ], [RA3953; F, H, Me, H, Me, Me], [R A3954; F, H, Me, H, Me, Et], [RA3955; F, H, Me, H, Me, Pr], [RA3956; F, H, Me, H, Me, i-Pr], [ RA3957; F, H, Me, H, Me, c-Pr], [RA3958; F, H, Me, H, Me, Bu], [RA3959; F, H, Me, H, Me, i-Bu] , [RA3960; F, H, Me, H, Me, t-Bu], [RA3961; F, H, Me, H, Me, c-PrCH ₂ ], [RA3962; F, H, Me, H, Me , Ph], [RA3963; F, H, Me, H, Me, Bn], [RA3964; F, H, Me, H, Me, CF ₃ ], [RA3965; F, H, Me, H, Me, CF ₃ CH ₂ ], [RA3966; F, H, Me, H, Me, CF ₃ CF ₂ ], [RA3967; F, H, Me, H, Me, CF ₂ H], [RA3968; F, H, Me, H, Me, CF ₂ HCH ₂ ], [RA3969; F, H, Me, Me, Me, Me], [RA3970; F, H, Me, Me, Me, Et], [RA3971; F, H , Me, Me, Me, Pr], [RA3972; F, H, Me, Me, Me, i-Pr], [RA3973; F, H, Me, Me, Me, c-Pr], [RA3974; F , H, Me, Me, Me, Bu], [RA3975; F, H, Me, Me, Me, i-Bu], [RA3976; F, H, Me, Me, Me, t-Bu], [RA3977 ; F, H, Me, Me, Me, c-PrCH ₂ ], [RA3978; F, H, Me, Me, Me, Ph], [RA3979; F, H, Me, Me, Me, Bn], [ RA3980; F, H, Me, Me, Me, CF ₃ ], [RA3981; F, H, Me, Me, Me, CF ₃ CH ₂ ], [RA3982; F, H, Me, Me, Me, CF ₃ CF ₂ ], [RA3983; F, H, Me, Me, Me, CF ₂ H], [RA3984; F, H, Me, Me, Me, CF ₂ HCH ₂ ], [RA3985; F, H, Me, Et, Me, Me], [RA3986; F, H, Me, Et, Me, Et], [RA3987; F, H, Me, Et, Me, Pr], [RA3988; F, H, Me, Et, Me, i-Pr], [RA3989; F, H, Me, Et, Me, c-Pr], [RA3990; F, H, Me, Et, M e, Bu], [RA3991; F, H, Me, Et, Me, i-Bu], [RA3992; F, H, Me, Et, Me, t-Bu], [RA3993; F, H, Me, Et, Me, c-PrCH ₂ ], [RA3994; F, H, Me, Et, Me, Ph], [RA3995; F, H, Me, Et, Me, Bn], [RA3996; F, H, Me , Et, Me, CF ₃ ], [RA3997; F, H, Me, Et, Me, CF ₃ CH ₂ ], [RA3998; F, H, Me, Et, Me, CF ₃ CF ₂ ], [RA3999; F, H, Me, Et, Me, CF ₂ H], [RA4000; F, H, Me, Et, Me, CF ₂ HCH ₂ ],

[RA4001; F, H, Me, F, Me, Me], [RA4002; F, H, Me, F, Me, Et], [RA4003; F, H, Me, F, Me, Pr], [RA4004 ; F, H, Me, F, Me, i-Pr], [RA4005; F, H, Me, F, Me, c-Pr], [RA4006; F, H, Me, F, Me, Bu], [RA4007; F, H, Me, F, Me, i-Bu], [RA4008; F, H, Me, F, Me, t-Bu], [RA4009; F, H, Me, F, Me, c -PrCH ₂ ], [RA4010; F, H, Me, F, Me, Ph], [RA4011; F, H, Me, F, Me, Bn], [RA4012; F, H, Me, F, Me, CF ₃ ], [RA4013; F, H, Me, F, Me, CF ₃ CH ₂ ], [RA4014; F, H, Me, F, Me, CF ₃ CF ₂ ], [RA4015; F, H, Me , F, Me, CF ₂ H], [RA4016; F, H, Me, F, Me, CF ₂ HCH ₂ ], [RA4017; F, H, Me, Cl, Me, Me], [RA4018; F, H, Me, Cl, Me, Et], [RA4019; F, H, Me, Cl, Me, Pr], [RA4020; F, H, Me, Cl, Me, i-Pr], [RA4021; F, H, Me, Cl, Me, c-Pr], [RA4022; F, H, Me, Cl, Me, Bu], [RA4023; F, H, Me, Cl, Me, i-Bu], [RA4024; F, H, Me, Cl, Me, t-Bu], [RA4025; F, H, Me, Cl, Me, c-PrCH ₂ ], [RA4026; F, H, Me, Cl, Me, Ph], [RA4027; F, H, Me, Cl, Me, Bn], [RA4028; F, H, Me, Cl, Me, CF ₃ ], [RA4029; F, H, Me, Cl, Me, CF ₃ CH ₂ ], [RA4030; F, H, Me, Cl, Me, CF ₃ CF ₂ ], [RA4031; F, H, Me, Cl, Me, CF ₂ H], [RA4032; F, H, Me, Cl, Me, CF ₂ HCH ₂ ], [RA4033; F, H, Et, H, Me, Me], [RA4034; F, H, Et, H, Me, Et], [RA4035; F, H, Et, H , Me, Pr], [RA4036; F, H, Et, H, Me, i-Pr], [RA4037; F, H, Et, H, Me, c-Pr ], [RA4038; F, H, Et, H, Me, Bu], [RA4039; F, H, Et, H, Me, i-Bu], [RA4040; F, H, Et, H, Me, t -Bu], [RA4041; F, H, Et, H, Me, c-PrCH ₂ ], [RA4042; F, H, Et, H, Me, Ph], [RA4043; F, H, Et, H, Me, Bn], [RA4044; F, H, Et, H, Me, CF ₃ ], [RA4045; F, H, Et, H, Me, CF ₃ CH ₂ ], [RA4046; F, H, Et, H, Me, CF ₃ CF ₂ ], [RA4047; F, H, Et, H, Me, CF ₂ H], [RA4048; F, H, Et, H, Me, CF ₂ HCH ₂ ], [RA4049; F, H, Et, F, Me, Me], [RA4050; F, H, Et, F, Me, Et], [RA4051; F, H, Et, F, Me, Pr], [RA4052; F, H, Et, F, Me, i-Pr], [RA4053; F, H, Et, F, Me, c-Pr], [RA4054; F, H, Et, F, Me, Bu], [RA4055; F, H, Et, F, Me, i-Bu], [RA4056; F, H, Et, F, Me, t-Bu], [RA4057; F, H, Et, F, Me, c-PrCH ₂ ], [RA4058; F, H, Et, F, Me, Ph], [RA4059; F, H, Et, F, Me, Bn], [RA4060; F, H, Et, F, Me, CF ₃ ] , [RA4061; F, H, Et, F, Me, CF ₃ CH ₂ ], [RA4062; F, H, Et, F, Me, CF ₃ CF ₂ ], [RA4063; F, H, Et, F, Me, CF ₂ H], [RA4064; F, H, Et, F, Me, CF ₂ HCH ₂ ], [RA4065; F, H, Et, Cl, Me, Me], [RA4066; F, H, Et , Cl, Me, Et], [RA4067; F, H, Et, Cl, Me, Pr], [RA4068; F, H, Et, Cl, Me, i-Pr], [RA4069; F, H, Et , Cl, Me, c-Pr], [RA4070; F, H, Et, Cl, Me, Bu], [RA4071; F, H, Et, Cl, Me, i-Bu], [RA4072; F, H , Et, Cl, Me, t-Bu], [RA4073; F, H, Et, Cl, Me, c-PrCH ₂ ], [RA4074; F, H, Et, Cl, Me , Ph], [RA4075; F, H, Et, Cl, Me, Bn], [RA4076; F, H, Et, Cl, Me, CF ₃ ], [RA4077; F, H, Et, Cl, Me, CF ₃ CH ₂ ], [RA4078; F, H, Et, Cl, Me, CF ₃ CF ₂ ], [RA4079; F, H, Et, Cl, Me, CF ₂ H], [RA4080; F, H, Et, Cl, Me, CF ₂ HCH ₂ ], [RA4081; F, H, F, H, Me, Me], [RA4082; F, H, F, H, Me, Et], [RA4083; F, H , F, H, Me, Pr], [RA4084; F, H, F, H, Me, i-Pr], [RA4085; F, H, F, H, Me, c-Pr], [RA4086; F , H, F, H, Me, Bu], [RA4087; F, H, F, H, Me, i-Bu], [RA4088; F, H, F, H, Me, t-Bu], [RA4089 ; F, H, F, H, Me, c-PrCH ₂ ], [RA4090; F, H, F, H, Me, Ph], [RA4091; F, H, F, H, Me, Bn], [ RA4092; F, H, F, H, Me, CF ₃ ], [RA4093; F, H, F, H, Me, CF ₃ CH ₂ ], [RA4094; F, H, F, H, Me, CF ₃ CF ₂ ], [RA4095; F, H, F, H, Me, CF ₂ H], [RA4096; F, H, F, H, Me, CF ₂ HCH ₂ ], [RA4097; F, H, F, F, Me, Me], [RA4098; F, H, F, F, Me, Et], [RA4099; F, H, F, F, Me, Pr], [RA4100; F, H, F, F, Me, i-Pr], [RA4101; F, H, F, F, Me, c-Pr], [RA4102; F, H, F, F, Me, Bu], [RA4103; F, H, F, F, Me, i-Bu], [RA4104; F, H, F, F, Me, t-Bu], [RA4105; F, H, F, F, Me, c-PrCH ₂ ], [RA4106; F , H, F, F, Me, Ph], [RA4107; F, H, F, F, Me, Bn], [RA4108; F, H, F, F, Me, CF ₃ ], [RA4109; F, H, F, F, Me, CF ₃ CH ₂ ], [RA4110; F, H, F, F, Me, CF ₃ CF ₂ ], [RA4111; F, H, F, F, Me, CF ₂ H] , [RA4112; F, H, F, F , Me, CF ₂ HCH ₂ ], [RA4113; F, H, F, Cl, Me, Me], [RA4114; F, H, F, Cl, Me, Et], [RA4115; F, H, F, Cl, Me, Pr], [RA4116; F, H, F, Cl, Me, i-Pr], [RA4117; F, H, F, Cl, Me, c-Pr], [RA4118; F, H, F, Cl, Me, Bu], [RA4119; F, H, F, Cl, Me, i-Bu], [RA4120; F, H, F, Cl, Me, t-Bu], [RA4121; F, H, F, Cl, Me, c-PrCH ₂ ], [RA4122; F, H, F, Cl, Me, Ph], [RA4123; F, H, F, Cl, Me, Bn], [RA4124; F , H, F, Cl, Me, CF ₃ ], [RA4125; F, H, F, Cl, Me, CF ₃ CH ₂ ], [RA4126; F, H, F, Cl, Me, CF ₃ CF ₂ ] , [RA4127; F, H, F, Cl, Me, CF ₂ H], [RA4128; F, H, F, Cl, Me, CF ₂ HCH ₂ ], [RA4129; F, H, Cl, H, Me , Me], [RA4130; F, H, Cl, H, Me, Et], [RA4131; F, H, Cl, H, Me, Pr], [RA4132; F, H, Cl, H, Me, i -Pr], [RA4133; F, H, Cl, H, Me, c-Pr], [RA4134; F, H, Cl, H, Me, Bu], [RA4135; F, H, Cl, H, Me , i-Bu], [RA4136; F, H, Cl, H, Me, t-Bu], [RA4137; F, H, Cl, H, Me, c-PrCH ₂ ], [RA4138; F, H, Cl, H, Me, Ph], [RA4139; F, H, Cl, H, Me, Bn], [RA4140; F, H, Cl, H, Me, CF ₃ ], [RA4141; F, H, Cl , H, Me, CF ₃ CH ₂ ], [RA4142; F, H, Cl, H, Me, CF ₃ CF ₂ ], [RA4143; F, H, Cl, H, Me, CF ₂ H], [RA4144 ; F, H, Cl, H, Me, CF ₂ HCH ₂ ], [RA4145; F, H, Cl, Cl, Me, Me], [RA4146; F, H, Cl, Cl, Me, Et], [ RA4147; F, H, Cl, Cl, Me, Pr], [RA4148; F, H, Cl, Cl, Me, i-Pr], [RA4149; F, H, Cl, Cl, M e, c-Pr], [RA4150; F, H, Cl, Cl, Me, Bu], [RA4151; F, H, Cl, Cl, Me, i-Bu], [RA4152; F, H, Cl, Cl, Me, t-Bu], [RA4153; F, H, Cl, Cl, Me, c-PrCH ₂ ], [RA4154; F, H, Cl, Cl, Me, Ph], [RA4155; F, H , Cl, Cl, Me, Bn], [RA4156; F, H, Cl, Cl, Me, CF ₃ ], [RA4157; F, H, Cl, Cl, Me, CF ₃ CH ₂ ], [RA4158; F , H, Cl, Cl, Me, CF ₃ CF ₂ ], [RA4159; F, H, Cl, Cl, Me, CF ₂ H], [RA4160; F, H, Cl, Cl, Me, CF ₂ HCH ₂ ], [RA4161; F, H, Me, H, Et, Me], [RA4162; F, H, Me, H, Et, Et], [RA4163; F, H, Me, H, Et, Pr], [RA4164; F, H, Me, H, Et, i-Pr], [RA4165; F, H, Me, H, Et, c-Pr], [RA4166; F, H, Me, H, Et, Bu ], [RA4167; F, H, Me, H, Et, i-Bu], [RA4168; F, H, Me, H, Et, t-Bu], [RA4169; F, H, Me, H, Et , c-PrCH ₂ ], [RA4170; F, H, Me, H, Et, Ph], [RA4171; F, H, Me, H, Et, Bn], [RA4172; F, H, Me, H, Et, CF ₃ ], [RA4173; F, H, Me, H, Et, CF ₃ CH ₂ ], [RA4174; F, H, Me, H, Et, CF ₃ CF ₂ ], [RA4175; F, H , Me, H, Et, CF ₂ H], [RA4176; F, H, Me, H, Et, CF ₂ HCH ₂ ], [RA4177; F, H, Me, Me, Et, Me], [RA4178; F, H, Me, Me, Et, Et], [RA4179; F, H, Me, Me, Et, Pr], [RA4180; F, H, Me, Me, Et, i-Pr], [RA4181; F, H, Me, Me, Et, c-Pr], [RA4182; F, H, Me, Me, Et, Bu], [RA4183; F, H, Me, Me, Et, i-Bu], [ RA4184; F, H, Me, Me, Et, t-Bu], [RA4185; F, H, Me, Me, Et, c-PrCH ₂ ], [RA 4186; F, H, Me, Me, Et, Ph], [RA4187; F, H, Me, Me, Et, Bn], [RA4188; F, H, Me, Me, Et, CF ₃ ], [RA4189 ; F, H, Me, Me, Et, CF ₃ CH ₂ ], [RA4190; F, H, Me, Me, Et, CF ₃ CF ₂ ], [RA4191; F, H, Me, Me, Et, CF ₂ H], [RA4192; F, H, Me, Me, Et, CF ₂ HCH ₂ ], [RA4193; F, H, Me, Et, Et, Me], [RA4194; F, H, Me, Et, Et, Et], [RA4195; F, H, Me, Et, Et, Pr], [RA4196; F, H, Me, Et, Et, i-Pr], [RA4197; F, H, Me, Et, Et, c-Pr], [RA4198; F, H, Me, Et, Et, Bu], [RA4199; F, H, Me, Et, Et, i-Bu], [RA4200; F, H, Me, Et, Et, t-Bu],

[RA4201; F, H, Me, Et, Et, c-PrCH ₂ ], [RA4202; F, H, Me, Et, Et, Ph], [RA4203; F, H, Me, Et, Et, Bn] , [RA4204; F, H, Me, Et, Et, CF ₃ ], [RA4205; F, H, Me, Et, Et, CF ₃ CH ₂ ], [RA4206; F, H, Me, Et, Et, CF ₃ CF ₂ ], [RA4207; F, H, Me, Et, Et, CF ₂ H], [RA4208; F, H, Me, Et, Et, CF ₂ HCH ₂ ], [RA4209; F, H, Me, F, Et, Me], [RA4210; F, H, Me, F, Et, Et], [RA4211; F, H, Me, F, Et, Pr], [RA4212; F, H, Me, F, Et, i-Pr], [RA4213; F, H, Me, F, Et, c-Pr], [RA4214; F, H, Me, F, Et, Bu], [RA4215; F, H, Me, F, Et, i-Bu], [RA4216; F, H, Me, F, Et, t-Bu], [RA4217; F, H, Me, F, Et, c-PrCH ₂ ], [RA4218 ; F, H, Me, F, Et, Ph], [RA4219; F, H, Me, F, Et, Bn], [RA4220; F, H, Me, F, Et, CF ₃ ], [RA4221; F, H, Me, F, Et, CF ₃ CH ₂ ], [RA4222; F, H, Me, F, Et, CF ₃ CF ₂ ], [RA4223; F, H, Me, F, Et, CF ₂ H], [RA4224; F, H, Me, F, Et, CF ₂ HCH ₂ ], [RA4225; F, H, Me, Cl, Et, Me], [RA4226; F, H, Me, Cl, Et , Et], [RA4227; F, H, Me, Cl, Et, Pr], [RA4228; F, H, Me, Cl, Et, i-Pr], [RA4229; F, H, Me, Cl, Et , c-Pr], [RA4230; F, H, Me, Cl, Et, Bu], [RA4231; F, H, Me, Cl, Et, i-Bu], [RA4232; F, H, Me, Cl , Et, t-Bu], [RA4233; F, H, Me, Cl, Et, c-PrCH ₂ ], [RA4234; F, H, Me, Cl, Et, Ph], [RA4235; F, H, Me, Cl, Et, Bn], [RA4236; F, H, Me, Cl, Et, CF ₃ ], [RA4237; F, H, Me, Cl, Et, CF ₃ CH ₂ ], [RA4238; F, H, Me, Cl, Et, CF ₃ CF ₂ ], [RA4239; F, H, Me, Cl, Et, CF ₂ H], [ RA4240; F, H, Me, Cl, Et, CF ₂ HCH ₂ ], [RA4241; F, H, Et, H, Et, Me], [RA4242; F, H, Et, H, Et, Et], [RA4243; F, H, Et, H, Et, Pr], [RA4244; F, H, Et, H, Et, i-Pr], [RA4245; F, H, Et, H, Et, c-Pr ], [RA4246; F, H, Et, H, Et, Bu], [RA4247; F, H, Et, H, Et, i-Bu], [RA4248; F, H, Et, H, Et, t -Bu], [RA4249; F, H, Et, H, Et, c-PrCH ₂ ], [RA4250; F, H, Et, H, Et, Ph], [RA4251; F, H, Et, H, Et, Bn], [RA4252; F, H, Et, H, Et, CF ₃ ], [RA4253; F, H, Et, H, Et, CF ₃ CH ₂ ], [RA4254; F, H, Et, H, Et, CF ₃ CF ₂ ], [RA4255; F, H, Et, H, Et, CF ₂ H], [RA4256; F, H, Et, H, Et, CF ₂ HCH ₂ ], [RA4257; F, H, Et, F, Et, Me], [RA4258; F, H, Et, F, Et, Et], [RA4259; F, H, Et, F, Et, Pr], [RA4260; F, H, Et, F, Et, i-Pr], [RA4261; F, H, Et, F, Et, c-Pr], [RA4262; F, H, Et, F, Et, Bu], [RA4263; F, H, Et, F, Et, i-Bu], [RA4264; F, H, Et, F, Et, t-Bu], [RA4265; F, H, Et, F, Et, c-PrCH ₂ ], [RA4266; F, H, Et, F, Et, Ph], [RA4267; F, H, Et, F, Et, Bn], [RA4268; F, H, Et, F, Et, CF ₃ ] , [RA4269; F, H, Et, F, Et, CF ₃ CH ₂ ], [RA4270; F, H, Et, F, Et, CF ₃ CF ₂ ], [RA4271; F, H, Et, F, Et, CF ₂ H], [RA4272; F, H, Et, F, Et, CF ₂ HCH ₂ ], [RA4273; F, H, Et, Cl, Et, Me], [RA4274; F, H, Et, Cl, Et, Et], [RA4275; F, H, Et, Cl, Et, Pr], [RA4276; F, H, Et, Cl, Et, i- Pr], [RA4277; F, H, Et, Cl, Et, c-Pr], [RA4278; F, H, Et, Cl, Et, Bu], [RA4279; F, H, Et, Cl, Et, i-Bu], [RA4280; F, H, Et, Cl, Et, t-Bu], [RA4281; F, H, Et, Cl, Et, c-PrCH ₂ ], [RA4282; F, H, Et , Cl, Et, Ph], [RA4283; F, H, Et, Cl, Et, Bn], [RA4284; F, H, Et, Cl, Et, CF ₃ ], [RA4285; F, H, Et, Cl, Et, CF ₃ CH ₂ ], [RA4286; F, H, Et, Cl, Et, CF ₃ CF ₂ ], [RA4287; F, H, Et, Cl, Et, CF ₂ H], [RA4288; F, H, Et, Cl, Et, CF ₂ HCH ₂ ], [RA4289; F, H, F, H, Et, Me], [RA4290; F, H, F, H, Et, Et], [RA4291 ; F, H, F, H, Et, Pr], [RA4292; F, H, F, H, Et, i-Pr], [RA4293; F, H, F, H, Et, c-Pr], [RA4294; F, H, F, H, Et, Bu], [RA4295; F, H, F, H, Et, i-Bu], [RA4296; F, H, F, H, Et, t-Bu ], [RA4297; F, H, F, H, Et, c-PrCH ₂ ], [RA4298; F, H, F, H, Et, Ph], [RA4299; F, H, F, H, Et, Bn], [RA4300; F, H, F, H, Et, CF ₃ ], [RA4301; F, H, F, H, Et, CF ₃ CH ₂ ], [RA4302; F, H, F, H, Et, CF ₃ CF ₂ ], [RA4303; F, H, F, H, Et, CF ₂ H], [RA4304; F, H, F, H, Et, CF ₂ HCH ₂ ], [RA4305; F, H, F, F, Et, Me], [RA4306; F, H, F, F, Et, Et], [RA4307; F, H, F, F, Et, Pr], [RA4308; F, H, F, F, Et, i-Pr], [RA4309; F, H, F, F, Et, c-Pr], [RA4310; F, H, F, F, Et, Bu], [RA4311; F, H, F, F, E t, i-Bu], [RA4312; F, H, F, F, Et, t-Bu], [RA4313; F, H, F, F, Et, c-PrCH ₂ ], [RA4314; F, H , F, F, Et, Ph], [RA4315; F, H, F, F, Et, Bn], [RA4316; F, H, F, F, Et, CF ₃ ], [RA4317; F, H, F, F, Et, CF ₃ CH ₂ ], [RA4318; F, H, F, F, Et, CF ₃ CF ₂ ], [RA4319; F, H, F, F, Et, CF ₂ H], [ RA4320; F, H, F, F, Et, CF ₂ HCH ₂ ], [RA4321; F, H, F, Cl, Et, Me], [RA4322; F, H, F, Cl, Et, Et], [RA4323; F, H, F, Cl, Et, Pr], [RA4324; F, H, F, Cl, Et, i-Pr], [RA4325; F, H, F, Cl, Et, c-Pr ], [RA4326; F, H, F, Cl, Et, Bu], [RA4327; F, H, F, Cl, Et, i-Bu], [RA4328; F, H, F, Cl, Et, t -Bu], [RA4329; F, H, F, Cl, Et, c-PrCH ₂ ], [RA4330; F, H, F, Cl, Et, Ph], [RA4331; F, H, F, Cl, Et, Bn], [RA4332; F, H, F, Cl, Et, CF ₃ ], [RA4333; F, H, F, Cl, Et, CF ₃ CH ₂ ], [RA4334; F, H, F, Cl, Et, CF ₃ CF ₂ ], [RA4335; F, H, F, Cl, Et, CF ₂ H], [RA4336; F, H, F, Cl, Et, CF ₂ HCH ₂ ], [RA4337; F, H, Cl, H, Et, Me], [RA4338; F, H, Cl, H, Et, Et], [RA4339; F, H, Cl, H, Et, Pr], [RA4340; F, H, Cl, H, Et, i-Pr], [RA4341; F, H, Cl, H, Et, c-Pr], [RA4342; F, H, Cl, H, Et, Bu], [RA4343; F, H, Cl, H, Et, i-Bu], [RA4344; F, H, Cl, H, Et, t-Bu], [RA4345; F, H, Cl, H, Et, c-PrCH ₂ ], [RA4346; F, H, Cl, H, Et, Ph], [RA4347; F, H, Cl, H, Et, Bn], [RA4348; F, H, Cl, H, Et, CF ₃ ] , [RA4349 ; F, H, Cl, H, Et, CF ₃ CH ₂ ], [RA4350; F, H, Cl, H, Et, CF ₃ CF ₂ ], [RA4351; F, H, Cl, H, Et, CF ₂ H], [RA4352; F, H, Cl, H, Et, CF ₂ HCH ₂ ], [RA4353; F, H, Cl, Cl, Et, Me], [RA4354; F, H, Cl, Cl, Et, Et], [RA4355; F, H, Cl, Cl, Et, Pr], [RA4356; F, H, Cl, Cl, Et, i-Pr], [RA4357; F, H, Cl, Cl, Et, c-Pr], [RA4358; F, H, Cl, Cl, Et, Bu], [RA4359; F, H, Cl, Cl, Et, i-Bu], [RA4360; F, H, Cl, Cl, Et, t-Bu], [RA4361; F, H, Cl, Cl, Et, c-PrCH ₂ ], [RA4362; F, H, Cl, Cl, Et, Ph], [RA4363; F, H , Cl, Cl, Et, Bn], [RA4364; F, H, Cl, Cl, Et, CF ₃ ], [RA4365; F, H, Cl, Cl, Et, CF ₃ CH ₂ ], [RA4366; F , H, Cl, Cl, Et, CF ₃ CF ₂ ], [RA4367; F, H, Cl, Cl, Et, CF ₂ H], [RA4368; F, H, Cl, Cl, Et, CF ₂ HCH ₂ ], [RA4369; F, H, Me, H, Pr, Me], [RA4370; F, H, Me, H, Pr, Et], [RA4371; F, H, Me, H, Pr, Pr], [RA4372; F, H, Me, H, Pr, i-Pr], [RA4373; F, H, Me, H, Pr, c-Pr], [RA4374; F, H, Me, H, Pr, Bu ], [RA4375; F, H, Me, H, Pr, i-Bu], [RA4376; F, H, Me, H, Pr, t-Bu], [RA4377; F, H, Me, H, Pr , c-PrCH ₂ ], [RA4378; F, H, Me, H, Pr, Ph], [RA4379; F, H, Me, H, Pr, Bn], [RA4380; F, H, Me, H, Pr, CF ₃ ], [RA4381; F, H, Me, H, Pr, CF ₃ CH ₂ ], [RA4382; F, H, Me, H, Pr, CF ₃ CF ₂ ], [RA4383; F, H , Me, H, Pr, CF ₂ H], [RA4384; F, H, Me, H, Pr, CF ₂ HCH ₂ ], [RA4 385; F, H, Me, Me, Pr, Me], [RA4386; F, H, Me, Me, Pr, Et], [RA4387; F, H, Me, Me, Pr, Pr], [RA4388; F, H, Me, Me, Pr, i-Pr], [RA4389; F, H, Me, Me, Pr, c-Pr], [RA4390; F, H, Me, Me, Pr, Bu], [ RA4391; F, H, Me, Me, Pr, i-Bu], [RA4392; F, H, Me, Me, Pr, t-Bu], [RA4393; F, H, Me, Me, Pr, c- PrCH ₂ ], [RA4394; F, H, Me, Me, Pr, Ph], [RA4395; F, H, Me, Me, Pr, Bn], [RA4396; F, H, Me, Me, Pr, CF ₃ ], [RA4397; F, H, Me, Me, Pr, CF ₃ CH ₂ ], [RA4398; F, H, Me, Me, Pr, CF ₃ CF ₂ ], [RA4399; F, H, Me, Me, Pr, CF ₂ H], [RA4400; F, H, Me, Me, Pr, CF ₂ HCH ₂ ],

[RA4401; F, H, Me, Et, Pr, Me], [RA4402; F, H, Me, Et, Pr, Et], [RA4403; F, H, Me, Et, Pr, Pr], [RA4404 ; F, H, Me, Et, Pr, i-Pr], [RA4405; F, H, Me, Et, Pr, c-Pr], [RA4406; F, H, Me, Et, Pr, Bu], [RA4407; F, H, Me, Et, Pr, i-Bu], [RA4408; F, H, Me, Et, Pr, t-Bu], [RA4409; F, H, Me, Et, Pr, c -PrCH ₂ ], [RA4410; F, H, Me, Et, Pr, Ph], [RA4411; F, H, Me, Et, Pr, Bn], [RA4412; F, H, Me, Et, Pr, CF ₃ ], [RA4413; F, H, Me, Et, Pr, CF ₃ CH ₂ ], [RA4414; F, H, Me, Et, Pr, CF ₃ CF ₂ ], [RA4415; F, H, Me , Et, Pr, CF ₂ H], [RA4416; F, H, Me, Et, Pr, CF ₂ HCH ₂ ], [RA4417; F, H, Me, F, Pr, Me], [RA4418; F, H, Me, F, Pr, Et], [RA4419; F, H, Me, F, Pr, Pr], [RA4420; F, H, Me, F, Pr, i-Pr], [RA4421; F, H, Me, F, Pr, c-Pr], [RA4422; F, H, Me, F, Pr, Bu], [RA4423; F, H, Me, F, Pr, i-Bu], [RA4424; F, H, Me, F, Pr, t-Bu], [RA4425; F, H, Me, F, Pr, c-PrCH ₂ ], [RA4426; F, H, Me, F, Pr, Ph], [RA4427; F, H, Me, F, Pr, Bn], [RA4428; F, H, Me, F, Pr, CF ₃ ], [RA4429; F, H, Me, F, Pr, CF ₃ CH ₂ ], [RA4430; F, H, Me, F, Pr, CF ₃ CF ₂ ], [RA4431; F, H, Me, F, Pr, CF ₂ H], [RA4432; F, H, Me, F, Pr, CF ₂ HCH ₂ ], [RA4433; F, H, Me, Cl, Pr, Me], [RA4434; F, H, Me, Cl, Pr, Et], [RA4435; F, H, Me, Cl , Pr, Pr], [RA4436; F, H, Me, Cl, Pr, i-Pr], [RA4437; F, H, Me, Cl, Pr , c-Pr], [RA4438; F, H, Me, Cl, Pr, Bu], [RA4439; F, H, Me, Cl, Pr, i-Bu], [RA4440; F, H, Me, Cl , Pr, t-Bu], [RA4441; F, H, Me, Cl, Pr, c-PrCH ₂ ], [RA4442; F, H, Me, Cl, Pr, Ph], [RA4443; F, H, Me, Cl, Pr, Bn], [RA4444; F, H, Me, Cl, Pr, CF ₃ ], [RA4445; F, H, Me, Cl, Pr, CF ₃ CH ₂ ], [RA4446; F, H, Me, Cl, Pr, CF ₃ CF ₂ ], [RA4447; F, H, Me, Cl, Pr, CF ₂ H], [RA4448; F, H, Me, Cl, Pr, CF ₂ HCH ₂ ] , [RA4449; F, H, Et, H, Pr, Me], [RA4450; F, H, Et, H, Pr, Et], [RA4451; F, H, Et, H, Pr, Pr], [ RA4452; F, H, Et, H, Pr, i-Pr], [RA4453; F, H, Et, H, Pr, c-Pr], [RA4454; F, H, Et, H, Pr, Bu] , [RA4455; F, H, Et, H, Pr, i-Bu], [RA4456; F, H, Et, H, Pr, t-Bu], [RA4457; F, H, Et, H, Pr, c-PrCH ₂ ], [RA4458; F, H, Et, H, Pr, Ph], [RA4459; F, H, Et, H, Pr, Bn], [RA4460; F, H, Et, H, Pr , CF ₃ ], [RA4461; F, H, Et, H, Pr, CF ₃ CH ₂ ], [RA4462; F, H, Et, H, Pr, CF ₃ CF ₂ ], [RA4463; F, H, Et, H, Pr, CF ₂ H], [RA4464; F, H, Et, H, Pr, CF ₂ HCH ₂ ], [RA4465; F, H, Et, F, Pr, Me], [RA4466; F , H, Et, F, Pr, Et], [RA4467; F, H, Et, F, Pr, Pr], [RA4468; F, H, Et, F, Pr, i-Pr], [RA4469; F , H, Et, F, Pr, c-Pr], [RA4470; F, H, Et, F, Pr, Bu], [RA4471; F, H, Et, F, Pr, i-Bu], [RA4472 ; F, H, Et, F, Pr, t-Bu], [RA4473; F, H, Et, F, Pr, c-PrCH ₂ ], [RA4474; F, H, E t, F, Pr, Ph], [RA4475; F, H, Et, F, Pr, Bn], [RA4476; F, H, Et, F, Pr, CF ₃ ], [RA4477; F, H, Et , F, Pr, CF ₃ CH ₂ ], [RA4478; F, H, Et, F, Pr, CF ₃ CF ₂ ], [RA4479; F, H, Et, F, Pr, CF ₂ H], [RA4480 ; F, H, Et, F, Pr, CF ₂ HCH ₂ ], [RA4481; F, H, Et, Cl, Pr, Me], [RA4482; F, H, Et, Cl, Pr, Et], [ RA4483; F, H, Et, Cl, Pr, Pr], [RA4484; F, H, Et, Cl, Pr, i-Pr], [RA4485; F, H, Et, Cl, Pr, c-Pr] , [RA4486; F, H, Et, Cl, Pr, Bu], [RA4487; F, H, Et, Cl, Pr, i-Bu], [RA4488; F, H, Et, Cl, Pr, t- Bu], [RA4489; F, H, Et, Cl, Pr, c-PrCH ₂ ], [RA4490; F, H, Et, Cl, Pr, Ph], [RA4491; F, H, Et, Cl, Pr , Bn], [RA4492; F, H, Et, Cl, Pr, CF ₃ ], [RA4493; F, H, Et, Cl, Pr, CF ₃ CH ₂ ], [RA4494; F, H, Et, Cl , Pr, CF ₃ CF ₂ ], [RA4495; F, H, Et, Cl, Pr, CF ₂ H], [RA4496; F, H, Et, Cl, Pr, CF ₂ HCH ₂ ], [RA4497; F , H, F, H, Pr, Me], [RA4498; F, H, F, H, Pr, Et], [RA4499; F, H, F, H, Pr, Pr], [RA4500; F, H , F, H, Pr, i-Pr], [RA4501; F, H, F, H, Pr, c-Pr], [RA4502; F, H, F, H, Pr, Bu], [RA4503; F , H, F, H, Pr, i-Bu], [RA4504; F, H, F, H, Pr, t-Bu], [RA4505; F, H, F, H, Pr, c-PrCH ₂ ] , [RA4506; F, H, F, H, Pr, Ph], [RA4507; F, H, F, H, Pr, Bn], [RA4508; F, H, F, H, Pr, CF ₃ ], [RA4509; F, H, F, H, Pr, CF ₃ CH ₂ ], [RA4510; F, H, F, H, Pr, CF ₃ CF ₂ ], [RA4511; F, H, F, H, Pr, CF ₂ H], [RA4512; F, H, F, H, Pr, CF ₂ HCH ₂ ], [RA4513; F, H, F, F, Pr, Me], [RA4514 ; F, H, F, F, Pr, Et], [RA4515; F, H, F, F, Pr, Pr], [RA4516; F, H, F, F, Pr, i-Pr], [RA4517 ; F, H, F, F, Pr, c-Pr], [RA4518; F, H, F, F, Pr, Bu], [RA4519; F, H, F, F, Pr, i-Bu], [RA4520; F, H, F, F, Pr, t-Bu], [RA4521; F, H, F, F, Pr, c-PrCH ₂ ], [RA4522; F, H, F, F, Pr, Ph], [RA4523; F, H, F, F, Pr, Bn], [RA4524; F, H, F, F, Pr, CF ₃ ], [RA4525; F, H, F, F, Pr, CF ₃ CH ₂ ], [RA4526; F, H, F, F, Pr, CF ₃ CF ₂ ], [RA4527; F, H, F, F, Pr, CF ₂ H], [RA4528; F, H, F , F, Pr, CF ₂ HCH ₂ ], [RA4529; F, H, F, Cl, Pr, Me], [RA4530; F, H, F, Cl, Pr, Et], [RA4531; F, H, F, Cl, Pr, Pr], [RA4532; F, H, F, Cl, Pr, i-Pr], [RA4533; F, H, F, Cl, Pr, c-Pr], [RA4534; F, H, F, Cl, Pr, Bu], [RA4535; F, H, F, Cl, Pr, i-Bu], [RA4536; F, H, F, Cl, Pr, t-Bu], [RA4537; F, H, F, Cl, Pr, c-PrCH ₂ ], [RA4538; F, H, F, Cl, Pr, Ph], [RA4539; F, H, F, Cl, Pr, Bn], [RA4540 ; F, H, F, Cl, Pr, CF ₃ ], [RA4541; F, H, F, Cl, Pr, CF ₃ CH ₂ ], [RA4542; F, H, F, Cl, Pr, CF ₃ CF ₂ ], [RA4543; F, H, F, Cl, Pr, CF ₂ H], [RA4544; F, H, F, Cl, Pr, CF ₂ HCH ₂ ], [RA4545; F, H, Cl, H , Pr, Me], [RA4546; F, H, Cl, H, Pr, Et], [RA4547; F, H, Cl, H, Pr, Pr], [RA4548; F, H, Cl, H, Pr , i-Pr], [RA4549 ; F, H, Cl, H, Pr, c-Pr], [RA4550; F, H, Cl, H, Pr, Bu], [RA4551; F, H, Cl, H, Pr, i-Bu], [RA4552; F, H, Cl, H, Pr, t-Bu], [RA4553; F, H, Cl, H, Pr, c-PrCH ₂ ], [RA4554; F, H, Cl, H, Pr, Ph], [RA4555; F, H, Cl, H, Pr, Bn], [RA4556; F, H, Cl, H, Pr, CF ₃ ], [RA4557; F, H, Cl, H, Pr, CF ₃ CH ₂ ], [RA4558; F, H, Cl, H, Pr, CF ₃ CF ₂ ], [RA4559; F, H, Cl, H, Pr, CF ₂ H], [RA4560; F, H, Cl , H, Pr, CF ₂ HCH ₂ ], [RA4561; F, H, Cl, Cl, Pr, Me], [RA4562; F, H, Cl, Cl, Pr, Et], [RA4563; F, H, Cl, Cl, Pr, Pr], [RA4564; F, H, Cl, Cl, Pr, i-Pr], [RA4565; F, H, Cl, Cl, Pr, c-Pr], [RA4566; F, H, Cl, Cl, Pr, Bu], [RA4567; F, H, Cl, Cl, Pr, i-Bu], [RA4568; F, H, Cl, Cl, Pr, t-Bu], [RA4569; F, H, Cl, Cl, Pr, c-PrCH ₂ ], [RA4570; F, H, Cl, Cl, Pr, Ph], [RA4571; F, H, Cl, Cl, Pr, Bn], [RA4572 ; F, H, Cl, Cl, Pr, CF ₃ ], [RA4573; F, H, Cl, Cl, Pr, CF ₃ CH ₂ ], [RA4574; F, H, Cl, Cl, Pr, CF ₃ CF ₂ ], [RA4575; F, H, Cl, Cl, Pr, CF ₂ H], [RA4576; F, H, Cl, Cl, Pr, CF ₂ HCH ₂ ], [RA4577; F, H, Me, H , Bu, Me], [RA4578; F, H, Me, H, Bu, Et], [RA4579; F, H, Me, H, Bu, Pr], [RA4580; F, H, Me, H, Bu , i-Pr], [RA4581; F, H, Me, H, Bu, c-Pr], [RA4582; F, H, Me, H, Bu, Bu], [RA4583; F, H, Me, H , Bu, i-Bu], [RA4584; F, H, Me, H, Bu, t-Bu], [RA4585; F, H, Me, H, Bu, c-PrCH ₂ ], [RA4586; F, H, Me, H, Bu, Ph], [RA4587; F, H, Me, H, Bu, Bn], [RA4588; F, H, Me, H, Bu, CF ₃ ], [RA4589; F, H, Me, H, Bu, CF ₃ CH ₂ ], [RA4590; F, H, Me, H, Bu, CF ₃ CF ₂ ], [RA4591; F, H, Me, H , Bu, CF ₂ H], [RA4592; F, H, Me, H, Bu, CF ₂ HCH ₂ ], [RA4593; F, H, Me, Me, Bu, Me], [RA4594; F, H, Me, Me, Bu, Et], [RA4595; F, H, Me, Me, Bu, Pr], [RA4596; F, H, Me, Me, Bu, i-Pr], [RA4597; F, H, Me, Me, Bu, c-Pr], [RA4598; F, H, Me, Me, Bu, Bu], [RA4599; F, H, Me, Me, Bu, i-Bu], [RA4600; F, H, Me, Me, Bu, t-Bu],

[RA4601; F, H, Me, Me, Bu, c-PrCH ₂ ], [RA4602; F, H, Me, Me, Bu, Ph], [RA4603; F, H, Me, Me, Bu, Bn] , [RA4604; F, H, Me, Me, Bu, CF ₃ ], [RA4605; F, H, Me, Me, Bu, CF ₃ CH ₂ ], [RA4606; F, H, Me, Me, Bu, CF ₃ CF ₂ ], [RA4607; F, H, Me, Me, Bu, CF ₂ H], [RA4608; F, H, Me, Me, Bu, CF ₂ HCH ₂ ], [RA4609; F, H, Me, Et, Bu, Me], [RA4610; F, H, Me, Et, Bu, Et], [RA4611; F, H, Me, Et, Bu, Pr], [RA4612; F, H, Me, Et, Bu, i-Pr], [RA4613; F, H, Me, Et, Bu, c-Pr], [RA4614; F, H, Me, Et, Bu, Bu], [RA4615; F, H, Me, Et, Bu, i-Bu], [RA4616; F, H, Me, Et, Bu, t-Bu], [RA4617; F, H, Me, Et, Bu, c-PrCH ₂ ], [RA4618 ; F, H, Me, Et, Bu, Ph], [RA4619; F, H, Me, Et, Bu, Bn], [RA4620; F, H, Me, Et, Bu, CF ₃ ], [RA4621; F, H, Me, Et, Bu, CF ₃ CH ₂ ], [RA4622; F, H, Me, Et, Bu, CF ₃ CF ₂ ], [RA4623; F, H, Me, Et, Bu, CF ₂ H], [RA4624; F, H, Me, Et, Bu, CF ₂ HCH ₂ ], [RA4625; F, H, Me, F, Bu, Me], [RA4626; F, H, Me, F, Bu , Et], [RA4627; F, H, Me, F, Bu, Pr], [RA4628; F, H, Me, F, Bu, i-Pr], [RA4629; F, H, Me, F, Bu , c-Pr], [RA4630; F, H, Me, F, Bu, Bu], [RA4631; F, H, Me, F, Bu, i-Bu], [RA4632; F, H, Me, F , Bu, t-Bu], [RA4633; F, H, Me, F, Bu, c-PrCH ₂ ], [RA4634; F, H, Me, F, Bu, Ph], [RA4635; F, H, Me, F, Bu, Bn], [RA4636; F, H, Me, F, Bu, CF ₃ ], [RA4637; F, H, Me, F, Bu, CF ₃ CH ₂ ], [RA4638; F, H, Me, F, Bu, CF ₃ CF ₂ ], [RA4639; F, H, Me, F, Bu, CF ₂ H], [RA4640; F, H, Me, F, Bu, CF ₂ HCH ₂ ], [RA4641; F, H, Me, Cl, Bu, Me], [RA4642; F, H, Me, Cl, Bu , Et], [RA4643; F, H, Me, Cl, Bu, Pr], [RA4644; F, H, Me, Cl, Bu, i-Pr], [RA4645; F, H, Me, Cl, Bu , c-Pr], [RA4646; F, H, Me, Cl, Bu, Bu], [RA4647; F, H, Me, Cl, Bu, i-Bu], [RA4648; F, H, Me, Cl , Bu, t-Bu], [RA4649; F, H, Me, Cl, Bu, c-PrCH ₂ ], [RA4650; F, H, Me, Cl, Bu, Ph], [RA4651; F, H, Me, Cl, Bu, Bn], [RA4652; F, H, Me, Cl, Bu, CF ₃ ], [RA4653; F, H, Me, Cl, Bu, CF ₃ CH ₂ ], [RA4654; F, H, Me, Cl, Bu, CF ₃ CF ₂ ], [RA4655; F, H, Me, Cl, Bu, CF ₂ H], [RA4656; F, H, Me, Cl, Bu, CF ₂ HCH ₂ ] , [RA4657; F, H, Et, H, Bu, Me], [RA4658; F, H, Et, H, Bu, Et], [RA4659; F, H, Et, H, Bu, Pr], [ RA4660; F, H, Et, H, Bu, i-Pr], [RA4661; F, H, Et, H, Bu, c-Pr], [RA4662; F, H, Et, H, Bu, Bu] , [RA4663; F, H, Et, H, Bu, i-Bu], [RA4664; F, H, Et, H, Bu, t-Bu], [RA4665; F, H, Et, H, Bu, c-PrCH ₂ ], [RA4666; F, H, Et, H, Bu, Ph], [RA4667; F, H, Et, H, Bu, Bn], [RA4668; F, H, Et, H, Bu , CF ₃ ], [RA4669; F, H, Et, H, Bu, CF ₃ CH ₂ ], [RA4670; F, H, Et, H, Bu, CF ₃ CF ₂ ], [RA4671; F, H, Et, H, Bu, CF ₂ H], [RA4672; F, H, Et, H, Bu, CF ₂ HCH ₂ ], [RA46 73; F, H, Et, F, Bu, Me], [RA4674; F, H, Et, F, Bu, Et], [RA4675; F, H, Et, F, Bu, Pr], [RA4676; F, H, Et, F, Bu, i-Pr], [RA4677; F, H, Et, F, Bu, c-Pr], [RA4678; F, H, Et, F, Bu, Bu], [ RA4679; F, H, Et, F, Bu, i-Bu], [RA4680; F, H, Et, F, Bu, t-Bu], [RA4681; F, H, Et, F, Bu, c- PrCH ₂ ], [RA4682; F, H, Et, F, Bu, Ph], [RA4683; F, H, Et, F, Bu, Bn], [RA4684; F, H, Et, F, Bu, CF ₃ ], [RA4685; F, H, Et, F, Bu, CF ₃ CH ₂ ], [RA4686; F, H, Et, F, Bu, CF ₃ CF ₂ ], [RA4687; F, H, Et, F, Bu, CF ₂ H], [RA4688; F, H, Et, F, Bu, CF ₂ HCH ₂ ], [RA4689; F, H, Et, Cl, Bu, Me], [RA4690; F, H , Et, Cl, Bu, Et], [RA4691; F, H, Et, Cl, Bu, Pr], [RA4692; F, H, Et, Cl, Bu, i-Pr], [RA4693; F, H , Et, Cl, Bu, c-Pr], [RA4694; F, H, Et, Cl, Bu, Bu], [RA4695; F, H, Et, Cl, Bu, i-Bu], [RA4696; F , H, Et, Cl, Bu, t-Bu], [RA4697; F, H, Et, Cl, Bu, c-PrCH ₂ ], [RA4698; F, H, Et, Cl, Bu, Ph], [ RA4699; F, H, Et, Cl, Bu, Bn], [RA4700; F, H, Et, Cl, Bu, CF ₃ ], [RA4701; F, H, Et, Cl, Bu, CF ₃ CH ₂ ] , [RA4702; F, H, Et, Cl, Bu, CF ₃ CF ₂ ], [RA4703; F, H, Et, Cl, Bu, CF ₂ H], [RA4704; F, H, Et, Cl, Bu , CF ₂ HCH ₂ ], [RA4705; F, H, F, H, Bu, Me], [RA4706; F, H, F, H, Bu, Et], [RA4707; F, H, F, H, Bu, Pr], [RA4708; F, H, F, H, Bu, i-Pr], [RA4709; F, H, F, H, Bu, c-Pr], [RA4710; F, H, F, H, Bu, Bu], [RA4711; F, H, F, H, Bu, i-Bu], [RA4712; F, H, F, H, Bu, t-Bu], [ RA4713; F, H, F, H, Bu, c-PrCH ₂ ], [RA4714; F, H, F, H, Bu, Ph], [RA4715; F, H, F, H, Bu, Bn], [RA4716; F, H, F, H, Bu, CF ₃ ], [RA4717; F, H, F, H, Bu, CF ₃ CH ₂ ], [RA4718; F, H, F, H, Bu, CF ₃ CF ₂ ], [RA4719; F, H, F, H, Bu, CF ₂ H], [RA4720; F, H, F, H, Bu, CF ₂ HCH ₂ ], [RA4721; F, H, F , F, Bu, Me], [RA4722; F, H, F, F, Bu, Et], [RA4723; F, H, F, F, Bu, Pr], [RA4724; F, H, F, F , Bu, i-Pr], [RA4725; F, H, F, F, Bu, c-Pr], [RA4726; F, H, F, F, Bu, Bu], [RA4727; F, H, F , F, Bu, i-Bu], [RA4728; F, H, F, F, Bu, t-Bu], [RA4729; F, H, F, F, Bu, c-PrCH ₂ ], [RA4730; F, H, F, F, Bu, Ph], [RA4731; F, H, F, F, Bu, Bn], [RA4732; F, H, F, F, Bu, CF ₃ ], [RA4733; F , H, F, F, Bu, CF ₃ CH ₂ ], [RA4734; F, H, F, F, Bu, CF ₃ CF ₂ ], [RA4735; F, H, F, F, Bu, CF ₂ H ], [RA4736; F, H, F, F, Bu, CF ₂ HCH ₂ ], [RA4737; F, H, F, Cl, Bu, Me], [RA4738; F, H, F, Cl, Bu, Et], [RA4739; F, H, F, Cl, Bu, Pr], [RA4740; F, H, F, Cl, Bu, i-Pr], [RA4741; F, H, F, Cl, Bu, c-Pr], [RA4742; F, H, F, Cl, Bu, Bu], [RA4743; F, H, F, Cl, Bu, i-Bu], [RA4744; F, H, F, Cl, Bu, t-Bu], [RA4745; F, H, F, Cl, Bu, c-PrCH ₂ ], [RA4746; F, H, F, Cl, Bu, Ph], [RA4747; F, H, F , Cl, Bu, Bn], [RA4748; F, H, F, Cl, B u, CF ₃ ], [RA4749; F, H, F, Cl, Bu, CF ₃ CH ₂ ], [RA4750; F, H, F, Cl, Bu, CF ₃ CF ₂ ], [RA4751; F, H , F, Cl, Bu, CF ₂ H], [RA4752; F, H, F, Cl, Bu, CF ₂ HCH ₂ ], [RA4753; F, H, Cl, H, Bu, Me], [RA4754; F, H, Cl, H, Bu, Et], [RA4755; F, H, Cl, H, Bu, Pr], [RA4756; F, H, Cl, H, Bu, i-Pr], [RA4757; F, H, Cl, H, Bu, c-Pr], [RA4758; F, H, Cl, H, Bu, Bu], [RA4759; F, H, Cl, H, Bu, i-Bu], [ RA4760; F, H, Cl, H, Bu, t-Bu], [RA4761; F, H, Cl, H, Bu, c-PrCH ₂ ], [RA4762; F, H, Cl, H, Bu, Ph ], [RA4763; F, H, Cl, H, Bu, Bn], [RA4764; F, H, Cl, H, Bu, CF ₃ ], [RA4765; F, H, Cl, H, Bu, CF ₃ CH ₂ ], [RA4766; F, H, Cl, H, Bu, CF ₃ CF ₂ ], [RA4767; F, H, Cl, H, Bu, CF ₂ H], [RA4768; F, H, Cl, H, Bu, CF ₂ HCH ₂ ], [RA4769; F, H, Cl, Cl, Bu, Me], [RA4770; F, H, Cl, Cl, Bu, Et], [RA4771; F, H, Cl , Cl, Bu, Pr], [RA4772; F, H, Cl, Cl, Bu, i-Pr], [RA4773; F, H, Cl, Cl, Bu, c-Pr], [RA4774; F, H , Cl, Cl, Bu, Bu], [RA4775; F, H, Cl, Cl, Bu, i-Bu], [RA4776; F, H, Cl, Cl, Bu, t-Bu], [RA4777; F , H, Cl, Cl, Bu, c-PrCH ₂ ], [RA4778; F, H, Cl, Cl, Bu, Ph], [RA4779; F, H, Cl, Cl, Bu, Bn], [RA4780; F, H, Cl, Cl, Bu, CF ₃ ], [RA4781; F, H, Cl, Cl, Bu, CF ₃ CH ₂ ], [RA4782; F, H, Cl, Cl, Bu, CF ₃ CF ₂ ], [RA4783; F, H, Cl, Cl, Bu, CF ₂ H], [RA4784; F, H, Cl, Cl, Bu, C F ₂ HCH ₂ ], [RA4785; F, H, Me, H, i-Pr, Me], [RA4786; F, H, Me, H, i-Pr, Et], [RA4787; F, H, Me , H, i-Pr, Pr], [RA4788; F, H, Me, H, i-Pr, i-Pr], [RA4789; F, H, Me, H, i-Pr, c-Pr], [RA4790; F, H, Me, H, i-Pr, Bu], [RA4791; F, H, Me, H, i-Pr, i-Bu], [RA4792; F, H, Me, H, i -Pr, t-Bu], [RA4793; F, H, Me, H, i-Pr, c-PrCH ₂ ], [RA4794; F, H, Me, H, i-Pr, Ph], [RA4795; F, H, Me, H, i-Pr, Bn], [RA4796; F, H, Me, H, i-Pr, CF ₃ ], [RA4797; F, H, Me, H, i-Pr, CF ₃ CH ₂ ], [RA4798; F, H, Me, H, i-Pr, CF ₃ CF ₂ ], [RA4799; F, H, Me, H, i-Pr, CF ₂ H], [RA4800; F , H, Me, H, i-Pr, CF ₂ HCH ₂ ],

[RA4801; F, H, Me, Me, i-Pr, Me], [RA4802; F, H, Me, Me, i-Pr, Et], [RA4803; F, H, Me, Me, i-Pr , Pr], [RA4804; F, H, Me, Me, i-Pr, i-Pr], [RA4805; F, H, Me, Me, i-Pr, c-Pr], [RA4806; F, H , Me, Me, i-Pr, Bu], [RA4807; F, H, Me, Me, i-Pr, i-Bu], [RA4808; F, H, Me, Me, i-Pr, t-Bu ], [RA4809; F, H, Me, Me, i-Pr, c-PrCH ₂ ], [RA4810; F, H, Me, Me, i-Pr, Ph], [RA4811; F, H, Me, Me, i-Pr, Bn], [RA4812; F, H, Me, Me, i-Pr, CF ₃ ], [RA4813; F, H, Me, Me, i-Pr, CF ₃ CH ₂ ], [ RA4814; F, H, Me, Me, i-Pr, CF ₃ CF ₂ ], [RA4815; F, H, Me, Me, i-Pr, CF ₂ H], [RA4816; F, H, Me, Me , i-Pr, CF ₂ HCH ₂ ], [RA4817; F, H, Me, Et, i-Pr, Me], [RA4818; F, H, Me, Et, i-Pr, Et], [RA4819; F, H, Me, Et, i-Pr, Pr], [RA4820; F, H, Me, Et, i-Pr, i-Pr], [RA4821; F, H, Me, Et, i-Pr, c-Pr], [RA4822; F, H, Me, Et, i-Pr, Bu], [RA4823; F, H, Me, Et, i-Pr, i-Bu], [RA4824; F, H, Me, Et, i-Pr, t-Bu], [RA4825; F, H, Me, Et, i-Pr, c-PrCH ₂ ], [RA4826; F, H, Me, Et, i-Pr, Ph ], [RA4827; F, H, Me, Et, i-Pr, Bn], [RA4828; F, H, Me, Et, i-Pr, CF ₃ ], [RA4829; F, H, Me, Et, i-Pr, CF ₃ CH ₂ ], [RA4830; F, H, Me, Et, i-Pr, CF ₃ CF ₂ ], [RA4831; F, H, Me, Et, i-Pr, CF ₂ H] , [RA4832; F, H, Me, Et, i-Pr, CF ₂ HCH ₂ ], [RA4833; F, H, Me, F, i-Pr, Me], [RA4834; F, H, Me, F , i-Pr, Et], [RA4835; F, H, Me, F, i-Pr, Pr], [RA4836; F, H, Me, F, i-Pr, i-Pr], [RA4837; F , H, Me, F, i-Pr, c-Pr], [RA4838; F, H, Me, F, i-Pr, Bu], [RA4839; F, H, Me, F, i-Pr, i -Bu], [RA4840; F, H, Me, F, i-Pr, t-Bu], [RA4841; F, H, Me, F, i-Pr, c-PrCH ₂ ], [RA4842; F, H, Me, F, i-Pr, Ph], [RA4843; F, H, Me, F, i-Pr, Bn], [RA4844; F, H, Me, F, i-Pr, CF ₃ ], [RA4845; F, H, Me, F, i-Pr, CF ₃ CH ₂ ], [RA4846; F, H, Me, F, i-Pr, CF ₃ CF ₂ ], [RA4847; F, H, Me , F, i-Pr, CF ₂ H], [RA4848; F, H, Me, F, i-Pr, CF ₂ HCH ₂ ], [RA4849; F, H, Me, Cl, i-Pr, Me] , [RA4850; F, H, Me, Cl, i-Pr, Et], [RA4851; F, H, Me, Cl, i-Pr, Pr], [RA4852; F, H, Me, Cl, i- Pr, i-Pr], [RA4853; F, H, Me, Cl, i-Pr, c-Pr], [RA4854; F, H, Me, Cl, i-Pr, Bu], [RA4855; F, H, Me, Cl, i-Pr, i-Bu], [RA4856; F, H, Me, Cl, i-Pr, t-Bu], [RA4857; F, H, Me, Cl, i-Pr, c-PrCH ₂ ], [RA4858; F, H, Me, Cl, i-Pr, Ph], [RA4859; F, H, Me, Cl, i-Pr, Bn], [RA4860; F, H, Me , Cl, i-Pr, CF ₃ ], [RA4861; F, H, Me, Cl, i-Pr, CF ₃ CH ₂ ], [RA4862; F, H, Me, Cl, i-Pr, CF ₃ CF ₂ ], [RA4863; F, H, Me, Cl, i-Pr, CF ₂ H], [RA4864; F, H, Me, Cl, i-Pr, CF ₂ HCH ₂ ], [RA4865; F, H , Et, H, i-Pr, Me], [RA4866; F, H, Et, H, i-Pr, Et], [RA4867; F, H, Et, H, i-Pr, Pr], [RA4868 ; F, H, Et, H, i-Pr, i-Pr], [RA4869; F, H, Et, H, i-Pr, c-Pr], [RA4870; F, H, Et, H, i-Pr, Bu], [RA4871; F, H, Et, H, i-Pr, i-Bu], [RA4872; F, H, Et, H, i-Pr, t-Bu], [RA4873; F, H, Et, H, i-Pr, c- PrCH ₂ ], [RA4874; F, H, Et, H, i-Pr, Ph], [RA4875; F, H, Et, H, i-Pr, Bn], [RA4876; F, H, Et, H , i-Pr, CF ₃ ], [RA4877; F, H, Et, H, i-Pr, CF ₃ CH ₂ ], [RA4878; F, H, Et, H, i-Pr, CF ₃ CF ₂ ] , [RA4879; F, H, Et, H, i-Pr, CF ₂ H], [RA4880; F, H, Et, H, i-Pr, CF ₂ HCH ₂ ], [RA4881; F, H, Et , F, i-Pr, Me], [RA4882; F, H, Et, F, i-Pr, Et], [RA4883; F, H, Et, F, i-Pr, Pr], [RA4884; F , H, Et, F, i-Pr, i-Pr], [RA4885; F, H, Et, F, i-Pr, c-Pr], [RA4886; F, H, Et, F, i-Pr , Bu], [RA4887; F, H, Et, F, i-Pr, i-Bu], [RA4888; F, H, Et, F, i-Pr, t-Bu], [RA4889; F, H , Et, F, i-Pr, c-PrCH ₂ ], [RA4890; F, H, Et, F, i-Pr, Ph], [RA4891; F, H, Et, F, i-Pr, Bn] , [RA4892; F, H, Et, F, i-Pr, CF ₃ ], [RA4893; F, H, Et, F, i-Pr, CF ₃ CH ₂ ], [RA4894; F, H, Et, F, i-Pr, CF ₃ CF ₂ ], [RA4895; F, H, Et, F, i-Pr, CF ₂ H], [RA4896; F, H, Et, F, i-Pr, CF ₂ HCH ₂ ], [RA4897; F, H, Et, Cl, i-Pr, Me], [RA4898; F, H, Et, Cl, i-Pr, Et], [RA4899; F, H, Et, Cl, i-Pr, Pr], [RA4900; F, H, Et, Cl, i-Pr, i-Pr], [RA4901; F, H, Et, Cl, i-Pr, c-Pr], [RA4902; F, H, Et, Cl, i-Pr, Bu], [RA4903; F, H, Et, Cl, i-Pr, i-Bu], [RA4904; F, H, Et, Cl, i-Pr, t-Bu], [RA4905; F, H, Et, Cl, i- Pr, c-PrCH ₂ ], [RA4906; F, H, Et, Cl, i-Pr, Ph], [RA4907; F, H, Et, Cl, i-Pr, Bn], [RA4908; F, H , Et, Cl, i-Pr, CF ₃ ], [RA4909; F, H, Et, Cl, i-Pr, CF ₃ CH ₂ ], [RA4910; F, H, Et, Cl, i-Pr, CF ₃ CF ₂ ], [RA4911; F, H, Et, Cl, i-Pr, CF ₂ H], [RA4912; F, H, Et, Cl, i-Pr, CF ₂ HCH ₂ ], [RA4913; F , H, F, H, i-Pr, Me], [RA4914; F, H, F, H, i-Pr, Et], [RA4915; F, H, F, H, i-Pr, Pr], [RA4916; F, H, F, H, i-Pr, i-Pr], [RA4917; F, H, F, H, i-Pr, c-Pr], [RA4918; F, H, F, H , i-Pr, Bu], [RA4919; F, H, F, H, i-Pr, i-Bu], [RA4920; F, H, F, H, i-Pr, t-Bu], [RA4921 ; F, H, F, H, i-Pr, c-PrCH ₂ ], [RA4922; F, H, F, H, i-Pr, Ph], [RA4923; F, H, F, H, i- Pr, Bn], [RA4924; F, H, F, H, i-Pr, CF ₃ ], [RA4925; F, H, F, H, i-Pr, CF ₃ CH ₂ ], [RA4926; F, H, F, H, i-Pr, CF ₃ CF ₂ ], [RA4927; F, H, F, H, i-Pr, CF ₂ H], [RA4928; F, H, F, H, i-Pr , CF ₂ HCH ₂ ], [RA4929; F, H, F, F, i-Pr, Me], [RA4930; F, H, F, F, i-Pr, Et], [RA4931; F, H, F, F, i-Pr, Pr], [RA4932; F, H, F, F, i-Pr, i-Pr], [RA4933; F, H, F, F, i-Pr, c-Pr] , [RA4934; F, H, F, F, i-Pr, Bu], [RA4935; F, H, F, F, i-Pr, i-Bu], [RA4936; F, H, F, F, i-Pr, t-Bu], [RA4937; F, H, F, F, i-Pr, c-PrCH ₂ ], [RA4938; F, H, F, F, i-Pr, Ph], [RA4939; F, H, F, F, i-Pr, Bn], [RA4940; F, H, F, F, i-Pr, CF ₃ ], [RA4941; F, H, F, F, i-Pr, CF ₃ CH ₂ ], [RA4942; F, H, F, F, i-Pr, CF ₃ CF ₂ ], [RA4943; F, H , F, F, i-Pr, CF ₂ H], [RA4944; F, H, F, F, i-Pr, CF ₂ HCH ₂ ], [RA4945; F, H, F, Cl, i-Pr, Me], [RA4946; F, H, F, Cl, i-Pr, Et], [RA4947; F, H, F, Cl, i-Pr, Pr], [RA4948; F, H, F, Cl, i-Pr, i-Pr], [RA4949; F, H, F, Cl, i-Pr, c-Pr], [RA4950; F, H, F, Cl, i-Pr, Bu], [RA4951; F, H, F, Cl, i-Pr, i-Bu], [RA4952; F, H, F, Cl, i-Pr, t-Bu], [RA4953; F, H, F, Cl, i- Pr, c-PrCH ₂ ], [RA4954; F, H, F, Cl, i-Pr, Ph], [RA4955; F, H, F, Cl, i-Pr, Bn], [RA4956; F, H , F, Cl, i-Pr, CF ₃ ], [RA4957; F, H, F, Cl, i-Pr, CF ₃ CH ₂ ], [RA4958; F, H, F, Cl, i-Pr, CF ₃ CF ₂ ], [RA4959; F, H, F, Cl, i-Pr, CF ₂ H], [RA4960; F, H, F, Cl, i-Pr, CF ₂ HCH ₂ ], [RA4961; F , H, Cl, H, i-Pr, Me], [RA4962; F, H, Cl, H, i-Pr, Et], [RA4963; F, H, Cl, H, i-Pr, Pr], [RA4964; F, H, Cl, H, i-Pr, i-Pr], [RA4965; F, H, Cl, H, i-Pr, c-Pr], [RA4966; F, H, Cl, H , i-Pr, Bu], [RA4967; F, H, Cl, H, i-Pr, i-Bu], [RA4968; F, H, Cl, H, i-Pr, t-Bu], [RA4969 ; F, H, Cl, H, i-Pr, c-PrCH ₂ ], [RA4970; F, H, Cl, H, i-Pr, Ph], [RA4971; F, H, Cl, H, i- Pr, Bn], [RA4972; F, H, Cl, H, i-Pr, CF ₃ ], [RA4973; F, H, Cl, H, i-Pr, CF ₃ CH ₂ ], [RA4974; F, H, Cl, H, i-Pr, CF ₃ CF ₂ ], [RA4975; F, H, Cl, H, i-Pr, CF ₂ H], [RA4976; F, H, Cl, H, i-Pr, CF ₂ HCH ₂ ], [RA4977; F, H, Cl, Cl, i-Pr, Me], [RA4978 ; F, H, Cl, Cl, i-Pr, Et], [RA4979; F, H, Cl, Cl, i-Pr, Pr], [RA4980; F, H, Cl, Cl, i-Pr, i -Pr], [RA4981; F, H, Cl, Cl, i-Pr, c-Pr], [RA4982; F, H, Cl, Cl, i-Pr, Bu], [RA4983; F, H, Cl , Cl, i-Pr, i-Bu], [RA4984; F, H, Cl, Cl, i-Pr, t-Bu], [RA4985; F, H, Cl, Cl, i-Pr, c-PrCH ₂ ], [RA4986; F, H, Cl, Cl, i-Pr, Ph], [RA4987; F, H, Cl, Cl, i-Pr, Bn], [RA4988; F, H, Cl, Cl, i-Pr, CF ₃ ], [RA4989; F, H, Cl, Cl, i-Pr, CF ₃ CH ₂ ], [RA4990; F, H, Cl, Cl, i-Pr, CF ₃ CF ₂ ], [RA4991; F, H, Cl, Cl, i-Pr, CF ₂ H], [RA4992; F, H, Cl, Cl, i-Pr, CF ₂ HCH ₂ ], [RA4993; F, H, Me, H, c-Pr, Me], [RA4994; F, H, Me, H, c-Pr, Et], [RA4995; F, H, Me, H, c-Pr, Pr], [RA4996; F, H, Me, H, c-Pr, i-Pr], [RA4997; F, H, Me, H, c-Pr, c-Pr], [RA4998; F, H, Me, H, c-Pr, Bu], [RA4999; F, H, Me, H, c-Pr, i-Bu], [RA5000; F, H, Me, H, c-Pr, t-Bu],

[RA5001; F, H, Me, H, c-Pr, c-PrCH ₂ ], [RA5002; F, H, Me, H, c-Pr, Ph], [RA5003; F, H, Me, H, c-Pr, Bn], [RA5004; F, H, Me, H, c-Pr, CF ₃ ], [RA5005; F, H, Me, H, c-Pr, CF ₃ CH ₂ ], [RA5006; F, H, Me, H, c-Pr, CF ₃ CF ₂ ], [RA5007; F, H, Me, H, c-Pr, CF ₂ H], [RA5008; F, H, Me, H, c -Pr, CF ₂ HCH ₂ ], [RA5009; F, H, Me, Me, c-Pr, Me], [RA5010; F, H, Me, Me, c-Pr, Et], [RA5011; F, H, Me, Me, c-Pr, Pr], [RA5012; F, H, Me, Me, c-Pr, i-Pr], [RA5013; F, H, Me, Me, c-Pr, c- Pr], [RA5014; F, H, Me, Me, c-Pr, Bu], [RA5015; F, H, Me, Me, c-Pr, i-Bu], [RA5016; F, H, Me, Me, c-Pr, t-Bu], [RA5017; F, H, Me, Me, c-Pr, c-PrCH ₂ ], [RA5018; F, H, Me, Me, c-Pr, Ph], [RA5019; F, H, Me, Me, c-Pr, Bn], [RA5020; F, H, Me, Me, c-Pr, CF ₃ ], [RA5021; F, H, Me, Me, c- Pr, CF ₃ CH ₂ ], [RA5022; F, H, Me, Me, c-Pr, CF ₃ CF ₂ ], [RA5023; F, H, Me, Me, c-Pr, CF ₂ H], [ RA5024; F, H, Me, Me, c-Pr, CF ₂ HCH ₂ ], [RA5025; F, H, Me, Et, c-Pr, Me], [RA5026; F, H, Me, Et, c -Pr, Et], [RA5027; F, H, Me, Et, c-Pr, Pr], [RA5028; F, H, Me, Et, c-Pr, i-Pr], [RA5029; F, H , Me, Et, c-Pr, c-Pr], [RA5030; F, H, Me, Et, c-Pr, Bu], [RA5031; F, H, Me, Et, c-Pr, i-Bu ], [RA5032; F, H, Me, Et, c-Pr, t-Bu], [RA5033; F, H, Me, Et, c-Pr, c-PrCH ₂ ], [RA5034; F, H, Me, E t, c-Pr, Ph], [RA5035; F, H, Me, Et, c-Pr, Bn], [RA5036; F, H, Me, Et, c-Pr, CF ₃ ], [RA5037; F , H, Me, Et, c-Pr, CF ₃ CH ₂ ], [RA5038; F, H, Me, Et, c-Pr, CF ₃ CF ₂ ], [RA5039; F, H, Me, Et, c -Pr, CF ₂ H], [RA5040; F, H, Me, Et, c-Pr, CF ₂ HCH ₂ ], [RA5041; F, H, Me, F, c-Pr, Me], [RA5042; F, H, Me, F, c-Pr, Et], [RA5043; F, H, Me, F, c-Pr, Pr], [RA5044; F, H, Me, F, c-Pr, i- Pr], [RA5045; F, H, Me, F, c-Pr, c-Pr], [RA5046; F, H, Me, F, c-Pr, Bu], [RA5047; F, H, Me, F, c-Pr, i-Bu], [RA5048; F, H, Me, F, c-Pr, t-Bu], [RA5049; F, H, Me, F, c-Pr, c-PrCH ₂ ], [RA5050; F, H, Me, F, c-Pr, Ph], [RA5051; F, H, Me, F, c-Pr, Bn], [RA5052; F, H, Me, F, c -Pr, CF ₃ ], [RA5053; F, H, Me, F, c-Pr, CF ₃ CH ₂ ], [RA5054; F, H, Me, F, c-Pr, CF ₃ CF ₂ ], [ RA5055; F, H, Me, F, c-Pr, CF ₂ H], [RA5056; F, H, Me, F, c-Pr, CF ₂ HCH ₂ ], [RA5057; F, H, Me, Cl , c-Pr, Me], [RA5058; F, H, Me, Cl, c-Pr, Et], [RA5059; F, H, Me, Cl, c-Pr, Pr], [RA5060; F, H , Me, Cl, c-Pr, i-Pr], [RA5061; F, H, Me, Cl, c-Pr, c-Pr], [RA5062; F, H, Me, Cl, c-Pr, Bu ], [RA5063; F, H, Me, Cl, c-Pr, i-Bu], [RA5064; F, H, Me, Cl, c-Pr, t-Bu], [RA5065; F, H, Me , Cl, c-Pr, c-PrCH ₂ ], [RA5066; F, H, Me, Cl, c-Pr, Ph], [RA5067; F, H, Me, Cl, c-Pr, Bn], [ RA5068; F, H, Me, Cl, c- Pr, CF ₃ ], [RA5069; F, H, Me, Cl, c-Pr, CF ₃ CH ₂ ], [RA5070; F, H, Me, Cl, c-Pr, CF ₃ CF ₂ ], [RA5071 ; F, H, Me, Cl, c-Pr, CF ₂ H], [RA5072; F, H, Me, Cl, c-Pr, CF ₂ HCH ₂ ], [RA5073; F, H, Et, H, c-Pr, Me], [RA5074; F, H, Et, H, c-Pr, Et], [RA5075; F, H, Et, H, c-Pr, Pr], [RA5076; F, H, Et, H, c-Pr, i-Pr], [RA5077; F, H, Et, H, c-Pr, c-Pr], [RA5078; F, H, Et, H, c-Pr, Bu] , [RA5079; F, H, Et, H, c-Pr, i-Bu], [RA5080; F, H, Et, H, c-Pr, t-Bu], [RA5081; F, H, Et, H, c-Pr, c-PrCH ₂ ], [RA5082; F, H, Et, H, c-Pr, Ph], [RA5083; F, H, Et, H, c-Pr, Bn], [RA5084 ; F, H, Et, H, c-Pr, CF ₃ ], [RA5085; F, H, Et, H, c-Pr, CF ₃ CH ₂ ], [RA5086; F, H, Et, H, c -Pr, CF ₃ CF ₂ ], [RA5087; F, H, Et, H, c-Pr, CF ₂ H], [RA5088; F, H, Et, H, c-Pr, CF ₂ HCH ₂ ], [RA5089; F, H, Et, F, c-Pr, Me], [RA5090; F, H, Et, F, c-Pr, Et], [RA5091; F, H, Et, F, c-Pr , Pr], [RA5092; F, H, Et, F, c-Pr, i-Pr], [RA5093; F, H, Et, F, c-Pr, c-Pr], [RA5094; F, H , Et, F, c-Pr, Bu], [RA5095; F, H, Et, F, c-Pr, i-Bu], [RA5096; F, H, Et, F, c-Pr, t-Bu ], [RA5097; F, H, Et, F, c-Pr, c-PrCH ₂ ], [RA5098; F, H, Et, F, c-Pr, Ph], [RA5099; F, H, Et, F, c-Pr, Bn], [RA5100; F, H, Et, F, c-Pr, CF ₃ ], [RA5101; F, H, Et, F, c-Pr, CF ₃ CH ₂ ], [ RA5102; F, H, Et, F, c-Pr, CF ₃ CF ₂ ], [RA5103; F, H, Et, F, c-Pr, CF ₂ H], [RA5104; F, H, Et, F, c-Pr, CF ₂ HCH ₂ ], [RA5105; F, H, Et, Cl, c-Pr, Me], [RA5106; F, H, Et, Cl, c-Pr, Et], [RA5107; F, H, Et, Cl, c-Pr, Pr], [ RA5108; F, H, Et, Cl, c-Pr, i-Pr], [RA5109; F, H, Et, Cl, c-Pr, c-Pr], [RA5110; F, H, Et, Cl, c-Pr, Bu], [RA5111; F, H, Et, Cl, c-Pr, i-Bu], [RA5112; F, H, Et, Cl, c-Pr, t-Bu], [RA5113; F, H, Et, Cl, c-Pr, c-PrCH ₂ ], [RA5114; F, H, Et, Cl, c-Pr, Ph], [RA5115; F, H, Et, Cl, c-Pr , Bn], [RA5116; F, H, Et, Cl, c-Pr, CF ₃ ], [RA5117; F, H, Et, Cl, c-Pr, CF ₃ CH ₂ ], [RA5118; F, H , Et, Cl, c-Pr, CF ₃ CF ₂ ], [RA5119; F, H, Et, Cl, c-Pr, CF ₂ H], [RA5120; F, H, Et, Cl, c-Pr, CF ₂ HCH ₂ ], [RA5121; F, H, F, H, c-Pr, Me], [RA5122; F, H, F, H, c-Pr, Et], [RA5123; F, H, F , H, c-Pr, Pr], [RA5124; F, H, F, H, c-Pr, i-Pr], [RA5125; F, H, F, H, c-Pr, c-Pr], [RA5126; F, H, F, H, c-Pr, Bu], [RA5127; F, H, F, H, c-Pr, i-Bu], [RA5128; F, H, F, H, c -Pr, t-Bu], [RA5129; F, H, F, H, c-Pr, c-PrCH ₂ ], [RA5130; F, H, F, H, c-Pr, Ph], [RA5131; F, H, F, H, c-Pr, Bn], [RA5132; F, H, F, H, c-Pr, CF ₃ ], [RA5133; F, H, F, H, c-Pr, CF ₃ CH ₂ ], [RA5134; F, H, F, H, c-Pr, CF ₃ CF ₂ ], [RA5135; F, H, F, H, c-Pr, CF ₂ H], [RA5136; F , H, F, H, c-Pr, CF ₂ HCH ₂ ], [ RA5137; F, H, F, F, c-Pr, Me], [RA5138; F, H, F, F, c-Pr, Et], [RA5139; F, H, F, F, c-Pr, Pr], [RA5140; F, H, F, F, c-Pr, i-Pr], [RA5141; F, H, F, F, c-Pr, c-Pr], [RA5142; F, H, F, F, c-Pr, Bu], [RA5143; F, H, F, F, c-Pr, i-Bu], [RA5144; F, H, F, F, c-Pr, t-Bu] , [RA5145; F, H, F, F, c-Pr, c-PrCH ₂ ], [RA5146; F, H, F, F, c-Pr, Ph], [RA5147; F, H, F, F , c-Pr, Bn], [RA5148; F, H, F, F, c-Pr, CF ₃ ], [RA5149; F, H, F, F, c-Pr, CF ₃ CH ₂ ], [RA5150 ; F, H, F, F, c-Pr, CF ₃ CF ₂ ], [RA5151; F, H, F, F, c-Pr, CF ₂ H], [RA5152; F, H, F, F, c-Pr, CF ₂ HCH ₂ ], [RA5153; F, H, F, Cl, c-Pr, Me], [RA5154; F, H, F, Cl, c-Pr, Et], [RA5155; F , H, F, Cl, c-Pr, Pr], [RA5156; F, H, F, Cl, c-Pr, i-Pr], [RA5157; F, H, F, Cl, c-Pr, c -Pr], [RA5158; F, H, F, Cl, c-Pr, Bu], [RA5159; F, H, F, Cl, c-Pr, i-Bu], [RA5160; F, H, F , Cl, c-Pr, t-Bu], [RA5161; F, H, F, Cl, c-Pr, c-PrCH ₂ ], [RA5162; F, H, F, Cl, c-Pr, Ph] , [RA5163; F, H, F, Cl, c-Pr, Bn], [RA5164; F, H, F, Cl, c-Pr, CF ₃ ], [RA5165; F, H, F, Cl, c -Pr, CF ₃ CH ₂ ], [RA5166; F, H, F, Cl, c-Pr, CF ₃ CF ₂ ], [RA5167; F, H, F, Cl, c-Pr, CF ₂ H], [RA5168; F, H, F, Cl, c-Pr, CF ₂ HCH ₂ ], [RA5169; F, H, Cl, H, c-Pr, Me], [RA5170; F, H, Cl, H, c-Pr, Et], [RA5171; F, H, Cl, H, c-Pr, Pr], [RA5172; F, H, C l, H, c-Pr, i-Pr], [RA5173; F, H, Cl, H, c-Pr, c-Pr], [RA5174; F, H, Cl, H, c-Pr, Bu] , [RA5175; F, H, Cl, H, c-Pr, i-Bu], [RA5176; F, H, Cl, H, c-Pr, t-Bu], [RA5177; F, H, Cl, H, c-Pr, c-PrCH ₂ ], [RA5178; F, H, Cl, H, c-Pr, Ph], [RA5179; F, H, Cl, H, c-Pr, Bn], [RA5180 ; F, H, Cl, H, c-Pr, CF ₃ ], [RA5181; F, H, Cl, H, c-Pr, CF ₃ CH ₂ ], [RA5182; F, H, Cl, H, c -Pr, CF ₃ CF ₂ ], [RA5183; F, H, Cl, H, c-Pr, CF ₂ H], [RA5184; F, H, Cl, H, c-Pr, CF ₂ HCH ₂ ], [RA5185; F, H, Cl, Cl, c-Pr, Me], [RA5186; F, H, Cl, Cl, c-Pr, Et], [RA5187; F, H, Cl, Cl, c-Pr , Pr], [RA5188; F, H, Cl, Cl, c-Pr, i-Pr], [RA5189; F, H, Cl, Cl, c-Pr, c-Pr], [RA5190; F, H , Cl, Cl, c-Pr, Bu], [RA5191; F, H, Cl, Cl, c-Pr, i-Bu], [RA5192; F, H, Cl, Cl, c-Pr, t-Bu ], [RA5193; F, H, Cl, Cl, c-Pr, c-PrCH ₂ ], [RA5194; F, H, Cl, Cl, c-Pr, Ph], [RA5195; F, H, Cl, Cl, c-Pr, Bn], [RA5196; F, H, Cl, Cl, c-Pr, CF ₃ ], [RA5197; F, H, Cl, Cl, c-Pr, CF ₃ CH ₂ ], [ RA5198; F, H, Cl, Cl, c-Pr, CF ₃ CF ₂ ], [RA5199; F, H, Cl, Cl, c-Pr, CF ₂ H], [RA5200; F, H, Cl, Cl , c-Pr, CF ₂ HCH ₂ ],

[RA5201; F, H, Me, H, i-Bu, Me], [RA5202; F, H, Me, H, i-Bu, Et], [RA5203; F, H, Me, H, i-Bu , Pr], [RA5204; F, H, Me, H, i-Bu, i-Pr], [RA5205; F, H, Me, H, i-Bu, c-Pr], [RA5206; F, H , Me, H, i-Bu, Bu], [RA5207; F, H, Me, H, i-Bu, i-Bu], [RA5208; F, H, Me, H, i-Bu, t-Bu ], [RA5209; F, H, Me, H, i-Bu, c-PrCH ₂ ], [RA5210; F, H, Me, H, i-Bu, Ph], [RA5211; F, H, Me, H, i-Bu, Bn], [RA5212; F, H, Me, H, i-Bu, CF ₃ ], [RA5213; F, H, Me, H, i-Bu, CF ₃ CH ₂ ], [ RA5214; F, H, Me, H, i-Bu, CF ₃ CF ₂ ], [RA5215; F, H, Me, H, i-Bu, CF ₂ H], [RA5216; F, H, Me, H , i-Bu, CF ₂ HCH ₂ ], [RA5217; F, H, Me, Me, i-Bu, Me], [RA5218; F, H, Me, Me, i-Bu, Et], [RA5219; F, H, Me, Me, i-Bu, Pr], [RA5220; F, H, Me, Me, i-Bu, i-Pr], [RA5221; F, H, Me, Me, i-Bu, c-Pr], [RA5222; F, H, Me, Me, i-Bu, Bu], [RA5223; F, H, Me, Me, i-Bu, i-Bu], [RA5224; F, H, Me, Me, i-Bu, t-Bu], [RA5225; F, H, Me, Me, i-Bu, c-PrCH ₂ ], [RA5226; F, H, Me, Me, i-Bu, Ph ], [RA5227; F, H, Me, Me, i-Bu, Bn], [RA5228; F, H, Me, Me, i-Bu, CF ₃ ], [RA5229; F, H, Me, Me, i-Bu, CF ₃ CH ₂ ], [RA5230; F, H, Me, Me, i-Bu, CF ₃ CF ₂ ], [RA5231; F, H, Me, Me, i-Bu, CF ₂ H] , [RA5232; F, H, Me, Me, i-Bu, CF ₂ HCH ₂ ], [RA5233; F, H, Me, Et, i-Bu, Me], [RA5234; F, H, Me, Et , i-Bu, Et], [RA5 235; F, H, Me, Et, i-Bu, Pr], [RA5236; F, H, Me, Et, i-Bu, i-Pr], [RA5237; F, H, Me, Et, i- Bu, c-Pr], [RA5238; F, H, Me, Et, i-Bu, Bu], [RA5239; F, H, Me, Et, i-Bu, i-Bu], [RA5240; F, H, Me, Et, i-Bu, t-Bu], [RA5241; F, H, Me, Et, i-Bu, c-PrCH ₂ ], [RA5242; F, H, Me, Et, i-Bu , Ph], [RA5243; F, H, Me, Et, i-Bu, Bn], [RA5244; F, H, Me, Et, i-Bu, CF ₃ ], [RA5245; F, H, Me, Et, i-Bu, CF ₃ CH ₂ ], [RA5246; F, H, Me, Et, i-Bu, CF ₃ CF ₂ ], [RA5247; F, H, Me, Et, i-Bu, CF ₂ H], [RA5248; F, H, Me, Et, i-Bu, CF ₂ HCH ₂ ], [RA5249; F, H, Me, F, i-Bu, Me], [RA5250; F, H, Me , F, i-Bu, Et], [RA5251; F, H, Me, F, i-Bu, Pr], [RA5252; F, H, Me, F, i-Bu, i-Pr], [RA5253 ; F, H, Me, F, i-Bu, c-Pr], [RA5254; F, H, Me, F, i-Bu, Bu], [RA5255; F, H, Me, F, i-Bu , i-Bu], [RA5256; F, H, Me, F, i-Bu, t-Bu], [RA5257; F, H, Me, F, i-Bu, c-PrCH ₂ ], [RA5258; F, H, Me, F, i-Bu, Ph], [RA5259; F, H, Me, F, i-Bu, Bn], [RA5260; F, H, Me, F, i-Bu, CF ₃ ], [RA5261; F, H, Me, F, i-Bu, CF ₃ CH ₂ ], [RA5262; F, H, Me, F, i-Bu, CF ₃ CF ₂ ], [RA5263; F, H , Me, F, i-Bu, CF ₂ H], [RA5264; F, H, Me, F, i-Bu, CF ₂ HCH ₂ ], [RA5265; F, H, Me, Cl, i-Bu, Me], [RA5266; F, H, Me, Cl, i-Bu, Et], [RA5267; F, H, Me, Cl, i-Bu, Pr], [RA5268; F, H, Me, Cl, i-Bu, i-Pr], [RA526 9; F, H, Me, Cl, i-Bu, c-Pr], [RA5270; F, H, Me, Cl, i-Bu, Bu], [RA5271; F, H, Me, Cl, i- Bu, i-Bu], [RA5272; F, H, Me, Cl, i-Bu, t-Bu], [RA5273; F, H, Me, Cl, i-Bu, c-PrCH ₂ ], [RA5274 ; F, H, Me, Cl, i-Bu, Ph], [RA5275; F, H, Me, Cl, i-Bu, Bn], [RA5276; F, H, Me, Cl, i-Bu, CF ₃ ], [RA5277; F, H, Me, Cl, i-Bu, CF ₃ CH ₂ ], [RA5278; F, H, Me, Cl, i-Bu, CF ₃ CF ₂ ], [RA5279; F, H, Me, Cl, i-Bu, CF ₂ H], [RA5280; F, H, Me, Cl, i-Bu, CF ₂ HCH ₂ ], [RA5281; F, H, Et, H, i-Bu , Me], [RA5282; F, H, Et, H, i-Bu, Et], [RA5283; F, H, Et, H, i-Bu, Pr], [RA5284; F, H, Et, H , i-Bu, i-Pr], [RA5285; F, H, Et, H, i-Bu, c-Pr], [RA5286; F, H, Et, H, i-Bu, Bu], [RA5287 ; F, H, Et, H, i-Bu, i-Bu], [RA5288; F, H, Et, H, i-Bu, t-Bu], [RA5289; F, H, Et, H, i -Bu, c-PrCH ₂ ], [RA5290; F, H, Et, H, i-Bu, Ph], [RA5291; F, H, Et, H, i-Bu, Bn], [RA5292; F, H, Et, H, i-Bu, CF ₃ ], [RA5293; F, H, Et, H, i-Bu, CF ₃ CH ₂ ], [RA5294; F, H, Et, H, i-Bu, CF ₃ CF ₂ ], [RA5295; F, H, Et, H, i-Bu, CF ₂ H], [RA5296; F, H, Et, H, i-Bu, CF ₂ HCH ₂ ], [RA5297; F, H, Et, F, i-Bu, Me], [RA5298; F, H, Et, F, i-Bu, Et], [RA5299; F, H, Et, F, i-Bu, Pr] , [RA5300; F, H, Et, F, i-Bu, i-Pr], [RA5301; F, H, Et, F, i-Bu, c-Pr], [RA5302; F, H, Et, F, i-Bu, Bu], [RA5303; F, H, Et , F, i-Bu, i-Bu], [RA5304; F, H, Et, F, i-Bu, t-Bu], [RA5305; F, H, Et, F, i-Bu, c-PrCH ₂ ], [RA5306; F, H, Et, F, i-Bu, Ph], [RA5307; F, H, Et, F, i-Bu, Bn], [RA5308; F, H, Et, F, i-Bu, CF ₃ ], [RA5309; F, H, Et, F, i-Bu, CF ₃ CH ₂ ], [RA5310; F, H, Et, F, i-Bu, CF ₃ CF ₂ ], [RA5311; F, H, Et, F, i-Bu, CF ₂ H], [RA5312; F, H, Et, F, i-Bu, CF ₂ HCH ₂ ], [RA5313; F, H, Et, Cl, i-Bu, Me], [RA5314; F, H, Et, Cl, i-Bu, Et], [RA5315; F, H, Et, Cl, i-Bu, Pr], [RA5316; F, H, Et, Cl, i-Bu, i-Pr], [RA5317; F, H, Et, Cl, i-Bu, c-Pr], [RA5318; F, H, Et, Cl, i-Bu, Bu], [RA5319; F, H, Et, Cl, i-Bu, i-Bu], [RA5320; F, H, Et, Cl, i-Bu, t-Bu], [RA5321; F, H, Et, Cl, i-Bu, c-PrCH ₂ ], [RA5322; F, H, Et, Cl, i-Bu, Ph], [RA5323; F, H, Et, Cl, i-Bu, Bn], [RA5324; F, H, Et, Cl, i-Bu, CF ₃ ], [RA5325; F, H, Et, Cl, i-Bu, CF ₃ CH ₂ ], [RA5326; F, H, Et, Cl , i-Bu, CF ₃ CF ₂ ], [RA5327; F, H, Et, Cl, i-Bu, CF ₂ H], [RA5328; F, H, Et, Cl, i-Bu, CF ₂ HCH ₂ ], [RA5329; F, H, F, H, i-Bu, Me], [RA5330; F, H, F, H, i-Bu, Et], [RA5331; F, H, F, H, i -Bu, Pr], [RA5332; F, H, F, H, i-Bu, i-Pr], [RA5333; F, H, F, H, i-Bu, c-Pr], [RA5334; F , H, F, H, i-Bu, Bu], [RA5335; F, H, F, H, i-Bu, i-Bu], [RA5336; F, H, F, H, i-Bu, t -Bu], [RA5337; F, H, F, H, i-Bu, cP rCH ₂ ], [RA5338; F, H, F, H, i-Bu, Ph], [RA5339; F, H, F, H, i-Bu, Bn], [RA5340; F, H, F, H , i-Bu, CF ₃ ], [RA5341; F, H, F, H, i-Bu, CF ₃ CH ₂ ], [RA5342; F, H, F, H, i-Bu, CF ₃ CF ₂ ] , [RA5343; F, H, F, H, i-Bu, CF ₂ H], [RA5344; F, H, F, H, i-Bu, CF ₂ HCH ₂ ], [RA5345; F, H, F , F, i-Bu, Me], [RA5346; F, H, F, F, i-Bu, Et], [RA5347; F, H, F, F, i-Bu, Pr], [RA5348; F , H, F, F, i-Bu, i-Pr], [RA5349; F, H, F, F, i-Bu, c-Pr], [RA5350; F, H, F, F, i-Bu , Bu], [RA5351; F, H, F, F, i-Bu, i-Bu], [RA5352; F, H, F, F, i-Bu, t-Bu], [RA5353; F, H , F, F, i-Bu, c-PrCH ₂ ], [RA5354; F, H, F, F, i-Bu, Ph], [RA5355; F, H, F, F, i-Bu, Bn] , [RA5356; F, H, F, F, i-Bu, CF ₃ ], [RA5357; F, H, F, F, i-Bu, CF ₃ CH ₂ ], [RA5358; F, H, F, F, i-Bu, CF ₃ CF ₂ ], [RA5359; F, H, F, F, i-Bu, CF ₂ H], [RA5360; F, H, F, F, i-Bu, CF ₂ HCH ₂ ], [RA5361; F, H, F, Cl, i-Bu, Me], [RA5362; F, H, F, Cl, i-Bu, Et], [RA5363; F, H, F, Cl, i-Bu, Pr], [RA5364; F, H, F, Cl, i-Bu, i-Pr], [RA5365; F, H, F, Cl, i-Bu, c-Pr], [RA5366; F, H, F, Cl, i-Bu, Bu], [RA5367; F, H, F, Cl, i-Bu, i-Bu], [RA5368; F, H, F, Cl, i-Bu, t-Bu], [RA5369; F, H, F, Cl, i-Bu, c-PrCH ₂ ], [RA5370; F, H, F, Cl, i-Bu, Ph], [RA5371; F, H , F, Cl, i-Bu, Bn], [RA5372; F, H, F, Cl, i-Bu, CF ₃ ], [RA5373; F, H, F, Cl, i-Bu, CF ₃ CH ₂ ], [RA5374; F, H, F, Cl, i-Bu, CF ₃ CF ₂ ], [RA5375; F, H, F, Cl, i-Bu, CF ₂ H], [RA5376; F, H, F, Cl, i-Bu, CF ₂ HCH ₂ ], [RA5377; F, H, Cl, H, i-Bu, Me], [RA5378 ; F, H, Cl, H, i-Bu, Et], [RA5379; F, H, Cl, H, i-Bu, Pr], [RA5380; F, H, Cl, H, i-Bu, i -Pr], [RA5381; F, H, Cl, H, i-Bu, c-Pr], [RA5382; F, H, Cl, H, i-Bu, Bu], [RA5383; F, H, Cl , H, i-Bu, i-Bu], [RA5384; F, H, Cl, H, i-Bu, t-Bu], [RA5385; F, H, Cl, H, i-Bu, c-PrCH ₂ ], [RA5386; F, H, Cl, H, i-Bu, Ph], [RA5387; F, H, Cl, H, i-Bu, Bn], [RA5388; F, H, Cl, H, i-Bu, CF ₃ ], [RA5389; F, H, Cl, H, i-Bu, CF ₃ CH ₂ ], [RA5390; F, H, Cl, H, i-Bu, CF ₃ CF ₂ ], [RA5391; F, H, Cl, H, i-Bu, CF ₂ H], [RA5392; F, H, Cl, H, i-Bu, CF ₂ HCH ₂ ], [RA5393; F, H, Cl, Cl, i-Bu, Me], [RA5394; F, H, Cl, Cl, i-Bu, Et], [RA5395; F, H, Cl, Cl, i-Bu, Pr], [RA5396; F, H, Cl, Cl, i-Bu, i-Pr], [RA5397; F, H, Cl, Cl, i-Bu, c-Pr], [RA5398; F, H, Cl, Cl, i-Bu, Bu], [RA5399; F, H, Cl, Cl, i-Bu, i-Bu], [RA5400; F, H, Cl, Cl, i-Bu, t-Bu],

[RA5401; F, H, Cl, Cl, i-Bu, c-PrCH ₂ ], [RA5402; F, H, Cl, Cl, i-Bu, Ph], [RA5403; F, H, Cl, Cl, i-Bu, Bn], [RA5404; F, H, Cl, Cl, i-Bu, CF ₃ ], [RA5405; F, H, Cl, Cl, i-Bu, CF ₃ CH ₂ ], [RA5406; F, H, Cl, Cl, i-Bu, CF ₃ CF ₂ ], [RA5407; F, H, Cl, Cl, i-Bu, CF ₂ H], [RA5408; F, H, Cl, Cl, i -Bu, CF ₂ HCH ₂ ], [RA5409; F, H, Me, H, t-Bu, Me], [RA5410; F, H, Me, H, t-Bu, Et], [RA5411; F, H, Me, H, t-Bu, Pr], [RA5412; F, H, Me, H, t-Bu, i-Pr], [RA5413; F, H, Me, H, t-Bu, c- Pr], [RA5414; F, H, Me, H, t-Bu, Bu], [RA5415; F, H, Me, H, t-Bu, i-Bu], [RA5416; F, H, Me, H, t-Bu, t-Bu], [RA5417; F, H, Me, H, t-Bu, c-PrCH ₂ ], [RA5418; F, H, Me, H, t-Bu, Ph], [RA5419; F, H, Me, H, t-Bu, Bn], [RA5420; F, H, Me, H, t-Bu, CF ₃ ], [RA5421; F, H, Me, H, t- Bu, CF ₃ CH ₂ ], [RA5422; F, H, Me, H, t-Bu, CF ₃ CF ₂ ], [RA5423; F, H, Me, H, t-Bu, CF ₂ H], [ RA5424; F, H, Me, H, t-Bu, CF ₂ HCH ₂ ], [RA5425; F, H, Me, Me, t-Bu, Me], [RA5426; F, H, Me, Me, t -Bu, Et], [RA5427; F, H, Me, Me, t-Bu, Pr], [RA5428; F, H, Me, Me, t-Bu, i-Pr], [RA5429; F, H , Me, Me, t-Bu, c-Pr], [RA5430; F, H, Me, Me, t-Bu, Bu], [RA5431; F, H, Me, Me, t-Bu, i-Bu ], [RA5432; F, H, Me, Me, t-Bu, t-Bu], [RA5433; F, H, Me, Me, t-Bu, c-PrCH ₂ ], [RA5434; F, H, Me, Me, t-Bu, P h], [RA5435; F, H, Me, Me, t-Bu, Bn], [RA5436; F, H, Me, Me, t-Bu, CF ₃ ], [RA5437; F, H, Me, Me , t-Bu, CF ₃ CH ₂ ], [RA5438; F, H, Me, Me, t-Bu, CF ₃ CF ₂ ], [RA5439; F, H, Me, Me, t-Bu, CF ₂ H ], [RA5440; F, H, Me, Me, t-Bu, CF ₂ HCH ₂ ], [RA5441; F, H, Me, Et, t-Bu, Me], [RA5442; F, H, Me, Et, t-Bu, Et], [RA5443; F, H, Me, Et, t-Bu, Pr], [RA5444; F, H, Me, Et, t-Bu, i-Pr], [RA5445; F, H, Me, Et, t-Bu, c-Pr], [RA5446; F, H, Me, Et, t-Bu, Bu], [RA5447; F, H, Me, Et, t-Bu, i-Bu], [RA5448; F, H, Me, Et, t-Bu, t-Bu], [RA5449; F, H, Me, Et, t-Bu, c-PrCH ₂ ], [RA5450; F , H, Me, Et, t-Bu, Ph], [RA5451; F, H, Me, Et, t-Bu, Bn], [RA5452; F, H, Me, Et, t-Bu, CF ₃ ] , [RA5453; F, H, Me, Et, t-Bu, CF ₃ CH ₂ ], [RA5454; F, H, Me, Et, t-Bu, CF ₃ CF ₂ ], [RA5455; F, H, Me, Et, t-Bu, CF ₂ H], [RA5456; F, H, Me, Et, t-Bu, CF ₂ HCH ₂ ], [RA5457; F, H, Me, F, t-Bu, Me ], [RA5458; F, H, Me, F, t-Bu, Et], [RA5459; F, H, Me, F, t-Bu, Pr], [RA5460; F, H, Me, F, t -Bu, i-Pr], [RA5461; F, H, Me, F, t-Bu, c-Pr], [RA5462; F, H, Me, F, t-Bu, Bu], [RA5463; F , H, Me, F, t-Bu, i-Bu], [RA5464; F, H, Me, F, t-Bu, t-Bu], [RA5465; F, H, Me, F, t-Bu , c-PrCH ₂ ], [RA5466; F, H, Me, F, t-Bu, Ph], [RA5467; F, H, Me, F, t-Bu, Bn], [RA5468; F, H, Me, F, t-Bu, C F ₃ ], [RA5469; F, H, Me, F, t-Bu, CF ₃ CH ₂ ], [RA5470; F, H, Me, F, t-Bu, CF ₃ CF ₂ ], [RA5471; F , H, Me, F, t-Bu, CF ₂ H], [RA5472; F, H, Me, F, t-Bu, CF ₂ HCH ₂ ], [RA5473; F, H, Me, Cl, t- Bu, Me], [RA5474; F, H, Me, Cl, t-Bu, Et], [RA5475; F, H, Me, Cl, t-Bu, Pr], [RA5476; F, H, Me, Cl, t-Bu, i-Pr], [RA5477; F, H, Me, Cl, t-Bu, c-Pr], [RA5478; F, H, Me, Cl, t-Bu, Bu], [ RA5479; F, H, Me, Cl, t-Bu, i-Bu], [RA5480; F, H, Me, Cl, t-Bu, t-Bu], [RA5481; F, H, Me, Cl, t-Bu, c-PrCH ₂ ], [RA5482; F, H, Me, Cl, t-Bu, Ph], [RA5483; F, H, Me, Cl, t-Bu, Bn], [RA5484; F , H, Me, Cl, t-Bu, CF ₃ ], [RA5485; F, H, Me, Cl, t-Bu, CF ₃ CH ₂ ], [RA5486; F, H, Me, Cl, t-Bu , CF ₃ CF ₂ ], [RA5487; F, H, Me, Cl, t-Bu, CF ₂ H], [RA5488; F, H, Me, Cl, t-Bu, CF ₂ HCH ₂ ], [RA5489 ; F, H, Et, H, t-Bu, Me], [RA5490; F, H, Et, H, t-Bu, Et], [RA5491; F, H, Et, H, t-Bu, Pr ], [RA5492; F, H, Et, H, t-Bu, i-Pr], [RA5493; F, H, Et, H, t-Bu, c-Pr], [RA5494; F, H, Et , H, t-Bu, Bu], [RA5495; F, H, Et, H, t-Bu, i-Bu], [RA5496; F, H, Et, H, t-Bu, t-Bu], [RA5497; F, H, Et, H, t-Bu, c-PrCH ₂ ], [RA5498; F, H, Et, H, t-Bu, Ph], [RA5499; F, H, Et, H, t-Bu, Bn], [RA5500; F, H, Et, H, t-Bu, CF ₃ ], [RA5501; F, H, Et, H, t-Bu, CF ₃ CH ₂ ], [RA5502; F, H, Et, H, t -Bu, CF ₃ CF ₂ ], [RA5503; F, H, Et, H, t-Bu, CF ₂ H], [RA5504; F, H, Et, H, t-Bu, CF ₂ HCH ₂ ], [RA5505; F, H, Et, F, t-Bu, Me], [RA5506; F, H, Et, F, t-Bu, Et], [RA5507; F, H, Et, F, t-Bu , Pr], [RA5508; F, H, Et, F, t-Bu, i-Pr], [RA5509; F, H, Et, F, t-Bu, c-Pr], [RA5510; F, H , Et, F, t-Bu, Bu], [RA5511; F, H, Et, F, t-Bu, i-Bu], [RA5512; F, H, Et, F, t-Bu, t-Bu ], [RA5513; F, H, Et, F, t-Bu, c-PrCH ₂ ], [RA5514; F, H, Et, F, t-Bu, Ph], [RA5515; F, H, Et, F, t-Bu, Bn], [RA5516; F, H, Et, F, t-Bu, CF ₃ ], [RA5517; F, H, Et, F, t-Bu, CF ₃ CH ₂ ], [ RA5518; F, H, Et, F, t-Bu, CF ₃ CF ₂ ], [RA5519; F, H, Et, F, t-Bu, CF ₂ H], [RA5520; F, H, Et, F , t-Bu, CF ₂ HCH ₂ ], [RA5521; F, H, Et, Cl, t-Bu, Me], [RA5522; F, H, Et, Cl, t-Bu, Et], [RA5523; F, H, Et, Cl, t-Bu, Pr], [RA5524; F, H, Et, Cl, t-Bu, i-Pr], [RA5525; F, H, Et, Cl, t-Bu, c-Pr], [RA5526; F, H, Et, Cl, t-Bu, Bu], [RA5527; F, H, Et, Cl, t-Bu, i-Bu], [RA5528; F, H, Et, Cl, t-Bu, t-Bu], [RA5529; F, H, Et, Cl, t-Bu, c-PrCH ₂ ], [RA5530; F, H, Et, Cl, t-Bu, Ph ], [RA5531; F, H, Et, Cl, t-Bu, Bn], [RA5532; F, H, Et, Cl, t-Bu, CF ₃ ], [RA5533; F, H, Et, Cl, t-Bu, CF ₃ CH ₂ ], [RA5534; F, H, Et, Cl, t-Bu, CF ₃ CF ₂ ], [RA5535; F, H, Et, Cl, t-Bu, CF ₂ H] , [RA5536; F, H, E t, Cl, t-Bu, CF ₂ HCH ₂ ], [RA5537; F, H, F, H, t-Bu, Me], [RA5538; F, H, F, H, t-Bu, Et], [RA5539; F, H, F, H, t-Bu, Pr], [RA5540; F, H, F, H, t-Bu, i-Pr], [RA5541; F, H, F, H, t -Bu, c-Pr], [RA5542; F, H, F, H, t-Bu, Bu], [RA5543; F, H, F, H, t-Bu, i-Bu], [RA5544; F , H, F, H, t-Bu, t-Bu], [RA5545; F, H, F, H, t-Bu, c-PrCH ₂ ], [RA5546; F, H, F, H, t- Bu, Ph], [RA5547; F, H, F, H, t-Bu, Bn], [RA5548; F, H, F, H, t-Bu, CF ₃ ], [RA5549; F, H, F , H, t-Bu, CF ₃ CH ₂ ], [RA5550; F, H, F, H, t-Bu, CF ₃ CF ₂ ], [RA5551; F, H, F, H, t-Bu, CF ₂ H], [RA5552; F, H, F, H, t-Bu, CF ₂ HCH ₂ ], [RA5553; F, H, F, F, t-Bu, Me], [RA5554; F, H, F, F, t-Bu, Et], [RA5555; F, H, F, F, t-Bu, Pr], [RA5556; F, H, F, F, t-Bu, i-Pr], [ RA5557; F, H, F, F, t-Bu, c-Pr], [RA5558; F, H, F, F, t-Bu, Bu], [RA5559; F, H, F, F, t- Bu, i-Bu], [RA5560; F, H, F, F, t-Bu, t-Bu], [RA5561; F, H, F, F, t-Bu, c-PrCH ₂ ], [RA5562 ; F, H, F, F, t-Bu, Ph], [RA5563; F, H, F, F, t-Bu, Bn], [RA5564; F, H, F, F, t-Bu, CF ₃ ], [RA5565; F, H, F, F, t-Bu, CF ₃ CH ₂ ], [RA5566; F, H, F, F, t-Bu, CF ₃ CF ₂ ], [RA5567; F, H, F, F, t-Bu, CF ₂ H], [RA5568; F, H, F, F, t-Bu, CF ₂ HCH ₂ ], [RA5569; F, H, F, Cl, t-Bu , Me], [RA5570; F, H, F, Cl, t-Bu, Et], [RA5571; F, H, F, Cl, t-Bu, Pr], [RA55 72; F, H, F, Cl, t-Bu, i-Pr], [RA5573; F, H, F, Cl, t-Bu, c-Pr], [RA5574; F, H, F, Cl, t-Bu, Bu], [RA5575; F, H, F, Cl, t-Bu, i-Bu], [RA5576; F, H, F, Cl, t-Bu, t-Bu], [RA5577; F, H, F, Cl, t-Bu, c-PrCH ₂ ], [RA5578; F, H, F, Cl, t-Bu, Ph], [RA5579; F, H, F, Cl, t-Bu , Bn], [RA5580; F, H, F, Cl, t-Bu, CF ₃ ], [RA5581; F, H, F, Cl, t-Bu, CF ₃ CH ₂ ], [RA5582; F, H , F, Cl, t-Bu, CF ₃ CF ₂ ], [RA5583; F, H, F, Cl, t-Bu, CF ₂ H], [RA5584; F, H, F, Cl, t-Bu, CF ₂ HCH ₂ ], [RA5585; F, H, Cl, H, t-Bu, Me], [RA5586; F, H, Cl, H, t-Bu, Et], [RA5587; F, H, Cl , H, t-Bu, Pr], [RA5588; F, H, Cl, H, t-Bu, i-Pr], [RA5589; F, H, Cl, H, t-Bu, c-Pr], [RA5590; F, H, Cl, H, t-Bu, Bu], [RA5591; F, H, Cl, H, t-Bu, i-Bu], [RA5592; F, H, Cl, H, t -Bu, t-Bu], [RA5593; F, H, Cl, H, t-Bu, c-PrCH ₂ ], [RA5594; F, H, Cl, H, t-Bu, Ph], [RA5595; F, H, Cl, H, t-Bu, Bn], [RA5596; F, H, Cl, H, t-Bu, CF ₃ ], [RA5597; F, H, Cl, H, t-Bu, CF ₃ CH ₂ ], [RA5598; F, H, Cl, H, t-Bu, CF ₃ CF ₂ ], [RA5599; F, H, Cl, H, t-Bu, CF ₂ H], [RA5600; F , H, Cl, H, t-Bu, CF ₂ HCH ₂ ],

[RA5601; F, H, Cl, Cl, t-Bu, Me], [RA5602; F, H, Cl, Cl, t-Bu, Et], [RA5603; F, H, Cl, Cl, t-Bu , Pr], [RA5604; F, H, Cl, Cl, t-Bu, i-Pr], [RA5605; F, H, Cl, Cl, t-Bu, c-Pr], [RA5606; F, H , Cl, Cl, t-Bu, Bu], [RA5607; F, H, Cl, Cl, t-Bu, i-Bu], [RA5608; F, H, Cl, Cl, t-Bu, t-Bu ], [RA5609; F, H, Cl, Cl, t-Bu, c-PrCH ₂ ], [RA5610; F, H, Cl, Cl, t-Bu, Ph], [RA5611; F, H, Cl, Cl, t-Bu, Bn], [RA5612; F, H, Cl, Cl, t-Bu, CF ₃ ], [RA5613; F, H, Cl, Cl, t-Bu, CF ₃ CH ₂ ], [ RA5614; F, H, Cl, Cl, t-Bu, CF ₃ CF ₂ ], [RA5615; F, H, Cl, Cl, t-Bu, CF ₂ H], [RA5616; F, H, Cl, Cl , t-Bu, CF ₂ HCH ₂ ], [RA5617; F, H, Me, H, CF ₂ H, Me], [RA5618; F, H, Me, H, CF ₂ H, Et], [RA5619; F, H, Me, H, CF ₂ H, Pr], [RA5620; F, H, Me, H, CF ₂ H, i-Pr], [RA5621; F, H, Me, H, CF ₂ H, c-Pr], [RA5622; F, H, Me, H, CF ₂ H, Bu], [RA5623; F, H, Me, H, CF ₂ H, i-Bu], [RA5624; F, H, Me, H, CF ₂ H, t-Bu], [RA5625; F, H, Me, H, CF ₂ H, c-PrCH ₂ ], [RA5626; F, H, Me, H, CF ₂ H, Ph ], [RA5627; F, H, Me, H, CF ₂ H, Bn], [RA5628; F, H, Me, H, CF ₂ H, CF ₃ ], [RA5629; F, H, Me, H, CF ₂ H, CF ₃ CH ₂ ], [RA5630; F, H, Me, H, CF ₂ H, CF ₃ CF ₂ ], [RA5631; F, H, Me, H, CF ₂ H, CF ₂ H] , [RA5632; F, H, Me, H, CF ₂ H, CF ₂ HCH ₂ ], [RA5633; F, H, Me, Me, CF ₂ H, M e], [RA5634; F, H, Me, Me, CF ₂ H, Et], [RA5635; F, H, Me, Me, CF ₂ H, Pr], [RA5636; F, H, Me, Me, CF ₂ H, i-Pr], [RA5637; F, H, Me, Me, CF ₂ H, c-Pr], [RA5638; F, H, Me, Me, CF ₂ H, Bu], [RA5639; F, H, Me, Me, CF ₂ H, i-Bu], [RA5640; F, H, Me, Me, CF ₂ H, t-Bu], [RA5641; F, H, Me, Me, CF ₂ H, c-PrCH ₂ ], [RA5642; F, H, Me, Me, CF ₂ H, Ph], [RA5643; F, H, Me, Me, CF ₂ H, Bn], [RA5644; F, H , Me, Me, CF ₂ H, CF ₃ ], [RA5645; F, H, Me, Me, CF ₂ H, CF ₃ CH ₂ ], [RA5646; F, H, Me, Me, CF ₂ H, CF ₃ CF ₂ ], [RA5647; F, H, Me, Me, CF ₂ H, CF ₂ H], [RA5648; F, H, Me, Me, CF ₂ H, CF ₂ HCH ₂ ], [RA5649; F , H, Me, Et, CF ₂ H, Me], [RA5650; F, H, Me, Et, CF ₂ H, Et], [RA5651; F, H, Me, Et, CF ₂ H, Pr], [RA5652; F, H, Me, Et, CF ₂ H, i-Pr], [RA5653; F, H, Me, Et, CF ₂ H, c-Pr], [RA5654; F, H, Me, Et , CF ₂ H, Bu], [RA5655; F, H, Me, Et, CF ₂ H, i-Bu], [RA5656; F, H, Me, Et, CF ₂ H, t-Bu], [RA5657 ; F, H, Me, Et, CF ₂ H, c-PrCH ₂ ], [RA5658; F, H, Me, Et, CF ₂ H, Ph], [RA5659; F, H, Me, Et, CF ₂ H, Bn], [RA5660; F, H, Me, Et, CF ₂ H, CF ₃ ], [RA5661; F, H, Me, Et, CF ₂ H, CF ₃ CH ₂ ], [RA5662; F, H, Me, Et, CF ₂ H, CF ₃ CF ₂ ], [RA5663; F, H, Me, Et, CF ₂ H, CF ₂ H], [RA5664; F, H, Me, Et, CF ₂ H , CF ₂ HCH ₂ ], [RA5 665; F, H, Me, F, CF ₂ H, Me], [RA5666; F, H, Me, F, CF ₂ H, Et], [RA5667; F, H, Me, F, CF ₂ H, Pr], [RA5668; F, H, Me, F, CF ₂ H, i-Pr], [RA5669; F, H, Me, F, CF ₂ H, c-Pr], [RA5670; F, H, Me, F, CF ₂ H, Bu], [RA5671; F, H, Me, F, CF ₂ H, i-Bu], [RA5672; F, H, Me, F, CF ₂ H, t-Bu] , [RA5673; F, H, Me, F, CF ₂ H, c-PrCH ₂ ], [RA5674; F, H, Me, F, CF ₂ H, Ph], [RA5675; F, H, Me, F , CF ₂ H, Bn], [RA5676; F, H, Me, F, CF ₂ H, CF ₃ ], [RA5677; F, H, Me, F, CF ₂ H, CF ₃ CH ₂ ], [RA5678 ; F, H, Me, F, CF ₂ H, CF ₃ CF ₂ ], [RA5679; F, H, Me, F, CF ₂ H, CF ₂ H], [RA5680; F, H, Me, F, CF ₂ H, CF ₂ HCH ₂ ], [RA5681; F, H, Me, Cl, CF ₂ H, Me], [RA5682; F, H, Me, Cl, CF ₂ H, Et], [RA5683; F , H, Me, Cl, CF ₂ H, Pr], [RA5684; F, H, Me, Cl, CF ₂ H, i-Pr], [RA5685; F, H, Me, Cl, CF ₂ H, c -Pr], [RA5686; F, H, Me, Cl, CF ₂ H, Bu], [RA5687; F, H, Me, Cl, CF ₂ H, i-Bu], [RA5688; F, H, Me , Cl, CF ₂ H, t-Bu], [RA5689; F, H, Me, Cl, CF ₂ H, c-PrCH ₂ ], [RA5690; F, H, Me, Cl, CF ₂ H, Ph] , [RA5691; F, H, Me, Cl, CF ₂ H, Bn], [RA5692; F, H, Me, Cl, CF ₂ H, CF ₃ ], [RA5693; F, H, Me, Cl, CF ₂ H, CF ₃ CH ₂ ], [RA5694; F, H, Me, Cl, CF ₂ H, CF ₃ CF ₂ ], [RA5695; F, H, Me, Cl, CF ₂ H, CF ₂ H], [RA5696; F, H, Me, Cl, CF ₂ H, CF ₂ HCH ₂ ], [RA5697; F, H, Et, H, CF ₂ H, Me], [RA5698; F, H, Et, H, CF ₂ H, Et], [RA5699; F, H, Et, H, CF ₂ H, Pr], [RA5700; F, H, Et, H, CF ₂ H, i-Pr], [RA5701; F, H, Et, H, CF ₂ H, c-Pr], [RA5702; F , H, Et, H, CF ₂ H, Bu], [RA5703; F, H, Et, H, CF ₂ H, i-Bu], [RA5704; F, H, Et, H, CF ₂ H, t -Bu], [RA5705; F, H, Et, H, CF ₂ H, c-PrCH ₂ ], [RA5706; F, H, Et, H, CF ₂ H, Ph], [RA5707; F, H, Et, H, CF ₂ H, Bn], [RA5708; F, H, Et, H, CF ₂ H, CF ₃ ], [RA5709; F, H, Et, H, CF ₂ H, CF ₃ CH ₂ ] , [RA5710; F, H, Et, H, CF ₂ H, CF ₃ CF ₂ ], [RA5711; F, H, Et, H, CF ₂ H, CF ₂ H], [RA5712; F, H, Et , H, CF ₂ H, CF ₂ HCH ₂ ], [RA5713; F, H, Et, F, CF ₂ H, Me], [RA5714; F, H, Et, F, CF ₂ H, Et], [ RA5715; F, H, Et, F, CF ₂ H, Pr], [RA5716; F, H, Et, F, CF ₂ H, i-Pr], [RA5717; F, H, Et, F, CF ₂ H, c-Pr], [RA5718; F, H, Et, F, CF ₂ H, Bu], [RA5719; F, H, Et, F, CF ₂ H, i-Bu], [RA5720; F, H, Et, F, CF ₂ H, t-Bu], [RA5721; F, H, Et, F, CF ₂ H, c-PrCH ₂ ], [RA5722; F, H, Et, F, CF ₂ H , Ph], [RA5723; F, H, Et, F, CF ₂ H, Bn], [RA5724; F, H, Et, F, CF ₂ H, CF ₃ ], [RA5725; F, H, Et, F, CF ₂ H, CF ₃ CH ₂ ], [RA5726; F, H, Et, F, CF ₂ H, CF ₃ CF ₂ ], [RA5727; F, H, Et, F, CF ₂ H, CF ₂ H], [RA5728; F, H, Et, F, CF ₂ H, CF ₂ HCH ₂ ], [RA5729; F, H, Et, Cl, CF ₂ H, Me], [RA5730; F, H, Et, Cl, CF ₂ H, Et], [RA5731; F, H, Et, Cl, CF ₂ H, Pr] , [RA5732; F, H, Et, Cl, CF ₂ H, i-Pr], [RA5733; F, H, Et, Cl, CF ₂ H, c-Pr], [RA5734; F, H, Et, Cl, CF ₂ H, Bu], [RA5735; F, H, Et, Cl, CF ₂ H, i-Bu], [RA5736; F, H, Et, Cl, CF ₂ H, t-Bu], [ RA5737; F, H, Et, Cl, CF ₂ H, c-PrCH ₂ ], [RA5738; F, H, Et, Cl, CF ₂ H, Ph], [RA5739; F, H, Et, Cl, CF ₂ H, Bn], [RA5740; F, H, Et, Cl, CF ₂ H, CF ₃ ], [RA5741; F, H, Et, Cl, CF ₂ H, CF ₃ CH ₂ ], [RA5742; F , H, Et, Cl, CF ₂ H, CF ₃ CF ₂ ], [RA5743; F, H, Et, Cl, CF ₂ H, CF ₂ H], [RA5744; F, H, Et, Cl, CF ₂ H, CF ₂ HCH ₂ ], [RA5745; F, H, F, H, CF ₂ H, Me], [RA5746; F, H, F, H, CF ₂ H, Et], [RA5747; F, H , F, H, CF ₂ H, Pr], [RA5748; F, H, F, H, CF ₂ H, i-Pr], [RA5749; F, H, F, H, CF ₂ H, c-Pr ], [RA5750; F, H, F, H, CF ₂ H, Bu], [RA5751; F, H, F, H, CF ₂ H, i-Bu], [RA5752; F, H, F, H , CF ₂ H, t-Bu], [RA5753; F, H, F, H, CF ₂ H, c-PrCH ₂ ], [RA5754; F, H, F, H, CF ₂ H, Ph], [ RA5755; F, H, F, H, CF ₂ H, Bn], [RA5756; F, H, F, H, CF ₂ H, CF ₃ ], [RA5757; F, H, F, H, CF ₂ H , CF ₃ CH ₂ ], [RA5758; F, H, F, H, CF ₂ H, CF ₃ CF ₂ ], [RA5759; F, H, F, H, CF ₂ H, CF ₂ H], [RA5760 ; F, H, F, H, CF ₂ H, CF ₂ HCH ₂ ], [RA5761; F, H, F, F, CF ₂ H, Me], [RA5762; F, H, F, F, CF ₂ H, Et], [RA5763; F, H, F, F, CF ₂ H, Pr], [RA5764; F, H, F , F, CF ₂ H, i-Pr], [RA5765; F, H, F, F, CF ₂ H, c-Pr], [RA5766; F, H, F, F, CF ₂ H, Bu], [RA5767; F, H, F, F, CF ₂ H, i-Bu], [RA5768; F, H, F, F, CF ₂ H, t-Bu], [RA5769; F, H, F, F , CF ₂ H, c-PrCH ₂ ], [RA5770; F, H, F, F, CF ₂ H, Ph], [RA5771; F, H, F, F, CF ₂ H, Bn], [RA5772; F, H, F, F, CF ₂ H, CF ₃ ], [RA5773; F, H, F, F, CF ₂ H, CF ₃ CH ₂ ], [RA5774; F, H, F, F, CF ₂ H, CF ₃ CF ₂ ], [RA5775; F, H, F, F, CF ₂ H, CF ₂ H], [RA5776; F, H, F, F, CF ₂ H, CF ₂ HCH ₂ ], [ RA5777; F, H, F, Cl, CF ₂ H, Me], [RA5778; F, H, F, Cl, CF ₂ H, Et], [RA5779; F, H, F, Cl, CF ₂ H, Pr], [RA5780; F, H, F, Cl, CF ₂ H, i-Pr], [RA5781; F, H, F, Cl, CF ₂ H, c-Pr], [RA5782; F, H, F, Cl, CF ₂ H, Bu], [RA5783; F, H, F, Cl, CF ₂ H, i-Bu], [RA5784; F, H, F, Cl, CF ₂ H, t-Bu] , [RA5785; F, H, F, Cl, CF ₂ H, c-PrCH ₂ ], [RA5786; F, H, F, Cl, CF ₂ H, Ph], [RA5787; F, H, F, Cl , CF ₂ H, Bn], [RA5788; F, H, F, Cl, CF ₂ H, CF ₃ ], [RA5789; F, H, F, Cl, CF ₂ H, CF ₃ CH ₂ ], [RA5790 ; F, H, F, Cl, CF ₂ H, CF ₃ CF ₂ ], [RA5791; F, H, F, Cl, CF ₂ H, CF ₂ H], [RA5792; F, H, F, Cl, CF ₂ H, CF ₂ HCH ₂ ], [RA5793; F, H, Cl, H, CF ₂ H, Me], [RA5794; F, H, Cl, H , CF ₂ H, Et], [RA5795; F, H, Cl, H, CF ₂ H, Pr], [RA5796; F, H, Cl, H, CF ₂ H, i-Pr], [RA5797; F , H, Cl, H, CF ₂ H, c-Pr], [RA5798; F, H, Cl, H, CF ₂ H, Bu], [RA5799; F, H, Cl, H, CF ₂ H, i -Bu], [RA5800; F, H, Cl, H, CF ₂ H, t-Bu],

[RA5801; F, H, Cl, H, CF ₂ H, c-PrCH ₂ ], [RA5802; F, H, Cl, H, CF ₂ H, Ph], [RA5803; F, H, Cl, H, CF ₂ H, Bn], [RA5804; F, H, Cl, H, CF ₂ H, CF ₃ ], [RA5805; F, H, Cl, H, CF ₂ H, CF ₃ CH ₂ ], [RA5806; F, H, Cl, H, CF ₂ H, CF ₃ CF ₂ ], [RA5807; F, H, Cl, H, CF ₂ H, CF ₂ H], [RA5808; F, H, Cl, H, CF ₂ H, CF ₂ HCH ₂ ], [RA5809; F, H, Cl, Cl, CF ₂ H, Me], [RA5810; F, H, Cl, Cl, CF ₂ H, Et], [RA5811; F, H, Cl, Cl, CF ₂ H, Pr], [RA5812; F, H, Cl, Cl, CF ₂ H, i-Pr], [RA5813; F, H, Cl, Cl, CF ₂ H, c- Pr], [RA5814; F, H, Cl, Cl, CF ₂ H, Bu], [RA5815; F, H, Cl, Cl, CF ₂ H, i-Bu], [RA5816; F, H, Cl, Cl, CF ₂ H, t-Bu], [RA5817; F, H, Cl, Cl, CF ₂ H, c-PrCH ₂ ], [RA5818; F, H, Cl, Cl, CF ₂ H, Ph], [RA5819; F, H, Cl, Cl, CF ₂ H, Bn], [RA5820; F, H, Cl, Cl, CF ₂ H, CF ₃ ], [RA5821; F, H, Cl, Cl, CF ₂ H, CF ₃ CH ₂ ], [RA5822; F, H, Cl, Cl, CF ₂ H, CF ₃ CF ₂ ], [RA5823; F, H, Cl, Cl, CF ₂ H, CF ₂ H], [ RA5824; F, H, Cl, Cl, CF ₂ H, CF ₂ HCH ₂ ], [RA5825; F, H, Me, H, CF ₃ , Me], [RA5826; F, H, Me, H, CF ₃ , Et], [RA5827; F, H, Me, H, CF ₃ , Pr], [RA5828; F, H, Me, H, CF ₃ , i-Pr], [RA5829; F, H, Me, H , CF ₃ , c-Pr], [RA5830; F, H, Me, H, CF ₃ , Bu], [RA5831; F, H, Me, H, CF ₃ , i-Bu], [RA5832; F, H, Me, H, CF ₃ , t-Bu], [R A5833; F, H, Me, H, CF ₃ , c-PrCH ₂ ], [RA5834; F, H, Me, H, CF ₃ , Ph], [RA5835; F, H, Me, H, CF ₃ , Bn], [RA5836; F, H, Me, H, CF ₃ , CF ₃ ], [RA5837; F, H, Me, H, CF ₃ , CF ₃ CH ₂ ], [RA5838; F, H, Me, H, CF ₃ , CF ₃ CF ₂ ], [RA5839; F, H, Me, H, CF ₃ , CF ₂ H], [RA5840; F, H, Me, H, CF ₃ , CF ₂ HCH ₂ ], [RA5841; F, H, Me, Me, CF ₃ , Me], [RA5842; F, H, Me, Me, CF ₃ , Et], [RA5843; F, H, Me, Me, CF ₃ , Pr] , [RA5844; F, H, Me, Me, CF ₃ , i-Pr], [RA5845; F, H, Me, Me, CF ₃ , c-Pr], [RA5846; F, H, Me, Me, CF ₃ , Bu], [RA5847; F, H, Me, Me, CF ₃ , i-Bu], [RA5848; F, H, Me, Me, CF ₃ , t-Bu], [RA5849; F, H , Me, Me, CF ₃ , c-PrCH ₂ ], [RA5850; F, H, Me, Me, CF ₃ , Ph], [RA5851; F, H, Me, Me, CF ₃ , Bn], [RA5852 ; F, H, Me, Me, CF ₃ , CF ₃ ], [RA5853; F, H, Me, Me, CF ₃ , CF ₃ CH ₂ ], [RA5854; F, H, Me, Me, CF ₃ , CF ₃ CF ₂ ], [RA5855; F, H, Me, Me, CF ₃ , CF ₂ H], [RA5856; F, H, Me, Me, CF ₃ , CF ₂ HCH ₂ ], [RA5857; F, H, Me, Et, CF ₃ , Me], [RA5858; F, H, Me, Et, CF ₃ , Et], [RA5859; F, H, Me, Et, CF ₃ , Pr], [RA5860; F , H, Me, Et, CF ₃ , i-Pr], [RA5861; F, H, Me, Et, CF ₃ , c-Pr], [RA5862; F, H, Me, Et, CF ₃ , Bu] , [RA5863; F, H, Me, Et, CF ₃ , i-Bu], [RA5864; F, H, Me, Et, CF ₃ , t-Bu], [RA5865; F, H, Me, Et, CF ₃ , c-PrCH ₂ ], [RA5866; F, H, Me, Et, CF ₃ , Ph], [RA5867; F, H, Me, Et, CF ₃ , Bn], [RA5868; F, H, Me , Et, CF ₃ , CF ₃ ], [RA5869; F, H, Me, Et, CF ₃ , CF ₃ CH ₂ ], [RA5870; F, H, Me, Et, CF ₃ , CF ₃ CF ₂ ], [RA5871; F, H, Me, Et, CF ₃ , CF ₂ H], [RA5872; F, H, Me, Et, CF ₃ , CF ₂ HCH ₂ ], [RA5873; F, H, Me, F, CF ₃ , Me], [RA5874; F, H, Me, F, CF ₃ , Et], [RA5875; F, H, Me, F, CF ₃ , Pr], [RA5876; F, H, Me, F , CF ₃ , i-Pr], [RA5877; F, H, Me, F, CF ₃ , c-Pr], [RA5878; F, H, Me, F, CF ₃ , Bu], [RA5879; F, H, Me, F, CF ₃ , i-Bu], [RA5880; F, H, Me, F, CF ₃ , t-Bu], [RA5881; F, H, Me, F, CF ₃ , c-PrCH ₂ ], [RA5882; F, H, Me, F, CF ₃ , Ph], [RA5883; F, H, Me, F, CF ₃ , Bn], [RA5884; F, H, Me, F, CF ₃ , CF ₃ ], [RA5885; F, H, Me, F, CF ₃ , CF ₃ CH ₂ ], [RA5886; F, H, Me, F, CF ₃ , CF ₃ CF ₂ ], [RA5887; F, H, Me, F, CF ₃ , CF ₂ H], [RA5888; F, H, Me, F, CF ₃ , CF ₂ HCH ₂ ], [RA5889; F, H, Me, Cl, CF ₃ , Me] , [RA5890; F, H, Me, Cl, CF ₃ , Et], [RA5891; F, H, Me, Cl, CF ₃ , Pr], [RA5892; F, H, Me, Cl, CF ₃ , i -Pr], [RA5893; F, H, Me, Cl, CF ₃ , c-Pr], [RA5894; F, H, Me, Cl, CF ₃ , Bu], [RA5895; F, H, Me, Cl , CF ₃ , i-Bu], [RA5896; F, H, Me, Cl, CF ₃ , t-Bu], [RA5897; F, H, Me, Cl, CF ₃ , c-PrCH ₂ ], [RA5898 ; F, H , Me, Cl, CF ₃ , Ph], [RA5899; F, H, Me, Cl, CF ₃ , Bn], [RA5900; F, H, Me, Cl, CF ₃ , CF ₃ ], [RA5901; F , H, Me, Cl, CF ₃ , CF ₃ CH ₂ ], [RA5902; F, H, Me, Cl, CF ₃ , CF ₃ CF ₂ ], [RA5903; F, H, Me, Cl, CF ₃ , CF ₂ H], [RA5904; F, H, Me, Cl, CF ₃ , CF ₂ HCH ₂ ], [RA5905; F, H, Et, H, CF ₃ , Me], [RA5906; F, H, Et , H, CF ₃ , Et], [RA5907; F, H, Et, H, CF ₃ , Pr], [RA5908; F, H, Et, H, CF ₃ , i-Pr], [RA5909; F, H, Et, H, CF ₃ , c-Pr], [RA5910; F, H, Et, H, CF ₃ , Bu], [RA5911; F, H, Et, H, CF ₃ , i-Bu], [RA5912; F, H, Et, H, CF ₃ , t-Bu], [RA5913; F, H, Et, H, CF ₃ , c-PrCH ₂ ], [RA5914; F, H, Et, H, CF ₃ , Ph], [RA5915; F, H, Et, H, CF ₃ , Bn], [RA5916; F, H, Et, H, CF ₃ , CF ₃ ], [RA5917; F, H, Et, H, CF ₃ , CF ₃ CH ₂ ], [RA5918; F, H, Et, H, CF ₃ , CF ₃ CF ₂ ], [RA5919; F, H, Et, H, CF ₃ , CF ₂ H], [RA5920; F, H, Et, H, CF ₃ , CF ₂ HCH ₂ ], [RA5921; F, H, Et, F, CF ₃ , Me], [RA5922; F, H, Et, F, CF ₃ , Et], [RA5923; F, H, Et, F, CF ₃ , Pr], [RA5924; F, H, Et, F, CF ₃ , i-Pr], [RA5925; F, H, Et, F , CF ₃ , c-Pr], [RA5926; F, H, Et, F, CF ₃ , Bu], [RA5927; F, H, Et, F, CF ₃ , i-Bu], [RA5928; F, H, Et, F, CF ₃ , t-Bu], [RA5929; F, H, Et, F, CF ₃ , c-PrCH ₂ ], [RA5930; F, H, Et, F, CF ₃ , Ph] , [RA5931; F, H, Et, F, CF ₃ , Bn], [RA5932; F, H, Et, F, CF ₃ , CF ₃ ], [RA5933; F, H, Et, F, CF ₃ , CF ₃ CH ₂ ], [RA5934; F, H, Et, F, CF ₃ , CF ₃ CF ₂ ], [RA5935; F, H, Et, F, CF ₃ , CF ₂ H], [RA5936; F, H, Et, F, CF ₃ , CF ₂ HCH ₂ ], [RA5937; F, H, Et, Cl, CF ₃ , Me], [RA5938; F, H, Et, Cl, CF ₃ , Et], [RA5939; F, H, Et, Cl, CF ₃ , Pr], [RA5940; F, H, Et, Cl, CF ₃ , i-Pr], [RA5941; F, H, Et, Cl, CF ₃ , c-Pr], [RA5942; F, H, Et, Cl, CF ₃ , Bu], [RA5943; F, H, Et, Cl, CF ₃ , i-Bu], [RA5944; F, H, Et, Cl, CF ₃ , t-Bu], [RA5945; F , H, Et, Cl, CF ₃ , c-PrCH ₂ ], [RA5946; F, H, Et, Cl, CF ₃ , Ph], [RA5947; F, H, Et, Cl, CF ₃ , Bn], [RA5948; F, H, Et, Cl, CF ₃ , CF ₃ ], [RA5949; F, H, Et, Cl, CF ₃ , CF ₃ CH ₂ ], [RA5950; F, H, Et, Cl, CF ₃ , CF ₃ CF ₂ ], [RA5951; F, H, Et, Cl, CF ₃ , CF ₂ H], [RA5952; F, H, Et, Cl, CF ₃ , CF ₂ HCH ₂ ], [RA5953; F, H, F, H, CF ₃ , Me], [RA5954; F, H, F, H, CF ₃ , Et], [RA5955; F, H, F, H, CF ₃ , Pr], [RA5956 ; F, H, F, H, CF ₃ , i-Pr], [RA5957; F, H, F, H, CF ₃ , c-Pr], [RA5958; F, H, F, H, CF ₃ , Bu], [RA5959; F, H, F, H, CF ₃ , i-Bu], [RA5960; F, H, F, H, CF ₃ , t-Bu], [RA5961; F, H, F, H, CF ₃ , c-PrCH ₂ ], [RA5962; F, H, F, H, CF ₃ , Ph], [RA5963; F, H, F, H, CF ₃ , Bn], [RA5964; F, H, F, H, CF ₃ , CF ₃ ], [RA5965; F, H, F, H, CF ₃ , CF ₃ CH ₂ ], [RA5966; F, H, F, H, CF ₃ , CF ₃ CF ₂ ], [RA5967; F, H, F, H , CF ₃ , CF ₂ H], [RA5968; F, H, F, H, CF ₃ , CF ₂ HCH ₂ ], [RA5969; F, H, F, F, CF ₃ , Me], [RA5970; F , H, F, F, CF ₃ , Et], [RA5971; F, H, F, F, CF ₃ , Pr], [RA5972; F, H, F, F, CF ₃ , i-Pr], [ RA5973; F, H, F, F, CF ₃ , c-Pr], [RA5974; F, H, F, F, CF ₃ , Bu], [RA5975; F, H, F, F, CF ₃ , i -Bu], [RA5976; F, H, F, F, CF ₃ , t-Bu], [RA5977; F, H, F, F, CF ₃ , c-PrCH ₂ ], [RA5978; F, H, F, F, CF ₃ , Ph], [RA5979; F, H, F, F, CF ₃ , Bn], [RA5980; F, H, F, F, CF ₃ , CF ₃ ], [RA5981; F, H, F, F, CF ₃ , CF ₃ CH ₂ ], [RA5982; F, H, F, F, CF ₃ , CF ₃ CF ₂ ], [RA5983; F, H, F, F, CF ₃ , CF ₂ H], [RA5984; F, H, F, F, CF ₃ , CF ₂ HCH ₂ ], [RA5985; F, H, F, Cl, CF ₃ , Me], [RA5986; F, H, F, Cl, CF ₃ , Et], [RA5987; F, H, F, Cl, CF ₃ , Pr], [RA5988; F, H, F, Cl, CF ₃ , i-Pr], [RA5989; F, H , F, Cl, CF ₃ , c-Pr], [RA5990; F, H, F, Cl, CF ₃ , Bu], [RA5991; F, H, F, Cl, CF ₃ , i-Bu], [ RA5992; F, H, F, Cl, CF ₃ , t-Bu], [RA5993; F, H, F, Cl, CF ₃ , c-PrCH ₂ ], [RA5994; F, H, F, Cl, CF ₃ , Ph], [RA5995; F, H, F, Cl, CF ₃ , Bn], [RA5996; F, H, F, Cl, CF ₃ , CF ₃ ], [RA5997; F, H, F, Cl , CF ₃ , CF ₃ CH ₂ ], [RA5998; F, H, F, Cl, CF ₃ , CF ₃ CF ₂ ], [RA5999; F, H, F, Cl, CF ₃ , CF ₂ H], [RA6000; F, H, F, Cl, CF ₃ , CF ₂ HCH ₂ ],

[RA6001; F, H, Cl, H, CF ₃ , Me], [RA6002; F, H, Cl, H, CF ₃ , Et], [RA6003; F, H, Cl, H, CF ₃ , Pr] , [RA6004; F, H, Cl, H, CF ₃ , i-Pr], [RA6005; F, H, Cl, H, CF ₃ , c-Pr], [RA6006; F, H, Cl, H, CF ₃ , Bu], [RA6007; F, H, Cl, H, CF ₃ , i-Bu], [RA6008; F, H, Cl, H, CF ₃ , t-Bu], [RA6009; F, H , Cl, H, CF ₃ , c-PrCH ₂ ], [RA6010; F, H, Cl, H, CF ₃ , Ph], [RA6011; F, H, Cl, H, CF ₃ , Bn], [RA6012 ; F, H, Cl, H, CF ₃ , CF ₃ ], [RA6013; F, H, Cl, H, CF ₃ , CF ₃ CH ₂ ], [RA6014; F, H, Cl, H, CF ₃ , CF ₃ CF ₂ ], [RA6015; F, H, Cl, H, CF ₃ , CF ₂ H], [RA6016; F, H, Cl, H, CF ₃ , CF ₂ HCH ₂ ], [RA6017; F, H, Cl, Cl, CF ₃ , Me], [RA6018; F, H, Cl, Cl, CF ₃ , Et], [RA6019; F, H, Cl, Cl, CF ₃ , Pr], [RA6020; F , H, Cl, Cl, CF ₃ , i-Pr], [RA6021; F, H, Cl, Cl, CF ₃ , c-Pr], [RA6022; F, H, Cl, Cl, CF ₃ , Bu] , [RA6023; F, H, Cl, Cl, CF ₃ , i-Bu], [RA6024; F, H, Cl, Cl, CF ₃ , t-Bu], [RA6025; F, H, Cl, Cl, CF ₃ , c-PrCH ₂ ], [RA6026; F, H, Cl, Cl, CF ₃ , Ph], [RA6027; F, H, Cl, Cl, CF ₃ , Bn], [RA6028; F, H, Cl, Cl, CF ₃ , CF ₃ ], [RA6029; F, H, Cl, Cl, CF ₃ , CF ₃ CH ₂ ], [RA6030; F, H, Cl, Cl, CF ₃ , CF ₃ CF ₂ ] , [RA6031; F, H, Cl, Cl, CF ₃ , CF ₂ H], [RA6032; F, H, Cl, Cl, CF ₃ , CF ₂ HCH ₂ ], [RA6033; F, H, Me, H , CF ₂ HCH ₂ , Me], [RA6034; F, H, Me, H, CF ₂ HCH ₂ , Et], [RA6035; F, H, Me, H, CF ₂ HCH ₂ , Pr], [RA6036; F, H, Me, H, CF ₂ HCH ₂ , i-Pr], [RA6037; F, H, Me, H, CF ₂ HCH ₂ , c-Pr], [RA6038; F, H, Me, H, CF ₂ HCH ₂ , Bu], [RA6039; F, H, Me, H, CF ₂ HCH ₂ , i-Bu], [RA6040; F, H, Me, H, CF ₂ HCH ₂ , t-Bu], [RA6041; F , H, Me, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA6042; F, H, Me, H, CF ₂ HCH ₂ , Ph], [RA6043; F, H, Me, H, CF ₂ HCH ₂ , Bn], [RA6044; F, H, Me, H, CF ₂ HCH ₂ , CF ₃ ], [RA6045; F, H, Me, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA6046 ; F, H, Me, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA6047; F, H, Me, H, CF ₂ HCH ₂ , CF ₂ H], [RA6048; F, H, Me, H, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA6049; F, H, Me, Me, CF ₂ HCH ₂ , Me], [RA6050; F, H, Me, Me, CF ₂ HCH ₂ , Et] , [RA6051; F, H, Me, Me, CF ₂ HCH ₂ , Pr], [RA6052; F, H, Me, Me, CF ₂ HCH ₂ , i-Pr], [RA6053; F, H, Me, Me, CF ₂ HCH ₂ , c-Pr], [RA6054; F, H, Me, Me, CF ₂ HCH ₂ , Bu], [RA6055; F, H, Me, Me, CF ₂ HCH ₂ , i-Bu ], [RA6056; F, H, Me, Me, CF ₂ HCH ₂ , t-Bu], [RA6057; F, H, Me, Me, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA6058; F, H, Me, Me, CF ₂ HCH ₂ , Ph], [RA6059; F, H, Me, Me, CF ₂ HCH ₂ , Bn], [RA6060; F, H, Me, Me, CF ₂ HCH ₂ , CF ₃ ], [RA6061; F, H, Me, Me, CF ₂ HC H ₂ , CF ₃ CH ₂ ], [RA6062; F, H, Me, Me, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA6063; F, H, Me, Me, CF ₂ HCH ₂ , CF ₂ H ], [RA6064; F, H, Me, Me, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA6065; F, H, Me, Et, CF ₂ HCH ₂ , Me], [RA6066; F, H, Me, Et, CF ₂ HCH ₂ , Et], [RA6067; F, H, Me, Et, CF ₂ HCH ₂ , Pr], [RA6068; F, H, Me, Et, CF ₂ HCH ₂ , i-Pr ], [RA6069; F, H, Me, Et, CF ₂ HCH ₂ , c-Pr], [RA6070; F, H, Me, Et, CF ₂ HCH ₂ , Bu], [RA6071; F, H, Me , Et, CF ₂ HCH ₂ , i-Bu], [RA6072; F, H, Me, Et, CF ₂ HCH ₂ , t-Bu], [RA6073; F, H, Me, Et, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA6074; F, H, Me, Et, CF ₂ HCH ₂ , Ph], [RA6075; F, H, Me, Et, CF ₂ HCH ₂ , Bn], [RA6076; F, H , Me, Et, CF ₂ HCH ₂ , CF ₃ ], [RA6077; F, H, Me, Et, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA6078; F, H, Me, Et, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA6079; F, H, Me, Et, CF ₂ HCH ₂ , CF ₂ H], [RA6080; F, H, Me, Et, CF ₂ HCH ₂ , CF ₂ HCH ₂ ] , [RA6081; F, H, Me, F, CF ₂ HCH ₂ , Me], [RA6082; F, H, Me, F, CF ₂ HCH ₂ , Et], [RA6083; F, H, Me, F, CF ₂ HCH ₂ , Pr], [RA6084; F, H, Me, F, CF ₂ HCH ₂ , i-Pr], [RA6085; F, H, Me, F, CF ₂ HCH ₂ , c-Pr], [RA6086; F, H, Me, F, CF ₂ HCH ₂ , Bu], [RA6087; F, H, Me, F, CF ₂ HCH ₂ , i-Bu], [RA6088; F, H, Me, F , CF ₂ HCH ₂ , t-B u], [RA6089; F, H, Me, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA6090; F, H, Me, F, CF ₂ HCH ₂ , Ph], [RA6091; F, H , Me, F, CF ₂ HCH ₂ , Bn], [RA6092; F, H, Me, F, CF ₂ HCH ₂ , CF ₃ ], [RA6093; F, H, Me, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA6094; F, H, Me, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA6095; F, H, Me, F, CF ₂ HCH ₂ , CF ₂ H], [RA6096 ; F, H, Me, F, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA6097; F, H, Me, Cl, CF ₂ HCH ₂ , Me], [RA6098; F, H, Me, Cl, CF ₂ HCH ₂ , Et], [RA6099; F, H, Me, Cl, CF ₂ HCH ₂ , Pr], [RA6100; F, H, Me, Cl, CF ₂ HCH ₂ , i-Pr], [RA6101 ; F, H, Me, Cl, CF ₂ HCH ₂ , c-Pr], [RA6102; F, H, Me, Cl, CF ₂ HCH ₂ , Bu], [RA6103; F, H, Me, Cl, CF ₂ HCH ₂ , i-Bu], [RA6104; F, H, Me, Cl, CF ₂ HCH ₂ , t-Bu], [RA6105; F, H, Me, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA6106; F, H, Me, Cl, CF ₂ HCH ₂ , Ph], [RA6107; F, H, Me, Cl, CF ₂ HCH ₂ , Bn], [RA6108; F, H, Me, Cl , CF ₂ HCH ₂ , CF ₃ ], [RA6109; F, H, Me, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA6110; F, H, Me, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA6111; F, H, Me, Cl, CF ₂ HCH ₂ , CF ₂ H], [RA6112; F, H, Me, Cl, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA6113; F, H, Et, H, CF ₂ HCH ₂ , Me], [RA6114; F, H, Et, H, CF ₂ HCH ₂ , Et], [RA6115; F, H, Et, H, CF ₂ HCH ₂ , Pr], [RA6 116; F, H, Et, H, CF ₂ HCH ₂ , i-Pr], [RA6117; F, H, Et, H, CF ₂ HCH ₂ , c-Pr], [RA6118; F, H, Et, H, CF ₂ HCH ₂ , Bu], [RA6119; F, H, Et, H, CF ₂ HCH ₂ , i-Bu], [RA6120; F, H, Et, H, CF ₂ HCH ₂ , t-Bu ], [RA6121; F, H, Et, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA6122; F, H, Et, H, CF ₂ HCH ₂ , Ph], [RA6123; F, H, Et, H, CF ₂ HCH ₂ , Bn], [RA6124; F, H, Et, H, CF ₂ HCH ₂ , CF ₃ ], [RA6125; F, H, Et, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA6126; F, H, Et, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA6127; F, H, Et, H, CF ₂ HCH ₂ , CF ₂ H], [RA6128; F, H, Et, H, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA6129; F, H, Et, F, CF ₂ HCH ₂ , Me], [RA6130; F, H, Et, F, CF ₂ HCH ₂ , Et], [RA6131; F, H, Et, F, CF ₂ HCH ₂ , Pr], [RA6132; F, H, Et, F, CF ₂ HCH ₂ , i-Pr], [RA6133; F, H, Et, F, CF ₂ HCH ₂ , c-Pr], [RA6134; F, H, Et, F, CF ₂ HCH ₂ , Bu], [RA6135; F, H, Et, F, CF ₂ HCH ₂ , i-Bu], [RA6136; F, H, Et, F, CF ₂ HCH ₂ , t-Bu], [RA6137; F, H, Et, F, CF ₂ HCH ₂ , c-PrCH ₂ ] , [RA6138; F, H, Et, F, CF ₂ HCH ₂ , Ph], [RA6139; F, H, Et, F, CF ₂ HCH ₂ , Bn], [RA6140; F, H, Et, F, CF ₂ HCH ₂ , CF ₃ ], [RA6141; F, H, Et, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA6142; F, H, Et, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA6143; F, H, Et, F, CF ₂ HCH ₂ , CF ₂ H], [RA6144; F, H, Et, F, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA6145; F, H, Et, Cl, CF ₂ HCH ₂ , Me], [RA6146; F, H, Et, Cl, CF ₂ HCH ₂ , Et], [RA6147; F, H, Et, Cl, CF ₂ HCH ₂ , Pr], [RA6148; F, H, Et, Cl, CF ₂ HCH ₂ , i -Pr], [RA6149; F, H, Et, Cl, CF ₂ HCH ₂ , c-Pr], [RA6150; F, H, Et, Cl, CF ₂ HCH ₂ , Bu], [RA6151; F, H , Et, Cl, CF ₂ HCH ₂ , i-Bu], [RA6152; F, H, Et, Cl, CF ₂ HCH ₂ , t-Bu], [RA6153; F, H, Et, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA6154; F, H, Et, Cl, CF ₂ HCH ₂ , Ph], [RA6155; F, H, Et, Cl, CF ₂ HCH ₂ , Bn], [RA6156; F , H, Et, Cl, CF ₂ HCH ₂ , CF ₃ ], [RA6157; F, H, Et, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA6158; F, H, Et, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA6159; F, H, Et, Cl, CF ₂ HCH ₂ , CF ₂ H], [RA6160; F, H, Et, Cl, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA6161; F, H, F, H, CF ₂ HCH ₂ , Me], [RA6162; F, H, F, H, CF ₂ HCH ₂ , Et], [RA6163; F, H, F, H, CF ₂ HCH ₂ , Pr], [RA6164; F, H, F, H, CF ₂ HCH ₂ , i-Pr], [RA6165; F, H, F, H, CF ₂ HCH ₂ , c-Pr ], [RA6166; F, H, F, H, CF ₂ HCH ₂ , Bu], [RA6167; F, H, F, H, CF ₂ HCH ₂ , i-Bu], [RA6168; F, H, F , H, CF ₂ HCH ₂ , t-Bu], [RA6169; F, H, F, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA6170; F, H, F, H, CF ₂ HCH ₂ , Ph], [RA6171; F, H, F, H, CF ₂ HCH ₂ , Bn], [RA6172; F, H, F, H, CF ₂ HCH ₂ , CF ₃ ], [RA6173; F, H, F, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA6174; F , H, F, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA6175; F, H, F, H, CF ₂ HCH ₂ , CF ₂ H], [RA6176; F, H, F, H, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA6177; F, H, F, F, CF ₂ HCH ₂ , Me], [RA6178; F, H, F, F, CF ₂ HCH ₂ , Et], [ RA6179; F, H, F, F, CF ₂ HCH ₂ , Pr], [RA6180; F, H, F, F, CF ₂ HCH ₂ , i-Pr], [RA6181; F, H, F, F, CF ₂ HCH ₂ , c-Pr], [RA6182; F, H, F, F, CF
₂ HCH ₂ , Bu], [RA6183; F, H, F, F, CF ₂ HCH ₂ , i-Bu], [RA6184; F, H, F, F, CF ₂ HCH ₂ , t-Bu], [ RA6185; F, H, F, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA6186; F, H, F, F, CF ₂ HCH ₂ , Ph], [RA6187; F, H, F, F , CF ₂ HCH ₂ , Bn], [RA6188; F, H, F, F, CF ₂ HCH ₂ , CF ₃ ], [RA6189; F, H, F, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ] , [RA6190; F, H, F, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA6191; F, H, F, F, CF ₂ HCH ₂ , CF ₂ H], [RA6192; F, H , F, F, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA6193; F, H, F, Cl, CF ₂ HCH ₂ , Me], [RA6194; F, H, F, Cl, CF ₂ HCH ₂ , Et], [RA6195; F, H, F, Cl, CF ₂ HCH ₂ , Pr], [RA6196; F, H, F, Cl, CF ₂ HCH ₂ , i-Pr], [RA6197; F, H , F, Cl, CF ₂ HCH ₂ , c-Pr], [RA6198; F, H, F, Cl, CF ₂ HCH ₂ , Bu], [RA6199; F, H, F, Cl, CF ₂ HCH ₂ , i-Bu], [RA6200; F, H, F, Cl, CF ₂ HCH ₂ , t-Bu],

[RA6201; F, H, F, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA6202; F, H, F, Cl, CF ₂ HCH ₂ , Ph], [RA6203; F, H, F, Cl, CF ₂ HCH ₂ , Bn], [RA6204; F, H, F, Cl, CF ₂ HCH ₂ , CF ₃ ], [RA6205; F, H, F, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA6206; F, H, F, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA6207; F, H, F, Cl, CF ₂ HCH ₂ , CF ₂ H], [RA6208; F, H, F, Cl, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA6209; F, H, Cl, H, CF ₂ HCH ₂ , Me], [RA6210; F, H, Cl, H, CF ₂ HCH ₂ , Et], [RA6211; F, H, Cl, H, CF ₂ HCH ₂ , Pr], [RA6212; F, H, Cl, H, CF ₂ HCH ₂ , i-Pr], [RA6213; F, H, Cl, H, CF ₂ HCH ₂ , c-Pr], [RA6214; F, H, Cl, H, CF ₂ HCH ₂ , Bu], [RA6215; F, H, Cl, H, CF ₂ HCH ₂ , i-Bu], [RA6216; F, H, Cl, H, CF ₂ HCH ₂ , t-Bu], [RA6217; F, H, Cl, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [ RA6218; F, H, Cl, H, CF ₂ HCH ₂ , Ph], [RA6219; F, H, Cl, H, CF ₂ HCH ₂ , Bn], [RA6220; F, H, Cl, H, CF ₂ HCH ₂ , CF ₃ ], [RA6221; F, H, Cl, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA6222; F, H, Cl, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ] , [RA6223; F, H, Cl, H, CF ₂ HCH ₂ , CF ₂ H], [RA6224; F, H, Cl, H, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA6225; F, H , Cl, Cl, CF ₂ HCH ₂ , Me], [RA6226; F, H, Cl, Cl, CF ₂ HCH ₂ , Et], [RA6227; F, H, Cl, Cl, CF ₂ HCH ₂ , Pr] , [RA6228; F, H, Cl, Cl, CF ₂ HCH ₂ , i-Pr], [RA6229; F, H, Cl, Cl, CF ₂ HCH ₂ , c-Pr], [RA6230; F, H, Cl, Cl, CF ₂ HCH ₂ , Bu], [ RA6231; F, H, Cl, Cl, CF ₂ HCH ₂ , i-Bu], [RA6232; F, H, Cl, Cl, CF ₂ HCH ₂ , t-Bu], [RA6233; F, H, Cl, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA6234; F, H, Cl, Cl, CF ₂ HCH ₂ , Ph], [RA6235; F, H, Cl, Cl, CF ₂ HCH ₂ , Bn] , [RA6236; F, H, Cl, Cl, CF ₂ HCH ₂ , CF ₃ ], [RA6237; F, H, Cl, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA6238; F, H, Cl, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA6239; F, H, Cl, Cl, CF ₂ HCH ₂ , CF ₂ H], [RA6240; F, H, Cl, Cl, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA6241; F, H, Me, H, CF ₃ CH ₂ , Me], [RA6242; F, H, Me, H, CF ₃ CH ₂ , Et], [RA6243; F , H, Me, H, CF ₃ CH ₂ , Pr], [RA6244; F, H, Me, H, CF ₃ CH ₂ , i-Pr], [RA6245; F, H, Me, H, CF ₃ CH ₂ , c-Pr], [RA6246; F, H, Me, H, CF ₃ CH ₂ , Bu], [RA6247; F, H, Me, H, CF ₃ CH ₂ , i-Bu], [RA6248; F, H, Me, H, CF ₃ CH ₂ , t-Bu], [RA6249; F, H, Me, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RA6250; F, H, Me, H , CF ₃ CH ₂ , Ph], [RA6251; F, H, Me, H, CF ₃ CH ₂ , Bn], [RA6252; F, H, Me, H, CF ₃ CH ₂ , CF ₃ ], [RA6253 ; F, H, Me, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA6254; F, H, Me, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA6255; F, H, Me , H, CF ₃ CH ₂ , CF ₂ H], [RA6256; F, H, M e, H, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA6257; F, H, Me, Me, CF ₃ CH ₂ , Me], [RA6258; F, H, Me, Me, CF ₃ CH ₂ , Et], [RA6259; F, H, Me, Me, CF ₃ CH ₂ , Pr], [RA6260; F, H, Me, Me, CF ₃ CH ₂ , i-Pr], [RA6261; F, H, Me, Me, CF ₃ CH ₂ , c-Pr], [RA6262; F, H, Me, Me, CF ₃ CH ₂ , Bu], [RA6263; F, H, Me, Me, CF ₃ CH ₂ , i -Bu], [RA6264; F, H, Me, Me, CF ₃ CH ₂ , t-Bu], [RA6265; F, H, Me, Me, CF ₃ CH ₂ , c-PrCH ₂ ], [RA6266; F, H, Me, Me, CF ₃ CH ₂ , Ph], [RA6267; F, H, Me, Me, CF ₃ CH ₂ , Bn], [RA6268; F, H, Me, Me, CF ₃ CH ₂ , CF ₃ ], [RA6269; F, H, Me, Me, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA6270; F, H, Me, Me, CF ₃ CH ₂ , CF ₃ CF ₂ ], [ RA6271; F, H, Me, Me, CF ₃ CH ₂ , CF ₂ H], [RA6272; F, H, Me, Me, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA6273; F, H, Me , Et, CF ₃ CH ₂ , Me], [RA6274; F, H, Me, Et, CF ₃ CH ₂ , Et], [RA6275; F, H, Me, Et, CF ₃ CH ₂ , Pr], [ RA6276; F, H, Me, Et, CF ₃ CH ₂ , i-Pr], [RA6277; F, H, Me, Et, CF ₃ CH ₂ , c-Pr], [RA6278; F, H, Me, Et, CF ₃ CH ₂ , Bu], [RA6279; F, H, Me, Et, CF ₃ CH ₂ , i-Bu], [RA6280; F, H, Me, Et, CF ₃ CH ₂ , t-Bu ], [RA6281; F, H, Me, Et, CF ₃ CH ₂ , c-PrCH ₂ ], [RA6282; F, H, Me, Et, CF ₃ CH ₂ , Ph], [RA6283; F, H, Me, Et, CF ₃ CH ₂ , Bn], [RA6284; F, H, Me, Et, C F ₃ CH ₂ , CF ₃ ], [RA6285; F, H, Me, Et, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA6286; F, H, Me, Et, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA6287; F, H, Me, Et, CF ₃ CH ₂ , CF ₂ H], [RA6288; F, H, Me, Et, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA6289; F , H, Me, F, CF ₃ CH ₂ , Me], [RA6290; F, H, Me, F, CF ₃ CH ₂ , Et], [RA6291; F, H, Me, F, CF ₃ CH ₂ , Pr], [RA6292; F, H, Me, F, CF ₃ CH ₂ , i-Pr], [RA6293; F, H, Me, F, CF ₃ CH ₂ , c-Pr], [RA6294; F, H, Me, F, CF ₃ CH ₂ , Bu], [RA6295; F, H, Me, F, CF ₃ CH ₂ , i-Bu], [RA6296; F, H, Me, F, CF ₃ CH ₂ , t-Bu], [RA6297; F, H, Me, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RA6298; F, H, Me, F, CF ₃ CH ₂ , Ph], [RA6299; F, H, Me, F, CF ₃ CH ₂ , Bn], [RA6300; F, H, Me, F, CF ₃ CH ₂ , CF ₃ ], [RA6301; F, H, Me, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA6302; F, H, Me, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA6303; F, H, Me, F, CF ₃ CH ₂ , CF ₂ H] , [RA6304; F, H, Me, F, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA6305; F, H, Me, Cl, CF ₃ CH ₂ , Me], [RA6306; F, H, Me , Cl, CF ₃ CH ₂ , Et], [RA6307; F, H, Me, Cl, CF ₃ CH ₂ , Pr], [RA6308; F, H, Me, Cl, CF ₃ CH ₂ , i-Pr] , [RA6309; F, H, Me, Cl, CF ₃ CH ₂ , c-Pr], [RA6310; F, H, Me, Cl, CF ₃ CH ₂ , Bu], [RA6311; F, H, Me, Cl, CF ₃ CH ₂ , i-Bu], [RA6312; F, H, Me, Cl, CF ₃ CH ₂ , t-Bu], [RA6313; F, H, Me, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RA6314; F, H, Me, Cl, CF ₃ CH ₂ , Ph], [RA6315 ; F, H, Me, Cl, CF ₃ CH ₂ , Bn], [RA6316; F, H, Me, Cl, CF ₃ CH ₂ , CF ₃ ], [RA6317; F, H, Me, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA6318; F, H, Me, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA6319; F, H, Me, Cl, CF ₃ CH ₂ , CF ₂ H ], [RA6320; F, H, Me, Cl, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA6321; F, H, Et, H, CF ₃ CH ₂ , Me], [RA6322; F, H, Et, H, CF ₃ CH ₂ , Et], [RA6323; F, H, Et, H, CF ₃ CH ₂ , Pr], [RA6324; F, H, Et, H, CF ₃ CH ₂ , i-Pr ], [RA6325; F, H, Et, H, CF ₃ CH ₂ , c-Pr], [RA6326; F, H, Et, H, CF ₃ CH ₂ , Bu], [RA6327; F, H, Et , H, CF ₃ CH ₂ , i-Bu], [RA6328; F, H, Et, H, CF ₃ CH ₂ , t-Bu], [RA6329; F, H, Et, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RA6330; F, H, Et, H, CF ₃ CH ₂ , Ph], [RA6331; F, H, Et, H, CF ₃ CH ₂ , Bn], [RA6332; F, H , Et, H, CF ₃ CH ₂ , CF ₃ ], [RA6333; F, H, Et, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA6334; F, H, Et, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA6335; F, H, Et, H, CF ₃ CH ₂ , CF ₂ H], [RA6336; F, H, Et, H, CF ₃ CH ₂ , CF ₂ HCH ₂ ] , [RA6337; F, H, Et, F, CF ₃ CH ₂ , Me], [RA6338; F, H, Et, F, CF ₃ CH ₂ , Et], [RA6339; F, H, Et, F, CF ₃ CH ₂ , Pr], [RA6340; F, H, Et, F, CF ₃ CH ₂ , i-Pr] , [RA6341; F, H, Et, F, CF ₃ CH ₂ , c-Pr], [RA6342; F, H, Et, F, CF ₃ CH ₂ , Bu], [RA6343; F, H, Et, F, CF ₃ CH ₂ , i-Bu], [RA6344; F, H, Et, F, CF ₃ CH ₂ , t-Bu], [RA6345; F, H, Et, F, CF ₃ CH ₂ , c -PrCH ₂ ], [RA6346; F, H, Et, F, CF ₃ CH ₂ , Ph], [RA6347; F, H, Et, F, CF ₃ CH ₂ , Bn], [RA6348; F, H, Et, F, CF ₃ CH ₂ , CF ₃ ], [RA6349; F, H, Et, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA6350; F, H, Et, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA6351; F, H, Et, F, CF ₃ CH ₂ , CF ₂ H], [RA6352; F, H, Et, F, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA6353; F, H, Et, Cl, CF ₃ CH ₂ , Me], [RA6354; F, H, Et, Cl, CF ₃ CH ₂ , Et], [RA6355; F, H, Et, Cl, CF ₃ CH ₂ , Pr], [RA6356; F, H, Et, Cl, CF ₃ CH ₂ , i-Pr], [RA6357; F, H, Et, Cl, CF ₃ CH ₂ , c-Pr], [ RA6358; F, H, Et, Cl, CF ₃ CH ₂ , Bu], [RA6359; F, H, Et, Cl, CF ₃ CH ₂ , i-Bu], [RA6360; F, H, Et, Cl, CF ₃ CH ₂ , t-Bu], [RA6361; F, H, Et, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RA6362; F, H, Et, Cl, CF ₃ CH ₂ , Ph] , [RA6363; F, H, Et, Cl, CF ₃ CH ₂ , Bn], [RA6364; F, H, Et, Cl, CF ₃ CH ₂ , CF ₃ ], [RA6365; F, H, Et, Cl , CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA6366; F, H, Et, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA6367; F, H, Et, Cl, CF ₃ CH ₂ , CF ₂ H], [RA6368; F, H, Et, Cl, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA6369; F, H, F, H, CF ₃ CH ₂ , Me], [RA6370; F, H, F, H, CF ₃ CH ₂ , Et], [RA6371; F, H, F, H, CF ₃ CH ₂ , Pr], [RA6372; F, H, F, H, CF ₃ CH ₂ , i-Pr], [RA6373; F, H, F, H, CF ₃ CH ₂ , c-Pr ], [RA6374; F, H, F, H, CF ₃ CH ₂ , Bu], [RA6375; F, H, F, H, CF
₃ CH ₂ , i-Bu], [RA6376; F, H, F, H, CF ₃ CH ₂ , t-Bu], [RA6377; F, H, F, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RA6378; F, H, F, H, CF ₃ CH ₂ , Ph], [RA6379; F, H, F, H, CF ₃ CH ₂ , Bn], [RA6380; F, H, F, H , CF ₃ CH ₂ , CF ₃ ], [RA6381; F, H, F, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA6382; F, H, F, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA6383; F, H, F, H, CF ₃ CH ₂ , CF ₂ H], [RA6384; F, H, F, H, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA6385; F, H, F, F, CF ₃ CH ₂ , Me], [RA6386; F, H, F, F, CF ₃ CH ₂ , Et], [RA6387; F, H, F, F, CF ₃ CH ₂ , Pr], [RA6388; F, H, F, F, CF ₃ CH ₂ , i-Pr], [RA6389; F, H, F, F, CF ₃ CH ₂ , c-Pr], [RA6390; F , H, F, F, CF ₃ CH ₂ , Bu], [RA6391; F, H, F, F, CF ₃ CH ₂ , i-Bu], [RA6392; F, H, F, F, CF ₃ CH ₂ , t-Bu], [RA6393; F, H, F, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RA6394; F, H, F, F, CF ₃ CH ₂ , Ph], [RA6395 ; F, H, F, F, CF ₃ CH ₂ , Bn], [RA6396; F, H, F, F, CF ₃ CH ₂ , CF ₃ ], [RA6397; F, H, F, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA6398; F, H, F, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA6399; F, H, F, F, CF ₃ CH ₂ , CF ₂ H ], [RA6400; F, H, F, F, CF ₃ CH ₂ , CF ₂ HCH ₂ ],

[RA6401; F, H, F, Cl, CF ₃ CH ₂ , Me], [RA6402; F, H, F, Cl, CF ₃ CH ₂ , Et], [RA6403; F, H, F, Cl, CF ₃ CH ₂ , Pr], [RA6404; F, H, F, Cl, CF ₃ CH ₂ , i-Pr], [RA6405; F, H, F, Cl, CF ₃ CH ₂ , c-Pr], [ RA6406; F, H, F, Cl, CF ₃ CH ₂ , Bu], [RA6407; F, H, F, Cl, CF ₃ CH ₂ , i-Bu], [RA6408; F, H, F, Cl, CF ₃ CH ₂ , t-Bu], [RA6409; F, H, F, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RA6410; F, H, F, Cl, CF ₃ CH ₂ , Ph] , [RA6411; F, H, F, Cl, CF ₃ CH ₂ , Bn], [RA6412; F, H, F, Cl, CF ₃ CH ₂ , CF ₃ ], [RA6413; F, H, F, Cl , CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA6414; F, H, F, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA6415; F, H, F, Cl, CF ₃ CH ₂ , CF ₂ H], [RA6416; F, H, F, Cl, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA6417; F, H, Cl, H, CF ₃ CH ₂ , Me], [RA6418; F , H, Cl, H, CF ₃ CH ₂ , Et], [RA6419; F, H, Cl, H, CF ₃ CH ₂ , Pr], [RA6420; F, H, Cl, H, CF ₃ CH ₂ , i-Pr], [RA6421; F, H, Cl, H, CF ₃ CH ₂ , c-Pr], [RA6422; F, H, Cl, H, CF ₃ CH ₂ , Bu], [RA6423; F, H, Cl, H, CF ₃ CH ₂ , i-Bu], [RA6424; F, H, Cl, H, CF ₃ CH ₂ , t-Bu], [RA6425; F, H, Cl, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RA6426; F, H, Cl, H, CF ₃ CH ₂ , Ph], [RA6427; F, H, Cl, H, CF ₃ CH ₂ , Bn], [RA6428; F, H, Cl, H, CF ₃ CH ₂ , CF ₃ ], [RA6429; F, H, Cl, H, CF ₃ CH ₂ , CF ₃ CH ₂ ] , [RA6430; F, H, Cl, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA6431; F, H, Cl, H, CF ₃ CH ₂ , CF ₂ H], [RA6432; F, H , Cl, H, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA6433; F, H, Cl, Cl, CF ₃ CH ₂ , Me], [RA6434; F, H, Cl, Cl, CF ₃ CH ₂ , Et], [RA6435; F, H, Cl, Cl, CF ₃ CH ₂ , Pr], [RA6436; F, H, Cl, Cl, CF ₃ CH ₂ , i-Pr], [RA6437; F, H , Cl, Cl, CF ₃ CH ₂ , c-Pr], [RA6438; F, H, Cl, Cl, CF ₃ CH ₂ , Bu], [RA6439; F, H, Cl, Cl, CF ₃ CH ₂ , i-Bu], [RA6440; F, H, Cl, Cl, CF ₃ CH ₂ , t-Bu], [RA6441; F, H, Cl, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RA6442 ; F, H, Cl, Cl, CF ₃ CH ₂ , Ph], [RA6443; F, H, Cl, Cl, CF ₃ CH ₂ , Bn], [RA6444; F, H, Cl, Cl, CF ₃ CH ₂ , CF ₃ ], [RA6445; F, H, Cl, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA6446; F, H, Cl, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA6447; F, H, Cl, Cl, CF ₃ CH ₂ , CF ₂ H], [RA6448; F, H, Cl, Cl, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA6449; F, H, Me, H, HCCCH ₂ , Me], [RA6450; F, H, Me, H, HCCCH ₂ , Et], [RA6451; F, H, Me, H, HCCCH ₂ , Pr], [RA6452; F, H , Me, H, HCCCH ₂ , i-Pr], [RA6453; F, H, Me, H, HCCCH ₂ , c-Pr], [RA6454; F, H, Me, H, HCCCH ₂ , Bu], [ RA6455; F, H, Me, H, HCCCH ₂ , i-Bu], [RA6456; F, H, Me, H, HCCCH ₂ , t-Bu], [RA6457; F, H, Me, H, HCCCH ₂ , c-PrCH ₂ ], [RA6458; F, H, Me, H, HCCCH ₂ , Ph], [RA6459; F, H, Me, H, HCCCH ₂ , Bn], [RA6460; F, H, Me, H, HCCCH ₂ , CF ₃ ], [RA6461; F, H, Me, H , HCCCH ₂ , CF ₃ CH ₂ ], [RA6462; F, H, Me, H, HCCCH ₂ , CF ₃ CF ₂ ], [RA6463; F, H, Me, H, HCCCH ₂ , CF ₂ H], [ RA6464; F, H, Me, H, HCCCH ₂ , CF ₂ HCH ₂ ], [RA6465; F, H, Me, Me, HCCCH ₂ , Me], [RA6466; F, H, Me, Me, HCCCH ₂ , Et], [RA6467; F, H, Me, Me, HCCCH ₂ , Pr], [RA6468; F, H, Me, Me, HCCCH ₂ , i-Pr], [RA6469; F, H, Me, Me, HCCCH ₂ , c-Pr], [RA6470; F, H, Me, Me, HCCCH ₂ , Bu], [RA6471; F, H, Me, Me, HCCCH ₂ , i-Bu], [RA6472; F, H , Me, Me, HCCCH ₂ , t-Bu], [RA6473; F, H, Me, Me, HCCCH ₂ , c-PrCH ₂ ], [RA6474; F, H, Me, Me, HCCCH ₂ , Ph], [RA6475; F, H, Me, Me, HCCCH ₂ , Bn], [RA6476; F, H, Me, Me, HCCCH ₂ , CF ₃ ], [RA6477; F, H, Me, Me, HCCCH ₂ , CF ₃ CH ₂ ], [RA6478; F, H, Me, Me, HCCCH ₂ , CF ₃ CF ₂ ], [RA6479; F, H, Me, Me, HCCCH ₂ , CF ₂ H], [RA6480; F, H , Me, Me, HCCCH ₂ , CF ₂ HCH ₂ ], [RA6481; F, H, Me, Et, HCCCH ₂ , Me], [RA6482; F, H, Me, Et, HCCCH ₂ , Et], [RA6483 ; F, H, Me, Et, HCCCH ₂ , Pr], [RA6484; F, H, Me, Et, HCCCH ₂ , i-Pr], [RA6485; F, H, Me, Et, HCCCH ₂ , c- Pr], [RA6486; F, H, Me, Et, HCCCH ₂ , Bu], [RA6487; F, H, Me, Et, HCCCH ₂ , i-Bu], [RA6488; F, H, Me , Et, HCCCH ₂ , t-Bu], [RA6489; F, H, Me, Et, HCCCH ₂ , c-PrCH ₂ ], [RA6490; F, H, Me, Et, HCCCH ₂ , Ph], [RA6491 ; F, H, Me, Et, HCCCH ₂ , Bn], [RA6492; F, H, Me, Et, HCCCH ₂ , CF ₃ ], [RA6493; F, H, Me, Et, HCCCH ₂ , CF ₃ CH ₂ ], [RA6494; F, H, Me, Et, HCCCH ₂ , CF ₃ CF ₂ ], [RA6495; F, H, Me, Et, HCCCH ₂ , CF ₂ H], [RA6496; F, H, Me , Et, HCCCH ₂ , CF ₂ HCH ₂ ], [RA6497; F, H, Me, F, HCCCH ₂ , Me], [RA6498; F, H, Me, F, HCCCH ₂ , Et], [RA6499; F , H, Me, F, HCCCH ₂ , Pr], [RA6500; F, H, Me, F, HCCCH ₂ , i-Pr], [RA6501; F, H, Me, F, HCCCH ₂ , c-Pr] , [RA6502; F, H, Me, F, HCCCH ₂ , Bu], [RA6503; F, H, Me, F, HCCCH ₂ , i-Bu], [RA6504; F, H, Me, F, HCCCH ₂ , t-Bu], [RA6505; F, H, Me, F, HCCCH ₂ , c-PrCH ₂ ], [RA6506; F, H, Me, F, HCCCH ₂ , Ph], [RA6507; F, H, Me, F, HCCCH ₂ , Bn], [RA6508; F, H, Me, F, HCCCH ₂ , CF ₃ ], [RA6509; F, H, Me, F, HCCCH ₂ , CF ₃ CH ₂ ], [RA6510 ; F, H, Me, F, HCCCH ₂ , CF ₃ CF ₂ ], [RA6511; F, H, Me, F, HCCCH ₂ , CF ₂ H], [RA6512; F, H, Me, F, HCCCH ₂ , CF ₂ HCH ₂ ], [RA6513; F, H, Me, Cl, HCCCH ₂ , Me], [RA6514; F, H, Me, Cl, HCCCH ₂ , Et], [RA6515; F, H, Me, Cl, HCCCH ₂ , Pr], [RA6516; F, H, Me, Cl, HCCCH ₂ , i-Pr], [RA6517; F, H, Me, Cl, HCCCH ₂ , c-Pr], [RA6518; F, H, Me, Cl, HCCCH ₂ , Bu], [RA6519; F, H, Me, Cl, HCCCH ₂ , i-Bu], [RA6520; F, H, Me, Cl, HCCCH ₂ , t-Bu ], [RA6521; F, H, Me, Cl, HCCCH ₂ , c-PrCH ₂ ], [RA6522; F, H, Me, Cl, HCCCH ₂ , Ph], [RA6523; F, H, Me, Cl, HCCCH ₂ , Bn], [RA6524; F, H, Me, Cl, HCCCH ₂ , CF ₃ ], [RA6525; F, H, Me, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RA6526; F, H , Me, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RA6527; F, H, Me, Cl, HCCCH ₂ , CF ₂ H], [RA6528; F, H, Me, Cl, HCCCH ₂ , CF ₂ HCH ₂ ], [RA6529; F, H, Et, H, HCCCH ₂ , Me], [RA6530; F, H, Et, H, HCCCH ₂ , Et], [RA6531; F, H, Et, H, HCCCH ₂ , Pr], [RA6532; F, H, Et, H, HCCCH ₂ , i-Pr], [RA6533; F, H, Et, H, HCCCH ₂ , c-Pr], [RA6534; F, H, Et , H, HCCCH ₂ , Bu], [RA6535; F, H, Et, H, HCCCH ₂ , i-Bu], [RA6536; F, H, Et, H, HCCCH ₂ , t-Bu], [RA6537; F, H, Et, H, HCCCH ₂ , c-PrCH ₂ ], [RA6538; F, H, Et, H, HCCCH ₂ , Ph], [RA6539; F, H, Et, H, HCCCH ₂ , Bn] , [RA6540; F, H, Et, H, HCCCH ₂ , CF ₃ ], [RA6541; F, H, Et, H, HCCCH ₂ , CF ₃ CH ₂ ], [RA6542; F, H, Et, H, HCCCH ₂ , CF ₃ CF ₂ ], [RA6543; F, H, Et, H, HCCCH ₂ , CF ₂ H], [RA6544; F, H, Et, H, HCCCH ₂ , CF ₂ HCH ₂ ], [RA6545 ; F, H, Et, F, HCCCH ₂ , Me], [RA6546; F, H, Et, F, HCCCH ₂ , Et], [RA6547; F, H, Et, F, HCCCH ₂ , Pr], [ RA6548 ; F, H, Et, F, HCCCH ₂ , i-Pr], [RA6549; F, H, Et, F, HCCCH ₂ , c-Pr], [RA6550; F, H, Et, F, HCCCH ₂ , Bu], [RA6551; F, H, Et, F, HCCCH ₂ , i-Bu], [RA6552; F, H, Et, F, HCCCH ₂ , t-Bu], [RA6553; F, H, Et, F, HCCCH ₂ , c-PrCH ₂ ], [RA6554; F, H, Et, F, HCCCH ₂ , Ph], [RA6555; F, H, Et, F, HCCCH ₂ , Bn], [RA6556; F, H, Et, F, HCCCH ₂ , CF ₃ ], [RA6557; F, H, Et, F, HCCCH ₂ , CF ₃ CH ₂ ], [RA6558; F, H, Et, F, HCCCH ₂ , CF ₃ CF ₂ ], [RA6559; F, H, Et, F, HCCCH ₂ , CF ₂ H], [RA6560; F, H, Et, F, HCCCH ₂ , CF ₂ HCH ₂ ], [RA6561; F, H, Et , Cl, HCCCH ₂ , Me], [RA6562; F, H, Et, Cl, HCCCH ₂ , Et], [RA6563; F, H, Et, Cl, HCCCH ₂ , Pr], [RA6564; F, H, Et, Cl, HCCCH ₂ , i-Pr], [RA6565; F, H, Et, Cl, HCCCH ₂ , c-Pr], [RA6566; F, H, Et, Cl, HCCCH ₂ , Bu], [RA6567 ; F, H, Et, Cl, HCCCH ₂ , i-Bu], [RA6568; F, H, Et, Cl, HCCCH ₂ , t-Bu], [RA6569; F, H, Et, Cl, HCCCH ₂ , c-PrCH ₂ ], [RA6570; F, H, Et, Cl, HCCCH ₂ , Ph], [RA6571; F, H, Et, Cl, HCCCH ₂ , Bn], [RA6572; F, H, Et, Cl , HCCCH ₂ , CF ₃ ], [RA6573; F, H, Et, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RA6574; F, H, Et, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RA6575 ; F, H, Et, Cl, HCCCH ₂ , CF ₂ H], [RA6576; F, H, Et, Cl, HCCCH ₂ , CF ₂ HCH ₂ ], [RA6577; F, H, F, H, HCCCH ₂ , Me ], [RA6578; F, H, F, H, HCCCH ₂ , Et], [RA6579; F, H, F, H, HCCCH ₂ , Pr], [RA6580; F, H, F, H, HCCCH ₂ , i-Pr], [RA6581; F, H, F, H, HCCCH ₂ , c-Pr], [RA6582; F, H, F, H, HCCCH ₂ , Bu], [RA6583; F, H, F, H, HCCCH ₂ , i-Bu], [RA6584; F, H, F, H, HCCCH ₂ , t-Bu], [RA6585; F, H, F, H, HCCCH ₂ , c-PrCH ₂ ], [ RA6586; F, H, F, H, HCCCH ₂ , Ph], [RA6587; F, H, F, H, HCCCH ₂ , Bn], [RA6588; F, H, F, H, HCCCH ₂ , CF ₃ ] , [RA6589; F, H, F, H, HCCCH ₂ , CF ₃ CH ₂ ], [RA6590; F, H, F, H, HCCCH ₂ , CF ₃ CF ₂ ], [RA6591; F, H, F, H, HCCCH ₂ , CF ₂ H], [RA6592; F, H, F, H, HCCCH ₂ , CF ₂ HCH ₂ ], [RA6593; F, H, F, F, HCCCH ₂ , Me], [RA6594; F, H, F, F, HCCCH ₂ , Et], [RA6595; F, H, F, F, HCCCH ₂ , Pr], [RA6596; F, H, F, F, HCCCH ₂ , i-Pr], [RA6597; F, H, F, F, HCCCH ₂ , c-Pr], [RA6598; F, H, F, F, HCCCH ₂ , Bu], [RA6599; F, H, F, F, HCCCH ₂ , i-Bu], [RA6600; F, H, F, F, HCCCH ₂ , t-Bu],

[RA6601; F, H, F, F, HCCCH ₂ , c-PrCH ₂ ], [RA6602; F, H, F, F, HCCCH ₂ , Ph], [RA6603; F, H, F, F, HCCCH ₂ , Bn], [RA6604; F, H, F, F, HCCCH ₂ , CF ₃ ], [RA6605; F, H, F, F, HCCCH ₂ , CF ₃ CH ₂ ], [RA6606; F, H, F , F, HCCCH ₂ , CF ₃ CF ₂ ], [RA6607; F, H, F, F, HCCCH ₂ , CF ₂ H], [RA6608; F, H, F, F, HCCCH ₂ , CF ₂ HCH ₂ ] , [RA6609; F, H, F, Cl, HCCCH ₂ , Me], [RA6610; F, H, F, Cl, HCCCH ₂ , Et], [RA6611; F, H, F, Cl, HCCCH ₂ , Pr ], [RA6612; F, H, F, Cl, HCCCH ₂ , i-Pr], [RA6613; F, H, F, Cl, HCCCH ₂ , c-Pr], [RA6614; F, H, F, Cl , HCCCH ₂ , Bu], [RA6615; F, H, F, Cl, HCCCH ₂ , i-Bu], [RA6616; F, H, F, Cl, HCCCH ₂ , t-Bu], [RA6617; F, H, F, Cl, HCCCH ₂ , c-PrCH ₂ ], [RA6618; F, H, F, Cl, HCCCH ₂ , Ph], [RA6619; F, H, F, Cl, HCCCH ₂ , Bn], [ RA6620; F, H, F, Cl, HCCCH ₂ , CF ₃ ], [RA6621; F, H, F, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RA6622; F, H, F, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RA6623; F, H, F, Cl, HCCCH ₂ , CF ₂ H], [RA6624; F, H, F, Cl, HCCCH ₂ , CF ₂ HCH ₂ ], [RA6625; F , H, Cl, H, HCCCH ₂ , Me], [RA6626; F, H, Cl, H, HCCCH ₂ , Et], [RA6627; F, H, Cl, H, HCCCH ₂ , Pr], [RA6628; F, H, Cl, H, HCCCH ₂ , i-Pr], [RA6629; F, H, Cl, H, HCCCH ₂ , c-Pr], [RA6630; F, H, Cl, H, HCCCH ₂ , Bu ], [RA6631; F, H, Cl, H, H CCCH ₂ , i-Bu], [RA6632; F, H, Cl, H, HCCCH ₂ , t-Bu], [RA6633; F, H, Cl, H, HCCCH ₂ , c-PrCH ₂ ], [RA6634; F, H, Cl, H, HCCCH ₂ , Ph], [RA6635; F, H, Cl, H, HCCCH ₂ , Bn], [RA6636; F, H, Cl, H, HCCCH ₂ , CF ₃ ], [ RA6637; F, H, Cl, H, HCCCH ₂ , CF ₃ CH ₂ ], [RA6638; F, H, Cl, H, HCCCH ₂ , CF ₃ CF ₂ ], [RA6639; F, H, Cl, H, HCCCH ₂ , CF ₂ H], [RA6640; F, H, Cl, H, HCCCH ₂ , CF ₂ HCH ₂ ], [RA6641; F, H, Cl, Cl, HCCCH ₂ , Me], [RA6642; F, H, Cl, Cl, HCCCH ₂ , Et], [RA6643; F, H, Cl, Cl, HCCCH ₂ , Pr], [RA6644; F, H, Cl, Cl, HCCCH ₂ , i-Pr], [RA6645 ; F, H, Cl, Cl, HCCCH ₂ , c-Pr], [RA6646; F, H, Cl, Cl, HCCCH ₂ , Bu], [RA6647; F, H, Cl, Cl, HCCCH ₂ , i- Bu], [RA6648; F, H, Cl, Cl, HCCCH ₂ , t-Bu], [RA6649; F, H, Cl, Cl, HCCCH ₂ , c-PrCH ₂ ], [RA6650; F, H, Cl , Cl, HCCCH ₂ , Ph], [RA6651; F, H, Cl, Cl, HCCCH ₂ , Bn], [RA6652; F, H, Cl, Cl, HCCCH ₂ , CF ₃ ], [RA6653; F, H , Cl, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RA6654; F, H, Cl, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RA6655; F, H, Cl, Cl, HCCCH ₂ , CF ₂ H], [RA6656; F, H, Cl, Cl, HCCCH ₂ , CF ₂ HCH ₂ ], [RA6657; F, H, Me, H, CH ₃ CCCH ₂ , Me], [RA6658; F, H, Me , H, CH ₃ CCCH ₂ , Et], [RA6659; F, H, Me, H, CH ₃ CCCH ₂ , Pr], [RA6660; F, H, Me, H, CH ₃ CCCH ₂ , i-Pr], [RA6661; F, H, Me, H, CH ₃ CCCH ₂ , c-Pr], [RA6662; F, H, Me, H, CH ₃ CCCH ₂ , Bu], [RA6663; F, H, Me, H, CH ₃ CCCH ₂ , i-Bu], [RA6664; F, H, Me, H, CH ₃ CCCH ₂ , t-Bu], [RA6665; F, H, Me, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA6666; F, H, Me, H, CH ₃ CCCH ₂ , Ph], [RA6667; F, H, Me, H, CH ₃ CCCH ₂ , Bn], [RA6668; F, H, Me, H, CH ₃ CCCH ₂ , CF ₃ ], [RA6669; F, H, Me, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA6670; F, H, Me, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA6671; F, H, Me, H, CH ₃ CCCH ₂ , CF ₂ H], [RA6672; F, H, Me, H, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA6673; F, H, Me, Me, CH ₃ CCCH ₂ , Me], [RA6674; F, H, Me, Me, CH ₃ CCCH ₂ , Et], [RA6675; F, H, Me , Me, CH ₃ CCCH ₂ , Pr], [RA6676; F, H, Me, Me, CH ₃ CCCH ₂ , i-Pr], [RA6677; F, H, Me, Me, CH ₃ CCCH ₂ , c- Pr], [RA6678; F, H, Me, Me, CH ₃ CCCH ₂ , Bu], [RA6679; F, H, Me, Me, CH ₃ CCCH ₂ , i-Bu], [RA6680; F, H, Me, Me, CH ₃ CCCH ₂ , t-Bu], [RA6681; F, H, Me, Me, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA6682; F, H, Me, Me, CH ₃ CCCH ₂ , Ph], [RA6683; F, H, Me, Me, CH ₃ CCCH ₂ , Bn], [RA6684; F, H, Me, Me, CH ₃ CCCH ₂ , CF ₃ ], [RA6685; F, H , Me, Me, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA6686; F, H, Me, Me, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA6687; F, H, Me, Me , CH ₃ CCCH ₂ , CF ₂ H], [RA6688; F, H, Me, Me, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA6689; F, H, Me, Et, CH ₃ CCCH ₂ , Me ], [RA6690; F, H, Me, Et, CH ₃ CCCH ₂ , Et], [RA6691; F, H, Me, Et, CH ₃ CCCH ₂ , Pr], [RA6692; F, H, Me, Et , CH ₃ CCCH ₂ , i-Pr], [RA6693; F, H, Me, Et, CH ₃ CCCH ₂ , c-Pr], [RA6694; F, H, Me, Et, CH ₃ CCCH ₂ , Bu] , [RA6695; F, H, Me, Et, CH ₃ CCCH ₂ , i-Bu], [RA6696; F, H, Me, Et, CH ₃ CCCH ₂ , t-Bu], [RA6697; F, H, Me, Et, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA6698; F, H, Me, Et, CH ₃ CCCH ₂ , Ph], [RA6699; F, H, Me, Et, CH ₃ CCCH ₂ , Bn], [RA6700; F, H, Me, Et, CH ₃ CCCH ₂ , CF ₃ ], [RA6701; F, H, Me, Et, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA6702; F, H, Me, Et, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA6703; F, H, Me, Et, CH ₃ CCCH ₂ , CF ₂ H], [RA6704; F, H, Me, Et, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA6705; F, H, Me, F, CH ₃ CCCH ₂ , Me], [RA6706; F, H, Me, F, CH ₃ CCCH ₂ , Et], [RA6707 ; F, H, Me, F, CH ₃ CCCH ₂ , Pr], [RA6708; F, H, Me, F, CH ₃ CCCH ₂ , i-Pr], [RA6709; F, H, Me, F, CH ₃ CCCH ₂ , c-Pr], [RA6710; F, H, Me, F, CH ₃ CCCH ₂ , Bu], [RA6711; F, H, Me, F, CH ₃ CCCH ₂ , i-Bu], [ RA6712; F, H, Me, F, CH ₃ CCCH ₂ , t-Bu], [RA6713; F, H, Me, F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA671 4; F, H, Me, F, CH ₃ CCCH ₂ , Ph], [RA6715; F, H, Me, F, CH ₃ CCCH ₂ , Bn], [RA6716; F, H, Me, F, CH ₃ CCCH ₂ , CF ₃ ], [RA6717; F, H, Me, F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA6718; F, H, Me, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ] , [RA6719; F, H, Me, F, CH ₃ CCCH ₂ , CF ₂ H], [RA6720; F, H, Me, F, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA6721; F, H , Me, Cl, CH ₃ CCCH ₂ , Me], [RA6722; F, H, Me, Cl, CH ₃ CCCH ₂ , Et], [RA6723; F, H, Me, Cl, CH ₃ CCCH ₂ , Pr] , [RA6724; F, H, Me, Cl, CH ₃ CCCH ₂ , i-Pr], [RA6725; F, H, Me, Cl, CH ₃ CCCH ₂ , c-Pr], [RA6726; F, H, Me, Cl, CH ₃ CCCH ₂ , Bu], [RA6727; F, H, Me, Cl, CH ₃ CCCH ₂ , i-Bu], [RA6728; F, H, Me, Cl, CH ₃ CCCH ₂ , t -Bu], [RA6729; F, H, Me, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA6730; F, H, Me, Cl, CH ₃ CCCH ₂ , Ph], [RA6731; F, H, Me, Cl, CH ₃ CCCH ₂ , Bn], [RA6732; F, H, Me, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RA6733; F, H, Me, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA6734; F, H, Me, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA6735; F, H, Me, Cl, CH ₃ CCCH ₂ , CF ₂ H], [ RA6736; F, H, Me, Cl, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA6737; F, H, Et, H, CH ₃ CCCH ₂ , Me], [RA6738; F, H, Et, H , CH ₃ CCCH ₂ , Et], [RA6739; F, H, Et, H, CH ₃ CCCH ₂ , Pr], [RA6740; F, H, Et, H, CH ₃ CCCH ₂ , i-Pr], [RA6741; F, H, Et, H, CH ₃ CCCH ₂ , c-Pr], [RA6742; F, H, Et, H, CH ₃ CCCH ₂ , Bu], [RA6743; F, H, Et, H, CH ₃ CCCH ₂ , i-Bu], [RA6744; F, H, Et, H, CH ₃ CCCH ₂ , t-Bu], [RA6745; F, H, Et, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA6746; F, H, Et, H, CH ₃ CCCH ₂ , Ph], [RA6747; F, H, Et, H, CH ₃ CCCH ₂ , Bn], [ RA6748; F, H, Et, H, CH ₃ CCCH ₂ , CF ₃ ], [RA6749; F, H, Et, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA6750; F, H, Et, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA6751; F, H, Et, H, CH ₃ CCCH ₂ , CF ₂ H], [RA6752; F, H, Et, H, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA6753; F, H, Et, F, CH ₃ CCCH ₂ , Me], [RA6754; F, H, Et, F, CH ₃ CCCH ₂ , Et], [RA6755; F, H , Et, F, CH ₃ CCCH ₂ , Pr], [RA6756; F, H, Et, F, CH ₃ CCCH ₂ , i-Pr], [RA6757; F, H, Et, F, CH ₃ CCCH ₂ , c-Pr], [RA6758; F, H, Et, F, CH ₃ CCCH ₂ , Bu], [RA6759; F, H, Et, F, CH ₃ CCCH ₂ , i-Bu], [RA6760; F, H, Et, F, CH ₃ CCCH ₂ , t-Bu], [RA6761; F, H, Et, F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA6762; F, H, Et, F, CH ₃ CCCH ₂ , Ph], [RA6763; F, H, Et, F, CH ₃ CCCH ₂ , Bn], [RA6764; F, H, Et, F, CH ₃ CCCH ₂ , CF ₃ ], [RA6765; F , H, Et, F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA6766; F, H, Et, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA6767; F, H, Et, F , CH ₃ CCCH ₂ , CF ₂ H], [RA6768; F, H, Et, F, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA6769; F, H, Et, Cl, CH ₃ CCCH ₂ , Me], [RA6770; F, H, Et, Cl, CH ₃ CCCH ₂ , Et], [RA6771; F, H, Et, Cl, CH ₃ CCCH ₂ , Pr], [RA6772; F, H, Et, Cl, CH ₃ CCCH ₂ , i-Pr], [RA6773; F, H, Et, Cl, CH ₃ CCCH ₂ , c-Pr], [RA6774; F, H, Et, Cl, CH ₃ CCCH ₂ , Bu], [RA6775; F , H, Et, Cl, CH ₃ CCCH ₂ , i-Bu], [RA6776; F, H, Et, Cl, CH ₃ CCCH ₂ , t-Bu], [RA6777; F, H, Et, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA6778; F, H, Et, Cl, CH ₃ CCCH ₂ , Ph], [RA6779; F, H, Et, Cl, CH ₃ CCCH ₂ , Bn], [RA6780 ; F, H, Et, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RA6781; F, H, Et, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA6782; F, H, Et, Cl , CH ₃
CCCH ₂ , CF ₃ CF ₂ ], [RA6783; F, H, Et, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RA6784; F, H, Et, Cl, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA6785; F, H, F, H, CH ₃ CCCH ₂ , Me], [RA6786; F, H, F, H, CH ₃ CCCH ₂ , Et], [RA6787; F, H, F, H , CH ₃ CCCH ₂ , Pr], [RA6788; F, H, F, H, CH ₃ CCCH ₂ , i-Pr], [RA6789; F, H, F, H, CH ₃ CCCH ₂ , c-Pr] , [RA6790; F, H, F, H, CH ₃ CCCH ₂ , Bu], [RA6791; F, H, F, H, CH ₃ CCCH ₂ , i-Bu], [RA6792; F, H, F, H, CH ₃ CCCH ₂ , t-Bu], [RA6793; F, H, F, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA6794; F, H, F, H, CH ₃ CCCH ₂ , Ph], [RA6795; F, H, F, H, CH ₃ CCCH ₂ , Bn], [RA6796; F, H, F, H, CH ₃ CCCH ₂ , CF ₃ ], [RA6797; F, H, F , H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA6798; F, H, F, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA6799; F, H, F, H, CH ₃ CCCH ₂ , CF ₂ H], [RA6800; F, H, F, H, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ],

[RA6801; F, H, F, F, CH ₃ CCCH ₂ , Me], [RA6802; F, H, F, F, CH ₃ CCCH ₂ , Et], [RA6803; F, H, F, F, CH ₃ CCCH ₂ , Pr], [RA6804; F, H, F, F, CH ₃ CCCH ₂ , i-Pr], [RA6805; F, H, F, F, CH ₃ CCCH ₂ , c-Pr], [ RA6806; F, H, F, F, CH ₃ CCCH ₂ , Bu], [RA6807; F, H, F, F, CH ₃ CCCH ₂ , i-Bu], [RA6808; F, H, F, F, CH ₃ CCCH ₂ , t-Bu], [RA6809; F, H, F, F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA6810; F, H, F, F, CH ₃ CCCH ₂ , Ph] , [RA6811; F, H, F, F, CH ₃ CCCH ₂ , Bn], [RA6812; F, H, F, F, CH ₃ CCCH ₂ , CF ₃ ], [RA6813; F, H, F, F , CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA6814; F, H, F, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA6815; F, H, F, F, CH ₃ CCCH ₂ , CF ₂ H], [RA6816; F, H, F, F, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA6817; F, H, F, Cl, CH ₃ CCCH ₂ , Me], [RA6818; F , H, F, Cl, CH ₃ CCCH ₂ , Et], [RA6819; F, H, F, Cl, CH ₃ CCCH ₂ , Pr], [RA6820; F, H, F, Cl, CH ₃ CCCH ₂ , i-Pr], [RA6821; F, H, F, Cl, CH ₃ CCCH ₂ , c-Pr], [RA6822; F, H, F, Cl, CH ₃ CCCH ₂ , Bu], [RA6823; F, H, F, Cl, CH ₃ CCCH ₂ , i-Bu], [RA6824; F, H, F, Cl, CH ₃ CCCH ₂ , t-Bu], [RA6825; F, H, F, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA6826; F, H, F, Cl, CH ₃ CCCH ₂ , Ph], [RA6827; F, H, F, Cl, CH ₃ CCCH ₂ , Bn], [RA6828; F, H, F, Cl, CH ₃ CCCH ₂ , CF ₃ ] , [RA6829; F, H, F, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA6830; F, H, F, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA6831; F, H, F, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RA6832; F, H, F, Cl, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA6833; F, H, Cl, H, CH ₃ CCCH ₂ , Me], [RA6834; F, H, Cl, H, CH ₃ CCCH ₂ , Et], [RA6835; F, H, Cl, H, CH ₃ CCCH ₂ , Pr], [RA6836; F, H, Cl, H, CH ₃ CCCH ₂ , i-Pr], [RA6837; F, H, Cl, H, CH ₃ CCCH ₂ , c-Pr], [RA6838; F, H, Cl, H, CH ₃ CCCH ₂ , Bu], [RA6839; F, H, Cl, H, CH ₃ CCCH ₂ , i-Bu], [RA6840; F, H, Cl, H, CH ₃ CCCH ₂ , t-Bu], [RA6841 ; F, H, Cl, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA6842; F, H, Cl, H, CH ₃ CCCH ₂ , Ph], [RA6843; F, H, Cl, H, CH ₃ CCCH ₂ , Bn], [RA6844; F, H, Cl, H, CH ₃ CCCH ₂ , CF ₃ ], [RA6845; F, H, Cl, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA6846; F, H, Cl, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA6847; F, H, Cl, H, CH ₃ CCCH ₂ , CF ₂ H], [RA6848; F, H, Cl, H, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA6849; F, H, Cl, Cl, CH ₃ CCCH ₂ , Me], [RA6850; F, H, Cl, Cl, CH ₃ CCCH ₂ , Et], [RA6851; F, H, Cl, Cl, CH ₃ CCCH ₂ , Pr], [RA6852; F, H, Cl, Cl, CH ₃ CCCH ₂ , i-Pr], [RA6853; F, H, Cl, Cl, CH ₃ CCCH ₂ , c-Pr], [RA6854; F, H, Cl, Cl, CH ₃ CCCH ₂ , Bu], [RA6855; F, H, Cl, Cl, CH ₃ CCCH ₂ , i-Bu], [RA6856; F, H, Cl, Cl, CH ₃ CCCH ₂ , t-Bu], [RA6857; F, H, Cl, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [ RA6858; F, H, Cl, Cl, CH ₃ CCCH ₂ , Ph], [RA6859; F, H, Cl, Cl, CH ₃ CCCH ₂ , Bn], [RA6860; F, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RA6861; F, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA6862; F, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ] , [RA6863; F, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RA6864; F, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA6865; F, H , Me, H, c-PrCH ₂ , Me], [RA6866; F, H, Me, H, c-PrCH ₂ , Et], [RA6867; F, H, Me, H, c-PrCH ₂ , Pr] , [RA6868; F, H, Me, H, c-PrCH ₂ , i-Pr], [RA6869; F, H, Me, H, c-PrCH ₂ , c-Pr], [RA6870; F, H, Me, H, c-PrCH ₂ , Bu], [RA6871; F, H, Me, H, c-PrCH ₂ , i-Bu], [RA6872; F, H, Me, H, c-PrCH ₂ , t -Bu], [RA6873; F, H, Me, H, c-PrCH ₂ , c-PrCH ₂ ], [RA6874; F, H, Me, H, c-PrCH ₂ , Ph], [RA6875; F, H, Me, H, c-PrCH ₂ , Bn], [RA6876; F, H, Me, H, c-PrCH ₂ , CF ₃ ], [RA6877; F, H, Me, H, c-PrCH ₂ , CF ₃ CH ₂ ], [RA6878; F, H, Me, H, c-PrCH ₂ , CF ₃ CF ₂ ], [RA6879; F, H, Me, H, c-PrCH ₂ , CF ₂ H], [ RA6880; F, H, Me, H, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA6881; F, H, Me, Me, c-PrCH ₂ , Me], [RA6882; F, H, Me, Me , c-PrCH ₂ , Et], [RA6883; F, H, Me, Me, c-PrCH ₂ , P r], [RA6884; F, H, Me, Me, c-PrCH ₂ , i-Pr], [RA6885; F, H, Me, Me, c-PrCH ₂ , c-Pr], [RA6886; F, H, Me, Me, c-PrCH ₂ , Bu], [RA6887; F, H, Me, Me, c-PrCH ₂ , i-Bu], [RA6888; F, H, Me, Me, c-PrCH ₂ , t-Bu], [RA6889; F, H, Me, Me, c-PrCH ₂ , c-PrCH ₂ ], [RA6890; F, H, Me, Me, c-PrCH ₂ , Ph], [RA6891; F, H, Me, Me, c-PrCH ₂ , Bn], [RA6892; F, H, Me, Me, c-PrCH ₂ , CF ₃ ], [RA6893; F, H, Me, Me, c-PrCH ₂ , CF ₃ CH ₂ ], [RA6894; F, H, Me, Me, c-PrCH ₂ , CF ₃ CF ₂ ], [RA6895; F, H, Me, Me, c-PrCH ₂ , CF ₂ H] , [RA6896; F, H, Me, Me, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA6897; F, H, Me, Et, c-PrCH ₂ , Me], [RA6898; F, H, Me , Et, c-PrCH ₂ , Et], [RA6899; F, H, Me, Et, c-PrCH ₂ , Pr], [RA6900; F, H, Me, Et, c-PrCH ₂ , i-Pr] , [RA6901; F, H, Me, Et, c-PrCH ₂ , c-Pr], [RA6902; F, H, Me, Et, c-PrCH ₂ , Bu], [RA6903; F, H, Me, Et, c-PrCH ₂ , i-Bu], [RA6904; F, H, Me, Et, c-PrCH ₂ , t-Bu], [RA6905; F, H, Me, Et, c-PrCH ₂ , c -PrCH ₂ ], [RA6906; F, H, Me, Et, c-PrCH ₂ , Ph], [RA6907; F, H, Me, Et, c-PrCH ₂ , Bn], [RA6908; F, H, Me, Et, c-PrCH ₂ , CF ₃ ], [RA6909; F, H, Me, Et, c-PrCH ₂ , CF ₃ CH ₂ ], [RA6910; F, H, Me, Et, c-PrCH ₂ , CF ₃ CF ₂ ], [RA6911; F, H, Me, Et, c-PrCH ₂ , CF ₂ H], [RA6912; F, H, Me, E t, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA6913; F, H, Me, F, c-PrCH ₂ , Me], [RA6914; F, H, Me, F, c-PrCH ₂ , Et] , [RA6915; F, H, Me, F, c-PrCH ₂ , Pr], [RA6916; F, H, Me, F, c-PrCH ₂ , i-Pr], [RA6917; F, H, Me, F, c-PrCH ₂ , c-Pr], [RA6918; F, H, Me, F, c-PrCH ₂ , Bu], [RA6919; F, H, Me, F, c-PrCH ₂ , i-Bu ], [RA6920; F, H, Me, F, c-PrCH ₂ , t-Bu], [RA6921; F, H, Me, F, c-PrCH ₂ , c-PrCH ₂ ], [RA6922; F, H, Me, F, c-PrCH ₂ , Ph], [RA6923; F, H, Me, F, c-PrCH ₂ , Bn], [RA6924; F, H, Me, F, c-PrCH ₂ , CF ₃ ], [RA6925; F, H, Me, F, c-PrCH ₂ , CF ₃ CH ₂ ], [RA6926; F, H, Me, F, c-PrCH ₂ , CF ₃ CF ₂ ], [RA6927; F, H, Me, F, c-PrCH ₂ , CF ₂ H], [RA6928; F, H, Me, F, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA6929; F, H, Me, Cl , c-PrCH ₂ , Me], [RA6930; F, H, Me, Cl, c-PrCH ₂ , Et], [RA6931; F, H, Me, Cl, c-PrCH ₂ , Pr], [RA6932; F, H, Me, Cl, c-PrCH ₂ , i-Pr], [RA6933; F, H, Me, Cl, c-PrCH ₂ , c-Pr], [RA6934; F, H, Me, Cl, c-PrCH ₂ , Bu], [RA6935; F, H, Me, Cl, c-PrCH ₂ , i-Bu], [RA6936; F, H, Me, Cl, c-PrCH ₂ , t-Bu], [RA6937; F, H, Me, Cl, c-PrCH ₂ , c-PrCH ₂ ], [RA6938; F, H, Me, Cl, c-PrCH ₂ , Ph], [RA6939; F, H, Me, Cl, c-PrCH ₂ , Bn], [RA6940; F, H, Me, Cl, c-PrCH ₂ , CF ₃ ], [RA6941; F, H, Me, Cl, c-PrCH ₂ , CF ₃ CH ₂ ], [RA6942; F, H, Me, Cl, c-PrCH ₂ , CF ₃ CF ₂ ], [RA6943; F, H, Me, Cl, c-PrCH ₂ , CF ₂ H], [RA6944 ; F, H, Me, Cl, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA6945; F, H, Et, H, c-PrCH ₂ , Me], [RA6946; F, H, Et, H, c-PrCH ₂ , Et], [RA6947; F, H, Et, H, c-PrCH ₂ , Pr], [RA6948; F, H, Et, H, c-PrCH ₂ , i-Pr], [RA6949 ; F, H, Et, H, c-PrCH ₂ , c-Pr], [RA6950; F, H, Et, H, c-PrCH ₂ , Bu], [RA6951; F, H, Et, H, c -PrCH ₂ , i-Bu], [RA6952; F, H, Et, H, c-PrCH ₂ , t-Bu], [RA6953; F, H, Et, H, c-PrCH ₂ , c-PrCH ₂ ], [RA6954; F, H, Et, H, c-PrCH ₂ , Ph], [RA6955; F, H, Et, H, c-PrCH ₂ , Bn], [RA6956; F, H, Et, H , c-PrCH ₂ , CF ₃ ], [RA6957; F, H, Et, H, c-PrCH ₂ , CF ₃ CH ₂ ], [RA6958; F, H, Et, H, c-PrCH ₂ , CF ₃ CF ₂ ], [RA6959; F, H, Et, H, c-PrCH ₂ , CF ₂ H], [RA6960; F, H, Et, H, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA6961; F, H, Et, F, c-PrCH ₂ , Me], [RA6962; F, H, Et, F, c-PrCH ₂ , Et], [RA6963; F, H, Et, F, c-PrCH ₂ , Pr], [RA6964; F, H, Et, F, c-PrCH ₂ , i-Pr], [RA6965; F, H, Et, F, c-PrCH ₂ , c-Pr], [RA6966; F , H, Et, F, c-PrCH ₂ , Bu], [RA6967; F, H, Et, F, c-PrCH ₂ , i-Bu], [RA6968; F, H, Et, F, c-PrCH ₂ , t-Bu], [RA6969; F, H, Et, F, c-PrCH ₂ , c-PrCH ₂ ], [RA6970; F, H, Et, F, c-PrCH ₂ , Ph], [RA69 71; F, H, Et, F, c-PrCH ₂ , Bn], [RA6972; F, H, Et, F, c-PrCH ₂ , CF ₃ ], [RA6973; F, H, Et, F, c -PrCH ₂ , CF ₃ CH ₂ ], [RA6974; F, H, Et, F, c-PrCH ₂ , CF ₃ CF ₂ ], [RA6975; F, H, Et, F, c-PrCH ₂ , CF ₂ H], [RA6976; F, H, Et, F, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA6977; F, H, Et, Cl, c-PrCH ₂ , Me], [RA6978; F, H , Et, Cl, c-PrCH ₂ , Et], [RA6979; F, H, Et, Cl, c-PrCH ₂ , Pr], [RA6980; F, H, Et, Cl, c-PrCH ₂ , i- Pr], [RA6981; F, H, Et, Cl, c-PrCH ₂ , c-Pr], [RA6982; F, H, Et, Cl, c-PrCH ₂ , Bu], [RA6983; F, H, Et, Cl, c-PrCH ₂ , i-Bu], [RA6984; F, H, Et, Cl, c-PrCH ₂ , t-Bu], [RA6985; F, H, Et, Cl, c-PrCH ₂ , c-PrCH ₂ ], [RA6986; F, H, Et, Cl, c-PrCH ₂ , Ph], [RA6987; F, H, Et, Cl, c-PrCH ₂ , Bn], [RA6988; F, H, Et, Cl, c-PrCH ₂ , CF ₃ ], [RA6989; F, H, Et, Cl, c-PrCH ₂ , CF ₃ CH ₂ ], [RA6990; F, H, Et, Cl, c- PrCH ₂ , CF ₃ CF ₂ ], [RA6991; F, H, Et, Cl, c-PrCH ₂ , CF ₂ H], [RA6992; F, H, Et, Cl, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA6993; F, H, F, H, c-PrCH ₂ , Me], [RA6994; F, H, F, H, c-PrCH ₂ , Et], [RA6995; F, H, F, H , c-PrCH ₂ , Pr], [RA6996; F, H, F, H, c-PrCH ₂ , i-Pr], [RA6997; F, H, F, H, c-PrCH ₂ ,
c-Pr], [RA6998; F, H, F, H, c-PrCH ₂ , Bu], [RA6999; F, H, F, H, c-PrCH ₂ , i-Bu], [RA7000; F, H, F, H, c-PrCH ₂ , t-Bu],
[RA7001; F, H, F, H, c-PrCH ₂ , c-PrCH ₂ ], [RA7002; F, H, F, H, c-PrCH ₂ , Ph], [RA7003; F, H, F, H, c-PrCH ₂ , Bn], [RA7004; F, H, F, H, c-PrCH ₂ , CF ₃ ], [RA7005; F, H, F, H, c-PrCH ₂ , CF ₃ CH ₂ ], [RA7006; F, H, F, H, c-PrCH ₂ , CF ₃ CF ₂ ], [RA7007; F, H, F, H, c-PrCH ₂ , CF ₂ H], [RA7008; F, H, F, H, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA7009; F, H, F, F, c-PrCH ₂ , Me], [RA7010; F, H, F, F, c-PrCH ₂ , Et], [RA7011; F, H, F, F, c-PrCH ₂ , Pr], [RA7012; F, H, F, F, c-PrCH ₂ , i-Pr], [RA7013; F, H, F, F, c-PrCH ₂ , c-Pr], [RA7014; F, H, F, F, c-PrCH ₂ , Bu], [RA7015; F, H, F, F, c-PrCH ₂ , i-Bu], [RA7016; F, H, F, F, c-PrCH ₂ , t-Bu], [RA7017; F, H, F, F, c-PrCH ₂ , c-PrCH ₂ ], [ RA7018; F, H, F, F, c-PrCH ₂ , Ph], [RA7019; F, H, F, F, c-PrCH ₂ , Bn], [RA7020; F, H, F, F, c- PrCH ₂ , CF ₃ ], [RA7021; F, H, F, F, c-PrCH ₂ , CF ₃ CH ₂ ], [RA7022; F, H, F, F, c-PrCH ₂ , CF ₃ CF ₂ ] , [RA7023; F, H, F, F, c-PrCH ₂ , CF ₂ H], [RA7024; F, H, F, F, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA7025; F, H , F, Cl, c-PrCH ₂ , Me], [RA7026; F, H, F, Cl, c-PrCH ₂ , Et], [RA7027; F, H, F, Cl, c-PrCH ₂ , Pr] , [RA7028; F, H, F, Cl, c-PrCH ₂ , i-Pr], [RA7029; F, H, F, Cl, c-PrCH ₂ , c-Pr], [RA7030; F, H, F, Cl, c-PrCH ₂ , Bu], [RA7 031; F, H, F, Cl, c-PrCH ₂ , i-Bu], [RA7032; F, H, F, Cl, c-PrCH ₂ , t-Bu], [RA7033; F, H, F, Cl, c-PrCH ₂ , c-PrCH ₂ ], [RA7034; F, H, F, Cl, c-PrCH ₂ , Ph], [RA7035; F, H, F, Cl, c-PrCH ₂ , Bn] , [RA7036; F, H, F, Cl, c-PrCH ₂ , CF ₃ ], [RA7037; F, H, F, Cl, c-PrCH ₂ , CF ₃ CH ₂ ], [RA7038; F, H, F, Cl, c-PrCH ₂ , CF ₃ CF ₂ ], [RA7039; F, H, F, Cl, c-PrCH ₂ , CF ₂ H], [RA7040; F, H, F, Cl, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA7041; F, H, Cl, H, c-PrCH ₂ , Me], [RA7042; F, H, Cl, H, c-PrCH ₂ , Et], [RA7043; F , H, Cl, H, c-PrCH ₂ , Pr], [RA7044; F, H, Cl, H, c-PrCH ₂ , i-Pr], [RA7045; F, H, Cl, H, c-PrCH _{2, c-Pr], [} RA7046; F, H, Cl, H, c-PrCH 2, Bu], [RA7047; F, H, Cl, H, c-PrCH 2, i-Bu], [RA7048; F, H, Cl, H, c-PrCH ₂ , t-Bu], [RA7049; F, H, Cl, H, c-PrCH ₂ , c-PrCH ₂ ], [RA7050; F, H, Cl, H , c-PrCH ₂ , Ph], [RA7051; F, H, Cl, H, c-PrCH ₂ , Bn], [RA7052; F, H, Cl, H, c-PrCH ₂ , CF ₃ ], [RA7053 ; F, H, Cl, H, c-PrCH ₂ , CF ₃ CH ₂ ], [RA7054; F, H, Cl, H, c-PrCH ₂ , CF ₃ CF ₂ ], [RA7055; F, H, Cl , H, c-PrCH ₂ , CF ₂ H], [RA7056; F, H, Cl, H, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA7057; F, H, Cl, Cl, c-PrCH ₂ , Me], [RA7058; F, H, Cl, Cl, c-PrCH ₂ , Et], [RA7059; F, H, Cl, Cl, c-PrCH ₂ , Pr], [RA7060; F, H, Cl, Cl, c-PrCH ₂ , i-Pr], [RA7061; F, H, Cl, Cl, c-PrCH ₂ , c-Pr], [RA7062; F, H, Cl, Cl, c-PrCH ₂ , Bu], [RA7063; F, H, Cl, Cl, c-PrCH ₂ , i-Bu], [RA7064; F, H, Cl, Cl, c-PrCH ₂ , t-Bu], [RA7065; F , H, Cl, Cl, c-PrCH ₂ , c-PrCH ₂ ], [RA7066; F, H, Cl, Cl, c-PrCH ₂ , Ph], [RA7067; F, H, Cl, Cl, c- PrCH ₂ , Bn], [RA7068; F, H, Cl, Cl, c-PrCH ₂ , CF ₃ ], [RA7069; F, H, Cl, Cl, c-PrCH ₂ , CF ₃ CH ₂ ], [RA7070 ; F, H, Cl, Cl, c-PrCH ₂ , CF ₃ CF ₂ ], [RA7071; F, H, Cl, Cl, c-PrCH ₂ , CF ₂ H], [RA7072; F, H, Cl, Cl, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA7073; F, H, Me, H, Bn, Me], [RA7074; F, H, Me, H, Bn, Et], [RA7075; F, H, Me, H, Bn, Pr], [RA7076; F, H, Me, H, Bn, i-Pr], [RA7077; F, H, Me, H, Bn, c-Pr], [RA7078; F, H, Me, H, Bn, Bu], [RA7079; F, H, Me, H, Bn, i-Bu], [RA7080; F, H, Me, H, Bn, t-Bu], [ RA7081; F, H, Me, H, Bn, c-PrCH ₂ ], [RA7082; F, H, Me, H, Bn, Ph], [RA7083; F, H, Me, H, Bn, Bn], [RA7084; F, H, Me, H, Bn, CF ₃ ], [RA7085; F, H, Me, H, Bn, CF ₃ CH ₂ ], [RA7086; F, H, Me, H, Bn, CF ₃ CF ₂ ], [RA7087; F, H, Me, H, Bn, CF ₂ H], [RA7088; F, H, Me, H, Bn, CF ₂ HCH ₂ ], [RA7089; F, H, Me , Me, Bn, Me], [RA7090; F, H, Me, Me, Bn, Et], [RA7091; F, H, Me, Me, Bn, Pr], [RA7092; F, H, Me, Me , Bn, i-Pr], [RA7093; F, H, Me, M e, Bn, c-Pr], [RA7094; F, H, Me, Me, Bn, Bu], [RA7095; F, H, Me, Me, Bn, i-Bu], [RA7096; F, H, Me, Me, Bn, t-Bu], [RA7097; F, H, Me, Me, Bn, c-PrCH ₂ ], [RA7098; F, H, Me, Me, Bn, Ph], [RA7099; F , H, Me, Me, Bn, Bn], [RA7100; F, H, Me, Me, Bn, CF ₃ ], [RA7101; F, H, Me, Me, Bn, CF ₃ CH ₂ ], [RA7102 ; F, H, Me, Me, Bn, CF ₃ CF ₂ ], [RA7103; F, H, Me, Me, Bn, CF ₂ H], [RA7104; F, H, Me, Me, Bn, CF ₂ HCH ₂ ], [RA7105; F, H, Me, Et, Bn, Me], [RA7106; F, H, Me, Et, Bn, Et], [RA7107; F, H, Me, Et, Bn, Pr ], [RA7108; F, H, Me, Et, Bn, i-Pr], [RA7109; F, H, Me, Et, Bn, c-Pr], [RA7110; F, H, Me, Et, Bn , Bu], [RA7111; F, H, Me, Et, Bn, i-Bu], [RA7112; F, H, Me, Et, Bn, t-Bu], [RA7113; F, H, Me, Et , Bn, c-PrCH ₂ ], [RA7114; F, H, Me, Et, Bn, Ph], [RA7115; F, H, Me, Et, Bn, Bn], [RA7116; F, H, Me, Et, Bn, CF ₃ ], [RA7117; F, H, Me, Et, Bn, CF ₃ CH ₂ ], [RA7118; F, H, Me, Et, Bn, CF ₃ CF ₂ ], [RA7119; F , H, Me, Et, Bn, CF ₂ H], [RA7120; F, H, Me, Et, Bn, CF ₂ HCH ₂ ], [RA7121; F, H, Me, F, Bn, Me], [ RA7122; F, H, Me, F, Bn, Et], [RA7123; F, H, Me, F, Bn, Pr], [RA7124; F, H, Me, F, Bn, i-Pr], [ RA7125; F, H, Me, F, Bn, c-Pr], [RA7126; F, H, Me, F, Bn, Bu], [RA7127; F, H, Me, F, Bn, i-Bu] , [RA7128; F, H, Me, F, Bn, t-Bu], [RA7129; F, H, Me, F, Bn, c-Pr CH ₂ ], [RA7130; F, H, Me, F, Bn, Ph], [RA7131; F, H, Me, F, Bn, Bn], [RA7132; F, H, Me, F, Bn, CF ₃ ], [RA7133; F, H, Me, F, Bn, CF ₃ CH ₂ ], [RA7134; F, H, Me, F, Bn, CF ₃ CF ₂ ], [RA7135; F, H, Me, F, Bn, CF ₂ H], [RA7136; F, H, Me, F, Bn, CF ₂ HCH ₂ ], [RA7137; F, H, Me, Cl, Bn, Me], [RA7138; F, H , Me, Cl, Bn, Et], [RA7139; F, H, Me, Cl, Bn, Pr], [RA7140; F, H, Me, Cl, Bn, i-Pr], [RA7141; F, H , Me, Cl, Bn, c-Pr], [RA7142; F, H, Me, Cl, Bn, Bu], [RA7143; F, H, Me, Cl, Bn, i-Bu], [RA7144; F , H, Me, Cl, Bn, t-Bu], [RA7145; F, H, Me, Cl, Bn, c-PrCH ₂ ], [RA7146; F, H, Me, Cl, Bn, Ph], [ RA7147; F, H, Me, Cl, Bn, Bn], [RA7148; F, H, Me, Cl, Bn, CF ₃ ], [RA7149; F, H, Me, Cl, Bn, CF ₃ CH ₂ ] , [RA7150; F, H, Me, Cl, Bn, CF ₃ CF ₂ ], [RA7151; F, H, Me, Cl, Bn, CF ₂ H], [RA7152; F, H, Me, Cl, Bn , CF ₂ HCH ₂ ], [RA7153; F, H, Et, H, Bn, Me], [RA7154; F, H, Et, H, Bn, Et], [RA7155; F, H, Et, H, Bn, Pr], [RA7156; F, H, Et, H, Bn, i-Pr], [RA7157; F, H, Et, H, Bn, c-Pr], [RA7158; F, H, Et, H, Bn, Bu], [RA7159; F, H, Et, H, Bn, i-Bu], [RA7160; F, H, Et, H, Bn, t-Bu], [RA7161; F, H, Et, H, Bn, c-PrCH ₂ ], [RA7162; F, H, Et, H, Bn, Ph], [RA7163; F, H, Et, H, Bn, Bn], [RA7164; F, H , Et, H, Bn, CF ₃ ], [RA7165; F, H, Et, H, Bn, CF ₃ CH ₂ ], [RA7166; F, H, Et, H, Bn, CF ₃ CF ₂ ], [RA7167; F, H, Et, H, Bn, CF ₂ H], [RA7168; F, H, Et, H, Bn, CF ₂ HCH ₂ ], [RA7169; F, H, Et, F, Bn, Me], [RA7170; F, H, Et, F, Bn, Et], [RA7171; F, H, Et, F, Bn, Pr] , [RA7172; F, H, Et, F, Bn, i-Pr], [RA7173; F, H, Et, F, Bn, c-Pr], [RA7174; F, H, Et, F, Bn, Bu], [RA7175; F, H, Et, F, Bn, i-Bu], [RA7176; F, H, Et, F, Bn, t-Bu], [RA7177; F, H, Et, F, Bn, c-PrCH ₂ ], [RA7178; F, H, Et, F, Bn, Ph], [RA7179; F, H, Et, F, Bn, Bn], [RA7180; F, H, Et, F , Bn, CF ₃ ], [RA7181; F, H, Et, F, Bn, CF ₃ CH ₂ ], [RA7182; F, H, Et, F, Bn, CF ₃ CF ₂ ], [RA7183; F, H, Et, F, Bn, CF ₂ H], [RA7184; F, H, Et, F, Bn, CF ₂ HCH ₂ ], [RA7185; F, H, Et, Cl, Bn, Me], [RA7186 ; F, H, Et, Cl, Bn, Et], [RA7187; F, H, Et, Cl, Bn, Pr], [RA7188; F, H, Et, Cl, Bn, i-Pr], [RA7189 ; F, H, Et, Cl, Bn, c-Pr], [RA7190; F, H, Et, Cl, Bn, Bu], [RA7191; F, H, Et, Cl, Bn, i-Bu], [RA7192; F, H, Et, Cl, Bn, t-Bu], [RA7193; F, H, Et, Cl, Bn, c-PrCH ₂ ], [RA7194; F, H, Et, Cl, Bn, Ph], [RA7195; F, H, Et, Cl, Bn, Bn], [RA7196; F, H, Et, Cl, Bn, CF ₃ ], [RA7197; F, H, Et, Cl, Bn, CF ₃ CH ₂ ], [RA7198; F, H, Et, Cl, Bn, CF ₃ CF ₂ ], [RA7199; F, H, Et, Cl, Bn, CF ₂ H], [RA7200; F, H, Et , Cl, Bn, CF ₂ HCH ₂ ],

[RA7201; F, H, F, H, Bn, Me], [RA7202; F, H, F, H, Bn, Et], [RA7203; F, H, F, H, Bn, Pr], [RA7204 ; F, H, F, H, Bn, i-Pr], [RA7205; F, H, F, H, Bn, c-Pr], [RA7206; F, H, F, H, Bn, Bu], [RA7207; F, H, F, H, Bn, i-Bu], [RA7208; F, H, F, H, Bn, t-Bu], [RA7209; F, H, F, H, Bn, c -PrCH ₂ ], [RA7210; F, H, F, H, Bn, Ph], [RA7211; F, H, F, H, Bn, Bn], [RA7212; F, H, F, H, Bn, CF ₃ ], [RA7213; F, H, F, H, Bn, CF ₃ CH ₂ ], [RA7214; F, H, F, H, Bn, CF ₃ CF ₂ ], [RA7215; F, H, F , H, Bn, CF ₂ H], [RA7216; F, H, F, H, Bn, CF ₂ HCH ₂ ], [RA7217; F, H, F, F, Bn, Me], [RA7218; F, H, F, F, Bn, Et], [RA7219; F, H, F, F, Bn, Pr], [RA7220; F, H, F, F, Bn, i-Pr], [RA7221; F, H, F, F, Bn, c-Pr], [RA7222; F, H, F, F, Bn, Bu], [RA7223; F, H, F, F, Bn, i-Bu], [RA7224; F, H, F, F, Bn, t-Bu], [RA7225; F, H, F, F, Bn, c-PrCH ₂ ], [RA7226; F, H, F, F, Bn, Ph], [RA7227; F, H, F, F, Bn, Bn], [RA7228; F, H, F, F, Bn, CF ₃ ], [RA7229; F, H, F, F, Bn, CF ₃ CH ₂ ], [RA7230; F, H, F, F, Bn, CF ₃ CF ₂ ], [RA7231; F, H, F, F, Bn, CF ₂ H], [RA7232; F, H, F, F, Bn, CF ₂ HCH ₂ ], [RA7233; F, H, F, Cl, Bn, Me], [RA7234; F, H, F, Cl, Bn, Et], [RA7235; F, H, F, Cl , Bn, Pr], [RA7236; F, H, F, Cl, Bn, i-Pr], [RA7237; F, H, F, Cl, Bn, c-Pr], [RA7238; F, H, F , Cl, Bn, Bu], [RA7239; F, H, F, Cl, Bn, i- Bu], [RA7240; F, H, F, Cl, Bn, t-Bu], [RA7241; F, H, F, Cl, Bn, c-PrCH ₂ ], [RA7242; F, H, F, Cl , Bn, Ph], [RA7243; F, H, F, Cl, Bn, Bn], [RA7244; F, H, F, Cl, Bn, CF ₃ ], [RA7245; F, H, F, Cl, Bn, CF ₃ CH ₂ ], [RA7246; F, H, F, Cl, Bn, CF ₃ CF ₂ ], [RA7247; F, H, F, Cl, Bn, CF ₂ H], [RA7248; F, H, F, Cl, Bn, CF ₂ HCH ₂ ], [RA7249; F, H, Cl, H, Bn, Me], [RA7250; F, H, Cl, H, Bn, Et], [RA7251; F , H, Cl, H, Bn, Pr], [RA7252; F, H, Cl, H, Bn, i-Pr], [RA7253; F, H, Cl, H, Bn, c-Pr], [RA7254 ; F, H, Cl, H, Bn, Bu], [RA7255; F, H, Cl, H, Bn, i-Bu], [RA7256; F, H, Cl, H, Bn, t-Bu], [RA7257; F, H, Cl, H, Bn, c-PrCH ₂ ], [RA7258; F, H, Cl, H, Bn, Ph], [RA7259; F, H, Cl, H, Bn, Bn] , [RA7260; F, H, Cl, H, Bn, CF ₃ ], [RA7261; F, H, Cl, H, Bn, CF ₃ CH ₂ ], [RA7262; F, H, Cl, H, Bn, CF ₃ CF ₂ ], [RA7263; F, H, Cl, H, Bn, CF ₂ H], [RA7264; F, H, Cl, H, Bn, CF ₂ HCH ₂ ], [RA7265; F, H, Cl, Cl, Bn, Me], [RA7266; F, H, Cl, Cl, Bn, Et], [RA7267; F, H, Cl, Cl, Bn, Pr], [RA7268; F, H, Cl, Cl, Bn, i-Pr], [RA7269; F, H, Cl, Cl, Bn, c-Pr], [RA7270; F, H, Cl, Cl, Bn, Bu], [RA7271; F, H, Cl, Cl, Bn, i-Bu], [RA7272; F, H, Cl, Cl, Bn, t-Bu], [RA7273; F, H, Cl, Cl, Bn, c-PrCH ₂ ], [RA7274 ; F, H, Cl, Cl, Bn, Ph], [RA7275; F, H, Cl, Cl, Bn, Bn], [RA7276; F, H, Cl, Cl, Bn, CF ₃ ], [RA7277; F, H, Cl, Cl, Bn, CF ₃ CH ₂ ], [RA7278; F, H, Cl, Cl, Bn, CF ₃ CF ₂ ], [RA7279; F, H , Cl, Cl, Bn, CF ₂ H], [RA7280; F, H, Cl, Cl, Bn, CF ₂ HCH ₂ ], [RA7281; F, H, Me, H, Ph, Me], [RA7282; F, H, Me, H, Ph, Et], [RA7283; F, H, Me, H, Ph, Pr], [RA7284; F, H, Me, H, Ph, i-Pr], [RA7285; F, H, Me, H, Ph, c-Pr], [RA7286; F, H, Me, H, Ph, Bu], [RA7287; F, H, Me, H, Ph, i-Bu], [ RA7288; F, H, Me, H, Ph, t-Bu], [RA7289; F, H, Me, H, Ph, c-PrCH ₂ ], [RA7290; F, H, Me, H, Ph, Ph ], [RA7291; F, H, Me, H, Ph, Bn], [RA7292; F, H, Me, H, Ph, CF ₃ ], [RA7293; F, H, Me, H, Ph, CF ₃ CH ₂ ], [RA7294; F, H, Me, H, Ph, CF ₃ CF ₂ ], [RA7295; F, H, Me, H, Ph, CF ₂ H], [RA7296; F, H, Me, H, Ph, CF ₂ HCH ₂ ], [RA7297; F, H, Me, Me, Ph, Me], [RA7298; F, H, Me, Me, Ph, Et], [RA7299; F, H, Me , Me, Ph, Pr], [RA7300; F, H, Me, Me, Ph, i-Pr], [RA7301; F, H, Me, Me, Ph, c-Pr], [RA7302; F, H , Me, Me, Ph, Bu], [RA7303; F, H, Me, Me, Ph, i-Bu], [RA7304; F, H, Me, Me, Ph, t-Bu], [RA7305; F , H, Me, Me, Ph, c-PrCH ₂ ], [RA7306; F, H, Me, Me, Ph, Ph], [RA7307; F, H, Me, Me, Ph, Bn], [RA7308; F, H, Me, Me, Ph, CF ₃ ], [RA7309; F, H, Me, Me, Ph, CF ₃ CH ₂ ], [RA7310; F, H, Me, Me, Ph, CF ₃ CF ₂ ], [RA7311; F, H, Me, Me, Ph, CF ₂ H], [RA7312; F, H, Me, Me , Ph, CF ₂ HCH ₂ ], [RA7313; F, H, Me, Et, Ph, Me], [RA7314; F, H, Me, Et, Ph, Et], [RA7315; F, H, Me, Et, Ph, Pr], [RA7316; F, H, Me, Et, Ph, i-Pr], [RA7317; F, H, Me, Et, Ph, c-Pr], [RA7318; F, H, Me, Et, Ph, Bu], [RA7319; F, H, Me, Et, Ph, i-Bu], [RA7320; F, H, Me, Et, Ph, t-Bu], [RA7321; F, H, Me, Et, Ph, c-PrCH ₂ ], [RA7322; F, H, Me, Et, Ph, Ph], [RA7323; F, H, Me, Et, Ph, Bn], [RA7324; F , H, Me, Et, Ph, CF ₃ ], [RA7325; F, H, Me, Et, Ph, CF ₃ CH ₂ ], [RA7326; F, H, Me, Et, Ph, CF ₃ CF ₂ ] , [RA7327; F, H, Me, Et, Ph, CF ₂ H], [RA7328; F, H, Me, Et, Ph, CF ₂ HCH ₂ ], [RA7329; F, H, Me, F, Ph , Me], [RA7330; F, H, Me, F, Ph, Et], [RA7331; F, H, Me, F, Ph, Pr], [RA7332; F, H, Me, F, Ph, i -Pr], [RA7333; F, H, Me, F, Ph, c-Pr], [RA7334; F, H, Me, F, Ph, Bu], [RA7335; F, H, Me, F, Ph , i-Bu], [RA7336; F, H, Me, F, Ph, t-Bu], [RA7337; F, H, Me, F, Ph, c-PrCH ₂ ], [RA7338; F, H, Me, F, Ph, Ph], [RA7339; F, H, Me, F, Ph, Bn], [RA7340; F, H, Me, F, Ph, CF ₃ ], [RA7341; F, H, Me , F, Ph, CF ₃ CH ₂ ], [RA7342; F, H, Me, F, Ph, CF ₃ CF ₂ ], [RA7343; F, H, Me, F, Ph, CF ₂ H], [RA7344 ; F, H, Me, F, Ph, CF ₂ HCH ₂ ], [RA7345; F, H, Me, Cl, Ph, Me], [RA7346; F, H, Me, Cl, Ph, Et], [ RA7347; F, H, Me, Cl, Ph, Pr], [RA7348; F, H, Me, Cl, Ph, i-Pr], [RA 7349; F, H, Me, Cl, Ph, c-Pr], [RA7350; F, H, Me, Cl, Ph, Bu], [RA7351; F, H, Me, Cl, Ph, i-Bu] , [RA7352; F, H, Me, Cl, Ph, t-Bu], [RA7353; F, H, Me, Cl, Ph, c-PrCH ₂ ], [RA7354; F, H, Me, Cl, Ph , Ph], [RA7355; F, H, Me, Cl, Ph, Bn], [RA7356; F, H, Me, Cl, Ph, CF ₃ ], [RA7357; F, H, Me, Cl, Ph, CF ₃ CH ₂ ], [RA7358; F, H, Me, Cl, Ph, CF ₃ CF ₂ ], [RA7359; F, H, Me, Cl, Ph, CF ₂ H], [RA7360; F, H, Me, Cl, Ph, CF ₂ HCH ₂ ], [RA7361; F, H, Et, H, Ph, Me], [RA7362; F, H, Et, H, Ph, Et], [RA7363; F, H , Et, H, Ph, Pr], [RA7364; F, H, Et, H, Ph, i-Pr], [RA7365; F, H, Et, H, Ph, c-Pr], [RA7366; F , H, Et, H, Ph, Bu], [RA7367; F, H, Et, H, Ph, i-Bu], [RA7368; F, H, Et, H, Ph, t-Bu], [RA7369 ; F, H, Et, H, Ph, c-PrCH ₂ ], [RA7370; F, H, Et, H, Ph, Ph], [RA7371; F, H, Et, H, Ph, Bn], [ RA7372; F, H, Et, H, Ph, CF ₃ ], [RA7373; F, H, Et, H, Ph, CF ₃ CH ₂ ], [RA7374; F, H, Et, H, Ph, CF ₃ CF ₂ ], [RA7375; F, H, Et, H, Ph, CF ₂ H], [RA7376; F, H, Et, H, Ph, CF ₂ HCH ₂ ], [RA7377; F, H, Et, F, Ph, Me], [RA7378; F, H, Et, F, Ph, Et], [RA7379; F, H, Et, F, Ph, Pr], [RA7380; F, H, Et, F, Ph, i-Pr], [RA7381; F, H, Et, F, Ph, c-Pr], [RA7382; F, H, Et, F, Ph, Bu], [RA7383; F, H, Et, F, Ph, i-Bu], [RA7384; F, H, Et, F, Ph, t-Bu], [RA7385; F, H, Et, F, Ph, c-PrCH ₂ ], [RA7386; F, H, Et, F, Ph, Ph], [RA7387; F, H, Et, F, Ph, Bn], [RA7388; F, H, Et, F, Ph, CF ₃ ], [RA7389; F, H, Et, F, Ph, CF ₃ CH ₂ ], [RA7390; F, H, Et, F, Ph, CF ₃ CF ₂ ], [RA7391; F, H, Et, F , Ph, CF ₂ H], [RA7392; F, H, Et, F, Ph, CF ₂ HCH ₂ ], [RA7393; F, H, Et, Cl, Ph, Me], [RA7394; F, H, Et, Cl, Ph, Et], [RA7395; F, H, Et, Cl, Ph, Pr], [RA7396; F, H, Et, Cl, Ph, i-Pr], [RA7397; F, H, Et, Cl, Ph, c-Pr], [RA7398; F, H, Et, Cl, Ph, Bu], [RA7399; F, H, Et, Cl, Ph, i-Bu], [RA7400; F, H, Et, Cl, Ph, t-Bu],

[RA7401; F, H, Et, Cl, Ph, c-PrCH ₂ ], [RA7402; F, H, Et, Cl, Ph, Ph], [RA7403; F, H, Et, Cl, Ph, Bn] , [RA7404; F, H, Et, Cl, Ph, CF ₃ ], [RA7405; F, H, Et, Cl, Ph, CF ₃ CH ₂ ], [RA7406; F, H, Et, Cl, Ph, CF ₃ CF ₂ ], [RA7407; F, H, Et, Cl, Ph, CF ₂ H], [RA7408; F, H, Et, Cl, Ph, CF ₂ HCH ₂ ], [RA7409; F, H, F, H, Ph, Me], [RA7410; F, H, F, H, Ph, Et], [RA7411; F, H, F, H, Ph, Pr], [RA7412; F, H, F, H, Ph, i-Pr], [RA7413; F, H, F, H, Ph, c-Pr], [RA7414; F, H, F, H, Ph, Bu], [RA7415; F, H, F, H, Ph, i-Bu], [RA7416; F, H, F, H, Ph, t-Bu], [RA7417; F, H, F, H, Ph, c-PrCH ₂ ], [RA7418 ; F, H, F, H, Ph, Ph], [RA7419; F, H, F, H, Ph, Bn], [RA7420; F, H, F, H, Ph, CF ₃ ], [RA7421; F, H, F, H, Ph, CF ₃ CH ₂ ], [RA7422; F, H, F, H, Ph, CF ₃ CF ₂ ], [RA7423; F, H, F, H, Ph, CF ₂ H], [RA7424; F, H, F, H, Ph, CF ₂ HCH ₂ ], [RA7425; F, H, F, F, Ph, Me], [RA7426; F, H, F, F, Ph , Et], [RA7427; F, H, F, F, Ph, Pr], [RA7428; F, H, F, F, Ph, i-Pr], [RA7429; F, H, F, F, Ph , c-Pr], [RA7430; F, H, F, F, Ph, Bu], [RA7431; F, H, F, F, Ph, i-Bu], [RA7432; F, H, F, F , Ph, t-Bu], [RA7433; F, H, F, F, Ph, c-PrCH ₂ ], [RA7434; F, H, F, F, Ph, Ph], [RA7435; F, H, F, F, Ph, Bn], [RA7436; F, H, F, F, Ph, CF ₃ ], [RA7437; F, H, F, F, Ph, CF ₃ CH ₂ ], [RA7438; F, H, F, F, Ph, CF ₃ CF ₂ ], [RA7439; F, H, F, F, Ph, CF ₂ H], [RA7440; F, H, F, F, Ph, CF ₂ HCH ₂ ], [RA7441; F, H, F , Cl, Ph, Me], [RA7442; F, H, F, Cl, Ph, Et], [RA7443; F, H, F, Cl, Ph, Pr], [RA7444; F, H, F, Cl , Ph, i-Pr], [RA7445; F, H, F, Cl, Ph, c-Pr], [RA7446; F, H, F, Cl, Ph, Bu], [RA7447; F, H, F , Cl, Ph, i-Bu], [RA7448; F, H, F, Cl, Ph, t-Bu], [RA7449; F, H, F, Cl, Ph, c-PrCH ₂ ], [RA7500; H, F, Me, H, H, CF ₃ ], [RA7501; H, F, Me, H, H, CF ₃ CH ₂ ], [RA7502; H, F, Me, H, H, CF ₃ CF ₂ ], [RA7503; H, F, Me, H, H, CF ₂ H], [RA7504; H, F, Me, H, H, CF ₂ HCH ₂ ], [RA7505; H, F, Me, Me, H, Me], [RA7506; H, F, Me, Me, H, Et], [RA7507; H, F, Me, Me, H, Pr], [RA7508; H, F, Me, Me, H, i-Pr], [RA7509; H, F, Me, Me, H, c-Pr], [RA7510; H, F, Me, Me, H, Bu], [RA7511; H, F, Me, Me, H, i-Bu], [RA7512; H, F, Me, Me, H, t-Bu], [RA7513; H, F, Me, Me, H, c-PrCH ₂ ], [RA7514; H, F , Me, Me, H, Ph], [RA7515; H, F, Me, Me, H, Bn], [RA7516; H, F, Me, Me, H, CF ₃ ], [RA7517; H, F, Me, Me, H, CF ₃ CH ₂ ], [RA7518; H, F, Me, Me, H, CF ₃ CF ₂ ], [RA7519; H, F, Me, Me, H, CF ₂ H], [ RA7520; H, F, Me, Me, H, CF ₂ HCH ₂ ], [RA7521; H, F, Me, Et, H, Me], [RA7522; H, F, Me, Et, H, Et], [RA7523; H, F, Me, Et, H, Pr], [RA7524; H, F, Me, Et, H, i-Pr], [RA7525; H, F, Me, Et, H, cP r], [RA7526; H, F, Me, Et, H, Bu], [RA7527; H, F, Me, Et, H, i-Bu], [RA7528; H, F, Me, Et, H, t-Bu], [RA7529; H, F, Me, Et, H, c-PrCH ₂ ], [RA7530; H, F, Me, Et, H, Ph], [RA7531; H, F, Me, Et , H, Bn], [RA7532; H, F, Me, Et, H, CF ₃ ], [RA7533; H, F, Me, Et, H, CF ₃ CH ₂ ], [RA7534; H, F, Me , Et, H, CF ₃ CF ₂ ], [RA7535; H, F, Me, Et, H, CF ₂ H], [RA7536; H, F, Me, Et, H, CF ₂ HCH ₂ ], [RA7537 ; H, F, Me, F, H, Me], [RA7538; H, F, Me, F, H, Et], [RA7539; H, F, Me, F, H, Pr], [RA7540; H , F, Me, F, H, i-Pr], [RA7541; H, F, Me, F, H, c-Pr], [RA7542; H, F, Me, F, H, Bu], [RA7543 ; H, F, Me, F, H, i-Bu], [RA7544; H, F, Me, F, H, t-Bu], [RA7545; H, F, Me, F, H, c-PrCH ₂ ], [RA7546; H, F, Me, F, H, Ph], [RA7547; H, F, Me, F, H, Bn], [RA7548; H, F, Me, F, H, CF ₃ ], [RA7549; H, F, Me, F, H, CF ₃ CH ₂ ], [RA7550; H, F, Me, F, H, CF ₃ CF ₂ ], [RA7551; H, F, Me, F , H, CF ₂ H], [RA7552; H, F, Me, F, H, CF ₂ HCH ₂ ], [RA7553; H, F, Me, Cl, H, Me], [RA7554; H, F, Me, Cl, H, Et], [RA7555; H, F, Me, Cl, H, Pr], [RA7556; H, F, Me, Cl, H, i-Pr], [RA7557; H, F, Me, Cl, H, c-Pr], [RA7558; H, F, Me, Cl, H, Bu], [RA7559; H, F, Me, Cl, H, i-Bu], [RA7560; H, F, Me, Cl, H, t-Bu], [RA7561; H, F, Me, Cl, H, c-PrCH ₂ ], [RA7562; H, F, Me, Cl, H, Ph], [RA7563 ; H, F, Me, Cl, H, Bn], [RA7564; H, F, Me, Cl, H, CF ₃ ], [RA7565; H, F, Me, Cl, H, CF ₃ CH ₂ ], [RA7566; H, F, Me, Cl, H, CF ₃ CF ₂ ], [RA7567; H, F, Me, Cl, H, CF ₂ H], [RA7568; H, F, Me, Cl, H, CF ₂ HCH ₂ ], [RA7569; H, F, Et, H, H, Me], [RA7570; H, F, Et, H, H, Et], [RA7571; H, F, Et, H, H, Pr], [RA7572; H, F, Et, H, H, i-Pr], [RA7573; H, F, Et, H, H, c-Pr], [RA7574; H, F, Et, H, H, Bu], [RA7575; H, F, Et, H, H, i-Bu], [RA7576; H, F, Et, H, H, t-Bu], [RA7577; H, F, Et, H, H, c-PrCH ₂ ], [RA7578; H, F, Et, H, H, Ph], [RA7579; H, F, Et, H, H, Bn], [RA7580; H, F, Et, H, H, CF ₃ ], [ RA7581; H, F, Et, H, H, CF ₃ CH ₂ ], [RA7582; H, F, Et, H, H, CF ₃ CF ₂ ], [RA7583; H, F, Et, H, H, CF ₂ H], [RA7584; H, F, Et, H, H, CF ₂ HCH ₂ ], [RA7585; H, F, Et, F, H, Me], [RA7586; H, F, Et, F , H, Et], [RA7587; H, F, Et, F, H, Pr], [RA7588; H, F, Et, F, H, i-Pr], [RA7589; H, F, Et, F , H, c-Pr], [RA7590; H, F, Et, F, H, Bu], [RA7591; H, F, Et, F, H, i-Bu], [RA7592; H, F, Et , F, H, t-Bu], [RA7593; H, F, Et, F, H, c-PrCH ₂ ], [RA7594; H, F, Et, F, H, Ph], [RA7595; H, F, Et, F, H, Bn], [RA7596; H, F, Et, F, H, CF ₃ ], [RA7597; H, F, Et, F, H, CF ₃ CH ₂ ], [RA7598; H, F, Et, F, H, CF ₃ CF ₂ ], [RA7599; H, F, Et, F, H, CF ₂ H], [RA7600; H, F, Et, F, H, CF ₂ HCH ₂ ],

[RA7601; H, F, Et, Cl, H, Me], [RA7602; H, F, Et, Cl, H, Et], [RA7603; H, F, Et, Cl, H, Pr], [RA7604 ; H, F, Et, Cl, H, i-Pr], [RA7605; H, F, Et, Cl, H, c-Pr], [RA7606; H, F, Et, Cl, H, Bu], [RA7607; H, F, Et, Cl, H, i-Bu], [RA7608; H, F, Et, Cl, H, t-Bu], [RA7609; H, F, Et, Cl, H, c -PrCH ₂ ], [RA7610; H, F, Et, Cl, H, Ph], [RA7611; H, F, Et, Cl, H, Bn], [RA7612; H, F, Et, Cl, H, CF ₃ ], [RA7613; H, F, Et, Cl, H, CF ₃ CH ₂ ], [RA7614; H, F, Et, Cl, H, CF ₃ CF ₂ ], [RA7615; H, F, Et , Cl, H, CF ₂ H], [RA7616; H, F, Et, Cl, H, CF ₂ HCH ₂ ], [RA7617; H, F, F, H, H, Me], [RA7618; H, F, F, H, H, Et], [RA7619; H, F, F, H, H, Pr], [RA7620; H, F, F, H, H, i-Pr], [RA7621; H, F, F, H, H, c-Pr], [RA7622; H, F, F, H, H, Bu], [RA7623; H, F, F, H, H, i-Bu], [RA7624; H, F, F, H, H, t-Bu], [RA7625; H, F, F, H, H, c-PrCH ₂ ], [RA7626; H, F, F, H, H, Ph], [RA7627; H, F, F, H, H, Bn], [RA7628; H, F, F, H, H, CF ₃ ], [RA7629; H, F, F, H, H, CF ₃ CH ₂ ], [RA7630; H, F, F, H, H, CF ₃ CF ₂ ], [RA7631; H, F, F, H, H, CF ₂ H], [RA7632; H, F, F, H, H, CF ₂ HCH ₂ ], [RA7633; H, F, F, F, H, Me], [RA7634; H, F, F, F, H, Et], [RA7635; H, F, F, F , H, Pr], [RA7636; H, F, F, F, H, i-Pr], [RA7637; H, F, F, F, H, c-Pr], [RA7638; H, F, F , F, H, Bu], [RA7639; H, F, F, F, H, i-Bu], [RA7640; H, F, F, F, H, t-Bu], [RA7641; H, F, F, F, H, c-PrCH ₂ ], [RA7642; H, F, F, F, H, Ph], [RA7643 ; H, F, F, F, H, Bn], [RA7644; H, F, F, F, H, CF ₃ ], [RA7645; H, F, F, F, H, CF ₃ CH ₂ ], [RA7646; H, F, F, F, H, CF ₃ CF ₂ ], [RA7647; H, F, F, F, H, CF ₂ H], [RA7648; H, F, F, F, H, CF ₂ HCH ₂ ], [RA7649; H, F, F, Cl, H, Me], [RA7650; H, F, F, Cl, H, Et], [RA7651; H, F, F, Cl, H , Pr], [RA7652; H, F, F, Cl, H, i-Pr], [RA7653; H, F, F, Cl, H, c-Pr], [RA7654; H, F, F, Cl , H, Bu], [RA7655; H, F, F, Cl, H, i-Bu], [RA7656; H, F, F, Cl, H, t-Bu], [RA7657; H, F, F , Cl, H, c-PrCH ₂ ], [RA7658; H, F, F, Cl, H, Ph], [RA7659; H, F, F, Cl, H, Bn], [RA7660; H, F, F, Cl, H, CF ₃ ], [RA7661; H, F, F, Cl, H, CF ₃ CH ₂ ], [RA7662; H, F, F, Cl, H, CF ₃ CF ₂ ], [RA7663 ; H, F, F, Cl, H, CF ₂ H], [RA7664; H, F, F, Cl, H, CF ₂ HCH ₂ ], [RA7665; H, F, Cl, H, H, Me] , [RA7666; H, F, Cl, H, H, Et], [RA7667; H, F, Cl, H, H, Pr], [RA7668; H, F, Cl, H, H, i-Pr] , [RA7669; H, F, Cl, H, H, c-Pr], [RA7670; H, F, Cl, H, H, Bu], [RA7671; H, F, Cl, H, H, i- Bu], [RA7672; H, F, Cl, H, H, t-Bu], [RA7673; H, F, Cl, H, H, c-PrCH ₂ ], [RA7674; H, F, Cl, H , H, Ph], [RA7675; H, F, Cl, H, H, Bn], [RA7676; H, F, Cl, H, H, CF ₃ ], [RA7677; H, F, Cl, H, H, CF ₃ CH ₂ ], [RA7678; H, F, Cl, H, H, CF ₃ CF ₂ ], [RA7679; H, F, Cl, H, H, CF ₂ H], [RA7680; H, F, Cl, H, H, CF ₂ HCH ₂ ], [RA7681; H, F, Cl, Cl, H, Me], [RA7682; H, F, Cl, Cl, H, Et], [RA7683; H, F, Cl, Cl, H, Pr], [RA7684; H, F, Cl, Cl, H, i- Pr], [RA7685; H, F, Cl, Cl, H, c-Pr], [RA7686; H, F, Cl, Cl, H, Bu], [RA7687; H, F, Cl, Cl, H, i-Bu], [RA7688; H, F, Cl, Cl, H, t-Bu], [RA7689; H, F, Cl, Cl, H, c-PrCH ₂ ], [RA7690; H, F, Cl , Cl, H, Ph], [RA7691; H, F, Cl, Cl, H, Bn], [RA7692; H, F, Cl, Cl, H, CF ₃ ], [RA7693; H, F, Cl, Cl, H, CF ₃ CH ₂ ], [RA7694; H, F, Cl, Cl, H, CF ₃ CF ₂ ], [RA7695; H, F, Cl, Cl, H, CF ₂ H], [RA7696; H, F, Cl, Cl, H, CF ₂ HCH ₂ ], [RA7697; H, F, Me, H, Me, Me], [RA7698; H, F, Me, H, Me, Et], [RA7699 ; H, F, Me, H, Me, Pr], [RA7700; H, F, Me, H, Me, i-Pr], [RA7701; H, F, Me, H, Me, c-Pr], [RA7702; H, F, Me, H, Me, Bu], [RA7703; H, F, Me, H, Me, i-Bu], [RA7704; H, F, Me, H, Me, t-Bu ], [RA7705; H, F, Me, H, Me, c-PrCH ₂ ], [RA7706; H, F, Me, H, Me, Ph], [RA7707; H, F, Me, H, Me, Bn], [RA7708; H, F, Me, H, Me, CF ₃ ], [RA7709; H, F, Me, H, Me, CF ₃ CH ₂ ], [RA7710; H, F, Me, H, Me, CF ₃ CF ₂ ], [RA7711; H, F, Me, H, Me, CF ₂ H], [RA7712; H, F, Me, H, Me, CF ₂ HCH ₂ ], [RA7713; H, F, Me, Me, Me, Me], [RA7714; H, F, Me, Me, Me, Et], [RA7715; H, F, Me, Me, Me, Pr], [RA7 716; H, F, Me, Me, Me, i-Pr], [RA7717; H, F, Me, Me, Me, c-Pr], [RA7718; H, F, Me, Me, Me, Bu] , [RA7719; H, F, Me, Me, Me, i-Bu], [RA7720; H, F, Me, Me, Me, t-Bu], [RA7721; H, F, Me, Me, Me, c-PrCH ₂ ], [RA7722; H, F, Me, Me, Me, Ph], [RA7723; H, F, Me, Me, Me, Bn], [RA7724; H, F, Me, Me, Me , CF ₃ ], [RA7725; H, F, Me, Me, Me, CF ₃ CH ₂ ], [RA7726; H, F, Me, Me, Me, CF ₃ CF ₂ ], [RA7727; H, F, Me, Me, Me, CF ₂ H], [RA7728; H, F, Me, Me, Me, CF ₂ HCH ₂ ], [RA7729; H, F, Me, Et, Me, Me], [RA7730; H , F, Me, Et, Me, Et], [RA7731; H, F, Me, Et, Me, Pr], [RA7732; H, F, Me, Et, Me, i-Pr], [RA7733; H , F, Me, Et, Me, c-Pr], [RA7734; H, F, Me, Et, Me, Bu], [RA7735; H, F, Me, Et, Me, i-Bu], [RA7736 ; H, F, Me, Et, Me, t-Bu], [RA7737; H, F, Me, Et, Me, c-PrCH ₂ ], [RA7738; H, F, Me, Et, Me, Ph] , [RA7739; H, F, Me, Et, Me, Bn], [RA7740; H, F, Me, Et, Me, CF ₃ ], [RA7741; H, F, Me, Et, Me, CF ₃ CH ₂ ], [RA7742; H, F, Me, Et, Me, CF ₃ CF ₂ ], [RA7743; H, F, Me, Et, Me, CF ₂ H], [RA7744; H, F, Me, Et , Me, CF ₂ HCH ₂ ], [RA7745; H, F, Me, F, Me, Me], [RA7746; H, F, Me, F, Me, Et], [RA7747; H, F, Me, F, Me, Pr], [RA7748; H, F, Me, F, Me, i-Pr], [RA7749; H, F, Me, F, Me, c-Pr], [RA7750; H, F, Me, F, Me, Bu], [RA7751; H, F, Me, F, Me, i-Bu], [RA7752; H, F , Me, F, Me, t-Bu], [RA7753; H, F, Me, F, Me, c-PrCH ₂ ], [RA7754; H, F, Me, F, Me, Ph], [RA7755; H, F, Me, F, Me, Bn], [RA7756; H, F, Me, F, Me, CF ₃ ], [RA7757; H, F, Me, F, Me, CF ₃ CH ₂ ], [ RA7758; H, F, Me, F, Me, CF ₃ CF ₂ ], [RA7759; H, F, Me, F, Me, CF ₂ H], [RA7760; H, F, Me, F, Me, CF ₂ HCH ₂ ], [RA7761; H, F, Me, Cl, Me, Me], [RA7762; H, F, Me, Cl, Me, Et], [RA7763; H, F, Me, Cl, Me, Pr], [RA7764; H, F, Me, Cl, Me, i-Pr], [RA7765; H, F, Me, Cl, Me, c-Pr], [RA7766; H, F, Me, Cl, Me, Bu], [RA7767; H, F, Me, Cl, Me, i-Bu], [RA7768; H, F, Me, Cl, Me, t-Bu], [RA7769; H, F, Me, Cl, Me, c-PrCH ₂ ], [RA7770; H, F, Me, Cl, Me, Ph], [RA7771; H, F, Me, Cl, Me, Bn], [RA7772; H, F, Me , Cl, Me, CF ₃ ], [RA7773; H, F, Me, Cl, Me, CF ₃ CH ₂ ], [RA7774; H, F, Me, Cl, Me, CF ₃ CF ₂ ], [RA7775; H, F, Me, Cl, Me, CF ₂ H], [RA7776; H, F, Me, Cl, Me, CF ₂ HCH ₂ ], [RA7777; H, F, Et, H, Me, Me], [RA7778; H, F, Et, H, Me, Et], [RA7779; H, F, Et, H, Me, Pr], [RA7780; H, F, Et, H, Me, i-Pr], [RA7781; H, F, Et, H, Me, c-Pr], [RA7782; H, F, Et, H, Me, Bu], [RA7783; H, F, Et, H, Me, i-Bu ], [RA7784; H, F, Et, H, Me, t-Bu], [RA7785; H, F, Et, H, Me, c-PrCH ₂ ], [RA7786; H, F, Et, H, Me, Ph], [RA7787; H, F, Et, H, Me, Bn], [RA7788; H, F, Et, H, Me, CF ₃ ], [ RA7789; H, F, Et, H, Me, CF ₃ CH ₂ ], [RA7790; H, F, Et, H, Me, CF ₃ CF ₂ ], [RA7791; H, F, Et, H, Me, CF ₂ H], [RA7792; H, F, Et, H, Me, CF ₂ HCH ₂ ], [RA7793; H, F, Et, F, Me, Me], [RA7794; H, F, Et, F , Me, Et], [RA7795; H, F, Et, F, Me, Pr], [RA7796; H, F, Et, F, Me, i-Pr], [RA7797; H, F, Et, F , Me, c-Pr], [RA7798; H, F, Et, F, Me, Bu], [RA7799; H, F, Et, F, Me, i-Bu], [RA7800; H, F, Et , F, Me, t-Bu],

[RA7801; H, F, Et, F, Me, c-PrCH ₂ ], [RA7802; H, F, Et, F, Me, Ph], [RA7803; H, F, Et, F, Me, Bn] , [RA7804; H, F, Et, F, Me, CF ₃ ], [RA7805; H, F, Et, F, Me, CF ₃ CH ₂ ], [RA7806; H, F, Et, F, Me, CF ₃ CF ₂ ], [RA7807; H, F, Et, F, Me, CF ₂ H], [RA7808; H, F, Et, F, Me, CF ₂ HCH ₂ ], [RA7809; H, F, Et, Cl, Me, Me], [RA7810; H, F, Et, Cl, Me, Et], [RA7811; H, F, Et, Cl, Me, Pr], [RA7812; H, F, Et, Cl, Me, i-Pr], [RA7813; H, F, Et, Cl, Me, c-Pr], [RA7814; H, F, Et, Cl, Me, Bu], [RA7815; H, F, Et, Cl, Me, i-Bu], [RA7816; H, F, Et, Cl, Me, t-Bu], [RA7817; H, F, Et, Cl, Me, c-PrCH ₂ ], [RA7818 ; H, F, Et, Cl, Me, Ph], [RA7819; H, F, Et, Cl, Me, Bn], [RA7820; H, F, Et, Cl, Me, CF ₃ ], [RA7821; H, F, Et, Cl, Me, CF ₃ CH ₂ ], [RA7822; H, F, Et, Cl, Me, CF ₃ CF ₂ ], [RA7823; H, F, Et, Cl, Me, CF ₂ H], [RA7824; H, F, Et, Cl, Me, CF ₂ HCH ₂ ], [RA7825; H, F, F, H, Me, Me], [RA7826; H, F, F, H, Me , Et], [RA7827; H, F, F, H, Me, Pr], [RA7828; H, F, F, H, Me, i-Pr], [RA7829; H, F, F, H, Me , c-Pr], [RA7830; H, F, F, H, Me, Bu], [RA7831; H, F, F, H, Me, i-Bu], [RA7832; H, F, F, H , Me, t-Bu], [RA7833; H, F, F, H, Me, c-PrCH ₂ ], [RA7834; H, F, F, H, Me, Ph], [RA7835; H, F, F, H, Me, Bn], [RA7836; H, F, F, H, Me, CF ₃ ], [RA7837; H, F, F, H, Me, CF ₃ CH ₂ ], [RA7838; H, F, F, H, Me, CF ₃ CF ₂ ], [RA7839; H, F, F, H, Me, CF ₂ H], [RA7840; H, F, F, H, Me, CF ₂ HCH ₂ ], [RA7841; H, F, F, F, Me, Me], [RA7842; H, F, F, F, Me, Et], [RA7843; H, F, F, F , Me, Pr], [RA7844; H, F, F, F, Me, i-Pr], [RA7845; H, F, F, F, Me, c-Pr], [RA7846; H, F, F , F, Me, Bu], [RA7847; H, F, F, F, Me, i-Bu], [RA7848; H, F, F, F, Me, t-Bu], [RA7849; H, F , F, F, Me, c-PrCH ₂ ], [RA7850; H, F, F, F, Me, Ph], [RA7851; H, F, F, F, Me, Bn], [RA7852; H, F, F, F, Me, CF ₃ ], [RA7853; H, F, F, F, Me, CF ₃ CH ₂ ], [RA7854; H, F, F, F, Me, CF ₃ CF ₂ ], [RA7855; H, F, F, F, Me, CF ₂ H], [RA7856; H, F, F, F, Me, CF ₂ HCH ₂ ], [RA7857; H, F, F, Cl, Me, Me], [RA7858; H, F, F, Cl, Me, Et], [RA7859; H, F, F, Cl, Me, Pr], [RA7860; H, F, F, Cl, Me, i- Pr], [RA7861; H, F, F, Cl, Me, c-Pr], [RA7862; H, F, F, Cl, Me, Bu], [RA7863; H, F, F, Cl, Me, i-Bu], [RA7864; H, F, F, Cl, Me, t-Bu], [RA7865; H, F, F, Cl, Me, c-PrCH ₂ ], [RA7866; H, F, F , Cl, Me, Ph], [RA7867; H, F, F, Cl, Me, Bn], [RA7868; H, F, F, Cl, Me, CF ₃ ], [RA7869; H, F, F, Cl, Me, CF ₃ CH ₂ ], [RA7870; H, F, F, Cl, Me, CF ₃ CF ₂ ], [RA7871; H, F, F, Cl, Me, CF ₂ H], [RA7872; H, F, F, Cl, Me, CF ₂ HCH ₂ ], [RA7873; H, F, Cl, H, Me, Me], [RA7874; H, F, Cl, H, Me, Et], [RA7875 ; H, F, C l, H, Me, Pr], [RA7876; H, F, Cl, H, Me, i-Pr], [RA7877; H, F, Cl, H, Me, c-Pr], [RA7878; H, F, Cl, H, Me, Bu], [RA7879; H, F, Cl, H, Me, i-Bu], [RA7880; H, F, Cl, H, Me, t-Bu], [RA7881; H, F, Cl, H, Me, c-PrCH ₂ ], [RA7882; H, F, Cl, H, Me, Ph], [RA7883; H, F, Cl, H, Me, Bn], [RA7884 ; H, F, Cl, H, Me, CF ₃ ], [RA7885; H, F, Cl, H, Me, CF ₃ CH ₂ ], [RA7886; H, F, Cl, H, Me, CF ₃ CF ₂ ], [RA7887; H, F, Cl, H, Me, CF ₂ H], [RA7888; H, F, Cl, H, Me, CF ₂ HCH ₂ ], [RA7889; H, F, Cl, Cl , Me, Me], [RA7890; H, F, Cl, Cl, Me, Et], [RA7891; H, F, Cl, Cl, Me, Pr], [RA7892; H, F, Cl, Cl, Me , i-Pr], [RA7893; H, F, Cl, Cl, Me, c-Pr], [RA7894; H, F, Cl, Cl, Me, Bu], [RA7895; H, F, Cl, Cl , Me, i-Bu], [RA7896; H, F, Cl, Cl, Me, t-Bu], [RA7897; H, F, Cl, Cl, Me, c-PrCH ₂ ], [RA7898; H, F, Cl, Cl, Me, Ph], [RA7899; H, F, Cl, Cl, Me, Bn], [RA7900; H, F, Cl, Cl, Me, CF ₃ ], [RA7901; H, F , Cl, Cl, Me, CF ₃ CH ₂ ], [RA7902; H, F, Cl, Cl, Me, CF ₃ CF ₂ ], [RA7903; H, F, Cl, Cl, Me, CF ₂ H], [RA7904; H, F, Cl, Cl, Me, CF ₂ HCH ₂ ], [RA7905; H, F, Me, H, Et, Me], [RA7906; H, F, Me, H, Et, Et] , [RA7907; H, F, Me, H, Et, Pr], [RA7908; H, F, Me, H, Et, i-Pr], [RA7909; H, F, Me, H, Et, c- Pr], [RA7910; H, F, Me, H, Et, Bu], [RA7911; H, F, Me, H, Et, i-Bu], [RA7912; H , F, Me, H, Et, t-Bu], [RA7913; H, F, Me, H, Et, c-PrCH ₂ ], [RA7914; H, F, Me, H, Et, Ph], [ RA7915; H, F, Me, H, Et, Bn], [RA7916; H, F, Me, H, Et, CF ₃ ], [RA7917; H, F, Me, H, Et, CF ₃ CH ₂ ] , [RA7918; H, F, Me, H, Et, CF ₃ CF ₂ ], [RA7919; H, F, Me, H, Et, CF ₂ H], [RA7920; H, F, Me, H, Et , CF ₂ HCH ₂ ], [RA7921; H, F, Me, Me, Et, Me], [RA7922; H, F, Me, Me, Et, Et], [RA7923; H, F, Me, Me, Et, Pr], [RA7924; H, F, Me, Me, Et, i-Pr], [RA7925; H, F, Me, Me, Et, c-Pr], [RA7926; H, F, Me, Me, Et, Bu], [RA7927; H, F, Me, Me, Et, i-Bu], [RA7928; H, F, Me, Me, Et, t-Bu], [RA7929; H, F, Me, Me, Et, c-PrCH ₂ ], [RA7930; H, F, Me, Me, Et, Ph], [RA7931; H, F, Me, Me, Et, Bn], [RA7932; H, F , Me, Me, Et, CF ₃ ], [RA7933; H, F, Me, Me, Et, CF ₃ CH ₂ ], [RA7934; H, F, Me, Me, Et, CF ₃ CF ₂ ], [ RA7935; H, F, Me, Me, Et, CF ₂ H], [RA7936; H, F, Me, Me, Et, CF ₂ HCH ₂ ], [RA7937; H, F, Me, Et, Et, Me ], [RA7938; H, F, Me, Et, Et, Et], [RA7939; H, F, Me, Et, Et, Pr], [RA7940; H, F, Me, Et, Et, i-Pr ], [RA7941; H, F, Me, Et, Et, c-Pr], [RA7942; H, F, Me, Et, Et, Bu], [RA7943; H, F, Me, Et, Et, i -Bu], [RA7944; H, F, Me, Et, Et, t-Bu], [RA7945; H, F, Me, Et, Et, c-PrCH ₂ ], [RA7946; H, F, Me, Et, Et, Ph], [RA7947; H, F, Me, Et, Et, Bn], [RA7948; H, F, Me, Et, Et, CF ₃ ], [RA7949; H, F, Me, Et, Et, CF ₃ CH ₂ ], [RA7950; H, F, Me, Et, Et, CF ₃ CF ₂ ], [RA7951; H , F, Me, Et, Et, CF ₂ H], [RA7952; H, F, Me, Et, Et, CF ₂ HCH ₂ ], [RA7953; H, F, Me, F, Et, Me], [ RA7954; H, F, Me, F, Et, Et], [RA7955; H, F, Me, F, Et, Pr], [RA7956; H, F, Me, F, Et, i-Pr], [ RA7957; H, F, Me, F, Et, c-Pr], [RA7958; H, F, Me, F, Et, Bu], [RA7959; H, F, Me, F, Et, i-Bu] , [RA7960; H, F, Me, F, Et, t-Bu], [RA7961; H, F, Me, F, Et, c-PrCH ₂ ], [RA7962; H, F, Me, F, Et , Ph], [RA7963; H, F, Me, F, Et, Bn], [RA7964; H, F, Me, F, Et, CF ₃ ], [RA7965; H, F, Me, F, Et, CF ₃ CH ₂ ], [RA7966; H, F, Me, F, Et, CF ₃ CF ₂ ], [RA7967; H, F, Me, F, Et, CF ₂ H], [RA7968; H, F, Me, F, Et, CF ₂ HCH ₂ ], [RA7969; H, F, Me, Cl, Et, Me], [RA7970; H, F, Me, Cl, Et, Et], [RA7971; H, F , Me, Cl, Et, Pr], [RA7972; H, F, Me, Cl, Et, i-Pr], [RA7973; H, F, Me, Cl, Et, c-Pr], [RA7974; H , F, Me, Cl, Et, Bu], [RA7975; H, F, Me, Cl, Et, i-Bu], [RA7976; H, F, Me, Cl, Et, t-Bu], [RA7977 ; H, F, Me, Cl, Et, c-PrCH ₂ ], [RA7978; H, F, Me, Cl, Et, Ph], [RA7979; H, F, Me, Cl, Et, Bn], [ RA7980; H, F, Me, Cl, Et, CF ₃ ], [RA7981; H, F, Me, Cl, Et, CF ₃ CH ₂ ], [RA7982; H, F, Me, Cl, Et, CF ₃ CF ₂ ], [RA7983; H, F, Me, Cl, Et, CF ₂ H], [RA7984; H, F, Me , Cl, Et, CF ₂ HCH ₂ ], [RA7985; H, F, Et, H, Et, Me], [RA7986; H, F, Et, H, Et, Et], [RA7987; H, F, Et, H, Et, Pr], [RA7988; H, F, Et, H, Et, i-Pr], [RA7989; H, F, Et, H, Et, c-Pr], [RA7990; H, F, Et, H, Et, Bu], [RA7991; H, F, Et, H, Et, i-Bu], [RA7992; H, F, Et, H, Et, t-Bu], [RA7993; H, F, Et, H, Et, c-PrCH ₂ ], [RA7994; H, F, Et, H, Et, Ph], [RA7995; H, F, Et, H, Et, Bn], [RA7996 ; H, F, Et, H, Et, CF ₃ ], [RA7997; H, F, Et, H, Et, CF ₃ CH ₂ ], [RA7998; H, F, Et, H, Et, CF ₃ CF ₂ ], [RA7999; H, F, Et, H, Et, CF ₂ H], [RA8000; H, F, Et, H, Et, CF ₂ HCH ₂ ],

[RA8001; H, F, Et, F, Et, Me], [RA8002; H, F, Et, F, Et, Et], [RA8003; H, F, Et, F, Et, Pr], [RA8004 ; H, F, Et, F, Et, i-Pr], [RA8005; H, F, Et, F, Et, c-Pr], [RA8006; H, F, Et, F, Et, Bu], [RA8007; H, F, Et, F, Et, i-Bu], [RA8008; H, F, Et, F, Et, t-Bu], [RA8009; H, F, Et, F, Et, c -PrCH ₂ ], [RA8010; H, F, Et, F, Et, Ph], [RA8011; H, F, Et, F, Et, Bn], [RA8012; H, F, Et, F, Et, CF ₃ ], [RA8013; H, F, Et, F, Et, CF ₃ CH ₂ ], [RA8014; H, F, Et, F, Et, CF ₃ CF ₂ ], [RA8015; H, F, Et , F, Et, CF ₂ H], [RA8016; H, F, Et, F, Et, CF ₂ HCH ₂ ], [RA8017; H, F, Et, Cl, Et, Me], [RA8018; H, F, Et, Cl, Et, Et], [RA8019; H, F, Et, Cl, Et, Pr], [RA8020; H, F, Et, Cl, Et, i-Pr], [RA8021; H, F, Et, Cl, Et, c-Pr], [RA8022; H, F, Et, Cl, Et, Bu], [RA8023; H, F, Et, Cl, Et, i-Bu], [RA8024; H, F, Et, Cl, Et, t-Bu], [RA8025; H, F, Et, Cl, Et, c-PrCH ₂ ], [RA8026; H, F, Et, Cl, Et, Ph], [RA8027; H, F, Et, Cl, Et, Bn], [RA8028; H, F, Et, Cl, Et, CF ₃ ], [RA8029; H, F, Et, Cl, Et, CF ₃ CH ₂ ], [RA8030; H, F, Et, Cl, Et, CF ₃ CF ₂ ], [RA8031; H, F, Et, Cl, Et, CF ₂ H], [RA8032; H, F, Et, Cl, Et, CF ₂ HCH ₂ ], [RA8033; H, F, F, H, Et, Me], [RA8034; H, F, F, H, Et, Et], [RA8035; H, F, F, H , Et, Pr], [RA8036; H, F, F, H, Et, i-Pr], [RA8037; H, F, F, H, Et, c-Pr], [RA 8038; H, F, F, H, Et, Bu], [RA8039; H, F, F, H, Et, i-Bu], [RA8040; H, F, F, H, Et, t-Bu] , [RA8041; H, F, F, H, Et, c-PrCH ₂ ], [RA8042; H, F, F, H, Et, Ph], [RA8043; H, F, F, H, Et, Bn ], [RA8044; H, F, F, H, Et, CF ₃ ], [RA8045; H, F, F, H, Et, CF ₃ CH ₂ ], [RA8046; H, F, F, H, Et , CF ₃ CF ₂ ], [RA8047; H, F, F, H, Et, CF ₂ H], [RA8048; H, F, F, H, Et, CF ₂ HCH ₂ ], [RA8049; H, F , F, F, Et, Me], [RA8050; H, F, F, F, Et, Et], [RA8051; H, F, F, F, Et, Pr], [RA8052; H, F, F , F, Et, i-Pr], [RA8053; H, F, F, F, Et, c-Pr], [RA8054; H, F, F, F, Et, Bu], [RA8055; H, F , F, F, Et, i-Bu], [RA8056; H, F, F, F, Et, t-Bu], [RA8057; H, F, F, F, Et, c-PrCH ₂ ], [ RA8058; H, F, F, F, Et, Ph], [RA8059; H, F, F, F, Et, Bn], [RA8060; H, F, F, F, Et, CF ₃ ], [RA8061 ; H, F, F, F, Et, CF ₃ CH ₂ ], [RA8062; H, F, F, F, Et, CF ₃ CF ₂ ], [RA8063; H, F, F, F, Et, CF ₂ H], [RA8064; H, F, F, F, Et, CF ₂ HCH ₂ ], [RA8065; H, F, F, Cl, Et, Me], [RA8066; H, F, F, Cl, Et, Et], [RA8067; H, F, F, Cl, Et, Pr], [RA8068; H, F, F, Cl, Et, i-Pr], [RA8069; H, F, F, Cl, Et, c-Pr], [RA8070; H, F, F, Cl, Et, Bu], [RA8071; H, F, F, Cl, Et, i-Bu], [RA8072; H, F, F, Cl, Et, t-Bu], [RA8073; H, F, F, Cl, Et, c-PrCH ₂ ], [RA8074; H, F, F, Cl, Et, Ph], [RA8075; H, F , F, Cl, Et, Bn], [RA8076; H, F, F , Cl, Et, CF ₃ ], [RA8077; H, F, F, Cl, Et, CF ₃ CH ₂ ], [RA8078; H, F, F, Cl, Et, CF ₃ CF ₂ ], [RA8079; H, F, F, Cl, Et, CF ₂ H], [RA8080; H, F, F, Cl, Et, CF ₂ HCH ₂ ], [RA8081; H, F, Cl, H, Et, Me], [RA8082; H, F, Cl, H, Et, Et], [RA8083; H, F, Cl, H, Et, Pr], [RA8084; H, F, Cl, H, Et, i-Pr], [RA8085; H, F, Cl, H, Et, c-Pr], [RA8086; H, F, Cl, H, Et, Bu], [RA8087; H, F, Cl, H, Et, i-Bu ], [RA8088; H, F, Cl, H, Et, t-Bu], [RA8089; H, F, Cl, H, Et, c-PrCH ₂ ], [RA8090; H, F, Cl, H, Et, Ph], [RA8091; H, F, Cl, H, Et, Bn], [RA8092; H, F, Cl, H, Et, CF ₃ ], [RA8093; H, F, Cl, H, Et , CF ₃ CH ₂ ], [RA8094; H, F, Cl, H, Et, CF ₃ CF ₂ ], [RA8095; H, F, Cl, H, Et, CF ₂ H], [RA8096; H, F , Cl, H, Et, CF ₂ HCH ₂ ], [RA8097; H, F, Cl, Cl, Et, Me], [RA8098; H, F, Cl, Cl, Et, Et], [RA8099; H, F, Cl, Cl, Et, Pr], [RA8100; H, F, Cl, Cl, Et, i-Pr], [RA8101; H, F, Cl, Cl, Et, c-Pr], [RA8102; H, F, Cl, Cl, Et, Bu], [RA8103; H, F, Cl, Cl, Et, i-Bu], [RA8104; H, F, Cl, Cl, Et, t-Bu], [ RA8105; H, F, Cl, Cl, Et, c-PrCH ₂ ], [RA8106; H, F, Cl, Cl, Et, Ph], [RA8107; H, F, Cl, Cl, Et, Bn], [RA8108; H, F, Cl, Cl, Et, CF ₃ ], [RA8109; H, F, Cl, Cl, Et, CF ₃ CH ₂ ], [RA8110; H, F, Cl, Cl, Et, CF ₃ CF ₂ ], [RA8111; H, F, Cl, Cl, Et, CF ₂ H], [RA8112; H, F, Cl, Cl , Et, CF ₂ HCH ₂ ], [RA8113; H, F, Me, H, Pr, Me], [RA8114; H, F, Me, H, Pr, Et], [RA8115; H, F, Me, H, Pr, Pr], [RA8116; H, F, Me, H, Pr, i-Pr], [RA8117; H, F, Me, H, Pr, c-Pr], [RA8118; H, F, Me, H, Pr, Bu], [RA8119; H, F, Me, H, Pr, i-Bu], [RA8120; H, F, Me, H, Pr, t-Bu], [RA8121; H, F, Me, H, Pr, c-PrCH ₂ ], [RA8122; H, F, Me, H, Pr, Ph], [RA8123; H, F, Me, H, Pr, Bn], [RA8124; H , F, Me, H, Pr, CF ₃ ], [RA8125; H, F, Me, H, Pr, CF ₃ CH ₂ ], [RA8126; H, F, Me, H, Pr, CF ₃ CF ₂ ] , [RA8127; H, F, Me, H, Pr, CF ₂ H], [RA8128; H, F, Me, H, Pr, CF ₂ HCH ₂ ], [RA8129; H, F, Me, Me, Pr , Me], [RA8130; H, F, Me, Me, Pr, Et], [RA8131; H, F, Me, Me, Pr, Pr], [RA8132; H, F, Me, Me, Pr, i -Pr], [RA8133; H, F, Me, Me, Pr, c-Pr], [RA8134; H, F, Me, Me, Pr, Bu], [RA8135; H, F, Me, Me, Pr , i-Bu], [RA8136; H, F, Me, Me, Pr, t-Bu], [RA8137; H, F, Me, Me, Pr, c-PrCH ₂ ], [RA8138; H, F, Me, Me, Pr, Ph], [RA8139; H, F, Me, Me, Pr, Bn], [RA8140; H, F, Me, Me, Pr, CF ₃ ], [RA8141; H, F, Me , Me, Pr, CF ₃ CH ₂ ], [RA8142; H, F, Me, Me, Pr, CF ₃ CF ₂ ], [RA8143; H, F, Me, Me, Pr, CF ₂ H], [RA8144 ; H, F, Me, Me, Pr, CF ₂ HCH ₂ ], [RA8145; H, F, Me, Et, Pr, Me], [RA8146; H, F, Me, Et, Pr, Et], [ RA8147; H, F, Me, Et, Pr, Pr], [RA8148; H, F, Me, Et, Pr, i-Pr], [RA 8149; H, F, Me, Et, Pr, c-Pr], [RA8150; H, F, Me, Et, Pr, Bu], [RA8151; H, F, Me, Et, Pr, i-Bu] , [RA8152; H, F, Me, Et, Pr, t-Bu], [RA8153; H, F, Me, Et, Pr, c-PrCH ₂ ], [RA8154; H, F, Me, Et, Pr , Ph], [RA8155; H, F, Me, Et, Pr, Bn], [RA8156; H, F, Me, Et, Pr, CF ₃ ], [RA8157; H, F, Me, Et, Pr, CF ₃ CH ₂ ], [RA8158; H, F, Me, Et, Pr, CF ₃ CF ₂ ], [RA8159; H, F, Me, Et, Pr, CF ₂ H], [RA8160; H, F, Me, Et, Pr, CF ₂ HCH ₂ ], [RA8161; H, F, Me, F, Pr, Me], [RA8162; H, F, Me, F, Pr, Et], [RA8163; H, F , Me, F, Pr, Pr], [RA8164; H, F, Me, F, Pr, i-Pr], [RA8165; H, F, Me, F, Pr, c-Pr], [RA8166; H , F, Me, F, Pr, Bu], [RA8167; H, F, Me, F, Pr, i-Bu], [RA8168; H, F, Me, F, Pr, t-Bu], [RA8169 ; H, F, Me, F, Pr, c-PrCH ₂ ], [RA8170; H, F, Me, F, Pr, Ph], [RA8171; H, F, Me, F, Pr, Bn], [ RA8172; H, F, Me, F, Pr, CF ₃ ], [RA8173; H, F, Me, F, Pr, CF ₃ CH ₂ ], [RA8174; H, F, Me, F, Pr, CF ₃ CF ₂ ], [RA8175; H, F, Me, F, Pr, CF ₂ H], [RA8176; H, F, Me, F, Pr, CF ₂ HCH ₂ ], [RA8177; H, F, Me, Cl, Pr, Me], [RA8178; H, F, Me, Cl, Pr, Et], [RA8179; H, F, Me, Cl, Pr, Pr], [RA8180; H, F, Me, Cl, Pr, i-Pr], [RA8181; H, F, Me, Cl, Pr, c-Pr], [RA8182; H, F, Me, Cl, Pr, Bu], [RA8183; H, F, Me, Cl, Pr, i-Bu], [RA8184; H, F, Me, Cl, Pr, t-Bu], [RA8185; H, F, Me, Cl, P r, c-PrCH ₂ ], [RA8186; H, F, Me, Cl, Pr, Ph], [RA8187; H, F, Me, Cl, Pr, Bn], [RA8188; H, F, Me, Cl , Pr, CF ₃ ], [RA8189; H, F, Me, Cl, Pr, CF ₃ CH ₂ ], [RA8190; H, F, Me, Cl, Pr, CF ₃ CF ₂ ], [RA8191; H, F, Me, Cl, Pr, CF ₂ H], [RA8192; H, F, Me, Cl, Pr, CF ₂ HCH ₂ ], [RA8193; H, F, Et, H, Pr, Me], [RA8194 ; H, F, Et, H, Pr, Et], [RA8195; H, F, Et, H, Pr, Pr], [RA8196; H, F, Et, H, Pr, i-Pr], [RA8197 ; H, F, Et, H, Pr, c-Pr], [RA8198; H, F, Et, H, Pr, Bu], [RA8199; H, F, Et, H, Pr, i-Bu], [RA8200; H, F, Et, H, Pr, t-Bu],

[RA8201; H, F, Et, H, Pr, c-PrCH ₂ ], [RA8202; H, F, Et, H, Pr, Ph], [RA8203; H, F, Et, H, Pr, Bn] , [RA8204; H, F, Et, H, Pr, CF ₃ ], [RA8205; H, F, Et, H, Pr, CF ₃ CH ₂ ], [RA8206; H, F, Et, H, Pr, CF ₃ CF ₂ ], [RA8207; H, F, Et, H, Pr, CF ₂ H], [RA8208; H, F, Et, H, Pr, CF ₂ HCH ₂ ], [RA8209; H, F, Et, F, Pr, Me], [RA8210; H, F, Et, F, Pr, Et], [RA8211; H, F, Et, F, Pr, Pr], [RA8212; H, F, Et, F, Pr, i-Pr], [RA8213; H, F, Et, F, Pr, c-Pr], [RA8214; H, F, Et, F, Pr, Bu], [RA8215; H, F, Et, F, Pr, i-Bu], [RA8216; H, F, Et, F, Pr, t-Bu], [RA8217; H, F, Et, F, Pr, c-PrCH ₂ ], [RA8218 ; H, F, Et, F, Pr, Ph], [RA8219; H, F, Et, F, Pr, Bn], [RA8220; H, F, Et, F, Pr, CF ₃ ], [RA8221; H, F, Et, F, Pr, CF ₃ CH ₂ ], [RA8222; H, F, Et, F, Pr, CF ₃ CF ₂ ], [RA8223; H, F, Et, F, Pr, CF ₂ H], [RA8224; H, F, Et, F, Pr, CF ₂ HCH ₂ ], [RA8225; H, F, Et, Cl, Pr, Me], [RA8226; H, F, Et, Cl, Pr , Et], [RA8227; H, F, Et, Cl, Pr, Pr], [RA8228; H, F, Et, Cl, Pr, i-Pr], [RA8229; H, F, Et, Cl, Pr , c-Pr], [RA8230; H, F, Et, Cl, Pr, Bu], [RA8231; H, F, Et, Cl, Pr, i-Bu], [RA8232; H, F, Et, Cl , Pr, t-Bu], [RA8233; H, F, Et, Cl, Pr, c-PrCH ₂ ], [RA8234; H, F, Et, Cl, Pr, Ph], [RA8235; H, F, Et, Cl, Pr, Bn], [RA8236; H, F, Et, Cl, Pr, CF ₃ ], [RA8237; H, F, Et, Cl, Pr , CF ₃ CH ₂ ], [RA8238; H, F, Et, Cl, Pr, CF ₃ CF ₂ ], [RA8239; H, F, Et, Cl, Pr, CF ₂ H], [RA8240; H, F , Et, Cl, Pr, CF ₂ HCH ₂ ], [RA8241; H, F, F, H, Pr, Me], [RA8242; H, F, F, H, Pr, Et], [RA8243; H, F, F, H, Pr, Pr], [RA8244; H, F, F, H, Pr, i-Pr], [RA8245; H, F, F, H, Pr, c-Pr], [RA8246; H, F, F, H, Pr, Bu], [RA8247; H, F, F, H, Pr, i-Bu], [RA8248; H, F, F, H, Pr, t-Bu], [ RA8249; H, F, F, H, Pr, c-PrCH ₂ ], [RA8250; H, F, F, H, Pr, Ph], [RA8251; H, F, F, H, Pr, Bn], [RA8252; H, F, F, H, Pr, CF ₃ ], [RA8253; H, F, F, H, Pr, CF ₃ CH ₂ ], [RA8254; H, F, F, H, Pr, CF ₃ CF ₂ ], [RA8255; H, F, F, H, Pr, CF ₂ H], [RA8256; H, F, F, H, Pr, CF ₂ HCH ₂ ], [RA8257; H, F, F , F, Pr, Me], [RA8258; H, F, F, F, Pr, Et], [RA8259; H, F, F, F, Pr, Pr], [RA8260; H, F, F, F , Pr, i-Pr], [RA8261; H, F, F, F, Pr, c-Pr], [RA8262; H, F, F, F, Pr, Bu], [RA8263; H, F, F , F, Pr, i-Bu], [RA8264; H, F, F, F, Pr, t-Bu], [RA8265; H, F, F, F, Pr, c-PrCH ₂ ], [RA8266; H, F, F, F, Pr, Ph], [RA8267; H, F, F, F, Pr, Bn], [RA8268; H, F, F, F, Pr, CF ₃ ], [RA8269; H , F, F, F, Pr, CF ₃ CH ₂ ], [RA8270; H, F, F, F, Pr, CF ₃ CF ₂ ], [RA8271; H, F, F, F, Pr, CF ₂ H ], [RA8272; H, F, F, F, Pr, CF ₂ HCH ₂ ], [RA8273; H, F, F, Cl, Pr, Me], [RA8274; H, F, F, Cl, Pr, Et], [RA8275; H, F, F , Cl, Pr, Pr], [RA8276; H, F, F, Cl, Pr, i-Pr], [RA8277; H, F, F, Cl, Pr, c-Pr], [RA8278; H, F , F, Cl, Pr, Bu], [RA8279; H, F, F, Cl, Pr, i-Bu], [RA8280; H, F, F, Cl, Pr, t-Bu], [RA8281; H , F, F, Cl, Pr, c-PrCH ₂ ], [RA8282; H, F, F, Cl, Pr, Ph], [RA8283; H, F, F, Cl, Pr, Bn], [RA8284; H, F, F, Cl, Pr, CF ₃ ], [RA8285; H, F, F, Cl, Pr, CF ₃ CH ₂ ], [RA8286; H, F, F, Cl, Pr, CF ₃ CF ₂ ], [RA8287; H, F, F, Cl, Pr, CF ₂ H], [RA8288; H, F, F, Cl, Pr, CF ₂ HCH ₂ ], [RA8289; H, F, Cl, H, Pr, Me], [RA8290; H, F, Cl, H, Pr, Et], [RA8291; H, F, Cl, H, Pr, Pr], [RA8292; H, F, Cl, H, Pr, i-Pr], [RA8293; H, F, Cl, H, Pr, c-Pr], [RA8294; H, F, Cl, H, Pr, Bu], [RA8295; H, F, Cl, H, Pr, i-Bu], [RA8296; H, F, Cl, H, Pr, t-Bu], [RA8297; H, F, Cl, H, Pr, c-PrCH ₂ ], [RA8298; H, F , Cl, H, Pr, Ph], [RA8299; H, F, Cl, H, Pr, Bn], [RA8300; H, F, Cl, H, Pr, CF ₃ ], [RA8301; H, F, Cl, H, Pr, CF ₃ CH ₂ ], [RA8302; H, F, Cl, H, Pr, CF ₃ CF ₂ ], [RA8303; H, F, Cl, H, Pr, CF ₂ H], [ RA8304; H, F, Cl, H, Pr, CF ₂ HCH ₂ ], [RA8305; H, F, Cl, Cl, Pr, Me], [RA8306; H, F, Cl, Cl, Pr, Et], [RA8307; H, F, Cl, Cl, Pr, Pr], [RA8308; H, F, Cl, Cl, Pr, i-Pr], [RA8309; H, F, Cl, Cl, Pr, c-Pr ], [RA8310; H, F, Cl, Cl, Pr, Bu], [RA8311; H, F, Cl, Cl, Pr, i-Bu], [RA8312; H, F, Cl, Cl, Pr, t-Bu], [RA8313; H, F, Cl, Cl, Pr, c-PrCH ₂ ], [RA8314; H, F, Cl, Cl, Pr, Ph], [RA8315; H, F, Cl , Cl, Pr, Bn], [RA8316; H, F, Cl, Cl, Pr, CF ₃ ], [RA8317; H, F, Cl, Cl, Pr, CF ₃ CH ₂ ], [RA8318; H, F , Cl, Cl, Pr, CF ₃ CF ₂ ], [RA8319; H, F, Cl, Cl, Pr, CF ₂ H], [RA8320; H, F, Cl, Cl, Pr, CF ₂ HCH ₂ ], [RA8321; H, F, Me, H, Bu, Me], [RA8322; H, F, Me, H, Bu, Et], [RA8323; H, F, Me, H, Bu, Pr], [RA8324 ; H, F, Me, H, Bu, i-Pr], [RA8325; H, F, Me, H, Bu, c-Pr], [RA8326; H, F, Me, H, Bu, Bu], [RA8327; H, F, Me, H, Bu, i-Bu], [RA8328; H, F, Me, H, Bu, t-Bu], [RA8329; H, F, Me, H, Bu, c -PrCH ₂ ], [RA8330; H, F, Me, H, Bu, Ph], [RA8331; H, F, Me, H, Bu, Bn], [RA8332; H, F, Me, H, Bu, CF ₃ ], [RA8333; H, F, Me, H, Bu, CF ₃ CH ₂ ], [RA8334; H, F, Me, H, Bu, CF ₃ CF ₂ ], [RA8335; H, F, Me , H, Bu, CF ₂ H], [RA8336; H, F, Me, H, Bu, CF ₂ HCH ₂ ], [RA8337; H, F, Me, Me, Bu, Me], [RA8338; H, F, Me, Me, Bu, Et], [RA8339; H, F, Me, Me, Bu, Pr], [RA8340; H, F, Me, Me, Bu, i-Pr], [RA8341; H, F, Me, Me, Bu, c-Pr], [RA8342; H, F, Me, Me, Bu, Bu], [RA8343; H, F, Me, Me, Bu, i-Bu], [RA8344; H, F, Me, Me, Bu, t-Bu], [RA8345; H, F, Me, Me, Bu, c-PrCH ₂ ], [RA8346; H, F, Me, Me, Bu, Ph], [RA8347; H, F, Me, Me, Bu, Bn], [RA8348; H, F, Me, Me, Bu, CF ₃ ], [RA 8349; H, F, Me, Me, Bu, CF ₃ CH ₂ ], [RA8350; H, F, Me, Me, Bu, CF ₃ CF ₂ ], [RA8351; H, F, Me, Me, Bu, CF ₂ H], [RA8352; H, F, Me, Me, Bu, CF ₂ HCH ₂ ], [RA8353; H, F, Me, Et, Bu, Me], [RA8354; H, F, Me, Et , Bu, Et], [RA8355; H, F, Me, Et, Bu, Pr], [RA8356; H, F, Me, Et, Bu, i-Pr], [RA8357; H, F, Me, Et , Bu, c-Pr], [RA8358; H, F, Me, Et, Bu, Bu], [RA8359; H, F, Me, Et, Bu, i-Bu], [RA8360; H, F, Me , Et, Bu, t-Bu], [RA8361; H, F, Me, Et, Bu, c-PrCH ₂ ], [RA8362; H, F, Me, Et, Bu, Ph], [RA8363; H, F, Me, Et, Bu, Bn], [RA8364; H, F, Me, Et, Bu, CF ₃ ], [RA8365; H, F, Me, Et, Bu, CF ₃ CH ₂ ], [RA8366; H, F, Me, Et, Bu, CF ₃ CF ₂ ], [RA8367; H, F, Me, Et, Bu, CF ₂ H], [RA8368; H, F, Me, Et, Bu, CF ₂ HCH ₂ ], [RA8369; H, F, Me, F, Bu, Me], [RA8370; H, F, Me, F, Bu, Et], [RA8371; H, F, Me, F, Bu, Pr] , [RA8372; H, F, Me, F, Bu, i-Pr], [RA8373; H, F, Me, F, Bu, c-Pr], [RA8374; H, F, Me, F, Bu, Bu], [RA8375; H, F, Me, F, Bu, i-Bu], [RA8376; H, F, Me, F, Bu, t-Bu], [RA8377; H, F, Me, F, Bu, c-PrCH ₂ ], [RA8378; H, F, Me, F, Bu, Ph], [RA8379; H, F, Me, F, Bu, Bn], [RA8380; H, F, Me, F , Bu, CF ₃ ], [RA8381; H, F, Me, F, Bu, CF ₃ CH ₂ ], [RA8382; H, F, Me, F, Bu, CF ₃ CF ₂ ], [RA8383; H, F, Me, F, Bu, CF ₂ H], [RA8384; H, F, Me, F, Bu, CF ₂ HCH ₂ ], [RA8385; H, F, Me, Cl, Bu, Me], [RA8386; H, F, Me, Cl, Bu, Et], [RA8387; H, F, Me, Cl, Bu, Pr] , [RA8388; H, F, Me, Cl, Bu, i-Pr], [RA8389; H, F, Me, Cl, Bu, c-Pr], [RA8390; H, F, Me, Cl, Bu, Bu], [RA8391; H, F, Me, Cl, Bu, i-Bu], [RA8392; H, F, Me, Cl, Bu, t-Bu], [RA8393; H, F, Me, Cl, Bu, c-PrCH ₂ ], [RA8394; H, F, Me, Cl, Bu, Ph], [RA8395; H, F, Me, Cl, Bu, Bn], [RA8396; H, F, Me, Cl , Bu, CF ₃ ], [RA8397; H, F, Me, Cl, Bu, CF ₃ CH ₂ ], [RA8398; H, F, Me, Cl, Bu, CF ₃ CF ₂ ], [RA8399; H, F, Me, Cl, Bu, CF ₂ H], [RA8400; H, F, Me, Cl, Bu, CF ₂ HCH ₂ ],

[RA8401; H, F, Et, H, Bu, Me], [RA8402; H, F, Et, H, Bu, Et], [RA8403; H, F, Et, H, Bu, Pr], [RA8404 ; H, F, Et, H, Bu, i-Pr], [RA8405; H, F, Et, H, Bu, c-Pr], [RA8406; H, F, Et, H, Bu, Bu], [RA8407; H, F, Et, H, Bu, i-Bu], [RA8408; H, F, Et, H, Bu, t-Bu], [RA8409; H, F, Et, H, Bu, c -PrCH ₂ ], [RA8410; H, F, Et, H, Bu, Ph], [RA8411; H, F, Et, H, Bu, Bn], [RA8412; H, F, Et, H, Bu, CF ₃ ], [RA8413; H, F, Et, H, Bu, CF ₃ CH ₂ ], [RA8414; H, F, Et, H, Bu, CF ₃ CF ₂ ], [RA8415; H, F, Et , H, Bu, CF ₂ H], [RA8416; H, F, Et, H, Bu, CF ₂ HCH ₂ ], [RA8417; H, F, Et, F, Bu, Me], [RA8418; H, F, Et, F, Bu, Et], [RA8419; H, F, Et, F, Bu, Pr], [RA8420; H, F, Et, F, Bu, i-Pr], [RA8421; H, F, Et, F, Bu, c-Pr], [RA8422; H, F, Et, F, Bu, Bu], [RA8423; H, F, Et, F, Bu, i-Bu], [RA8424; H, F, Et, F, Bu, t-Bu], [RA8425; H, F, Et, F, Bu, c-PrCH ₂ ], [RA8426; H, F, Et, F, Bu, Ph], [RA8427; H, F, Et, F, Bu, Bn], [RA8428; H, F, Et, F, Bu, CF ₃ ], [RA8429; H, F, Et, F, Bu, CF ₃ CH ₂ ], [RA8430; H, F, Et, F, Bu, CF ₃ CF ₂ ], [RA8431; H, F, Et, F, Bu, CF ₂ H], [RA8432; H, F, Et, F, Bu, CF ₂ HCH ₂ ], [RA8433; H, F, Et, Cl, Bu, Me], [RA8434; H, F, Et, Cl, Bu, Et], [RA8435; H, F, Et, Cl , Bu, Pr], [RA8436; H, F, Et, Cl, Bu, i-Pr], [RA8437; H, F, Et, Cl, Bu, c-Pr], [RA8438; H , F, Et, Cl, Bu, Bu], [RA8439; H, F, Et, Cl, Bu, i-Bu], [RA8440; H, F, Et, Cl, Bu, t-Bu], [RA8441 ; H, F, Et, Cl, Bu, c-PrCH ₂ ], [RA8442; H, F, Et, Cl, Bu, Ph], [RA8443; H, F, Et, Cl, Bu, Bn], [ RA8444; H, F, Et, Cl, Bu, CF ₃ ], [RA8445; H, F, Et, Cl, Bu, CF ₃ CH ₂ ], [RA8446; H, F, Et, Cl, Bu, CF ₃ CF ₂ ], [RA8447; H, F, Et, Cl, Bu, CF ₂ H], [RA8448; H, F, Et, Cl, Bu, CF ₂ HCH ₂ ], [RA8449; H, F, F, H, Bu, Me], [RA8450; H, F, F, H, Bu, Et], [RA8451; H, F, F, H, Bu, Pr], [RA8452; H, F, F, H, Bu, i-Pr], [RA8453; H, F, F, H, Bu, c-Pr], [RA8454; H, F, F, H, Bu, Bu], [RA8455; H, F, F, H, Bu, i-Bu], [RA8456; H, F, F, H, Bu, t-Bu], [RA8457; H, F, F, H, Bu, c-PrCH ₂ ], [RA8458; H , F, F, H, Bu, Ph], [RA8459; H, F, F, H, Bu, Bn], [RA8460; H, F, F, H, Bu, CF ₃ ], [RA8461; H, F, F, H, Bu, CF ₃ CH ₂ ], [RA8462; H, F, F, H, Bu, CF ₃ CF ₂ ], [RA8463; H, F, F, H, Bu, CF ₂ H] , [RA8464; H, F, F, H, Bu, CF ₂ HCH ₂ ], [RA8465; H, F, F, F, Bu, Me], [RA8466; H, F, F, F, Bu, Et ], [RA8467; H, F, F, F, Bu, Pr], [RA8468; H, F, F, F, Bu, i-Pr], [RA8469; H, F, F, F, Bu, c -Pr], [RA8470; H, F, F, F, Bu, Bu], [RA8471; H, F, F, F, Bu, i-Bu], [RA8472; H, F, F, F, Bu , t-Bu], [RA8473; H, F, F, F, Bu, c-PrCH ₂ ], [RA8474; H, F, F, F, Bu, Ph], [RA8475; H, F, F, F, Bu, Bn], [RA8476; H, F, F, F, Bu, CF ₃ ], [RA8477; H, F, F, F, Bu, CF ₃ CH ₂ ], [RA8478; H, F, F, F, Bu, CF ₃ CF ₂ ], [RA8479; H, F, F, F, Bu, CF ₂ H], [RA8480; H, F, F, F, Bu, CF ₂ HCH ₂ ], [RA8481; H, F, F, Cl, Bu, Me], [RA8482; H, F, F, Cl, Bu, Et], [RA8483; H, F, F, Cl, Bu, Pr], [RA8484; H, F, F, Cl, Bu, i-Pr], [RA8485; H, F, F, Cl, Bu, c-Pr], [RA8486; H, F, F, Cl, Bu, Bu], [RA8487; H, F, F, Cl, Bu, i-Bu], [RA8488; H, F, F, Cl, Bu, t-Bu], [RA8489; H, F, F, Cl, Bu, c-PrCH ₂ ], [RA8490; H, F , F, Cl, Bu, Ph], [RA8491; H, F, F, Cl, Bu, Bn], [RA8492; H, F, F, Cl, Bu, CF ₃ ], [RA8493; H, F, F, Cl, Bu, CF ₃ CH ₂ ], [RA8494; H, F, F, Cl, Bu, CF ₃ CF ₂ ], [RA8495; H, F, F, Cl, Bu, CF ₂ H], [ RA8496; H, F, F, Cl, Bu, CF ₂ HCH ₂ ], [RA8497; H, F, Cl, H, Bu, Me], [RA8498; H, F, Cl, H, Bu, Et], [RA8499; H, F, Cl, H, Bu, Pr], [RA8500; H, F, Cl, H, Bu, i-Pr], [RA8501; H, F, Cl, H, Bu, c-Pr ], [RA8502; H, F, Cl, H, Bu, Bu], [RA8503; H, F, Cl, H, Bu, i-Bu], [RA8504; H, F, Cl, H, Bu, t -Bu], [RA8505; H, F, Cl, H, Bu, c-PrCH ₂ ], [RA8506; H, F, Cl, H, Bu, Ph], [RA8507; H, F, Cl, H, Bu, Bn], [RA8508; H, F, Cl, H, Bu, CF ₃ ], [RA8509; H, F, Cl, H, Bu, CF ₃ CH ₂ ], [RA8510; H, F, Cl, H, Bu, CF ₃ CF ₂ ], [RA8511; H, F, Cl, H, Bu, CF ₂ H], [RA8512; H, F, Cl, H, Bu, CF ₂ HCH ₂ ] , [RA8513; H, F, Cl, Cl, Bu, Me], [RA8514; H, F, Cl, Cl, Bu, Et], [RA8515; H, F, Cl, Cl, Bu, Pr], [ RA8516; H, F, Cl, Cl, Bu, i-Pr], [RA8517; H, F, Cl, Cl, Bu, c-Pr], [RA8518; H, F, Cl, Cl, Bu, Bu] , [RA8519; H, F, Cl, Cl, Bu, i-Bu], [RA8520; H, F, Cl, Cl, Bu, t-Bu], [RA8521; H, F, Cl, Cl, Bu, c-PrCH ₂ ], [RA8522; H, F, Cl, Cl, Bu, Ph], [RA8523; H, F, Cl, Cl, Bu, Bn], [RA8524; H, F, Cl, Cl, Bu , CF ₃ ], [RA8525; H, F, Cl, Cl, Bu, CF ₃ CH ₂ ], [RA8526; H, F, Cl, Cl, Bu, CF ₃ CF ₂ ], [RA8527; H, F, Cl, Cl, Bu, CF ₂ H], [RA8528; H, F, Cl, Cl, Bu, CF ₂ HCH ₂ ], [RA8529; H, F, Me, H, i-Pr, Me], [RA8530 ; H, F, Me, H, i-Pr, Et], [RA8531; H, F, Me, H, i-Pr, Pr], [RA8532; H, F, Me, H, i-Pr, i -Pr], [RA8533; H, F, Me, H, i-Pr, c-Pr], [RA8534; H, F, Me, H, i-Pr, Bu], [RA8535; H, F, Me , H, i-Pr, i-Bu], [RA8536; H, F, Me, H, i-Pr, t-Bu], [RA8537; H, F, Me, H, i-Pr, c-PrCH ₂ ], [RA8538; H, F, Me, H, i-Pr, Ph], [RA8539; H, F, Me, H, i-Pr, Bn], [RA8540; H, F, Me, H, i-Pr, CF ₃ ], [RA8541; H, F, Me, H, i-Pr, CF ₃ CH ₂ ], [RA8542; H, F, Me, H, i-Pr, CF ₃ CF ₂ ], [RA8543; H, F, Me, H, i-Pr, CF ₂ H], [RA8544; H, F, Me, H, i-Pr, CF ₂ HCH ₂ ], [RA8545; H, F, Me, Me, i-Pr, Me], [RA8546; H, F, Me, Me, i-Pr, Et], [RA8547; H, F, Me, Me, i-Pr, Pr], [RA8548; H, F, Me, Me, i-Pr, i-Pr], [RA8549; H, F, Me, Me, i-Pr, c-Pr], [RA8550; H, F, Me, Me, i- Pr, Bu], [RA8551; H, F, Me, Me, i-Pr, i-Bu], [RA8552; H, F, Me, Me, i-Pr, t-Bu], [RA8553; H, F, Me, Me, i-Pr, c-PrCH ₂ ], [RA8554; H, F, Me, Me, i-Pr, Ph], [RA8555; H, F, Me, Me, i-Pr, Bn ], [RA8556; H, F, Me, Me, i-Pr, CF ₃ ], [RA8557; H, F, Me, Me, i-Pr, CF ₃ CH ₂ ], [RA8558; H, F, Me , Me, i-Pr, CF ₃ CF ₂ ], [RA8559; H, F, Me, Me, i-Pr, CF ₂ H], [RA8560; H, F, Me, Me, i-Pr, CF ₂ HCH ₂ ], [RA8561; H, F, Me, Et, i-Pr, Me], [RA8562; H, F, Me, Et, i-Pr, Et], [RA8563; H, F, Me, Et , i-Pr, Pr], [RA8564; H, F, Me, Et, i-Pr, i-Pr], [RA8565; H, F, Me, Et, i-Pr, c-Pr], [RA8566 ; H, F, Me, Et, i-Pr, Bu], [RA8567; H, F, Me, Et, i-Pr, i-Bu], [RA8568; H, F, Me, Et, i-Pr , t-Bu], [RA8569; H, F, Me, Et, i-Pr, c-PrCH ₂ ], [RA8570; H, F, Me, Et, i-Pr, Ph], [RA8571; H, F, Me, Et, i-Pr, Bn], [RA8572; H, F, Me, Et, i-Pr, CF ₃ ], [RA8573; H, F, Me, Et, i-Pr, CF ₃ CH ₂ ], [RA8574; H, F, Me, Et, i-Pr, CF ₃ CF ₂ ], [RA8575; H, F, Me, Et, i-Pr, CF ₂ H], [RA8576; H, F , Me, Et, i-Pr, CF ₂ HCH ₂ ], [RA8577; H, F, Me, F, i-Pr, Me], [RA8578; H, F, Me, F, i-Pr, Et] , [RA8579; H, F, Me, F, i-Pr, Pr], [RA8580; H, F, Me, F, i-Pr, i-Pr], [RA8581; H, F, Me, F, i-Pr, cP r], [RA8582; H, F, Me, F, i-Pr, Bu], [RA8583; H, F, Me, F, i-Pr, i-Bu], [RA8584; H, F, Me, F, i-Pr, t-Bu], [RA8585; H, F, Me, F, i-Pr, c-PrCH ₂ ], [RA8586; H, F, Me, F, i-Pr, Ph], [RA8587; H, F, Me, F, i-Pr, Bn], [RA8588; H, F, Me, F, i-Pr, CF ₃ ], [RA8589; H, F, Me, F, i- Pr, CF ₃ CH ₂ ], [RA8590; H, F, Me, F, i-Pr, CF ₃ CF ₂ ], [RA8591; H, F, Me, F, i-Pr, CF ₂ H], [ RA8592; H, F, Me, F, i-Pr, CF ₂ HCH ₂ ], [RA8593; H, F, Me, Cl, i-Pr, Me], [RA8594; H, F, Me, Cl, i -Pr, Et], [RA8595; H, F, Me, Cl, i-Pr, Pr], [RA8596; H, F, Me, Cl, i-Pr, i-Pr], [RA8597; H, F , Me, Cl, i-Pr, c-Pr], [RA8598; H, F, Me, Cl, i-Pr, Bu], [RA8599; H, F, Me, Cl, i-Pr, i-Bu ], [RA8600; H, F, Me, Cl, i-Pr, t-Bu],

[RA8601; H, F, Me, Cl, i-Pr, c-PrCH ₂ ], [RA8602; H, F, Me, Cl, i-Pr, Ph], [RA8603; H, F, Me, Cl, i-Pr, Bn], [RA8604; H, F, Me, Cl, i-Pr, CF ₃ ], [RA8605; H, F, Me, Cl, i-Pr, CF ₃ CH ₂ ], [RA8606; H, F, Me, Cl, i-Pr, CF ₃ CF ₂ ], [RA8607; H, F, Me, Cl, i-Pr, CF ₂ H], [RA8608; H, F, Me, Cl, i -Pr, CF ₂ HCH ₂ ], [RA8609; H, F, Et, H, i-Pr, Me], [RA8610; H, F, Et, H, i-Pr, Et], [RA8611; H, F, Et, H, i-Pr, Pr], [RA8612; H, F, Et, H, i-Pr, i-Pr], [RA8613; H, F, Et, H, i-Pr, c- Pr], [RA8614; H, F, Et, H, i-Pr, Bu], [RA8615; H, F, Et, H, i-Pr, i-Bu], [RA8616; H, F, Et, H, i-Pr, t-Bu], [RA8617; H, F, Et, H, i-Pr, c-PrCH ₂ ], [RA8618; H, F, Et, H, i-Pr, Ph], [RA8619; H, F, Et, H, i-Pr, Bn], [RA8620; H, F, Et, H, i-Pr, CF ₃ ], [RA8621; H, F, Et, H, i- Pr, CF ₃ CH ₂ ], [RA8622; H, F, Et, H, i-Pr, CF ₃ CF ₂ ], [RA8623; H, F, Et, H, i-Pr, CF ₂ H], [ RA8624; H, F, Et, H, i-Pr, CF ₂ HCH ₂ ], [RA8625; H, F, Et, F, i-Pr, Me], [RA8626; H, F, Et, F, i -Pr, Et], [RA8627; H, F, Et, F, i-Pr, Pr], [RA8628; H, F, Et, F, i-Pr, i-Pr], [RA8629; H, F , Et, F, i-Pr, c-Pr], [RA8630; H, F, Et, F, i-Pr, Bu], [RA8631; H, F, Et, F, i-Pr, i-Bu ], [RA8632; H, F, Et, F, i-Pr, t-Bu], [RA8633; H, F, Et, F, i-Pr, c-PrCH ₂ ], [RA8634; H, F, Et, F, i-Pr, Ph], [RA8635 ; H, F, Et, F, i-Pr, Bn], [RA8636; H, F, Et, F, i-Pr, CF ₃ ], [RA8637; H, F, Et, F, i-Pr, CF ₃ CH ₂ ], [RA8638; H, F, Et, F, i-Pr, CF ₃ CF ₂ ], [RA8639; H, F, Et, F, i-Pr, CF ₂ H], [RA8640; H, F, Et, F, i-Pr, CF ₂ HCH ₂ ], [RA8641; H, F, Et, Cl, i-Pr, Me], [RA8642; H, F, Et, Cl, i-Pr , Et], [RA8643; H, F, Et, Cl, i-Pr, Pr], [RA8644; H, F, Et, Cl, i-Pr, i-Pr], [RA8645; H, F, Et , Cl, i-Pr, c-Pr], [RA8646; H, F, Et, Cl, i-Pr, Bu], [RA8647; H, F, Et, Cl, i-Pr, i-Bu], [RA8648; H, F, Et, Cl, i-Pr, t-Bu], [RA8649; H, F, Et, Cl, i-Pr, c-PrCH ₂ ], [RA8650; H, F, Et, Cl, i-Pr, Ph], [RA8651; H, F, Et, Cl, i-Pr, Bn], [RA8652; H, F, Et, Cl, i-Pr, CF ₃ ], [RA8653; H , F, Et, Cl, i-Pr, CF ₃ CH ₂ ], [RA8654; H, F, Et, Cl, i-Pr, CF ₃ CF ₂ ], [RA8655; H, F, Et, Cl, i -Pr, CF ₂ H], [RA8656; H, F, Et, Cl, i-Pr, CF ₂ HCH ₂ ], [RA8657; H, F, F, H, i-Pr, Me], [RA8658; H, F, F, H, i-Pr, Et], [RA8659; H, F, F, H, i-Pr, Pr], [RA8660; H, F, F, H, i-Pr, i- Pr], [RA8661; H, F, F, H, i-Pr, c-Pr], [RA8662; H, F, F, H, i-Pr, Bu], [RA8663; H, F, F, H, i-Pr, i-Bu], [RA8664; H, F, F, H, i-Pr, t-Bu], [RA8665; H, F, F, H, i-Pr, c-PrCH ₂ ], [RA8666; H, F, F, H, i-Pr, Ph], [RA8667; H, F, F, H, i-Pr, Bn], [RA8668; H, F, F, H, i -Pr, CF ₃ ], [RA8669; H, F, F, H, i-Pr, C F ₃ CH ₂ ], [RA8670; H, F, F, H, i-Pr, CF ₃ CF ₂ ], [RA8671; H, F, F, H, i-Pr, CF ₂ H], [RA8672; H, F, F, H, i-Pr, CF ₂ HCH ₂ ], [RA8673; H, F, F, F, i-Pr, Me], [RA8674; H, F, F, F, i-Pr , Et], [RA8675; H, F, F, F, i-Pr, Pr], [RA8676; H, F, F, F, i-Pr, i-Pr], [RA8677; H, F, F , F, i-Pr, c-Pr], [RA8678; H, F, F, F, i-Pr, Bu], [RA8679; H, F, F, F, i-Pr, i-Bu], [RA8680; H, F, F, F, i-Pr, t-Bu], [RA8681; H, F, F, F, i-Pr, c-PrCH ₂ ], [RA8682; H, F, F, F, i-Pr, Ph], [RA8683; H, F, F, F, i-Pr, Bn], [RA8684; H, F, F, F, i-Pr, CF ₃ ], [RA8685; H , F, F, F, i-Pr, CF ₃ CH ₂ ], [RA8686; H, F, F, F, i-Pr, CF ₃ CF ₂ ], [RA8687; H, F, F, F, i -Pr, CF ₂ H], [RA8688; H, F, F, F, i-Pr, CF ₂ HCH ₂ ], [RA8689; H, F, F, Cl, i-Pr, Me], [RA8690; H, F, F, Cl, i-Pr, Et], [RA8691; H, F, F, Cl, i-Pr, Pr], [RA8692; H, F, F, Cl, i-Pr, i- Pr], [RA8693; H, F, F, Cl, i-Pr, c-Pr], [RA8694; H, F, F, Cl, i-Pr, Bu], [RA8695; H, F, F, Cl, i-Pr, i-Bu], [RA8696; H, F, F, Cl, i-Pr, t-Bu], [RA8697; H, F, F, Cl, i-Pr, c-PrCH ₂ ], [RA8698; H, F, F, Cl, i-Pr, Ph], [RA8699; H, F, F, Cl, i-Pr, Bn], [RA8700; H, F, F, Cl, i -Pr, CF ₃ ], [RA8701; H, F, F, Cl, i-Pr, CF ₃ CH ₂ ], [RA8702; H, F, F, Cl, i-Pr, CF ₃ CF ₂ ], [ RA8703; H, F, F, Cl, i-Pr, CF ₂ H], [RA8704; H, F, F, Cl, i -Pr, CF ₂ HCH ₂ ], [RA8705; H, F, Cl, H, i-Pr, Me], [RA8706; H, F, Cl, H, i-Pr, Et], [RA8707; H, F, Cl, H, i-Pr, Pr], [RA8708; H, F, Cl, H, i-Pr, i-Pr], [RA8709; H, F, Cl, H, i-Pr, c- Pr], [RA8710; H, F, Cl, H, i-Pr, Bu], [RA8711; H, F, Cl, H, i-Pr, i-Bu], [RA8712; H, F, Cl, H, i-Pr, t-Bu], [RA8713; H, F, Cl, H, i-Pr, c-PrCH ₂ ], [RA8714; H, F, Cl, H, i-Pr, Ph], [RA8715; H, F, Cl, H, i-Pr, Bn], [RA8716; H, F, Cl, H, i-Pr, CF ₃ ], [RA8717; H, F, Cl, H, i- Pr, CF ₃ CH ₂ ], [RA8718; H, F, Cl, H, i-Pr, CF ₃ CF ₂ ], [RA8719; H, F, Cl, H, i-Pr, CF ₂ H], [ RA8720; H, F, Cl, H, i-Pr, CF ₂ HCH ₂ ], [RA8721; H, F, Cl, Cl, i-Pr, Me], [RA8722; H, F, Cl, Cl, i -Pr, Et], [RA8723; H, F, Cl, Cl, i-Pr, Pr], [RA8724; H, F, Cl, Cl, i-Pr, i-Pr], [RA8725; H, F , Cl, Cl, i-Pr, c-Pr], [RA8726; H, F, Cl, Cl, i-Pr, Bu], [RA8727; H, F, Cl, Cl, i-Pr, i-Bu ], [RA8728; H, F, Cl, Cl, i-Pr, t-Bu], [RA8729; H, F, Cl, Cl, i-Pr, c-PrCH ₂ ], [RA8730; H, F, Cl, Cl, i-Pr, Ph], [RA8731; H, F, Cl, Cl, i-Pr, Bn], [RA8732; H, F, Cl, Cl, i-Pr, CF ₃ ], [RA8733 ; H, F, Cl, Cl, i-Pr, CF ₃ CH ₂ ], [RA8734; H, F, Cl, Cl, i-Pr, CF ₃ CF ₂ ], [RA8735; H, F, Cl, Cl , i-Pr, CF ₂ H], [RA8736; H, F, Cl, Cl, i-Pr, CF ₂ HCH ₂ ], [RA8737; H, F, Me, H, c-Pr, Me], [ RA8738; H, F, Me, H, c-Pr, Et], [RA8739; H, F, Me, H, c-Pr, Pr], [RA8740; H, F, Me, H, c-Pr, i-Pr], [RA8741; H, F, Me, H, c-Pr, c-Pr], [RA8742; H, F, Me, H, c-Pr, Bu], [RA8743; H, F, Me, H, c-Pr, i-Bu], [RA8744; H, F, Me, H, c-Pr, t-Bu], [RA8745; H, F, Me, H, c-Pr, c-PrCH ₂ ], [RA8746; H , F, Me, H, c-Pr, Ph], [RA8747; H, F, Me, H, c-Pr, Bn], [RA8748; H, F, Me, H, c-Pr, CF ₃ ] , [RA8749; H, F, Me, H, c-Pr, CF ₃ CH ₂ ], [RA8750; H, F, Me, H, c-Pr, CF ₃ CF ₂ ], [RA8751; H, F, Me, H, c-Pr, CF ₂ H], [RA8752; H, F, Me, H, c-Pr, CF ₂ HCH ₂ ], [RA8753; H, F, Me, Me, c-Pr, Me ], [RA8754; H, F, Me, Me, c-Pr, Et], [RA8755; H, F, Me, Me, c-Pr, Pr], [RA8756; H, F, Me, Me, c -Pr, i-Pr], [RA8757; H, F, Me, Me, c-Pr, c-Pr], [RA8758; H, F, Me, Me, c-Pr, Bu], [RA8759; H , F, Me, Me, c-Pr, i-Bu], [RA8760; H, F, Me, Me, c-Pr, t-Bu], [RA8761; H, F, Me, Me, c-Pr , c-PrCH ₂ ], [RA8762; H, F, Me, Me, c-Pr, Ph], [RA8763; H, F, Me, Me, c-Pr, Bn], [RA8764; H, F, Me, Me, c-Pr, CF ₃ ], [RA8765; H, F, Me, Me, c-Pr, CF ₃ CH ₂ ], [RA8766; H, F, Me, Me, c-Pr, CF ₃ CF ₂ ], [RA8767; H, F, Me, Me, c-Pr, CF ₂ H], [RA8768; H, F, Me, Me, c-Pr, CF ₂ HCH ₂ ], [RA8769; H, F, Me, Et, c-Pr, Me], [RA8770; H, F, Me, Et, c-Pr, Et], [RA8771; H, F, Me, Et, c-Pr, Pr], [ RA8772; H, F, Me, Et, c-Pr, i-Pr], [RA8773; H, F, Me, Et, c-Pr, c-Pr], [RA8774; H, F, Me, Et, c-Pr, Bu], [RA8775; H, F, Me, Et, c-Pr, i-Bu], [RA8776; H, F, Me, Et, c-Pr, t-Bu], [RA8777; H, F, Me, Et, c- Pr, c-PrCH ₂ ], [RA8778; H, F, Me, Et, c-Pr, Ph], [RA8779; H, F, Me, Et, c-Pr, Bn], [RA8780; H, F , Me, Et, c-Pr, CF ₃ ], [RA8781; H, F, Me, Et, c-Pr, CF ₃ CH ₂ ], [RA8782; H, F, Me, Et, c-Pr, CF ₃ CF ₂ ], [RA8783; H, F, Me, Et, c-Pr, CF ₂ H], [RA8784; H, F, Me, Et, c-Pr, CF ₂ HCH ₂ ], [RA8785; H , F, Me, F, c-Pr, Me], [RA8786; H, F, Me, F, c-Pr, Et], [RA8787; H, F, Me, F, c-Pr, Pr], [RA8788; H, F, Me, F, c-Pr, i-Pr], [RA8789; H, F, Me, F, c-Pr, c-Pr], [RA8790; H, F, Me, F , c-Pr, Bu], [RA8791; H, F, Me, F, c-Pr, i-Bu], [RA8792; H, F, Me, F, c-Pr, t-Bu], [RA8793 ; H, F, Me, F, c-Pr, c-PrCH ₂ ], [RA8794; H, F, Me, F, c-Pr, Ph], [RA8795; H, F, Me, F, c- Pr, Bn], [RA8796; H, F, Me, F, c-Pr, CF ₃ ], [RA8797; H, F, Me, F, c-Pr, CF ₃ CH ₂ ], [RA8798; H, F, Me, F, c-Pr, CF ₃ CF ₂ ], [RA8799; H, F, Me, F, c-Pr, CF ₂ H], [RA8800; H, F, Me, F, c-Pr , CF ₂ HCH ₂ ],

[RA8801; H, F, Me, Cl, c-Pr, Me], [RA8802; H, F, Me, Cl, c-Pr, Et], [RA8803; H, F, Me, Cl, c-Pr , Pr], [RA8804; H, F, Me, Cl, c-Pr, i-Pr], [RA8805; H, F, Me, Cl, c-Pr, c-Pr], [RA8806; H, F , Me, Cl, c-Pr, Bu], [RA8807; H, F, Me, Cl, c-Pr, i-Bu], [RA8808; H, F, Me, Cl, c-Pr, t-Bu ], [RA8809; H, F, Me, Cl, c-Pr, c-PrCH ₂ ], [RA8810; H, F, Me, Cl, c-Pr, Ph], [RA8811; H, F, Me, Cl, c-Pr, Bn], [RA8812; H, F, Me, Cl, c-Pr, CF ₃ ], [RA8813; H, F, Me, Cl, c-Pr, CF ₃ CH ₂ ], [ RA8814; H, F, Me, Cl, c-Pr, CF ₃ CF ₂ ], [RA8815; H, F, Me, Cl, c-Pr, CF ₂ H], [RA8816; H, F, Me, Cl , c-Pr, CF ₂ HCH ₂ ], [RA8817; H, F, Et, H, c-Pr, Me], [RA8818; H, F, Et, H, c-Pr, Et], [RA8819; H, F, Et, H, c-Pr, Pr], [RA8820; H, F, Et, H, c-Pr, i-Pr], [RA8821; H, F, Et, H, c-Pr, c-Pr], [RA8822; H, F, Et, H, c-Pr, Bu], [RA8823; H, F, Et, H, c-Pr, i-Bu], [RA8824; H, F, Et, H, c-Pr, t-Bu], [RA8825; H, F, Et, H, c-Pr, c-PrCH ₂ ], [RA8826; H, F, Et, H, c-Pr, Ph ], [RA8827; H, F, Et, H, c-Pr, Bn], [RA8828; H, F, Et, H, c-Pr, CF ₃ ], [RA8829; H, F, Et, H, c-Pr, CF ₃ CH ₂ ], [RA8830; H, F, Et, H, c-Pr, CF ₃ CF ₂ ], [RA8831; H, F, Et, H, c-Pr, CF ₂ H] , [RA8832; H, F, Et, H, c-Pr, CF ₂ HCH ₂ ], [RA8833; H, F, Et, F, c-Pr, Me], [RA8834; H, F, Et, F , c-Pr, Et], [RA883 5; H, F, Et, F, c-Pr, Pr], [RA8836; H, F, Et, F, c-Pr, i-Pr], [RA8837; H, F, Et, F, c- Pr, c-Pr], [RA8838; H, F, Et, F, c-Pr, Bu], [RA8839; H, F, Et, F, c-Pr, i-Bu], [RA8840; H, F, Et, F, c-Pr, t-Bu], [RA8841; H, F, Et, F, c-Pr, c-PrCH ₂ ], [RA8842; H, F, Et, F, c-Pr , Ph], [RA8843; H, F, Et, F, c-Pr, Bn], [RA8844; H, F, Et, F, c-Pr, CF ₃ ], [RA8845; H, F, Et, F, c-Pr, CF ₃ CH ₂ ], [RA8846; H, F, Et, F, c-Pr, CF ₃ CF ₂ ], [RA8847; H, F, Et, F, c-Pr, CF ₂ H], [RA8848; H, F, Et, F, c-Pr, CF ₂ HCH ₂ ], [RA8849; H, F, Et, Cl, c-Pr, Me], [RA8850; H, F, Et , Cl, c-Pr, Et], [RA8851; H, F, Et, Cl, c-Pr, Pr], [RA8852; H, F, Et, Cl, c-Pr, i-Pr], [RA8853 ; H, F, Et, Cl, c-Pr, c-Pr], [RA8854; H, F, Et, Cl, c-Pr, Bu], [RA8855; H, F, Et, Cl, c-Pr , i-Bu], [RA8856; H, F, Et, Cl, c-Pr, t-Bu], [RA8857; H, F, Et, Cl, c-Pr, c-PrCH ₂ ], [RA8858; H, F, Et, Cl, c-Pr, Ph], [RA8859; H, F, Et, Cl, c-Pr, Bn], [RA8860; H, F, Et, Cl, c-Pr, CF ₃ ], [RA8861; H, F, Et, Cl, c-Pr, CF ₃ CH ₂ ], [RA8862; H, F, Et, Cl, c-Pr, CF ₃ CF ₂ ], [RA8863; H, F , Et, Cl, c-Pr, CF ₂ H], [RA8864; H, F, Et, Cl, c-Pr, CF ₂ HCH ₂ ], [RA8865; H, F, F, H, c-Pr, Me], [RA8866; H, F, F, H, c-Pr, Et], [RA8867; H, F, F, H, c-Pr, Pr], [RA8868; H, F, F, H, c-Pr, i-Pr], [RA8869; H, F, F, H, c-Pr, c-Pr], [RA8870; H, F, F, H, c-Pr, Bu], [RA8871; H, F, F, H, c-Pr, i-Bu], [ RA8872; H, F, F, H, c-Pr, t-Bu], [RA8873; H, F, F, H, c-Pr, c-PrCH ₂ ], [RA8874; H, F, F, H , c-Pr, Ph], [RA8875; H, F, F, H, c-Pr, Bn], [RA8876; H, F, F, H, c-Pr, CF ₃ ], [RA8877; H, F, F, H, c-Pr, CF ₃ CH ₂ ], [RA8878; H, F, F, H, c-Pr, CF ₃ CF ₂ ], [RA8879; H, F, F, H, c- Pr, CF ₂ H], [RA8880; H, F, F, H, c-Pr, CF ₂ HCH ₂ ], [RA8881; H, F, F, F, c-Pr, Me], [RA8882; H , F, F, F, c-Pr, Et], [RA8883; H, F, F, F, c-Pr, Pr], [RA8884; H, F, F, F, c-Pr, i-Pr ], [RA8885; H, F, F, F, c-Pr, c-Pr], [RA8886; H, F, F, F, c-Pr, Bu], [RA8887; H, F, F, F , c-Pr, i-Bu], [RA8888; H, F, F, F, c-Pr, t-Bu], [RA8889; H, F, F, F, c-Pr, c-PrCH ₂ ] , [RA8890; H, F, F, F, c-Pr, Ph], [RA8891; H, F, F, F, c-Pr, Bn], [RA8892; H, F, F, F, c- Pr, CF ₃ ], [RA8893; H, F, F, F, c-Pr, CF ₃ CH ₂ ], [RA8894; H, F, F, F, c-Pr, CF ₃ CF ₂ ], [RA8895 ; H, F, F, F, c-Pr, CF ₂ H], [RA8896; H, F, F, F, c-Pr, CF ₂ HCH ₂ ], [RA8897; H, F, F, Cl, c-Pr, Me], [RA8898; H, F, F, Cl, c-Pr, Et], [RA8899; H, F, F, Cl, c-Pr, Pr], [RA8900; H, F, F, Cl, c-Pr, i-Pr], [RA8901; H, F, F, Cl, c-Pr, c-Pr], [RA8902; H, F, F, Cl, c-Pr, Bu] , [RA8903; H, F, F, Cl, c-Pr, i-Bu], [RA8904; H, F, F, Cl, c-Pr, t-Bu], [RA890 5; H, F, F, Cl, c-Pr, c-PrCH ₂ ], [RA8906; H, F, F, Cl, c-Pr, Ph], [RA8907; H, F, F, Cl, c -Pr, Bn], [RA8908; H, F, F, Cl, c-Pr, CF ₃ ], [RA8909; H, F, F, Cl, c-Pr, CF ₃ CH ₂ ], [RA8910; H , F, F, Cl, c-Pr, CF ₃ CF ₂ ], [RA8911; H, F, F, Cl, c-Pr, CF ₂ H], [RA8912; H, F, F, Cl, c- Pr, CF ₂ HCH ₂ ], [RA8913; H, F, Cl, H, c-Pr, Me], [RA8914; H, F, Cl, H, c-Pr, Et], [RA8915; H, F , Cl, H, c-Pr, Pr], [RA8916; H, F, Cl, H, c-Pr, i-Pr], [RA8917; H, F, Cl, H, c-Pr, c-Pr ], [RA8918; H, F, Cl, H, c-Pr, Bu], [RA8919; H, F, Cl, H, c-Pr, i-Bu], [RA8920; H, F, Cl, H , c-Pr, t-Bu], [RA8921; H, F, Cl, H, c-Pr, c-PrCH ₂ ], [RA8922; H, F, Cl, H, c-Pr, Ph], [ RA8923; H, F, Cl, H, c-Pr, Bn], [RA8924; H, F, Cl, H, c-Pr, CF ₃ ], [RA8925; H, F, Cl, H, c-Pr , CF ₃ CH ₂ ], [RA8926; H, F, Cl, H, c-Pr, CF ₃ CF ₂ ], [RA8927; H, F, Cl, H, c-Pr, CF ₂ H], [RA8928 ; H, F, Cl, H, c-Pr, CF ₂ HCH ₂ ], [RA8929; H, F, Cl, Cl, c-Pr, Me], [RA8930; H, F, Cl, Cl, c- Pr, Et], [RA8931; H, F, Cl, Cl, c-Pr, Pr], [RA8932; H, F, Cl, Cl, c-Pr, i-Pr], [RA8933; H, F, Cl, Cl, c-Pr, c-Pr], [RA8934; H, F, Cl, Cl, c-Pr, Bu], [RA8935; H, F, Cl, Cl, c-Pr, i-Bu] , [RA8936; H, F, Cl, Cl, c-Pr, t-Bu], [RA8937; H, F, Cl, Cl, c-Pr, c-PrCH ₂ ], [RA8938; H, F, Cl , Cl, c-Pr, Ph], [RA8939; H, F , Cl, Cl, c-Pr, Bn], [RA8940; H, F, Cl, Cl, c-Pr, CF ₃ ], [RA8941; H, F, Cl, Cl, c-Pr, CF ₃ CH ₂ ], [RA8942; H, F, Cl, Cl, c-Pr, CF ₃ CF ₂ ], [RA8943; H, F, Cl, Cl, c-Pr, CF ₂ H], [RA8944; H, F, Cl, Cl, c-Pr, CF ₂ HCH ₂ ], [RA8945; H, F, Me, H, i-Bu, Me], [RA8946; H, F, Me, H, i-Bu, Et], [RA8947; H, F, Me, H, i-Bu, Pr], [RA8948; H, F, Me, H, i-Bu, i-Pr], [RA8949; H, F, Me, H, i -Bu, c-Pr], [RA8950; H, F, Me, H, i-Bu, Bu], [RA8951; H, F, Me, H, i-Bu, i-Bu], [RA8952; H , F, Me, H, i-Bu, t-Bu], [RA8953; H, F, Me, H, i-Bu, c-PrCH ₂ ], [RA8954; H, F, Me, H, i- Bu, Ph], [RA8955; H, F, Me, H, i-Bu, Bn], [RA8956; H, F, Me, H, i-Bu, CF ₃ ], [RA8957; H, F, Me , H, i-Bu, CF ₃ CH ₂ ], [RA8958; H, F, Me, H, i-Bu, CF ₃ CF ₂ ], [RA8959; H, F, Me, H, i-Bu, CF ₂ H], [RA8960; H, F, Me, H, i-Bu, CF ₂ HCH ₂ ], [RA8961; H, F, Me, Me, i-Bu, Me], [RA8962; H, F, Me, Me, i-Bu, Et], [RA8963; H, F, Me, Me, i-Bu, Pr], [RA8964; H, F, Me, Me, i-Bu, i-Pr], [ RA8965; H, F, Me, Me, i-Bu, c-Pr], [RA8966; H, F, Me, Me, i-Bu, Bu], [RA8967; H, F, Me, Me, i- Bu, i-Bu], [RA8968; H, F, Me, Me, i-Bu, t-Bu], [RA8969; H, F, Me, Me, i-Bu, c-PrCH ₂ ], [RA8970 ; H, F, Me, Me, i-Bu, Ph], [RA8971; H, F, Me, Me, i-Bu, Bn], [RA8972; H, F, Me, Me, i-Bu, CF ₃ ], [RA8973; H, F, Me, Me, i-Bu, CF ₃ CH ₂ ], [RA8974; H, F, Me, Me, i-Bu, CF ₃ CF ₂ ], [RA8975; H, F, Me, Me, i-Bu, CF ₂ H], [RA8976; H, F, Me, Me, i-Bu, CF ₂ HCH ₂ ], [RA8977; H, F, Me, Et, i-Bu, Me], [RA8978; H, F , Me, Et, i-Bu, Et], [RA8979; H, F, Me, Et, i-Bu, Pr], [RA8980; H, F, Me, Et, i-Bu, i-Pr], [RA8981; H, F, Me, Et, i-Bu, c-Pr], [RA8982; H, F, Me, Et, i-Bu, Bu], [RA8983; H, F, Me, Et, i -Bu, i-Bu], [RA8984; H, F, Me, Et, i-Bu, t-Bu], [RA8985; H, F, Me, Et, i-Bu, c-PrCH ₂ ], [ RA8986; H, F, Me, Et, i-Bu, Ph], [RA8987; H, F, Me, Et, i-Bu, Bn], [RA8988; H, F, Me, Et, i-Bu, CF ₃ ], [RA8989; H, F, Me, Et, i-Bu, CF ₃ CH ₂ ], [RA8990; H, F, Me, Et, i-Bu, CF ₃ CF ₂ ], [RA8991; H , F, Me, Et, i-Bu, CF ₂ H], [RA8992; H, F, Me, Et, i-Bu, CF ₂ HCH ₂ ], [RA8993; H, F, Me, F, i- Bu, Me], [RA8994; H, F, Me, F, i-Bu, Et], [RA8995; H, F, Me, F, i-Bu, Pr], [RA8996; H, F, Me, F, i-Bu, i-Pr], [RA8997; H, F, Me, F, i-Bu, c-Pr], [RA8998; H, F, Me, F, i-Bu, Bu], [ RA8999; H, F, Me, F, i-Bu, i-Bu], [RA9000; H, F, Me, F, i-Bu, t-Bu],

[RA9001; H, F, Me, F, i-Bu, c-PrCH ₂ ], [RA9002; H, F, Me, F, i-Bu, Ph], [RA9003; H, F, Me, F, i-Bu, Bn], [RA9004; H, F, Me, F, i-Bu, CF ₃ ], [RA9005; H, F, Me, F, i-Bu, CF ₃ CH ₂ ], [RA9006; H, F, Me, F, i-Bu, CF ₃ CF ₂ ], [RA9007; H, F, Me, F, i-Bu, CF ₂ H], [RA9008; H, F, Me, F, i -Bu, CF ₂ HCH ₂ ], [RA9009; H, F, Me, Cl, i-Bu, Me], [RA9010; H, F, Me, Cl, i-Bu, Et], [RA9011; H, F, Me, Cl, i-Bu, Pr], [RA9012; H, F, Me, Cl, i-Bu, i-Pr], [RA9013; H, F, Me, Cl, i-Bu, c- Pr], [RA9014; H, F, Me, Cl, i-Bu, Bu], [RA9015; H, F, Me, Cl, i-Bu, i-Bu], [RA9016; H, F, Me, Cl, i-Bu, t-Bu], [RA9017; H, F, Me, Cl, i-Bu, c-PrCH ₂ ], [RA9018; H, F, Me, Cl, i-Bu, Ph], [RA9019; H, F, Me, Cl, i-Bu, Bn], [RA9020; H, F, Me, Cl, i-Bu, CF ₃ ], [RA9021; H, F, Me, Cl, i- Bu, CF ₃ CH ₂ ], [RA9022; H, F, Me, Cl, i-Bu, CF ₃ CF ₂ ], [RA9023; H, F, Me, Cl, i-Bu, CF ₂ H], [ RA9024; H, F, Me, Cl, i-Bu, CF ₂ HCH ₂ ], [RA9025; H, F, Et, H, i-Bu, Me], [RA9026; H, F, Et, H, i -Bu, Et], [RA9027; H, F, Et, H, i-Bu, Pr], [RA9028; H, F, Et, H, i-Bu, i-Pr], [RA9029; H, F , Et, H, i-Bu, c-Pr], [RA9030; H, F, Et, H, i-Bu, Bu], [RA9031; H, F, Et, H, i-Bu, i-Bu ], [RA9032; H, F, Et, H, i-Bu, t-Bu], [RA9033; H, F, Et, H, i-Bu, c-PrCH ₂ ], [RA9034; H, F, Et, H, i-Bu, Ph] , [RA9035; H, F, Et, H, i-Bu, Bn], [RA9036; H, F, Et, H, i-Bu, CF ₃ ], [RA9037; H, F, Et, H, i -Bu, CF ₃ CH ₂ ], [RA9038; H, F, Et, H, i-Bu, CF ₃ CF ₂ ], [RA9039; H, F, Et, H, i-Bu, CF ₂ H], [RA9040; H, F, Et, H, i-Bu, CF ₂ HCH ₂ ], [RA9041; H, F, Et, F, i-Bu, Me], [RA9042; H, F, Et, F, i-Bu, Et], [RA9043; H, F, Et, F, i-Bu, Pr], [RA9044; H, F, Et, F, i-Bu, i-Pr], [RA9045; H, F, Et, F, i-Bu, c-Pr], [RA9046; H, F, Et, F, i-Bu, Bu], [RA9047; H, F, Et, F, i-Bu, i- Bu], [RA9048; H, F, Et, F, i-Bu, t-Bu], [RA9049; H, F, Et, F, i-Bu, c-PrCH ₂ ], [RA9050; H, F , Et, F, i-Bu, Ph], [RA9051; H, F, Et, F, i-Bu, Bn], [RA9052; H, F, Et, F, i-Bu, CF ₃ ], [ RA9053; H, F, Et, F, i-Bu, CF ₃ CH ₂ ], [RA9054; H, F, Et, F, i-Bu, CF ₃ CF ₂ ], [RA9055; H, F, Et, F, i-Bu, CF ₂ H], [RA9056; H, F, Et, F, i-Bu, CF ₂ HCH ₂ ], [RA9057; H, F, Et, Cl, i-Bu, Me], [RA9058; H, F, Et, Cl, i-Bu, Et], [RA9059; H, F, Et, Cl, i-Bu, Pr], [RA9060; H, F, Et, Cl, i-Bu , i-Pr], [RA9061; H, F, Et, Cl, i-Bu, c-Pr], [RA9062; H, F, Et, Cl, i-Bu, Bu], [RA9063; H, F , Et, Cl, i-Bu, i-Bu], [RA9064; H, F, Et, Cl, i-Bu, t-Bu], [RA9065; H, F, Et, Cl, i-Bu, c -PrCH ₂ ], [RA9066; H, F, Et, Cl, i-Bu, Ph], [RA9067; H, F, Et, Cl, i-Bu, Bn], [RA9068; H, F, Et, Cl, i-Bu, CF ₃ ], [RA906 9; H, F, Et, Cl, i-Bu, CF ₃ CH ₂ ], [RA9070; H, F, Et, Cl, i-Bu, CF ₃ CF ₂ ], [RA9071; H, F, Et, Cl, i-Bu, CF ₂ H], [RA9072; H, F, Et, Cl, i-Bu, CF ₂ HCH ₂ ], [RA9073; H, F, F, H, i-Bu, Me], [RA9074; H, F, F, H, i-Bu, Et], [RA9075; H, F, F, H, i-Bu, Pr], [RA9076; H, F, F, H, i-Bu , i-Pr], [RA9077; H, F, F, H, i-Bu, c-Pr], [RA9078; H, F, F, H, i-Bu, Bu], [RA9079; H, F , F, H, i-Bu, i-Bu], [RA9080; H, F, F, H, i-Bu, t-Bu], [RA9081; H, F, F, H, i-Bu, c -PrCH ₂ ], [RA9082; H, F, F, H, i-Bu, Ph], [RA9083; H, F, F, H, i-Bu, Bn], [RA9084; H, F, F, H, i-Bu, CF ₃ ], [RA9085; H, F, F, H, i-Bu, CF ₃ CH ₂ ], [RA9086; H, F, F, H, i-Bu, CF ₃ CF ₂ ], [RA9087; H, F, F, H, i-Bu, CF ₂ H], [RA9088; H, F, F, H, i-Bu, CF ₂ HCH ₂ ], [RA9089; H, F, F, F, i-Bu, Me], [RA9090; H, F, F, F, i-Bu, Et], [RA9091; H, F, F, F, i-Bu, Pr], [RA9092; H, F, F, F, i-Bu, i-Pr], [RA9093; H, F, F, F, i-Bu, c-Pr], [RA9094; H, F, F, F, i- Bu, Bu], [RA9095; H, F, F, F, i-Bu, i-Bu], [RA9096; H, F, F, F, i-Bu, t-Bu], [RA9097; H, F, F, F, i-Bu, c-PrCH ₂ ], [RA9098; H, F, F, F, i-Bu, Ph], [RA9099; H, F, F, F, i-Bu, Bn ], [RA9100; H, F, F, F, i-Bu, CF ₃ ], [RA9101; H, F, F, F, i-Bu, CF ₃ CH ₂ ], [RA9102; H, F, F , F, i-Bu, CF ₃ CF ₂ ], [RA9103; H, F, F, F, i-Bu, CF ₂ H], [RA9104; H , F, F, F, i-Bu, CF ₂ HCH ₂ ], [RA9105; H, F, F, Cl, i-Bu, Me], [RA9106; H, F, F, Cl, i-Bu, Et], [RA9107; H, F, F, Cl, i-Bu, Pr], [RA9108; H, F, F, Cl, i-Bu, i-Pr], [RA9109; H, F, F, Cl, i-Bu, c-Pr], [RA9110; H, F, F, Cl, i-Bu, Bu], [RA9111; H, F, F, Cl, i-Bu, i-Bu], [ RA9112; H, F, F, Cl, i-Bu, t-Bu], [RA9113; H, F, F, Cl, i-Bu, c-PrCH ₂ ], [RA9114; H, F, F, Cl , i-Bu, Ph], [RA9115; H, F, F, Cl, i-Bu, Bn], [RA9116; H, F, F, Cl, i-Bu, CF ₃ ], [RA9117; H, F, F, Cl, i-Bu, CF ₃ CH ₂ ], [RA9118; H, F, F, Cl, i-Bu, CF ₃ CF ₂ ], [RA9119; H, F, F, Cl, i- Bu, CF ₂ H], [RA9120; H, F, F, Cl, i-Bu, CF ₂ HCH ₂ ], [RA9121; H, F, Cl, H, i-Bu, Me], [RA9122; H , F, Cl, H, i-Bu, Et], [RA9123; H, F, Cl, H, i-Bu, Pr], [RA9124; H, F, Cl, H, i-Bu, i-Pr ], [RA9125; H, F, Cl, H, i-Bu, c-Pr], [RA9126; H, F, Cl, H, i-Bu, Bu], [RA9127; H, F, Cl, H , i-Bu, i-Bu], [RA9128; H, F, Cl, H, i-Bu, t-Bu], [RA9129; H, F, Cl, H, i-Bu, c-PrCH ₂ ] , [RA9130; H, F, Cl, H, i-Bu, Ph], [RA9131; H, F, Cl, H, i-Bu, Bn], [RA9132; H, F, Cl, H, i- Bu, CF ₃ ], [RA9133; H, F, Cl, H, i-Bu, CF ₃ CH ₂ ], [RA9134; H, F, Cl, H, i-Bu, CF ₃ CF ₂ ], [RA9135 ; H, F, Cl, H, i-Bu, CF ₂ H], [RA9136; H, F, Cl, H, i-Bu, CF ₂ HCH ₂ ], [RA9137; H, F, Cl, Cl, i-Bu, Me], [RA9138; H, F, Cl, Cl, i-Bu , Et], [RA9139; H, F, Cl, Cl, i-Bu, Pr], [RA9140; H, F, Cl, Cl, i-Bu, i-Pr], [RA9141; H, F, Cl , Cl, i-Bu, c-Pr], [RA9142; H, F, Cl, Cl, i-Bu, Bu], [RA9143; H, F, Cl, Cl, i-Bu, i-Bu], [RA9144; H, F, Cl, Cl, i-Bu, t-Bu], [RA9145; H, F, Cl, Cl, i-Bu, c-PrCH ₂ ], [RA9146; H, F, Cl, Cl, i-Bu, Ph], [RA9147; H, F, Cl, Cl, i-Bu, Bn], [RA9148; H, F, Cl, Cl, i-Bu, CF ₃ ], [RA9149; H , F, Cl, Cl, i-Bu, CF ₃ CH ₂ ], [RA9150; H, F, Cl, Cl, i-Bu, CF ₃ CF ₂ ], [RA9151; H, F, Cl, Cl, i -Bu, CF ₂ H], [RA9152; H, F, Cl, Cl, i-Bu, CF ₂ HCH ₂ ], [RA9153; H, F, Me, H, t-Bu, Me], [RA9154; H, F, Me, H, t-Bu, Et], [RA9155; H, F, Me, H, t-Bu, Pr], [RA9156; H, F, Me, H, t-Bu, i- Pr], [RA9157; H, F, Me, H, t-Bu, c-Pr], [RA9158; H, F, Me, H, t-Bu, Bu], [RA9159; H, F, Me, H, t-Bu, i-Bu], [RA9160; H, F, Me, H, t-Bu, t-Bu], [RA9161; H, F, Me, H, t-Bu, c-PrCH ₂ ], [RA9162; H, F, Me, H, t-Bu, Ph], [RA9163; H, F, Me, H, t-Bu, Bn], [RA9164; H, F, Me, H, t -Bu, CF ₃ ], [RA9165; H, F, Me, H, t-Bu, CF ₃ CH ₂ ], [RA9166; H, F, Me, H, t-Bu, CF ₃ CF ₂ ], [ RA9167; H, F, Me, H, t-Bu, CF ₂ H], [RA9168; H, F, Me, H, t-Bu, CF ₂ HCH ₂ ], [RA9169; H, F, Me, Me , t-Bu, Me], [RA9170; H, F, Me, Me, t-Bu, Et], [RA9171; H, F, Me, Me, t-Bu, Pr], [RA9172; H, F , Me, Me, t-Bu, iP r], [RA9173; H, F, Me, Me, t-Bu, c-Pr], [RA9174; H, F, Me, Me, t-Bu, Bu], [RA9175; H, F, Me, Me, t-Bu, i-Bu], [RA9176; H, F, Me, Me, t-Bu, t-Bu], [RA9177; H, F, Me, Me, t-Bu, c-PrCH ₂ ], [RA9178; H, F, Me, Me, t-Bu, Ph], [RA9179; H, F, Me, Me, t-Bu, Bn], [RA9180; H, F, Me, Me, t -Bu, CF ₃ ], [RA9181; H, F, Me, Me, t-Bu, CF ₃ CH ₂ ], [RA9182; H, F, Me, Me, t-Bu, CF ₃ CF ₂ ], [ RA9183; H, F, Me, Me, t-Bu, CF ₂ H], [RA9184; H, F, Me, Me, t-Bu, CF ₂ HCH ₂ ], [RA9185; H, F, Me, Et , t-Bu, Me], [RA9186; H, F, Me, Et, t-Bu, Et], [RA9187; H, F, Me, Et, t-Bu, Pr], [RA9188; H, F , Me, Et, t-Bu, i-Pr], [RA9189; H, F, Me, Et, t-Bu, c-Pr], [RA9190; H, F, Me, Et, t-Bu, Bu ], [RA9191; H, F, Me, Et, t-Bu, i-Bu], [RA9192; H, F, Me, Et, t-Bu, t-Bu], [RA9193; H, F, Me , Et, t-Bu, c-PrCH ₂ ], [RA9194; H, F, Me, Et, t-Bu, Ph], [RA9195; H, F, Me, Et, t-Bu, Bn], [ RA9196; H, F, Me, Et, t-Bu, CF ₃ ], [RA9197; H, F, Me, Et, t-Bu, CF ₃ CH ₂ ], [RA9198; H, F, Me, Et, t-Bu, CF ₃ CF ₂ ], [RA9199; H, F, Me, Et, t-Bu, CF ₂ H], [RA9200; H, F, Me, Et, t-Bu, CF ₂ HCH ₂ ] ,

[RA9201; H, F, Me, F, t-Bu, Me], [RA9202; H, F, Me, F, t-Bu, Et], [RA9203; H, F, Me, F, t-Bu , Pr], [RA9204; H, F, Me, F, t-Bu, i-Pr], [RA9205; H, F, Me, F, t-Bu, c-Pr], [RA9206; H, F , Me, F, t-Bu, Bu], [RA9207; H, F, Me, F, t-Bu, i-Bu], [RA9208; H, F, Me, F, t-Bu, t-Bu ], [RA9209; H, F, Me, F, t-Bu, c-PrCH ₂ ], [RA9210; H, F, Me, F, t-Bu, Ph], [RA9211; H, F, Me, F, t-Bu, Bn], [RA9212; H, F, Me, F, t-Bu, CF ₃ ], [RA9213; H, F, Me, F, t-Bu, CF ₃ CH ₂ ], [ RA9214; H, F, Me, F, t-Bu, CF ₃ CF ₂ ], [RA9215; H, F, Me, F, t-Bu, CF ₂ H], [RA9216; H, F, Me, F , t-Bu, CF ₂ HCH ₂ ], [RA9217; H, F, Me, Cl, t-Bu, Me], [RA9218; H, F, Me, Cl, t-Bu, Et], [RA9219; H, F, Me, Cl, t-Bu, Pr], [RA9220; H, F, Me, Cl, t-Bu, i-Pr], [RA9221; H, F, Me, Cl, t-Bu, c-Pr], [RA9222; H, F, Me, Cl, t-Bu, Bu], [RA9223; H, F, Me, Cl, t-Bu, i-Bu], [RA9224; H, F, Me, Cl, t-Bu, t-Bu], [RA9225; H, F, Me, Cl, t-Bu, c-PrCH ₂ ], [RA9226; H, F, Me, Cl, t-Bu, Ph ], [RA9227; H, F, Me, Cl, t-Bu, Bn], [RA9228; H, F, Me, Cl, t-Bu, CF ₃ ], [RA9229; H, F, Me, Cl, t-Bu, CF ₃ CH ₂ ], [RA9230; H, F, Me, Cl, t-Bu, CF ₃ CF ₂ ], [RA9231; H, F, Me, Cl, t-Bu, CF ₂ H] , [RA9232; H, F, Me, Cl, t-Bu, CF ₂ HCH ₂ ], [RA9233; H, F, Et, H, t-Bu, Me], [RA9234; H, F, Et, H , t-Bu, Et], [RA923 5; H, F, Et, H, t-Bu, Pr], [RA9236; H, F, Et, H, t-Bu, i-Pr], [RA9237; H, F, Et, H, t- Bu, c-Pr], [RA9238; H, F, Et, H, t-Bu, Bu], [RA9239; H, F, Et, H, t-Bu, i-Bu], [RA9240; H, F, Et, H, t-Bu, t-Bu], [RA9241; H, F, Et, H, t-Bu, c-PrCH ₂ ], [RA9242; H, F, Et, H, t-Bu , Ph], [RA9243; H, F, Et, H, t-Bu, Bn], [RA9244; H, F, Et, H, t-Bu, CF ₃ ], [RA9245; H, F, Et, H, t-Bu, CF ₃ CH ₂ ], [RA9246; H, F, Et, H, t-Bu, CF ₃ CF ₂ ], [RA9247; H, F, Et, H, t-Bu, CF ₂ H], [RA9248; H, F, Et, H, t-Bu, CF ₂ HCH ₂ ], [RA9249; H, F, Et, F, t-Bu, Me], [RA9250; H, F, Et , F, t-Bu, Et], [RA9251; H, F, Et, F, t-Bu, Pr], [RA9252; H, F, Et, F, t-Bu, i-Pr], [RA9253 ; H, F, Et, F, t-Bu, c-Pr], [RA9254; H, F, Et, F, t-Bu, Bu], [RA9255; H, F, Et, F, t-Bu , i-Bu], [RA9256; H, F, Et, F, t-Bu, t-Bu], [RA9257; H, F, Et, F, t-Bu, c-PrCH ₂ ], [RA9258; H, F, Et, F, t-Bu, Ph], [RA9259; H, F, Et, F, t-Bu, Bn], [RA9260; H, F, Et, F, t-Bu, CF ₃ ], [RA9261; H, F, Et, F, t-Bu, CF ₃ CH ₂ ], [RA9262; H, F, Et, F, t-Bu, CF ₃ CF ₂ ], [RA9263; H, F , Et, F, t-Bu, CF ₂ H], [RA9264; H, F, Et, F, t-Bu, CF ₂ HCH ₂ ], [RA9265; H, F, Et, Cl, t-Bu, Me], [RA9266; H, F, Et, Cl, t-Bu, Et], [RA9267; H, F, Et, Cl, t-Bu, Pr], [RA9268; H, F, Et, Cl, t-Bu, i-Pr], [RA9269; H, F, Et, Cl, t-Bu , c-Pr], [RA9270; H, F, Et, Cl, t-Bu, Bu], [RA9271; H, F, Et, Cl, t-Bu, i-Bu], [RA9272; H, F , Et, Cl, t-Bu, t-Bu], [RA9273; H, F, Et, Cl, t-Bu, c-PrCH ₂ ], [RA9274; H, F, Et, Cl, t-Bu, Ph], [RA9275; H, F, Et, Cl, t-Bu, Bn], [RA9276; H, F, Et, Cl, t-Bu, CF ₃ ], [RA9277; H, F, Et, Cl , t-Bu, CF ₃ CH ₂ ], [RA9278; H, F, Et, Cl, t-Bu, CF ₃ CF ₂ ], [RA9279; H, F, Et, Cl, t-Bu, CF ₂ H ], [RA9280; H, F, Et, Cl, t-Bu, CF ₂ HCH ₂ ], [RA9281; H, F, F, H, t-Bu, Me], [RA9282; H, F, F, H, t-Bu, Et], [RA9283; H, F, F, H, t-Bu, Pr], [RA9284; H, F, F, H, t-Bu, i-Pr], [RA9285; H, F, F, H, t-Bu, c-Pr], [RA9286; H, F, F, H, t-Bu, Bu], [RA9287; H, F, F, H, t-Bu, i-Bu], [RA9288; H, F, F, H, t-Bu, t-Bu], [RA9289; H, F, F, H, t-Bu, c-PrCH ₂ ], [RA9290; H , F, F, H, t-Bu, Ph], [RA9291; H, F, F, H, t-Bu, Bn], [RA9292; H, F, F, H, t-Bu, CF ₃ ] , [RA9293; H, F, F, H, t-Bu, CF ₃ CH ₂ ], [RA9294; H, F, F, H, t-Bu, CF ₃ CF ₂ ], [RA9295; H, F, F, H, t-Bu, CF ₂ H], [RA9296; H, F, F, H, t-Bu, CF ₂ HCH ₂ ], [RA9297; H, F, F, F, t-Bu, Me ], [RA9298; H, F, F, F, t-Bu, Et], [RA9299; H, F, F, F, t-Bu, Pr], [RA9300; H, F, F, F, t -Bu, i-Pr], [RA9301; H, F, F, F, t-Bu, c-Pr], [RA9302; H, F, F, F, t-Bu, Bu], [RA9303; H , F, F, F, t-Bu, i-Bu], [RA9304; H, F, F, F, t-Bu, t-Bu ], [RA9305; H, F, F, F, t-Bu, c-PrCH ₂ ], [RA9306; H, F, F, F, t-Bu, Ph], [RA9307; H, F, F, F, t-Bu, Bn], [RA9308; H, F, F, F, t-Bu, CF ₃ ], [RA9309; H, F, F, F, t-Bu, CF ₃ CH ₂ ], [ RA9310; H, F, F, F, t-Bu, CF ₃ CF ₂ ], [RA9311; H, F, F, F, t-Bu, CF ₂ H], [RA9312; H, F, F, F , t-Bu, CF ₂ HCH ₂ ], [RA9313; H, F, F, Cl, t-Bu, Me], [RA9314; H, F, F, Cl, t-Bu, Et], [RA9315; H, F, F, Cl, t-Bu, Pr], [RA9316; H, F, F, Cl, t-Bu, i-Pr], [RA9317; H, F, F, Cl, t-Bu, c-Pr], [RA9318; H, F, F, Cl, t-Bu, Bu], [RA9319; H, F, F, Cl, t-Bu, i-Bu], [RA9320; H, F, F, Cl, t-Bu, t-Bu], [RA9321; H, F, F, Cl, t-Bu, c-PrCH ₂ ], [RA9322; H, F, F, Cl, t-Bu, Ph ], [RA9323; H, F, F, Cl, t-Bu, Bn], [RA9324; H, F, F, Cl, t-Bu, CF ₃ ], [RA9325; H, F, F, Cl, t-Bu, CF ₃ CH ₂ ], [RA9326; H, F, F, Cl, t-Bu, CF ₃ CF ₂ ], [RA9327; H, F, F, Cl, t-Bu, CF ₂ H] , [RA9328; H, F, F, Cl, t-Bu, CF ₂ HCH ₂ ], [RA9329; H, F, Cl, H, t-Bu, Me], [RA9330; H, F, Cl, H , t-Bu, Et], [RA9331; H, F, Cl, H, t-Bu, Pr], [RA9332; H, F, Cl, H, t-Bu, i-Pr], [RA9333; H , F, Cl, H, t-Bu, c-Pr], [RA9334; H, F, Cl, H, t-Bu, Bu], [RA9335; H, F, Cl, H, t-Bu, i -Bu], [RA9336; H, F, Cl, H, t-Bu, t-Bu], [RA9337; H, F, Cl, H, t-Bu, c-PrCH ₂ ], [RA9338; H, F, Cl, H, t-Bu, Ph], [RA9339; H, F, Cl, H, t-Bu , Bn], [RA9340; H, F, Cl, H, t-Bu, CF ₃ ], [RA9341; H, F, Cl, H, t-Bu, CF ₃ CH ₂ ], [RA9342; H, F , Cl, H, t-Bu, CF ₃ CF ₂ ], [RA9343; H, F, Cl, H, t-Bu, CF ₂ H], [RA9344; H, F, Cl, H, t-Bu, CF ₂ HCH ₂ ], [RA9345; H, F, Cl, Cl, t-Bu, Me], [RA9346; H, F, Cl, Cl, t-Bu, Et], [RA9347; H, F, Cl , Cl, t-Bu, Pr], [RA9348; H, F, Cl, Cl, t-Bu, i-Pr], [RA9349; H, F, Cl, Cl, t-Bu, c-Pr], [RA9350; H, F, Cl, Cl, t-Bu, Bu], [RA9351; H, F, Cl, Cl, t-Bu, i-Bu], [RA9352; H, F, Cl, Cl, t -Bu, t-Bu], [RA9353; H, F, Cl, Cl, t-Bu, c-PrCH ₂ ], [RA9354; H, F, Cl, Cl, t-Bu, Ph], [RA9355; H, F, Cl, Cl, t-Bu, Bn], [RA9356; H, F, Cl, Cl, t-Bu, CF ₃ ], [RA9357; H, F, Cl, Cl, t-Bu, CF ₃ CH ₂ ], [RA9358; H, F, Cl, Cl, t-Bu, CF ₃ CF ₂ ], [RA9359; H, F, Cl, Cl, t-Bu, CF ₂ H], [RA9360; H , F, Cl, Cl, t-Bu, CF ₂ HCH ₂ ], [RA9361; H, F, Me, H, CF ₂ H, Me], [RA9362; H, F, Me, H, CF ₂ H, Et], [RA9363; H, F, Me, H, CF ₂ H, Pr], [RA9364; H, F, Me, H, CF ₂ H, i-Pr], [RA9365; H, F, Me, H, CF ₂ H, c-Pr], [RA9366; H, F, Me, H, CF ₂ H, Bu], [RA9367; H, F, Me, H, CF ₂ H, i-Bu], [ RA9368; H, F, Me, H, CF ₂ H, t-Bu], [RA9369; H, F, Me, H, CF ₂ H, c-PrCH ₂ ], [RA9370; H, F, Me, H , CF ₂ H, Ph], [RA9371; H, F, Me, H, CF ₂ H, Bn], [RA9372; H, F, Me, H, CF ₂ H, CF ₃ ], [RA9373; H, F, Me, H, CF ₂ H, CF ₃ CH ₂ ], [RA9374; H, F, Me, H, CF ₂ H, CF ₃ CF ₂ ], [RA9375; H, F, Me , H, CF ₂ H, CF ₂ H], [RA9376; H, F, Me, H, CF ₂ H, CF ₂ HCH ₂ ], [RA9377; H, F, Me, Me, CF ₂ H, Me] , [RA9378; H, F, Me, Me, CF ₂ H, Et], [RA9379; H, F, Me, Me, CF ₂ H, Pr], [RA9380; H, F, Me, Me, CF ₂ H, i-Pr], [RA9381; H, F, Me, Me, CF ₂ H, c-Pr], [RA9382; H, F, Me, Me, CF ₂ H, Bu], [RA9383; H, F, Me, Me, CF ₂ H, i-Bu], [RA9384; H, F, Me, Me, CF ₂ H, t-Bu], [RA9385; H, F, Me, Me, CF ₂ H, c-PrCH ₂ ], [RA9386; H, F, Me, Me, CF ₂ H, Ph], [RA9387; H, F, Me, Me, CF ₂ H, Bn], [RA9388; H, F, Me , Me, CF ₂ H, CF ₃ ], [RA9389; H, F, Me, Me, CF ₂ H, CF ₃ CH ₂ ], [RA9390; H, F, Me, Me, CF ₂ H, CF ₃ CF ₂ ], [RA9391; H, F, Me, Me, CF ₂ H, CF ₂ H], [RA9392; H, F, Me, Me, CF ₂ H, CF ₂ HCH ₂ ], [RA9393; H, F , Me, Et, CF ₂ H, Me], [RA9394; H, F, Me, Et, CF ₂ H, Et], [RA9395; H, F, Me, Et, CF ₂ H, Pr], [RA9396 ; H, F, Me, Et, CF ₂ H, i-Pr], [RA9397; H, F, Me, Et, CF ₂ H, c-Pr], [RA9398; H, F, Me, Et, CF ₂ H, Bu], [RA9399; H, F, Me, Et, CF ₂ H, i-Bu], [RA9400; H, F, Me, Et, CF ₂ H, t-Bu],

[RA9401; H, F, Me, Et, CF ₂ H, c-PrCH ₂ ], [RA9402; H, F, Me, Et, CF ₂ H, Ph], [RA9403; H, F, Me, Et, CF ₂ H, Bn], [RA9404; H, F, Me, Et, CF ₂ H, CF ₃ ], [RA9405; H, F, Me, Et, CF ₂ H, CF ₃ CH ₂ ], [RA9406; H, F, Me, Et, CF ₂ H, CF ₃ CF ₂ ], [RA9407; H, F, Me, Et, CF ₂ H, CF ₂ H], [RA9408; H, F, Me, Et, CF ₂ H, CF ₂ HCH ₂ ], [RA9409; H, F, Me, F, CF ₂ H, Me], [RA9410; H, F, Me, F, CF ₂ H, Et], [RA9411; H, F, Me, F, CF ₂ H, Pr], [RA9412; H, F, Me, F, CF ₂ H, i-Pr], [RA9413; H, F, Me, F, CF ₂ H, c- Pr], [RA9414; H, F, Me, F, CF ₂ H, Bu], [RA9415; H, F, Me, F, CF ₂ H, i-Bu], [RA9416; H, F, Me, F, CF ₂ H, t-Bu], [RA9417; H, F, Me, F, CF ₂ H, c-PrCH ₂ ], [RA9418; H, F, Me, F, CF ₂ H, Ph], [RA9419; H, F, Me, F, CF ₂ H, Bn], [RA9420; H, F, Me, F, CF ₂ H, CF ₃ ], [RA9421; H, F, Me, F, CF ₂ H, CF ₃ CH ₂ ], [RA9422; H, F, Me, F, CF ₂ H, CF ₃ CF ₂ ], [RA9423; H, F, Me, F, CF ₂ H, CF ₂ H], [ RA9424; H, F, Me, F, CF ₂ H, CF ₂ HCH ₂ ], [RA9425; H, F, Me, Cl, CF ₂ H, Me], [RA9426; H, F, Me, Cl, CF ₂ H, Et], [RA9427; H, F, Me, Cl, CF ₂ H, Pr], [RA9428; H, F, Me, Cl, CF ₂ H, i-Pr], [RA9429; H, F , Me, Cl, CF ₂ H, c-Pr], [RA9430; H, F, Me, Cl, CF ₂ H, Bu], [RA9431; H, F, Me, Cl, CF ₂ H, i-Bu ], [RA9432; H, F, Me, Cl, CF ₂ H, t-Bu], [RA9433; H, F, Me, Cl, CF ₂ H, c-PrCH ₂ ], [RA9434; H, F, Me, Cl, CF ₂ H, Ph], [RA9435; H, F , Me, Cl, CF ₂ H, Bn], [RA9436; H, F, Me, Cl, CF ₂ H, CF ₃ ], [RA9437; H, F, Me, Cl, CF ₂ H, CF ₃ CH ₂ ], [RA9438; H, F, Me, Cl, CF ₂ H, CF ₃ CF ₂ ], [RA9439; H, F, Me, Cl, CF ₂ H, CF ₂ H], [RA9440; H, F, Me, Cl, CF ₂ H, CF ₂ HCH ₂ ], [RA9441; H, F, Et, H, CF ₂ H, Me], [RA9442; H, F, Et, H, CF ₂ H, Et], [RA9443; H, F, Et, H, CF ₂ H, Pr], [RA9444; H, F, Et, H, CF ₂ H, i-Pr], [RA9445; H, F, Et, H, CF ₂ H, c-Pr], [RA9446; H, F, Et, H, CF ₂ H, Bu], [RA9447; H, F, Et, H, CF ₂ H, i-Bu], [RA9448; H , F, Et, H, CF ₂ H, t-Bu], [RA9449; H, F, Et, H, CF ₂ H, c-PrCH ₂ ], [RA9450; H, F, Et, H, CF ₂ H, Ph], [RA9451; H, F, Et, H, CF ₂ H, Bn], [RA9452; H, F, Et, H, CF ₂ H, CF ₃ ], [RA9453; H, F, Et , H, CF ₂ H, CF ₃ CH ₂ ], [RA9454; H, F, Et, H, CF ₂ H, CF ₃ CF ₂ ], [RA9455; H, F, Et, H, CF ₂ H, CF ₂ H], [RA9456; H, F, Et, H, CF ₂ H, CF ₂ HCH ₂ ], [RA9457; H, F, Et, F, CF ₂ H, Me], [RA9458; H, F, Et, F, CF ₂ H, Et], [RA9459; H, F, Et, F, CF ₂ H, Pr], [RA9460; H, F, Et, F, CF ₂ H, i-Pr], [ RA9461; H, F, Et, F, CF ₂ H, c-Pr], [RA9462; H, F, Et, F, CF ₂ H, Bu], [RA9463; H, F, Et, F, CF ₂ H, i-Bu], [RA9464; H, F, Et, F, CF ₂ H, t- Bu], [RA9465; H, F, Et, F, CF ₂ H, c-PrCH ₂ ], [RA9466; H, F, Et, F, CF ₂ H, Ph], [RA9467; H, F, Et , F, CF ₂ H, Bn], [RA9468; H, F, Et, F, CF ₂ H, CF ₃ ], [RA9469; H, F, Et, F, CF ₂ H, CF ₃ CH ₂ ], [RA9470; H, F, Et, F, CF ₂ H, CF ₃ CF ₂ ], [RA9471; H, F, Et, F, CF ₂ H, CF ₂ H], [RA9472; H, F, Et, F, CF ₂ H, CF ₂ HCH ₂ ], [RA9473; H, F, Et, Cl, CF ₂ H, Me], [RA9474; H, F, Et, Cl, CF ₂ H, Et], [RA9475 ; H, F, Et, Cl, CF ₂ H, Pr], [RA9476; H, F, Et, Cl, CF ₂ H, i-Pr], [RA9477; H, F, Et, Cl, CF ₂ H , c-Pr], [RA9478; H, F, Et, Cl, CF ₂ H, Bu], [RA9479; H, F, Et, Cl, CF ₂ H, i-Bu], [RA9480; H, F , Et, Cl, CF ₂ H, t-Bu], [RA9481; H, F, Et, Cl, CF ₂ H, c-PrCH ₂ ], [RA9482; H, F, Et, Cl, CF ₂ H, Ph], [RA9483; H, F, Et, Cl, CF ₂ H, Bn], [RA9484; H, F, Et, Cl, CF ₂ H, CF ₃ ], [RA9485; H, F, Et, Cl , CF ₂ H, CF ₃ CH ₂ ], [RA9486; H, F, Et, Cl, CF ₂ H, CF ₃ CF ₂ ], [RA9487; H, F, Et, Cl, CF ₂ H, CF ₂ H ], [RA9488; H, F, Et, Cl, CF ₂ H, CF ₂ HCH ₂ ], [RA9489; H, F, F, H, CF ₂ H, Me], [RA9490; H, F, F, H, CF ₂ H, Et], [RA9491; H, F, F, H, CF ₂ H, Pr], [RA9492; H, F, F, H, CF ₂ H, i-Pr], [RA9493; H, F, F, H, CF ₂ H, c-Pr], [RA9494; H, F, F, H, CF ₂ H, Bu], [RA9495; H, F, F, H, CF ₂ H, i-Bu], [RA9496; H, F, F, H, CF ₂ H, t-Bu ], [RA9497; H, F, F, H, CF ₂ H, c-PrCH ₂ ], [RA9498; H, F, F, H, CF ₂ H, Ph], [RA9499; H, F, F, H, CF ₂ H, Bn], [RA9500; H, F, F, H, CF ₂ H, CF ₃ ], [RA9501; H, F, F, H, CF ₂ H, CF ₃ CH ₂ ], [ RA9502; H, F, F, H, CF ₂ H, CF ₃ CF ₂ ], [RA9503; H, F, F, H, CF ₂ H, CF ₂ H], [RA9504; H, F, F, H , CF ₂ H, CF ₂ HCH ₂ ], [RA9505; H, F, F, F, CF ₂ H, Me], [RA9506; H, F, F, F, CF ₂ H, Et], [RA9507; H, F, F, F, CF ₂ H, Pr], [RA9508; H, F, F, F, CF ₂ H, i-Pr], [RA9509; H, F, F, F, CF ₂ H, c-Pr], [RA9510; H, F, F, F, CF ₂ H, Bu], [RA9511; H, F, F, F, CF ₂ H, i-Bu], [RA9512; H, F, F, F, CF ₂ H, t-Bu], [RA9513; H, F, F, F, CF ₂ H, c-PrCH ₂ ], [RA9514; H, F, F, F, CF ₂ H, Ph ], [RA9515; H, F, F, F, CF ₂ H, Bn], [RA9516; H, F, F, F, CF ₂ H, CF ₃ ], [RA9517; H, F, F, F, CF ₂ H, CF ₃ CH ₂ ], [RA9518; H, F, F, F, CF ₂ H, CF ₃ CF ₂ ], [RA9519; H, F, F, F, CF ₂ H, CF ₂ H] , [RA9520; H, F, F, F, CF ₂ H, CF ₂ HCH ₂ ], [RA9521; H, F, F, Cl, CF ₂ H, Me], [RA9522; H, F, F, Cl , CF ₂ H, Et], [RA9523; H, F, F, Cl, CF ₂ H, Pr], [RA9524; H, F, F, Cl, CF ₂ H, i-Pr], [RA9525; H , F, F, Cl, CF ₂ H, c-Pr], [RA9526; H, F, F, Cl, CF ₂ H, Bu], [RA9527; H, F, F, Cl, CF ₂ H, i -Bu], [RA9528; H, F, F, Cl, CF ₂ H, t-Bu], [RA9529; H, F, F, Cl, CF ₂ H, c-PrCH ₂ ], [RA9530; H, F, F, Cl, CF ₂ H, Ph], [RA9531; H, F, F, Cl, CF ₂ H, Bn], [RA9532; H, F, F, Cl, CF ₂ H, CF ₃ ], [RA9533; H, F, F, Cl, CF ₂ H, CF ₃ CH ₂ ], [RA9534; H, F, F, Cl, CF ₂ H, CF ₃ CF ₂ ], [ RA9535; H, F, F, Cl, CF ₂ H, CF ₂ H], [RA9536; H, F, F, Cl, CF ₂ H, CF ₂ HCH ₂ ], [RA9537; H, F, Cl, H , CF ₂ H, Me], [RA9538; H, F, Cl, H, CF ₂ H, Et], [RA9539; H, F, Cl, H, CF ₂ H, Pr], [RA9540; H, F , Cl, H, CF ₂ H, i-Pr], [RA9541; H, F, Cl, H, CF ₂ H, c-Pr], [RA9542; H, F, Cl, H, CF ₂ H, Bu ], [RA9543; H, F, Cl, H, CF ₂ H, i-Bu], [RA9544; H, F, Cl, H, CF ₂ H, t-Bu], [RA9545; H, F, Cl , H, CF ₂ H, c-PrCH ₂ ], [RA9546; H, F, Cl, H, CF ₂ H, Ph], [RA9547; H, F, Cl, H, CF ₂ H, Bn], [ RA9548; H, F, Cl, H, CF ₂ H, CF ₃ ], [RA9549; H, F, Cl, H, CF ₂ H, CF ₃ CH ₂ ], [RA9550; H, F, Cl, H, CF ₂ H, CF ₃ CF ₂ ], [RA9551; H, F, Cl, H, CF ₂ H, CF ₂ H], [RA9552; H, F, Cl, H, CF ₂ H, CF ₂ HCH ₂ ] , [RA9553; H, F, Cl, Cl, CF ₂ H, Me], [RA9554; H, F, Cl, Cl, CF ₂ H, Et], [RA9555; H, F, Cl, Cl, CF ₂ H, Pr], [RA9556; H, F, Cl, Cl, CF ₂ H, i-Pr], [RA9557; H, F, Cl, Cl, CF ₂ H, c-Pr], [RA9558; H, F, Cl, Cl, CF ₂ H, Bu], [RA9559; H, F, Cl, Cl, CF ₂ H, i-Bu], [RA9560; H, F, Cl, Cl, CF ₂ H, t- Bu], [RA9561; H, F, Cl, Cl, CF ₂ H, c-PrCH ₂ ], [RA9562; H, F, Cl, Cl, CF ₂ H, Ph], [RA9563; H, F, Cl, Cl, CF ₂ H, Bn], [RA9564; H, F, Cl, Cl, CF ₂ H, CF ₃ ], [RA9565; H, F, Cl, Cl, CF ₂ H, CF ₃ CH ₂ ], [RA9566; H, F, Cl, Cl, CF ₂ H, CF ₃ CF ₂ ], [ RA9567; H, F, Cl, Cl, CF ₂ H, CF ₂ H], [RA9568; H, F, Cl, Cl, CF ₂ H, CF ₂ HCH ₂ ], [RA9569; H, F, Me, H , CF ₃ , Me], [RA9570; H, F, Me, H, CF ₃ , Et], [RA9571; H, F, Me, H, CF ₃ , Pr], [RA9572; H, F, Me, H, CF ₃ , i-Pr], [RA9573; H, F, Me, H, CF ₃ , c-Pr], [RA9574; H, F, Me, H, CF ₃ , Bu], [RA9575; H , F, Me, H, CF ₃ , i-Bu], [RA9576; H, F, Me, H, CF ₃ , t-Bu], [RA9577; H, F, Me, H, CF ₃ , c- PrCH ₂ ], [RA9578; H, F, Me, H, CF ₃ , Ph], [RA9579; H, F, Me, H, CF ₃ , Bn], [RA9580; H, F, Me, H, CF ₃ , CF ₃ ], [RA9581; H, F, Me, H, CF ₃ , CF ₃ CH ₂ ], [RA9582; H, F, Me, H, CF ₃ , CF ₃ CF ₂ ], [RA9583; H , F, Me, H, CF ₃ , CF ₂ H], [RA9584; H, F, Me, H, CF ₃ , CF ₂ HCH ₂ ], [RA9585; H, F, Me, Me, CF ₃ , Me ], [RA9586; H, F, Me, Me, CF ₃ , Et], [RA9587; H, F, Me, Me, CF ₃ , Pr], [RA9588; H, F, Me, Me, CF ₃ , i-Pr], [RA9589; H, F, Me, Me, CF ₃ , c-Pr], [RA9590; H, F, Me, Me, CF ₃ , Bu], [RA9591; H, F, Me, Me, CF ₃ , i-Bu], [RA9592; H, F, Me, Me, CF ₃ , t-Bu], [RA9593; H, F, Me, Me, CF ₃ , c-PrCH ₂ ], [ RA9594; H, F, Me, Me , CF ₃ , Ph], [RA9595; H, F, Me, Me, CF ₃ , Bn], [RA9596; H, F, Me, Me, CF ₃ , CF ₃ ], [RA9597; H, F, Me , Me, CF ₃ , CF ₃ CH ₂ ], [RA9598; H, F, Me, Me, CF ₃ , CF ₃ CF ₂ ], [RA9599; H, F, Me, Me, CF ₃ , CF ₂ H] , [RA9600; H, F, Me, Me, CF ₃ , CF ₂ HCH ₂ ],

[RA9601; H, F, Me, Et, CF ₃ , Me], [RA9602; H, F, Me, Et, CF ₃ , Et], [RA9603; H, F, Me, Et, CF ₃ , Pr] , [RA9604; H, F, Me, Et, CF ₃ , i-Pr], [RA9605; H, F, Me, Et, CF ₃ , c-Pr], [RA9606; H, F, Me, Et, CF ₃ , Bu], [RA9607; H, F, Me, Et, CF ₃ , i-Bu], [RA9608; H, F, Me, Et, CF ₃ , t-Bu], [RA9609; H, F , Me, Et, CF ₃ , c-PrCH ₂ ], [RA9610; H, F, Me, Et, CF ₃ , Ph], [RA9611; H, F, Me, Et, CF ₃ , Bn], [RA9612 ; H, F, Me, Et, CF ₃ , CF ₃ ], [RA9613; H, F, Me, Et, CF ₃ , CF ₃ CH ₂ ], [RA9614; H, F, Me, Et, CF ₃ , CF ₃ CF ₂ ], [RA9615; H, F, Me, Et, CF ₃ , CF ₂ H], [RA9616; H, F, Me, Et, CF ₃ , CF ₂ HCH ₂ ], [RA9617; H, F, Me, F, CF ₃ , Me], [RA9618; H, F, Me, F, CF ₃ , Et], [RA9619; H, F, Me, F, CF ₃ , Pr], [RA9620; H , F, Me, F, CF ₃ , i-Pr], [RA9621; H, F, Me, F, CF ₃ , c-Pr], [RA9622; H, F, Me, F, CF ₃ , Bu] , [RA9623; H, F, Me, F, CF ₃ , i-Bu], [RA9624; H, F, Me, F, CF ₃ , t-Bu], [RA9625; H, F, Me, F, CF ₃ , c-PrCH ₂ ], [RA9626; H, F, Me, F, CF ₃ , Ph], [RA9627; H, F, Me, F, CF ₃ , Bn], [RA9628; H, F, Me, F, CF ₃ , CF ₃ ], [RA9629; H, F, Me, F, CF ₃ , CF ₃ CH ₂ ], [RA9630; H, F, Me, F, CF ₃ , CF ₃ CF ₂ ] , [RA9631; H, F, Me, F, CF ₃ , CF ₂ H], [RA9632; H, F, Me, F, CF ₃ , CF ₂ HCH ₂ ], [RA9633; H, F, Me, Cl , CF ₃ , Me ], [RA9634; H, F, Me, Cl, CF ₃ , Et], [RA9635; H, F, Me, Cl, CF ₃ , Pr], [RA9636; H, F, Me, Cl, CF ₃ , i-Pr], [RA9637; H, F, Me, Cl, CF ₃ , c-Pr], [RA9638; H, F, Me, Cl, CF ₃ , Bu], [RA9639; H, F, Me, Cl, CF ₃ , i-Bu], [RA9640; H, F, Me, Cl, CF ₃ , t-Bu], [RA9641; H, F, Me, Cl, CF ₃ , c-PrCH ₂ ], [ RA9642; H, F, Me, Cl, CF ₃ , Ph], [RA9643; H, F, Me, Cl, CF ₃ , Bn], [RA9644; H, F, Me, Cl, CF ₃ , CF ₃ ] , [RA9645; H, F, Me, Cl, CF ₃ , CF ₃ CH ₂ ], [RA9646; H, F, Me, Cl, CF ₃ , CF ₃ CF ₂ ], [RA9647; H, F, Me, Cl, CF ₃ , CF ₂ H], [RA9648; H, F, Me, Cl, CF ₃ , CF ₂ HCH ₂ ], [RA9649; H, F, Et, H, CF ₃ , Me], [RA9650; H, F, Et, H, CF ₃ , Et], [RA9651; H, F, Et, H, CF ₃ , Pr], [RA9652; H, F, Et, H, CF ₃ , i-Pr], [RA9653; H, F, Et, H, CF ₃ , c-Pr], [RA9654; H, F, Et, H, CF ₃ , Bu], [RA9655; H, F, Et, H, CF ₃ , i-Bu], [RA9656; H, F, Et, H, CF ₃ , t-Bu], [RA9657; H, F, Et, H, CF ₃ , c-PrCH ₂ ], [RA9658; H, F , Et, H, CF ₃ , Ph], [RA9659; H, F, Et, H, CF ₃ , Bn], [RA9660; H, F, Et, H, CF ₃ , CF ₃ ], [RA9661; H , F, Et, H, CF ₃ , CF ₃ CH ₂ ], [RA9662; H, F, Et, H, CF ₃ , CF ₃ CF ₂ ], [RA9663; H, F, Et, H, CF ₃ , CF ₂ H], [RA9664; H, F, Et, H, CF ₃ , CF ₂ HCH ₂ ], [RA9665; H, F, Et, F, CF ₃ , Me], [RA9666; H, F, Et , F, CF ₃ , Et ], [RA9667; H, F, Et, F, CF ₃ , Pr], [RA9668; H, F, Et, F, CF ₃ , i-Pr], [RA9669; H, F, Et, F, CF ₃ , c-Pr], [RA9670; H, F, Et, F, CF ₃ , Bu], [RA9671; H, F, Et, F, CF ₃ , i-Bu], [RA9672; H, F, Et, F, CF ₃ , t-Bu], [RA9673; H, F, Et, F, CF ₃ , c-PrCH ₂ ], [RA9674; H, F, Et, F, CF ₃ , Ph], [ RA9675; H, F, Et, F, CF ₃ , Bn], [RA9676; H, F, Et, F, CF ₃ , CF ₃ ], [RA9677; H, F, Et, F, CF ₃ , CF ₃ CH ₂ ], [RA9678; H, F, Et, F, CF ₃ , CF ₃ CF ₂ ], [RA9679; H, F, Et, F, CF ₃ , CF ₂ H], [RA9680; H, F, Et, F, CF ₃ , CF ₂ HCH ₂ ], [RA9681; H, F, Et, Cl, CF ₃ , Me], [RA9682; H, F, Et, Cl, CF ₃ , Et], [RA9683; H, F, Et, Cl, CF ₃ , Pr], [RA9684; H, F, Et, Cl, CF ₃ , i-Pr], [RA9685; H, F, Et, Cl, CF ₃ , c-Pr ], [RA9686; H, F, Et, Cl, CF ₃ , Bu], [RA9687; H, F, Et, Cl, CF ₃ , i-Bu], [RA9688; H, F, Et, Cl, CF ₃ , t-Bu], [RA9689; H, F, Et, Cl, CF ₃ , c-PrCH ₂ ], [RA9690; H, F, Et, Cl, CF ₃ , Ph], [RA9691; H, F , Et, Cl, CF ₃ , Bn], [RA9692; H, F, Et, Cl, CF ₃ , CF ₃ ], [RA9693; H, F, Et, Cl, CF ₃ , CF ₃ CH ₂ ], [ RA9694; H, F, Et, Cl, CF ₃ , CF ₃ CF ₂ ], [RA9695; H, F, Et, Cl, CF ₃ , CF ₂ H], [RA9696; H, F, Et, Cl, CF ₃ , CF ₂ HCH ₂ ], [RA9697; H, F, F, H, CF ₃ , Me], [RA9698; H, F, F, H, CF ₃ , Et], [RA9699; H, F, F , H, CF ₃ , Pr], [RA9700; H, F, F, H, CF ₃ , i-Pr], [RA9701; H, F, F, H, CF ₃ , c-Pr], [RA9702; H, F, F, H, CF ₃ , Bu], [RA9703; H, F, F, H, CF ₃ , i-Bu], [RA9704; H, F, F, H, CF ₃ , t-Bu], [RA9705; H, F, F, H, CF ₃ , c-PrCH ₂ ], [RA9706; H, F, F, H, CF ₃ , Ph], [RA9707; H, F, F, H, CF ₃ , Bn], [RA9708; H, F, F, H, CF ₃ , CF ₃ ], [RA9709; H, F, F, H, CF ₃ , CF ₃ CH ₂ ], [RA9710; H, F, F, H, CF ₃ , CF ₃ CF ₂ ], [RA9711; H, F, F, H, CF ₃ , CF ₂ H], [RA9712; H, F, F, H, CF ₃ , CF ₂ HCH ₂ ], [RA9713; H, F , F, F, CF ₃ , Me], [RA9714; H, F, F, F, CF ₃ , Et], [RA9715; H, F, F, F, CF ₃ , Pr], [RA9716; H, F, F, F, CF ₃ , i-Pr], [RA9717; H, F, F, F, CF ₃ , c-Pr], [RA9718; H, F, F, F, CF ₃ , Bu], [RA9719; H, F, F, F, CF ₃ , i-Bu], [RA9720; H, F, F, F, CF ₃ , t-Bu], [RA9721; H, F, F, F, CF ₃ , c-PrCH ₂ ], [RA9722; H, F, F, F, CF ₃ , Ph], [RA9723; H, F, F, F, CF ₃ , Bn], [RA9724; H, F, F , F, CF ₃ , CF ₃ ], [RA9725; H, F, F, F, CF ₃ , CF ₃ CH ₂ ], [RA9726; H, F, F, F, CF ₃ , CF ₃ CF ₂ ], [RA9727; H, F, F, F, CF ₃ , CF ₂ H], [RA9728; H, F, F, F, CF ₃ , CF ₂ HCH ₂ ], [RA9729; H, F, F, Cl, CF ₃ , Me], [RA9730; H, F, F, Cl, CF ₃ , Et], [RA9731; H, F, F, Cl, CF ₃ , Pr], [RA9732; H, F, F, Cl , CF ₃ , i-Pr], [RA9733; H, F, F, Cl, CF ₃ , c-Pr], [RA9734; H, F, F , Cl, CF ₃ , Bu], [RA9735; H, F, F, Cl, CF ₃ , i-Bu], [RA9736; H, F, F, Cl, CF ₃ , t-Bu], [RA9737; H, F, F, Cl, CF ₃ , c-PrCH ₂ ], [RA9738; H, F, F, Cl, CF ₃ , Ph], [RA9739; H, F, F, Cl, CF ₃ , Bn] , [RA9740; H, F, F, Cl, CF ₃ , CF ₃ ], [RA9741; H, F, F, Cl, CF ₃ , CF ₃ CH ₂ ], [RA9742; H, F, F, Cl, CF ₃ , CF ₃ CF ₂ ], [RA9743; H, F, F, Cl, CF ₃ , CF ₂ H], [RA9744; H, F, F, Cl, CF ₃ , CF ₂ HCH ₂ ], [RA9745 ; H, F, Cl, H, CF ₃ , Me], [RA9746; H, F, Cl, H, CF ₃ , Et], [RA9747; H, F, Cl, H, CF ₃ , Pr], [ RA9748; H, F, Cl, H, CF ₃ , i-Pr], [RA9749; H, F, Cl, H, CF ₃ , c-Pr], [RA9750; H, F, Cl, H, CF ₃ , Bu], [RA9751; H, F, Cl, H, CF ₃ , i-Bu], [RA9752; H, F, Cl, H, CF ₃ , t-Bu], [RA9753; H, F, Cl , H, CF ₃ , c-PrCH ₂ ], [RA9754; H, F, Cl, H, CF ₃ , Ph], [RA9755; H, F, Cl, H, CF ₃ , Bn], [RA9756; H , F, Cl, H, CF ₃ , CF ₃ ], [RA9757; H, F, Cl, H, CF ₃ , CF ₃ CH ₂ ], [RA9758; H, F, Cl, H, CF ₃ , CF ₃ CF ₂ ], [RA9759; H, F, Cl, H, CF ₃ , CF ₂ H], [RA9760; H, F, Cl, H, CF ₃ , CF ₂ HCH ₂ ], [RA9761; H, F, Cl, Cl, CF ₃ , Me], [RA9762; H, F, Cl, Cl, CF ₃ , Et], [RA9763; H, F, Cl, Cl, CF ₃ , Pr], [RA9764; H, F , Cl, Cl, CF ₃ , i-Pr], [RA9765; H, F, Cl, Cl, CF ₃ , c-Pr], [RA9766; H, F, Cl, Cl, CF ₃ , Bu], [ RA9767; H, F, Cl, Cl, CF ₃ , i-Bu], [RA9768; H, F, Cl, Cl, CF ₃ , t-Bu], [RA9769; H, F, Cl, Cl, CF ₃ , c-PrCH ₂ ], [RA9770; H, F, Cl, Cl, CF ₃ , Ph], [RA9771; H, F, Cl, Cl, CF ₃ , Bn], [RA9772; H, F, Cl, Cl, CF ₃ , CF ₃ ], [RA9773; H, F, Cl, Cl, CF ₃ , CF ₃ CH ₂ ], [RA9774; H, F, Cl, Cl, CF ₃ , CF ₃ CF ₂ ], [RA9775; H, F, Cl, Cl, CF ₃ , CF ₂ H], [RA9776; H, F, Cl, Cl, CF ₃ , CF ₂ HCH ₂ ], [RA9777; H, F, Me, H, CF ₂ HCH ₂ , Me], [RA9778; H, F, Me, H, CF ₂ HCH ₂ , Et], [RA9779; H, F, Me, H, CF ₂ HCH ₂ , Pr], [RA9780; H, F, Me, H, CF ₂ HCH ₂ , i -Pr], [RA9781; H, F, Me, H, CF ₂ HCH ₂ , c-Pr], [RA9782; H, F, Me, H, CF ₂ HCH ₂ , Bu], [RA9783; H, F , Me, H, CF ₂ HCH ₂ , i-Bu], [RA9784; H, F, Me, H, CF ₂ HCH ₂ , t-Bu], [RA9785; H, F, Me, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA9786; H, F, Me, H, CF ₂ HCH ₂ , Ph], [RA9787; H, F, Me, H, CF ₂ HCH ₂ , Bn], [RA9788; H , F, Me, H, CF ₂ HCH ₂ , CF ₃ ], [RA9789; H, F, Me, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA9790; H, F, Me, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA9791; H, F, Me, H, CF ₂ HCH ₂ , CF ₂ H], [RA9792; H, F, Me, H, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA9793; H, F, Me, Me, CF ₂ HCH ₂ , Me], [RA9794; H, F, Me, Me, CF ₂ HCH ₂ , Et], [RA9795; H, F, Me, Me, CF ₂ HCH ₂ , Pr], [RA9796; H, F, Me, Me, CF ₂ HCH ₂ , i-Pr], [RA9797; H, F, Me, Me, CF ₂ HCH ₂ , c-Pr], [RA9798; H, F, Me, Me, CF ₂ HCH ₂ , Bu], [RA9799 ; H, F, Me, Me, CF ₂ HCH ₂ , i-Bu], [RA9800; H, F, Me, Me, CF ₂ HCH ₂ , t-Bu],

[RA9801; H, F, Me, Me, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA9802; H, F, Me, Me, CF ₂ HCH ₂ , Ph], [RA9803; H, F, Me, Me, CF ₂ HCH ₂ , Bn], [RA9804; H, F, Me, Me, CF ₂ HCH ₂ , CF ₃ ], [RA9805; H, F, Me, Me, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA9806; H, F, Me, Me, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA9807; H, F, Me, Me, CF ₂ HCH ₂ , CF ₂ H], [RA9808; H, F, Me, Me, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA9809; H, F, Me, Et, CF ₂ HCH ₂ , Me], [RA9810; H, F, Me, Et, CF ₂ HCH ₂ , Et], [RA9811; H, F, Me, Et, CF ₂ HCH ₂ , Pr], [RA9812; H, F, Me, Et, CF ₂ HCH ₂ , i-Pr], [RA9813; H, F, Me, Et, CF ₂ HCH ₂ , c-Pr], [RA9814; H, F, Me, Et, CF ₂ HCH ₂ , Bu], [RA9815; H, F, Me, Et, CF ₂ HCH ₂ , i-Bu], [RA9816; H, F, Me, Et, CF ₂ HCH ₂ , t-Bu], [RA9817; H, F, Me, Et, CF ₂ HCH ₂ , c-PrCH ₂ ], [ RA9818; H, F, Me, Et, CF ₂ HCH ₂ , Ph], [RA9819; H, F, Me, Et, CF ₂ HCH ₂ , Bn], [RA9820; H, F, Me, Et, CF ₂ HCH ₂ , CF ₃ ], [RA9821; H, F, Me, Et, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA9822; H, F, Me, Et, CF ₂ HCH ₂ , CF ₃ CF ₂ ] , [RA9823; H, F, Me, Et, CF ₂ HCH ₂ , CF ₂ H], [RA9824; H, F, Me, Et, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA9825; H, F , Me, F, CF ₂ HCH ₂ , Me], [RA9826; H, F, Me, F, CF ₂ HCH ₂ , Et], [RA9827; H, F, Me, F, CF ₂ HCH ₂ , Pr] , [RA9828; H, F, Me, F, CF ₂ HCH ₂ , i-Pr], [RA9829; H, F, Me, F, CF ₂ HCH ₂ , c-Pr], [RA9830; H, F, Me, F, CF ₂ HCH ₂ , Bu], [RA9831; H, F, Me, F, CF ₂ HCH ₂ , i-Bu], [RA9832; H, F, Me, F, CF ₂ HCH ₂ , t -Bu], [RA9833; H, F, Me, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA9834; H, F, Me, F, CF ₂ HCH ₂ , Ph], [RA9835; H, F, Me, F, CF ₂ HCH ₂ , Bn], [RA9836; H, F, Me, F, CF ₂ HCH ₂ , CF ₃ ], [RA9837; H, F, Me, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA9838; H, F, Me, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA9839; H, F, Me, F, CF ₂ HCH ₂ , CF ₂ H], [ RA9840; H, F, Me, F, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA9841; H, F, Me, Cl, CF ₂ HCH ₂ , Me], [RA9842; H, F, Me, Cl , CF ₂ HCH ₂ , Et], [RA9843; H, F, Me, Cl, CF ₂ HCH ₂ , Pr], [RA9844; H, F, Me, Cl, CF ₂ HCH ₂ , i-Pr], [ RA9845; H, F, Me, Cl, CF ₂ HCH ₂ , c-Pr], [RA9846; H, F, Me, Cl, CF ₂ HCH ₂ , Bu], [RA9847; H, F, Me, Cl, CF ₂ HCH ₂ , i-Bu], [RA9848; H, F, Me, Cl, CF ₂ HCH ₂ , t-Bu], [RA9849; H, F, Me, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA9850; H, F, Me, Cl, CF ₂ HCH ₂ , Ph], [RA9851; H, F, Me, Cl, CF ₂ HCH ₂ , Bn], [RA9852; H, F, Me, Cl, CF ₂ HCH ₂ , CF ₃ ], [RA9853; H, F, Me, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA9854; H, F, Me, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA9855; H, F, M e, Cl, CF ₂ HCH ₂ , CF ₂ H], [RA9856; H, F, Me, Cl, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA9857; H, F, Et, H, CF ₂ HCH ₂ , Me], [RA9858; H, F, Et, H, CF ₂ HCH ₂ , Et], [RA9859; H, F, Et, H, CF ₂ HCH ₂ , Pr], [RA9860; H, F, Et, H, CF ₂ HCH ₂ , i-Pr], [RA9861; H, F, Et, H, CF ₂ HCH ₂ , c-Pr], [RA9862; H, F, Et, H, CF ₂ HCH ₂ , Bu], [RA9863; H, F, Et, H, CF ₂ HCH ₂ , i-Bu], [RA9864; H, F, Et, H, CF ₂ HCH ₂ , t-Bu], [RA9865; H , F, Et, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA9866; H, F, Et, H, CF ₂ HCH ₂ , Ph], [RA9867; H, F, Et, H, CF ₂ HCH ₂ , Bn], [RA9868; H, F, Et, H, CF ₂ HCH ₂ , CF ₃ ], [RA9869; H, F, Et, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA9870 ; H, F, Et, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA9871; H, F, Et, H, CF ₂ HCH ₂ , CF ₂ H], [RA9872; H, F, Et, H, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA9873; H, F, Et, F, CF ₂ HCH ₂ , Me], [RA9874; H, F, Et, F, CF ₂ HCH ₂ , Et] , [RA9875; H, F, Et, F, CF ₂ HCH ₂ , Pr], [RA9876; H, F, Et, F, CF ₂ HCH ₂ , i-Pr], [RA9877; H, F, Et, F, CF ₂ HCH ₂ , c-Pr], [RA9878; H, F, Et, F, CF ₂ HCH ₂ , Bu], [RA9879; H, F, Et, F, CF ₂ HCH ₂ , i-Bu ], [RA9880; H, F, Et, F, CF ₂ HCH ₂ , t-Bu], [RA9881; H, F, Et, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA9882; H, F, Et, F, CF ₂ HCH ₂ , Ph], [RA9883; H, F, Et, F, CF ₂ HCH ₂ , Bn], [RA9884; H, F, Et, F, CF ₂ HCH ₂ , CF ₃ ], [RA9885; H, F, Et, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA9886; H, F, Et, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA9887; H, F, Et, F, CF ₂ HCH ₂ , CF ₂ H], [RA9888; H, F, Et, F, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA9889; H, F, Et, Cl, CF ₂ HCH ₂ , Me], [RA9890; H, F, Et, Cl, CF ₂ HCH ₂ , Et], [RA9891; H, F, Et, Cl, CF ₂ HCH ₂ , Pr], [RA9892; H, F, Et, Cl, CF ₂ HCH ₂ , i-Pr], [RA9893; H, F, Et, Cl, CF ₂ HCH ₂ , c-Pr], [RA9894; H, F, Et, Cl, CF ₂ HCH ₂ , Bu], [RA9895; H, F, Et, Cl, CF ₂ HCH ₂ , i-Bu], [RA9896; H, F, Et, Cl, CF ₂ HCH ₂ , t-Bu], [RA9897; H, F, Et, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ] , [RA9898; H, F, Et, Cl, CF ₂ HCH ₂ , Ph], [RA9899; H, F, Et, Cl, CF ₂ HCH ₂ , Bn], [RA9900; H, F, Et, Cl, CF ₂ HCH ₂ , CF ₃ ], [RA9901; H, F, Et, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA9902; H, F, Et, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA9903; H, F, Et, Cl, CF ₂ HCH ₂ , CF ₂ H], [RA9904; H, F, Et, Cl, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA9905; H , F, F, H, CF ₂ HCH ₂ , Me], [RA9906; H, F, F, H, CF ₂ HCH ₂ , Et], [RA9907; H, F, F, H, CF ₂ HCH ₂ , Pr], [RA9908; H, F, F, H, CF ₂ HCH ₂ , i-Pr], [RA9909; H, F, F, H, CF ₂ HCH ₂ , c-Pr], [RA9910; H, F, F, H, CF ₂ HCH ₂ , Bu], [RA9911; H, F, F, H, CF ₂ HCH ₂ , i-Bu], [RA9912; H, F, F, H, CF ₂ HCH ₂ , t-Bu], [RA9913; H , F, F, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA9914; H, F, F, H, CF ₂ HCH ₂ , Ph], [RA9915; H, F, F, H, CF ₂ HCH ₂ , Bn], [RA9916; H, F, F, H, CF ₂ HCH ₂ , CF ₃ ], [RA9917; H, F, F, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA9918 ; H, F, F, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA9919; H, F, F, H, CF ₂ HCH ₂ , CF ₂ H], [RA9920; H, F, F, H, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA9921; H, F, F, F, CF ₂ HCH ₂ , Me], [RA9922; H, F, F, F, CF ₂ HCH ₂ , Et] , [RA9923; H, F, F, F, CF ₂ HCH ₂ , Pr], [RA9924; H, F, F, F, CF ₂ HCH ₂ , i-Pr], [RA9925; H, F, F, F, CF ₂ HCH ₂ , c-Pr], [RA9926; H, F, F, F, CF ₂ HCH ₂ , Bu], [RA9927; H, F, F, F, CF ₂ HCH ₂ , i-Bu ], [RA9928; H, F, F, F, CF ₂ HCH ₂ , t-Bu], [RA9929; H, F, F, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA9930; H, F, F, F, CF ₂ HCH ₂ , Ph], [RA9931; H, F, F, F, CF ₂ HCH ₂ , Bn], [RA9932; H, F, F, F, CF ₂ HCH ₂ , CF ₃ ], [RA9933; H, F, F, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA9934; H, F, F, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA9935; H, F, F, F, CF ₂ HCH ₂ , CF ₂ H], [RA9936; H, F, F, F, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA9937; H, F, F, Cl , CF ₂ HCH ₂ , Me], [RA9938; H, F, F, Cl, CF ₂ HCH ₂ , Et], [RA9939 ; H, F, F, Cl, CF ₂ HCH ₂ , Pr], [RA9940; H, F, F, Cl, CF ₂ HCH ₂ , i-Pr], [RA9941; H, F, F, Cl, CF ₂ HCH ₂ , c-Pr], [RA9942; H, F, F, Cl, CF ₂ HCH ₂ , Bu], [RA9943; H, F, F, Cl, CF ₂ HCH ₂ , i-Bu], [ RA9944; H, F, F, Cl, CF ₂ HCH ₂ , t-Bu], [RA9945; H, F, F, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA9946; H, F, F , Cl, CF ₂ HCH ₂ , Ph], [RA9947; H, F, F, Cl, CF ₂ HCH ₂ , Bn], [RA9948; H, F, F, Cl, CF ₂ HCH ₂ , CF ₃ ], [RA9949; H, F, F, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA9950; H, F, F, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA9951; H, F , F, Cl, CF ₂ HCH ₂ , CF ₂ H], [RA9952; H, F, F, Cl, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA9953; H, F, Cl, H, CF _{2 HCH 2, Me], [RA9954} ; H, F, Cl, H, CF 2 HCH 2, Et], [RA9955; H, F, Cl, H, CF 2 HCH 2, Pr], [RA9956; H, F , Cl, H, CF ₂ HCH ₂ , i-Pr], [RA9957; H, F, Cl, H, CF ₂ HCH ₂ , c-Pr], [RA9958; H, F, Cl, H, CF ₂ HCH ₂ , Bu], [RA9959; H, F, Cl, H, CF ₂ HCH ₂ , i-Bu], [RA9960; H, F, Cl, H, CF ₂ HCH ₂ , t-Bu], [RA9961; H, F, Cl, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA9962; H, F, Cl, H, CF ₂ HCH ₂ , Ph], [RA9963; H, F, Cl, H, CF ₂ HCH ₂ , Bn], [RA9964; H, F, Cl, H, CF ₂ HCH ₂ , CF ₃ ], [RA9965; H, F, Cl, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [ RA9966; H, F, Cl, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [R A9967; H, F, Cl, H, CF ₂ HCH ₂ , CF ₂ H], [RA9968; H, F, Cl, H, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA9969; H, F, Cl , Cl, CF ₂ HCH ₂ , Me], [RA9970; H, F, Cl, Cl, CF ₂ HCH ₂ , Et], [RA9971; H, F, Cl, Cl, CF ₂ HCH ₂ , Pr], [ RA9972; H, F, Cl, Cl, CF ₂ HCH ₂ , i-Pr], [RA9973; H, F, Cl, Cl, CF ₂ HCH
₂ , c-Pr], [RA9974; H, F, Cl, Cl, CF ₂ HCH ₂ , Bu], [RA9975; H, F, Cl, Cl, CF ₂ HCH ₂ , i-Bu], [RA9976; H, F, Cl, Cl, CF ₂ HCH ₂ , t-Bu], [RA9977; H, F, Cl, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RA9978; H, F, Cl, Cl , CF ₂ HCH ₂ , Ph], [RA9979; H, F, Cl, Cl, CF ₂ HCH ₂ , Bn], [RA9980; H, F, Cl, Cl, CF ₂ HCH ₂ , CF ₃ ], [RA9981 ; H, F, Cl, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RA9982; H, F, Cl, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RA9983; H, F, Cl , Cl, CF ₂ HCH ₂ , CF ₂ H], [RA9984; H, F, Cl, Cl, CF ₂ HCH ₂ , CF ₂ HCH ₂ ], [RA9985; H, F, Me, H, CF ₃ CH ₂ , Me], [RA9986; H, F, Me, H, CF ₃ CH ₂ , Et], [RA9987; H, F, Me, H, CF ₃ CH ₂ , Pr], [RA9988; H, F, Me , H, CF ₃ CH ₂ , i-Pr], [RA9989; H, F, Me, H, CF ₃ CH ₂ , c-Pr], [RA9990; H, F, Me, H, CF ₃ CH ₂ , Bu], [RA9991; H, F, Me, H, CF ₃ CH ₂ , i-Bu], [RA9992; H, F, Me, H, CF ₃ CH ₂ , t-Bu], [RA9993; H, F, Me, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RA9994; H, F, Me, H, CF ₃ CH ₂ , Ph], [RA9995; H, F, Me, H, CF ₃ CH ₂ , Bn], [RA9996; H, F, Me, H, CF ₃ CH ₂ , CF ₃ ], [RA9997; H, F, Me, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA9998; H, F, Me, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA9999; H, F, Me, H, CF ₃ CH ₂ , CF ₂ H], [RA10000; H, F, Me, H , CF ₃ CH ₂ , CF ₂ HCH ₂ ],

[RA10001; H, F, Me, Me, CF ₃ CH ₂ , Me], [RA10002; H, F, Me, Me, CF ₃ CH ₂ , Et], [RA10003; H, F, Me, Me, CF ₃ CH ₂ , Pr], [RA10004; H, F, Me, Me, CF ₃ CH ₂ , i-Pr], [RA10005; H, F, Me, Me, CF ₃ CH ₂ , c-Pr], [ RA10006; H, F, Me, Me, CF ₃ CH ₂ , Bu], [RA10007; H, F, Me, Me, CF ₃ CH ₂ , i-Bu], [RA10008; H, F, Me, Me, CF ₃ CH ₂ , t-Bu], [RA10009; H, F, Me, Me, CF ₃ CH ₂ , c-PrCH ₂ ], [RA10010; H, F, Me, Me, CF ₃ CH ₂ , Ph] , [RA10011; H, F, Me, Me, CF ₃ CH ₂ , Bn], [RA10012; H, F, Me, Me, CF ₃ CH ₂ , CF ₃ ], [RA10013; H, F, Me, Me , CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA10014; H, F, Me, Me, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA10015; H, F, Me, Me, CF ₃ CH ₂ , CF ₂ H], [RA10016; H, F, Me, Me, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA10017; H, F, Me, Et, CF ₃ CH ₂ , Me], [RA10018; H , F, Me, Et, CF ₃ CH ₂ , Et], [RA10019; H, F, Me, Et, CF ₃ CH ₂ , Pr], [RA10020; H, F, Me, Et, CF ₃ CH ₂ , i-Pr], [RA10021; H, F, Me, Et, CF ₃ CH ₂ , c-Pr], [RA10022; H, F, Me, Et, CF ₃ CH ₂ , Bu], [RA10023; H, F, Me, Et, CF ₃ CH ₂ , i-Bu], [RA10024; H, F, Me, Et, CF ₃ CH ₂ , t-Bu], [RA10025; H, F, Me, Et, CF _{3 CH 2, c-PrCH 2]} , [RA10026; H, F, Me, Et, CF 3 CH 2, Ph], [RA10027; H, F, Me, Et, CF 3 CH 2, Bn], [RA10028; H, F, Me, Et, C F ₃ CH ₂ , CF ₃ ], [RA10029; H, F, Me, Et, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA10030; H, F, Me, Et, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA10031; H, F, Me, Et, CF ₃ CH ₂ , CF ₂ H], [RA10032; H, F, Me, Et, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA10033; H , F, Me, F, CF ₃ CH ₂ , Me], [RA10034; H, F, Me, F, CF ₃ CH ₂ , Et], [RA10035; H, F, Me, F, CF ₃ CH ₂ , Pr], [RA10036; H, F, Me, F, CF ₃ CH ₂ , i-Pr], [RA10037; H, F, Me, F, CF ₃ CH ₂ , c-Pr], [RA10038; H, F, Me, F, CF ₃ CH ₂ , Bu], [RA10039; H, F, Me, F, CF ₃ CH ₂ , i-Bu], [RA10040; H, F, Me, F, CF ₃ CH ₂ , t-Bu], [RA10041; H, F, Me, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RA10042; H, F, Me, F, CF ₃ CH ₂ , Ph], [RA10043; H, F, Me, F, CF ₃ CH ₂ , Bn], [RA10044; H, F, Me, F, CF ₃ CH ₂ , CF ₃ ], [RA10045; H, F, Me, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA10046; H, F, Me, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA10047; H, F, Me, F, CF ₃ CH ₂ , CF ₂ H] , [RA10048; H, F, Me, F, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA10049; H, F, Me, Cl, CF ₃ CH ₂ , Me], [RA10050; H, F, Me , Cl, CF ₃ CH ₂ , Et], [RA10051; H, F, Me, Cl, CF ₃ CH ₂ , Pr], [RA10052; H, F, Me, Cl, CF ₃ CH ₂ , i-Pr] , [RA10053; H, F, Me, Cl, CF ₃ CH ₂ , c-Pr], [RA10054; H, F, Me, Cl, CF ₃ CH ₂ , Bu], [RA10055; H, F, Me, Cl, CF ₃ CH ₂ , i-Bu] , [RA10056; H, F, Me, Cl, CF ₃ CH ₂ , t-Bu], [RA10057; H, F, Me, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RA10058; H, F , Me, Cl, CF ₃ CH ₂ , Ph], [RA10059; H, F, Me, Cl, CF ₃ CH ₂ , Bn], [RA10060; H, F, Me, Cl, CF ₃ CH ₂ , CF ₃ ], [RA10061; H, F, Me, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA10062; H, F, Me, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA10063; H , F, Me, Cl, CF ₃ CH ₂ , CF ₂ H], [RA10064; H, F, Me, Cl, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA10065; H, F, Et, H, CF ₃ CH ₂ , Me], [RA10066; H, F, Et, H, CF ₃ CH ₂ , Et], [RA10067; H, F, Et, H, CF ₃ CH ₂ , Pr], [RA10068; H , F, Et, H, CF ₃ CH ₂ , i-Pr], [RA10069; H, F, Et, H, CF ₃ CH ₂ , c-Pr], [RA10070; H, F, Et, H, CF ₃ CH ₂ , Bu], [RA10071; H, F, Et, H, CF ₃ CH ₂ , i-Bu], [RA10072; H, F, Et, H, CF ₃ CH ₂ , t-Bu], [ RA10073; H, F, Et, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RA10074; H, F, Et, H, CF ₃ CH ₂ , Ph], [RA10075; H, F, Et, H , CF ₃ CH ₂ , Bn], [RA10076; H, F, Et, H, CF ₃ CH ₂ , CF ₃ ], [RA10077; H, F, Et, H, CF ₃ CH ₂ , CF ₃ CH ₂ ] , [RA10078; H, F, Et, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA10079; H, F, Et, H, CF ₃ CH ₂ , CF ₂ H], [RA10080; H, F , Et, H, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA10081; H, F, Et, F, CF ₃ CH ₂ , Me], [RA10082; H, F, Et, F, CF ₃ CH ₂ , Et], [RA10083; H, F, Et, F, CF ₃ CH ₂ , Pr], [RA10084; H, F, Et, F, CF ₃ CH ₂ , i-Pr], [RA10085; H, F, Et, F, CF ₃ CH ₂ , c-Pr], [RA10086; H, F, Et, F, CF ₃ CH ₂ , Bu], [RA10087; H, F, Et, F, CF ₃ CH ₂ , i-Bu], [RA10088; H , F, Et, F, CF ₃ CH ₂ , t-Bu], [RA10089; H, F, Et, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RA10090; H, F, Et, F, CF ₃ CH ₂ , Ph], [RA10091; H, F, Et, F, CF ₃ CH ₂ , Bn], [RA10092; H, F, Et, F, CF ₃ CH ₂ , CF ₃ ], [RA10093; H, F, Et, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA10094; H, F, Et, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA10095; H, F, Et, F, CF ₃ CH ₂ , CF ₂ H], [RA10096; H, F, Et, F, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA10097; H, F, Et, Cl, CF ₃ CH ₂ , Me], [RA10098; H, F, Et, Cl, CF ₃ CH ₂ , Et], [RA10099; H, F, Et, Cl, CF ₃ CH ₂ , Pr], [RA10100; H, F, Et, Cl, CF ₃ CH ₂ , i-Pr], [RA10101; H, F, Et, Cl, CF ₃ CH ₂ , c-Pr], [RA10102; H, F, Et, Cl, CF ₃ CH ₂ , Bu ], [RA10103; H, F, Et, Cl, CF ₃ CH ₂ , i-Bu], [RA10104; H, F, Et, Cl, CF ₃ CH ₂ , t-Bu], [RA10105; H, F , Et, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RA10106; H, F, Et, Cl, CF ₃ CH ₂ , Ph], [RA10107; H, F, Et, Cl, CF ₃ CH ₂ , Bn], [RA10108; H, F, Et, Cl, CF ₃ CH ₂ , CF ₃ ], [RA10109; H, F, Et, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA10110; H , F, Et, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA10111; H, F, Et, Cl, CF ₃ CH ₂ , CF ₂ H], [RA10112; H, F, Et, Cl, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA10113; H, F, F, H, CF ₃ CH ₂ , Me], [RA10114; H, F, F, H, CF ₃ CH ₂ , Et], [RA10115; H, F, F, H, CF ₃ CH ₂ , Pr], [RA10116; H, F, F, H, CF ₃ CH ₂ , i-Pr], [RA10117; H, F, F, H, CF ₃ CH ₂ , c-Pr], [RA10118; H , F, F, H, CF ₃ CH ₂ , Bu], [RA10119; H, F, F, H, CF ₃ CH ₂ , i-Bu], [RA10120; H, F, F, H, CF ₃ CH ₂ , t-Bu], [RA10121; H, F, F, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RA10122; H, F, F, H, CF ₃ CH ₂ , Ph], [RA10123 ; H, F, F, H, CF ₃ CH ₂ , Bn], [RA10124; H, F, F, H, CF ₃ CH ₂ , CF ₃ ], [RA10125; H, F, F, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA10126; H, F, F, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA10127; H, F, F, H, CF ₃ CH ₂ , CF ₂ H ], [RA10128; H, F, F, H, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA10129; H, F, F, F, CF ₃ CH ₂ , Me], [RA10130; H, F, F, F, CF ₃ CH ₂ , Et], [RA10131; H, F, F, F, CF ₃ CH ₂ , Pr], [RA10132; H, F, F, F, CF ₃ CH ₂ , i-Pr ], [RA10133; H, F, F, F, CF ₃ CH ₂ , c-Pr], [RA10134; H, F, F, F, CF ₃ CH ₂ , Bu], [RA10135; H, F, F , F, CF ₃ CH ₂ , i-Bu], [RA10136; H, F, F, F, CF ₃ CH ₂ , t-Bu], [RA10137; H, F, F, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RA10138; H, F, F, F, CF ₃ CH ₂ , Ph], [RA10139; H, F, F, F, CF ₃ CH ₂ , Bn], [RA10140; H, F, F, F, CF ₃ CH ₂ , CF ₃ ], [RA10141; H, F, F, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA10142; H, F, F, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA10143; H, F, F, F, CF ₃ CH ₂ , CF ₂ H], [RA10144; H, F, F, F, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA10145; H, F, F, Cl, CF ₃ CH ₂ , Me], [RA10146; H, F, F, Cl, CF ₃ CH ₂ , Et], [RA10147; H, F, F, Cl, CF ₃ CH ₂ , Pr], [RA10148; H, F, F, Cl, CF ₃ CH ₂ , i-Pr], [RA10149; H, F, F, Cl, CF ₃ CH ₂ , c-Pr], [RA10150; H, F, F, Cl, CF ₃ CH ₂ , Bu], [RA10151; H, F, F, Cl, CF ₃ CH ₂ , i -Bu], [RA10152; H, F, F, Cl, CF ₃ CH ₂ , t-Bu], [RA10153; H, F, F, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RA10154; H, F, F, Cl, CF ₃ CH ₂ , Ph], [RA10155; H, F, F, Cl, CF ₃ CH ₂ , Bn], [RA10156; H, F, F, Cl, CF ₃ CH ₂ , CF ₃ ], [RA10157; H, F, F, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA10158; H, F, F, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [ RA10159; H, F, F, Cl, CF ₃ CH ₂ , CF ₂ H], [RA10160; H, F, F, Cl, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA10161; H, F, Cl , H, CF ₃ CH ₂ , Me], [RA10162; H, F, Cl, H, CF ₃ CH ₂ , Et], [RA10163; H, F, Cl, H, CF ₃ CH ₂ , Pr], [ RA10164; H, F, Cl, H, CF ₃ CH ₂ , i-Pr], [RA10165; H, F, Cl, H, CF ₃ CH ₂ , c-Pr], [RA10166; H, F, Cl, H, CF ₃ CH ₂ , Bu], [RA10167; H, F, Cl, H, CF ₃ CH ₂ , i-Bu], [RA10168; H, F, Cl, H, CF ₃ CH ₂ , t-Bu], [RA10169; H, F, Cl, H, CF ₃ CH ₂ , c -PrCH ₂ ], [RA10170; H, F, Cl, H, CF ₃ CH ₂ , Ph], [RA10171; H, F, Cl, H, CF ₃ CH ₂ , Bn], [RA10172; H, F, Cl, H, CF ₃ CH ₂ , CF ₃ ], [RA10173; H, F, Cl, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA10174; H, F, Cl, H, CF ₃ CH ₂
, CF ₃ CF ₂ ], [RA10175; H, F, Cl, H, CF ₃ CH ₂ , CF ₂ H], [RA10176; H, F, Cl, H, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA10177; H, F, Cl, Cl, CF ₃ CH ₂ , Me], [RA10178; H, F, Cl, Cl, CF ₃ CH ₂ , Et], [RA10179; H, F, Cl, Cl, CF ₃ CH ₂ , Pr], [RA10180; H, F, Cl, Cl, CF ₃ CH ₂ , i-Pr], [RA10181; H, F, Cl, Cl, CF ₃ CH ₂ , c-Pr], [ RA10182; H, F, Cl, Cl, CF ₃ CH ₂ , Bu], [RA10183; H, F, Cl, Cl, CF ₃ CH ₂ , i-Bu], [RA10184; H, F, Cl, Cl, CF ₃ CH ₂ , t-Bu], [RA10185; H, F, Cl, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RA10186; H, F, Cl, Cl, CF ₃ CH ₂ , Ph] , [RA10187; H, F, Cl, Cl, CF ₃ CH ₂ , Bn], [RA10188; H, F, Cl, Cl, CF ₃ CH ₂ , CF ₃ ], [RA10189; H, F, Cl, Cl , CF ₃ CH ₂ , CF ₃ CH ₂ ], [RA10190; H, F, Cl, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RA10191; H, F, Cl, Cl, CF ₃ CH ₂ , CF ₂ H], [RA10192; H, F, Cl, Cl, CF ₃ CH ₂ , CF ₂ HCH ₂ ], [RA10193; H, F, Me, H, HCCCH ₂ , Me], [RA10194; H, F _{, Me, H, HCCCH 2,} Et], [RA10195; H, F, Me, H, HCCCH 2, Pr], [RA10196; H, F, Me, H, HCCCH 2, i-Pr], [RA10197; H, F, Me, H, HCCCH ₂ , c-Pr], [RA10198; H, F, Me, H, HCCCH ₂ , Bu], [RA10199; H, F, Me, H, HCCCH ₂ , i-Bu ], [RA10200; H, F, Me, H, HCCCH ₂ , t-Bu],

[RA10201; H, F, Me, H, HCCCH ₂ , c-PrCH ₂ ], [RA10202; H, F, Me, H, HCCCH ₂ , Ph], [RA10203; H, F, Me, H, HCCCH ₂ , Bn], [RA10204; H, F, Me, H, HCCCH ₂ , CF ₃ ], [RA10205; H, F, Me, H, HCCCH ₂ , CF ₃ CH ₂ ], [RA10206; H, F, Me , H, HCCCH ₂ , CF ₃ CF ₂ ], [RA10207; H, F, Me, H, HCCCH ₂ , CF ₂ H], [RA10208; H, F, Me, H, HCCCH ₂ , CF ₂ HCH ₂ ] , [RA10209; H, F, Me, Me, HCCCH ₂ , Me], [RA10210; H, F, Me, Me, HCCCH ₂ , Et], [RA10211; H, F, Me, Me, HCCCH ₂ , Pr ], [RA10212; H, F, Me, Me, HCCCH ₂ , i-Pr], [RA10213; H, F, Me, Me, HCCCH ₂ , c-Pr], [RA10214; H, F, Me, Me , HCCCH ₂ , Bu], [RA10215; H, F, Me, Me, HCCCH ₂ , i-Bu], [RA10216; H, F, Me, Me, HCCCH ₂ , t-Bu], [RA10217; H, F, Me, Me, HCCCH ₂ , c-PrCH ₂ ], [RA10218; H, F, Me, Me, HCCCH ₂ , Ph], [RA10219; H, F, Me, Me, HCCCH ₂ , Bn], [ RA10220; H, F, Me, Me, HCCCH ₂ , CF ₃ ], [RA10221; H, F, Me, Me, HCCCH ₂ , CF ₃ CH ₂ ], [RA10222; H, F, Me, Me, HCCCH ₂ , CF ₃ CF ₂ ], [RA10223; H, F, Me, Me, HCCCH ₂ , CF ₂ H], [RA10224; H, F, Me, Me, HCCCH ₂ , CF ₂ HCH ₂ ], [RA10225; H , F, Me, Et, HCCCH ₂ , Me], [RA10226; H, F, Me, Et, HCCCH ₂ , Et], [RA10227; H, F, Me, Et, HCCCH ₂ , Pr], [RA10228; H, F, Me, Et, HCCCH ₂ , i-Pr], [RA10229; H, F, Me, Et, HCCCH _{2, c-Pr], [} RA10230; H, F, Me, Et, HCCCH 2, Bu], [RA10231; H, F, Me, Et, HCCCH 2, i-Bu], [RA10232; H, F, _{Me, Et, HCCCH 2, t} -Bu], [RA10233; H, F, Me, Et, HCCCH 2, c-PrCH 2], [RA10234; H, F, Me, Et, HCCCH 2, Ph], [ RA10235; H, F, Me, Et, HCCCH ₂ , Bn], [RA10236; H, F, Me, Et, HCCCH ₂ , CF ₃ ], [RA10237; H, F, Me, Et, HCCCH ₂ , CF ₃ CH ₂ ], [RA10238; H, F, Me, Et, HCCCH ₂ , CF ₃ CF ₂ ], [RA10239; H, F, Me, Et, HCCCH ₂ , CF ₂ H], [RA10240; H, F, Me, Et, HCCCH ₂ , CF ₂ HCH ₂ ], [RA10241; H, F, Me, F, HCCCH ₂ , Me], [RA10242; H, F, Me, F, HCCCH ₂ , Et], [RA10243; H, F, Me, F, HCCCH ₂ , Pr], [RA10244; H, F, Me, F, HCCCH ₂ , i-Pr], [RA10245; H, F, Me, F, HCCCH ₂ , c-Pr ], [RA10246; H, F, Me, F, HCCCH ₂ , Bu], [RA10247; H, F, Me, F, HCCCH ₂ , i-Bu], [RA10248; H, F, Me, F, HCCCH ₂ , t-Bu], [RA10249; H, F, Me, F, HCCCH ₂ , c-PrCH ₂ ], [RA10250; H, F, Me, F, HCCCH ₂ , Ph], [RA10251; H, F , Me, F, HCCCH ₂ , Bn], [RA10252; H, F, Me, F, HCCCH ₂ , CF ₃ ], [RA10253; H, F, Me, F, HCCCH ₂ , CF ₃ CH ₂ ], [ RA10254; H, F, Me, F, HCCCH ₂ , CF ₃ CF ₂ ], [RA10255; H, F, Me, F, HCCCH ₂ , CF ₂ H], [RA10256; H, F, Me, F, HCCCH ₂ , CF ₂ HCH ₂ ], [RA10257; H, F, Me, Cl, HCCCH ₂ , Me], [RA10258; H, F, Me, Cl, H CCCH ₂ , Et], [RA10259; H, F, Me, Cl, HCCCH ₂ , Pr], [RA10260; H, F, Me, Cl, HCCCH ₂ , i-Pr], [RA10261; H, F, Me , Cl, HCCCH ₂ , c-Pr], [RA10262; H, F, Me, Cl, HCCCH ₂ , Bu], [RA10263; H, F, Me, Cl, HCCCH ₂ , i-Bu], [RA10264; H, F, Me, Cl, HCCCH ₂ , t-Bu], [RA10265; H, F, Me, Cl, HCCCH ₂ , c-PrCH ₂ ], [RA10266; H, F, Me, Cl, HCCCH ₂ , Ph], [RA10267; H, F, Me, Cl, HCCCH ₂ , Bn], [RA10268; H, F, Me, Cl, HCCCH ₂ , CF ₃ ], [RA10269; H, F, Me, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RA10270; H, F, Me, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RA10271; H, F, Me, Cl, HCCCH ₂ , CF ₂ H], [RA10272; H, F, Me, Cl, HCCCH ₂ , CF ₂ HCH ₂ ], [RA10273; H, F, Et, H, HCCCH ₂ , Me], [RA10274; H, F, Et, H, HCCCH ₂ , Et] , [RA10275; H, F, Et, H, HCCCH ₂ , Pr], [RA10276; H, F, Et, H, HCCCH ₂ , i-Pr], [RA10277; H, F, Et, H, HCCCH ₂ , c-Pr], [RA10278; H, F, Et, H, HCCCH ₂ , Bu], [RA10279; H, F, Et, H, HCCCH ₂ , i-Bu], [RA10280; H, F, Et , H, HCCCH ₂ , t-Bu], [RA10281; H, F, Et, H, HCCCH ₂ , c-PrCH ₂ ], [RA10282; H, F, Et, H, HCCCH ₂ , Ph], [RA10283 ; H, F, Et, H, HCCCH ₂ , Bn], [RA10284; H, F, Et, H, HCCCH ₂ , CF ₃ ], [RA10285; H, F, Et, H, HCCCH ₂ , CF ₃ CH ₂ ], [RA10286; H, F, Et, H, HCCCH ₂ , CF ₃ CF ₂ ], [RA10287; H, F, Et, H, HCCCH ₂ , CF ₂ H], [RA10288; H, F, Et, H, HCCCH ₂ , CF ₂ HCH ₂ ], [RA10289; H, F, Et, F, HCCCH ₂ , Me], [RA10290; H, F, Et, F, HCCCH ₂ , Et], [RA10291; H, F, Et, F, HCCCH ₂ , Pr], [RA10292; H, F, Et, F, HCCCH ₂ , i-Pr], [RA10293; H , F, Et, F, HCCCH ₂ , c-Pr], [RA10294; H, F, Et, F, HCCCH ₂ , Bu], [RA10295; H, F, Et, F, HCCCH ₂ , i-Bu] , [RA10296; H, F, Et, F, HCCCH ₂ , t-Bu], [RA10297; H, F, Et, F, HCCCH ₂ , c-PrCH ₂ ], [RA10298; H, F, Et, F , HCCCH ₂ , Ph], [RA10299; H, F, Et, F, HCCCH ₂ , Bn], [RA10300; H, F, Et, F, HCCCH ₂ , CF ₃ ], [RA10301; H, F, Et , F, HCCCH ₂ , CF ₃ CH ₂ ], [RA10302; H, F, Et, F, HCCCH ₂ , CF ₃ CF ₂ ], [RA10303; H, F, Et, F, HCCCH ₂ , CF ₂ H] , [RA10304; H, F, Et, F, HCCCH ₂ , CF ₂ HCH ₂ ], [RA10305; H, F, Et, Cl, HCCCH ₂ , Me], [RA10306; H, F, Et, Cl, HCCCH ₂ , Et], [RA10307; H, F, Et, Cl, HCCCH ₂ , Pr], [RA10308; H, F, Et, Cl, HCCCH ₂ , i-Pr], [RA10309; H, F, Et, Cl, HCCCH ₂ , c-Pr], [RA10310; H, F, Et, Cl, HCCCH ₂ , Bu], [RA10311; H, F, Et, Cl, HCCCH ₂ , i-Bu], [RA10312; H , F, Et, Cl, HCCCH ₂ , t-Bu], [RA10313; H, F, Et, Cl, HCCCH ₂ , c-PrCH ₂ ], [RA10314; H, F, Et, Cl, HCCCH ₂ , Ph ], [RA10315; H, F, Et, Cl, HCCCH ₂ , Bn], [RA10316; H, F, Et, Cl, HCCCH ₂ , CF ₃ ], [RA10 317; H, F, Et, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RA10318; H, F, Et, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RA10319; H, F, Et, Cl, HCCCH ₂ , CF ₂ H], [RA10320; H, F, Et, Cl, HCCCH ₂ , CF ₂ HCH ₂ ], [RA10321; H, F, F, H, HCCCH ₂ , Me], [RA10322; H, F, F, H, HCCCH ₂ , Et], [RA10323; H, F, F, H, HCCCH ₂ , Pr], [RA10324; H, F, F, H, HCCCH ₂ , i-Pr], [RA10325 ; H, F, F, H, HCCCH ₂ , c-Pr], [RA10326; H, F, F, H, HCCCH ₂ , Bu], [RA10327; H, F, F, H, HCCCH ₂ , i- Bu], [RA10328; H, F, F, H, HCCCH ₂ , t-Bu], [RA10329; H, F, F, H, HCCCH ₂ , c-PrCH ₂ ], [RA10330; H, F, F , H, HCCCH ₂ , Ph], [RA10331; H, F, F, H, HCCCH ₂ , Bn], [RA10332; H, F, F, H, HCCCH ₂ , CF ₃ ], [RA10333; H, F , F, H, HCCCH ₂ , CF ₃ CH ₂ ], [RA10334; H, F, F, H, HCCCH ₂ , CF ₃ CF ₂ ], [RA10335; H, F, F, H, HCCCH ₂ , CF ₂ H], [RA10336; H, F, F, H, HCCCH ₂ , CF ₂ HCH ₂ ], [RA10337; H, F, F, F, HCCCH ₂ , Me], [RA10338; H, F, F, F , HCCCH ₂ , Et], [RA10339; H, F, F, F, HCCCH ₂ , Pr], [RA10340; H, F, F, F, HCCCH ₂ , i-Pr], [RA10341; H, F, F, F, HCCCH ₂ , c-Pr], [RA10342; H, F, F, F, HCCCH ₂ , Bu], [RA10343; H, F, F, F, HCCCH ₂ , i-Bu], [RA10344 ; H, F, F, F, HCCCH ₂ , t-Bu], [RA10345; H, F, F, F, HCCCH ₂ , c-PrCH ₂ ], [RA10346; H, F, F, F, HCCCH ₂ , Ph], [RA103 47; H, F, F, F, HCCCH ₂ , Bn], [RA10348; H, F, F, F, HCCCH ₂ , CF ₃ ], [RA10349; H, F, F, F, HCCCH ₂ , CF ₃ CH ₂ ], [RA10350; H, F, F, F, HCCCH ₂ , CF ₃ CF ₂ ], [RA10351; H, F, F, F, HCCCH ₂ , CF ₂ H], [RA10352; H, F, F, F, HCCCH ₂ , CF ₂ HCH ₂ ], [RA10353; H, F, F, Cl, HCCCH ₂ , Me], [RA10354; H, F, F, Cl, HCCCH ₂ , Et], [RA10355; H, F, F, Cl, HCCCH ₂ , Pr], [RA10356; H, F, F, Cl, HCCCH ₂ , i-Pr], [RA10357; H, F, F, Cl, HCCCH ₂ , c-Pr ], [RA10358; H, F, F, Cl, HCCCH ₂ , Bu], [RA10359; H, F, F, Cl, HCCCH ₂ , i-Bu], [RA10360; H, F, F, Cl, HCCCH ₂ , t-Bu], [RA10361; H, F, F, Cl, HCCCH ₂ , c-PrCH ₂ ], [RA10362; H, F, F, Cl, HCCCH ₂ , Ph], [RA10363; H, F , F, Cl, HCCCH ₂ , Bn], [RA10364; H, F, F, Cl, HCCCH ₂ , CF ₃ ], [RA10365; H, F, F, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [ RA10366; H, F, F, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RA10367; H, F, F, Cl, HCCCH ₂ , CF ₂ H], [RA10368; H, F, F, Cl, HCCCH ₂ , CF ₂ HCH ₂ ], [RA10369; H, F, Cl, H, HCCCH ₂ , Me], [RA10370; H, F, Cl, H, HCCCH ₂ , Et], [RA10371; H, F, Cl , H, HCCCH ₂ , Pr], [RA10372; H, F, Cl, H, HCCCH ₂ , i-Pr], [RA10373; H, F, Cl, H, HCCCH ₂ , c-Pr], [RA10374; H, F, Cl, H, HCCCH ₂ , Bu], [RA10375; H, F, Cl, H, HCCCH ₂ , i-Bu], [RA10376; H, F, Cl, H, HCCCH ₂ , t -Bu], [RA10377; H, F, Cl, H, HCCCH ₂ , c-PrCH ₂ ], [RA10378; H, F, Cl, H, HCCCH ₂ , Ph], [RA10379; H, F, Cl, H, HCCCH ₂ , Bn], [RA10380; H, F, Cl, H, HCCCH ₂ , CF ₃ ], [RA10381; H, F, Cl, H, HCCCH ₂ , CF ₃ CH ₂ ], [RA10382; H , F, Cl, H, HCCCH ₂ , CF ₃ CF ₂ ], [RA10383; H, F, Cl, H, HCCCH ₂ , CF ₂ H], [RA10384; H, F, Cl, H, HCCCH ₂ , CF ₂ HCH ₂ ], [RA10385; H, F, Cl, Cl, HCCCH ₂ , Me], [RA10386; H, F, Cl, Cl, HCCCH ₂ , Et], [RA10387; H, F, Cl, Cl, HCCCH ₂ , Pr], [RA10388; H, F, Cl, Cl, HCCCH ₂ , i-Pr], [RA10389; H, F, Cl, Cl, HCCCH ₂ , c-Pr], [RA10390; H, F , Cl, Cl, HCCCH ₂ , Bu], [RA10391; H, F, Cl, Cl, HCCCH ₂ , i-Bu], [RA10392; H, F, Cl, Cl, HCCCH ₂ , t-Bu], [ RA10393; H, F, Cl, Cl, HCCCH ₂ , c-PrCH ₂ ], [RA10394; H, F, Cl, Cl, HCCCH ₂ , Ph], [RA10395; H, F, Cl, Cl, HCCCH ₂ , Bn], [RA10396; H, F, Cl, Cl, HCCCH ₂ , CF ₃ ], [RA10397; H, F, Cl, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RA10398; H, F, Cl, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RA10399; H, F, Cl, Cl, HCCCH ₂ , CF ₂ H], [RA10400; H, F, Cl, Cl, HCCCH ₂ , CF ₂ HCH ₂ ],

[RA10401; H, F, Me, H, CH ₃ CCCH ₂ , Me], [RA10402; H, F, Me, H, CH ₃ CCCH ₂ , Et], [RA10403; H, F, Me, H, CH ₃ CCCH ₂ , Pr], [RA10404; H, F, Me, H, CH ₃ CCCH ₂ , i-Pr], [RA10405; H, F, Me, H, CH ₃ CCCH ₂ , c-Pr], [ RA10406; H, F, Me, H, CH ₃ CCCH ₂ , Bu], [RA10407; H, F, Me, H, CH ₃ CCCH ₂ , i-Bu], [RA10408; H, F, Me, H, CH ₃ CCCH ₂ , t-Bu], [RA10409; H, F, Me, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA10410; H, F, Me, H, CH ₃ CCCH ₂ , Ph] , [RA10411; H, F, Me, H, CH ₃ CCCH ₂ , Bn], [RA10412; H, F, Me, H, CH ₃ CCCH ₂ , CF ₃ ], [RA10413; H, F, Me, H , CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA10414; H, F, Me, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA10415; H, F, Me, H, CH ₃ CCCH ₂ , CF ₂ H], [RA10416; H, F, Me, H, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA10417; H, F, Me, Me, CH ₃ CCCH ₂ , Me], [RA10418; H , F, Me, Me, CH ₃ CCCH ₂ , Et], [RA10419; H, F, Me, Me, CH ₃ CCCH ₂ , Pr], [RA10420; H, F, Me, Me, CH ₃ CCCH ₂ , i-Pr], [RA10421; H, F, Me, Me, CH ₃ CCCH ₂ , c-Pr], [RA10422; H, F, Me, Me, CH ₃ CCCH ₂ , Bu], [RA10423; H, F, Me, Me, CH ₃ CCCH ₂ , i-Bu], [RA10424; H, F, Me, Me, CH ₃ CCCH ₂ , t-Bu], [RA10425; H, F, Me, Me, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA10426; H, F, Me, Me, CH ₃ CCCH ₂ , Ph], [RA10427; H, F, Me, Me , CH ₃ CCCH ₂ , Bn], [RA10428; H, F, Me, Me, CH ₃ CCCH ₂ , CF ₃ ], [RA10429; H, F, Me, Me, CH ₃ CCCH ₂ , CF ₃ CH ₂ ] , [RA10430; H, F, Me, Me, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA10431; H, F, Me, Me, CH ₃ CCCH ₂ , CF ₂ H], [RA10432; H, F , Me, Me, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA10433; H, F, Me, Et, CH ₃ CCCH ₂ , Me], [RA10434; H, F, Me, Et, CH ₃ CCCH ₂ , Et], [RA10435; H, F, Me, Et, CH ₃ CCCH ₂ , Pr], [RA10436; H, F, Me, Et, CH ₃ CCCH ₂ , i-Pr], [RA10437; H, F , Me, Et, CH ₃ CCCH ₂ , c-Pr], [RA10438; H, F, Me, Et, CH ₃ CCCH ₂ , Bu], [RA10439; H, F, Me, Et, CH ₃ CCCH ₂ , i-Bu], [RA10440; H, F, Me, Et, CH ₃ CCCH ₂ , t-Bu], [RA10441; H, F, Me, Et, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA10442 ; H, F, Me, Et, CH ₃ CCCH ₂ , Ph], [RA10443; H, F, Me, Et, CH ₃ CCCH ₂ , Bn], [RA10444; H, F, Me, Et, CH ₃ CCCH ₂ , CF ₃ ], [RA10445; H, F, Me, Et, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA10446; H, F, Me, Et, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA10447; H, F, Me, Et, CH ₃ CCCH ₂ , CF ₂ H], [RA10448; H, F, Me, Et, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA10449; H, F, Me, F, CH ₃ CCCH ₂ , Me], [RA10450; H, F, Me, F, CH ₃ CCCH ₂ , Et], [RA10451; H, F, Me, F, CH ₃ CCCH ₂ , Pr], [RA10452; H, F, Me, F, CH ₃ CCCH ₂ , i-Pr], [RA10 453; H, F, Me, F, CH ₃ CCCH ₂ , c-Pr], [RA10454; H, F, Me, F, CH ₃ CCCH ₂ , Bu], [RA10455; H, F, Me, F, CH ₃ CCCH ₂ , i-Bu], [RA10456; H, F, Me, F, CH ₃ CCCH ₂ , t-Bu], [RA10457; H, F, Me, F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA10458; H, F, Me, F, CH ₃ CCCH ₂ , Ph], [RA10459; H, F, Me, F, CH ₃ CCCH ₂ , Bn], [RA10460; H, F, Me, F, CH ₃ CCCH ₂ , CF ₃ ], [RA10461; H, F, Me, F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA10462; H, F, Me, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA10463; H, F, Me, F, CH ₃ CCCH ₂ , CF ₂ H], [RA10464; H, F, Me, F, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA10465 ; H, F, Me, Cl, CH ₃ CCCH ₂ , Me], [RA10466; H, F, Me, Cl, CH ₃ CCCH ₂ , Et], [RA10467; H, F, Me, Cl, CH ₃ CCCH ₂ , Pr], [RA10468; H, F, Me, Cl, CH ₃ CCCH ₂ , i-Pr], [RA10469; H, F, Me, Cl, CH ₃ CCCH ₂ , c-Pr], [RA10470; H, F, Me, Cl, CH ₃ CCCH ₂ , Bu], [RA10471; H, F, Me, Cl, CH ₃ CCCH ₂ , i-Bu], [RA10472; H, F, Me, Cl, CH ₃ CCCH ₂ , t-Bu], [RA10473; H, F, Me, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA10474; H, F, Me, Cl, CH ₃ CCCH ₂ , Ph], [ RA10475; H, F, Me, Cl, CH ₃ CCCH ₂ , Bn], [RA10476; H, F, Me, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RA10477; H, F, Me, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA10478; H, F, Me, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [R A10479; H, F, Me, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RA10480; H, F, Me, Cl, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA10481; H, F, Et , H, CH ₃ CCCH ₂ , Me], [RA10482; H, F, Et, H, CH ₃ CCCH ₂ , Et], [RA10483; H, F, Et, H, CH ₃ CCCH ₂ , Pr], [ RA10484; H, F, Et, H, CH ₃ CCCH ₂ , i-Pr], [RA10485; H, F, Et, H, CH ₃ CCCH ₂ , c-Pr], [RA10486; H, F, Et, H, CH ₃ CCCH ₂ , Bu], [RA10487; H, F, Et, H, CH ₃ CCCH ₂ , i-Bu], [RA10488; H, F, Et, H, CH ₃ CCCH ₂ , t-Bu ], [RA10489; H, F, Et, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA10490; H, F, Et, H, CH ₃ CCCH ₂ , Ph], [RA10491; H, F, Et, H, CH ₃ CCCH ₂ , Bn], [RA10492; H, F, Et, H, CH ₃ CCCH ₂ , CF ₃ ], [RA10493; H, F, Et, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA10494; H, F, Et, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA10495; H, F, Et, H, CH ₃ CCCH ₂ , CF ₂ H], [RA10496; H, F, Et, H, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA10497; H, F, Et, F, CH ₃ CCCH ₂ , Me], [RA10498; H, F, Et, F, CH ₃ CCCH ₂ , Et], [RA10499; H, F, Et, F, CH ₃ CCCH ₂ , Pr], [RA10500; H, F, Et, F, CH ₃ CCCH ₂ , i-Pr], [RA10501; H, F, Et, F, CH ₃ CCCH ₂ , c-Pr], [RA10502; H, F, Et, F, CH ₃ CCCH ₂ , Bu], [RA10503; H, F, Et, F, CH ₃ CCCH ₂ , i-Bu], [RA10504; H, F, Et, F, CH ₃ CCCH ₂ , t-Bu], [RA10505; H, F, Et, F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA10506; H, F, Et, F, CH ₃ CCCH ₂ , Ph], [RA10507; H, F, Et, F, CH ₃ CCCH ₂ , Bn], [RA10508; H, F, Et, F, CH ₃ CCCH ₂ , CF ₃ ], [RA10509; H, F, Et, F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA10510; H, F, Et, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA10511; H, F, Et, F, CH ₃ CCCH ₂ , CF ₂ H], [RA10512; H, F, Et, F, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA10513; H, F, Et, Cl, CH ₃ CCCH ₂ , Me], [RA10514; H, F, Et, Cl, CH ₃ CCCH ₂ , Et], [RA10515; H, F, Et , Cl, CH ₃ CCCH ₂ , Pr], [RA10516; H, F, Et, Cl, CH ₃ CCCH ₂ , i-Pr], [RA10517; H, F, Et, Cl, CH ₃ CCCH ₂ , c- Pr], [RA10518; H, F, Et, Cl, CH ₃ CCCH ₂ , Bu], [RA10519; H, F, Et, Cl, CH ₃ CCCH ₂ , i-Bu], [RA10520; H, F, Et, Cl, CH ₃ CCCH ₂ , t-Bu], [RA10521; H, F, Et, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA10522; H, F, Et, Cl, CH ₃ CCCH ₂ , Ph], [RA10523; H, F, Et, Cl, CH ₃ CCCH ₂ , Bn], [RA10524; H, F, Et, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RA10525; H, F , Et, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA10526; H, F, Et, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA10527; H, F, Et, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RA10528; H, F, Et, Cl, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA10529; H, F, F, H, CH ₃ CCCH ₂ , Me], [RA10530; H, F, F, H, CH ₃ CCCH ₂ , Et], [RA10531; H, F , F, H, CH ₃ CCCH ₂ , Pr], [RA10532; H, F, F, H, CH ₃ CCCH ₂ , i-Pr], [RA10533; H, F, F, H, CH ₃ CCCH ₂ , c-Pr], [RA10534; H, F, F, H, CH ₃ CCCH ₂ , Bu], [RA10535; H, F, F, H, CH ₃ CCCH ₂ , i-Bu], [RA10536; H, F, F, H, CH ₃ CCCH ₂ , t-Bu], [RA10537; H, F, F, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA10538; H, F, F, H, CH ₃ CCCH ₂ , Ph], [RA10539; H, F, F, H, CH ₃ CCCH ₂ , Bn], [RA10540; H, F, F, H, CH ₃ CCCH ₂ , CF ₃ ], [RA10541; H , F, F, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA10542; H, F, F, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA10543; H, F, F, H , CH ₃ CCCH ₂ , CF ₂ H], [RA10544; H, F, F, H, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA10545; H, F, F, F, CH ₃ CCCH ₂ , Me ], [RA10546; H, F, F, F, CH ₃ CCCH ₂ , Et], [RA10547; H, F, F, F, CH ₃ CCCH ₂ , Pr], [RA10548; H, F, F, F , CH ₃ CCCH ₂ , i-Pr], [RA10549; H, F, F, F, CH ₃ CCCH ₂ , c-Pr], [RA10550; H, F, F, F, CH ₃ CCCH ₂ , Bu] , [RA10551; H, F, F, F, CH ₃ CCCH ₂ , i-Bu], [RA10552; H, F, F, F, CH ₃ CCCH ₂ , t-Bu], [RA10553; H, F, F, F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA10554; H, F, F, F, CH ₃ CCCH ₂ , Ph], [RA10555; H, F, F, F, CH ₃ CCCH ₂ , Bn], [RA10556; H, F, F, F, CH ₃ CCCH ₂ , CF ₃ ], [RA10557; H, F, F, F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA10558; H, F, F, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA10559; H, F, F, F, CH ₃ CCCH ₂ , CF ₂ H], [RA10560; H, F, F, F, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA10561; H, F, F, Cl, CH ₃ CCCH ₂ , Me], [RA10562; H, F, F, Cl, CH ₃ CCCH ₂ , Et], [RA10563; H, F, F, Cl , CH ₃ CCCH ₂ , Pr], [RA10564; H, F, F, Cl, CH ₃ CCCH ₂ , i-Pr], [RA10565; H, F, F, Cl, CH ₃ CCCH ₂ , c-Pr] , [RA10566; H, F, F, Cl, CH ₃ CCCH ₂ , Bu], [RA10567; H, F, F, Cl, CH ₃ CCCH ₂ , i-Bu], [RA10568; H, F, F, Cl, CH ₃ CCCH ₂ , t-Bu], [RA10569; H, F, F, Cl
, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA10570; H, F, F, Cl, CH ₃ CCCH ₂ , Ph], [RA10571; H, F, F, Cl, CH ₃ CCCH ₂ , Bn], [RA10572; H, F, F, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RA10573; H, F, F, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA10574; H, F, F , Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA10575; H, F, F, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RA10576; H, F, F, Cl, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA10577; H, F, Cl, H, CH ₃ CCCH ₂ , Me], [RA10578; H, F, Cl, H, CH ₃ CCCH ₂ , Et], [RA10579; H, F, Cl, H, CH ₃ CCCH ₂ , Pr], [RA10580; H, F, Cl, H, CH ₃ CCCH ₂ , i-Pr], [RA10581; H, F, Cl, H, CH ₃ CCCH ₂ , c-Pr], [RA10582; H, F, Cl, H, CH ₃ CCCH ₂ , Bu], [RA10583; H, F, Cl, H, CH ₃ CCCH ₂ , i-Bu], [RA10584; H , F, Cl, H, CH ₃ CCCH ₂ , t-Bu], [RA10585; H, F, Cl, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA10586; H, F, Cl, H, CH ₃ CCCH ₂ , Ph], [RA10587; H, F, Cl, H, CH ₃ CCCH ₂ , Bn], [RA10588; H, F, Cl, H, CH ₃ CCCH ₂ , CF ₃ ], [RA10589; H, F, Cl, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA10590; H, F, Cl, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA10591; H, F, Cl, H, CH ₃ CCCH ₂ , CF ₂ H], [RA10592; H, F, Cl, H, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA10593; H, F, Cl, Cl, CH ₃ CCCH ₂ , Me], [RA10594; H, F, Cl, Cl, CH ₃ CCCH ₂ , Et], [RA10595; H, F, Cl, Cl, CH ₃ CCCH ₂ , Pr], [RA10596; H, F, Cl, Cl, CH ₃ CCCH ₂ , i-Pr], [RA10597; H, F, Cl, Cl, CH ₃ CCCH ₂ , c-Pr], [RA10598; H, F, Cl, Cl, CH ₃ CCCH ₂ , Bu], [RA10599; H, F, Cl, Cl, CH ₃ CCCH ₂ , i-Bu], [RA10600; H, F, Cl, Cl , CH ₃ CCCH ₂ , t-Bu],

[RA10601; H, F, Cl, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RA10602; H, F, Cl, Cl, CH ₃ CCCH ₂ , Ph], [RA10603; H, F, Cl, Cl, CH ₃ CCCH ₂ , Bn], [RA10604; H, F, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RA10605; H, F, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RA10606; H, F, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RA10607; H, F, Cl, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RA10608; H, F, Cl, Cl, CH ₃ CCCH ₂ , CF ₂ HCH ₂ ], [RA10609; H, F, Me, H, c-PrCH ₂ , Me], [RA10610; H, F, Me, H, c-PrCH ₂ , Et], [RA10611; H, F, Me, H, c-PrCH ₂ , Pr], [RA10612; H, F, Me, H, c-PrCH ₂ , i-Pr], [RA10613; H, F, Me, H, c-PrCH ₂ , c-Pr], [RA10614; H, F, Me, H, c-PrCH ₂ , Bu], [RA10615; H, F, Me, H, c-PrCH ₂ , i-Bu], [RA10616; H, F, Me, H, c-PrCH ₂ , t-Bu], [RA10617; H, F, Me, H, c-PrCH ₂ , c-PrCH ₂ ], [ RA10618; H, F, Me, H, c-PrCH ₂ , Ph], [RA10619; H, F, Me, H, c-PrCH ₂ , Bn], [RA10620; H, F, Me, H, c- PrCH ₂ , CF ₃ ], [RA10621; H, F, Me, H, c-PrCH ₂ , CF ₃ CH ₂ ], [RA10622; H, F, Me, H, c-PrCH ₂ , CF ₃ CF ₂ ] , [RA10623; H, F, Me, H, c-PrCH ₂ , CF ₂ H], [RA10624; H, F, Me, H, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA10625; H, F , Me, Me, c-PrCH ₂ , Me], [RA10626; H, F, Me, Me, c-PrCH ₂ , Et], [RA10627; H, F, Me, Me, c-PrCH ₂ , Pr] , [RA10628; H, F, Me , Me, c-PrCH ₂ , i-Pr], [RA10629; H, F, Me, Me, c-PrCH ₂ , c-Pr], [RA10630; H, F, Me, Me, c-PrCH ₂ , Bu], [RA10631; H, F, Me, Me, c-PrCH ₂ , i-Bu], [RA10632; H, F, Me, Me, c-PrCH ₂ , t-Bu], [RA10633; H, F, Me, Me, c-PrCH ₂ , c-PrCH ₂ ], [RA10634; H, F, Me, Me, c-PrCH ₂ , Ph], [RA10635; H, F, Me, Me, c-PrCH _{2, Bn], [RA10636;} H, F, Me, Me, c-PrCH 2, CF 3], [RA10637; H, F, Me, Me, c-PrCH 2, CF 3 CH 2], [RA10638; H, F, Me, Me, c-PrCH ₂ , CF ₃ CF ₂ ], [RA10639; H, F, Me, Me, c-PrCH ₂ , CF ₂ H], [RA10640; H, F, Me, Me , c-PrCH ₂ , CF ₂ HCH ₂ ], [RA10641; H, F, Me, Et, c-PrCH ₂ , Me], [RA10642; H, F, Me, Et, c-PrCH ₂ , Et], [RA10643; H, F, Me, Et, c-PrCH ₂ , Pr], [RA10644; H, F, Me, Et, c-PrCH ₂ , i-Pr], [RA10645; H, F, Me, Et , c-PrCH ₂ , c-Pr], [RA10646; H, F, Me, Et, c-PrCH ₂ , Bu], [RA10647; H, F, Me, Et, c-PrCH ₂ , i-Bu] , [RA10648; H, F, Me, Et, c-PrCH ₂ , t-Bu], [RA10649; H, F, Me, Et, c-PrCH ₂ , c-PrCH ₂ ], [RA10650; H, F , Me, Et, c-PrCH ₂ , Ph], [RA10651; H, F, Me, Et, c-PrCH ₂ , Bn], [RA10652; H, F, Me, Et, c-PrCH ₂ , CF ₃ ], [RA10653; H, F, Me, Et, c-PrCH ₂ , CF ₃ CH ₂ ], [RA10654; H, F, Me, Et, c-PrCH ₂ , CF ₃ CF ₂ ], [RA10655; H , F, Me, Et, c-PrCH ₂ , CF ₂ H], [RA106 56; H, F, Me, Et, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA10657; H, F, Me, F, c-PrCH ₂ , Me], [RA10658; H, F, Me, F , c-PrCH ₂ , Et], [RA10659; H, F, Me, F, c-PrCH ₂ , Pr], [RA10660; H, F, Me, F, c-PrCH ₂ , i-Pr], [ RA10661; H, F, Me, F, c-PrCH ₂ , c-Pr], [RA10662; H, F, Me, F, c-PrCH ₂ , Bu], [RA10663; H, F, Me, F, c-PrCH ₂ , i-Bu], [RA10664; H, F, Me, F, c-PrCH ₂ , t-Bu], [RA10665; H, F, Me, F, c-PrCH ₂ , c-PrCH ₂ ], [RA10666; H, F, Me, F, c-PrCH ₂ , Ph], [RA10667; H, F, Me, F, c-PrCH ₂ , Bn], [RA10668; H, F, Me, F, c-PrCH ₂ , CF ₃ ], [RA10669; H, F, Me, F, c-PrCH ₂ , CF ₃ CH ₂ ], [RA10670; H, F, Me, F, c-PrCH ₂ , CF ₃ CF ₂ ], [RA10671; H, F, Me, F, c-PrCH ₂ , CF ₂ H], [RA10672; H, F, Me, F, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA10673 ; H, F, Me, Cl, c-PrCH ₂ , Me], [RA10674; H, F, Me, Cl, c-PrCH ₂ , Et], [RA10675; H, F, Me, Cl, c-PrCH ₂ , Pr], [RA10676; H, F, Me, Cl, c-PrCH ₂ , i-Pr], [RA10677; H, F, Me, Cl, c-PrCH ₂ , c-Pr], [RA10678; H, F, Me, Cl, c-PrCH ₂ , Bu], [RA10679; H, F, Me, Cl, c-PrCH ₂ , i-Bu], [RA10680; H, F, Me, Cl, c- PrCH ₂ , t-Bu], [RA10681; H, F, Me, Cl, c-PrCH ₂ , c-PrCH ₂ ], [RA10682; H, F, Me, Cl, c-PrCH ₂ , Ph], [ RA10683; H, F, Me, Cl, c-PrCH ₂ , Bn], [RA10684; H, F, Me, Cl, c-PrCH ₂ , CF ₃ ], [RA10685; H, F, Me, Cl, c-PrCH ₂ , CF ₃ CH ₂ ], [RA10686; H, F, Me, Cl, c-PrCH ₂ , CF ₃ CF ₂ ], [ RA10687; H, F, Me, Cl, c-PrCH ₂ , CF ₂ H], [RA10688; H, F, Me, Cl, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA10689; H, F, Et , H, c-PrCH ₂ , Me], [RA10690; H, F, Et, H, c-PrCH ₂ , Et], [RA10691; H, F, Et, H, c-PrCH ₂ , Pr], [ RA10692; H, F, Et, H, c-PrCH ₂ , i-Pr], [RA10693; H, F, Et, H, c-PrCH ₂ , c-Pr], [RA10694; H, F, Et, H, c-PrCH ₂ , Bu], [RA10695; H, F, Et, H, c-PrCH ₂ , i-Bu], [RA10696; H, F, Et, H, c-PrCH ₂ , t-Bu ], [RA10697; H, F, Et, H, c-PrCH ₂ , c-PrCH ₂ ], [RA10698; H, F, Et, H, c-PrCH ₂ , Ph], [RA10699; H, F, Et, H, c-PrCH ₂ , Bn], [RA10700; H, F, Et, H, c-PrCH ₂ , CF ₃ ], [RA10701; H, F, Et, H, c-PrCH ₂ , CF ₃ CH ₂ ], [RA10702; H, F, Et, H, c-PrCH ₂ , CF ₃ CF ₂ ], [RA10703; H, F, Et, H, c-PrCH ₂ , CF ₂ H], [RA10704; H, F, Et, H, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA10705; H, F, Et, F, c-PrCH ₂ , Me], [RA10706; H, F, Et, F, c -PrCH ₂ , Et], [RA10707; H, F, Et, F, c-PrCH ₂ , Pr], [RA10708; H, F, Et, F, c-PrCH ₂ , i-Pr], [RA10709; H, F, Et, F, c-PrCH ₂ , c-Pr], [RA10710; H, F, Et, F, c-PrCH ₂ , Bu], [RA10711; H, F, Et, F, c- PrCH ₂ , i-Bu], [RA10712; H, F, Et, F, c-PrCH ₂ , t-Bu], [RA1071 3; H, F, Et, F, c-PrCH ₂ , c-PrCH ₂ ], [RA10714; H, F, Et, F, c-PrCH ₂ , Ph], [RA10715; H, F, Et, F , c-PrCH ₂ , Bn], [RA10716; H, F, Et, F, c-PrCH ₂ , CF ₃ ], [RA10717; H, F, Et, F, c-PrCH ₂ , CF ₃ CH ₂ ] , [RA10718; H, F, Et, F, c-PrCH ₂ , CF ₃ CF ₂ ], [RA10719; H, F, Et, F, c-PrCH ₂ , CF ₂ H], [RA10720; H, F , Et, F, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA10721; H, F, Et, Cl, c-PrCH ₂ , Me], [RA10722; H, F, Et, Cl, c-PrCH ₂ , Et], [RA10723; H, F, Et, Cl, c-PrCH ₂ , Pr], [RA10724; H, F, Et, Cl, c-PrCH ₂ , i-Pr], [RA10725; H, F , Et, Cl, c-PrCH 2, c-Pr], [RA10726; H, F, Et, Cl, c-PrCH 2, Bu], [RA10727; H, F, Et, Cl, c-PrCH 2, i-Bu], [RA10728; H, F, Et, Cl, c-PrCH ₂ , t-Bu], [RA10729; H, F, Et, Cl, c-PrCH ₂ , c-PrCH ₂ ], [RA10730 ; H, F, Et, Cl, c-PrCH ₂ , Ph], [RA10731; H, F, Et, Cl, c-PrCH ₂ , Bn], [RA10732; H, F, Et, Cl, c-PrCH ₂ , CF ₃ ], [RA10733; H, F, Et, Cl, c-PrCH ₂ , CF ₃ CH ₂ ], [RA10734; H, F, Et, Cl, c-PrCH ₂ , CF ₃ CF ₂ ], [RA10735; H, F, Et, Cl, c-PrCH ₂ , CF ₂ H], [RA10736; H, F, Et, Cl, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA10737; H, F, F, H, c-PrCH ₂ , Me], [RA10738; H, F, F, H, c-PrCH ₂ , Et], [RA10739; H, F, F, H, c-PrCH ₂ , Pr], [RA10740; H, F, F, H, c-PrCH ₂ , i-Pr], [RA10741; H, F, F, H, c-PrCH ₂ , c-Pr], [RA10742; H, F, F, H, c-PrCH ₂ , Bu], [RA10743; H, F, F, H, c-PrCH ₂ , i-Bu], [RA10744; H, F, F, H, c-PrCH ₂ , t-Bu], [RA10745; H, F, F, H, c-PrCH ₂ , c-PrCH ₂ ], [ RA10746; H, F, F, H, c-PrCH ₂ , Ph], [RA10747; H, F, F, H, c-PrCH ₂ , Bn], [RA10748; H, F, F, H, c- PrCH ₂ , CF ₃ ], [RA10749; H, F, F, H, c-PrCH ₂ , CF ₃ CH ₂ ], [RA10750; H, F, F, H, c-PrCH ₂ , CF ₃ CF ₂ ] , [RA10751; H, F, F, H, c-PrCH ₂ , CF ₂ H], [RA10752; H, F, F, H, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA10753; H, F , F, F, c-PrCH ₂ , Me], [RA10754; H, F, F, F, c-PrCH ₂ , Et], [RA10755; H, F, F, F, c-PrCH ₂ , Pr] , [RA10756; H, F, F, F, c-PrCH ₂ , i-Pr], [RA10757; H, F, F, F, c-PrCH ₂ , c-Pr], [RA10758; H, F, F, F, c-PrCH ₂ , Bu], [RA10759; H, F, F, F, c-PrCH ₂ , i-Bu], [RA10760; H, F, F, F, c-PrCH ₂ , t -Bu], [RA10761; H, F, F, F, c-PrCH ₂ , c-PrCH ₂ ], [RA10762; H, F, F, F, c-PrCH ₂ , Ph], [RA10763; H, F, F, F, c-PrCH ₂ , Bn], [RA10764; H, F, F, F, c-PrCH ₂ , CF ₃ ], [RA10765; H, F, F, F, c-PrCH ₂ , CF ₃ CH ₂ ], [RA10766; H, F, F, F, c-PrCH ₂ , CF ₃ CF ₂ ], [RA10767; H, F, F, F, c-PrCH ₂ , CF ₂ H], [ RA10768; H, F, F, F, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA10769; H, F, F, Cl, c-PrCH ₂ , Me], [RA10770; H, F, F, Cl , c -PrCH ₂ , Et], [RA10771; H, F, F, Cl, c-PrCH ₂ , Pr], [RA10772; H, F, F, Cl, c-PrCH ₂ , i-Pr], [RA10773; H, F, F, Cl, c-PrCH ₂ , c-Pr], [RA10774; H, F, F, Cl, c-PrCH ₂ , Bu], [RA10775; H, F, F, Cl, c- PrCH ₂ , i-Bu], [RA10776; H, F, F, Cl, c-PrCH ₂ , t-Bu], [RA10777; H, F, F, Cl, c-PrCH ₂ , c-PrCH ₂ ] , [RA10778; H, F, F, Cl, c-PrCH ₂ , Ph], [RA10779; H, F, F, Cl, c-PrCH ₂ , Bn], [RA10780; H, F, F, Cl, c-PrCH ₂ , CF ₃ ], [RA10781; H, F, F, Cl, c-PrCH ₂ , CF ₃ CH ₂ ], [RA10782; H, F, F, Cl, c-PrCH ₂ , CF ₃ CF ₂ ], [RA10783; H, F, F, Cl, c-PrCH ₂ , CF ₂ H], [RA10784; H, F, F, Cl, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA10785; H , F, Cl, H, c-PrCH ₂ , Me], [RA10786; H, F, Cl, H, c-PrCH ₂ , Et], [RA10787; H, F, Cl, H, c-PrCH ₂ , Pr], [RA10788; H, F, Cl, H, c-PrCH ₂ , i-Pr], [RA10789; H, F, Cl, H, c-PrCH ₂ , c-Pr], [RA10790; H, F, Cl, H, c-PrCH ₂ , Bu], [RA10791; H, F, Cl, H, c-PrCH ₂ , i-Bu], [RA10792; H, F, Cl, H, c-PrCH ₂ , t-Bu], [RA10793; H, F, Cl, H, c-PrCH ₂ , c-PrCH ₂ ], [RA10794; H, F, Cl, H, c-PrCH ₂ , Ph], [RA10795; H, F, Cl, H, c-PrCH ₂ , Bn], [RA10796; H, F, Cl, H, c-PrCH ₂ , CF ₃ ], [RA10797; H, F, Cl, H, c-PrCH ₂ , CF ₃ CH ₂ ], [RA10798; H, F, Cl, H, c-PrCH ₂ , CF ₃ CF ₂ ], [RA10799; H , F, Cl, H, c-PrCH ₂ , CF ₂ H], [RA10800; H, F, Cl, H, c-PrCH ₂ , CF ₂ HCH ₂ ],

[RA10801; H, F, Cl, Cl, c-PrCH ₂ , Me], [RA10802; H, F, Cl, Cl, c-PrCH ₂ , Et], [RA10803; H, F, Cl, Cl, c -PrCH ₂ , Pr], [RA10804; H, F, Cl, Cl, c-PrCH ₂ , i-Pr], [RA10805; H, F, Cl, Cl, c-PrCH ₂ , c-Pr], [ RA10806; H, F, Cl, Cl, c-PrCH ₂ , Bu], [RA10807; H, F, Cl, Cl, c-PrCH ₂ , i-Bu], [RA10808; H, F, Cl, Cl, c-PrCH ₂ , t-Bu], [RA10809; H, F, Cl, Cl, c-PrCH ₂ , c-PrCH ₂ ], [RA10810; H, F, Cl, Cl, c-PrCH ₂ , Ph] , [RA10811; H, F, Cl, Cl, c-PrCH ₂ , Bn], [RA10812; H, F, Cl, Cl, c-PrCH ₂ , CF ₃ ], [RA10813; H, F, Cl, Cl , c-PrCH ₂ , CF ₃ CH ₂ ], [RA10814; H, F, Cl, Cl, c-PrCH ₂ , CF ₃ CF ₂ ], [RA10815; H, F, Cl, Cl, c-PrCH ₂ , CF ₂ H], [RA10816; H, F, Cl, Cl, c-PrCH ₂ , CF ₂ HCH ₂ ], [RA10817; H, F, Me, H, Bn, Me], [RA10818; H, F, Me, H, Bn, Et], [RA10819; H, F, Me, H, Bn, Pr], [RA10820; H, F, Me, H, Bn, i-Pr], [RA10821; H, F, Me, H, Bn, c-Pr], [RA10822; H, F, Me, H, Bn, Bu], [RA10823; H, F, Me, H, Bn, i-Bu], [RA10824; H, F, Me, H, Bn, t-Bu], [RA10825; H, F, Me, H, Bn, c-PrCH ₂ ], [RA10826; H, F, Me, H, Bn, Ph], [RA10827 ; H, F, Me, H, Bn, Bn], [RA10828; H, F, Me, H, Bn, CF ₃ ], [RA10829; H, F, Me, H, Bn, CF ₃ CH ₂ ], [RA10830; H, F, Me, H, Bn, CF ₃ CF ₂ ], [RA10831; H, F, Me, H, Bn, CF ₂ H], [RA10832; H, F , Me, H, Bn, CF ₂ HCH ₂ ], [RA10833; H, F, Me, Me, Bn, Me], [RA10834; H, F, Me, Me, Bn, Et], [RA10835; H, F, Me, Me, Bn, Pr], [RA10836; H, F, Me, Me, Bn, i-Pr], [RA10837; H, F, Me, Me, Bn, c-Pr], [RA10838; H, F, Me, Me, Bn, Bu], [RA10839; H, F, Me, Me, Bn, i-Bu], [RA10840; H, F, Me, Me, Bn, t-Bu], [ RA10841; H, F, Me, Me, Bn, c-PrCH ₂ ], [RA10842; H, F, Me, Me, Bn, Ph], [RA10843; H, F, Me, Me, Bn, Bn], [RA10844; H, F, Me, Me, Bn, CF ₃ ], [RA10845; H, F, Me, Me, Bn, CF ₃ CH ₂ ], [RA10846; H, F, Me, Me, Bn, CF ₃ CF ₂ ], [RA10847; H, F, Me, Me, Bn, CF ₂ H], [RA10848; H, F, Me, Me, Bn, CF ₂ HCH ₂ ], [RA10849; H, F, Me , Et, Bn, Me], [RA10850; H, F, Me, Et, Bn, Et], [RA10851; H, F, Me, Et, Bn, Pr], [RA10852; H, F, Me, Et , Bn, i-Pr], [RA10853; H, F, Me, Et, Bn, c-Pr], [RA10854; H, F, Me, Et, Bn, Bu], [RA10855; H, F, Me , Et, Bn, i-Bu], [RA10856; H, F, Me, Et, Bn, t-Bu], [RA10857; H, F, Me, Et, Bn, c-PrCH ₂ ], [RA10858; H, F, Me, Et, Bn, Ph], [RA10859; H, F, Me, Et, Bn, Bn], [RA10860; H, F, Me, Et, Bn, CF ₃ ], [RA10861; H , F, Me, Et, Bn, CF ₃ CH ₂ ], [RA10862; H, F, Me, Et, Bn, CF ₃ CF ₂ ], [RA10863; H, F, Me, Et, Bn, CF ₂ H ], [RA10864; H, F, Me, Et, Bn, CF ₂ HCH ₂ ], [RA10865; H, F, Me, F, Bn, Me], [RA10866; H, F, Me, F, Bn, Et], [R A10867; H, F, Me, F, Bn, Pr], [RA10868; H, F, Me, F, Bn, i-Pr], [RA10869; H, F, Me, F, Bn, c-Pr] , [RA10870; H, F, Me, F, Bn, Bu], [RA10871; H, F, Me, F, Bn, i-Bu], [RA10872; H, F, Me, F, Bn, t- Bu], [RA10873; H, F, Me, F, Bn, c-PrCH ₂ ], [RA10874; H, F, Me, F, Bn, Ph], [RA10875; H, F, Me, F, Bn , Bn], [RA10876; H, F, Me, F, Bn, CF ₃ ], [RA10877; H, F, Me, F, Bn, CF ₃ CH ₂ ], [RA10878; H, F, Me, F , Bn, CF ₃ CF ₂ ], [RA10879; H, F, Me, F, Bn, CF ₂ H], [RA10880; H, F, Me, F, Bn, CF ₂ HCH ₂ ], [RA10881; H , F, Me, Cl, Bn, Me], [RA10882; H, F, Me, Cl, Bn, Et], [RA10883; H, F, Me, Cl, Bn, Pr], [RA10884; H, F , Me, Cl, Bn, i-Pr], [RA10885; H, F, Me, Cl, Bn, c-Pr], [RA10886; H, F, Me, Cl, Bn, Bu], [RA10887; H , F, Me, Cl, Bn, i-Bu], [RA10888; H, F, Me, Cl, Bn, t-Bu], [RA10889; H, F, Me, Cl, Bn, c-PrCH ₂ ] , [RA10890; H, F, Me, Cl, Bn, Ph], [RA10891; H, F, Me, Cl, Bn, Bn], [RA10892; H, F, Me, Cl, Bn, CF ₃ ], [RA10893; H, F, Me, Cl, Bn, CF ₃ CH ₂ ], [RA10894; H, F, Me, Cl, Bn, CF ₃ CF ₂ ], [RA10895; H, F, Me, Cl, Bn , CF ₂ H], [RA10896; H, F, Me, Cl, Bn, CF ₂ HCH ₂ ], [RA10897; H, F, Et, H, Bn, Me], [RA10898; H, F, Et, H, Bn, Et], [RA10899; H, F, Et, H, Bn, Pr], [RA10900; H, F, Et, H, Bn, i-Pr], [RA10901; H, F, Et, H, Bn, c-Pr], [RA10902; H, F, Et, H, Bn, Bu], [RA10903; H, F, Et, H, Bn, i-Bu], [RA10904; H, F, Et, H, Bn, t-Bu], [RA10905; H, F, Et, H, Bn, c-PrCH ₂ ], [RA10906; H, F, Et, H, Bn, Ph], [RA10907; H, F, Et, H, Bn, Bn], [RA10908; H , F, Et, H, Bn, CF ₃ ], [RA10909; H, F, Et, H, Bn, CF ₃ CH ₂ ], [RA10910; H, F, Et, H, Bn, CF ₃ CF ₂ ] , [RA10911; H, F, Et, H, Bn, CF ₂ H], [RA10912; H, F, Et, H, Bn, CF ₂ HCH ₂ ], [RA10913; H, F, Et, F, Bn , Me], [RA10914; H, F, Et, F, Bn, Et], [RA10915; H, F, Et, F, Bn, Pr], [RA10916; H, F, Et, F, Bn, i -Pr], [RA10917; H, F, Et, F, Bn, c-Pr], [RA10918; H, F, Et, F, Bn, Bu], [RA10919; H, F, Et, F, Bn , i-Bu], [RA10920; H, F, Et, F, Bn, t-Bu], [RA10921; H, F, Et, F, Bn, c-PrCH ₂ ], [RA10922; H, F, Et, F, Bn, Ph], [RA10923; H, F, Et, F, Bn, Bn], [RA10924; H, F, Et, F, Bn, CF ₃ ], [RA10925; H, F, Et , F, Bn, CF ₃ CH ₂ ], [RA10926; H, F, Et, F, Bn, CF ₃ CF ₂ ], [RA10927; H, F, Et, F, Bn, CF ₂ H], [RA10928 ; H, F, Et, F, Bn, CF ₂ HCH ₂ ], [RA10929; H, F, Et, Cl, Bn, Me], [RA10930; H, F, Et, Cl, Bn, Et], [ RA10931; H, F, Et, Cl, Bn, Pr], [RA10932; H, F, Et, Cl, Bn, i-Pr], [RA10933; H, F, Et, Cl, Bn, c-Pr] , [RA10934; H, F, Et, Cl, Bn, Bu], [RA10935; H, F, Et, Cl, Bn, i-Bu], [RA10936; H, F, Et, Cl, Bn, t- Bu], [RA10937; H, F, Et, Cl, Bn, c-PrCH ₂ ] , [RA10938; H, F, Et, Cl, Bn, Ph], [RA10939; H, F, Et, Cl, Bn, Bn], [RA10940; H, F, Et, Cl, Bn, CF ₃ ], [RA10941; H, F, Et, Cl, Bn, CF ₃ CH ₂ ], [RA10942; H, F, Et, Cl, Bn, CF ₃ CF ₂ ], [RA10943; H, F, Et, Cl, Bn , CF ₂ H], [RA10944; H, F, Et, Cl, Bn, CF ₂ HCH ₂ ], [RA10945; H, F, F, H, Bn, Me], [RA10946; H, F, F, H, Bn, Et], [RA10947; H, F, F, H, Bn, Pr], [RA10948; H, F, F, H, Bn, i-Pr], [RA10949; H, F, F, H, Bn, c-Pr], [RA10950; H, F, F, H, Bn, Bu], [RA10951; H, F, F, H, Bn, i-Bu], [RA10952; H, F, F, H, Bn, t-Bu], [RA10953; H, F, F, H, Bn, c-PrCH ₂ ], [RA10954; H, F, F, H, Bn, Ph], [RA10955; H , F, F, H, Bn, Bn], [RA10956; H, F, F, H, Bn, CF ₃ ], [RA10957; H, F, F, H, Bn, CF ₃ CH ₂ ], [RA10958 ; H, F, F, H, Bn, CF ₃ CF ₂ ], [RA10959; H, F, F, H, Bn, CF ₂ H], [RA10960; H, F, F, H, Bn, CF ₂ HCH ₂ ], [RA10961; H, F, F, F, Bn, Me], [RA10962; H, F, F, F, Bn, Et], [RA10963; H, F, F, F, Bn, Pr ], [RA10964; H, F, F, F, Bn, i-Pr], [RA10965; H, F, F, F, Bn, c-Pr], [RA10966; H, F, F, F, Bn , Bu], [RA10967; H, F, F, F, Bn, i-Bu], [RA10968; H, F, F, F, Bn, t-Bu], [RA10969; H, F, F, F , Bn, c-PrCH ₂ ], [RA10970; H, F, F, F, Bn, Ph], [RA10971; H, F, F, F, Bn, Bn], [RA10972; H, F, F, F, Bn, CF ₃ ], [RA10973; H, F, F, F, Bn, CF ₃ CH ₂ ], [RA10974; H, F, F, F , Bn, CF ₃ CF ₂ ], [RA10975; H, F, F, F, Bn, CF ₂ H], [RA10976; H, F, F, F, Bn, CF ₂ HCH ₂ ], [RA10977; H , F, F, Cl, Bn, Me], [RA10978; H, F, F, Cl, Bn, Et], [RA10979; H, F, F, Cl, Bn, Pr], [RA10980; H, F , F, Cl, Bn, i-Pr], [RA10981; H, F, F, Cl, Bn, c-Pr], [RA10982; H, F, F, Cl, Bn, Bu], [RA10983; H , F, F, Cl, Bn, i-Bu], [RA10984; H, F, F, Cl, Bn, t-Bu], [RA10985; H, F, F, Cl, Bn, c-PrCH ₂ ] , [RA10986; H, F, F, Cl, Bn, Ph], [RA10987; H, F, F, Cl, Bn, Bn], [RA10988; H, F, F, Cl, Bn, CF ₃ ], [RA10989; H, F, F, Cl, Bn, CF ₃ CH ₂ ], [RA10990; H, F, F, Cl, Bn, CF ₃ CF ₂ ], [RA10991; H, F, F, Cl, Bn , CF ₂ H], [RA10992; H, F, F, Cl, Bn, CF ₂ HCH ₂ ], [RA10993; H, F, Cl, H, Bn, Me], [RA10994; H, F, Cl, H, Bn, Et], [RA10995; H, F, Cl, H, Bn, Pr], [RA10996; H, F, Cl, H, Bn, i-Pr], [RA10997; H, F, Cl, H, Bn, c-Pr], [RA10998; H, F, Cl, H, Bn, Bu], [RA10999; H, F, Cl, H, Bn, i-Bu], [RA11000; H, F, Cl, H, Bn, t-Bu],

[RA11001; H, F, Cl, H, Bn, c-PrCH ₂ ], [RA11002; H, F, Cl, H, Bn, Ph], [RA11003; H, F, Cl, H, Bn, Bn] , [RA11004; H, F, Cl, H, Bn, CF ₃ ], [RA11005; H, F, Cl, H, Bn, CF ₃ CH ₂ ], [RA11006; H, F, Cl, H, Bn, CF ₃ CF ₂ ], [RA11007; H, F, Cl, H, Bn, CF ₂ H], [RA11008; H, F, Cl, H, Bn, CF ₂ HCH ₂ ], [RA11009; H, F, Cl, Cl, Bn, Me], [RA11010; H, F, Cl, Cl, Bn, Et], [RA11011; H, F, Cl, Cl, Bn, Pr], [RA11012; H, F, Cl, Cl, Bn, i-Pr], [RA11013; H, F, Cl, Cl, Bn, c-Pr], [RA11014; H, F, Cl, Cl, Bn, Bu], [RA11015; H, F, Cl, Cl, Bn, i-Bu], [RA11016; H, F, Cl, Cl, Bn, t-Bu], [RA11017; H, F, Cl, Cl, Bn, c-PrCH ₂ ], [RA11018 ; H, F, Cl, Cl, Bn, Ph], [RA11019; H, F, Cl, Cl, Bn, Bn], [RA11020; H, F, Cl, Cl, Bn, CF ₃ ], [RA11021; H, F, Cl, Cl, Bn, CF ₃ CH ₂ ], [RA11022; H, F, Cl, Cl, Bn, CF ₃ CF ₂ ], [RA11023; H, F, Cl, Cl, Bn, CF ₂ H], [RA11024; H, F, Cl, Cl, Bn, CF ₂ HCH ₂ ], [RA11025; H, F, Me, H, Ph, Me], [RA11026; H, F, Me, H, Ph , Et], [RA11027; H, F, Me, H, Ph, Pr], [RA11028; H, F, Me, H, Ph, i-Pr], [RA11029; H, F, Me, H, Ph , c-Pr], [RA11030; H, F, Me, H, Ph, Bu], [RA11031; H, F, Me, H, Ph, i-Bu], [RA11032; H, F, Me, H , Ph, t-Bu], [RA11033; H, F, Me, H, Ph, c-PrCH ₂ ], [RA11034; H, F, Me, H, Ph, Ph], [RA11035; H, F, Me, H, Ph, Bn], [RA11036 ; H, F, Me, H, Ph, CF ₃ ], [RA11037; H, F, Me, H, Ph, CF ₃ CH ₂ ], [RA11038; H, F, Me, H, Ph, CF ₃ CF ₂ ], [RA11039; H, F, Me, H, Ph, CF ₂ H], [RA11040; H, F, Me, H, Ph, CF ₂ HCH ₂ ], [RA11041; H, F, Me, Me , Ph, Me], [RA11042; H, F, Me, Me, Ph, Et], [RA11043; H, F, Me, Me, Ph, Pr], [RA11044; H, F, Me, Me, Ph , i-Pr], [RA11045; H, F, Me, Me, Ph, c-Pr], [RA11046; H, F, Me, Me, Ph, Bu], [RA11047; H, F, Me, Me , Ph, i-Bu], [RA11048; H, F, Me, Me, Ph, t-Bu], [RA11049; H, F, Me, Me, Ph, c-PrCH ₂ ], [RA11050; H, F, Me, Me, Ph, Ph], [RA11051; H, F, Me, Me, Ph, Bn], [RA11052; H, F, Me, Me, Ph, CF ₃ ], [RA11053; H, F , Me, Me, Ph, CF ₃ CH ₂ ], [RA11054; H, F, Me, Me, Ph, CF ₃ CF ₂ ], [RA11055; H, F, Me, Me, Ph, CF ₂ H], [RA11056; H, F, Me, Me, Ph, CF ₂ HCH ₂ ], [RA11057; H, F, Me, Et, Ph, Me], [RA11058; H, F, Me, Et, Ph, Et] , [RA11059; H, F, Me, Et, Ph, Pr], [RA11060; H, F, Me, Et, Ph, i-Pr], [RA11061; H, F, Me, Et, Ph, c- Pr], [RA11062; H, F, Me, Et, Ph, Bu], [RA11063; H, F, Me, Et, Ph, i-Bu], [RA11064; H, F, Me, Et, Ph, t-Bu], [RA11065; H, F, Me, Et, Ph, c-PrCH ₂ ], [RA11066; H, F, Me, Et, Ph, Ph], [RA11067; H, F, Me, Et , Ph, Bn], [RA11068; H, F, Me, Et, Ph, CF ₃ ], [RA11069; H, F, Me, Et, Ph, CF ₃ CH ₂ ], [RA11070; H, F, Me , Et, Ph, CF ₃ CF ₂ ], [RA11071; H, F, Me, Et, Ph, CF ₂ H], [RA11072; H, F, Me, Et, Ph, CF ₂ HCH ₂ ], [RA11073; H, F, Me , F, Ph, Me], [RA11074; H, F, Me, F, Ph, Et], [RA11075; H, F, Me, F, Ph, Pr], [RA11076; H, F, Me, F , Ph, i-Pr], [RA11077; H, F, Me, F, Ph, c-Pr], [RA11078; H, F, Me, F, Ph, Bu], [RA11079; H, F, Me , F, Ph, i-Bu], [RA11080; H, F, Me, F, Ph, t-Bu], [RA11081; H, F, Me, F, Ph, c-PrCH ₂ ], [RA11082; H, F, Me, F, Ph, Ph], [RA11083; H, F, Me, F, Ph, Bn], [RA11084; H, F, Me, F, Ph, CF ₃ ], [RA11085; H , F, Me, F, Ph, CF ₃ CH ₂ ], [RA11086; H, F, Me, F, Ph, CF ₃ CF ₂ ], [RA11087; H, F, Me, F, Ph, CF ₂ H ], [RA11088; H, F, Me, F, Ph, CF ₂ HCH ₂ ], [RA11089; H, F, Me, Cl, Ph, Me], [RA11090; H, F, Me, Cl, Ph, Et], [RA11091; H, F, Me, Cl, Ph, Pr], [RA11092; H, F, Me, Cl, Ph, i-Pr], [RA11093; H, F, Me, Cl, Ph, c-Pr], [RA11094; H, F, Me, Cl, Ph, Bu], [RA11095; H, F, Me, Cl, Ph, i-Bu], [RA11096; H, F, Me, Cl, Ph, t-Bu], [RA11097; H, F, Me, Cl, Ph, c-PrCH ₂ ], [RA11098; H, F, Me, Cl, Ph, Ph], [RA11099; H, F, Me , Cl, Ph, Bn], [RA11100; H, F, Me, Cl, Ph, CF ₃ ], [RA11101; H, F, Me, Cl, Ph, CF ₃ CH ₂ ], [RA11102; H, F , Me, Cl, Ph, CF ₃ CF ₂ ], [RA11103; H, F, Me, Cl, Ph, CF ₂ H], [RA11104; H, F, Me, Cl, Ph, CF ₂ HCH ₂ ], [RA11105; H, F, Et , H, Ph, Me], [RA11106; H, F, Et, H, Ph, Et], [RA11107; H, F, Et, H, Ph, Pr], [RA11108; H, F, Et, H , Ph, i-Pr], [RA11109; H, F, Et, H, Ph, c-Pr], [RA11110; H, F, Et, H, Ph, Bu], [RA11111; H, F, Et , H, Ph, i-Bu], [RA11112; H, F, Et, H, Ph, t-Bu], [RA11113; H, F, Et, H, Ph, c-PrCH ₂ ], [RA11114; H, F, Et, H, Ph, Ph], [RA11115; H, F, Et, H, Ph, Bn], [RA11116; H, F, Et, H, Ph, CF ₃ ], [RA11117; H , F, Et, H, Ph, CF ₃ CH ₂ ], [RA11118; H, F, Et, H, Ph, CF ₃ CF ₂ ], [RA11119; H, F, Et, H, Ph, CF ₂ H ], [RA11120; H, F, Et, H, Ph, CF ₂ HCH ₂ ], [RA11121; H, F, Et, F, Ph, Me], [RA11122; H, F, Et, F, Ph, Et], [RA11123; H, F, Et, F, Ph, Pr], [RA11124; H, F, Et, F, Ph, i-Pr], [RA11125; H, F, Et, F, Ph, c-Pr], [RA11126; H, F, Et, F, Ph, Bu], [RA11127; H, F, Et, F, Ph, i-Bu], [RA11128; H, F, Et, F, Ph, t-Bu], [RA11129; H, F, Et, F, Ph, c-PrCH ₂ ], [RA11130; H, F, Et, F, Ph, Ph], [RA11131; H, F, Et , F, Ph, Bn], [RA11132; H, F, Et, F, Ph, CF ₃ ], [RA11133; H, F, Et, F, Ph, CF ₃ CH ₂ ], [RA11134; H, F , Et, F, Ph, CF ₃ CF ₂ ], [RA11135; H, F, Et, F, Ph, CF ₂ H], [RA11136; H, F, Et, F, Ph, CF ₂ HCH ₂ ], [RA11137; H, F, Et, Cl, Ph, Me], [RA11138; H, F, Et, Cl, Ph, Et], [RA11139; H, F, Et, Cl, Ph, Pr], [RA11140 ; H, F, Et, Cl, Ph, i-Pr], [RA11141; H, F, Et , Cl, Ph, c-Pr], [RA11142; H, F, Et, Cl, Ph, Bu], [RA11143; H, F, Et, Cl, Ph, i-Bu], [RA11144; H, F , Et, Cl, Ph, t-Bu], [RA11145; H, F, Et, Cl, Ph, c-PrCH ₂ ], [RA11146; H, F, Et, Cl, Ph, Ph], [RA11147; H, F, Et, Cl, Ph, Bn], [RA11148; H, F, Et, Cl, Ph, CF ₃ ], [RA11149; H, F, Et, Cl, Ph, CF ₃ CH ₂ ], [ RA11150; H, F, Et, Cl, Ph, CF ₃ CF ₂ ], [RA11151; H, F, Et, Cl, Ph, CF ₂ H], [RA11152; H, F, Et, Cl, Ph, CF ₂ HCH ₂ ], [RA11153; H, F, F, H, Ph, Me], [RA11154; H, F, F, H, Ph, Et], [RA11155; H, F, F, H, Ph, Pr], [RA11156; H, F, F, H, Ph, i-Pr], [RA11157; H, F, F, H, Ph, c-Pr], [RA11158; H, F, F, H, Ph, Bu], [RA11159; H, F, F, H, Ph, i-Bu], [RA11160; H, F, F, H, Ph, t-Bu], [RA11161; H, F, F, H, Ph, c-PrCH ₂ ], [RA11162; H, F, F, H, Ph, Ph], [RA11163; H, F, F, H, Ph, Bn], [RA11164; H, F, F , H, Ph, CF ₃ ], [RA11165; H, F, F, H, Ph, CF ₃ CH ₂ ], [RA11166; H, F, F, H, Ph, CF ₃ CF ₂ ], [RA11167; H, F, F, H, Ph, CF ₂ H], [RA11168; H, F, F, H, Ph, CF ₂ HCH ₂ ], [RA11169; H, F, F, F, Ph, Me], [RA11170; H, F, F, F, Ph, Et], [RA11171; H, F, F, F, Ph, Pr], [RA11172; H, F, F, F, Ph, i-Pr], [RA11173; H, F, F, F, Ph, c-Pr], [RA11174; H, F, F, F, Ph, Bu], [RA11175; H, F, F, F, Ph, i-Bu ], [RA11176; H, F, F, F, Ph, t-Bu], [RA11177; H, F, F, F, Ph, c-PrCH ₂ ], [RA11178; H, F, F, F, Ph, Ph], [RA11179; H, F, F, F, Ph, Bn], [RA11180; H, F, F, F, Ph, CF ₃ ], [RA11181; H, F, F, F, Ph, CF ₃ CH ₂ ], [RA11182; H, F, F, F, Ph, CF ₃ CF ₂ ], [RA11183; H, F, F, F , Ph, CF ₂ H], [RA11184; H, F, F, F, Ph, CF ₂ HCH ₂ ], [RA11185; H, F, F, Cl, Ph, Me], [RA11186; H, F, F, Cl, Ph, Et], [RA11187; H, F, F, Cl, Ph, Pr], [RA11188; H, F, F, Cl, Ph, i-Pr], [RA11189; H, F, F, Cl, Ph, c-Pr], [RA11190; H, F, F, Cl, Ph, Bu], [RA11191; H, F, F, Cl, Ph, i-Bu], [RA11192; H, F, F, Cl, Ph, t-Bu], [RA11193; H, F, F, Cl, Ph, c-PrCH ₂ ], [RA11194; H, F, F, Cl, Ph, Ph], [RA11195 ; H, F, F, Cl, Ph, Bn], [RA11196; H, F, F, Cl, Ph, CF ₃ ], [RA11197; H, F, F, Cl, Ph, CF ₃ CH ₂ ], [RA11198; H, F, F, Cl, Ph, CF ₃ CF ₂ ], [RA11199; H, F, F, Cl, Ph, CF ₂ H], [RA11200; H, F, F, Cl, Ph, CF ₂ HCH ₂ ],

[RA11201; H, F, Cl, H, Ph, Me], [RA11202; H, F, Cl, H, Ph, Et], [RA11203; H, F, Cl, H, Ph, Pr], [RA11204 ; H, F, Cl, H, Ph, i-Pr], [RA11205; H, F, Cl, H, Ph, c-Pr], [RA11206; H, F, Cl, H, Ph, Bu], [RA11207; H, F, Cl, H, Ph, i-Bu], [RA11208; H, F, Cl, H, Ph, t-Bu], [RA11209; H, F, Cl, H, Ph, c -PrCH ₂ ], [RA11210; H, F, Cl, H, Ph, Ph], [RA11211; H, F, Cl, H, Ph, Bn], [RA11212; H, F, Cl, H, Ph, CF ₃ ], [RA11213; H, F, Cl, H, Ph, CF ₃ CH ₂ ], [RA11214; H, F, Cl, H, Ph, CF ₃ CF ₂ ], [RA11215; H, F, Cl , H, Ph, CF ₂ H], [RA11216; H, F, Cl, H, Ph, CF ₂ HCH ₂ ], [RA11217; H, F, Cl, Cl, Ph, Me], [RA11218; H, F, Cl, Cl, Ph, Et], [RA11219; H, F, Cl, Cl, Ph, Pr], [RA11220; H, F, Cl, Cl, Ph, i-Pr], [RA11221; H, F, Cl, Cl, Ph, c-Pr], [RA11222; H, F, Cl, Cl, Ph, Bu], [RA11223; H, F, Cl, Cl, Ph, i-Bu], [RA11224; H, F, Cl, Cl, Ph, t-Bu], [RA11225; H, F, Cl, Cl, Ph, c-PrCH ₂ ], [RA11226; H, F, Cl, Cl, Ph, Ph], [RA11227; H, F, Cl, Cl, Ph, Bn], [RA11228; H, F, Cl, Cl, Ph, CF ₃ ], [RA11229; H, F, Cl, Cl, Ph, CF ₃ CH ₂ ], [RA11230; H, F, Cl, Cl, Ph, CF ₃ CF ₂ ], [RA11231; H, F, Cl, Cl, Ph, CF ₂ H], [RA11232; H, F, Cl, Cl, Ph, CF ₂ HCH ₂ ]

Formula (IV)

In which the combination of R ³¹ , R ³² , R ³³ , R ³⁴ and R ³⁵ is a combination described in any one of the substituent numbers ZA1 to ZA8289 (hereinafter referred to as formula (IV)) In the compounds shown, compounds having substituent numbers ZA1 to ZA8289 are represented as the present compounds RB1 to RB8289, and the present compounds RB1 to RB8289 are collectively represented as the present compound RB). it can.

Here, the substituent numbers ZA1 to ZA8289 are combinations of R ³¹ , R ³² , R ³³ , R ³⁴ and R ^{35 in} the compound represented by the formula (IV) or the compound represented by the formula (V). In the following, it will be referred to as [substituent group number; R ³¹ , R ³² , R ³³ , R ³⁴ , R ³⁵ ].
For example, the substituent number ZA2 represents a combination in which R ³¹ , R ³² , R ³³ and R ³⁴ are hydrogen atoms and R ³⁵ is NHEt.

For example, the present compound RB2 means a compound having a substituent number ZA2 in the compound represented by the formula (IV), and R ³¹ , R ³² , R ³³ and R in the compound represented by the formula (IV). ³⁴ represents a hydrogen atom, and R ³⁵ represents NHEt.

[Substituent number: R ³¹ , R ³² , R ³³ , R ³⁴ , R ³⁵ ]:
[ZA1; H, H, H, H, NHMe], [ZA2; H, H, H, H, NHEt], [ZA3; H, H, H, H, NHPr], [ZA4; H, H, H , H, NHBu], [ZA5; H, H, H, H, NHPen], [ZA6; H, H, H, H, NHHex], [ZA7; H, H, H, H, NH (i-Pr )], [ZA8; H, H, H, H, NH (i-Bu)], [ZA9; H, H, H, H, NH (c-Pr)], [ZA10; H, H, H, H, NH (c-Bu)], [ZA11; H, H, H, H, NH (c-Pen)], [ZA12; H, H, H, H, NH (c-Hex)], [ZA13 ; H, H, H, H, NHCH ₂ (c-Pr)], [ZA14; H, H, H, H, NHCH ₂ (c-Bu)], [ZA15; H, H, H, H, NHCH ₂ (c-Pen)], [ZA16; H, H, H, H, NHCH ₂ (c-Hex)], [ZA17; H, H, H, H, NHCH ₂ F], [ZA18; H, H , H, H, NHCHF ₂ ], [ZA19; H, H, H, H, NHCF ₃ ], [ZA20; H, H, H, H, NH (CH ₂ ) ₂ F], [ZA21; H, H , H, H, NHCH ₂ CHF ₂ ], [ZA22; H, H, H, H, NHCH ₂ CHF ₃ ], [ZA23; H, H, H, H, NH (CH ₂ ) ₃ F], [ZA24 ; H, H, H, H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA25; H, H, H, H, NH (CH ₂ ) ₂ CF ₃ ], [ZA26; H, H, H, H , NHCH ₂ CH (CF ₃ ) ₂ ], [ZA27; H, H, H, H, NHCH ₂ Cl], [ZA28; H, H, H, H, NH (CH ₂ ) ₂ Cl], [ZA29; H, H, H, H, NH (CH ₂ ) ₃ Cl], [ZA30; H, H, H, H, NH (CH ₂ ) ₄ Cl], [ZA31; H, H, H, H, NH ( CH ₂ ) ₅ Cl], [ZA32; H, H, H, H, NHCH ₂ OMe], [ZA33; H, H, H, H, NH (CH ₂ ) ₂ OMe], [ZA34; H, H, H, H, NH (CH ₂ ) ₃ OMe], [ZA35; H, H, H, H, NH (CH ₂ ) ₄ OMe], [ZA36; H, H, H, H, NHCH ₂ OEt], [ ZA37; H, H, H, H, NH (CH ₂ ) ₂ OEt], [ZA38; H, H, H, H , NH (CH ₂ ) ₃ OEt], [ZA39; H, H, H, H, NHCH ₂ OPr], [ZA40; H, H, H, H, NH (CH ₂ ) ₂ OPr], [ZA41; H , H, H, H, NH (CH ₂ ) ₃ OPr], [ZA42; H, H, H, H, NHCH ₂ CN], [ZA43; H, H, H, H, NH (CH ₂ ) ₂ CN ], [ZA44; H, H, H, H, NH (CH ₂ ) ₃ CN], [ZA45; H, H, H, H, NH (CH ₂ ) ₄ CN], [ZA46; H, H, H , H, NH (CH ₂ ) ₅ CN], [ZA47; H, H, H, H, NHCH ₂ CH = CH ₂ ], [ZA48; H, H, H, H, NHCH ₂ C≡CH], [ ZA49; H, H, H, H, NHCH ₂ C≡CCH ₃ ], [ZA50; H, H, H, H, NHCH ₂ Ph], [ZA51; H, H, H, H, NHCH ₂ (2- Py)], [ZA52; H, H, H, H, NHCH ₂ (3-Py)], [ZA53; H, H, H, H, NHCH ₂ (4-Py)], [ZA54; H, H , H, H, NH (CH ₂ ) ₂ Ph], [ZA55; H, H, H, H, NH (CH ₂ ) ₂ (2-Py)], [ZA56; H, H, H, H, NH (CH ₂ ) ₂ (3-Py)], [ZA57; H, H, H, H, NH (CH ₂ ) ₂ (4-Py)], [ZA58; H, H, H, H, NHPh], [ZA59; H, H, H, H, NH (2-Py)], [ZA60; H, H, H, H, NH (3-Py)], [ZA61; H, H, H, H, NH (4-Py)], [ZA62; H, H, H, H, NMe ₂ ], [ZA63; H, H, H, H, NMeEt], [ZA64; H, H, H, H, NMePr], [ZA65; H, H, H, H, NMeBu], [ZA66; H, H, H, H, NMePen], [ZA67; H, H, H, H, NMeHex], [ZA68; H, H, H , H, NMe (i-Pr)], [ZA69; H, H, H, H, NMe (i-Bu)], [ZA70; H, H, H, H, NMe (c-Pr)], [ ZA71; H, H, H, H, NMe (c-Bu)], [ZA72; H, H, H, H, NMe (c-Pen)], [ZA73; H, H, H, H, NMe ( c-Hex)], [ZA74; H, H, H, H, NMeCH ₂ (c-Pr)], [ZA75; H, H , H, H, NMeCH ₂ (c-Bu)], [ZA76; H, H, H, H, NMeCH ₂ (c-Pen)], [ZA77; H, H, H, H, NMeCH ₂ (c- Hex)], [ZA78; H, H, H, H, NMeCH ₂ F], [ZA79; H, H, H, H, NMeCHF ₂ ], [ZA80; H, H, H, H, NMeCF ₃ ], [ZA81; H, H, H, H, NMe (CH ₂ ) ₂ F], [ZA82; H, H, H, H, NMeCH ₂ CHF ₂ ], [ZA83; H, H, H, H, NMeCH ₂ CHF ₃ ], [ZA84; H, H, H, H, NMe (CH ₂ ) ₃ F], [ZA85; H, H, H, H, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA86; H, H, H, H, NMe (CH ₂ ) ₂ CF ₃ ], [ZA87; H, H, H, H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA88; H, H, H, H, NMeCH ₂ Cl], [ZA89; H, H, H, H, NMe (CH ₂ ) ₂ Cl], [ZA90; H, H, H, H, NMe (CH ₂ ) ₃ Cl], [ZA91; H, H, H, H, NMe (CH ₂ ) ₄ Cl], [ZA92; H, H, H, H, NMe (CH ₂ ) ₅ Cl], [ZA93; H, H, H, H, NMeCH ₂ OMe], [ ZA94; H, H, H, H, NMe (CH ₂ ) ₂ OMe], [ZA95; H, H, H, H, NMe (CH ₂ ) ₃ OMe], [ZA96; H, H, H, H, NMe (CH ₂ ) ₄ OMe], [ZA97; H, H, H, H, NMeCH ₂ OEt], [ZA98; H, H, H, H, NMe (CH ₂ ) ₂ OEt], [ZA99; H, H, H, H, NMe (CH ₂ ) ₃ OEt], [ZA100; H, H, H, H, NMeCH ₂ OPr], [ZA101; H, H, H, H, NMe (CH ₂ ) ₂ OPr] , [ZA102; H, H, H, H, NMe (CH ₂ ) ₃ OPr], [ZA103; H, H, H, H, NMeCH ₂ CN], [ZA104; H, H, H, H, NMe ( _{CH 2) 2 CN], [} ZA105; H, H, H, H, NMe (CH 2) 3 CN], [ZA106; H, H, H, H, NMe (CH 2) 4 CN], [ZA107; H, H, H, H, NMe (CH ₂ ) ₅ CN], [ZA10 8; H, H, H, H, NMeCH ₂ CH = CH ₂ ], [ZA109; H, H, H, H, NMeCH ₂ C≡CH], [ZA110; H, H, H, H, NMeCH ₂ C ≡CCH ₃ ], [ZA111; H, H, H, H, NMeCH ₂ Ph], [ZA112; H, H, H, H, NMeCH ₂ (2-Py)], [ZA113; H, H, H, H, NMeCH ₂ (3-Py)], [ZA114; H, H, H, H, NMeCH ₂ (4-Py)], [ZA115; H, H, H, H, NMe (CH ₂ ) ₂ Ph] , [ZA116; H, H, H, H, NMe (CH ₂ ) ₂ (2-Py)], [ZA117; H, H, H, H, NMe (CH ₂ ) ₂ (3-Py)], [ ZA118; H, H, H, H, NMe (CH ₂ ) ₂ (4-Py)], [ZA119; H, H, H, H, NMePh], [ZA120; H, H, H, H, NMe ( 2-Py)], [ZA121; H, H, H, H, NMe (3-Py)], [ZA122; H, H, H, H, NMe (4-Py)], [ZA123; H, H , H, H, NEt ₂ ], [ZA124; H, H, H, H, NEtPr], [ZA125; H, H, H, H, NEtBu], [ZA126; H, H, H, H, NEtPen] , [ZA127; H, H, H, H, NEtHex], [ZA128; H, H, H, H, NEt (i-Pr)], [ZA129; H, H, H, H, NEt (i-Bu )], [ZA130; H, H, H, H, NEt (c-Pr)], [ZA131; H, H, H, H, NEt (c-Bu)], [ZA132; H, H, H, H, NEt (c-Pen)], [ZA133; H, H, H, H, NEt (c-Hex)], [ZA134; H, H, H, H, NEtCH ₂ (c-Pr)], [ ZA135; H, H, H, H, NEtCH ₂ (c-Bu)], [ZA136; H, H, H, H, NEtCH ₂ (c-Pen)], [ZA137; H, H, H, H, NEtCH ₂ (c-Hex)], [ZA138; H, H, H, H, NEtCH ₂ F], [ZA139; H, H, H, H, NEtCHF ₂ ], [ZA140; H, H, H, H , NEtCF ₃ ], [ZA141; H, H, H, H, NEt (CH ₂ ) ₂ F], [ZA142; H, H, H, H, NEtCH ₂ CHF ₂ ], [ZA143; H, H , H, H, NEtCH ₂ CHF ₃ ], [ZA144; H, H, H, H, NEt (CH ₂ ) ₃ F], [ZA145; H, H, H, H, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA146; H, H, H, H, NEt (CH ₂ ) ₂ CF ₃ ], [ZA147; H, H, H, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA148; H, H , H, H, NEtCH ₂ Cl], [ZA149; H, H, H, H, NEt (CH ₂ ) ₂ Cl], [ZA150; H, H, H, H, NEt (CH ₂ ) ₃ Cl], [ZA151; H, H, H, H, NEt (CH ₂ ) ₄ Cl], [ZA152; H, H, H, H, NEt (CH ₂ ) ₅ Cl], [ZA153; H, H, H, H , NEtCH ₂ OMe], [ZA154; H, H, H, H, NEt (CH ₂ ) ₂ OMe], [ZA155; H, H, H, H, NEt (CH ₂ ) ₃ OMe], [ZA156; H , H, H, H, NEt (CH ₂ ) ₄ OMe], [ZA157; H, H, H, H, NEtCH ₂ OEt], [ZA158; H, H, H, H, NEt (CH ₂ ) ₂ OEt ], [ZA159; H, H, H, H, NEt (CH ₂ ) ₃ OEt], [ZA160; H, H, H, H, NEtCH ₂ OPr], [ZA161; H, H, H, H, NEt (CH ₂ ) ₂ OPr], [ZA162; H, H, H, H, NEt (CH ₂ ) ₃ OPr], [ZA163; H, H, H, H, NEtCH ₂ CN], [ZA164; H, H , H, H, NEt (CH ₂ ) ₂ CN], [ZA165; H, H, H, H, NEt (CH ₂ ) ₃ CN], [ZA166; H, H, H, H, NEt (CH ₂ ) ₄ CN], [ZA167; H, H, H, H, NEt (CH ₂ ) ₅ CN], [ZA168; H, H, H, H, NEtCH ₂ CH = CH ₂ ], [ZA169; H, H, H, H, NEtCH ₂ C≡CH], [ZA170; H, H, H, H, NEtCH ₂ C≡CCH ₃ ], [ZA171; H, H, H, H, NEtCH ₂ Ph], [ZA172; H , H, H, H, NEtCH ₂ (2-Py)], [ZA173; H, H, H, H, NEtCH ₂ (3-Py)], [ZA174; H, H, H, H, NEtCH ₂ ( 4-P y)], [ZA175; H, H, H, H, NEt (CH ₂ ) ₂ Ph], [ZA176; H, H, H, H, NEt (CH ₂ ) ₂ (2-Py)], [ZA177 ; H, H, H, H, NEt (CH ₂ ) ₂ (3-Py)], [ZA178; H, H, H, H, NEt (CH ₂ ) ₂ (4-Py)], [ZA179; H , H, H, H, NEtPh], [ZA180; H, H, H, H, NEt (2-Py)], [ZA181; H, H, H, H, NEt (3-Py)], [ZA182 ; H, H, H, H, NEt (4-Py)], [ZA183; H, H, H, H, Pyr], [ZA184; H, H, H, H, Pip], [ZA185; H, H, H, H, Mor], [ZA186; H, H, H, H, OMe], [ZA187; H, H, H, H, OEt], [ZA188; H, H, H, H, OPr] , [ZA189; H, H, H, H, OBu], [ZA190; H, H, H, H, OPen], [ZA191; H, H, H, H, OHex], [ZA192; H, H, H, H, O (i-Pr)], [ZA193; H, H, H, H, O (i-Bu)], [ZA194; H, H, H, H, O (c-Pr)], [ZA195; H, H, H, H, O (c-Bu)], [ZA196; H, H, H, H, O (c-Pen)], [ZA197; H, H, H, H, O (c-Hex)], [ZA198; H, H, H, H, OCH ₂ (c-Pr)], [ZA199; H, H, H, H, OCH ₂ (c-Bu)], [ZA200; H, H, H, H, OCH ₂ (c-Pen)], [ZA201; H, H, H, H, OCH ₂ (c-Hex)], [ZA202; H, H, H, H, OCH ₂ F], [ZA203; H, H, H, H, OCHF ₂ ], [ZA204; H, H, H, H, OCF ₃ ], [ZA205; H, H, H, H, O (CH ₂ ) ₂ F], [ZA206; H, H, H, H, OCH ₂ CHF ₂ ], [ZA207; H, H, H, H, OCH ₂ CHF ₃ ], [ZA208; H, H, H, H, O ( CH ₂ ) ₃ F], [ZA209; H, H, H, H, O (CH ₂ ) ₂ CHF ₂ ], [ZA210; H, H, H, H, O (CH ₂ ) ₂ CF ₃ ], [ ZA211; H, H, H, H, OCH ₂ CH (CF ₃ ) ₂ ], [ZA212; H, H, H, H, OCH ₂ Cl], [ZA213; H, H, H, H, O (CH ₂ ) ₂ Cl], [ZA214; H, H, H, H, O (CH ₂ ) ₃ Cl], [ZA215; H, H, H, H, O (CH ₂ ) ₄ Cl], [ZA216; H, H, H, H, O (CH ₂ ) ₅ Cl], [ZA217; H, H, H, H, OCH ₂ OMe], [ ZA218; H, H, H, H, O (CH ₂ ) ₂ OMe], [ZA219; H, H, H, H, O (CH ₂ ) ₃ OMe], [ZA220; H, H, H, H, O (CH ₂ ) ₄ OMe], [ZA221; H, H, H, H, OCH ₂ OEt], [ZA222; H, H, H, H, O (CH ₂ ) ₂ OEt], [ZA223; H, H, H, H, O (CH ₂ ) ₃ OEt], [ZA224; H, H, H, H, OCH ₂ OPr], [ZA225; H, H, H, H, O (CH ₂ ) ₂ OPr] , [ZA226; H, H, H, H, O (CH ₂ ) ₃ OPr], [ZA227; H, H, H, H, OCH ₂ CN], [ZA228; H, H, H, H, O ( _{CH 2) 2 CN], [} ZA229; H, H, H, H, O (CH 2) 3 CN], [ZA230; H, H, H, H, O (CH 2) 4 CN], [ZA231; H, H, H, H, O (CH ₂ ) ₅ CN], [ZA232; H, H, H, H, OCH ₂ CH = CH ₂ ], [ZA233; H, H, H, H, OCH ₂ C ≡CH], [ZA234; H, H, H, H, OCH ₂ C≡CCH ₃ ], [ZA235; H, H, H, H, OCH ₂ Ph], [ZA236; H, H, H, H, OCH ₂ (2-Py)], [ZA237; H, H, H, H, OCH ₂ (3-Py)], [ZA238; H, H, H, H, OCH ₂ (4-Py)], [ ZA239; H, H, H, H, O (CH ₂ ) ₂ Ph], [ZA240; H, H, H, H, O (CH ₂ ) ₂ (2-Py)], [ZA241; H, H, H, H, O (CH ₂ ) ₂ (3-Py)], [ZA242; H, H, H, H, O (CH ₂ ) ₂ (4-Py)], [ZA243; H, H, H, H, OPh], [ZA244; H, H, H, H, O (2-Py)], [ZA245; H, H, H, H, O (3-Py)], [ZA246; H, H, H, H, O (4-Py)], [ZA247; H, H, H, H, Me], [ZA248; H, H, H, H, Et], [ZA249; H, H, H, H, Pr], [ZA250; H, H, H, H, Bu],

[ZA251; H, H, H, H, Pen], [ZA252; H, H, H, H, Hex], [ZA253; H, H, H, H, (i-Pr)], [ZA254; H , H, H, H, (i-Bu)], [ZA255; H, H, H, H, (c-Pr)], [ZA256; H, H, H, H, (c-Bu)], [ZA257; H, H, H, H, (c-Pen)], [ZA258; H, H, H, H, (c-Hex)], [ZA259; H, H, H, H, CH ₂ ( c-Pr)], [ZA260; H, H, H, H, CH ₂ (c-Bu)], [ZA261; H, H, H, H, CH ₂ (c-Pen)], [ZA262; H , H, H, H, CH ₂ (c-Hex)], [ZA263; H, H, H, H, CH ₂ F], [ZA264; H, H, H, H, CHF ₂ ], [ZA265; H, H, H, H, CF ₃ ], [ZA266; H, H, H, H, (CH ₂ ) ₂ F], [ZA267; H, H, H, H, CH ₂ CHF ₂ ], [ZA268 ; H, H, H, H, CH ₂ CHF ₃ ], [ZA269; H, H, H, H, (CH ₂ ) ₃ F], [ZA270; H, H, H, H, (CH ₂ ) ₂ CHF ₂ ], [ZA271; H, H, H, H, (CH ₂ ) ₂ CF ₃ ], [ZA272; H, H, H, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA273; H, H, H, H, CH ₂ Cl], [ZA274; H, H, H, H, (CH ₂ ) ₂ Cl], [ZA275; H, H, H, H, (CH ₂ ) ₃ Cl], [ ZA276; H, H, H, H, (CH ₂ ) ₄ Cl], [ZA277; H, H, H, H, (CH ₂ ) ₅ Cl], [ZA278; H, H, H, H, CH ₂ OMe], [ZA279; H, H, H, H, (CH ₂ ) ₂ OMe], [ZA280; H, H, H, H, (CH ₂ ) ₃ OMe], [ZA281; H, H, H, H, (CH ₂ ) ₄ OMe], [ZA282; H, H, H, H, CH ₂ OEt], [ZA283; H, H, H, H, (CH ₂ ) ₂ OEt], [ZA284; H, H, H, H, (CH ₂ ) ₃ OEt], [ZA285; H, H, H, H, CH ₂ OPr], [ZA286; H, H, H, H, (CH ₂ ) ₂ OPr], [ ZA287; H, H, H, H, (CH ₂ ) ₃ OPr], [Z A288; H, H, H, H, CH ₂ CN], [ZA289; H, H, H, H, (CH ₂ ) ₂ CN], [ZA290; H, H, H, H, (CH ₂ ) ₃ CN], [ZA291; H, H, H, H, (CH ₂ ) ₄ CN], [ZA292; H, H, H, H, (CH ₂ ) ₅ CN], [ZA293; H, H, H, H, CH ₂ CH = CH ₂ ], [ZA294; H, H, H, H, CH ₂ C≡CH], [ZA295; H, H, H, H, CH ₂ C≡CCH ₃ ], [ZA296; H, H, H, H, CH ₂ Ph], [ZA297; H, H, H, H, CH ₂ (2-Py)], [ZA298; H, H, H, H, CH ₂ (3-Py )], [ZA299; H, H, H, H, CH ₂ (4-Py)], [ZA300; H, H, H, H, (CH ₂ ) ₂ Ph], [ZA301; H, H, H , H, (CH ₂ ) ₂ (2-Py)], [ZA302; H, H, H, H, (CH ₂ ) ₂ (3-Py)], [ZA303; H, H, H, H, ( CH ₂ ) ₂ (4-Py)], [ZA304; H, H, H, H, Ph], [ZA305; H, H, H, H, 2-Py], [ZA306; H, H, H, H, 3-Py], [ZA307; H, H, H, H, 4-Py], [ZA308; H, H, Me, H, NHMe], [ZA309; H, H, Me, H, NHEt] , [ZA310; H, H, Me, H, NHPr], [ZA311; H, H, Me, H, NHBu], [ZA312; H, H, Me, H, NHPen], [ZA313; H, H, Me, H, NHHex], [ZA314; H, H, Me, H, NH (i-Pr)], [ZA315; H, H, Me, H, NH (i-Bu)], [ZA316; H, H, Me, H, NH (c-Pr)], [ZA317; H, H, Me, H, NH (c-Bu)], [ZA318; H, H, Me, H, NH (c-Pen) ], [ZA319; H, H, Me, H, NH (c-Hex)], [ZA320; H, H, Me, H, NHCH ₂ (c-Pr)], [ZA321; H, H, Me, H, NHCH ₂ (c-Bu)], [ZA322; H, H, Me, H, NHCH ₂ (c-Pen)], [ZA323; H, H, Me, H, NHCH ₂ (c-Hex)] , [ZA324; H, H, Me, H, NHCH ₂ F], [ZA325; H, H , Me, H, NHCHF ₂ ], [ZA326; H, H, Me, H, NHCF ₃ ], [ZA327; H, H, Me, H, NH (CH ₂ ) ₂ F], [ZA328; H, H , Me, H, NHCH ₂ CHF ₂ ], [ZA329; H, H, Me, H, NHCH ₂ CHF ₃ ], [ZA330; H, H, Me, H, NH (CH ₂ ) ₃ F], [ZA331 ; H, H, Me, H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA332; H, H, Me, H, NH (CH ₂ ) ₂ CF ₃ ], [ZA333; H, H, Me, H , NHCH ₂ CH (CF ₃ ) ₂ ], [ZA334; H, H, Me, H, NHCH ₂ Cl], [ZA335; H, H, Me, H, NH (CH ₂ ) ₂ Cl], [ZA336; H, H, Me, H, NH (CH ₂ ) ₃ Cl], [ZA337; H, H, Me, H, NH (CH ₂ ) ₄ Cl], [ZA338; H, H, Me, H, NH ( CH ₂ ) ₅ Cl], [ZA339; H, H, Me, H, NHCH ₂ OMe], [ZA340; H, H, Me, H, NH (CH ₂ ) ₂ OMe], [ZA341; H, H, Me, H, NH (CH ₂ ) ₃ OMe], [ZA342; H, H, Me, H, NH (CH ₂ ) ₄ OMe], [ZA343; H, H, Me, H, NHCH ₂ OEt], [ ZA344; H, H, Me, H, NH (CH ₂ ) ₂ OEt], [ZA345; H, H, Me, H, NH (CH ₂ ) ₃ OEt], [ZA346; H, H, Me, H, NHCH ₂ OPr], [ZA347; H, H, Me, H, NH (CH ₂ ) ₂ OPr], [ZA348; H, H, Me, H, NH (CH ₂ ) ₃ OPr], [ZA349; H, H, Me, H, NHCH ₂ CN], [ZA350; H, H, Me, H, NH (CH ₂ ) ₂ CN], [ZA351; H, H, Me, H, NH (CH ₂ ) ₃ CN] , [ZA352; H, H, Me, H, NH (CH ₂ ) ₄ CN], [ZA353; H, H, Me, H, NH (CH ₂ ) ₅ CN], [ZA354; H, H, Me, H, NHCH ₂ CH = CH ₂ ], [ZA355; H, H, Me, H, NHCH ₂ C≡CH], [ZA356; H, H, Me, H, NHCH ₂ C≡CCH ₃ ], [ZA 357; H, H, Me, H, NHCH ₂ Ph], [ZA358; H, H, Me, H, NHCH ₂ (2-Py)], [ZA359; H, H, Me, H, NHCH ₂ (3 -Py)], [ZA360; H, H, Me, H, NHCH ₂ (4-Py)], [ZA361; H, H, Me, H, NH (CH ₂ ) ₂ Ph], [ZA362; H, H, Me, H, NH (CH ₂ ) ₂ (2-Py)], [ZA363; H, H, Me, H, NH (CH ₂ ) ₂ (3-Py)], [ZA364; H, H, Me, H, NH (CH ₂ ) ₂ (4-Py)], [ZA365; H, H, Me, H, NHPh], [ZA366; H, H, Me, H, NH (2-Py)], [ZA367; H, H, Me, H, NH (3-Py)], [ZA368; H, H, Me, H, NH (4-Py)], [ZA369; H, H, Me, H, NMe ₂ ], [ZA370; H, H, Me, H, NMeEt], [ZA371; H, H, Me, H, NMePr], [ZA372; H, H, Me, H, NMeBu], [ZA373; H, H, Me, H, NMePen], [ZA374; H, H, Me, H, NMeHex], [ZA375; H, H, Me, H, NMe (i-Pr)], [ZA376; H, H, Me , H, NMe (i-Bu)], [ZA377; H, H, Me, H, NMe (c-Pr)], [ZA378; H, H, Me, H, NMe (c-Bu)], [ ZA379; H, H, Me, H, NMe (c-Pen)], [ZA380; H, H, Me, H, NMe (c-Hex)], [ZA381; H, H, Me, H, NMeCH ₂ (c-Pr)], [ZA382; H, H, Me, H, NMeCH ₂ (c-Bu)], [ZA383; H, H, Me, H, NMeCH ₂ (c-Pen)], [ZA384; H, H, Me, H, NMeCH ₂ (c-Hex)], [ZA385; H, H, Me, H, NMeCH ₂ F], [ZA386; H, H, Me, H, NMeCHF ₂ ], [ZA387 ; H, H, Me, H, NMeCF ₃ ], [ZA388; H, H, Me, H, NMe (CH ₂ ) ₂ F], [ZA389; H, H, Me, H, NMeCH ₂ CHF ₂ ], [ZA390; H, H, Me, H, NMeCH ₂ CHF ₃ ], [ZA391; H, H, Me, H, NMe (CH ₂ ) ₃ F], [ZA392; H, H, Me, H, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA393; H, H, Me, H, NMe (CH ₂ ) ₂ CF ₃ ], [ZA394; H, H, Me , H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA395; H, H, Me, H, NMeCH ₂ Cl], [ZA396; H, H, Me, H, NMe (CH ₂ ) ₂ Cl], [ ZA397; H, H, Me, H, NMe (CH ₂ ) ₃ Cl], [ZA398; H, H, Me, H, NMe (CH ₂ ) ₄ Cl], [ZA399; H, H, Me, H, NMe (CH ₂ ) ₅ Cl], [ZA400; H, H, Me, H, NMeCH ₂ OMe], [ZA401; H, H, Me, H, NMe (CH ₂ ) ₂ OMe], [ZA402; H, H, Me, H, NMe (CH ₂ ) ₃ OMe], [ZA403; H, H, Me, H, NMe (CH ₂ ) ₄ OMe], [ZA404; H, H, Me, H, NMeCH ₂ OEt] , [ZA405; H, H, Me, H, NMe (CH ₂ ) ₂ OEt], [ZA406; H, H, Me, H, NMe (CH ₂ ) ₃ OEt], [ZA407; H, H, Me, H, NMeCH ₂ OPr], [ZA408; H, H, Me, H, NMe (CH ₂ ) ₂ OPr], [ZA409; H, H, Me, H, NMe (CH ₂ ) ₃ OPr], [ZA410; H, H, Me, H, NMeCH ₂ CN], [ZA411; H, H, Me, H, NMe (CH ₂ ) ₂ CN], [ZA412; H, H, Me, H, NMe (CH ₂ ) ₃ CN], [ZA413; H, H, Me, H, NMe (CH ₂ ) ₄ CN], [ZA414; H, H, Me, H, NMe (CH ₂ ) ₅ CN], [ZA415; H, H, Me, H, NMeCH ₂ CH = CH ₂ ], [ZA416; H, H, Me, H, NMeCH ₂ C≡CH], [ZA417; H, H, Me, H, NMeCH ₂ C≡CCH ₃ ], [ ZA418; H, H, Me, H, NMeCH ₂ Ph], [ZA419; H, H, Me, H, NMeCH ₂ (2-Py)], [ZA420; H, H, Me, H, NMeCH ₂ (3 -Py)], [ZA421; H, H, Me, H, NMeCH ₂ (4-Py)], [ZA422; H, H, Me, H, NM e (CH ₂ ) ₂ Ph], [ZA423; H, H, Me, H, NMe (CH ₂ ) ₂ (2-Py)], [ZA424; H, H, Me, H, NMe (CH ₂ ) ₂ (3-Py)], [ZA425; H, H, Me, H, NMe (CH ₂ ) ₂ (4-Py)], [ZA426; H, H, Me, H, NMePh], [ZA427; H, H, Me, H, NMe (2-Py)], [ZA428; H, H, Me, H, NMe (3-Py)], [ZA429; H, H, Me, H, NMe (4-Py) ], [ZA430; H, H, Me, H, NEt ₂ ], [ZA431; H, H, Me, H, NEtPr], [ZA432; H, H, Me, H, NEtBu], [ZA433; H, H, Me, H, NEtPen], [ZA434; H, H, Me, H, NEtHex], [ZA435; H, H, Me, H, NEt (i-Pr)], [ZA436; H, H, Me , H, NEt (i-Bu)], [ZA437; H, H, Me, H, NEt (c-Pr)], [ZA438; H, H, Me, H, NEt (c-Bu)], [ ZA439; H, H, Me, H, NEt (c-Pen)], [ZA440; H, H, Me, H, NEt (c-Hex)], [ZA441; H, H, Me, H, NEtCH ₂ (c-Pr)], [ZA442; H, H, Me, H, NEtCH ₂ (c-Bu)], [ZA443; H, H, Me, H, NEtCH ₂ (c-Pen)], [ZA444; H, H, Me, H, NEtCH ₂ (c-Hex)], [ZA445; H, H, Me, H, NEtCH ₂ F], [ZA446; H, H, Me, H, NEtCHF ₂ ], [ZA447 ; H, H, Me, H, NEtCF ₃ ], [ZA448; H, H, Me, H, NEt (CH ₂ ) ₂ F], [ZA449; H, H, Me, H, NEtCH ₂ CHF ₂ ], [ZA450; H, H, Me, H, NEtCH ₂ CHF ₃ ], [ZA451; H, H, Me, H, NEt (CH ₂ ) ₃ F], [ZA452; H, H, Me, H, NEt ( CH ₂ ) ₂ CHF ₂ ], [ZA453; H, H, Me, H, NEt (CH ₂ ) ₂ CF ₃ ], [ZA454; H, H, Me, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA455; H, H, Me, H, NEtCH ₂ Cl], [ZA456; H, H, Me, H, NEt (CH ₂ ) ₂ Cl], [ZA457; H, H, Me, H, NEt (CH ₂ ) ₃ Cl], [ZA458; H, H, Me, H, NEt (CH ₂ ) ₄ Cl], [ZA459; H, H, Me, H, NEt (CH ₂ ) ₅ Cl], [ZA460; H, H, Me, H, NEtCH ₂ OMe], [ZA461; H, H, Me, H, NEt (CH ₂ ) ₂ OMe], [ZA462; H, H, Me, H, NEt (CH ₂ ) ₃ OMe], [ZA463; H, H, Me, H, NEt (CH ₂ ) ₄ OMe], [ ZA464; H, H, Me, H, NEtCH ₂ OEt], [ZA465; H, H, Me, H, NEt (CH ₂ ) ₂ OEt], [ZA466; H, H, Me, H, NEt (CH ₂ ) ₃ OEt], [ZA467; H, H, Me, H, NEtCH ₂ OPr], [ZA468; H, H, Me, H, NEt (CH ₂ ) ₂ OPr], [ZA469; H, H, Me, _{H, NEt (CH 2) 3} OPr], [ZA470; H, H, Me, H, NEtCH 2 CN], [ZA471; H, H, Me, H, NEt (CH 2) 2 CN], [ZA472; H, H, Me, H, NEt (CH ₂ ) ₃ CN], [ZA473; H, H, Me, H, NEt (CH ₂ ) ₄ CN], [ZA474; H, H, Me, H, NEt ( CH ₂ ) ₅ CN], [ZA475; H, H, Me, H, NEtCH ₂ CH = CH ₂ ], [ZA476; H, H, Me, H, NEtCH ₂ C≡CH], [ZA477; H, H , Me, H, NEtCH ₂ C≡CCH ₃ ], [ZA478; H, H, Me, H, NEtCH ₂ Ph], [ZA479; H, H, Me, H, NEtCH ₂ (2-Py)], [ ZA480; H, H, Me, H, NEtCH ₂ (3-Py)], [ZA481; H, H, Me, H, NEtCH ₂ (4-Py)], [ZA482; H, H, Me, H, NEt (CH ₂ ) ₂ Ph], [ZA483; H, H, Me, H, NEt (CH ₂ ) ₂ (2-Py)], [ZA484; H, H, Me, H, NEt (CH ₂ ) ₂ (3-Py)], [ZA485; H, H, Me, H, NEt (CH ₂ ) ₂ (4-Py)], [ZA486; H, H, Me, H, NEtPh], [ ZA487; H, H, Me, H, NEt (2-Py)], [ZA488; H, H, Me, H, NEt (3-Py)], [ZA489; H, H, Me, H, NEt ( 4-Py)], [ZA490; H, H, Me, H, Pyr], [ZA491; H, H, Me, H, Pip], [ZA492; H, H, Me, H, Mor], [ZA493 ; H, H, Me, H, OMe], [ZA494; H, H, Me, H, OEt], [ZA495; H, H, Me, H, OPr], [ZA496; H, H, Me, H , OBu], [ZA497; H, H, Me, H, OPen], [ZA498; H, H, Me, H, OHex], [ZA499; H, H, Me, H, O (i-Pr)] , [ZA500; H, H, Me, H, O (i-Bu)],

[ZA501; H, H, Me, H, O (c-Pr)], [ZA502; H, H, Me, H, O (c-Bu)], [ZA503; H, H, Me, H, O (c-Pen)], [ZA504; H, H, Me, H, O (c-Hex)], [ZA505; H, H, Me, H, OCH ₂ (c-Pr)], [ZA506; H , H, Me, H, OCH ₂ (c-Bu)], [ZA507; H, H, Me, H, OCH ₂ (c-Pen)], [ZA508; H, H, Me, H, OCH ₂ ( c-Hex)], [ZA509; H, H, Me, H, OCH ₂ F], [ZA510; H, H, Me, H, OCHF ₂ ], [ZA511; H, H, Me, H, OCF ₃ ], [ZA512; H, H, Me, H, O (CH ₂ ) ₂ F], [ZA513; H, H, Me, H, OCH ₂ CHF ₂ ], [ZA514; H, H, Me, H, OCH ₂ CHF ₃ ], [ZA515; H, H, Me, H, O (CH ₂ ) ₃ F], [ZA516; H, H, Me, H, O (CH ₂ ) ₂ CHF ₂ ], [ZA517; H, H, Me, H, O (CH ₂ ) ₂ CF ₃ ], [ZA518; H, H, Me, H, OCH ₂ CH (CF ₃ ) ₂ ], [ZA519; H, H, Me, H, OCH ₂ Cl], [ZA520; H, H, Me, H, O (CH ₂ ) ₂ Cl], [ZA521; H, H, Me, H, O (CH ₂ ) ₃ Cl], [ZA522; H, H, Me, H, O (CH ₂ ) ₄ Cl], [ZA523; H, H, Me, H, O (CH ₂ ) ₅ Cl], [ZA524; H, H, Me, H, OCH ₂ OMe] , [ZA525; H, H, Me, H, O (CH ₂ ) ₂ OMe], [ZA526; H, H, Me, H, O (CH ₂ ) ₃ OMe], [ZA527; H, H, Me, H, O (CH ₂ ) ₄ OMe], [ZA528; H, H, Me, H, OCH ₂ OEt], [ZA529; H, H, Me, H, O (CH ₂ ) ₂ OEt], [ZA530; H, H, Me, H, O (CH ₂ ) ₃ OEt], [ZA531; H, H, Me, H, OCH ₂ OPr], [ZA532; H, H, Me, H, O (CH ₂ ) ₂ OPr], [ZA533; H, H, Me, H, O (CH ₂ ) ₃ OPr], [ZA534; H, H, Me, H, OCH ₂ CN], [ZA535; H, H, Me, H, O (CH ₂ ) ₂ CN], [ZA536; H, H, Me, H, O (CH ₂ ) ₃ CN], [ZA537; H, H, Me, H, O (CH ₂ ) ₄ CN], [ZA538; H, H, Me, H, O (CH ₂ ) ₅ CN], [ZA539; H, H, Me, H, OCH ₂ CH = CH ₂ ], [ZA540; H, H, Me, H, OCH ₂ C≡CH], [ZA541; H, H, Me, H, OCH ₂ C≡CCH ₃ ], [ZA542; H, H, Me, H, OCH ₂ Ph], [ZA543; H, H, Me, H, OCH ₂ (2-Py)], [ZA544; H, H, Me, H, OCH ₂ (3-Py)], [ZA545; H, H, Me, H, OCH ₂ (4-Py)], [ZA546; H, H, Me, H, O (CH ₂ ) ₂ Ph], [ZA547; H, H, Me, H, O (CH ₂ ) ₂ (2-Py)], [ZA548; H, H, Me, H, O (CH ₂ ) ₂ (3-Py)], [ZA549; H, H, Me, H, O (CH ₂ ) ₂ (4-Py)], [ZA550; H, H, Me, H, OPh], [ZA551; H, H, Me, H, O (2-Py)], [ZA552; H, H, Me, H , O (3-Py)], [ZA553; H, H, Me, H, O (4-Py)], [ZA554; H, H, Me, H, Me], [ZA555; H, H, Me , H, Et], [ZA556; H, H, Me, H, Pr], [ZA557; H, H, Me, H, Bu], [ZA558; H, H, Me, H, Pen], [ZA559 ; H, H, Me, H, Hex], [ZA560; H, H, Me, H, (i-Pr)], [ZA561; H, H, Me, H, (i-Bu)], [ZA562 ; H, H, Me, H, (c-Pr)], [ZA563; H, H, Me, H, (c-Bu)], [ZA564; H, H, Me, H, (c-Pen) ], [ZA565; H, H, Me, H, (c-Hex)], [ZA566; H, H, Me, H, CH ₂ (c-Pr)], [ZA567; H, H, Me, H , CH ₂ (c-Bu)], [ZA568; H, H, Me, H, CH ₂ (c-Pen)], [ZA569; H, H, Me, H, CH ₂ (c-Hex)], [ZA570; H, H, Me, H, CH ₂ F], [ZA571; H, H, Me, H, CH F ₂ ], [ZA572; H, H, Me, H, CF ₃ ], [ZA573; H, H, Me, H, (CH ₂ ) ₂ F], [ZA574; H, H, Me, H, CH ₂ CHF ₂ ], [ZA575; H, H, Me, H, CH ₂ CHF ₃ ], [ZA576; H, H, Me, H, (CH ₂ ) ₃ F], [ZA577; H, H, Me, H, (CH ₂ ) ₂ CHF ₂ ], [ZA578; H, H, Me, H, (CH ₂ ) ₂ CF ₃ ], [ZA579; H, H, Me, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA580; H, H, Me, H, CH ₂ Cl], [ZA581; H, H, Me, H, (CH ₂ ) ₂ Cl], [ZA582; H, H, Me, H, (CH _{2) 3 Cl], [ZA583} ; H, H, Me, H, (CH 2) 4 Cl], [ZA584; H, H, Me, H, (CH 2) 5 Cl], [ZA585; H, H , Me, H, CH ₂ OMe], [ZA586; H, H, Me, H, (CH ₂ ) ₂ OMe], [ZA587; H, H, Me, H, (CH ₂ ) ₃ OMe], [ZA588 ; H, H, Me, H, (CH ₂ ) ₄ OMe], [ZA589; H, H, Me, H, CH ₂ OEt], [ZA590; H, H, Me, H, (CH ₂ ) ₂ OEt ], [ZA591; H, H, Me, H, (CH ₂ ) ₃ OEt], [ZA592; H, H, Me, H, CH ₂ OPr], [ZA593; H, H, Me, H, (CH ₂ ) ₂ OPr], [ZA594; H, H, Me, H, (CH ₂ ) ₃ OPr], [ZA595; H, H, Me, H, CH ₂ CN], [ZA596; H, H, Me, H, (CH ₂ ) ₂ CN], [ZA597; H, H, Me, H, (CH ₂ ) ₃ CN], [ZA598; H, H, Me, H, (CH ₂ ) ₄ CN], [ZA599 ; H, H, Me, H, (CH ₂ ) ₅ CN], [ZA600; H, H, Me, H, CH ₂ CH = CH ₂ ], [ZA601; H, H, Me, H, CH ₂ C ≡CH], [ZA602; H, H, Me, H, CH ₂ C≡CCH ₃ ], [ZA603; H, H, Me, H, CH ₂ Ph], [ZA604; H, H, Me, H, CH ₂ (2-Py)], [ZA605; H, H, Me, H, CH ₂ (3-Py)], [ZA606; H, H, Me, H, CH ₂ (4-Py)], [ZA607; H, H, Me, H, (CH ₂ ) ₂ Ph], [ZA608; H , H, Me, H, (CH ₂ ) ₂ (2-Py)], [ZA609; H, H, Me, H, (CH ₂ ) ₂ (3-Py)], [ZA610; H, H, Me , H, (CH ₂ ) ₂ (4-Py)], [ZA611; H, H, Me, H, Ph], [ZA612; H, H, Me, H, 2-Py], [ZA613; H, H, Me, H, 3-Py], [ZA614; H, H, Me, H, 4-Py], [ZA615; H, H, Me, Me, NHMe], [ZA616; H, H, Me, Me, NHEt], [ZA617; H, H, Me, Me, NHPr], [ZA618; H, H, Me, Me, NHBu], [ZA619; H, H, Me, Me, NHPen], [ZA620; H, H, Me, Me, NHHex], [ZA621; H, H, Me, Me, NH (i-Pr)], [ZA622; H, H, Me, Me, NH (i-Bu)], [ ZA623; H, H, Me, Me, NH (c-Pr)], [ZA624; H, H, Me, Me, NH (c-Bu)], [ZA625; H, H, Me, Me, NH ( c-Pen)], [ZA626; H, H, Me, Me, NH (c-Hex)], [ZA627; H, H, Me, Me, NHCH ₂ (c-Pr)], [ZA628; H, H, Me, Me, NHCH ₂ (c-Bu)], [ZA629; H, H, Me, Me, NHCH ₂ (c-Pen)], [ZA630; H, H, Me, Me, NHCH ₂ (c -Hex)], [ZA631; H, H, Me, Me, NHCH ₂ F], [ZA632; H, H, Me, Me, NHCHF ₂ ], [ZA633; H, H, Me, Me, NHCF ₃ ] , [ZA634; H, H, Me, Me, NH (CH ₂ ) ₂ F], [ZA635; H, H, Me, Me, NHCH ₂ CHF ₂ ], [ZA636; H, H, Me, Me, NHCH ₂ CHF ₃ ], [ZA637; H, H, Me, Me, NH (CH ₂ ) ₃ F], [ZA638; H, H, Me, Me, NH (CH ₂ ) ₂ CHF ₂ ], [ZA639; H , H, Me, Me, NH (CH ₂ ) ₂ CF ₃ ], [ZA640; H, H, Me, Me, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA641; H, H, Me, Me, NHCH ₂ Cl], [ZA642; H, H, Me, Me, NH (CH ₂ ) ₂ Cl], [ZA643; H, H, Me, Me, NH (CH ₂ ) ₃ Cl], [ZA644; H, H, Me, Me, NH (CH ₂ ) ₄ Cl], [ZA645; H, H, Me, Me, NH (CH ₂ ) ₅ Cl] , [ZA646; H, H, Me, Me, NHCH ₂ OMe], [ZA647; H, H, Me, Me, NH (CH ₂ ) ₂ OMe], [ZA648; H, H, Me, Me, NH ( CH ₂ ) ₃ OMe], [ZA649; H, H, Me, Me, NH (CH ₂ ) ₄ OMe], [ZA650; H, H, Me, Me, NHCH ₂ OEt], [ZA651; H, H, Me, Me, NH (CH ₂ ) ₂ OEt], [ZA652; H, H, Me, Me, NH (CH ₂ ) ₃ OEt], [ZA653; H, H, Me, Me, NHCH ₂ OPr], [ ZA654; H, H, Me, Me, NH (CH ₂ ) ₂ OPr], [ZA655; H, H, Me, Me, NH (CH ₂ ) ₃ OPr], [ZA656; H, H, Me, Me, NHCH ₂ CN], [ZA657; H, H, Me, Me, NH (CH ₂ ) ₂ CN], [ZA658; H, H, Me, Me, NH (CH ₂ ) ₃ CN], [ZA659; H, H, Me, Me, NH (CH ₂ ) ₄ CN], [ZA660; H, H, Me, Me, NH (CH ₂ ) ₅ CN], [ZA661; H, H, Me, Me, NHCH ₂ CH = CH ₂ ], [ZA662; H, H, Me, Me, NHCH ₂ C≡CH], [ZA663; H, H, Me, Me, NHCH ₂ C≡CCH ₃ ], [ZA664; H, H, Me, Me, NHCH ₂ Ph], [ZA665; H, H, Me, Me, NHCH ₂ (2-Py)], [ZA666; H, H, Me, Me, NHCH ₂ (3-Py)], [ZA667; H, H, Me, Me, NHCH ₂ (4-Py)], [ZA668; H, H, Me, Me, NH (CH ₂ ) ₂ Ph], [ZA669; H, H, Me, Me, NH ( CH ₂ ) ₂ (2-Py)], [ZA670; H, H, Me, Me, NH (CH ₂ ) ₂ (3-Py)], [ZA671; H, H, Me, Me, NH (CH ₂ ) ₂ (4-Py)], [ZA672; H, H, Me, Me, NHPh], [ZA673; H, H, Me, Me, NH (2-Py)], [ZA674 ; H, H, Me, Me, NH (3-Py)], [ZA675; H, H, Me, Me, NH (4-Py)], [ZA676; H, H, Me, Me, NMe ₂ ] , [ZA677; H, H, Me, Me, NMeEt], [ZA678; H, H, Me, Me, NMePr], [ZA679; H, H, Me, Me, NMeBu], [ZA680; H, H, Me, Me, NMePen], [ZA681; H, H, Me, Me, NMeHex], [ZA682; H, H, Me, Me, NMe (i-Pr)], [ZA683; H, H, Me, Me , NMe (i-Bu)], [ZA684; H, H, Me, Me, NMe (c-Pr)], [ZA685; H, H, Me, Me, NMe (c-Bu)], [ZA686; H, H, Me, Me, NMe (c-Pen)], [ZA687; H, H, Me, Me, NMe (c-Hex)], [ZA688; H, H, Me, Me, NMeCH ₂ (c -Pr)], [ZA689; H, H, Me, Me, NMeCH ₂ (c-Bu)], [ZA690; H, H, Me, Me, NMeCH ₂ (c-Pen)], [ZA691; H, H, Me, Me, NMeCH ₂ (c-Hex)], [ZA692; H, H, Me, Me, NMeCH ₂ F], [ZA693; H, H, Me, Me, NMeCHF ₂ ], [ZA694; H , H, Me, Me, NMeCF ₃ ], [ZA695; H, H, Me, Me, NMe (CH ₂ ) ₂ F], [ZA696; H, H, Me, Me, NMeCH ₂ CHF ₂ ], [ZA697 ; H, H, Me, Me, NMeCH ₂ CHF ₃ ], [ZA698; H, H, Me, Me, NMe (CH ₂ ) ₃ F], [ZA699; H, H, Me, Me, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA700; H, H, Me, Me, NMe (CH ₂ ) ₂ CF ₃ ], [ZA701; H, H, Me, Me, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA702 ; H, H, Me, Me, NMeCH ₂ Cl], [ZA703; H, H, Me, Me, NMe (CH ₂ ) ₂ Cl], [ZA704; H, H, Me, Me, NMe (CH ₂ ) _Three Cl], [ZA705; H, H, Me, Me, NMe (CH ₂ ) ₄ Cl], [ZA706; H, H, Me, Me, NMe (CH ₂ ) ₅ Cl], [ZA707; H, H, Me, Me, NMeCH ₂ OMe], [ZA708; H, H, Me, Me, NMe (CH ₂ ) ₂ OMe], [ZA709; H, H, Me, Me, NMe (CH ₂ ) ₃ OMe], [ ZA710; H, H, Me, Me, NMe (CH ₂ ) ₄ OMe], [ZA711; H, H, Me, Me, NMeCH ₂ OEt], [ZA712; H, H, Me, Me, NMe (CH ₂ ) ₂ OEt], [ZA713; H, H, Me, Me, NMe (CH ₂ ) ₃ OEt], [ZA714; H, H, Me, Me, NMeCH ₂ OPr], [ZA715; H, H, Me, Me, NMe (CH ₂ ) ₂ OPr], [ZA716; H, H, Me, Me, NMe (CH ₂ ) ₃ OPr], [ZA717; H, H, Me, Me, NMeCH ₂ CN], [ZA718; H, H, Me, Me, NMe (CH ₂ ) ₂ CN], [ZA719; H, H, Me, Me, NMe (CH ₂ ) ₃ CN], [ZA720; H, H, Me, Me, NMe ( CH ₂ ) ₄ CN], [ZA721; H, H, Me, Me, NMe (CH ₂ ) ₅ CN], [ZA722; H, H, Me, Me, NMeCH ₂ CH = CH ₂ ], [ZA723; H , H, Me, Me, NMeCH ₂ C≡CH], [ZA724; H, H, Me, Me, NMeCH ₂ C≡CCH ₃ ], [ZA725; H, H, Me, Me, NMeCH ₂ Ph], [ ZA726; H, H, Me, Me, NMeCH ₂ (2-Py)], [ZA727; H, H, Me, Me, NMeCH ₂ (3-Py)], [ZA728; H, H, Me, Me, NMeCH ₂ (4-Py)], [ZA729; H, H, Me, Me, NMe (CH ₂ ) ₂ Ph], [ZA730; H, H, Me, Me, NMe (CH ₂ ) ₂ (2-Py )], [ZA731; H, H, Me, Me, NMe (CH ₂ ) ₂ (3-Py)], [ZA732; H, H, Me, Me, NMe (CH ₂ ) ₂ (4-Py)] , [ZA733; H, H, Me, Me, NMePh], [ZA734; H, H, Me, Me, NMe (2- Py)], [ZA735; H, H, Me, Me, NMe (3-Py)], [ZA736; H, H, Me, Me, NMe (4-Py)], [ZA737; H, H, Me , Me, NEt ₂ ], [ZA738; H, H, Me, Me, NEtPr], [ZA739; H, H, Me, Me, NEtBu], [ZA740; H, H, Me, Me, NEtPen], [ ZA741; H, H, Me, Me, NEtHex], [ZA742; H, H, Me, Me, NEt (i-Pr)], [ZA743; H, H, Me, Me, NEt (i-Bu)] , [ZA744; H, H, Me, Me, NEt (c-Pr)], [ZA745; H, H, Me, Me, NEt (c-Bu)], [ZA746; H, H, Me, Me, NEt (c-Pen)], [ZA747; H, H, Me, Me, NEt (c-Hex)], [ZA748; H, H, Me, Me, NEtCH ₂ (c-Pr)], [ZA749; H, H, Me, Me, NEtCH ₂ (c-Bu)], [ZA750; H, H, Me, Me, NEtCH ₂ (c-Pen)],

[ZA751; H, H, Me, Me, NEtCH ₂ (c-Hex)], [ZA752; H, H, Me, Me, NEtCH ₂ F], [ZA753; H, H, Me, Me, NEtCHF ₂ ] , [ZA754; H, H, Me, Me, NEtCF ₃ ], [ZA755; H, H, Me, Me, NEt (CH ₂ ) ₂ F], [ZA756; H, H, Me, Me, NEtCH ₂ CHF ₂ ], [ZA757; H, H, Me, Me, NEtCH ₂ CHF ₃ ], [ZA758; H, H, Me, Me, NEt (CH ₂ ) ₃ F], [ZA759; H, H, Me, Me , NEt (CH ₂ ) ₂ CHF ₂ ], [ZA760; H, H, Me, Me, NEt (CH ₂ ) ₂ CF ₃ ], [ZA761; H, H, Me, Me, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA762; H, H, Me, Me, NEtCH ₂ Cl], [ZA763; H, H, Me, Me, NEt (CH ₂ ) ₂ Cl], [ZA764; H, H, Me, Me, NEt (CH ₂ ) ₃ Cl], [ZA765; H, H, Me, Me, NEt (CH ₂ ) ₄ Cl], [ZA766; H, H, Me, Me, NEt (CH ₂ ) ₅ Cl], [ ZA767; H, H, Me, Me, NEtCH ₂ OMe], [ZA768; H, H, Me, Me, NEt (CH ₂ ) ₂ OMe], [ZA769; H, H, Me, Me, NEt (CH ₂ ) ₃ OMe], [ZA770; H, H, Me, Me, NEt (CH ₂ ) ₄ OMe], [ZA771; H, H, Me, Me, NEtCH ₂ OEt], [ZA772; H, H, Me, Me, NEt (CH ₂ ) ₂ OEt], [ZA773; H, H, Me, Me, NEt (CH ₂ ) ₃ OEt], [ZA774; H, H, Me, Me, NEtCH ₂ OPr], [ZA775; H, H, Me, Me, NEt (CH ₂ ) ₂ OPr], [ZA776; H, H, Me, Me, NEt (CH ₂ ) ₃ OPr], [ZA777; H, H, Me, Me, NEtCH ₂ CN], [ZA778; H, H, Me, Me, NEt (CH ₂ ) ₂ CN], [ZA779; H, H, Me, Me, NEt (CH ₂ ) ₃ CN], [ZA780; H, H, Me, Me, NEt (CH ₂ ) ₄ CN], [ZA781 ; H, H, Me, Me, NEt (CH ₂ ) ₅ CN], [ZA782; H, H, Me, Me, NEtCH ₂ CH = CH ₂ ], [ZA783; H, H, Me, Me, NEtCH ₂ C≡CH], [ZA784; H, H, Me, Me, NEtCH ₂ C≡CCH ₃ ], [ZA785; H, H, Me, Me, NEtCH ₂ Ph], [ZA786; H, H, Me, Me , NEtCH ₂ (2-Py)], [ZA787; H, H, Me, Me, NEtCH ₂ (3-Py)], [ZA788; H, H, Me, Me, NEtCH ₂ (4-Py)], [ZA789; H, H, Me, Me, NEt (CH ₂ ) ₂ Ph], [ZA790; H, H, Me, Me, NEt (CH ₂ ) ₂ (2-Py)], [ZA791; H, H , Me, Me, NEt (CH ₂ ) ₂ (3-Py)], [ZA792; H, H, Me, Me, NEt (CH ₂ ) ₂ (4-Py)], [ZA793; H, H, Me , Me, NEtPh], [ZA794; H, H, Me, Me, NEt (2-Py)], [ZA795; H, H, Me, Me, NEt (3-Py)], [ZA796; H, H , Me, Me, NEt (4-Py)], [ZA797; H, H, Me, Me, Pyr], [ZA798; H, H, Me, Me, Pip], [ZA799; H, H, Me, Me, Mor], [ZA800; H, H, Me, Me, OMe], [ZA801; H, H, Me, Me, OEt], [ZA802; H, H, Me, Me, OPr], [ZA803; H, H, Me, Me, OBu], [ZA804; H, H, Me, Me, OPen], [ZA805; H, H, Me, Me, OHex], [ZA806; H, H, Me, Me, O (i-Pr)], [ZA807; H, H, Me, Me, O (i-Bu)], [ZA808; H, H, Me, Me, O (c-Pr)], [ZA809; H , H, Me, Me, O (c-Bu)], [ZA810; H, H, Me, Me, O (c-Pen)], [ZA811; H, H, Me, Me, O (c-Hex )], [ZA812; H, H, Me, Me, OCH ₂ (c-Pr)], [ZA813; H, H, Me, Me, OCH ₂ (c-Bu)], [ZA814; H, H, Me, Me, OCH ₂ (c-Pen)], [ZA815; H, H, Me, Me, OCH ₂ (c-Hex)] , [ZA816; H, H, Me, Me, OCH ₂ F], [ZA817; H, H, Me, Me, OCHF ₂ ], [ZA818; H, H, Me, Me, OCF ₃ ], [ZA819; H, H, Me, Me, O (CH ₂ ) ₂ F], [ZA820; H, H, Me, Me, OCH ₂ CHF ₂ ], [ZA821; H, H, Me, Me, OCH ₂ CHF ₃ ] , [ZA822; H, H, Me, Me, O (CH ₂ ) ₃ F], [ZA823; H, H, Me, Me, O (CH ₂ ) ₂ CHF ₂ ], [ZA824; H, H, Me , Me, O (CH ₂ ) ₂ CF ₃ ], [ZA825; H, H, Me, Me, OCH ₂ CH (CF ₃ ) ₂ ], [ZA826; H, H, Me, Me, OCH ₂ Cl], [ZA827; H, H, Me, Me, O (CH ₂ ) ₂ Cl], [ZA828; H, H, Me, Me, O (CH ₂ ) ₃ Cl], [ZA829; H, H, Me, Me , O (CH ₂ ) ₄ Cl], [ZA830; H, H, Me, Me, O (CH ₂ ) ₅ Cl], [ZA831; H, H, Me, Me, OCH ₂ OMe], [ZA832; H , H, Me, Me, O (CH ₂ ) ₂ OMe], [ZA833; H, H, Me, Me, O (CH ₂ ) ₃ OMe], [ZA834; H, H, Me, Me, O (CH ₂ ) ₄ OMe], [ZA835; H, H, Me, Me, OCH ₂ OEt], [ZA836; H, H, Me, Me, O (CH ₂ ) ₂ OEt], [ZA837; H, H, Me , Me, O (CH ₂ ) ₃ OEt], [ZA838; H, H, Me, Me, OCH ₂ OPr], [ZA839; H, H, Me, Me, O (CH ₂ ) ₂ OPr], [ZA840 ; H, H, Me, Me, O (CH ₂ ) ₃ OPr], [ZA841; H, H, Me, Me, OCH ₂ CN], [ZA842; H, H, Me, Me, O (CH ₂ ) ₂ CN], [ZA843; H, H, Me, Me, O (CH ₂ ) ₃ CN], [ZA844; H, H, Me, Me, O (CH ₂ ) ₄ CN], [ZA845; H, H , Me, Me, O (CH ₂ ) ₅ CN], [ZA846; H, H, Me, Me, OCH ₂ CH = CH ₂ ], [ZA847; H, H, Me, Me, OCH ₂ C≡CH] , [ ZA848; H, H, Me, Me, OCH ₂ C≡CCH ₃ ], [ZA849; H, H, Me, Me, OCH ₂ Ph], [ZA850; H, H, Me, Me, OCH ₂ (2- Py)], [ZA851; H, H, Me, Me, OCH ₂ (3-Py)], [ZA852; H, H, Me, Me, OCH ₂ (4-Py)], [ZA853; H, H , Me, Me, O (CH ₂ ) ₂ Ph], [ZA854; H, H, Me, Me, O (CH ₂ ) ₂ (2-Py)], [ZA855; H, H, Me, Me, O (CH ₂ ) ₂ (3-Py)], [ZA856; H, H, Me, Me, O (CH ₂ ) ₂ (4-Py)], [ZA857; H, H, Me, Me, OPh], [ZA858; H, H, Me, Me, O (2-Py)], [ZA859; H, H, Me, Me, O (3-Py)], [ZA860; H, H, Me, Me, O (4-Py)], [ZA861; H, H, Me, Me, Me], [ZA862; H, H, Me, Me, Et], [ZA863; H, H, Me, Me, Pr], [ ZA864; H, H, Me, Me, Bu], [ZA865; H, H, Me, Me, Pen], [ZA866; H, H, Me, Me, Hex], [ZA867; H, H, Me, Me, (i-Pr)], [ZA868; H, H, Me, Me, (i-Bu)], [ZA869; H, H, Me, Me, (c-Pr)], [ZA870; H, H, Me, Me, (c-Bu)], [ZA871; H, H, Me, Me, (c-Pen)], [ZA872; H, H, Me, Me, (c-Hex)], [ ZA873; H, H, Me, Me, CH ₂ (c-Pr)], [ZA874; H, H, Me, Me, CH ₂ (c-Bu)], [ZA875; H, H, Me, Me, CH ₂ (c-Pen)], [ZA876; H, H, Me, Me, CH ₂ (c-Hex)], [ZA877; H, H, Me, Me, CH ₂ F], [ZA878; H, H, Me, Me, CHF ₂ ], [ZA879; H, H, Me, Me, CF ₃ ], [ZA880; H, H, Me, Me, (CH ₂ ) ₂ F], [ZA881; H, H , Me, Me, CH ₂ CHF ₂ ], [ZA882; H, H, Me, Me, CH ₂ CHF ₃ ], [ZA883; H, H, Me, Me, (CH ₂ ) ₃ F], [ZA884; H, H , Me, Me, (CH ₂ ) ₂ CHF ₂ ], [ZA885; H, H, Me, Me, (CH ₂ ) ₂ CF ₃ ], [ZA886; H, H, Me, Me, CH ₂ CH (CF ₃ ) ₂ ], [ZA887; H, H, Me, Me, CH ₂ Cl], [ZA888; H, H, Me, Me, (CH ₂ ) ₂ Cl], [ZA889; H, H, Me, Me , (CH ₂ ) ₃ Cl], [ZA890; H, H, Me, Me, (CH ₂ ) ₄ Cl], [ZA891; H, H, Me, Me, (CH ₂ ) ₅ Cl], [ZA892; H, H, Me, Me, CH ₂ OMe], [ZA893; H, H, Me, Me, (CH ₂ ) ₂ OMe], [ZA894; H, H, Me, Me, (CH ₂ ) ₃ OMe] , [ZA895; H, H, Me, Me, (CH ₂ ) ₄ OMe], [ZA896; H, H, Me, Me, CH ₂ OEt], [ZA897; H, H, Me, Me, (CH ₂ ) ₂ OEt], [ZA898; H, H, Me, Me, (CH ₂ ) ₃ OEt], [ZA899; H, H, Me, Me, CH ₂ OPr], [ZA900; H, H, Me, Me , (CH ₂ ) ₂ OPr], [ZA901; H, H, Me, Me, (CH ₂ ) ₃ OPr], [ZA902; H, H, Me, Me, CH ₂ CN], [ZA903; H, H , Me, Me, (CH ₂ ) ₂ CN], [ZA904; H, H, Me, Me, (CH ₂ ) ₃ CN], [ZA905; H, H, Me, Me, (CH ₂ ) ₄ CN] , [ZA906; H, H, Me, Me, (CH ₂ ) ₅ CN], [ZA907; H, H, Me, Me, CH ₂ CH = CH ₂ ], [ZA908; H, H, Me, Me, CH ₂ C≡CH], [ZA909; H, H, Me, Me, CH ₂ C≡CCH ₃ ], [ZA910; H, H, Me, Me, CH ₂ Ph], [ZA911; H, H, Me , Me, CH ₂ (2-Py)], [ZA912; H, H, Me, Me, CH ₂ (3-Py)], [ZA913; H, H, Me, Me, CH ₂ (4-Py) ], [ZA914; H, H, Me, Me, (CH ₂ ) ₂ Ph], [ZA915; H, H, Me, Me, (CH ₂ ) ₂ (2-Py)], [ZA916; H, H , Me, Me, (CH ₂ ) ₂ (3-Py)], [ZA917; H, H, Me, Me, (CH ₂ ) ₂ (4-Py)], [ZA918; H, H, Me, Me, Ph], [ZA919; H , H, Me, Me, 2-Py], [ZA920; H, H, Me, Me, 3-Py], [ZA921; H, H, Me, Me, 4-Py], [ZA922; H, H , F, H, NHMe], [ZA923; H, H, F, H, NHEt], [ZA924; H, H, F, H, NHPr], [ZA925; H, H, F, H, NHBu], [ZA926; H, H, F, H, NHPen], [ZA927; H, H, F, H, NHHex], [ZA928; H, H, F, H, NH (i-Pr)], [ZA929; H, H, F, H, NH (i-Bu)], [ZA930; H, H, F, H, NH (c-Pr)], [ZA931; H, H, F, H, NH (c- Bu)], [ZA932; H, H, F, H, NH (c-Pen)], [ZA933; H, H, F, H, NH (c-Hex)], [ZA934; H, H, F , H, NHCH ₂ (c-Pr)], [ZA935; H, H, F, H, NHCH ₂ (c-Bu)], [ZA936; H, H, F, H, NHCH ₂ (c-Pen) ], [ZA937; H, H, F, H, NHCH ₂ (c-Hex)], [ZA938; H, H, F, H, NHCH ₂ F], [ZA939; H, H, F, H, NHCHF ₂ ], [ZA940; H, H, F, H, NHCF ₃ ], [ZA941; H, H, F, H, NH (CH ₂ ) ₂ F], [ZA942; H, H, F, H, NHCH ₂ CHF ₂ ], [ZA943; H, H, F, H, NHCH ₂ CHF ₃ ], [ZA944; H, H, F, H, NH (CH ₂ ) ₃ F], [ZA945; H, H, F , H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA946; H, H, F, H, NH (CH ₂ ) ₂ CF ₃ ], [ZA947; H, H, F, H, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA948; H, H, F, H, NHCH ₂ Cl], [ZA949; H, H, F, H, NH (CH ₂ ) ₂ Cl], [ZA950; H, H, F, H, NH (CH ₂ ) ₃ Cl], [ZA951; H, H, F, H, NH (CH ₂ ) ₄ Cl], [ZA952; H, H, F, H, NH (CH ₂ ) ₅ Cl] , [ZA953; H, H, F, H, NHCH ₂ OMe], [ZA954; H, H, F, H, NH (CH ₂ ) ₂ OMe], [ZA955; H, H, F, H, NH (CH ₂ ) ₃ OMe], [ ZA956; H, H, F, H, NH (CH ₂ ) ₄ OMe], [ZA957; H, H, F, H, NHCH ₂ OEt], [ZA958; H, H, F, H, NH (CH ₂ ) ₂ OEt], [ZA959; H, H, F, H, NH (CH ₂ ) ₃ OEt], [ZA960; H, H, F, H, NHCH ₂ OPr], [ZA961; H, H, F, H, NH (CH ₂ ) ₂ OPr], [ZA962; H, H, F, H, NH (CH ₂ ) ₃ OPr], [ZA963; H, H, F, H, NHCH ₂ CN], [ZA964; H, H, F, H, NH (CH ₂ ) ₂ CN], [ZA965; H, H, F, H, NH (CH ₂ ) ₃ CN], [ZA966; H, H, F, H, NH ( CH ₂ ) ₄ CN], [ZA967; H, H, F, H, NH (CH ₂ ) ₅ CN], [ZA968; H, H, F, H, NHCH ₂ CH = CH ₂ ], [ZA969; H , H, F, H, NHCH ₂ C≡CH], [ZA970; H, H, F, H, NHCH ₂ C≡CCH ₃ ], [ZA971; H, H, F, H, NHCH ₂ Ph], [ ZA972; H, H, F, H, NHCH ₂ (2-Py)], [ZA973; H, H, F, H, NHCH ₂ (3-Py)], [ZA974; H, H, F, H, NHCH ₂ (4-Py)], [ZA975; H, H, F, H, NH (CH ₂ ) ₂ Ph], [ZA976; H, H, F, H, NH (CH ₂ ) ₂ (2-Py )], [ZA977; H, H, F, H, NH (CH ₂ ) ₂ (3-Py)], [ZA978; H, H, F, H, NH (CH ₂ ) ₂ (4-Py)] , [ZA979; H, H, F, H, NHPh], [ZA980; H, H, F, H, NH (2-Py)], [ZA981; H, H, F, H, NH (3-Py )], [ZA982; H, H, F, H, NH (4-Py)], [ZA983; H, H, F, H, NMe ₂ ], [ZA984; H, H, F, H, NMeEt] , [ZA985; H, H, F, H, NMePr], [ZA986; H, H, F, H, NMeBu], [ZA987; H, H, F, H, NMePen], [ZA988; H, H, F, H, NMeHex], [ZA989; H, H, F, H, NMe (i-Pr)], [ZA990; H, H, F, H, NMe (i-Bu) ], [ZA991; H, H, F, H, NMe (c-Pr)], [ZA992; H, H, F, H, NMe (c-Bu)], [ZA993; H, H, F, H , NMe (c-Pen)], [ZA994; H, H, F, H, NMe (c-Hex)], [ZA995; H, H, F, H, NMeCH ₂ (c-Pr)], [ZA996 ; H, H, F, H, NMeCH ₂ (c-Bu)], [ZA997; H, H, F, H, NMeCH ₂ (c-Pen)], [ZA998; H, H, F, H, NMeCH ₂ (c-Hex)], [ZA999; H, H, F, H, NMeCH ₂ F], [ZA1000; H, H, F, H, NMeCHF ₂ ],

[ZA1001; H, H, F, H, NMeCF ₃ ], [ZA1002; H, H, F, H, NMe (CH ₂ ) ₂ F], [ZA1003; H, H, F, H, NMeCH ₂ CHF ₂ ], [ZA1004; H, H, F, H, NMeCH ₂ CHF ₃ ], [ZA1005; H, H, F, H, NMe (CH ₂ ) ₃ F], [ZA1006; H, H, F, H, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA1007; H, H, F, H, NMe (CH ₂ ) ₂ CF ₃ ], [ZA1008; H, H, F, H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA1009; H, H, F, H, NMeCH ₂ Cl], [ZA1010; H, H, F, H, NMe (CH ₂ ) ₂ Cl], [ZA1011; H, H, F, H, NMe (CH ₂ ) ₃ Cl], [ZA1012; H, H, F, H, NMe (CH ₂ ) ₄ Cl], [ZA1013; H, H, F, H, NMe (CH ₂ ) ₅ Cl], [ZA1014 ; H, H, F, H, NMeCH ₂ OMe], [ZA1015; H, H, F, H, NMe (CH ₂ ) ₂ OMe], [ZA1016; H, H, F, H, NMe (CH ₂ ) ₃ OMe], [ZA1017; H, H, F, H, NMe (CH ₂ ) ₄ OMe], [ZA1018; H, H, F, H, NMeCH ₂ OEt], [ZA1019; H, H, F, H , NMe (CH ₂ ) ₂ OEt], [ZA1020; H, H, F, H, NMe (CH ₂ ) ₃ OEt], [ZA1021; H, H, F, H, NMeCH ₂ OPr], [ZA1022; H , H, F, H, NMe (CH ₂ ) ₂ OPr], [ZA1023; H, H, F, H, NMe (CH ₂ ) ₃ OPr], [ZA1024; H, H, F, H, NMeCH ₂ CN ], [ZA1025; H, H, F, H, NMe (CH ₂ ) ₂ CN], [ZA1026; H, H, F, H, NMe (CH ₂ ) ₃ CN], [ZA1027; H, H, F , H, NMe (CH ₂ ) ₄ CN], [ZA1028; H, H, F, H, NMe (CH ₂ ) ₅ CN], [ZA1029; H, H, F, H, NMeCH ₂ CH = CH ₂ ] , [ZA1030; H, H, F, H, NMeCH ₂ C≡CH], [ZA1031; H, H, F, H, NMeCH ₂ C≡CCH ₃ ], [ZA1032; H, H, F, H, NMeCH ₂ Ph], [ZA1033; H, H, F, H, NMeCH ₂ (2-Py)], [ZA1034; H, H, F , H, NMeCH ₂ (3-Py)], [ZA1035; H, H, F, H, NMeCH ₂ (4-Py)], [ZA1036; H, H, F, H, NMe (CH ₂ ) ₂ Ph ], [ZA1037; H, H, F, H, NMe (CH ₂ ) ₂ (2-Py)], [ZA1038; H, H, F, H, NMe (CH ₂ ) ₂ (3-Py)], [ZA1039; H, H, F, H, NMe (CH ₂ ) ₂ (4-Py)], [ZA1040; H, H, F, H, NMePh], [ZA1041; H, H, F, H, NMe (2-Py)], [ZA1042; H, H, F, H, NMe (3-Py)], [ZA1043; H, H, F, H, NMe (4-Py)], [ZA1044; H, H, F, H, NEt ₂ ], [ZA1045; H, H, F, H, NEtPr], [ZA1046; H, H, F, H, NEtBu], [ZA1047; H, H, F, H, NEtPen ], [ZA1048; H, H, F, H, NEtHex], [ZA1049; H, H, F, H, NEt (i-Pr)], [ZA1050; H, H, F, H, NEt (i- Bu)], [ZA1051; H, H, F, H, NEt (c-Pr)], [ZA1052; H, H, F, H, NEt (c-Bu)], [ZA1053; H, H, F , H, NEt (c-Pen)], [ZA1054; H, H, F, H, NEt (c-Hex)], [ZA1055; H, H, F, H, NEtCH ₂ (c-Pr)], [ZA1056; H, H, F, H, NEtCH ₂ (c-Bu)], [ZA1057; H, H, F, H, NEtCH ₂ (c-Pen)], [ZA1058; H, H, F, H , NEtCH ₂ (c-Hex)], [ZA1059; H, H, F, H, NEtCH ₂ F], [ZA1060; H, H, F, H, NEtCHF ₂ ], [ZA1061; H, H, F, H, NEtCF ₃ ], [ZA1062; H, H, F, H, NEt (CH ₂ ) ₂ F], [ZA1063; H, H, F, H, NEtCH ₂ CHF ₂ ], [ZA1064; H, H, F, H, NEtCH ₂ CHF ₃ ], [ZA1065; H, H, F, H, NEt (CH ₂ ) ₃ F], [ZA1066; H, H, F, H, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA1067; H, H, F, H, NEt (CH ₂ ) ₂ CF ₃ ], [ZA1068; H, H, F, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA1069; H, H, F, H, NEtCH ₂ Cl], [ZA1070; H, H, F, H, NEt (CH ₂ ) ₂ Cl ], [ZA1071; H, H, F, H, NEt (CH ₂ ) ₃ Cl], [ZA1072; H, H, F, H, NEt (CH ₂ ) ₄ Cl], [ZA1073; H, H, F , H, NEt (CH ₂ ) ₅ Cl], [ZA1074; H, H, F, H, NEtCH ₂ OMe], [ZA1075; H, H, F, H, NEt (CH ₂ ) ₂ OMe], [ZA1076 ; H, H, F, H, NEt (CH ₂ ) ₃ OMe], [ZA1077; H, H, F, H, NEt (CH ₂ ) ₄ OMe], [ZA1078; H, H, F, H, NEtCH ₂ OEt], [ZA1079; H, H, F, H, NEt (CH ₂ ) ₂ OEt], [ZA1080; H, H, F, H, NEt (CH ₂ ) ₃ OEt], [ZA1081; H, H , F, H, NEtCH ₂ OPr], [ZA1082; H, H, F, H, NEt (CH ₂ ) ₂ OPr], [ZA1083; H, H, F, H, NEt (CH ₂ ) ₃ OPr], [ZA1084; H, H, F, H, NEtCH ₂ CN], [ZA1085; H, H, F, H, NEt (CH ₂ ) ₂ CN], [ZA1086; H, H, F, H, NEt (CH _{2) 3 CN], [ZA1087} ; H, H, F, H, NEt (CH 2) 4 CN], [ZA1088; H, H, F, H, NEt (CH 2) 5 CN], [ZA1089; H , H, F, H, NEtCH ₂ CH = CH ₂ ], [ZA1090; H, H, F, H, NEtCH ₂ C≡CH], [ZA1091; H, H, F, H, NEtCH ₂ C≡CCH ₃ ], [ZA1092; H, H, F, H, NEtCH ₂ Ph], [ZA1093; H, H, F, H, NEtCH ₂ (2-Py)], [ZA1094; H, H, F, H, NEtCH ₂ (3-Py)], [ZA1095; H, H, F, H, NEtCH ₂ (4-Py)], [ZA1096; H, H, F, H, NEt (CH ₂ ) ₂ Ph], [ZA1097; H, H, F, H, NEt (CH ₂ ) ₂ (2-Py)], [ZA1098; H, H, F, H, NEt (CH ₂ ) ₂ (3-Py)], [ZA1099; H, H, F, H, NEt (CH ₂ ) ₂ (4-Py)], [ZA1100; H, H, F, H, NEtPh], [ZA1101; H, H, F, H, NEt (2-Py)], [ZA1102; H, H, F, H, NEt (3-Py)], [ZA1103; H, H, F, H, NEt (4- Py)], [ZA1104; H, H, F, H, Pyr], [ZA1105; H, H, F, H, Pip], [ZA1106; H, H, F, H, Mor], [ZA1107; H , H, F, H, OMe], [ZA1108; H, H, F, H, OEt], [ZA1109; H, H, F, H, OPr], [ZA1110; H, H, F, H, OBu ], [ZA1111; H, H, F, H, OPen], [ZA1112; H, H, F, H, OHex], [ZA1113; H, H, F, H, O (i-Pr)], [ ZA1114; H, H, F, H, O (i-Bu)], [ZA1115; H, H, F, H, O (c-Pr)], [ZA1116; H, H, F, H, O ( c-Bu)], [ZA1117; H, H, F, H, O (c-Pen)], [ZA1118; H, H, F, H, O (c-Hex)], [ZA1119; H, H , F, H, OCH ₂ (c-Pr)], [ZA1120; H, H, F, H, OCH ₂ (c-Bu)], [ZA1121; H, H, F, H, OCH ₂ (c- Pen)], [ZA1122; H, H, F, H, OCH ₂ (c-Hex)], [ZA1123; H, H, F, H, OCH ₂ F], [ZA1124; H, H, F, H , OCHF ₂ ], [ZA1125; H, H, F, H, OCF ₃ ], [ZA1126; H, H, F, H, O (CH ₂ ) ₂ F], [ZA1127; H, H, F, H , OCH ₂ CHF ₂ ], [ZA1128; H, H, F, H, OCH ₂ CHF ₃ ], [ZA1129; H, H, F, H, O (CH ₂ ) ₃ F], [ZA1130; H, H , F, H, O (CH ₂ ) ₂ CHF ₂ ], [ZA1131; H, H, F, H, O (CH ₂ ) ₂ CF ₃ ], [ZA1132; H, H, F, H, OCH ₂ CH (CF ₃ ) ₂ ], [Z A1133; H, H, F, H, OCH ₂ Cl], [ZA1134; H, H, F, H, O (CH ₂ ) ₂ Cl], [ZA1135; H, H, F, H, O (CH _{2 ) 3 Cl], [ZA1136;} H, H, F, H, O (CH 2) 4 Cl], [ZA1137; H, H, F, H, O (CH 2) 5 Cl], [ZA1138; H, H, F, H, OCH ₂ OMe], [ZA1139; H, H, F, H, O (CH ₂ ) ₂ OMe], [ZA1140; H, H, F, H, O (CH ₂ ) ₃ OMe] , [ZA1141; H, H, F, H, O (CH ₂ ) ₄ OMe], [ZA1142; H, H, F, H, OCH ₂ OEt], [ZA1143; H, H, F, H, O ( _{CH 2) 2 OEt], [} ZA1144; H, H, F, H, O (CH 2) 3 OEt], [ZA1145; H, H, F, H, OCH 2 OPr], [ZA1146; H, H, F, H, O (CH ₂ ) ₂ OPr], [ZA1147; H, H, F, H, O (CH ₂ ) ₃ OPr], [ZA1148; H, H, F, H, OCH ₂ CN], [ ZA1149; H, H, F, H, O (CH ₂ ) ₂ CN], [ZA1150; H, H, F, H, O (CH ₂ ) ₃ CN], [ZA1151; H, H, F, H, O (CH ₂ ) ₄ CN], [ZA1152; H, H, F, H, O (CH ₂ ) ₅ CN], [ZA1153; H, H, F, H, OCH ₂ CH = CH ₂ ], [ZA1154 ; H, H, F, H, OCH ₂ C≡CH], [ZA1155; H, H, F, H, OCH ₂ C≡CCH ₃ ], [ZA1156; H, H, F, H, OCH ₂ Ph] , [ZA1157; H, H, F, H, OCH ₂ (2-Py)], [ZA1158; H, H, F, H, OCH ₂ (3-Py)], [ZA1159; H, H, F, H, OCH ₂ (4-Py)], [ZA1160; H, H, F, H, O (CH ₂ ) ₂ Ph], [ZA1161; H, H, F, H, O (CH ₂ ) ₂ (2 -Py)], [ZA1162; H, H, F, H, O (CH ₂ ) ₂ (3-Py)], [ZA1163; H, H, F, H, O (CH ₂ ) ₂ (4-Py )], [ZA1164; H, H, F, H, OPh], [ZA1165; H, H, F, H, O (2-Py)], [ZA 1166; H, H, F, H, O (3-Py)], [ZA1167; H, H, F, H, O (4-Py)], [ZA1168; H, H, F, H, Me] , [ZA1169; H, H, F, H, Et], [ZA1170; H, H, F, H, Pr], [ZA1171; H, H, F, H, Bu], [ZA1172; H, H, F, H, Pen], [ZA1173; H, H, F, H, Hex], [ZA1174; H, H, F, H, (i-Pr)], [ZA1175; H, H, F, H, (i-Bu)], [ZA1176; H, H, F, H, (c-Pr)], [ZA1177; H, H, F, H, (c-Bu)], [ZA1178; H, H, F, H, (c-Pen)], [ZA1179; H, H, F, H, (c-Hex)], [ZA1180; H, H, F, H, CH ₂ (c-Pr)], [ ZA1181; H, H, F, H, CH ₂ (c-Bu)], [ZA1182; H, H, F, H, CH ₂ (c-Pen)], [ZA1183; H, H, F, H, CH ₂ (c-Hex)], [ZA1184; H, H, F, H, CH ₂ F], [ZA1185; H, H, F, H, CHF ₂ ], [ZA1186; H, H, F, H , CF ₃ ], [ZA1187; H, H, F, H, (CH ₂ ) ₂ F], [ZA1188; H, H, F, H, CH ₂ CHF ₂ ], [ZA1189; H, H, F, H, CH ₂ CHF ₃ ], [ZA1190; H, H, F, H, (CH ₂ ) ₃ F], [ZA1191; H, H, F, H, (CH ₂ ) ₂ CHF ₂ ], [ZA1192; H, H, F, H, (CH ₂ ) ₂ CF ₃ ], [ZA1193; H, H, F, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA1194; H, H, F, H, CH ₂ Cl], [ZA1195; H, H, F, H, (CH ₂ ) ₂ Cl], [ZA1196; H, H, F, H, (CH ₂ ) ₃ Cl], [ZA1197; H, H, F , H, (CH ₂ ) ₄ Cl], [ZA1198; H, H, F, H, (CH ₂ ) ₅ Cl], [ZA1199; H, H, F, H, CH ₂ OMe], [ZA1200; H , H, F, H, (CH ₂ ) ₂ OMe], [ZA1201; H, H, F, H, (CH ₂ ) ₃ OMe], [ZA1202; H, H, F, H, (CH ₂ ) ₄ OMe], [ZA1203; H, H, F, H, CH ₂ OEt], [ZA1204; H, H, F, H, (CH ₂ ) ₂ OEt], [ZA1205; H, H, F, H, (CH ₂ ) ₃ OEt], [ZA1206; H, H, F, H, CH ₂ OPr], [ZA1207; H, H, F, H, (CH ₂ ) ₂ OPr], [ZA1208; H, H, F, H, (CH ₂ ) ₃ OPr], [ ZA1209; H, H, F, H, CH ₂ CN], [ZA1210; H, H, F, H, (CH ₂ ) ₂ CN], [ZA1211; H, H, F, H, (CH ₂ ) ₃ CN], [ZA1212; H, H, F, H, (CH ₂ ) ₄ CN], [ZA1213; H, H, F, H, (CH ₂ ) ₅ CN], [ZA1214; H, H, F, H, CH ₂ CH = CH ₂ ], [ZA1215; H, H, F, H, CH ₂ C≡CH], [ZA1216; H, H, F, H, CH ₂ C≡CCH ₃ ], [ZA1217; H, H, F, H, CH ₂ Ph], [ZA1218; H, H, F, H, CH ₂ (2-Py)], [ZA1219; H, H, F, H, CH ₂ (3-Py )], [ZA1220; H, H, F, H, CH ₂ (4-Py)], [ZA1221; H, H, F, H, (CH ₂ ) ₂ Ph], [ZA1222; H, H, F , H, (CH ₂ ) ₂ (2-Py)], [ZA1223; H, H, F, H, (CH ₂ ) ₂ (3-Py)], [ZA1224; H, H, F, H, ( CH ₂ ) ₂ (4-Py)], [ZA1225; H, H, F, H, Ph], [ZA1226; H, H, F, H, 2-Py], [ZA1227; H, H, F, H, 3-Py], [ZA1228; H, H, F, H, 4-Py], [ZA1229; H, H, F, F, NHMe], [ZA1230; H, H, F, F, NHEt] , [ZA1231; H, H, F, F, NHPr], [ZA1232; H, H, F, F, NHBu], [ZA1233; H, H, F, F, NHPen], [ZA1234; H, H, F, F, NHHex], [ZA1235; H, H, F, F, NH (i-Pr)], [ZA1236; H, H, F, F, NH (i-Bu)], [ZA1237; H, H, F, F, NH (c-Pr)], [ZA1238; H, H, F, F, NH (c-Bu)], [ZA1239; H, H, F, F, NH (c-Pen) ], [ZA12 40; H, H, F, F, NH (c-Hex)], [ZA1241; H, H, F, F, NHCH ₂ (c-Pr)], [ZA1242; H, H, F, F, NHCH ₂ (c-Bu)], [ZA1243; H, H, F, F, NHCH ₂ (c-Pen)], [ZA1244; H, H, F, F, NHCH ₂ (c-Hex)], [ZA1245 ; H, H, F, F, NHCH ₂ F], [ZA1246; H, H, F, F, NHCHF ₂ ], [ZA1247; H, H, F, F, NHCF ₃ ], [ZA1248; H, H , F, F, NH (CH ₂ ) ₂ F], [ZA1249; H, H, F, F, NHCH ₂ CHF ₂ ], [ZA1250; H, H, F, F, NHCH ₂ CHF ₃ ],

[ZA1251; H, H, F, F, NH (CH ₂ ) ₃ F], [ZA1252; H, H, F, F, NH (CH ₂ ) ₂ CHF ₂ ], [ZA1253; H, H, F, F, NH (CH ₂ ) ₂ CF ₃ ], [ZA1254; H, H, F, F, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA1255; H, H, F, F, NHCH ₂ Cl], [ ZA1256; H, H, F, F, NH (CH ₂ ) ₂ Cl], [ZA1257; H, H, F, F, NH (CH ₂ ) ₃ Cl], [ZA1258; H, H, F, F, NH (CH ₂ ) ₄ Cl], [ZA1259; H, H, F, F, NH (CH ₂ ) ₅ Cl], [ZA1260; H, H, F, F, NHCH ₂ OMe], [ZA1261; H, H, F, F, NH (CH ₂ ) ₂ OMe], [ZA1262; H, H, F, F, NH (CH ₂ ) ₃ OMe], [ZA1263; H, H, F, F, NH (CH ₂ ) ₄ OMe], [ZA1264; H, H, F, F, NHCH ₂ OEt], [ZA1265; H, H, F, F, NH (CH ₂ ) ₂ OEt], [ZA1266; H, H, F, F, NH (CH ₂ ) ₃ OEt], [ZA1267; H, H, F, F, NHCH ₂ OPr], [ZA1268; H, H, F, F, NH (CH ₂ ) ₂ OPr], [ZA1269; H, H, F, F, NH (CH ₂ ) ₃ OPr], [ZA1270; H, H, F, F, NHCH ₂ CN], [ZA1271; H, H, F, F, NH (CH ₂ ) ₂ CN], [ZA1272; H, H, F, F, NH (CH ₂ ) ₃ CN], [ZA1273; H, H, F, F, NH (CH ₂ ) ₄ CN], [ZA1274; H, H, F, F, NH (CH ₂ ) ₅ CN], [ZA1275; H, H, F, F, NHCH ₂ CH = CH ₂ ], [ZA1276; H, H, F, F, NHCH ₂ C≡CH], [ZA1277; H, H, F, F, NHCH ₂ C≡CCH ₃ ], [ZA1278; H, H, F, F, NHCH ₂ Ph], [ZA1279; H, H, F, F, NHCH ₂ (2 -Py)], [ZA1280; H, H, F, F, NHCH ₂ (3-Py)], [ZA1281; H, H, F, F, NHCH ₂ (4-Py)], [ZA1282; H, H, F, F, N H (CH ₂ ) ₂ Ph], [ZA1283; H, H, F, F, NH (CH ₂ ) ₂ (2-Py)], [ZA1284; H, H, F, F, NH (CH ₂ ) ₂ (3-Py)], [ZA1285; H, H, F, F, NH (CH ₂ ) ₂ (4-Py)], [ZA1286; H, H, F, F, NHPh], [ZA1287; H, H, F, F, NH (2-Py)], [ZA1288; H, H, F, F, NH (3-Py)], [ZA1289; H, H, F, F, NH (4-Py) ], [ZA1290; H, H, F, F, NMe ₂ ], [ZA1291; H, H, F, F, NMeEt], [ZA1292; H, H, F, F, NMePr], [ZA1293; H, H, F, F, NMeBu], [ZA1294; H, H, F, F, NMePen], [ZA1295; H, H, F, F, NMeHex], [ZA1296; H, H, F, F, NMe ( i-Pr)], [ZA1297; H, H, F, F, NMe (i-Bu)], [ZA1298; H, H, F, F, NMe (c-Pr)], [ZA1299; H, H , F, F, NMe (c-Bu)], [ZA1300; H, H, F, F, NMe (c-Pen)], [ZA1301; H, H, F, F, NMe (c-Hex)] , [ZA1302; H, H, F, F, NMeCH ₂ (c-Pr)], [ZA1303; H, H, F, F, NMeCH ₂ (c-Bu)], [ZA1304; H, H, F, F, NMeCH ₂ (c-Pen)], [ZA1305; H, H, F, F, NMeCH ₂ (c-Hex)], [ZA1306; H, H, F, F, NMeCH ₂ F], [ZA1307; H, H, F, F, NMeCHF ₂ ], [ZA1308; H, H, F, F, NMeCF ₃ ], [ZA1309; H, H, F, F, NMe (CH ₂ ) ₂ F], [ZA1310; H, H, F, F, NMeCH ₂ CHF ₂ ], [ZA1311; H, H, F, F, NMeCH ₂ CHF ₃ ], [ZA1312; H, H, F, F, NMe (CH ₂ ) ₃ F] , [ZA1313; H, H, F, F, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA1314; H, H, F, F, NMe (CH ₂ ) ₂ CF ₃ ], [ZA1315; H, H, F, F, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA1316; H, H, F, F, NMeCH ₂ Cl], [ZA1317; H, H, F, F, NMe (CH ₂ ) ₂ Cl], [ZA1318; H, H, F, F, NMe (CH ₂ ) ₃ Cl], [ZA1319; H, H, F, F, NMe (CH ₂ ) ₄ Cl], [ZA1320; H, H, F, F, NMe (CH ₂ ) ₅ Cl], [ZA1321; H, H, F, F, NMeCH ₂ OMe], [ ZA1322; H, H, F, F, NMe (CH ₂ ) ₂ OMe], [ZA1323; H, H, F, F, NMe (CH ₂ ) ₃ OMe], [ZA1324; H, H, F, F, NMe (CH ₂ ) ₄ OMe], [ZA1325; H, H, F, F, NMeCH ₂ OEt], [ZA1326; H, H, F, F, NMe (CH ₂ ) ₂ OEt], [ZA1327; H, H, F, F, NMe (CH ₂ ) ₃ OEt], [ZA1328; H, H, F, F, NMeCH ₂ OPr], [ZA1329; H, H, F, F, NMe (CH ₂ ) ₂ OPr] , [ZA1330; H, H, F, F, NMe (CH ₂ ) ₃ OPr], [ZA1331; H, H, F, F, NMeCH ₂ CN], [ZA1332; H, H, F, F, NMe ( _{CH 2) 2 CN], [} ZA1333; H, H, F, F, NMe (CH 2) 3 CN], [ZA1334; H, H, F, F, NMe (CH 2) 4 CN], [ZA1335; H, H, F, F, NMe (CH ₂ ) ₅ CN], [ZA1336; H, H, F, F, NMeCH ₂ CH = CH ₂ ], [ZA1337; H, H, F, F, NMeCH ₂ C ≡CH], [ZA1338; H, H, F, F, NMeCH ₂ C≡CCH ₃ ], [ZA1339; H, H, F, F, NMeCH ₂ Ph], [ZA1340; H, H, F, F, NMeCH ₂ (2-Py)], [ZA1341; H, H, F, F, NMeCH ₂ (3-Py)], [ZA1342; H, H, F, F, NMeCH ₂ (4-Py)], [ ZA1343; H, H, F, F, NMe (CH ₂ ) ₂ Ph], [ZA1344; H, H, F, F, NMe (CH ₂ ) ₂ (2-Py)], [ZA1345; H, H, F, F, NMe (CH ₂ ) ₂ (3-Py)], [ZA1346; H, H, F, F, NMe (CH ₂ ) ₂ (4-Py)], [ZA1347; H, H, F, F, NMePh], [ZA1348; H, H, F, F, NMe (2-Py)], [ZA1349; H, H, F, F, NMe (3-Py)], [ ZA1350; H, H, F, F, NMe (4-Py)], [ZA1351; H, H, F, F, NEt ₂ ], [ZA1352; H, H, F, F, NEtPr], [ZA1353; H, H, F, F, NEtBu], [ZA1354; H, H, F, F, NEtPen], [ZA1355; H, H, F, F, NEtHex], [ZA1356; H, H, F, F, NEt (i-Pr)], [ZA1357; H, H, F, F, NEt (i-Bu)], [ZA1358; H, H, F, F, NEt (c-Pr)], [ZA1359; H , H, F, F, NEt (c-Bu)], [ZA1360; H, H, F, F, NEt (c-Pen)], [ZA1361; H, H, F, F, NEt (c-Hex )], [ZA1362; H, H, F, F, NEtCH ₂ (c-Pr)], [ZA1363; H, H, F, F, NEtCH ₂ (c-Bu)], [ZA1364; H, H, F, F, NEtCH ₂ (c-Pen)], [ZA1365; H, H, F, F, NEtCH ₂ (c-Hex)], [ZA1366; H, H, F, F, NEtCH ₂ F], [ ZA1367; H, H, F, F, NEtCHF ₂ ], [ZA1368; H, H, F, F, NEtCF ₃ ], [ZA1369; H, H, F, F, NEt (CH ₂ ) ₂ F], [ ZA1370; H, H, F, F, NEtCH ₂ CHF ₂ ], [ZA1371; H, H, F, F, NEtCH ₂ CHF ₃ ], [ZA1372; H, H, F, F, NEt (CH ₂ ) ₃ F], [ZA1373; H, H, F, F, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA1374; H, H, F, F, NEt (CH ₂ ) ₂ CF ₃ ], [ZA1375; H, H, F, F, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA1376; H, H, F, F, NEtCH ₂ Cl], [ZA1377; H, H, F, F, NEt (CH ₂ ) ₂ Cl ], [ZA1378; H, H, F, F, NEt (CH ₂ ) ₃ Cl], [ZA1379; H, H, F, F, NEt (CH ₂ ) ₄ Cl], [ZA1380; H, H, F , F, NEt (CH ₂ ) ₅ Cl], [ZA1381; H, H, F , F, NEtCH ₂ OMe], [ZA1382; H, H, F, F, NEt (CH ₂ ) ₂ OMe], [ZA1383; H, H, F, F, NEt (CH ₂ ) ₃ OMe], [ZA1384 ; H, H, F, F, NEt (CH ₂ ) ₄ OMe], [ZA1385; H, H, F, F, NEtCH ₂ OEt], [ZA1386; H, H, F, F, NEt (CH ₂ ) ₂ OEt], [ZA1387; H, H, F, F, NEt (CH ₂ ) ₃ OEt], [ZA1388; H, H, F, F, NEtCH ₂ OPr], [ZA1389; H, H, F, F , NEt (CH ₂ ) ₂ OPr], [ZA1390; H, H, F, F, NEt (CH ₂ ) ₃ OPr], [ZA1391; H, H, F, F, NEtCH ₂ CN], [ZA1392; H , H, F, F, NEt (CH ₂ ) ₂ CN], [ZA1393; H, H, F, F, NEt (CH ₂ ) ₃ CN], [ZA1394; H, H, F, F, NEt (CH _{2) 4 CN], [ZA1395} ; H, H, F, F, NEt (CH 2) 5 CN], [ZA1396; H, H, F, F, NEtCH 2 CH = CH 2], [ZA1397; H, H, F, F, NEtCH ₂ C≡CH], [ZA1398; H, H, F, F, NEtCH ₂ C≡CCH ₃ ], [ZA1399; H, H, F, F, NEtCH ₂ Ph], [ZA1400 ; H, H, F, F, NEtCH ₂ (2-Py)], [ZA1401; H, H, F, F, NEtCH ₂ (3-Py)], [ZA1402; H, H, F, F, NEtCH ₂ (4-Py)], [ZA1403; H, H, F, F, NEt (CH ₂ ) ₂ Ph], [ZA1404; H, H, F, F, NEt (CH ₂ ) ₂ (2-Py) ], [ZA1405; H, H, F, F, NEt (CH ₂ ) ₂ (3-Py)], [ZA1406; H, H, F, F, NEt (CH ₂ ) ₂ (4-Py)], [ZA1407; H, H, F, F, NEtPh], [ZA1408; H, H, F, F, NEt (2-Py)], [ZA1409; H, H, F, F, NEt (3-Py) ], [ZA1410; H, H, F, F, NEt (4-Py)], [ZA1411; H, H, F, F, Pyr], [ZA1412; H, H, F, F, Pip], [ ZA1413; H, H, F, F, Mor], [ZA1414; H, H, F, F, OMe], [ZA1415; H, H, F, F, OEt], [ZA1416; H, H, F, F, OPr], [ ZA1417; H, H, F, F, OBu], [ZA1418; H, H, F, F, OPen], [ZA1419; H, H, F, F, OHex], [ZA1420; H, H, F, F, O (i-Pr)], [ZA1421; H, H, F, F, O (i-Bu)], [ZA1422; H, H, F, F, O (c-Pr)], [ZA1423 ; H, H, F, F, O (c-Bu)], [ZA1424; H, H, F, F, O (c-Pen)], [ZA1425; H, H, F, F, O (c -Hex)], [ZA1426; H, H, F, F, OCH ₂ (c-Pr)], [ZA1427; H, H, F, F, OCH ₂ (c-Bu)], [ZA1428; H, H, F, F, OCH ₂ (c-Pen)], [ZA1429; H, H, F, F, OCH ₂ (c-Hex)], [ZA1430; H, H, F, F, OCH ₂ F] , [ZA1431; H, H, F, F, OCHF ₂ ], [ZA1432; H, H, F, F, OCF ₃ ], [ZA1433; H, H, F, F, O (CH ₂ ) ₂ F] , [ZA1434; H, H, F, F, OCH ₂ CHF ₂ ], [ZA1435; H, H, F, F, OCH ₂ CHF ₃ ], [ZA1436; H, H, F, F, O (CH ₂ ) ₃ F], [ZA1437; H, H, F, F, O (CH ₂ ) ₂ CHF ₂ ], [ZA1438; H, H, F, F, O (CH ₂ ) ₂ CF ₃ ], [ZA1439; H, H, F, F, OCH ₂ CH (CF ₃ ) ₂ ], [ZA1440; H, H, F, F, OCH ₂ Cl], [ZA1441; H, H, F, F, O (CH ₂ ) ₂ Cl], [ZA1442; H, H, F, F, O (CH ₂ ) ₃ Cl], [ZA1443; H, H, F, F, O (CH ₂ ) ₄ Cl], [ZA1444; H, H , F, F, O (CH ₂ ) ₅ Cl], [ZA1445; H, H, F, F, OCH ₂ OMe], [ZA1446; H, H, F, F, O (CH ₂ ) ₂ OMe], [ZA1447; H, H, F, F, O (CH ₂ ) ₃ OMe], [ZA1448; H, H, F, F, O (CH ₂ ) ₄ OMe], [ZA1449; H, H, F, F , O _{CH 2 OEt], [ZA1450;} H, H, F, F, O (CH 2) 2 OEt], [ZA1451; H, H, F, F, O (CH 2) 3 OEt], [ZA1452; H, H, F, F, OCH ₂ OPr], [ZA1453; H, H, F, F, O (CH ₂ ) ₂ OPr], [ZA1454; H, H, F, F, O (CH ₂ ) ₃ OPr] , [ZA1455; H, H, F, F, OCH ₂ CN], [ZA1456; H, H, F, F, O (CH ₂ ) ₂ CN], [ZA1457; H, H, F, F, O ( _{CH 2) 3 CN], [} ZA1458; H, H, F, F, O (CH 2) 4 CN], [ZA1459; H, H, F, F, O (CH 2) 5 CN], [ZA1460; H, H, F, F, OCH ₂ CH = CH ₂ ], [ZA1461; H, H, F, F, OCH ₂ C≡CH], [ZA1462; H, H, F, F, OCH ₂ C≡CCH ₃ ], [ZA1463; H, H, F, F, OCH ₂ Ph], [ZA1464; H, H, F, F, OCH ₂ (2-Py)], [ZA1465; H, H, F, F, OCH ₂ (3-Py)], [ZA1466; H, H, F, F, OCH ₂ (4-Py)], [ZA1467; H, H, F, F, O (CH ₂ ) ₂ Ph], [ ZA1468; H, H, F, F, O (CH ₂ ) ₂ (2-Py)], [ZA1469; H, H, F, F, O (CH ₂ ) ₂ (3-Py)], [ZA1470; H, H, F, F, O (CH ₂ ) ₂ (4-Py)], [ZA1471; H, H, F, F, OPh], [ZA1472; H, H, F, F, O (2- Py)], [ZA1473; H, H, F, F, O (3-Py)], [ZA1474; H, H, F, F, O (4-Py)], [ZA1475; H, H, F , F, Me], [ZA1476; H, H, F, F, Et], [ZA1477; H, H, F, F, Pr], [ZA1478; H, H, F, F, Bu], [ZA1479 ; H, H, F, F, Pen], [ZA1480; H, H, F, F, Hex], [ZA1481; H, H, F, F, (i-Pr)], [ZA1482; H, H , F, F, (i-Bu)], [ZA1483; H, H, F, F, (c-Pr)], [ZA1484; H, H, F, F, (c-Bu)], [ZA1485 ; H, H, F, F, (c-Pen) ], [ZA1486; H, H, F, F, (c-Hex)], [ZA1487; H, H, F, F, CH ₂ (c-Pr)], [ZA1488; H, H, F, F , CH ₂ (c-Bu)], [ZA1489; H, H, F, F, CH ₂ (c-Pen)], [ZA1490; H, H, F, F, CH ₂ (c-Hex)], [ZA1491; H, H, F, F, CH ₂ F], [ZA1492; H, H, F, F, CHF ₂ ], [ZA1493; H, H, F, F, CF ₃ ], [ZA1494; H , H, F, F, (CH ₂ ) ₂ F], [ZA1495; H, H, F, F, CH ₂ CHF ₂ ], [ZA1496; H, H, F, F, CH ₂ CHF ₃ ], [ ZA1497; H, H, F, F, (CH ₂ ) ₃ F], [ZA1498; H, H, F, F, (CH ₂ ) ₂ CHF ₂ ], [ZA1499; H, H, F, F, ( CH ₂ ) ₂ CF ₃ ], [ZA1500; H, H, F, F, CH
₂ CH (CF ₃ ) ₂ ],

[ZA1501; H, H, F, F, CH ₂ Cl], [ZA1502; H, H, F, F, (CH ₂ ) ₂ Cl], [ZA1503; H, H, F, F, (CH ₂ ) ₃ Cl], [ZA1504; H, H, F, F, (CH ₂ ) ₄ Cl], [ZA1505; H, H, F, F, (CH ₂ ) ₅ Cl], [ZA1506; H, H, F , F, CH ₂ OMe], [ZA1507; H, H, F, F, (CH ₂ ) ₂ OMe], [ZA1508; H, H, F, F, (CH ₂ ) ₃ OMe], [ZA1509; H , H, F, F, (CH ₂ ) ₄ OMe], [ZA1510; H, H, F, F, CH ₂ OEt], [ZA1511; H, H, F, F, (CH ₂ ) ₂ OEt], [ZA1512; H, H, F, F, (CH ₂ ) ₃ OEt], [ZA1513; H, H, F, F, CH ₂ OPr], [ZA1514; H, H, F, F, (CH ₂ ) ₂ OPr], [ZA1515; H, H, F, F, (CH ₂ ) ₃ OPr], [ZA1516; H, H, F, F, CH ₂ CN], [ZA1517; H, H, F, F, (CH ₂ ) ₂ CN], [ZA1518; H, H, F, F, (CH ₂ ) ₃ CN], [ZA1519; H, H, F, F, (CH ₂ ) ₄ CN], [ZA1520; H , H, F, F, (CH ₂ ) ₅ CN], [ZA1521; H, H, F, F, CH ₂ CH = CH ₂ ], [ZA1522; H, H, F, F, CH ₂ C≡CH ], [ZA1523; H, H, F, F, CH ₂ C≡CCH ₃ ], [ZA1524; H, H, F, F, CH ₂ Ph], [ZA1525; H, H, F, F, CH ₂ (2-Py)], [ZA1526; H, H, F, F, CH ₂ (3-Py)], [ZA1527; H, H, F, F, CH ₂ (4-Py)], [ZA1528; H, H, F, F, (CH ₂ ) ₂ Ph], [ZA1529; H, H, F, F, (CH ₂ ) ₂ (2-Py)], [ZA1530; H, H, F, F, (CH ₂ ) ₂ (3-Py)], [ZA1531; H, H, F, F, (CH ₂ ) ₂ (4-Py)], [ZA1532; H, H, F, F, Ph], [ ZA1533; H, H, F, F, 2-Py], [ZA1534; H, H, F, F, 3-Py], [ZA1535; H, H, F, F, 4-Py], [ZA1536; H, H, Cl, H, NHMe], [ZA1537; H, H, Cl, H, NHEt], [ZA1538; H, H, Cl, H, NHPr], [ ZA1539; H, H, Cl, H, NHBu], [ZA1540; H, H, Cl, H, NHPen], [ZA1541; H, H, Cl, H, NHHex], [ZA1542; H, H, Cl, H, NH (i-Pr)], [ZA1543; H, H, Cl, H, NH (i-Bu)], [ZA1544; H, H, Cl, H, NH (c-Pr)], [ZA1545 ; H, H, Cl, H, NH (c-Bu)], [ZA1546; H, H, Cl, H, NH (c-Pen)], [ZA1547; H, H, Cl, H, NH (c -Hex)], [ZA1548; H, H, Cl, H, NHCH ₂ (c-Pr)], [ZA1549; H, H, Cl, H, NHCH ₂ (c-Bu)], [ZA1550; H, H, Cl, H, NHCH ₂ (c-Pen)], [ZA1551; H, H, Cl, H, NHCH ₂ (c-Hex)], [ZA1552; H, H, Cl, H, NHCH ₂ F] , [ZA1553; H, H, Cl, H, NHCHF ₂ ], [ZA1554; H, H, Cl, H, NHCF ₃ ], [ZA1555; H, H, Cl, H, NH (CH ₂ ) ₂ F] , [ZA1556; H, H, Cl, H, NHCH ₂ CHF ₂ ], [ZA1557; H, H, Cl, H, NHCH ₂ CHF ₃ ], [ZA1558; H, H, Cl, H, NH (CH ₂ ) ₃ F], [ZA1559; H, H, Cl, H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA1560; H, H, Cl, H, NH (CH ₂ ) ₂ CF ₃ ], [ZA1561; H, H, Cl, H, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA1562; H, H, Cl, H, NHCH ₂ Cl], [ZA1563; H, H, Cl, H, NH (CH ₂ ) ₂ Cl], [ZA1564; H, H, Cl, H, NH (CH ₂ ) ₃ Cl], [ZA1565; H, H, Cl, H, NH (CH ₂ ) ₄ Cl], [ZA1566; H, H , Cl, H, NH (CH ₂ ) ₅ Cl], [ZA1567; H, H, Cl, H, NHCH ₂ OMe], [ZA1568; H, H, Cl, H, NH (CH ₂ ) ₂ OMe], [ZA1569; H, H, Cl, H , NH (CH ₂ ) ₃ OMe], [ZA1570; H, H, Cl, H, NH (CH ₂ ) ₄ OMe], [ZA1571; H, H, Cl, H, NHCH ₂ OEt], [ZA1572; H , H, Cl, H, NH (CH ₂ ) ₂ OEt], [ZA1573; H, H, Cl, H, NH (CH ₂ ) ₃ OEt], [ZA1574; H, H, Cl, H, NHCH ₂ OPr ], [ZA1575; H, H, Cl, H, NH (CH ₂ ) ₂ OPr], [ZA1576; H, H, Cl, H, NH (CH ₂ ) ₃ OPr], [ZA1577; H, H, Cl , H, NHCH ₂ CN], [ZA1578; H, H, Cl, H, NH (CH ₂ ) ₂ CN], [ZA1579; H, H, Cl, H, NH (CH ₂ ) ₃ CN], [ZA1580 ; H, H, Cl, H, NH (CH ₂ ) ₄ CN], [ZA1581; H, H, Cl, H, NH (CH ₂ ) ₅ CN], [ZA1582; H, H, Cl, H, NHCH ₂ CH = CH ₂ ], [ZA1583; H, H, Cl, H, NHCH ₂ C≡CH], [ZA1584; H, H, Cl, H, NHCH ₂ C≡CCH ₃ ], [ZA1585; H, H , Cl, H, NHCH ₂ Ph], [ZA1586; H, H, Cl, H, NHCH ₂ (2-Py)], [ZA1587; H, H, Cl, H, NHCH ₂ (3-Py)], [ZA1588; H, H, Cl, H, NHCH ₂ (4-Py)], [ZA1589; H, H, Cl, H, NH (CH ₂ ) ₂ Ph], [ZA1590; H, H, Cl, H , NH (CH ₂ ) ₂ (2-Py)], [ZA1591; H, H, Cl, H, NH (CH ₂ ) ₂ (3-Py)], [ZA1592; H, H, Cl, H, NH (CH ₂ ) ₂ (4-Py)], [ZA1593; H, H, Cl, H, NHPh], [ZA1594; H, H, Cl, H, NH (2-Py)], [ZA1595; H, H, Cl, H, NH (3-Py)], [ZA1596; H, H, Cl, H, NH (4-Py)], [ZA1597; H, H, Cl, H, NMe ₂ ], [ZA1598 ; H, H, Cl, H, NMeEt], [ZA1599; H, H, Cl, H, NMePr], [ZA1600; H, H, Cl, H, NMeBu], [ZA1601; H, H, Cl, H , NMePen ], [ZA1602; H, H, Cl, H, NMeHex], [ZA1603; H, H, Cl, H, NMe (i-Pr)], [ZA1604; H, H, Cl, H, NMe (i- Bu)], [ZA1605; H, H, Cl, H, NMe (c-Pr)], [ZA1606; H, H, Cl, H, NMe (c-Bu)], [ZA1607; H, H, Cl , H, NMe (c-Pen)], [ZA1608; H, H, Cl, H, NMe (c-Hex)], [ZA1609; H, H, Cl, H, NMeCH ₂ (c-Pr)], [ZA1610; H, H, Cl, H, NMeCH ₂ (c-Bu)], [ZA1611; H, H, Cl, H, NMeCH ₂ (c-Pen)], [ZA1612; H, H, Cl, H , NMeCH ₂ (c-Hex)], [ZA1613; H, H, Cl, H, NMeCH ₂ F], [ZA1614; H, H, Cl, H, NMeCHF ₂ ], [ZA1615; H, H, Cl, H, NMeCF ₃ ], [ZA1616; H, H, Cl, H, NMe (CH ₂ ) ₂ F], [ZA1617; H, H, Cl, H, NMeCH ₂ CHF ₂ ], [ZA1618; H, H, Cl, H, NMeCH ₂ CHF ₃ ], [ZA1619; H, H, Cl, H, NMe (CH ₂ ) ₃ F], [ZA1620; H, H, Cl, H, NMe (CH ₂ ) ₂ CHF ₂ ] , [ZA1621; H, H, Cl, H, NMe (CH ₂ ) ₂ CF ₃ ], [ZA1622; H, H, Cl, H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA1623; H, H, Cl, H, NMeCH ₂ Cl], [ZA1624; H, H, Cl, H, NMe (CH ₂ ) ₂ Cl], [ZA1625; H, H, Cl, H, NMe (CH ₂ ) ₃ Cl], [ ZA1626; H, H, Cl, H, NMe (CH ₂ ) ₄ Cl], [ZA1627; H, H, Cl, H, NMe (CH ₂ ) ₅ Cl], [ZA1628; H, H, Cl, H, NMeCH ₂ OMe], [ZA1629; H, H, Cl, H, NMe (CH ₂ ) ₂ OMe], [ZA1630; H, H, Cl, H, NMe (CH ₂ ) ₃ OMe], [ZA1631; H, H, Cl, H, NMe (CH ₂ ) ₄ OMe], [ZA1632; H, H, Cl, H, NMeCH ₂ OEt], [ZA1633; H, H, Cl, H, NMe (CH ₂ ) ₂ OEt], [ZA1634; H, H, Cl, H, NMe (CH ₂ ) ₃ OEt], [ZA1635; H, H, Cl, H, NMeCH ₂ OPr] , [ZA1636; H, H, Cl, H, NMe (CH ₂ ) ₂ OPr], [ZA1637; H, H, Cl, H, NMe (CH ₂ ) ₃ OPr], [ZA1638; H, H, Cl, H, NMeCH ₂ CN], [ZA1639; H, H, Cl, H, NMe (CH ₂ ) ₂ CN], [ZA1640; H, H, Cl, H, NMe (CH ₂ ) ₃ CN], [ZA1641; H, H, Cl, H, NMe (CH ₂ ) ₄ CN], [ZA1642; H, H, Cl, H, NMe (CH ₂ ) ₅ CN], [ZA1643; H, H, Cl, H, NMeCH ₂ CH = CH ₂ ], [ZA1644; H, H, Cl, H, NMeCH ₂ C≡CH], [ZA1645; H, H, Cl, H, NMeCH ₂ C≡CCH ₃ ], [ZA1646; H, H, Cl, H, NMeCH ₂ Ph], [ZA1647; H, H, Cl, H, NMeCH ₂ (2-Py)], [ZA1648; H, H, Cl, H, NMeCH ₂ (3-Py)], [ ZA1649; H, H, Cl, H, NMeCH ₂ (4-Py)], [ZA1650; H, H, Cl, H, NMe (CH ₂ ) ₂ Ph], [ZA1651; H, H, Cl, H, NMe (CH ₂ ) ₂ (2-Py)], [ZA1652; H, H, Cl, H, NMe (CH ₂ ) ₂ (3-Py)], [ZA1653; H, H, Cl, H, NMe ( CH ₂ ) ₂ (4-Py)], [ZA1654; H, H, Cl, H, NMePh], [ZA1655; H, H, Cl, H, NMe (2-Py)], [ZA1656; H, H , Cl, H, NMe (3-Py)], [ZA1657; H, H, Cl, H, NMe (4-Py)], [ZA1658; H, H, Cl, H, NEt ₂ ], [ZA1659; H, H, Cl, H, NEtPr], [ZA1660; H, H, Cl, H, NEtBu], [ZA1661; H, H, Cl, H, NEtPen], [ZA1662; H, H, Cl, H, NEtHex], [ZA1663; H, H, Cl, H, NEt (i-Pr)], [ZA1664; H, H, Cl, H, NEt (i-Bu)], [ZA1665 ; H, H, Cl, H, NEt (c-Pr)], [ZA1666; H, H, Cl, H, NEt (c-Bu)], [ZA1667; H, H, Cl, H, NEt (c -Pen)], [ZA1668; H, H, Cl, H, NEt (c-Hex)], [ZA1669; H, H, Cl, H, NEtCH ₂ (c-Pr)], [ZA1670; H, H , Cl, H, NEtCH ₂ (c-Bu)], [ZA1671; H, H, Cl, H, NEtCH ₂ (c-Pen)], [ZA1672; H, H, Cl, H, NEtCH ₂ (c- Hex)], [ZA1673; H, H, Cl, H, NEtCH ₂ F], [ZA1674; H, H, Cl, H, NEtCHF ₂ ], [ZA1675; H, H, Cl, H, NEtCF ₃ ], [ZA1676; H, H, Cl, H, NEt (CH ₂ ) ₂ F], [ZA1677; H, H, Cl, H, NEtCH ₂ CHF ₂ ], [ZA1678; H, H, Cl, H, NEtCH ₂ CHF ₃ ], [ZA1679; H, H, Cl, H, NEt (CH ₂ ) ₃ F], [ZA1680; H, H, Cl, H, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA1681; H, H, Cl, H, NEt (CH ₂ ) ₂ CF ₃ ], [ZA1682; H, H, Cl, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA1683; H, H, Cl, H, NEtCH ₂ Cl], [ZA1684; H, H, Cl, H, NEt (CH ₂ ) ₂ Cl], [ZA1685; H, H, Cl, H, NEt (CH ₂ ) ₃ Cl], [ZA1686; H, H, Cl, H, NEt (CH ₂ ) ₄ Cl], [ZA1687; H, H, Cl, H, NEt (CH ₂ ) ₅ Cl], [ZA1688; H, H, Cl, H, NEtCH ₂ OMe], [ ZA1689; H, H, Cl, H, NEt (CH ₂ ) ₂ OMe], [ZA1690; H, H, Cl, H, NEt (CH ₂ ) ₃ OMe], [ZA1691; H, H, Cl, H, NEt (CH ₂ ) ₄ OMe], [ZA1692; H, H, Cl, H, NEtCH ₂ OEt], [ZA1693; H, H, Cl, H, NEt (CH ₂ ) ₂ OEt], [ZA1694; H, H, Cl, H, NEt (CH ₂ ) ₃ OEt], [ZA1695; H, H, Cl, H, NEtCH ₂ OPr], [ZA1696; H, H, Cl, H, NEt (CH ₂ ) ₂ OPr], [ZA1697; H, H, Cl, H, NEt (CH ₂ ) ₃ OPr], [ZA1698; H, H, Cl, H , NEtCH ₂ CN], [ZA1699; H, H, Cl, H, NEt (CH ₂ ) ₂ CN], [ZA1700; H, H, Cl, H, NEt (CH ₂ ) ₃ CN], [ZA1701; H , H, Cl, H, NEt (CH ₂ ) ₄ CN], [ZA1702; H, H, Cl, H, NEt (CH ₂ ) ₅ CN], [ZA1703; H, H, Cl, H, NEtCH ₂ CH = CH ₂ ], [ZA1704; H, H, Cl, H, NEtCH ₂ C≡CH], [ZA1705; H, H, Cl, H, NEtCH ₂ C≡CCH ₃ ], [ZA1706; H, H, Cl , H, NEtCH ₂ Ph], [ZA1707; H, H, Cl, H, NEtCH ₂ (2-Py)], [ZA1708; H, H, Cl, H, NEtCH ₂ (3-Py)], [ZA1709 ; H, H, Cl, H, NEtCH ₂ (4-Py)], [ZA1710; H, H, Cl, H, NEt (CH ₂ ) ₂ Ph], [ZA1711; H, H, Cl, H, NEt (CH ₂ ) ₂ (2-Py)], [ZA1712; H, H, Cl, H, NEt (CH ₂ ) ₂ (3-Py)], [ZA1713; H, H, Cl, H, NEt (CH ₂ ) ₂ (4-Py)], [ZA1714; H, H, Cl, H, NEtPh], [ZA1715; H, H, Cl, H, NEt (2-Py)], [ZA1716; H, H, Cl, H, NEt (3-Py)], [ZA1717; H, H, Cl, H, NEt (4-Py)], [ZA1718; H, H, Cl, H, Pyr], [ZA1719; H, H, Cl, H, Pip], [ZA1720; H, H, Cl, H, Mor], [ZA1721; H, H, Cl, H, OMe], [ZA1722; H, H, Cl, H, OEt] , [ZA1723; H, H, Cl, H, OPr], [ZA1724; H, H, Cl, H, OBu], [ZA1725; H, H, Cl, H, OPen], [ZA1726; H, H, Cl, H, OHex], [ZA1727; H, H, Cl, H, O (i-Pr)], [ZA1728; H, H, Cl, H, O (i-Bu)], [ZA1729; H, H, Cl, H, O (c-Pr) ], [ZA1730; H, H, Cl, H, O (c-Bu)], [ZA1731; H, H, Cl, H, O (c-Pen)], [ZA1732; H, H, Cl, H , O (c-Hex)], [ZA1733; H, H, Cl, H, OCH ₂ (c-Pr)], [ZA1734; H, H, Cl, H, OCH ₂ (c-Bu)], [ ZA1735; H, H, Cl, H, OCH ₂ (c-Pen)], [ZA1736; H, H, Cl, H, OCH ₂ (c-Hex)], [ZA1737; H, H, Cl, H, OCH ₂ F], [ZA1738; H, H, Cl, H, OCHF ₂ ], [ZA1739; H, H, Cl, H, OCF ₃ ], [ZA1740; H, H, Cl, H, O (CH ₂ ) ₂ F], [ZA1741; H, H, Cl, H, OCH ₂ CHF ₂ ], [ZA1742; H, H, Cl, H, OCH ₂ CHF ₃ ], [ZA1743; H, H, Cl, H, O (CH ₂ ) ₃ F], [ZA1744; H, H, Cl, H, O (CH ₂ ) ₂ CHF ₂ ], [ZA1745; H, H, Cl, H, O (CH ₂ ) ₂ CF ₃ ] , [ZA1746; H, H, Cl, H, OCH ₂ CH (CF
_{3) 2], [ZA1747;} H, H, Cl, H, OCH 2 Cl], [ZA1748; H, H, Cl, H, O (CH 2) 2 Cl], [ZA1749; H, H, Cl, H, O (CH ₂ ) ₃ Cl], [ZA1750; H, H, Cl, H, O (CH ₂ ) ₄ Cl],

[ZA1751; H, H, Cl, H, O (CH ₂ ) ₅ Cl], [ZA1752; H, H, Cl, H, OCH ₂ OMe], [ZA1753; H, H, Cl, H, O (CH ₂ ) ₂ OMe], [ZA1754; H, H, Cl, H, O (CH ₂ ) ₃ OMe], [ZA1755; H, H, Cl, H, O (CH ₂ ) ₄ OMe], [ZA1756; H , H, Cl, H, OCH ₂ OEt], [ZA1757; H, H, Cl, H, O (CH ₂ ) ₂ OEt], [ZA1758; H, H, Cl, H, O (CH ₂ ) ₃ OEt ], [ZA1759; H, H, Cl, H, OCH ₂ OPr], [ZA1760; H, H, Cl, H, O (CH ₂ ) ₂ OPr], [ZA1761; H, H, Cl, H, O (CH ₂ ) ₃ OPr], [ZA1762; H, H, Cl, H, OCH ₂ CN], [ZA1763; H, H, Cl, H, O (CH ₂ ) ₂ CN], [ZA1764; H, H , Cl, H, O (CH ₂ ) ₃ CN], [ZA1765; H, H, Cl, H, O (CH ₂ ) ₄ CN], [ZA1766; H, H, Cl, H, O (CH ₂ ) ₅ CN], [ZA1767; H, H, Cl, H, OCH ₂ CH = CH ₂ ], [ZA1768; H, H, Cl, H, OCH ₂ C≡CH], [ZA1769; H, H, Cl, H, OCH ₂ C≡CCH ₃ ], [ZA1770; H, H, Cl, H, OCH ₂ Ph], [ZA1771; H, H, Cl, H, OCH ₂ (2-Py)], [ZA1772; H , H, Cl, H, OCH ₂ (3-Py)], [ZA1773; H, H, Cl, H, OCH ₂ (4-Py)], [ZA1774; H, H, Cl, H, O (CH ₂ ) ₂ Ph], [ZA1775; H, H, Cl, H, O (CH ₂ ) ₂ (2-Py)], [ZA1776; H, H, Cl, H, O (CH ₂ ) ₂ (3- Py)], [ZA1777; H, H, Cl, H, O (CH ₂ ) ₂ (4-Py)], [ZA1778; H, H, Cl, H, OPh], [ZA1779; H, H, Cl , H, O (2-Py)], [ZA1780; H, H, Cl, H, O (3-Py)], [ZA1781; H, H, Cl, H, O (4-Py)], [ ZA1782; H, H, Cl, H, Me], [ZA1783; H, H, Cl, H, E t], [ZA1784; H, H, Cl, H, Pr], [ZA1785; H, H, Cl, H, Bu], [ZA1786; H, H, Cl, H, Pen], [ZA1787; H, H, Cl, H, Hex], [ZA1788; H, H, Cl, H, (i-Pr)], [ZA1789; H, H, Cl, H, (i-Bu)], [ZA1790; H, H, Cl, H, (c-Pr)], [ZA1791; H, H, Cl, H, (c-Bu)], [ZA1792; H, H, Cl, H, (c-Pen)], [ ZA1793; H, H, Cl, H, (c-Hex)], [ZA1794; H, H, Cl, H, CH ₂ (c-Pr)], [ZA1795; H, H, Cl, H, CH ₂ (c-Bu)], [ZA1796; H, H, Cl, H, CH ₂ (c-Pen)], [ZA1797; H, H, Cl, H, CH ₂ (c-Hex)], [ZA1798; H, H, Cl, H, CH ₂ F], [ZA1799; H, H, Cl, H, CHF ₂ ], [ZA1800; H, H, Cl, H, CF ₃ ], [ZA1801; H, H, Cl, H, (CH ₂ ) ₂ F], [ZA1802; H, H, Cl, H, CH ₂ CHF ₂ ], [ZA1803; H, H, Cl, H, CH ₂ CHF ₃ ], [ZA1804; H , H, Cl, H, (CH ₂ ) ₃ F], [ZA1805; H, H, Cl, H, (CH ₂ ) ₂ CHF ₂ ], [ZA1806; H, H, Cl, H, (CH ₂ ) ₂ CF ₃ ], [ZA1807; H, H, Cl, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA1808; H, H, Cl, H, CH ₂ Cl], [ZA1809; H, H, Cl , H, (CH ₂ ) ₂ Cl], [ZA1810; H, H, Cl, H, (CH ₂ ) ₃ Cl], [ZA1811; H, H, Cl, H, (CH ₂ ) ₄ Cl], [ ZA1812; H, H, Cl, H, (CH ₂ ) ₅ Cl], [ZA1813; H, H, Cl, H, CH ₂ OMe], [ZA1814; H, H, Cl, H, (CH ₂ ) ₂ OMe], [ZA1815; H, H, Cl, H, (CH ₂ ) ₃ OMe], [ZA1816; H, H, Cl, H, (CH ₂ ) ₄ OMe], [ZA1817; H, H, Cl, H, CH ₂ OEt], [ZA1818; H, H, Cl, H, (CH ₂ ) ₂ OEt], [ZA181 9; H, H, Cl, H, (CH ₂ ) ₃ OEt], [ZA1820; H, H, Cl, H, CH ₂ OPr], [ZA1821; H, H, Cl, H, (CH ₂ ) ₂ OPr], [ZA1822; H, H, Cl, H, (CH ₂ ) ₃ OPr], [ZA1823; H, H, Cl, H, CH ₂ CN], [ZA1824; H, H, Cl, H, ( _{CH 2) 2 CN], [} ZA1825; H, H, Cl, H, (CH 2) 3 CN], [ZA1826; H, H, Cl, H, (CH 2) 4 CN], [ZA1827; H, H, Cl, H, (CH ₂ ) ₅ CN], [ZA1828; H, H, Cl, H, CH ₂ CH = CH ₂ ], [ZA1829; H, H, Cl, H, CH ₂ C≡CH] , [ZA1830; H, H, Cl, H, CH ₂ C≡CCH ₃ ], [ZA1831; H, H, Cl, H, CH ₂ Ph], [ZA1832; H, H, Cl, H, CH ₂ ( 2-Py)], [ZA1833; H, H, Cl, H, CH ₂ (3-Py)], [ZA1834; H, H, Cl, H, CH ₂ (4-Py)], [ZA1835; H , H, Cl, H, (CH ₂ ) ₂ Ph], [ZA1836; H, H, Cl, H, (CH ₂ ) ₂ (2-Py)], [ZA1837; H, H, Cl, H, ( CH ₂ ) ₂ (3-Py)], [ZA1838; H, H, Cl, H, (CH ₂ ) ₂ (4-Py)], [ZA1839; H, H, Cl, H, Ph], [ZA1840 ; H, H, Cl, H, 2-Py], [ZA1841; H, H, Cl, H, 3-Py], [ZA1842; H, H, Cl, H, 4-Py], [ZA1843; H , H, Cl, Cl, NHMe], [ZA1844; H, H, Cl, Cl, NHEt], [ZA1845; H, H, Cl, Cl, NHPr], [ZA1846; H, H, Cl, Cl, NHBu ], [ZA1847; H, H, Cl, Cl, NHPen], [ZA1848; H, H, Cl, Cl, NHHex], [ZA1849; H, H, Cl, Cl, NH (i-Pr)], [ ZA1850; H, H, Cl, Cl, NH (i-Bu)], [ZA1851; H, H, Cl, Cl, NH (c-Pr)], [ZA1852; H, H, Cl, Cl, NH ( c-Bu)], [ZA1853; H, H, Cl, Cl, NH (c-Pen)], [ZA1854; H, H, Cl, Cl, NH (c-Hex)], [ZA1855; H, H, Cl, Cl, NHCH ₂ (c-Pr)], [ZA1856; H, H, Cl, Cl, NHCH ₂ ( c-Bu)], [ZA1857; H, H, Cl, Cl, NHCH ₂ (c-Pen)], [ZA1858; H, H, Cl, Cl, NHCH ₂ (c-Hex)], [ZA1859; H , H, Cl, Cl, NHCH ₂ F], [ZA1860; H, H, Cl, Cl, NHCHF ₂ ], [ZA1861; H, H, Cl, Cl, NHCF ₃ ], [ZA1862; H, H, Cl , Cl, NH (CH ₂ ) ₂ F], [ZA1863; H, H, Cl, Cl, NHCH ₂ CHF ₂ ], [ZA1864; H, H, Cl, Cl, NHCH ₂ CHF ₃ ], [ZA1865; H , H, Cl, Cl, NH (CH ₂ ) ₃ F], [ZA1866; H, H, Cl, Cl, NH (CH ₂ ) ₂ CHF ₂ ], [ZA1867; H, H, Cl, Cl, NH ( CH ₂ ) ₂ CF ₃ ], [ZA1868; H, H, Cl, Cl, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA1869; H, H, Cl, Cl, NHCH ₂ Cl], [ZA1870; H, H, Cl, Cl, NH (CH ₂ ) ₂ Cl], [ZA1871; H, H, Cl, Cl, NH (CH ₂ ) ₃ Cl], [ZA1872; H, H, Cl, Cl, NH (CH ₂ ) ₄ Cl], [ZA1873; H, H, Cl, Cl, NH (CH ₂ ) ₅ Cl], [ZA1874; H, H, Cl, Cl, NHCH ₂ OMe], [ZA1875; H, H, Cl, Cl, NH (CH ₂ ) ₂ OMe], [ZA1876; H, H, Cl, Cl, NH (CH ₂ ) ₃ OMe], [ZA1877; H, H, Cl, Cl, NH (CH ₂ ) ₄ OMe] , [ZA1878; H, H, Cl, Cl, NHCH ₂ OEt], [ZA1879; H, H, Cl, Cl, NH (CH ₂ ) ₂ OEt], [ZA1880; H, H, Cl, Cl, NH ( CH ₂ ) ₃ OEt], [ZA1881; H, H, Cl, Cl, NHCH ₂ OPr], [ZA1882; H, H, Cl, Cl, NH (CH ₂ ) ₂ OPr], [ZA1883; H, H, Cl, Cl, NH (CH ₂ ) ₃ OPr], [ZA1884; H, H, Cl, C l, NHCH ₂ CN], [ZA1885; H, H, Cl, Cl, NH (CH ₂ ) ₂ CN], [ZA1886; H, H, Cl, Cl, NH (CH ₂ ) ₃ CN], [ZA1887; H, H, Cl, Cl, NH (CH ₂ ) ₄ CN], [ZA1888; H, H, Cl, Cl, NH (CH ₂ ) ₅ CN], [ZA1889; H, H, Cl, Cl, NHCH ₂ CH = CH ₂ ], [ZA1890; H, H, Cl, Cl, NHCH ₂ C≡CH], [ZA1891; H, H, Cl, Cl, NHCH ₂ C≡CCH ₃ ], [ZA1892; H, H, Cl, Cl, NHCH ₂ Ph], [ZA1893; H, H, Cl, Cl, NHCH ₂ (2-Py)], [ZA1894; H, H, Cl, Cl, NHCH ₂ (3-Py)], [ ZA1895; H, H, Cl, Cl, NHCH ₂ (4-Py)], [ZA1896; H, H, Cl, Cl, NH (CH ₂ ) ₂ Ph], [ZA1897; H, H, Cl, Cl, NH (CH ₂ ) ₂ (2-Py)], [ZA1898; H, H, Cl, Cl, NH (CH ₂ ) ₂ (3-Py)], [ZA1899; H, H, Cl, Cl, NH ( CH ₂ ) ₂ (4-Py)], [ZA1900; H, H, Cl, Cl, NHPh], [ZA1901; H, H, Cl, Cl, NH (2-Py)], [ZA1902; H, H , Cl, Cl, NH (3-Py)], [ZA1903; H, H, Cl, Cl, NH (4-Py)], [ZA1904; H, H, Cl, Cl, NMe ₂ ], [ZA1905; H, H, Cl, Cl, NMeEt], [ZA1906; H, H, Cl, Cl, NMePr], [ZA1907; H, H, Cl, Cl, NMeBu], [ZA1908; H, H, Cl, Cl, NMePen], [ZA1909; H, H, Cl, Cl, NMeHex], [ZA1910; H, H, Cl, Cl, NMe (i-Pr)], [ZA1911; H, H, Cl, Cl, NMe (i -Bu)], [ZA1912; H, H, Cl, Cl, NMe (c-Pr)], [ZA1913; H, H, Cl, Cl, NMe (c-Bu)], [ZA1914; H, H, Cl, Cl, NMe (c-Pen)], [ZA1915; H, H, Cl, Cl, NMe (c-Hex)], [ZA1916; H, H, Cl, Cl, NMeCH ₂ (c-Pr)] , [ZA1917; H, H, Cl, Cl, NMeCH ₂ (c-Bu)], [ZA1918; H, H, Cl, Cl, NMeCH ₂ (c-Pen)], [ZA1919; H, H, Cl, Cl, NMeCH ₂ (c-Hex)], [ZA1920; H, H, Cl, Cl, NMeCH ₂ F], [ZA1921; H, H, Cl, Cl, NMeCHF ₂ ], [ZA1922; H, H, Cl , Cl, NMeCF ₃ ], [ZA1923; H, H, Cl, Cl, NMe (CH ₂ ) ₂ F], [ZA1924; H, H, Cl, Cl, NMeCH ₂ CHF ₂ ], [ZA1925; H, H , Cl, Cl, NMeCH ₂ CHF ₃ ], [ZA1926; H, H, Cl, Cl, NMe (CH ₂ ) ₃ F], [ZA1927; H, H, Cl, Cl, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA1928; H, H, Cl, Cl, NMe (CH ₂ ) ₂ CF ₃ ], [ZA1929; H, H, Cl, Cl, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA1930; H, H , Cl, Cl, NMeCH ₂ Cl], [ZA1931; H, H, Cl, Cl, NMe (CH ₂ ) ₂ Cl], [ZA1932; H, H, Cl, Cl, NMe (CH ₂ ) ₃ Cl], [ZA1933; H, H, Cl, Cl, NMe (CH ₂ ) ₄ Cl], [ZA1934; H, H, Cl, Cl, NMe (CH ₂ ) ₅ Cl], [ZA1935; H, H, Cl, Cl , NMeCH ₂ OMe], [ZA1936; H, H, Cl, Cl, NMe (CH ₂ ) ₂ OMe], [ZA1937; H, H, Cl, Cl, NMe (CH ₂ ) ₃ OMe], [ZA1938; H , H, Cl, Cl, NMe (CH ₂ ) ₄ OMe], [ZA1939; H, H, Cl, Cl, NMeCH ₂ OEt], [ZA1940; H, H, Cl, Cl, NMe (CH ₂ ) ₂ OEt ], [ZA1941; H, H, Cl, Cl, NMe (CH ₂ ) ₃ OEt], [ZA1942; H, H, Cl, Cl, NMeCH ₂ OPr], [ZA1943; H, H, Cl, Cl, NMe (CH ₂ ) ₂ OPr], [ZA1944; H, H, Cl, Cl, NMe (CH ₂ ) ₃ OPr], [ZA1945; H, H, Cl, Cl, NMeCH ₂ CN], [ZA1946; H, H , Cl, Cl, NMe (CH ₂ ) ₂ CN], [ZA1947; H, H, Cl, Cl, NMe (CH ₂ ) ₃ CN], [ZA1948; H, H, Cl, Cl, NMe (CH ₂ ) ₄ CN], [ZA1949; H, H, Cl, Cl, NMe (CH ₂ ) ₅ CN], [ZA1950; H, H, Cl, Cl, NMeCH ₂ CH = CH ₂ ], [ZA1951; H, H, Cl, Cl, NMeCH ₂ C≡CH], [ZA1952; H, H, Cl, Cl, NMeCH ₂ C≡CCH ₃ ], [ZA1953; H, H, Cl, Cl, NMeCH ₂ Ph], [ZA1954; H , H, Cl, Cl, NMeCH ₂ (2-Py)], [ZA1955; H, H, Cl, Cl, NMeCH ₂ (3-Py)], [ZA1956; H, H, Cl, Cl, NMeCH ₂ ( 4-Py)], [ZA1957; H, H, Cl, Cl, NMe (CH ₂ ) ₂ Ph], [ZA1958; H, H, Cl, Cl, NMe (CH ₂ ) ₂ (2-Py)], [ZA1959; H, H, Cl, Cl, NMe (CH ₂ ) ₂ (3-Py)], [ZA1960; H, H, Cl, Cl, NMe (CH ₂ ) ₂ (4-Py)], [ZA1961 ; H, H, Cl, Cl, NMePh], [ZA1962; H, H, Cl, Cl, NMe (2-Py)], [ZA1963; H, H, Cl, Cl, NMe (3-Py)], [ZA1964; H, H, Cl, Cl, NMe (4-Py)], [ZA1965; H, H, Cl, Cl, NEt ₂ ], [ZA1966; H, H, Cl, Cl, NEtPr], [ZA1967 ; H, H, Cl, Cl, NEtBu], [ZA1968; H, H, Cl, Cl, NEtPen], [ZA1969; H, H, Cl, Cl, NEtHex], [ZA1970; H, H, Cl, Cl , NEt (i-Pr)], [ZA1971; H, H, Cl, Cl, NEt (i-Bu)], [ZA1972; H, H, Cl, Cl, NEt (c-Pr)], [ZA1973; H, H, Cl, Cl, NEt (c-Bu)], [ZA1974; H, H, Cl, Cl, NEt (c-Pen)], [ZA1975; H, H, Cl, Cl, NEt (c- Hex)], [ZA1976; H, H, Cl, Cl, NEtCH ₂ (c-Pr)], [ZA1977; H, H, Cl, Cl, NEtCH ₂ (c- Bu)], [ZA1978; H, H, Cl, Cl, NEtCH ₂ (c-Pen)], [ZA1979; H, H, Cl, Cl, NEtCH ₂ (c-Hex)], [ZA1980; H, H , Cl, Cl, NEtCH ₂ F], [ZA1981; H, H, Cl, Cl, NEtCHF ₂ ], [ZA1982; H, H, Cl, Cl, NEtCF ₃ ], [ZA1983; H, H, Cl, Cl , NEt (CH ₂ ) ₂ F], [ZA1984; H, H, Cl, Cl, NEtCH ₂ CHF ₂ ], [ZA1985; H, H, Cl, Cl, NEtCH ₂ CHF ₃ ], [ZA1986; H, H , Cl, Cl, NEt (CH ₂ ) ₃ F], [ZA1987; H, H, Cl, Cl, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA1988; H, H, Cl, Cl, NEt (CH ₂ ) ₂ CF ₃ ], [ZA1989; H, H, Cl, Cl, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA1990; H, H, Cl, Cl, NEtCH ₂ Cl], [ZA1991; H, H, Cl, Cl, NEt (CH ₂ ) ₂ Cl], [ZA1992; H, H, Cl, Cl, NEt (CH ₂ ) ₃ Cl
], [ZA1993; H, H, Cl, Cl, NEt (CH ₂ ) ₄ Cl], [ZA1994; H, H, Cl, Cl, NEt (CH ₂ ) ₅ Cl], [ZA1995; H, H, Cl , Cl, NEtCH ₂ OMe], [ZA1996; H, H, Cl, Cl, NEt (CH ₂ ) ₂ OMe], [ZA1997; H, H, Cl, Cl, NEt (CH ₂ ) ₃ OMe], [ZA1998 ; H, H, Cl, Cl, NEt (CH ₂ ) ₄ OMe], [ZA1999; H, H, Cl, Cl, NEtCH ₂ OEt], [ZA2000; H, H, Cl, Cl, NEt (CH ₂ ) ₂ OEt],

[ZA2001; H, H, Cl, Cl, NEt (CH ₂ ) ₃ OEt], [ZA2002; H, H, Cl, Cl, NEtCH ₂ OPr], [ZA2003; H, H, Cl, Cl, NEt (CH ₂ ) ₂ OPr], [ZA2004; H, H, Cl, Cl, NEt (CH ₂ ) ₃ OPr], [ZA2005; H, H, Cl, Cl, NEtCH ₂ CN], [ZA2006; H, H, Cl , Cl, NEt (CH ₂ ) ₂ CN], [ZA2007; H, H, Cl, Cl, NEt (CH ₂ ) ₃ CN], [ZA2008; H, H, Cl, Cl, NEt (CH ₂ ) ₄ CN ], [ZA2009; H, H, Cl, Cl, NEt (CH ₂ ) ₅ CN], [ZA2010; H, H, Cl, Cl, NEtCH ₂ CH = CH ₂ ], [ZA2011; H, H, Cl, Cl, NEtCH ₂ C≡CH], [ZA2012; H, H, Cl, Cl, NEtCH ₂ C≡CCH ₃ ], [ZA2013; H, H, Cl, Cl, NEtCH ₂ Ph], [ZA2014; H, H , Cl, Cl, NEtCH ₂ (2-Py)], [ZA2015; H, H, Cl, Cl, NEtCH ₂ (3-Py)], [ZA2016; H, H, Cl, Cl, NEtCH ₂ (4- Py)], [ZA2017; H, H, Cl, Cl, NEt (CH ₂ ) ₂ Ph], [ZA2018; H, H, Cl, Cl, NEt (CH ₂ ) ₂ (2-Py)], [ZA2019 ; H, H, Cl, Cl, NEt (CH ₂ ) ₂ (3-Py)], [ZA2020; H, H, Cl, Cl, NEt (CH ₂ ) ₂ (4-Py)], [ZA2021; H , H, Cl, Cl, NEtPh], [ZA2022; H, H, Cl, Cl, NEt (2-Py)], [ZA2023; H, H, Cl, Cl, NEt (3-Py)], [ZA2024 ; H, H, Cl, Cl, NEt (4-Py)], [ZA2025; H, H, Cl, Cl, Pyr], [ZA2026; H, H, Cl, Cl, Pip], [ZA2027; H, H, Cl, Cl, Mor], [ZA2028; H, H, Cl, Cl, OMe], [ZA2029; H, H, Cl, Cl, OEt], [ZA2030; H, H, Cl, Cl, OPr] , [ZA2031; H, H, Cl, Cl, OBu], [ZA2032; H, H, Cl, Cl, OPen], [Z A2033; H, H, Cl, Cl, OHex], [ZA2034; H, H, Cl, Cl, O (i-Pr)], [ZA2035; H, H, Cl, Cl, O (i-Bu)] , [ZA2036; H, H, Cl, Cl, O (c-Pr)], [ZA2037; H, H, Cl, Cl, O (c-Bu)], [ZA2038; H, H, Cl, Cl, O (c-Pen)], [ZA2039; H, H, Cl, Cl, O (c-Hex)], [ZA2040; H, H, Cl, Cl, OCH ₂ (c-Pr)], [ZA2041; H, H, Cl, Cl, OCH ₂ (c-Bu)], [ZA2042; H, H, Cl, Cl, OCH ₂ (c-Pen)], [ZA2043; H, H, Cl, Cl, OCH ₂ (c-Hex)], [ZA2044; H, H, Cl, Cl, OCH ₂ F], [ZA2045; H, H, Cl, Cl, OCHF ₂ ], [ZA2046; H, H, Cl, Cl, OCF ₃ ], [ZA2047; H, H, Cl, Cl, O (CH ₂ ) ₂ F], [ZA2048; H, H, Cl, Cl, OCH ₂ CHF ₂ ], [ZA2049; H, H, Cl, Cl , OCH ₂ CHF ₃ ], [ZA2050; H, H, Cl, Cl, O (CH ₂ ) ₃ F], [ZA2051; H, H, Cl, Cl, O (CH ₂ ) ₂ CHF ₂ ], [ZA2052 ; H, H, Cl, Cl, O (CH ₂ ) ₂ CF ₃ ], [ZA2053; H, H, Cl, Cl, OCH ₂ CH (CF ₃ ) ₂ ], [ZA2054; H, H, Cl, Cl , OCH ₂ Cl], [ZA2055; H, H, Cl, Cl, O (CH ₂ ) ₂ Cl], [ZA2056; H, H, Cl, Cl, O (CH ₂ ) ₃ Cl], [ZA2057; H , H, Cl, Cl, O (CH ₂ ) ₄ Cl], [ZA2058; H, H, Cl, Cl, O (CH ₂ ) ₅ Cl], [ZA2059; H, H, Cl, Cl, OCH ₂ OMe ], [ZA2060; H, H, Cl, Cl, O (CH ₂ ) ₂ OMe], [ZA2061; H, H, Cl, Cl, O (CH ₂ ) ₃ OMe], [ZA2062; H, H, Cl , Cl, O (CH ₂ ) ₄ OMe], [ZA2063; H, H, Cl, Cl, OCH ₂ OEt], [ZA2064; H, H, Cl, Cl, O (CH ₂ ) ₂ OEt], [ZA2065 ; H, H , Cl, Cl, O (CH ₂ ) ₃ OEt], [ZA2066; H, H, Cl, Cl, OCH ₂ OPr], [ZA2067; H, H, Cl, Cl, O (CH ₂ ) ₂ OPr], [ZA2068; H, H, Cl, Cl, O (CH ₂ ) ₃ OPr], [ZA2069; H, H, Cl, Cl, OCH ₂ CN], [ZA2070; H, H, Cl, Cl, O (CH _{2) 2 CN], [ZA2071} ; H, H, Cl, Cl, O (CH 2) 3 CN], [ZA2072; H, H, Cl, Cl, O (CH 2) 4 CN], [ZA2073; H , H, Cl, Cl, O (CH ₂ ) ₅ CN], [ZA2074; H, H, Cl, Cl, OCH ₂ CH = CH ₂ ], [ZA2075; H, H, Cl, Cl, OCH ₂ C≡ CH], [ZA2076; H, H, Cl, Cl, OCH ₂ C≡CCH ₃ ], [ZA2077; H, H, Cl, Cl, OCH ₂ Ph], [ZA2078; H, H, Cl, Cl, OCH ₂ (2-Py)], [ZA2079; H, H, Cl, Cl, OCH ₂ (3-Py)], [ZA2080; H, H, Cl, Cl, OCH ₂ (4-Py)], [ZA2081 ; H, H, Cl, Cl, O (CH ₂ ) ₂ Ph], [ZA2082; H, H, Cl, Cl, O (CH ₂ ) ₂ (2-Py)], [ZA2083; H, H, Cl , Cl, O (CH ₂ ) ₂ (3-Py)], [ZA2084; H, H, Cl, Cl, O (CH ₂ ) ₂ (4-Py)], [ZA2085; H, H, Cl, Cl , OPh], [ZA2086; H, H, Cl, Cl, O (2-Py)], [ZA2087; H, H, Cl, Cl, O (3-Py)], [ZA2088; H, H, Cl , Cl, O (4-Py)], [ZA2089; H, H, Cl, Cl, Me], [ZA2090; H, H, Cl, Cl, Et], [ZA2091; H, H, Cl, Cl, Pr], [ZA2092; H, H, Cl, Cl, Bu], [ZA2093; H, H, Cl, Cl, Pen], [ZA2094; H, H, Cl, Cl, Hex], [ZA2095; H, H, Cl, Cl, (i-Pr)], [ZA2096; H, H, Cl, Cl, (i-Bu)], [ZA2097; H, H, Cl, Cl, (c-Pr)], [ ZA2098; H, H, Cl, Cl, (c-Bu)], [ZA2099; H, H, Cl, Cl, (c-Pen)], [ZA2100; H, H, Cl, Cl, (c-Hex)], [ZA2101; H, H, Cl, Cl, CH ₂ (c-Pr )], [ZA2102; H, H, Cl, Cl, CH ₂ (c-Bu)], [ZA2103; H, H, Cl, Cl, CH ₂ (c-Pen)], [ZA2104; H, H, Cl, Cl, CH ₂ (c-Hex)], [ZA2105; H, H, Cl, Cl, CH ₂ F], [ZA2106; H, H, Cl, Cl, CHF ₂ ], [ZA2107; H, H , Cl, Cl, CF ₃ ], [ZA2108; H, H, Cl, Cl, (CH ₂ ) ₂ F], [ZA2109; H, H, Cl, Cl, CH ₂ CHF ₂ ], [ZA2110; H, H, Cl, Cl, CH ₂ CHF ₃ ], [ZA2111; H, H, Cl, Cl, (CH ₂ ) ₃ F], [ZA2112; H, H, Cl, Cl, (CH ₂ ) ₂ CHF ₂ ] , [ZA2113; H, H, Cl, Cl, (CH ₂ ) ₂ CF ₃ ], [ZA2114; H, H, Cl, Cl, CH ₂ CH (CF ₃ ) ₂ ], [ZA2115; H, H, Cl , Cl, CH ₂ Cl], [ZA2116; H, H, Cl, Cl, (CH ₂ ) ₂ Cl], [ZA2117; H, H, Cl, Cl, (CH ₂ ) ₃ Cl], [ZA2118; H , H, Cl, Cl, (CH ₂ ) ₄ Cl], [ZA2119; H, H, Cl, Cl, (CH ₂ ) ₅ Cl], [ZA2120; H, H, Cl, Cl, CH ₂ OMe], [ZA2121; H, H, Cl, Cl, (CH ₂ ) ₂ OMe], [ZA2122; H, H, Cl, Cl, (CH ₂ ) ₃ OMe], [ZA2123; H, H, Cl, Cl, ( CH ₂ ) ₄ OMe], [ZA2124; H, H, Cl, Cl, CH ₂ OEt], [ZA2125; H, H, Cl, Cl, (CH ₂ ) ₂ OEt], [ZA2126; H, H, Cl , Cl, (CH ₂ ) ₃ OEt], [ZA2127; H, H, Cl, Cl, CH ₂ OPr], [ZA2128; H, H, Cl, Cl, (CH ₂ ) ₂ OPr], [ZA2129; H , H, Cl, Cl, (CH ₂ ) ₃ OPr], [ZA2130; H, H, Cl, Cl, CH ₂ CN], [ZA2131; H, H, Cl, Cl, (CH _{2) 2 CN], [ZA2132} ; H, H, Cl, Cl, (CH 2) 3 CN], [ZA2133; H, H, Cl, Cl, (CH 2) 4 CN], [ZA2134; H, H , Cl, Cl, (CH ₂ ) ₅ CN], [ZA2135; H, H, Cl, Cl, CH ₂ CH = CH ₂ ], [ZA2136; H, H, Cl, Cl, CH ₂ C≡CH], [ZA2137; H, H, Cl, Cl, CH ₂ C≡CCH ₃ ], [ZA2138; H, H, Cl, Cl, CH ₂ Ph], [ZA2139; H, H, Cl, Cl, CH ₂ (2 -Py)], [ZA2140; H, H, Cl, Cl, CH ₂ (3-Py)], [ZA2141; H, H, Cl, Cl, CH ₂ (4-Py)], [ZA2142; H, H, Cl, Cl, (CH ₂ ) ₂ Ph], [ZA2143; H, H, Cl, Cl, (CH ₂ ) ₂ (2-Py)], [ZA2144; H, H, Cl, Cl, (CH ₂ ) ₂ (3-Py)], [ZA2145; H, H, Cl, Cl, (CH ₂ ) ₂ (4-Py)], [ZA2146; H, H, Cl, Cl, Ph], [ZA2147; H, H, Cl, Cl, 2-Py], [ZA2148; H, H, Cl, Cl, 3-Py], [ZA2149; H, H, Cl, Cl, 4-Py], [ZA2150; H, H, Et, H, NHMe], [ZA2151; H, H, Et, H, NHEt], [ZA2152; H, H, Et, H, NHPr], [ZA2153; H, H, Et, H, NHBu] , [ZA2154; H, H, Et, H, NHPen], [ZA2155; H, H, Et, H, NHHex], [ZA2156; H, H, Et, H, NH (i-Pr)], [ZA2157 ; H, H, Et, H, NH (i-Bu)], [ZA2158; H, H, Et, H, NH (c-Pr)], [ZA2159; H, H, Et, H, NH (c -Bu)], [ZA2160; H, H, Et, H, NH (c-Pen)], [ZA2161; H, H, Et, H, NH (c-Hex)], [ZA2162; H, H, Et, H, NHCH ₂ (c-Pr)], [ZA2163; H, H, Et, H, NHCH ₂ (c-Bu)], [ZA2164; H, H, Et, H, NHCH ₂ (c-Pen )], [ZA2165; H, H, Et, H, NHCH ₂ (c-Hex)], [ZA2166 ; H, H, Et, H, NHCH ₂ F], [ZA2167; H, H, Et, H, NHCHF ₂ ], [ZA2168; H, H, Et, H, NHCF ₃ ], [ZA2169; H, H , Et, H, NH (CH ₂ ) ₂ F], [ZA2170; H, H, Et, H, NHCH ₂ CHF ₂ ], [ZA2171; H, H, Et, H, NHCH ₂ CHF ₃ ], [ZA2172 ; H, H, Et, H, NH (CH ₂ ) ₃ F], [ZA2173; H, H, Et, H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA2174; H, H, Et, H, NH (CH ₂ ) ₂ CF ₃ ], [ZA2175; H, H, Et, H, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA2176; H, H, Et, H, NHCH ₂ Cl], [ZA2177; H, H, Et, H, NH (CH ₂ ) ₂ Cl], [ZA2178; H, H, Et, H, NH (CH ₂ ) ₃ Cl], [ZA2179; H, H, Et, H, NH ( _{CH 2) 4 Cl], [} ZA2180; H, H, Et, H, NH (CH 2) 5 Cl], [ZA2181; H, H, Et, H, NHCH 2 OMe], [ZA2182; H, H, Et, H, NH (CH ₂ ) ₂ OMe], [ZA2183; H, H, Et, H, NH (CH ₂ ) ₃ OMe], [ZA2184; H, H, Et, H, NH (CH ₂ ) ₄ OMe], [ZA2185; H, H, Et, H, NHCH ₂ OEt], [ZA2186; H, H, Et, H, NH (CH ₂ ) ₂ OEt], [ZA2187; H, H, Et, H, NH (CH ₂ ) ₃ OEt], [ZA2188; H, H, Et, H, NHCH ₂ OPr], [ZA2189; H, H, Et, H, NH (CH ₂ ) ₂ OPr], [ZA2190; H, H, Et, H, NH (CH ₂ ) ₃ OPr], [ZA2191; H, H, Et, H, NHCH ₂ CN], [ZA2192; H, H, Et, H, NH (CH ₂ ) ₂ CN] , [ZA2193; H, H, Et, H, NH (CH ₂ ) ₃ CN], [ZA2194; H, H, Et, H, NH (CH ₂ ) ₄ CN], [ZA2195; H, H, Et, H, NH (CH ₂ ) ₅ CN], [ZA2196; H, H, Et, H, NHCH ₂ CH = CH ₂ ], [ZA2197; H , H, Et, H, NHCH ₂ C≡CH], [ZA2198; H, H, Et, H, NHCH ₂ C≡CCH ₃ ], [ZA2199; H, H, Et, H, NHCH ₂ Ph], [ ZA2200; H, H, Et, H, NHCH ₂ (2-Py)], [ZA2201; H, H, Et, H, NHCH ₂ (3-Py)], [ZA2202; H, H, Et, H, NHCH ₂ (4-Py)], [ZA2203; H, H, Et, H, NH (CH ₂ ) ₂ Ph], [ZA2204; H, H, Et, H, NH (CH ₂ ) ₂ (2-Py )], [ZA2205; H, H, Et, H, NH (CH ₂ ) ₂ (3-Py)], [ZA2206; H, H, Et, H, NH (CH ₂ ) ₂ (4-Py)] , [ZA2207; H, H, Et, H, NHPh], [ZA2208; H, H, Et, H, NH (2-Py)], [ZA2209; H, H, Et, H, NH (3-Py )], [ZA2210; H, H, Et, H, NH (4-Py)], [ZA2211; H, H, Et, H, NMe ₂ ], [ZA2212; H, H, Et, H, NMeEt] , [ZA2213; H, H, Et, H, NMePr], [ZA2214; H, H, Et, H, NMeBu], [ZA2215; H, H, Et, H, NMePen], [ZA2216; H, H, Et, H, NMeHex], [ZA2217; H, H, Et, H, NMe (i-Pr)], [ZA2218; H, H, Et, H, NMe (i-Bu)], [ZA2219; H, H, Et, H, NMe (c-Pr)], [ZA2220; H, H, Et, H, NMe (c-Bu)], [ZA2221; H, H, Et, H, NMe (c-Pen) ], [ZA2222; H, H, Et, H, NMe (c-Hex)], [ZA2223; H, H, Et, H, NMeCH ₂ (c-Pr)], [ZA2224; H, H, Et, H, NMeCH ₂ (c-Bu)], [ZA2225; H, H, Et, H, NMeCH ₂ (c-Pen)], [ZA2226; H, H, Et, H, NMeCH ₂ (c-Hex)] , [ZA2227; H, H, Et, H, NMeCH ₂ F], [ZA2228; H, H, Et, H, NMeCHF ₂ ], [ZA2229; H, H, Et, H, NMeCF ₃ ], [ZA2230; H, H, Et, H, NMe (CH ₂ ) ₂ F], [Z A2231; H, H, Et, H, NMeCH ₂ CHF ₂ ], [ZA2232; H, H, Et, H, NMeCH ₂ CHF ₃ ], [ZA2233; H, H, Et, H, NMe (CH ₂ ) ₃ F], [ZA2234; H, H, Et, H, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA2235; H, H, Et, H, NMe (CH ₂ ) ₂ CF ₃ ], [ZA2236; H, H, Et, H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA2237; H, H, Et, H, NMeCH ₂ Cl], [ZA2238; H, H, Et, H, NMe (CH ₂ ) ₂ Cl ], [ZA2239; H, H, Et, H, NMe (CH ₂ ) ₃ Cl], [ZA2240; H, H, Et, H, NMe (CH ₂ ) ₄ Cl], [ZA2241; H, H, Et , H, NMe (CH ₂ ) ₅ Cl], [ZA2242; H, H, Et, H, NMeCH ₂ OMe], [ZA2243; H, H, Et, H, NMe (CH ₂ ) ₂ OMe], [ZA2244 ; H, H, Et, H, NMe (CH ₂ ) ₃ OMe], [ZA2245; H, H, Et, H, NMe (CH ₂ ) ₄ OMe], [ZA2246; H, H, Et, H, NM
eCH ₂ OEt], [ZA2247; H, H, Et, H, NMe (CH ₂ ) ₂ OEt], [ZA2248; H, H, Et, H, NMe (CH ₂ ) ₃ OEt], [ZA2249; H, H, Et, H, NMeCH ₂ OPr], [ZA2250; H, H, Et, H, NMe (CH ₂ ) ₂ OPr],

[ZA2251; H, H, Et, H, NMe (CH ₂ ) ₃ OPr], [ZA2252; H, H, Et, H, NMeCH ₂ CN], [ZA2253; H, H, Et, H, NMe (CH _{2) 2 CN], [ZA2254} ; H, H, Et, H, NMe (CH 2) 3 CN], [ZA2255; H, H, Et, H, NMe (CH 2) 4 CN], [ZA2256; H , H, Et, H, NMe (CH ₂ ) ₅ CN], [ZA2257; H, H, Et, H, NMeCH ₂ CH = CH ₂ ], [ZA2258; H, H, Et, H, NMeCH ₂ C≡ CH], [ZA2259; H, H, Et, H, NMeCH ₂ C≡CCH ₃ ], [ZA2260; H, H, Et, H, NMeCH ₂ Ph], [ZA2261; H, H, Et, H, NMeCH ₂ (2-Py)], [ZA2262; H, H, Et, H, NMeCH ₂ (3-Py)], [ZA2263; H, H, Et, H, NMeCH ₂ (4-Py)], [ZA2264 ; H, H, Et, H, NMe (CH ₂ ) ₂ Ph], [ZA2265; H, H, Et, H, NMe (CH ₂ ) ₂ (2-Py)], [ZA2266; H, H, Et , H, NMe (CH ₂ ) ₂ (3-Py)], [ZA2267; H, H, Et, H, NMe (CH ₂ ) ₂ (4-Py)], [ZA2268; H, H, Et, H , NMePh], [ZA2269; H, H, Et, H, NMe (2-Py)], [ZA2270; H, H, Et, H, NMe (3-Py)], [ZA2271; H, H, Et , H, NMe (4-Py)], [ZA2272; H, H, Et, H, NEt ₂ ], [ZA2273; H, H, Et, H, NEtPr], [ZA2274; H, H, Et, H , NEtBu], [ZA2275; H, H, Et, H, NEtPen], [ZA2276; H, H, Et, H, NEtHex], [ZA2277; H, H, Et, H, NEt (i-Pr)] , [ZA2278; H, H, Et, H, NEt (i-Bu)], [ZA2279; H, H, Et, H, NEt (c-Pr)], [ZA2280; H, H, Et, H, NEt (c-Bu)], [ZA2281; H, H, Et, H, NEt (c-Pen)], [ZA2282; H, H, Et, H, NEt (c-Hex)], [ZA2283; H , H, Et, H, N EtCH ₂ (c-Pr)], [ZA2284; H, H, Et, H, NEtCH ₂ (c-Bu)], [ZA2285; H, H, Et, H, NEtCH ₂ (c-Pen)], [ ZA2286; H, H, Et, H, NEtCH ₂ (c-Hex)], [ZA2287; H, H, Et, H, NEtCH ₂ F], [ZA2288; H, H, Et, H, NEtCHF ₂ ], [ZA2289; H, H, Et, H, NEtCF ₃ ], [ZA2290; H, H, Et, H, NEt (CH ₂ ) ₂ F], [ZA2291; H, H, Et, H, NEtCH ₂ CHF ₂ ], [ZA2292; H, H, Et, H, NEtCH ₂ CHF ₃ ], [ZA2293; H, H, Et, H, NEt (CH ₂ ) ₃ F], [ZA2294; H, H, Et, H, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA2295; H, H, Et, H, NEt (CH ₂ ) ₂ CF ₃ ], [ZA2296; H, H, Et, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA2297; H, H, Et, H, NEtCH ₂ Cl], [ZA2298; H, H, Et, H, NEt (CH ₂ ) ₂ Cl], [ZA2299; H, H, Et, H, NEt (CH ₂ ) ₃ Cl], [ZA2300; H, H, Et, H, NEt (CH ₂ ) ₄ Cl], [ZA2301; H, H, Et, H, NEt (CH ₂ ) ₅ Cl], [ZA2302 ; H, H, Et, H, NEtCH ₂ OMe], [ZA2303; H, H, Et, H, NEt (CH ₂ ) ₂ OMe], [ZA2304; H, H, Et, H, NEt (CH ₂ ) ₃ OMe], [ZA2305; H, H, Et, H, NEt (CH ₂ ) ₄ OMe], [ZA2306; H, H, Et, H, NEtCH ₂ OEt], [ZA2307; H, H, Et, H , NEt (CH ₂ ) ₂ OEt], [ZA2308; H, H, Et, H, NEt (CH ₂ ) ₃ OEt], [ZA2309; H, H, Et, H, NEtCH ₂ OPr], [ZA2310; H , H, Et, H, NEt (CH ₂ ) ₂ OPr], [ZA2311; H, H, Et, H, NEt (CH ₂ ) ₃ OPr], [ZA2312; H, H, Et, H, NEtCH ₂ CN ], [ZA2313; H, H, Et, H, NEt (CH ₂ ) ₂ CN], [ZA2314; H, H, Et, H, NEt (CH ₂ ) ₃ CN], [ZA2315; H, H, Et, H, NEt (CH ₂ ) ₄ CN], [ZA2316; H, H, Et, H, NEt (CH ₂ ) ₅ CN], [ZA2317; H, H, Et, H, NEtCH ₂ CH = CH ₂ ], [ZA2318; H, H, Et, H, NEtCH ₂ C≡CH ], [ZA2319; H, H, Et, H, NEtCH ₂ C≡CCH ₃ ], [ZA2320; H, H, Et, H, NEtCH ₂ Ph], [ZA2321; H, H, Et, H, NEtCH ₂ (2-Py)], [ZA2322; H, H, Et, H, NEtCH ₂ (3-Py)], [ZA2323; H, H, Et, H, NEtCH ₂ (4-Py)], [ZA2324; H, H, Et, H, NEt (CH ₂ ) ₂ Ph], [ZA2325; H, H, Et, H, NEt (CH ₂ ) ₂ (2-Py)], [ZA2326; H, H, Et, H, NEt (CH ₂ ) ₂ (3-Py)], [ZA2327; H, H, Et, H, NEt (CH ₂ ) ₂ (4-Py)], [ZA2328; H, H, Et, H, NEtPh], [ZA2329; H, H, Et, H, NEt (2-Py)], [ZA2330; H, H, Et, H, NEt (3-Py)], [ZA2331; H, H, Et, H, NEt (4-Py)], [ZA2332; H, H, Et, H, Pyr], [ZA2333; H, H, Et, H, Pip], [ZA2334; H, H, Et, H, Mor ], [ZA2335; H, H, Et, H, OMe], [ZA2336; H, H, Et, H, OEt], [ZA2337; H, H, Et, H, OPr], [ZA2338; H, H , Et, H, OBu], [ZA2339; H, H, Et, H, OPen], [ZA2340; H, H, Et, H, OHex], [ZA2341; H, H, Et, H, O (i -Pr)], [ZA2342; H, H, Et, H, O (i-Bu)], [ZA2343; H, H, Et, H, O (c-Pr)], [ZA2344; H, H, Et, H, O (c-Bu)], [ZA2345; H, H, Et, H, O (c-Pen)], [ZA2346; H, H, Et, H, O (c-Hex)], [ZA2347; H, H, Et, H, OCH ₂ (c-Pr)], [ZA2348; H, H, Et, H, OCH ₂ (c-Bu)], [ZA2349; H, H, Et, H, OCH ₂ (c-Pen)], [ZA2350; H, H, Et, H, OCH ₂ (c-Hex )], [ZA2351; H, H, Et, H, OCH ₂ F], [ZA2352; H, H, Et, H, OCHF ₂ ], [ZA2353; H, H, Et, H, OCF ₃ ], [ ZA2354; H, H, Et, H, O (CH ₂ ) ₂ F], [ZA2355; H, H, Et, H, OCH ₂ CHF ₂ ], [ZA2356; H, H, Et, H, OCH ₂ CHF ₃ ], [ZA2357; H, H, Et, H, O (CH ₂ ) ₃ F], [ZA2358; H, H, Et, H, O (CH ₂ ) ₂ CHF ₂ ], [ZA2359; H, H , Et, H, O (CH ₂ ) ₂ CF ₃ ], [ZA2360; H, H, Et, H, OCH ₂ CH (CF ₃ ) ₂ ], [ZA2361; H, H, Et, H, OCH ₂ Cl ], [ZA2362; H, H, Et, H, O (CH ₂ ) ₂ Cl], [ZA2363; H, H, Et, H, O (CH ₂ ) ₃ Cl], [ZA2364; H, H, Et , H, O (CH ₂ ) ₄ Cl], [ZA2365; H, H, Et, H, O (CH ₂ ) ₅ Cl], [ZA2366; H, H, Et, H, OCH ₂ OMe], [ZA2367 ; H, H, Et, H, O (CH ₂ ) ₂ OMe], [ZA2368; H, H, Et, H, O (CH ₂ ) ₃ OMe], [ZA2369; H, H, Et, H, O (CH ₂ ) ₄ OMe], [ZA2370; H, H, Et, H, OCH ₂ OEt], [ZA2371; H, H, Et, H, O (CH ₂ ) ₂ OEt], [ZA2372; H, H , Et, H, O (CH ₂ ) ₃ OEt], [ZA2373; H, H, Et, H, OCH ₂ OPr], [ZA2374; H, H, Et, H, O (CH ₂ ) ₂ OPr], [ZA2375; H, H, Et, H, O (CH ₂ ) ₃ OPr], [ZA2376; H, H, Et, H, OCH ₂ CN], [ZA2377; H, H, Et, H, O (CH _{2) 2 CN], [ZA2378} ; H, H, Et, H, O (CH 2) 3 CN], [ZA2379; H, H, Et, H, O (CH 2) 4 CN], [ZA2380; H , H, Et, H, O (CH ₂ ) ₅ CN], [ZA2381; H, H, Et, H, OCH ₂ CH = CH ₂ ], [ZA2382; H, H, Et, H, OCH ₂ C≡CH], [ZA2383 ; H, H, Et, H, OCH ₂ C≡CCH ₃ ], [ZA2384; H, H, Et, H, OCH ₂ Ph], [ZA2385; H, H, Et, H, OCH ₂ (2-Py )], [ZA2386; H, H, Et, H, OCH ₂ (3-Py)], [ZA2387; H, H, Et, H, OCH ₂ (4-Py)], [ZA2388; H, H, Et, H, O (CH ₂ ) ₂ Ph], [ZA2389; H, H, Et, H, O (CH ₂ ) ₂ (2-Py)], [ZA2390; H, H, Et, H, O ( CH ₂ ) ₂ (3-Py)], [ZA2391; H, H, Et, H, O (CH ₂ ) ₂ (4-Py)], [ZA2392; H, H, Et, H, OPh], [ ZA2393; H, H, Et, H, O (2-Py)], [ZA2394; H, H, Et, H, O (3-Py)], [ZA2395; H, H, Et, H, O ( 4-Py)], [ZA2396; H, H, Et, H, Me], [ZA2397; H, H, Et, H, Et], [ZA2398; H, H, Et, H, Pr], [ZA2399 ; H, H, Et, H, Bu], [ZA2400; H, H, Et, H, Pen], [ZA2401; H, H, Et, H, Hex], [ZA2402; H, H, Et, H , (i-Pr)], [ZA2403; H, H, Et, H, (i-Bu)], [ZA2404; H, H, Et, H, (c-Pr)], [ZA2405; H, H , Et, H, (c-Bu)], [ZA2406; H, H, Et, H, (c-Pen)], [ZA2407; H, H, Et, H, (c-Hex)], [ZA2408 ; H, H, Et, H, CH ₂ (c-Pr)], [ZA2409; H, H, Et, H, CH ₂ (c-Bu)], [ZA2410; H, H, Et, H, CH ₂ (c-Pen)], [ZA2411; H, H, Et, H, CH ₂ (c-Hex)], [ZA2412; H, H, Et, H, CH ₂ F], [ZA2413; H, H , Et, H, CHF ₂ ], [ZA2414; H, H, Et, H, CF ₃ ], [ZA2415; H, H, Et, H, (CH ₂ ) ₂ F], [ZA2416; H, H, Et, H, C H ₂ CHF ₂ ], [ZA2417; H, H, Et, H, CH ₂ CHF ₃ ], [ZA2418; H, H, Et, H, (CH ₂ ) ₃ F], [ZA2419; H, H, Et , H, (CH ₂ ) ₂ CHF ₂ ], [ZA2420; H, H, Et, H, (CH ₂ ) ₂ CF ₃ ], [ZA2421; H, H, Et, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA2422; H, H, Et, H, CH ₂ Cl], [ZA2423; H, H, Et, H, (CH ₂ ) ₂ Cl], [ZA2424; H, H, Et, H, ( CH ₂ ) ₃ Cl], [ZA2425; H, H, Et, H, (CH ₂ ) ₄ Cl], [ZA2426; H, H, Et, H, (CH ₂ ) ₅ Cl], [ZA2427; H, H, Et, H, CH ₂ OMe], [ZA2428; H, H, Et, H, (CH ₂ ) ₂ OMe], [ZA2429; H, H, Et, H, (CH ₂ ) ₃ OMe], [ ZA2430; H, H, Et, H, (CH ₂ ) ₄ OMe], [ZA2431; H, H, Et, H, CH ₂ OEt], [ZA2432; H, H, Et, H, (CH ₂ ) ₂ OEt], [ZA2433; H, H, Et, H, (CH ₂ ) ₃ OEt], [ZA2434; H, H, Et, H, CH ₂ OPr], [ZA2435; H, H, Et, H, ( CH ₂ ) ₂ OPr], [ZA2436; H, H, Et, H, (CH ₂ ) ₃ OPr], [ZA2437; H, H, Et, H, CH ₂ CN], [ZA2438; H, H, Et , H, (CH ₂ ) ₂ CN], [ZA2439; H, H, Et, H, (CH ₂ ) ₃ CN], [ZA2440; H, H, Et, H, (CH ₂ ) ₄ CN], [ ZA2441; H, H, Et, H, (CH ₂ ) ₅ CN], [ZA2442; H, H, Et, H, CH ₂ CH = CH ₂ ], [ZA2443; H, H, Et, H, CH ₂ C≡CH], [ZA2444; H, H, Et, H, CH ₂ C≡CCH ₃ ], [ZA2445; H, H, Et, H, CH ₂ Ph], [ZA2446; H, H, Et, H , CH ₂ (2-Py)], [ZA2447; H, H, Et, H, CH ₂ (3-Py)], [ZA2448; H, H, Et, H, CH ₂ (4-Py)], [ZA244 9; H, H, Et, H, (CH ₂ ) ₂ Ph], [ZA2450; H, H, Et, H, (CH ₂ ) ₂ (2-Py)], [ZA2451; H, H, Et, H, (CH ₂ ) ₂ (3-Py)], [ZA2452; H, H, Et, H, (CH ₂ ) ₂ (4-Py)], [ZA2453; H, H, Et, H, Ph] , [ZA2454; H, H, Et, H, 2-Py], [ZA2455; H, H, Et, H, 3-Py], [ZA2456; H, H, Et, H, 4-Py], [ ZA2457; H, H, Me, Et, NHMe], [ZA2458; H, H, Me, Et, NHEt], [ZA2459; H, H, Me, Et, NHPr], [ZA2460; H, H, Me, Et, NHBu], [ZA2461; H, H, Me, Et, NHPen], [ZA2462; H, H, Me, Et, NHHex], [ZA2463; H, H, Me, Et, NH (i-Pr) ], [ZA2464; H, H, Me, Et, NH (i-Bu)], [ZA2465; H, H, Me, Et, NH (c-Pr)], [ZA2466; H, H, Me, Et , NH (c-Bu)], [ZA2467; H, H, Me, Et, NH (c-Pen)], [ZA2468; H, H, Me, Et, NH (c-Hex)], [ZA2469; H, H, Me, Et, NHCH ₂ (c-Pr)], [ZA2470; H, H, Me, Et, NHCH ₂ (c-Bu)], [ZA2471; H, H, Me, Et, NHCH ₂ (c-Pen)], [ZA2472; H, H, Me, Et, NHCH ₂ (c-Hex)], [ZA2473; H, H, Me, Et, NHCH ₂ F], [ZA2474; H, H, Me, Et, NHCHF ₂ ], [ZA2475; H, H, Me, Et, NHCF ₃ ], [ZA2476; H, H, Me, Et, NH (CH ₂ ) ₂ F], [ZA2477; H, H, Me, Et, NHCH ₂ CHF ₂ ], [ZA2478; H, H, Me, Et, NHCH ₂ CHF ₃ ], [ZA2479; H, H, Me, Et, NH (CH ₂ ) ₃ F], [ZA2480; H, H, Me, Et, NH (CH ₂ ) ₂ CHF ₂ ], [ZA2481; H, H, Me, Et, NH (CH ₂ ) ₂ CF ₃ ], [ZA2482; H, H, Me, Et, NHCH ₂ CH (CF ₃ ) ₂ ], [ ZA2483; H, H, Me, Et, NHCH ₂ Cl], [ZA2484; H, H, Me, Et, NH (CH ₂ ) ₂ Cl], [ZA2485; H, H, Me, Et, NH (CH _{2 ) 3 Cl], [ZA2486;} H, H, Me, Et, NH (CH 2) 4 Cl], [ZA2487; H, H, Me, Et, NH (CH 2) 5 Cl], [ZA2488; H, H, Me, Et, NHCH ₂ OMe], [ZA2489; H, H, Me, Et, NH (CH ₂ ) ₂ OMe], [ZA2490; H, H, Me, Et, NH (CH ₂ ) ₃ OMe] , [ZA2491; H, H, Me, Et, NH (CH ₂ ) ₄ OMe], [ZA2492; H, H, Me, Et, NHCH ₂ OEt], [ZA2493; H, H, Me, Et, NH ( CH ₂ ) ₂ OEt], [ZA2494; H, H, Me, Et, NH (CH ₂ ) ₃ OEt], [ZA2495; H, H, Me, Et, NHCH ₂ OPr], [ZA2496; H, H, Me, Et, NH (CH ₂ ) ₂ OPr], [ZA2497; H, H, Me, Et, NH (CH ₂ )
₃ OPr], [ZA2498; H, H, Me, Et, NHCH ₂ CN], [ZA2499; H, H, Me, Et, NH (CH ₂ ) ₂ CN], [ZA2500; H, H, Me, Et , NH (CH ₂ ) ₃ CN],

[ZA2501; H, H, Me, Et, NH (CH ₂ ) ₄ CN], [ZA2502; H, H, Me, Et, NH (CH ₂ ) ₅ CN], [ZA2503; H, H, Me, Et , NHCH ₂ CH = CH ₂ ], [ZA2504; H, H, Me, Et, NHCH ₂ C≡CH], [ZA2505; H, H, Me, Et, NHCH ₂ C≡CCH ₃ ], [ZA2506; H , H, Me, Et, NHCH ₂ Ph], [ZA2507; H, H, Me, Et, NHCH ₂ (2-Py)], [ZA2508; H, H, Me, Et, NHCH ₂ (3-Py) ], [ZA2509; H, H, Me, Et, NHCH ₂ (4-Py)], [ZA2510; H, H, Me, Et, NH (CH ₂ ) ₂ Ph], [ZA2511; H, H, Me , Et, NH (CH ₂ ) ₂ (2-Py)], [ZA2512; H, H, Me, Et, NH (CH ₂ ) ₂ (3-Py)], [ZA2513; H, H, Me, Et , NH (CH ₂ ) ₂ (4-Py)], [ZA2514; H, H, Me, Et, NHPh], [ZA2515; H, H, Me, Et, NH (2-Py)], [ZA2516; H, H, Me, Et, NH (3-Py)], [ZA2517; H, H, Me, Et, NH (4-Py)], [ZA2518; H, H, Me, Et, NMe ₂ ], [ZA2519; H, H, Me, Et, NMeEt], [ZA2520; H, H, Me, Et, NMePr], [ZA2521; H, H, Me, Et, NMeBu], [ZA2522; H, H, Me , Et, NMePen], [ZA2523; H, H, Me, Et, NMeHex], [ZA2524; H, H, Me, Et, NMe (i-Pr)], [ZA2525; H, H, Me, Et, NMe (i-Bu)], [ZA2526; H, H, Me, Et, NMe (c-Pr)], [ZA2527; H, H, Me, Et, NMe (c-Bu)], [ZA2528; H , H, Me, Et, NMe (c-Pen)], [ZA2529; H, H, Me, Et, NMe (c-Hex)], [ZA2530; H, H, Me, Et, NMeCH ₂ (c- Pr)], [ZA2531; H, H, Me, Et, NMeCH ₂ (c-Bu)], [ZA2532; H, H, Me, Et, NMeCH ₂ (c-Pen)], [ZA2533; H, H , Me, Et, NMeCH ₂ (c-Hex)], [ZA2534; H, H, Me, Et, NMeCH ₂ F], [ZA2535; H, H, Me, Et, NMeCHF ₂ ], [ZA2536; H, H, Me, Et, NMeCF ₃ ], [ZA2537; H, H, Me, Et, NMe (CH ₂ ) ₂ F], [ZA2538; H, H, Me, Et, NMeCH ₂ CHF ₂ ], [ZA2539; H, H, Me, Et, NMeCH ₂ CHF ₃ ], [ZA2540; H, H, Me, Et, NMe (CH ₂ ) ₃ F], [ZA2541; H, H, Me, Et, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA2542; H, H, Me, Et, NMe (CH ₂ ) ₂ CF ₃ ], [ZA2543; H, H, Me, Et, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA2544; H, H, Me, Et, NMeCH ₂ Cl], [ZA2545; H, H, Me, Et, NMe (CH ₂ ) ₂ Cl], [ZA2546; H, H, Me, Et, NMe (CH ₂ ) ₃ Cl], [ZA2547; H, H, Me, Et, NMe (CH ₂ ) ₄ Cl], [ZA2548; H, H, Me, Et, NMe (CH ₂ ) ₅ Cl], [ZA2549; H, H, Me, Et, NMeCH ₂ OMe], [ZA2550; H, H, Me, Et, NMe (CH ₂ ) ₂ OMe], [ZA2551; H, H, Me, Et, NMe (CH ₂ ) ₃ OMe], [ ZA2552; H, H, Me, Et, NMe (CH ₂ ) ₄ OMe], [ZA2553; H, H, Me, Et, NMeCH ₂ OEt], [ZA2554; H, H, Me, Et, NMe (CH ₂ ) ₂ OEt], [ZA2555; H, H, Me, Et, NMe (CH ₂ ) ₃ OEt], [ZA2556; H, H, Me, Et, NMeCH ₂ OPr], [ZA2557; H, H, Me, Et, NMe (CH ₂ ) ₂ OPr], [ZA2558; H, H, Me, Et, NMe (CH ₂ ) ₃ OPr], [ZA2559; H, H, Me, Et, NMeCH ₂ CN], [ZA2560; H, H, Me, Et, NMe (CH ₂ ) ₂ CN], [ZA2561; H, H, Me, Et, NMe (CH ₂ ) ₃ CN], [ZA2562; H, H, Me, Et, NMe ( CH ₂ ) ₄ CN], [ZA2563; H, H, Me, Et, NMe (CH ₂ ) ₅ CN], [ZA2564; H, H, Me, Et, NMeCH ₂ CH = CH ₂ ], [ZA2565; H , H, Me, Et, NMeCH ₂ C≡CH], [ZA2566; H, H, Me, Et, NMeCH ₂ C≡CCH ₃ ], [ZA2567; H, H, Me, Et, NMeCH ₂ Ph], [ ZA2568; H, H, Me, Et, NMeCH ₂ (2-Py)], [ZA2569; H, H, Me, Et, NMeCH ₂ (3-Py)], [ZA2570; H, H, Me, Et, NMeCH ₂ (4-Py)], [ZA2571; H, H, Me, Et, NMe (CH ₂ ) ₂ Ph], [ZA2572; H, H, Me, Et, NMe (CH ₂ ) ₂ (2-Py )], [ZA2573; H, H, Me, Et, NMe (CH ₂ ) ₂ (3-Py)], [ZA2574; H, H, Me, Et, NMe (CH ₂ ) ₂ (4-Py)] , [ZA2575; H, H, Me, Et, NMePh], [ZA2576; H, H, Me, Et, NMe (2-Py)], [ZA2577; H, H, Me, Et, NMe (3-Py )], [ZA2578; H, H, Me, Et, NMe (4-Py)], [ZA2579; H, H, Me, Et, NEt ₂ ], [ZA2580; H, H, Me, Et, NEtPr] , [ZA2581; H, H, Me, Et, NEtBu], [ZA2582; H, H, Me, Et, NEtPen], [ZA2583; H, H, Me, Et, NEtHex], [ZA2584; H, H, Me, Et, NEt (i-Pr)], [ZA2585; H, H, Me, Et, NEt (i-Bu)], [ZA2586; H, H, Me, Et, NEt (c-Pr)], [ZA2587; H, H, Me, Et, NEt (c-Bu)], [ZA2588; H, H, Me, Et, NEt (c-Pen)], [ZA2589; H, H, Me, Et, NEt (c-Hex)], [ZA2590; H, H, Me, Et, NEtCH ₂ (c-Pr)], [ZA2591; H, H, Me, Et, NEtCH ₂ (c-Bu)], [ZA2592; H, H, Me, Et, NEtCH ₂ (c-Pen)], [ZA2593; H, H, Me, Et, NEtCH ₂ (c-Hex)], [ZA259 4; H, H, Me, Et, NEtCH ₂ F], [ZA2595; H, H, Me, Et, NEtCHF ₂ ], [ZA2596; H, H, Me, Et, NEtCF ₃ ], [ZA2597; H, H, Me, Et, NEt (CH ₂ ) ₂ F], [ZA2598; H, H, Me, Et, NEtCH ₂ CHF ₂ ], [ZA2599; H, H, Me, Et, NEtCH ₂ CHF ₃ ], [ ZA2600; H, H, Me, Et, NEt (CH ₂ ) ₃ F], [ZA2601; H, H, Me, Et, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA2602; H, H, Me, Et , NEt (CH ₂ ) ₂ CF ₃ ], [ZA2603; H, H, Me, Et, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA2604; H, H, Me, Et, NEtCH ₂ Cl], [ZA2605 ; H, H, Me, Et, NEt (CH ₂ ) ₂ Cl], [ZA2606; H, H, Me, Et, NEt (CH ₂ ) ₃ Cl], [ZA2607; H, H, Me, Et, NEt (CH ₂ ) ₄ Cl], [ZA2608; H, H, Me, Et, NEt (CH ₂ ) ₅ Cl], [ZA2609; H, H, Me, Et, NEtCH ₂ OMe], [ZA2610; H, H , Me, Et, NEt (CH ₂ ) ₂ OMe], [ZA2611; H, H, Me, Et, NEt (CH ₂ ) ₃ OMe], [ZA2612; H, H, Me, Et, NEt (CH ₂ ) ₄ OMe], [ZA2613; H, H, Me, Et, NEtCH ₂ OEt], [ZA2614; H, H, Me, Et, NEt (CH ₂ ) ₂ OEt], [ZA2615; H, H, Me, Et , NEt (CH ₂ ) ₃ OEt], [ZA2616; H, H, Me, Et, NEtCH ₂ OPr], [ZA2617; H, H, Me, Et, NEt (CH ₂ ) ₂ OPr], [ZA2618; H , H, Me, Et, NEt (CH ₂ ) ₃ OPr], [ZA2619; H, H, Me, Et, NEtCH ₂ CN], [ZA2620; H, H, Me, Et, NEt (CH ₂ ) ₂ CN ], [ZA2621; H, H, Me, Et, NEt (CH ₂ ) ₃ CN], [ZA2622; H, H, Me, Et, NEt (CH ₂ ) ₄ CN], [ZA2623; H, H, Me , Et , NEt (CH ₂ ) ₅ CN], [ZA2624; H, H, Me, Et, NEtCH ₂ CH = CH ₂ ], [ZA2625; H, H, Me, Et, NEtCH ₂ C≡CH], [ZA2626; H, H, Me, Et, NEtCH ₂ C≡CCH ₃ ], [ZA2627; H, H, Me, Et, NEtCH ₂ Ph], [ZA2628; H, H, Me, Et, NEtCH ₂ (2-Py) ], [ZA2629; H, H, Me, Et, NEtCH ₂ (3-Py)], [ZA2630; H, H, Me, Et, NEtCH ₂ (4-Py)], [ZA2631; H, H, Me , Et, NEt (CH ₂ ) ₂ Ph], [ZA2632; H, H, Me, Et, NEt (CH ₂ ) ₂ (2-Py)], [ZA2633; H, H, Me, Et, NEt (CH ₂ ) ₂ (3-Py)], [ZA2634; H, H, Me, Et, NEt (CH ₂ ) ₂ (4-Py)], [ZA2635; H, H, Me, Et, NEtPh], [ZA2636 ; H, H, Me, Et, NEt (2-Py)], [ZA2637; H, H, Me, Et, NEt (3-Py)], [ZA2638; H, H, Me, Et, NEt (4 -Py)], [ZA2639; H, H, Me, Et, Pyr], [ZA2640; H, H, Me, Et, Pip], [ZA2641; H, H, Me, Et, Mor], [ZA2642; H, H, Me, Et, OMe], [ZA2643; H, H, Me, Et, OEt], [ZA2644; H, H, Me, Et, OPr], [ZA2645; H, H, Me, Et, OBu], [ZA2646; H, H, Me, Et, OPen], [ZA2647; H, H, Me, Et, OHex], [ZA2648; H, H, Me, Et, O (i-Pr)], [ZA2649; H, H, Me, Et, O (i-Bu)], [ZA2650; H, H, Me, Et, O (c-Pr)], [ZA2651; H, H, Me, Et, O (c-Bu)], [ZA2652; H, H, Me, Et, O (c-Pen)], [ZA2653; H, H, Me, Et, O (c-Hex)], [ZA2654; H, H, Me, Et, OCH ₂ (c-Pr)], [ZA2655; H, H, Me, Et, OCH ₂ (c-Bu)], [ZA2656; H, H, Me, Et, OCH ₂ (c -Pen)], [ZA2657; H, H, Me, Et, OCH ₂ (c-Hex)], [ZA2658; H, H, Me, Et, OCH ₂ F], [ZA2659; H, H, Me, Et, OCHF ₂ ], [ZA2660 ; H, H, Me, Et, OCF ₃ ], [ZA2661; H, H, Me, Et, O (CH ₂ ) ₂ F], [ZA2662; H, H, Me, Et, OCH ₂ CHF ₂ ], [ZA2663; H, H, Me, Et, OCH ₂ CHF ₃ ], [ZA2664; H, H, Me, Et, O (CH ₂ ) ₃ F], [ZA2665; H, H, Me, Et, O ( CH ₂ ) ₂ CHF ₂ ], [ZA2666; H, H, Me, Et, O (CH ₂ ) ₂ CF ₃ ], [ZA2667; H, H, Me, Et, OCH ₂ CH (CF ₃ ) ₂ ], [ZA2668; H, H, Me, Et, OCH ₂ Cl], [ZA2669; H, H, Me, Et, O (CH ₂ ) ₂ Cl], [ZA2670; H, H, Me, Et, O (CH _{2) 3 Cl], [ZA2671} ; H, H, Me, Et, O (CH 2) 4 Cl], [ZA2672; H, H, Me, Et, O (CH 2) 5 Cl], [ZA2673; H , H, Me, Et, OCH ₂ OMe], [ZA2674; H, H, Me, Et, O (CH ₂ ) ₂ OMe], [ZA2675; H, H, Me, Et, O (CH ₂ ) ₃ OMe ], [ZA2676; H, H, Me, Et, O (CH ₂ ) ₄ OMe], [ZA2677; H, H, Me, Et, OCH ₂ OEt], [ZA2678; H, H, Me, Et, O (CH ₂ ) ₂ OEt], [ZA2679; H, H, Me, Et, O (CH ₂ ) ₃ OEt], [ZA2680; H, H, Me, Et, OCH ₂ OPr], [ZA2681; H, H , Me, Et, O (CH ₂ ) ₂ OPr], [ZA2682; H, H, Me, Et, O (CH ₂ ) ₃ OPr], [ZA2683; H, H, Me, Et, OCH ₂ CN], [ZA2684; H, H, Me, Et, O (CH ₂ ) ₂ CN], [ZA2685; H, H, Me, Et, O (CH ₂ ) ₃ CN], [ZA2686; H, H, Me, Et , O (CH ₂ ) ₄ CN], [ZA2687; H, H, Me, Et, O (CH ₂ ) ₅ CN], [ZA2688; H, H , Me, Et, OCH ₂ CH = CH ₂ ], [ZA2689; H, H, Me, Et, OCH ₂ C≡CH], [ZA2690; H, H, Me, Et, OCH ₂ C≡CCH ₃ ], [ZA2691; H, H, Me, Et, OCH ₂ Ph], [ZA2692; H, H, Me, Et, OCH ₂ (2-Py)], [ZA2693; H, H, Me, Et, OCH ₂ ( 3-Py)], [ZA2694; H, H, Me, Et, OCH ₂ (4-Py)], [ZA2695; H, H, Me, Et, O (CH ₂ ) ₂ Ph], [ZA2696; H , H, Me, Et, O (CH ₂ ) ₂ (2-Py)], [ZA2697; H, H, Me, Et, O (CH ₂ ) ₂ (3-Py)], [ZA2698; H, H , Me, Et, O (CH ₂ ) ₂ (4-Py)], [ZA2699; H, H, Me, Et, OPh], [ZA2700; H, H, Me, Et, O (2-Py)] , [ZA2701; H, H, Me, Et, O (3-Py)], [ZA2702; H, H, Me, Et, O (4-Py)], [ZA2703; H, H, Me, Et, Me], [ZA2704; H, H, Me, Et, Et], [ZA2705; H, H, Me, Et, Pr], [ZA2706; H, H, Me, Et, Bu], [ZA2707; H, H, Me, Et, Pen], [ZA2708; H, H, Me, Et, Hex], [ZA2709; H, H, Me, Et, (i-Pr)], [ZA2710; H, H, Me, Et, (i-Bu)], [ZA2711; H, H, Me, Et, (c-Pr)], [ZA2712; H, H, Me, Et, (c-Bu)], [ZA2713; H, H, Me, Et, (c-Pen)], [ZA2714; H, H, Me, Et, (c-Hex)], [ZA2715; H, H, Me, Et, CH ₂ (c-Pr)] , [ZA2716; H, H, Me, Et, CH ₂ (c-Bu)], [ZA2717; H, H, Me, Et, CH ₂ (c-Pen)], [ZA2718; H, H, Me, Et, CH ₂ (c-Hex)], [ZA2719; H, H, Me, Et, CH ₂ F], [ZA2720; H, H, Me, Et, CHF ₂ ], [ZA2721; H, H, Me , Et, CF ₃ ], [ZA2722; H, H, Me, Et, (CH ₂ ) ₂ F], [ZA2723; H, H , Me, Et, CH ₂ CHF ₂ ], [ZA2724; H, H, Me, Et, CH ₂ CHF ₃ ], [ZA2725; H, H, Me, Et, (CH ₂ ) ₃ F], [ZA2726; H, H, Me, Et, (CH ₂ ) ₂ CHF ₂ ], [ZA2727; H, H, Me, Et, (CH ₂ ) ₂ CF ₃ ], [ZA2728; H, H, Me, Et, CH ₂ CH (CF ₃ ) ₂ ], [ZA2729; H, H, Me, Et, CH ₂ Cl], [ZA2730; H, H, Me, Et, (CH ₂ ) ₂ Cl], [ZA2731; H, H, Me, Et, (CH ₂ ) ₃ Cl], [ZA2732; H, H, Me, Et, (CH ₂ ) ₄ Cl], [ZA2733; H, H, Me, Et, (CH ₂ ) ₅ Cl], [ZA2734; H, H, Me, Et, CH ₂ OMe], [ZA2735; H, H, Me, Et, (CH ₂ ) ₂ OMe], [ZA2736; H, H, Me, Et, (CH ₂ ) ₃ OMe], [ZA2737; H, H, Me, Et, (CH ₂ ) ₄ OMe], [ZA2738; H, H, Me, Et, CH ₂ OEt], [ZA2739; H, H, Me, Et, (CH ₂ ) ₂ OEt], [ZA2740; H, H, Me, Et, (CH ₂ ) ₃ OEt], [ZA2741; H, H, Me, Et,
CH ₂ OPr], [ZA2742; H, H, Me, Et, (CH ₂ ) ₂ OPr], [ZA2743; H, H, Me, Et, (CH ₂ ) ₃ OPr], [ZA2744; H, H, Me, Et, CH ₂ CN], [ZA2745; H, H, Me, Et, (CH ₂ ) ₂ CN], [ZA 2746; H, H, Me, Et, (CH ₂ ) ₃ CN], [ZA2747; H, H, Me, Et, (CH ₂ ) ₄ CN], [ZA2748; H, H, Me, Et, (CH ₂ ) ₅ CN], [ZA2749; H, H, Me, Et, CH ₂ CH = CH ₂ ], [ZA2750; H, H, Me, Et, CH ₂ C≡CH],

[ZA2751; H, H, Me, Et, CH ₂ C≡CCH ₃ ], [ZA2752; H, H, Me, Et, CH ₂ Ph], [ZA2753; H, H, Me, Et, CH ₂ (2 -Py)], [ZA2754; H, H, Me, Et, CH ₂ (3-Py)], [ZA2755; H, H, Me, Et, CH ₂ (4-Py)], [ZA2756; H, H, Me, Et, (CH ₂ ) ₂ Ph], [ZA2757; H, H, Me, Et, (CH ₂ ) ₂ (2-Py)], [ZA2758; H, H, Me, Et, (CH ₂ ) ₂ (3-Py)], [ZA2759; H, H, Me, Et, (CH ₂ ) ₂ (4-Py)], [ZA2760; H, H, Me, Et, Ph], [ZA2761; H, H, Me, Et, 2-Py], [ZA2762; H, H, Me, Et, 3-Py], [ZA2763; H, H, Me, Et, 4-Py], [ZA2764; F, H, H, H, NHMe], [ZA2765; F, H, H, H, NHEt], [ZA2766; F, H, H, H, NHPr], [ZA2767; F, H, H, H, NHBu] , [ZA2768; F, H, H, H, NHPen], [ZA2769; F, H, H, H, NHHex], [ZA2770; F, H, H, H, NH (i-Pr)], [ZA2771 ; F, H, H, H, NH (i-Bu)], [ZA2772; F, H, H, H, NH (c-Pr)], [ZA2773; F, H, H, H, NH (c -Bu)], [ZA2774; F, H, H, H, NH (c-Pen)], [ZA2775; F, H, H, H, NH (c-Hex)], [ZA2776; F, H, H, H, NHCH ₂ (c-Pr)], [ZA2777; F, H, H, H, NHCH ₂ (c-Bu)], [ZA2778; F, H, H, H, NHCH ₂ (c-Pen )], [ZA2779; F, H, H, H, NHCH ₂ (c-Hex)], [ZA2780; F, H, H, H, NHCH ₂ F], [ZA2781; F, H, H, H, NHCHF ₂ ], [ZA2782; F, H, H, H, NHCF ₃ ], [ZA2783; F, H, H, H, NH (CH ₂ ) ₂ F], [ZA2784; F, H, H, H, NHCH ₂ CHF ₂ ], [ZA2785; F, H, H, H, NHCH ₂ CHF ₃ ], [ZA2786; F, H, H, H, NH (CH ₂ ) ₃ F], [ZA2787; F, H, H, H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA2788; F, H, H, H, NH (CH ₂ ) ₂ CF ₃ ], [ZA2789; F, H, H, H, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA2790; F, H, H, H, NHCH ₂ Cl], [ZA2791; F, H, H, H, NH (CH ₂ ) ₂ Cl], [ZA2792; F, H, H, H, NH (CH ₂ ) ₃ Cl], [ZA2793; F, H, H, H, NH (CH ₂ ) ₄ Cl], [ZA2794; F, H , H, H, NH (CH ₂ ) ₅ Cl], [ZA2795; F, H, H, H, NHCH ₂ OMe], [ZA2796; F, H, H, H, NH (CH ₂ ) ₂ OMe], [ZA2797; F, H, H, H, NH (CH ₂ ) ₃ OMe], [ZA2798; F, H, H, H, NH (CH ₂ ) ₄ OMe], [ZA2799; F, H, H, H , NHCH ₂ OEt], [ZA2800; F, H, H, H, NH (CH ₂ ) ₂ OEt], [ZA2801; F, H, H, H, NH (CH ₂ ) ₃ OEt], [ZA2802; F , H, H, H, NHCH ₂ OPr], [ZA2803; F, H, H, H, NH (CH ₂ ) ₂ OPr], [ZA2804; F, H, H, H, NH (CH ₂ ) ₃ OPr ], [ZA2805; F, H, H, H, NHCH ₂ CN], [ZA2806; F, H, H, H, NH (CH ₂ ) ₂ CN], [ZA2807; F, H, H, H, NH (CH ₂ ) ₃ CN], [ZA2808; F, H, H, H, NH (CH ₂ ) ₄ CN], [ZA2809; F, H, H, H, NH (CH ₂ ) ₅ CN], [ZA2810 ; F, H, H, H, NHCH ₂ CH = CH ₂ ], [ZA2811; F, H, H, H, NHCH ₂ C≡CH], [ZA2812; F, H, H, H, NHCH ₂ C≡ CCH ₃ ], [ZA2813; F, H, H, H, NHCH ₂ Ph], [ZA2814; F, H, H, H, NHCH ₂ (2-Py)], [ZA2815; F, H, H, H , NHCH ₂ (3-Py)], [ZA2816; F, H, H, H, NHCH ₂ (4-Py)], [ZA2817; F, H, H, H, NH (CH ₂ ) ₂ Ph], [ZA2818; F, H, H, H, NH (CH ₂ ) ₂ (2-Py)], [ZA2819; F, H, H, H, NH (CH ₂ ) ₂ (3-Py)], [ZA2820; F, H, H, H, NH (CH ₂ ) ₂ (4-Py)], [ZA2821; F, H, H, H, NHPh], [ZA2822; F, H, H, H, NH (2-Py) ], [ZA2823; F, H, H, H, NH (3-Py)], [ZA2824; F, H, H, H, NH (4-Py)], [ZA2825; F, H, H, H , NMe ₂ ], [ZA2826; F, H, H, H, NMeEt], [ZA2827; F, H, H, H, NMePr], [ZA2828; F, H, H, H, NMeBu], [ZA2829; F, H, H, H, NMePen], [ZA2830; F, H, H, H, NMeHex], [ZA2831; F, H, H, H, NMe (i-Pr)], [ZA2832; F, H , H, H, NMe (i-Bu)], [ZA2833; F, H, H, H, NMe (c-Pr)], [ZA2834; F, H, H, H, NMe (c-Bu)] , [ZA2835; F, H, H, H, NMe (c-Pen)], [ZA2836; F, H, H, H, NMe (c-Hex)], [ZA2837; F, H, H, H, NMeCH ₂ (c-Pr)], [ZA2838; F, H, H, H, NMeCH ₂ (c-Bu)], [ZA2839; F, H, H, H, NMeCH ₂ (c-Pen)], [ ZA2840; F, H, H, H, NMeCH ₂ (c-Hex)], [ZA2841; F, H, H, H, NMeCH ₂ F], [ZA2842; F, H, H, H, NMeCHF ₂ ], [ZA2843; F, H, H, H, NMeCF ₃ ], [ZA2844; F, H, H, H, NMe (CH ₂ ) ₂ F], [ZA2845; F, H, H, H, NMeCH ₂ CHF ₂ ], [ZA2846; F, H, H, H, NMeCH ₂ CHF ₃ ], [ZA2847; F, H, H, H, NMe (CH ₂ ) ₃ F], [ZA2848; F, H, H, H, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA2849; F, H, H, H, NMe (CH ₂ ) ₂ CF ₃ ], [ZA2850; F, H, H, H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA2851; F, H, H, H, NMeCH ₂ Cl], [ZA2852; F, H, H, H, NM e (CH ₂ ) ₂ Cl], [ZA2853; F, H, H, H, NMe (CH ₂ ) ₃ Cl], [ZA2854; F, H, H, H, NMe (CH ₂ ) ₄ Cl], [ ZA2855; F, H, H, H, NMe (CH ₂ ) ₅ Cl], [ZA2856; F, H, H, H, NMeCH ₂ OMe], [ZA2857; F, H, H, H, NMe (CH ₂ ) ₂ OMe], [ZA2858; F, H, H, H, NMe (CH ₂ ) ₃ OMe], [ZA2859; F, H, H, H, NMe (CH ₂ ) ₄ OMe], [ZA2860; F, H, H, H, NMeCH ₂ OEt], [ZA2861; F, H, H, H, NMe (CH ₂ ) ₂ OEt], [ZA2862; F, H, H, H, NMe (CH ₂ ) ₃ OEt] , [ZA2863; F, H, H, H, NMeCH ₂ OPr], [ZA2864; F, H, H, H, NMe (CH ₂ ) ₂ OPr], [ZA2865; F, H, H, H, NMe ( _{CH 2) 3 OPr], [} ZA2866; F, H, H, H, NMeCH 2 CN], [ZA2867; F, H, H, H, NMe (CH 2) 2 CN], [ZA2868; F, H, H, H, NMe (CH ₂ ) ₃ CN], [ZA2869; F, H, H, H, NMe (CH ₂ ) ₄ CN], [ZA2870; F, H, H, H, NMe (CH ₂ ) ₅ CN], [ZA2871; F, H, H, H, NMeCH ₂ CH = CH ₂ ], [ZA2872; F, H, H, H, NMeCH ₂ C≡CH], [ZA2873; F, H, H, H , NMeCH ₂ C≡CCH ₃ ], [ZA2874; F, H, H, H, NMeCH ₂ Ph], [ZA2875; F, H, H, H, NMeCH ₂ (2-Py)], [ZA2876; F, H, H, H, NMeCH ₂ (3-Py)], [ZA2877; F, H, H, H, NMeCH ₂ (4-Py)], [ZA2878; F, H, H, H, NMe (CH ₂ ) ₂ Ph], [ZA2879; F, H, H, H, NMe (CH ₂ ) ₂ (2-Py)], [ZA2880; F, H, H, H, NMe (CH ₂ ) ₂ (3-Py )], [ZA2881; F, H, H, H, NMe (CH ₂ ) ₂ (4-Py)], [ZA2882; F, H, H, H, NMePh], [ZA2883; F, H, H, H, NMe (2-Py)], [ZA2884; F, H, H, H, NMe (3-Py)], [ZA2885; F, H, H, H, NMe (4- Py)], [ZA2886; F, H, H, H, NEt ₂ ], [ZA2887; F, H, H, H, NEtPr], [ZA2888; F, H, H, H, NEtBu], [ZA2889; F, H, H, H, NEtPen], [ZA2890; F, H, H, H, NEtHex], [ZA2891; F, H, H, H, NEt (i-Pr)], [ZA2892; F, H , H, H, NEt (i-Bu)], [ZA2893; F, H, H, H, NEt (c-Pr)], [ZA2894; F, H, H, H, NEt (c-Bu)] , [ZA2895; F, H, H, H, NEt (c-Pen)], [ZA2896; F, H, H, H, NEt (c-Hex)], [ZA2897; F, H, H, H, NEtCH ₂ (c-Pr)], [ZA2898; F, H, H, H, NEtCH ₂ (c-Bu)], [ZA2899; F, H, H, H, NEtCH ₂ (c-Pen)], [ ZA2900; F, H, H, H, NEtCH ₂ (c-Hex)], [ZA2901; F, H, H, H, NEtCH ₂ F], [ZA2902; F, H, H, H, NEtCHF ₂ ], [ZA2903; F, H, H, H, NEtCF ₃ ], [ZA2904; F, H, H, H, NEt (CH ₂ ) ₂ F], [ZA2905; F, H, H, H, NEtCH ₂ CHF ₂ ], [ZA2906; F, H, H, H, NEtCH ₂ CHF ₃ ], [ZA2907; F, H, H, H, NEt (CH ₂ ) ₃ F], [ZA2908; F, H, H, H, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA2909; F, H, H, H, NEt (CH ₂ ) ₂ CF ₃ ], [ZA2910; F, H, H, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA2911; F, H, H, H, NEtCH ₂ Cl], [ZA2912; F, H, H, H, NEt (CH ₂ ) ₂ Cl], [ZA2913; F, H, H, H, NEt (CH ₂ ) ₃ Cl], [ZA2914; F, H, H, H, NEt (CH ₂ ) ₄ Cl], [ZA2915; F, H, H, H, NEt (CH ₂ ) ₅ Cl], [ZA2916 ; F, H, H, H, NEtCH ₂ OMe], [ZA2917 ; F, H, H, H, NEt (CH ₂ ) ₂ OMe], [ZA2918; F, H, H, H, NEt (CH ₂ ) ₃ OMe], [ZA2919; F, H, H, H, NEt (CH ₂ ) ₄ OMe], [ZA2920; F, H, H, H, NEtCH ₂ OEt], [ZA2921; F, H, H, H, NEt (CH ₂ ) ₂ OEt], [ZA2922; F, H , H, H, NEt (CH ₂ ) ₃ OEt], [ZA2923; F, H, H, H, NEtCH ₂ OPr], [ZA2924; F, H, H, H, NEt (CH ₂ ) ₂ OPr], [ZA2925; F, H, H, H, NEt (CH ₂ ) ₃ OPr], [ZA2926; F, H, H, H, NEtCH ₂ CN], [ZA2927; F, H, H, H, NEt (CH _{2) 2 CN], [ZA2928} ; F, H, H, H, NEt (CH 2) 3 CN], [ZA2929; F, H, H, H, NEt (CH 2) 4 CN], [ZA2930; F , H, H, H, NEt (CH ₂ ) ₅ CN], [ZA2931; F, H, H, H, NEtCH ₂ CH = CH ₂ ], [ZA2932; F, H, H, H, NEtCH ₂ C≡ CH], [ZA2933; F, H, H, H, NEtCH ₂ C≡CCH ₃ ], [ZA2934; F, H, H, H, NEtCH ₂ Ph], [ZA2935; F, H, H, H, NEtCH ₂ (2-Py)], [ZA2936; F, H, H, H, NEtCH ₂ (3-Py)], [ZA2937; F, H, H, H, NEtCH ₂ (4-Py)], [ZA2938 ; F, H, H, H, NEt (CH ₂ ) ₂ Ph], [ZA2939; F, H, H, H, NEt (CH ₂ ) ₂ (2-Py)], [ZA2940; F, H, H , H, NEt (CH ₂ ) ₂ (3-Py)], [ZA2941; F, H, H, H, NEt (CH ₂ ) ₂ (4-Py)], [ZA2942; F, H, H, H , NEtPh], [ZA2943; F, H, H, H, NEt (2-Py)], [ZA2944; F, H, H, H, NEt (3-Py)], [ZA2945; F, H, H , H, NEt (4-Py)], [ZA2946; F, H, H, H, Pyr], [ZA2947; F, H, H, H, Pip], [ZA2948; F, H, H, H, Mor], [ZA2949; F, H, H, H, OMe], [ZA2950; F, H, H, H, OEt], [ZA2951; F, H, H, H, OPr], [ZA2952; F, H, H, H, OBu], [ZA2953; F, H, H, H, OPen], [ZA2954; F, H, H, H, OHex], [ZA2955; F, H, H, H, O (i-Pr)], [ZA2956; F, H , H, H, O (i-Bu)], [ZA2957; F, H, H, H, O (c-Pr)], [ZA2958; F, H, H, H, O (c-Bu)] , [ZA2959; F, H, H, H, O (c-Pen)], [ZA2960; F, H, H, H, O (c-Hex)], [ZA2961; F, H, H, H, OCH ₂ (c-Pr)], [ZA2962; F, H, H, H, OCH ₂ (c-Bu)], [ZA2963; F, H, H, H, OCH ₂ (c-Pen)], [ ZA2964; F, H, H, H, OCH ₂ (c-Hex)], [ZA2965; F, H, H, H, OCH ₂ F], [ZA2966; F, H, H, H, OCHF ₂ ], [ZA2967; F, H, H, H, OCF ₃ ], [ZA2968; F, H, H, H, O (CH ₂ ) ₂ F], [ZA2969; F, H, H, H, OCH ₂ CHF ₂ ], [ZA2970; F, H, H, H, OCH ₂ CHF ₃ ], [ZA2971; F, H, H, H, O (CH ₂ ) ₃ F], [ZA2972; F, H, H, H, O (CH ₂ ) ₂ CHF ₂ ], [ZA2973; F, H, H, H, O (CH ₂ ) ₂ CF ₃ ], [ZA2974; F, H, H, H, OCH ₂ CH (CF ₃ ) ₂ ], [ZA2975; F, H, H, H, OCH ₂ Cl], [ZA2976; F, H, H, H, O (CH ₂ ) ₂ Cl], [ZA2977; F, H, H, H, O (CH ₂ ) ₃ Cl], [ZA2978; F, H, H, H, O (CH ₂ ) ₄ Cl], [ZA2979; F, H, H, H, O (CH ₂ ) ₅ Cl], [ZA2980 ; F, H, H, H, OCH ₂ OMe], [ZA2981; F, H, H, H, O (CH ₂ ) ₂ OMe], [ZA2982; F, H, H, H, O (CH ₂ ) ₃ OMe], [ZA2983; F, H, H, H, O (CH ₂ ) ₄ OMe], [ZA2984; F, H, H, H, OCH ₂ OEt], [ZA2985; F, H, H , H, O (CH ₂ ) ₂ OEt], [ZA2986; F, H, H, H, O (CH ₂ ) ₃ OEt], [ZA2987; F, H, H, H, OCH ₂ OPr], [ZA2988 ; F, H, H, H, O (CH ₂ ) ₂ OPr], [ZA2989; F, H, H, H, O (CH ₂ ) ₃ OPr], [ZA2990; F, H, H, H, OCH ₂ CN], [ZA2991; F, H, H, H, O (CH ₂ ) ₂ CN], [ZA2992; F, H, H, H, O (CH ₂ ) ₃ CN], [ZA2993; F, H , H, H, O (CH ₂ ) ₄ CN], [ZA2994; F, H, H, H, O (CH ₂ ) ₅ CN], [ZA2995; F, H, H, H, OCH ₂ CH = CH ₂ ], [ZA2996; F, H, H, H, OCH ₂ C≡CH], [ZA2997; F, H, H, H, OCH ₂ C≡CCH ₃ ], [ZA2998; F, H, H, H , OCH ₂ Ph], [ZA2999; F, H, H, H, OCH ₂ (2-Py)], [ZA3000; F, H, H, H
, OCH ₂ (3-Py)],

[ZA3001; F, H, H, H, OCH ₂ (4-Py)], [ZA3002; F, H, H, H, O (CH ₂ ) ₂ Ph], [ZA3003; F, H, H, H , O (CH ₂ ) ₂ (2-Py)], [ZA3004; F, H, H, H, O (CH ₂ ) ₂ (3-Py)], [ZA3005; F, H, H, H, O (CH ₂ ) ₂ (4-Py)], [ZA3006; F, H, H, H, OPh], [ZA3007; F, H, H, H, O (2-Py)], [ZA3008; F, H, H, H, O (3-Py)], [ZA3009; F, H, H, H, O (4-Py)], [ZA3010; F, H, H, H, Me], [ZA3011; F, H, H, H, Et], [ZA3012; F, H, H, H, Pr], [ZA3013; F, H, H, H, Bu], [ZA3014; F, H, H, H, Pen], [ZA3015; F, H, H, H, Hex], [ZA3016; F, H, H, H, (i-Pr)], [ZA3017; F, H, H, H, (i-Bu )], [ZA3018; F, H, H, H, (c-Pr)], [ZA3019; F, H, H, H, (c-Bu)], [ZA3020; F, H, H, H, (c-Pen)], [ZA3021; F, H, H, H, (c-Hex)], [ZA3022; F, H, H, H, CH ₂ (c-Pr)], [ZA3023; F, H, H, H, CH ₂ (c-Bu)], [ZA3024; F, H, H, H, CH ₂ (c-Pen)], [ZA3025; F, H, H, H, CH ₂ (c -Hex)], [ZA3026; F, H, H, H, CH ₂ F], [ZA3027; F, H, H, H, CHF ₂ ], [ZA3028; F, H, H, H, CF ₃ ] , [ZA3029; F, H, H, H, (CH ₂ ) ₂ F], [ZA3030; F, H, H, H, CH ₂ CHF ₂ ], [ZA3031; F, H, H, H, CH ₂ CHF ₃ ], [ZA3032; F, H, H, H, (CH ₂ ) ₃ F], [ZA3033; F, H, H, H, (CH ₂ ) ₂ CHF ₂ ], [ZA3034; F, H, H, H, (CH ₂ ) ₂ CF ₃ ], [ZA3035; F, H, H, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA3036; F, H, H, H, CH ₂ Cl], [ZA3037; F, H, H, H, (CH ₂ ) ₂ Cl], [ZA3038; F, H, H, H, (CH ₂ ) ₃ Cl], [ZA3039; F, H, H, H, (CH ₂ ) ₄ Cl], [ZA3040; F, H, H, H, (CH ₂ ) ₅ Cl], [ZA3041; F, H, H, H, CH ₂ OMe], [ZA3042; F, H, H, H, (CH ₂ ) ₂ OMe], [ZA3043; F, H, H, H, (CH ₂ ) ₃ OMe], [ZA3044; F, H, H, H, (CH ₂ ) ₄ OMe], [ZA3045; F, H, H, H, CH ₂ OEt], [ZA3046; F, H, H, H, (CH ₂ ) ₂ OEt], [ZA3047; F, H, H, H, (CH ₂ ) ₃ OEt], [ZA3048; F, H, H, H, CH ₂ OPr], [ZA3049; F, H, H, H, (CH ₂ ) ₂ OPr], [ZA3050; F, H, H, H, (CH ₂ ) ₃ OPr], [ZA3051; F, H, H, H, CH ₂ CN] , [ZA3052; F, H, H, H, (CH ₂ ) ₂ CN], [ZA3053; F, H, H, H, (CH ₂ ) ₃ CN], [ZA3054; F, H, H, H, (CH ₂ ) ₄ CN], [ZA3055; F, H, H, H, (CH ₂ ) ₅ CN], [ZA3056; F, H, H, H, CH ₂ CH = CH ₂ ], [ZA3057; F , H, H, H, CH ₂ C≡CH], [ZA3058; F, H, H, H, CH ₂ C≡CCH ₃ ], [ZA3059; F, H, H, H, CH ₂ Ph], [ ZA3060; F, H, H, H, CH ₂ (2-Py)], [ZA3061; F, H, H, H, CH ₂ (3-Py)], [ZA3062; F, H, H, H, CH ₂ (4-Py)], [ZA3063; F, H, H, H, (CH ₂ ) ₂ Ph], [ZA3064; F, H, H, H, (CH ₂ ) ₂ (2-Py)] , [ZA3065; F, H, H, H, (CH ₂ ) ₂ (3-Py)], [ZA3066; F, H, H, H, (CH ₂ ) ₂ (4-Py)], [ZA3067; F, H, H, H, Ph], [ZA3068; F, H, H, H, 2-Py], [ZA3069; F, H, H, H, 3-Py], [ZA3070; F, H, H, H, 4-Py], [ZA3071; F, H, Me, H, NHMe], [ZA3072; F, H, Me, H, NHEt], [ZA3073; F , H, Me, H, NHPr], [ZA3074; F, H, Me, H, NHBu], [ZA3075; F, H, Me, H, NHPen], [ZA3076; F, H, Me, H, NHHex ], [ZA3077; F, H, Me, H, NH (i-Pr)], [ZA3078; F, H, Me, H, NH (i-Bu)], [ZA3079; F, H, Me, H , NH (c-Pr)], [ZA3080; F, H, Me, H, NH (c-Bu)], [ZA3081; F, H, Me, H, NH (c-Pen)], [ZA3082; F, H, Me, H, NH (c-Hex)], [ZA3083; F, H, Me, H, NHCH ₂ (c-Pr)], [ZA3084; F, H, Me, H, NHCH ₂ ( c-Bu)], [ZA3085; F, H, Me, H, NHCH ₂ (c-Pen)], [ZA3086; F, H, Me, H, NHCH ₂ (c-Hex)], [ZA3087; F , H, Me, H, NHCH ₂ F], [ZA3088; F, H, Me, H, NHCHF ₂ ], [ZA3089; F, H, Me, H, NHCF ₃ ], [ZA3090; F, H, Me , H, NH (CH ₂ ) ₂ F], [ZA3091; F, H, Me, H, NHCH ₂ CHF ₂ ], [ZA3092; F, H, Me, H, NHCH ₂ CHF ₃ ], [ZA3093; F , H, Me, H, NH (CH ₂ ) ₃ F], [ZA3094; F, H, Me, H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA3095; F, H, Me, H, NH ( CH ₂ ) ₂ CF ₃ ], [ZA3096; F, H, Me, H, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA3097; F, H, Me, H, NHCH ₂ Cl], [ZA3098; F, H, Me, H, NH (CH ₂ ) ₂ Cl], [ZA3099; F, H, Me, H, NH (CH ₂ ) ₃ Cl], [ZA3100; F, H, Me, H, NH (CH ₂ ) ₄ Cl], [ZA3101; F, H, Me, H, NH (CH ₂ ) ₅ Cl], [ZA3102; F, H, Me, H, NHCH ₂ OMe], [ZA3103; F, H, Me, H, NH (CH ₂ ) ₂ OMe], [ZA3104; F, H, Me, H, NH (CH ₂ ) ₃ OMe], [ZA3105; F, H, Me, H, NH (CH ₂ ) ₄ OMe] , [ZA3106; F, H , Me, H, NHCH ₂ OEt], [ZA3107; F, H, Me, H, NH (CH ₂ ) ₂ OEt], [ZA3108; F, H, Me, H, NH (CH ₂ ) ₃ OEt], [ZA3109; F, H, Me, H, NHCH ₂ OPr], [ZA3110; F, H, Me, H, NH (CH ₂ ) ₂ OPr], [ZA3111; F, H, Me, H, NH (CH ₂ ) ₃ OPr], [ZA3112; F, H, Me, H, NHCH ₂ CN], [ZA3113; F, H, Me, H, NH (CH ₂ ) ₂ CN], [ZA3114; F, H, Me , H, NH (CH ₂ ) ₃ CN], [ZA3115; F, H, Me, H, NH (CH ₂ ) ₄ CN], [ZA3116; F, H, Me, H, NH (CH ₂ ) ₅ CN ], [ZA3117; F, H, Me, H, NHCH ₂ CH = CH ₂ ], [ZA3118; F, H, Me, H, NHCH ₂ C≡CH], [ZA3119; F, H, Me, H, NHCH ₂ C≡CCH ₃ ], [ZA3120; F, H, Me, H, NHCH ₂ Ph], [ZA3121; F, H, Me, H, NHCH ₂ (2-Py)], [ZA3122; F, H , Me, H, NHCH ₂ (3-Py)], [ZA3123; F, H, Me, H, NHCH ₂ (4-Py)], [ZA3124; F, H, Me, H, NH (CH ₂ ) ₂ Ph], [ZA3125; F, H, Me, H, NH (CH ₂ ) ₂ (2-Py)], [ZA3126; F, H, Me, H, NH (CH ₂ ) ₂ (3-Py) ], [ZA3127; F, H, Me, H, NH (CH ₂ ) ₂ (4-Py)], [ZA3128; F, H, Me, H, NHPh], [ZA3129; F, H, Me, H , NH (2-Py)], [ZA3130; F, H, Me, H, NH (3-Py)], [ZA3131; F, H, Me, H, NH (4-Py)], [ZA3132; F, H, Me, H, NMe ₂ ], [ZA3133; F, H, Me, H, NMeEt], [ZA3134; F, H, Me, H, NMePr], [ZA3135; F, H, Me, H , NMeBu], [ZA3136; F, H, Me, H, NMePen], [ZA3137; F, H, Me, H, NMeHex], [ZA3138; F, H, Me, H, NMe (i-Pr)] , [ZA3139; F, H, Me, H, NMe (i-Bu)], [ZA3140; F, H, Me, H, NMe (c-Pr)], [ZA3141; F, H, Me, H, NMe (c- Bu)], [ZA3142; F, H, Me, H, NMe (c-Pen)], [ZA3143; F, H, Me, H, NMe (c-Hex)], [ZA3144; F, H, Me , H, NMeCH ₂ (c-Pr)], [ZA3145; F, H, Me, H, NMeCH ₂ (c-Bu)], [ZA3146; F, H, Me, H, NMeCH ₂ (c-Pen) ], [ZA3147; F, H, Me, H, NMeCH ₂ (c-Hex)], [ZA3148; F, H, Me, H, NMeCH ₂ F], [ZA3149; F, H, Me, H, NMeCHF ₂ ], [ZA3150; F, H, Me, H, NMeCF ₃ ], [ZA3151; F, H, Me, H, NMe (CH ₂ ) ₂ F], [ZA3152; F, H, Me, H, NMeCH ₂ CHF ₂ ], [ZA3153; F, H, Me, H, NMeCH ₂ CHF ₃ ], [ZA3154; F, H, Me, H, NMe (CH ₂ ) ₃ F], [ZA3155; F, H, Me , H, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA3156; F, H, Me, H, NMe (CH ₂ ) ₂ CF ₃ ], [ZA3157; F, H, Me, H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA3158; F, H, Me, H, NMeCH ₂ Cl], [ZA3159; F, H, Me, H, NMe (CH ₂ ) ₂ Cl], [ZA3160; F, H, Me, H, NMe (CH ₂ ) ₃ Cl], [ZA3161; F, H, Me, H, NMe (CH ₂ ) ₄ Cl], [ZA3162; F, H, Me, H, NMe (CH ₂ ) ₅ Cl] , [ZA3163; F, H, Me, H, NMeCH ₂ OMe], [ZA3164; F, H, Me, H, NMe (CH ₂ ) ₂ OMe], [ZA3165; F, H, Me, H, NMe ( CH ₂ ) ₃ OMe], [ZA3166; F, H, Me, H, NMe (CH ₂ ) ₄ OMe], [ZA3167; F, H, Me, H, NMeCH ₂ OEt], [ZA3168; F, H, Me, H, NMe (CH ₂ ) ₂ OEt], [ZA3169; F, H, Me, H, NMe (CH ₂ ) ₃ OEt], [ZA 3170; F, H, Me, H, NMeCH ₂ OPr], [ZA3171; F, H, Me, H, NMe (CH ₂ ) ₂ OPr], [ZA3172; F, H, Me, H, NMe (CH ₂ ) ₃ OPr], [ZA3173; F, H, Me, H, NMeCH ₂ CN], [ZA3174; F, H, Me, H, NMe (CH ₂ ) ₂ CN], [ZA3175; F, H, Me, H, NMe (CH ₂ ) ₃ CN], [ZA3176; F, H, Me, H, NMe (CH ₂ ) ₄ CN], [ZA3177; F, H, Me, H, NMe (CH ₂ ) ₅ CN] , [ZA3178; F, H, Me, H, NMeCH ₂ CH = CH ₂ ], [ZA3179; F, H, Me, H, NMeCH ₂ C≡CH], [ZA3180; F, H, Me, H, NMeCH ₂ C≡CCH ₃ ], [ZA3181; F, H, Me, H, NMeCH ₂ Ph], [ZA3182; F, H, Me, H, NMeCH ₂ (2-Py)], [ZA3183; F, H, Me, H, NMeCH ₂ (3-Py)], [ZA3184; F, H, Me, H, NMeCH ₂ (4-Py)], [ZA3185; F, H, Me, H, NMe (CH ₂ ) ₂ Ph], [ZA3186; F, H, Me, H, NMe (CH ₂ ) ₂ (2-Py)], [ZA3187; F, H, Me, H, NMe (CH ₂ ) ₂ (3-Py)] , [ZA3188; F, H, Me, H, NMe (CH ₂ ) ₂ (4-Py)], [ZA3189; F, H, Me, H, NMePh], [ZA3190; F, H, Me, H, NMe (2-Py)], [ZA3191; F, H, Me, H, NMe (3-Py)], [ZA3192; F, H, Me, H, NMe (4-Py)], [ZA3193; F , H, Me, H, NEt ₂ ], [ZA3194; F, H, Me, H, NEtPr], [ZA3195; F, H, Me, H, NEtBu], [ZA3196; F, H, Me, H, NEtPen], [ZA3197; F, H, Me, H, NEtHex], [ZA3198; F, H, Me, H, NEt (i-Pr)], [ZA3199; F, H, Me, H, NEt (i -Bu)], [ZA3200; F, H, Me, H, NEt (c-Pr)], [ZA3201; F, H, Me, H, NEt (c-Bu)], [ZA3202; F, H, Me , H, NEt (c-Pen)], [ZA3203; F, H, Me, H, NEt (c-Hex)], [ZA3204; F, H, Me, H, NEtCH ₂ (c-Pr)], [ZA3205; F, H, Me, H, NEtCH ₂ (c-Bu)], [ZA3206; F, H, Me, H, NEtCH ₂ (c-Pen)], [ZA3207; F, H, Me, H , NEtCH ₂ (c-Hex)], [ZA3208; F, H, Me, H, NEtCH ₂ F], [ZA3209; F, H, Me, H, NEtCHF ₂ ], [ZA3210; F, H, Me, H, NEtCF ₃ ], [ZA3211; F, H, Me, H, NEt (CH ₂ ) ₂ F], [ZA3212; F, H, Me, H, NEtCH ₂ CHF ₂ ], [ZA3213; F, H, Me, H, NEtCH ₂ CHF ₃ ], [ZA3214; F, H, Me, H, NEt (CH ₂ ) ₃ F], [ZA3215; F, H, Me, H, NEt (CH ₂ ) ₂ CHF ₂ ] , [ZA3216; F, H, Me, H, NEt (CH ₂ ) ₂ CF ₃ ], [ZA3217; F, H, Me, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA3218; F, H, Me, H, NEtCH ₂ Cl], [ZA3219; F, H, Me, H, NEt (CH ₂ ) ₂ Cl], [ZA3220; F, H, Me, H, NEt (CH ₂ ) ₃ Cl], [ ZA3221; F, H, Me, H, NEt (CH ₂ ) ₄ Cl], [ZA3222; F, H, Me, H, NEt (CH ₂ ) ₅ Cl], [ZA3223; F, H, Me, H, NEtCH ₂ OMe], [ZA3224; F, H, Me, H, NEt (CH ₂ ) ₂ OMe], [ZA3225; F, H, Me, H, NEt (CH ₂ ) ₃ OMe], [ZA3226; F, H, Me, H, NEt (CH ₂ ) ₄ OMe], [ZA3227; F, H, Me, H, NEtCH ₂ OEt], [ZA3228; F, H, Me, H, NEt (CH ₂ ) ₂ OEt] , [ZA3229; F, H, Me, H, NEt (CH ₂ ) ₃ OEt], [ZA3230; F, H, Me, H, NEtCH ₂ OPr], [ZA3231; F, H, Me, H, NEt ( CH ₂ ) ₂ OPr], [ZA3232; F, H, Me, H, NEt (CH ₂ ) ₃ OPr], [ZA3233; F, H, Me, H, NEtCH ₂ CN], [ZA3234; F, H, Me, H, NEt (CH ₂ ) ₂ CN], [ZA3235; F, H, Me, H , NEt (CH ₂ ) ₃ CN], [ZA3236; F, H, Me, H, NEt (CH ₂ ) ₄ CN], [ZA3237; F, H, Me, H, NEt (CH ₂ ) ₅ CN], [ZA3238; F, H, Me, H, NEtCH ₂ CH = CH ₂ ], [ZA3239; F, H, Me, H, NEtCH ₂ C≡CH], [ZA3240; F, H, Me, H, NEtCH ₂ C≡CCH ₃ ], [ZA3241; F, H, Me, H, NEtCH ₂ Ph], [ZA3242; F, H, Me, H, NEtCH ₂ (2-Py)], [ZA3243; F, H, Me , H, NEtCH ₂ (3-Py)], [ZA3244; F, H, Me, H, NEtCH ₂ (4-Py)], [ZA3245; F, H, Me, H, NEt (CH ₂ ) ₂ Ph ], [ZA3246; F, H, Me, H, NEt (CH
₂ ) ₂ (2-Py)], [ZA3247; F, H, Me, H, NEt (CH ₂ ) ₂ (3-Py)], [ZA3248; F, H, Me, H, NEt (CH ₂ ) ₂ (4-Py)], [ZA3249; F, H, Me, H, NEtPh], [ZA3250; F, H, Me, H, NEt (2-Py)],

[ZA3251; F, H, Me, H, NEt (3-Py)], [ZA3252; F, H, Me, H, NEt (4-Py)], [ZA3253; F, H, Me, H, Pyr ], [ZA3254; F, H, Me, H, Pip], [ZA3255; F, H, Me, H, Mor], [ZA3256; F, H, Me, H, OMe], [ZA3257; F, H , Me, H, OEt], [ZA3258; F, H, Me, H, OPr], [ZA3259; F, H, Me, H, OBu], [ZA3260; F, H, Me, H, OPen], [ZA3261; F, H, Me, H, OHex], [ZA3262; F, H, Me, H, O (i-Pr)], [ZA3263; F, H, Me, H, O (i-Bu) ], [ZA3264; F, H, Me, H, O (c-Pr)], [ZA3265; F, H, Me, H, O (c-Bu)], [ZA3266; F, H, Me, H , O (c-Pen)], [ZA3267; F, H, Me, H, O (c-Hex)], [ZA3268; F, H, Me, H, OCH ₂ (c-Pr)], [ZA3269 ; F, H, Me, H, OCH ₂ (c-Bu)], [ZA3270; F, H, Me, H, OCH ₂ (c-Pen)], [ZA3271; F, H, Me, H, OCH ₂ (c-Hex)], [ZA3272; F, H, Me, H, OCH ₂ F], [ZA3273; F, H, Me, H, OCHF ₂ ], [ZA3274; F, H, Me, H, OCF ₃ ], [ZA3275; F, H, Me, H, O (CH ₂ ) ₂ F], [ZA3276; F, H, Me, H, OCH ₂ CHF ₂ ], [ZA3277; F, H, Me, H, OCH ₂ CHF ₃ ], [ZA3278; F, H, Me, H, O (CH ₂ ) ₃ F], [ZA3279; F, H, Me, H, O (CH ₂ ) ₂ CHF ₂ ], [ ZA3280; F, H, Me, H, O (CH ₂ ) ₂ CF ₃ ], [ZA3281; F, H, Me, H, OCH ₂ CH (CF ₃ ) ₂ ], [ZA3282; F, H, Me, H, OCH ₂ Cl], [ZA3283; F, H, Me, H, O (CH ₂ ) ₂ Cl], [ZA3284; F, H, Me, H, O (CH ₂ ) ₃ Cl], [ZA3285; F, H, Me, H, O (CH ₂ ) ₄ Cl], [ZA3286; F, H, Me, H, O (CH ₂ ) ₅ Cl], [ZA3287; F, H, Me, H, OCH ₂ OMe], [ZA3288; F, H, Me, H, O (CH ₂ ) ₂ OMe], [ZA3289; F, H, Me, H, O (CH ₂ ) ₃ OMe], [ZA3290; F, H, Me, H, O (CH ₂ ) ₄ OMe], [ZA3291; F, H, Me, H, OCH ₂ OEt], [ZA3292; F, H, Me, H, O (CH ₂ ) ₂ OEt], [ZA3293; F, H, Me, H, O (CH ₂ ) ₃ OEt], [ZA3294; F, H, Me, H, OCH ₂ OPr] , [ZA3295; F, H, Me, H, O (CH ₂ ) ₂ OPr], [ZA3296; F, H, Me, H, O (CH ₂ ) ₃ OPr], [ZA3297; F, H, Me, H, OCH ₂ CN], [ZA3298; F, H, Me, H, O (CH ₂ ) ₂ CN], [ZA3299; F, H, Me, H, O (CH ₂ ) ₃ CN], [ZA3300; F, H, Me, H, O (CH ₂ ) ₄ CN], [ZA3301; F, H, Me, H, O (CH ₂ ) ₅ CN], [ZA3302; F, H, Me, H, OCH ₂ CH = CH ₂ ], [ZA3303; F, H, Me, H, OCH ₂ C≡CH], [ZA3304; F, H, Me, H, OCH ₂ C≡CCH ₃ ], [ZA3305; F, H, Me, H, OCH ₂ Ph], [ZA3306; F, H, Me, H, OCH ₂ (2-Py)], [ZA3307; F, H, Me, H, OCH ₂ (3-Py)], [ ZA3308; F, H, Me, H, OCH ₂ (4-Py)], [ZA3309; F, H, Me, H, O (CH ₂ ) ₂ Ph], [ZA3310; F, H, Me, H, O (CH ₂ ) ₂ (2-Py)], [ZA3311; F, H, Me, H, O (CH ₂ ) ₂ (3-Py)], [ZA3312; F, H, Me, H, O ( CH ₂ ) ₂ (4-Py)], [ZA3313; F, H, Me, H, OPh], [ZA3314; F, H, Me, H, O (2-Py)], [ZA3315; F, H , Me, H, O (3-Py)], [ZA3316; F, H, Me, H, O (4-Py)], [ZA3317; F, H, Me, H, Me], [ZA3318; F , H, Me, H, Et], [ZA3319; F, H, Me, H, Pr], [ZA3 320; F, H, Me, H, Bu], [ZA3321; F, H, Me, H, Pen], [ZA3322; F, H, Me, H, Hex], [ZA3323; F, H, Me, H, (i-Pr)], [ZA3324; F, H, Me, H, (i-Bu)], [ZA3325; F, H, Me, H, (c-Pr)], [ZA3326; F, H, Me, H, (c-Bu)], [ZA3327; F, H, Me, H, (c-Pen)], [ZA3328; F, H, Me, H, (c-Hex)], [ ZA3329; F, H, Me, H, CH ₂ (c-Pr)], [ZA3330; F, H, Me, H, CH ₂ (c-Bu)], [ZA3331; F, H, Me, H, CH ₂ (c-Pen)], [ZA3332; F, H, Me, H, CH ₂ (c-Hex)], [ZA3333; F, H, Me, H, CH ₂ F], [ZA3334; F, H, Me, H, CHF ₂ ], [ZA3335; F, H, Me, H, CF ₃ ], [ZA3336; F, H, Me, H, (CH ₂ ) ₂ F], [ZA3337; F, H , Me, H, CH ₂ CHF ₂ ], [ZA3338; F, H, Me, H, CH ₂ CHF ₃ ], [ZA3339; F, H, Me, H, (CH ₂ ) ₃ F], [ZA3340; F, H, Me, H, (CH ₂ ) ₂ CHF ₂ ], [ZA3341; F, H, Me, H, (CH ₂ ) ₂ CF ₃ ], [ZA3342; F, H, Me, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA3343; F, H, Me, H, CH ₂ Cl], [ZA3344; F, H, Me, H, (CH ₂ ) ₂ Cl], [ZA3345; F, H, Me, H, (CH ₂ ) ₃ Cl], [ZA3346; F, H, Me, H, (CH ₂ ) ₄ Cl], [ZA3347; F, H, Me, H, (CH ₂ ) ₅ Cl], [ZA3348; F, H, Me, H, CH ₂ OMe], [ZA3349; F, H, Me, H, (CH ₂ ) ₂ OMe], [ZA3350; F, H, Me, H, (CH ₂ ) ₃ OMe], [ZA3351; F, H, Me, H, (CH ₂ ) ₄ OMe], [ZA3352; F, H, Me, H, CH ₂ OEt], [ZA3353; F, H, Me, H, (CH ₂ ) ₂ OEt], [ZA3354; F, H, Me, H, (CH ₂ ) ₃ OEt], [Z A3355; F, H, Me, H, CH ₂ OPr], [ZA3356; F, H, Me, H, (CH ₂ ) ₂ OPr], [ZA3357; F, H, Me, H, (CH ₂ ) ₃ OPr], [ZA3358; F, H, Me, H, CH ₂ CN], [ZA3359; F, H, Me, H, (CH ₂ ) ₂ CN], [ZA3360; F, H, Me, H, ( _{CH 2) 3 CN], [} ZA3361; F, H, Me, H, (CH 2) 4 CN], [ZA3362; F, H, Me, H, (CH 2) 5 CN], [ZA3363; F, H, Me, H, CH ₂ CH = CH ₂ ], [ZA3364; F, H, Me, H, CH ₂ C≡CH], [ZA3365; F, H, Me, H, CH ₂ C≡CCH ₃ ] , [ZA3366; F, H, Me, H, CH ₂ Ph], [ZA3367; F, H, Me, H, CH ₂ (2-Py)], [ZA3368; F, H, Me, H, CH ₂ (3-Py)], [ZA3369; F, H, Me, H, CH ₂ (4-Py)], [ZA3370; F, H, Me, H, (CH ₂ ) ₂ Ph], [ZA3371; F , H, Me, H, (CH ₂ ) ₂ (2-Py)], [ZA3372; F, H, Me, H, (CH ₂ ) ₂ (3-Py)], [ZA3373; F, H, Me , H, (CH ₂ ) ₂ (4-Py)], [ZA3374; F, H, Me, H, Ph], [ZA3375; F, H, Me, H, 2-Py], [ZA3376; F, H, Me, H, 3-Py], [ZA3377; F, H, Me, H, 4-Py], [ZA3378; F, H, Me, Me, NHMe], [ZA3379; F, H, Me, Me, NHEt], [ZA3380; F, H, Me, Me, NHPr], [ZA3381; F, H, Me, Me, NHBu], [ZA3382; F, H, Me, Me, NHPen], [ZA3383; F, H, Me, Me, NHHex], [ZA3384; F, H, Me, Me, NH (i-Pr)], [ZA3385; F, H, Me, Me, NH (i-Bu)], [ ZA3386; F, H, Me, Me, NH (c-Pr)], [ZA3387; F, H, Me, Me, NH (c-Bu)], [ZA3388; F, H, Me, Me, NH ( c-Pen)], [ZA3389; F, H, Me, Me, NH (c-Hex)], [ZA3390 ; F, H, Me, Me, NHCH ₂ (c-Pr)], [ZA3391; F, H, Me, Me, NHCH ₂ (c-Bu)], [ZA3392; F, H, Me, Me, NHCH ₂ (c-Pen)], [ZA3393; F, H, Me, Me, NHCH ₂ (c-Hex)], [ZA3394; F, H, Me, Me, NHCH ₂ F], [ZA3395; F, H , Me, Me, NHCHF ₂ ], [ZA3396; F, H, Me, Me, NHCF ₃ ], [ZA3397; F, H, Me, Me, NH (CH ₂ ) ₂ F], [ZA3398; F, H , Me, Me, NHCH ₂ CHF ₂ ], [ZA3399; F, H, Me, Me, NHCH ₂ CHF ₃ ], [ZA3400; F, H, Me, Me, NH (CH ₂ ) ₃ F], [ZA3401 ; F, H, Me, Me, NH (CH ₂ ) ₂ CHF ₂ ], [ZA3402; F, H, Me, Me, NH (CH ₂ ) ₂ CF ₃ ], [ZA3403; F, H, Me, Me , NHCH ₂ CH (CF ₃ ) ₂ ], [ZA3404; F, H, Me, Me, NHCH ₂ Cl], [ZA3405; F, H, Me, Me, NH (CH ₂ ) ₂ Cl], [ZA3406; F, H, Me, Me, NH (CH ₂ ) ₃ Cl], [ZA3407; F, H, Me, Me, NH (CH ₂ ) ₄ Cl], [ZA3408; F, H, Me, Me, NH ( CH ₂ ) ₅ Cl], [ZA3409; F, H, Me, Me, NHCH ₂ OMe], [ZA3410; F, H, Me, Me, NH (CH ₂ ) ₂ OMe], [ZA3411; F, H, Me, Me, NH (CH ₂ ) ₃ OMe], [ZA3412; F, H, Me, Me, NH (CH ₂ ) ₄ OMe], [ZA3413; F, H, Me, Me, NHCH ₂ OEt], [ ZA3414; F, H, Me, Me, NH (CH ₂ ) ₂ OEt], [ZA3415; F, H, Me, Me, NH (CH ₂ ) ₃ OEt], [ZA3416; F, H, Me, Me, NHCH ₂ OPr], [ZA3417; F, H, Me, Me, NH (CH ₂ ) ₂ OPr], [ZA3418; F, H, Me, Me, NH (CH ₂ ) ₃ OPr], [ZA3419; F, H, Me, Me, NHCH ₂ CN], [ZA3420; F, H, Me, Me, NH (CH ₂ ) ₂ CN], [ZA3421; F, H, Me, Me, NH (CH ₂ ) ₃ CN], [ZA3422; F, H, Me, Me, NH (CH ₂ ) ₄ CN] , [ZA3423; F, H, Me, Me, NH (CH ₂ ) ₅ CN], [ZA3424; F, H, Me, Me, NHCH ₂ CH = CH ₂ ], [ZA3425; F, H, Me, Me , NHCH ₂ C≡CH], [ZA3426; F, H, Me, Me, NHCH ₂ C≡CCH ₃ ], [ZA3427; F, H, Me, Me, NHCH ₂ Ph], [ZA3428; F, H, Me, Me, NHCH ₂ (2-Py)], [ZA3429; F, H, Me, Me, NHCH ₂ (3-Py)], [ZA3430; F, H, Me, Me, NHCH ₂ (4-Py )], [ZA3431; F, H, Me, Me, NH (CH ₂ ) ₂ Ph], [ZA3432; F, H, Me, Me, NH (CH ₂ ) ₂ (2-Py)], [ZA3433; F, H, Me, Me, NH (CH ₂ ) ₂ (3-Py)], [ZA3434; F, H, Me, Me, NH (CH ₂ ) ₂ (4-Py)], [ZA3435; F, H, Me, Me, NHPh], [ZA3436; F, H, Me, Me, NH (2-Py)], [ZA3437; F, H, Me, Me, NH (3-Py)], [ZA3438; F, H, Me, Me, NH (4-Py)], [ZA3439; F, H, Me, Me, NMe ₂ ], [ZA3440; F, H, Me, Me, NMeEt], [ZA3441; F, H, Me, Me, NMePr], [ZA3442; F, H, Me, Me, NMeBu], [ZA3443; F, H, Me, Me, NMePen], [ZA3444; F, H, Me, Me, NMeHex] , [ZA3445; F, H, Me, Me, NMe (i-Pr)], [ZA3446; F, H, Me, Me, NMe (i-Bu)], [ZA3447; F, H, Me, Me, NMe (c-Pr)], [ZA3448; F, H, Me, Me, NMe (c-Bu)], [ZA3449; F, H, Me, Me, NMe (c-Pen)], [ZA3450; F , H, Me, Me, NMe (c-Hex)], [ZA3451; F, H, Me, Me, NMeCH ₂ (c-Pr)], [ZA3452; F, H, Me, Me, NMeCH ₂ ( c-Bu)], [ZA3453; F, H, Me, Me, NMeCH ₂ (c-Pen)], [ZA3454; F, H, Me, Me, NMeCH ₂ (c-Hex)], [ZA3455; F , H, Me, Me, NMeCH ₂ F], [ZA3456; F, H, Me, Me, NMeCHF ₂ ], [ZA3457; F, H, Me, Me, NMeCF ₃ ], [ZA3458; F, H, Me , Me, NMe (CH ₂ ) ₂ F], [ZA3459; F, H, Me, Me, NMeCH ₂ CHF ₂ ], [ZA3460; F, H, Me, Me, NMeCH ₂ CHF ₃ ], [ZA3461; F , H, Me, Me, NMe (CH ₂ ) ₃ F], [ZA3462; F, H, Me, Me, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA3463; F, H, Me, Me, NMe ( CH ₂ ) ₂ CF ₃ ], [ZA3464; F, H, Me, Me, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA3465; F, H, Me, Me, NMeCH ₂ Cl], [ZA3466; F, H, Me, Me, NMe (CH ₂ ) ₂ Cl], [ZA3467; F, H, Me, Me, NMe (CH ₂ ) ₃ Cl], [ZA3468; F, H, Me, Me, NMe (CH ₂ ) ₄ Cl], [ZA3469; F, H, Me, Me, NMe (CH ₂ ) ₅ Cl], [ZA3470; F, H, Me, Me, NMeCH ₂ OMe], [ZA3471; F, H, Me, Me, NMe (CH ₂ ) ₂ OMe], [ZA3472; F, H, Me, Me, NMe (CH ₂ ) ₃ OMe], [ZA3473; F, H, Me, Me, NMe (CH ₂ ) ₄ OMe] , [ZA3474; F, H, Me, Me, NMeCH ₂ OEt], [ZA3475; F, H, Me, Me, NMe (CH ₂ ) ₂ OEt], [ZA3476; F, H, Me, Me, NMe ( _{CH 2) 3 OEt], [} ZA3477; F, H, Me, Me, NMeCH 2 OPr], [ZA3478; F, H, Me, Me, NMe (CH 2) 2 OPr], [ZA3479; F, H, Me, Me, NMe (CH ₂ ) ₃ OPr], [ZA3480; F, H, Me, Me, NMeCH ₂ CN], [ZA3481; F, H, Me, Me, NMe (CH ₂ ) ₂ CN], [ ZA3 482; F, H, Me, Me, NMe (CH 2) 3 CN], [ZA3483; F, H, Me, Me, NMe (CH 2) 4 CN], [ZA3484; F, H, Me, Me, NMe (CH ₂ ) ₅ CN], [ZA3485; F, H, Me, Me, NMeCH ₂ CH = CH ₂ ], [ZA3486; F, H, Me, Me, NMeCH ₂ C≡CH], [ZA3487; F , H, Me, Me, NMeCH ₂ C≡CCH ₃ ], [ZA3488; F, H, Me, Me, NMeCH ₂ Ph], [ZA3489; F, H, Me, Me, NMeCH ₂ (2-Py)] , [ZA3490; F, H, Me, Me, NMeCH ₂ (3-Py)], [ZA3491; F, H, Me, Me, NMeCH ₂ (4-Py)], [ZA3492; F, H, Me, Me, NMe (CH ₂ ) ₂ Ph], [ZA3493; F, H, Me, Me, NMe (CH ₂ ) ₂ (2-Py)], [ZA3494; F, H, Me, Me, NMe (CH ₂ ) ₂ (3-Py)], [ZA3495; F, H, Me, Me, NMe (CH ₂ ) ₂ (4-Py)], [ZA3496; F,
H, Me, Me, NMePh], [ZA3497; F, H, Me, Me, NMe (2-Py)], [ZA3498; F, H, Me, Me, NMe (3-Py)], [ZA3499; F, H, Me, Me, NMe (4-Py)], [ZA3500; F, H, Me, Me, NEt ₂ ],

[ZA3501; F, H, Me, Me, NEtPr], [ZA3502; F, H, Me, Me, NEtBu], [ZA3503; F, H, Me, Me, NEtPen], [ZA3504; F, H, Me , Me, NEtHex], [ZA3505; F, H, Me, Me, NEt (i-Pr)], [ZA3506; F, H, Me, Me, NEt (i-Bu)], [ZA3507; F, H , Me, Me, NEt (c-Pr)], [ZA3508; F, H, Me, Me, NEt (c-Bu)], [ZA3509; F, H, Me, Me, NEt (c-Pen)] , [ZA3510; F, H, Me, Me, NEt (c-Hex)], [ZA3511; F, H, Me, Me, NEtCH ₂ (c-Pr)], [ZA3512; F, H, Me, Me , NEtCH ₂ (c-Bu)], [ZA3513; F, H, Me, Me, NEtCH ₂ (c-Pen)], [ZA3514; F, H, Me, Me, NEtCH ₂ (c-Hex)], [ZA3515; F, H, Me, Me, NEtCH ₂ F], [ZA3516; F, H, Me, Me, NEtCHF ₂ ], [ZA3517; F, H, Me, Me, NEtCF ₃ ], [ZA3518; F , H, Me, Me, NEt (CH ₂ ) ₂ F], [ZA3519; F, H, Me, Me, NEtCH ₂ CHF ₂ ], [ZA3520; F, H, Me, Me, NEtCH ₂ CHF ₃ ], [ZA3521; F, H, Me, Me, NEt (CH ₂ ) ₃ F], [ZA3522; F, H, Me, Me, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA3523; F, H, Me, Me, NEt (CH ₂ ) ₂ CF ₃ ], [ZA3524; F, H, Me, Me, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA3525; F, H, Me, Me, NEtCH ₂ Cl], [ ZA3526; F, H, Me, Me, NEt (CH ₂ ) ₂ Cl], [ZA3527; F, H, Me, Me, NEt (CH ₂ ) ₃ Cl], [ZA3528; F, H, Me, Me, NEt (CH ₂ ) ₄ Cl], [ZA3529; F, H, Me, Me, NEt (CH ₂ ) ₅ Cl], [ZA3530; F, H, Me, Me, NEtCH ₂ OMe], [ZA3531; F, H, Me, Me, NEt (CH ₂ ) ₂ OMe], [ZA3532; F, H, Me, Me, NEt (CH ₂ ) ₃ OMe], [ZA3533; F, H, Me, Me, NEt (CH ₂ ) ₄ OMe], [ZA3534; F, H, Me, Me, NEtCH ₂ OEt], [ZA3535; F, H, Me, Me, NEt (CH ₂ ) ₂ OEt], [ZA3536; F, H, Me, Me, NEt (CH ₂ ) ₃ OEt], [ZA3537; F, H, Me, Me, NEtCH ₂ OPr], [ZA3538; F, H, Me, Me, NEt (CH ₂ ) ₂ OPr], [ZA3539; F, H, Me, Me, NEt (CH ₂ ) ₃ OPr], [ ZA3540; F, H, Me, Me, NEtCH ₂ CN], [ZA3541; F, H, Me, Me, NEt (CH ₂ ) ₂ CN], [ZA3542; F, H, Me, Me, NEt (CH ₂ ) ₃ CN], [ZA3543; F, H, Me, Me, NEt (CH ₂ ) ₄ CN], [ZA3544; F, H, Me, Me, NEt (CH ₂ ) ₅ CN], [ZA3545; F, H, Me, Me, NEtCH ₂ CH = CH ₂ ], [ZA3546; F, H, Me, Me, NEtCH ₂ C≡CH], [ZA3547; F, H, Me, Me, NEtCH ₂ C≡CCH ₃ ] , [ZA3548; F, H, Me, Me, NEtCH ₂ Ph], [ZA3549; F, H, Me, Me, NEtCH ₂ (2-Py)], [ZA3550; F, H, Me, Me, NEtCH ₂ (3-Py)], [ZA3551; F, H, Me, Me, NEtCH ₂ (4-Py)], [ZA3552; F, H, Me, Me, NEt (CH ₂ ) ₂ Ph], [ZA3553; F, H, Me, Me, NEt (CH ₂ ) ₂ (2-Py)], [ZA3554; F, H, Me, Me, NEt (CH ₂ ) ₂ (3-Py)], [ZA3555; F, H, Me, Me, NEt (CH ₂ ) ₂ (4-Py)], [ZA3556; F, H, Me, Me, NEtPh], [ZA3557; F, H, Me, Me, NEt (2-Py) ], [ZA3558; F, H, Me, Me, NEt (3-Py)], [ZA3559; F, H, Me, Me, NEt (4-Py)], [ZA3560; F, H, Me, Me , Pyr], [ZA3561; F, H, Me, Me, Pip], [ZA3562; F, H, Me, Me, Mor], [ZA3563; F, H, Me, Me, OMe], [ZA3564; F, H, Me, Me, OEt], [ZA3565; F, H, Me, Me, OPr] , [ZA3566; F, H, Me, Me, OBu], [ZA3567; F, H, Me, Me, OPen], [ZA3568; F, H, Me, Me, OHex], [ZA3569; F, H, Me, Me, O (i-Pr)], [ZA3570; F, H, Me, Me, O (i-Bu)], [ZA3571; F, H, Me, Me, O (c-Pr)], [ZA3572; F, H, Me, Me, O (c-Bu)], [ZA3573; F, H, Me, Me, O (c-Pen)], [ZA3574; F, H, Me, Me, O (c-Hex)], [ZA3575; F, H, Me, Me, OCH ₂ (c-Pr)], [ZA3576; F, H, Me, Me, OCH ₂ (c-Bu)], [ZA3577; F, H, Me, Me, OCH ₂ (c-Pen)], [ZA3578; F, H, Me, Me, OCH ₂ (c-Hex)], [ZA3579; F, H, Me, Me, OCH ₂ F], [ZA3580; F, H, Me, Me, OCHF ₂ ], [ZA3581; F, H, Me, Me, OCF ₃ ], [ZA3582; F, H, Me, Me, O (CH ₂ ) ₂ F], [ZA3583; F, H, Me, Me, OCH ₂ CHF ₂ ], [ZA3584; F, H, Me, Me, OCH ₂ CHF ₃ ], [ZA3585; F, H, Me, Me, O ( CH ₂ ) ₃ F], [ZA3586; F, H, Me, Me, O (CH ₂ ) ₂ CHF ₂ ], [ZA3587; F, H, Me, Me, O (CH ₂ ) ₂ CF ₃ ], [ ZA3588; F, H, Me, Me, OCH ₂ CH (CF ₃ ) ₂ ], [ZA3589; F, H, Me, Me, OCH ₂ Cl], [ZA3590; F, H, Me, Me, O (CH _{2) 2 Cl], [ZA3591} ; F, H, Me, Me, O (CH 2) 3 Cl], [ZA3592; F, H, Me, Me, O (CH 2) 4 Cl], [ZA3593; F , H, Me, Me, O (CH ₂ ) ₅ Cl], [ZA3594; F, H, Me, Me, OCH ₂ OMe], [ZA3595; F, H, Me, Me, O (CH ₂ ) ₂ OMe ], [ZA3596; F, H , Me, Me, O (CH ₂ ) ₃ OMe], [ZA3597; F, H, Me, Me, O (CH ₂ ) ₄ OMe], [ZA3598; F, H, Me, Me, OCH ₂ OEt], [ZA3599; F, H, Me, Me, O (CH ₂ ) ₂ OEt], [ZA3600; F, H, Me, Me, O (CH ₂ ) ₃ OEt], [ZA3601; F, H, Me, Me , OCH ₂ OPr], [ZA3602; F, H, Me, Me, O (CH ₂ ) ₂ OPr], [ZA3603; F, H, Me, Me, O (CH ₂ ) ₃ OPr], [ZA3604; F , H, Me, Me, OCH ₂ CN], [ZA3605; F, H, Me, Me, O (CH ₂ ) ₂ CN], [ZA3606; F, H, Me, Me, O (CH ₂ ) ₃ CN ], [ZA3607; F, H, Me, Me, O (CH ₂ ) ₄ CN], [ZA3608; F, H, Me, Me, O (CH ₂ ) ₅ CN], [ZA3609; F, H, Me , Me, OCH ₂ CH = CH ₂ ], [ZA3610; F, H, Me, Me, OCH ₂ C≡CH], [ZA3611; F, H, Me, Me, OCH ₂ C≡CCH ₃ ], [ZA3612 ; F, H, Me, Me, OCH ₂ Ph], [ZA3613; F, H, Me, Me, OCH ₂ (2-Py)], [ZA3614; F, H, Me, Me, OCH ₂ (3- Py)], [ZA3615; F, H, Me, Me, OCH ₂ (4-Py)], [ZA3616; F, H, Me, Me, O (CH ₂ ) ₂ Ph], [ZA3617; F, H , Me, Me, O (CH ₂ ) ₂ (2-Py)], [ZA3618; F, H, Me, Me, O (CH ₂ ) ₂ (3-Py)], [ZA3619; F, H, Me , Me, O (CH ₂ ) ₂ (4-Py)], [ZA3620; F, H, Me, Me, OPh], [ZA3621; F, H, Me, Me, O (2-Py)], [ ZA3622; F, H, Me, Me, O (3-Py)], [ZA3623; F, H, Me, Me, O (4-Py)], [ZA3624; F, H, Me, Me, Me] , [ZA3625; F, H, Me, Me, Et], [ZA3626; F, H, Me, Me, Pr], [ZA3627; F, H, Me, Me, Bu], [ZA3628; F, H, Me, Me, Pen], [ZA3 629; F, H, Me, Me, Hex], [ZA3630; F, H, Me, Me, (i-Pr)], [ZA3631; F, H, Me, Me, (i-Bu)], [ ZA3632; F, H, Me, Me, (c-Pr)], [ZA3633; F, H, Me, Me, (c-Bu)], [ZA3634; F, H, Me, Me, (c-Pen )], [ZA3635; F, H, Me, Me, (c-Hex)], [ZA3636; F, H, Me, Me, CH ₂ (c-Pr)], [ZA3637; F, H, Me, Me, CH ₂ (c-Bu)], [ZA3638; F, H, Me, Me, CH ₂ (c-Pen)], [ZA3639; F, H, Me, Me, CH ₂ (c-Hex)] , [ZA3640; F, H, Me, Me, CH ₂ F], [ZA3641; F, H, Me, Me, CHF ₂ ], [ZA3642; F, H, Me, Me, CF ₃ ], [ZA3643; F, H, Me, Me, (CH ₂ ) ₂ F], [ZA3644; F, H, Me, Me, CH ₂ CHF ₂ ], [ZA3645; F, H, Me, Me, CH ₂ CHF ₃ ], [ZA3646; F, H, Me, Me, (CH ₂ ) ₃ F], [ZA3647; F, H, Me, Me, (CH ₂ ) ₂ CHF ₂ ], [ZA3648; F, H, Me, Me, (CH ₂ ) ₂ CF ₃ ], [ZA3649; F, H, Me, Me, CH ₂ CH (CF ₃ ) ₂ ], [ZA3650; F, H, Me, Me, CH ₂ Cl], [ZA3651; F , H, Me, Me, (CH ₂ ) ₂ Cl], [ZA3652; F, H, Me, Me, (CH ₂ ) ₃ Cl], [ZA3653; F, H, Me, Me, (CH ₂ ) ₄ Cl], [ZA3654; F, H, Me, Me, (CH ₂ ) ₅ Cl], [ZA3655; F, H, Me, Me, CH ₂ OMe], [ZA3656; F, H, Me, Me, ( CH ₂ ) ₂ OMe], [ZA3657; F, H, Me, Me, (CH ₂ ) ₃ OMe], [ZA3658; F, H, Me, Me, (CH ₂ ) ₄ OMe], [ZA3659; F, H, Me, Me, CH ₂ OEt], [ZA3660; F, H, Me, Me, (CH ₂ ) ₂ OEt], [ZA3661; F, H, Me, Me, (CH ₂ ) ₃ OEt], [ ZA3662; F, H, Me, Me, CH ₂ OPr], [ZA3663; F, H, Me, Me, (CH ₂ ) ₂ OPr], [ZA3664; F, H, Me, Me, (CH ₂ ) ₃ OPr], [ZA3665; F, H, Me, Me, CH ₂ CN], [ZA3666; F, H, Me, Me, (CH ₂ ) ₂ CN], [ZA3667; F, H, Me, Me, (CH ₂ ) ₃ CN] , [ZA3668; F, H, Me, Me, (CH ₂ ) ₄ CN], [ZA3669; F, H, Me, Me, (CH ₂ ) ₅ CN], [ZA3670; F, H, Me, Me, CH ₂ CH = CH ₂ ], [ZA3671; F, H, Me, Me, CH ₂ C≡CH], [ZA3672; F, H, Me, Me, CH ₂ C≡CCH ₃ ], [ZA3673; F, H, Me, Me, CH ₂ Ph], [ZA3674; F, H, Me, Me, CH ₂ (2-Py)], [ZA3675; F, H, Me, Me, CH ₂ (3-Py)] , [ZA3676; F, H, Me, Me, CH ₂ (4-Py)], [ZA3677; F, H, Me, Me, (CH ₂ ) ₂ Ph], [ZA3678; F, H, Me, Me , (CH ₂ ) ₂ (2-Py)], [ZA3679; F, H, Me, Me, (CH ₂ ) ₂ (3-Py)], [ZA3680; F, H, Me, Me, (CH ₂ ) ₂ (4-Py)], [ZA3681; F, H, Me, Me, Ph], [ZA3682; F, H, Me, Me, 2-Py], [ZA3683; F, H, Me, Me, 3-Py], [ZA3684; F, H, Me, Me, 4-Py], [ZA3685; F, H, F, H, NHMe], [ZA3686; F, H, F, H, NHEt], [ ZA3687; F, H, F, H, NHPr], [ZA3688; F, H, F, H, NHBu], [ZA3689; F, H, F, H, NHPen], [ZA3690; F, H, F, H, NHHex], [ZA3691; F, H, F, H, NH (i-Pr)], [ZA3692; F, H, F, H, NH (i-Bu)], [ZA3693; F, H, F, H, NH (c-Pr)], [ZA3694; F, H, F, H, NH (c-Bu)], [ZA3695; F, H, F, H, NH (c-Pen)], [ZA3696; F, H, F, H, NH (c-Hex)], [ZA3697; F, H, F, H, NH CH ₂ (c-Pr)], [ZA3698; F, H, F, H, NHCH ₂ (c-Bu)], [ZA3699; F, H, F, H, NHCH ₂ (c-Pen)], [ ZA3700; F, H, F, H, NHCH ₂ (c-Hex)], [ZA3701; F, H, F, H, NHCH ₂ F], [ZA3702; F, H, F, H, NHCHF ₂ ], [ZA3703; F, H, F, H, NHCF ₃ ], [ZA3704; F, H, F, H, NH (CH ₂ ) ₂ F], [ZA3705; F, H, F, H, NHCH ₂ CHF ₂ ], [ZA3706; F, H, F, H, NHCH ₂ CHF ₃ ], [ZA3707; F, H, F, H, NH (CH ₂ ) ₃ F], [ZA3708; F, H, F, H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA3709; F, H, F, H, NH (CH ₂ ) ₂ CF ₃ ], [ZA3710; F, H, F, H, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA3711; F, H, F, H, NHCH ₂ Cl], [ZA3712; F, H, F, H, NH (CH ₂ ) ₂ Cl], [ZA3713; F, H, F, H, NH (CH ₂ ) ₃ Cl], [ZA3714; F, H, F, H, NH (CH ₂ ) ₄ Cl], [ZA3715; F, H, F, H, NH (CH ₂ ) ₅ Cl], [ZA3716 ; F, H, F, H, NHCH ₂ OMe], [ZA3717; F, H, F, H, NH (CH ₂ ) ₂ OMe], [ZA3718; F, H, F, H, NH (CH ₂ ) ₃ OMe], [ZA3719; F, H, F, H, NH (CH ₂ ) ₄ OMe], [ZA3720; F, H, F, H, NHCH ₂ OEt], [ZA3721; F, H, F, H , NH (CH ₂ ) ₂ OEt], [ZA3722; F, H, F, H, NH (CH ₂ ) ₃ OEt], [ZA3723; F, H, F, H, NHCH ₂ OPr], [ZA3724; F , H, F, H, NH (CH ₂ ) ₂ OPr], [ZA3725; F, H, F, H, NH (CH ₂ ) ₃ OPr], [ZA3726; F, H, F, H, NHCH ₂ CN ], [ZA3727; F, H, F, H, NH (CH ₂ ) ₂ CN], [ZA3728; F, H, F, H, NH (CH ₂ ) ₃ CN], [ZA3729; F, H, F , H, NH (CH _{2) 4 CN], [ZA3730} ; F, H, F, H, NH (CH 2) 5 CN], [ZA3731; F, H, F, H, NHCH 2 CH = CH 2], [ZA3732; F, H, F, H, NHCH ₂ C≡CH], [ZA3733; F, H, F, H, NHCH ₂ C≡CCH ₃ ], [ZA3734; F, H, F, H, NHCH ₂ Ph], [ZA3735 ; F, H, F, H, NHCH ₂ (2-Py)], [ZA3736; F, H, F, H, NHCH ₂ (3-Py)], [ZA3737; F, H, F, H, NHCH ₂ (4-Py)], [ZA3738; F, H, F, H, NH (CH ₂ ) ₂ Ph], [ZA3739; F, H, F, H, NH (CH ₂ ) ₂ (2-Py) ], [ZA3740; F, H, F, H, NH (CH ₂ ) ₂ (3-Py)], [ZA3741; F, H, F, H, NH (CH ₂ ) ₂ (4-Py)], [ZA3742; F, H, F, H, NHPh], [ZA3743; F, H, F, H, NH (2-Py)], [ZA3744; F, H, F, H, NH (3-Py) ], [ZA3745; F, H, F, H, NH (4-Py)], [ZA3746; F, H
, F, H, NMe ₂ ], [ZA3747; F, H, F, H, NMeEt], [ZA3748; F, H, F, H, NMePr], [ZA3749; F, H, F, H, NMeBu] , [ZA3750; F, H, F, H, NMePen],

[ZA3751; F, H, F, H, NMeHex], [ZA3752; F, H, F, H, NMe (i-Pr)], [ZA3753; F, H, F, H, NMe (i-Bu) ], [ZA3754; F, H, F, H, NMe (c-Pr)], [ZA3755; F, H, F, H, NMe (c-Bu)], [ZA3756; F, H, F, H , NMe (c-Pen)], [ZA3757; F, H, F, H, NMe (c-Hex)], [ZA3758; F, H, F, H, NMeCH ₂ (c-Pr)], [ZA3759 ; F, H, F, H, NMeCH ₂ (c-Bu)], [ZA3760; F, H, F, H, NMeCH ₂ (c-Pen)], [ZA3761; F, H, F, H, NMeCH ₂ (c-Hex)], [ZA3762; F, H, F, H, NMeCH ₂ F], [ZA3763; F, H, F, H, NMeCHF ₂ ], [ZA3764; F, H, F, H, NMeCF ₃ ], [ZA3765; F, H, F, H, NMe (CH ₂ ) ₂ F], [ZA3766; F, H, F, H, NMeCH ₂ CHF ₂ ], [ZA3767; F, H, F, H, NMeCH ₂ CHF ₃ ], [ZA3768; F, H, F, H, NMe (CH ₂ ) ₃ F], [ZA3769; F, H, F, H, NMe (CH ₂ ) ₂ CHF ₂ ], [ ZA3770; F, H, F, H, NMe (CH ₂ ) ₂ CF ₃ ], [ZA3771; F, H, F, H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA3772; F, H, F, H, NMeCH ₂ Cl], [ZA3773; F, H, F, H, NMe (CH ₂ ) ₂ Cl], [ZA3774; F, H, F, H, NMe (CH ₂ ) ₃ Cl], [ZA3775; F, H, F, H, NMe (CH ₂ ) ₄ Cl], [ZA3776; F, H, F, H, NMe (CH ₂ ) ₅ Cl], [ZA3777; F, H, F, H, NMeCH ₂ OMe], [ZA3778; F, H, F, H, NMe (CH ₂ ) ₂ OMe], [ZA3779; F, H, F, H, NMe (CH ₂ ) ₃ OMe], [ZA3780; F, H, F, H, NMe (CH ₂ ) ₄ OMe], [ZA3781; F, H, F, H, NMeCH ₂ OEt], [ZA3782; F, H, F, H, NMe (CH ₂ ) ₂ OEt], [ ZA3783; F , H, F, H, NMe (CH ₂ ) ₃ OEt], [ZA3784; F, H, F, H, NMeCH ₂ OPr], [ZA3785; F, H, F, H, NMe (CH ₂ ) ₂ OPr ], [ZA3786; F, H, F, H, NMe (CH ₂ ) ₃ OPr], [ZA3787; F, H, F, H, NMeCH ₂ CN], [ZA3788; F, H, F, H, NMe (CH ₂ ) ₂ CN], [ZA3789; F, H, F, H, NMe (CH ₂ ) ₃ CN], [ZA3790; F, H, F, H, NMe (CH ₂ ) ₄ CN], [ZA3791 ; F, H, F, H, NMe (CH ₂ ) ₅ CN], [ZA3792; F, H, F, H, NMeCH ₂ CH = CH ₂ ], [ZA3793; F, H, F, H, NMeCH ₂ C≡CH], [ZA3794; F, H, F, H, NMeCH ₂ C≡CCH ₃ ], [ZA3795; F, H, F, H, NMeCH ₂ Ph], [ZA3796; F, H, F, H , NMeCH ₂ (2-Py)], [ZA3797; F, H, F, H, NMeCH ₂ (3-Py)], [ZA3798; F, H, F, H, NMeCH ₂ (4-Py)], [ZA3799; F, H, F, H, NMe (CH ₂ ) ₂ Ph], [ZA3800; F, H, F, H, NMe (CH ₂ ) ₂ (2-Py)], [ZA3801; F, H , F, H, NMe (CH ₂ ) ₂ (3-Py)], [ZA3802; F, H, F, H, NMe (CH ₂ ) ₂ (4-Py)], [ZA3803; F, H, F , H, NMePh], [ZA3804; F, H, F, H, NMe (2-Py)], [ZA3805; F, H, F, H, NMe (3-Py)], [ZA3806; F, H , F, H, NMe (4-Py)], [ZA3807; F, H, F, H, NEt ₂ ], [ZA3808; F, H, F, H, NEtPr], [ZA3809; F, H, F , H, NEtBu], [ZA3810; F, H, F, H, NEtPen], [ZA3811; F, H, F, H, NEtHex], [ZA3812; F, H, F, H, NEt (i-Pr )], [ZA3813; F, H, F, H, NEt (i-Bu)], [ZA3814; F, H, F, H, NEt (c-Pr)], [ZA3815; F, H, F, H, NEt (c-Bu)], [ZA3816; F, H, F, H, NE t (c-Pen)], [ZA3817; F, H, F, H, NEt (c-Hex)], [ZA3818; F, H, F, H, NEtCH ₂ (c-Pr)], [ZA3819; F, H, F, H, NEtCH ₂ (c-Bu)], [ZA3820; F, H, F, H, NEtCH ₂ (c-Pen)], [ZA3821; F, H, F, H, NEtCH ₂ (c-Hex)], [ZA3822; F, H, F, H, NEtCH ₂ F], [ZA3823; F, H, F, H, NEtCHF ₂ ], [ZA3824; F, H, F, H, NEtCF ₃ ], [ZA3825; F, H, F, H, NEt (CH ₂ ) ₂ F], [ZA3826; F, H, F, H, NEtCH ₂ CHF ₂ ], [ZA3827; F, H, F, H , NEtCH ₂ CHF ₃ ], [ZA3828; F, H, F, H, NEt (CH ₂ ) ₃ F], [ZA3829; F, H, F, H, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA3830 ; F, H, F, H, NEt (CH ₂ ) ₂ CF ₃ ], [ZA3831; F, H, F, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA3832; F, H, F, H , NEtCH ₂ Cl], [ZA3833; F, H, F, H, NEt (CH ₂ ) ₂ Cl], [ZA3834; F, H, F, H, NEt (CH ₂ ) ₃ Cl], [ZA3835; F , H, F, H, NEt (CH ₂ ) ₄ Cl], [ZA3836; F, H, F, H, NEt (CH ₂ ) ₅ Cl], [ZA3837; F, H, F, H, NEtCH ₂ OMe ], [ZA3838; F, H, F, H, NEt (CH ₂ ) ₂ OMe], [ZA3839; F, H, F, H, NEt (CH ₂ ) ₃ OMe], [ZA3840; F, H, F , H, NEt (CH ₂ ) ₄ OMe], [ZA3841; F, H, F, H, NEtCH ₂ OEt], [ZA3842; F, H, F, H, NEt (CH ₂ ) ₂ OEt], [ZA3843 ; F, H, F, H, NEt (CH ₂ ) ₃ OEt], [ZA3844; F, H, F, H, NEtCH ₂ OPr], [ZA3845; F, H, F, H, NEt (CH ₂ ) ₂ OPr], [ZA3846; F, H, F, H, NEt (CH ₂ ) ₃ OPr], [ZA3847; F, H, F, H, NEtCH ₂ CN], [ZA3848; F, H, F, H, NEt (CH ₂ ) ₂ CN], [ZA3849; F, H, F, H, NEt (CH ₂ ) ₃ CN], [ZA3850; F, H, F, H , NEt (CH ₂ ) ₄ CN], [ZA3851; F, H, F, H, NEt (CH ₂ ) ₅ CN], [ZA3852; F, H, F, H, NEtCH ₂ CH = CH ₂ ], [ ZA3853; F, H, F, H, NEtCH ₂ C≡CH], [ZA3854; F, H, F, H, NEtCH ₂ C≡CCH ₃ ], [ZA3855; F, H, F, H, NEtCH ₂ Ph ], [ZA3856; F, H, F, H, NEtCH ₂ (2-Py)], [ZA3857; F, H, F, H, NEtCH ₂ (3-Py)], [ZA3858; F, H, F , H, NEtCH ₂ (4-Py)], [ZA3859; F, H, F, H, NEt (CH ₂ ) ₂ Ph], [ZA3860; F, H, F, H, NEt (CH ₂ ) ₂ ( 2-Py)], [ZA3861; F, H, F, H, NEt (CH ₂ ) ₂ (3-Py)], [ZA3862; F, H, F, H, NEt (CH ₂ ) ₂ (4- Py)], [ZA3863; F, H, F, H, NEtPh], [ZA3864; F, H, F, H, NEt (2-Py)], [ZA3865; F, H, F, H, NEt ( 3-Py)], [ZA3866; F, H, F, H, NEt (4-Py)], [ZA3867; F, H, F, H, Pyr], [ZA3868; F, H, F, H, Pip], [ZA3869; F, H, F, H, Mor], [ZA3870; F, H, F, H, OMe], [ZA3871; F, H, F, H, OEt], [ZA3872; F, H, F, H, OPr], [ZA3873; F, H, F, H, OBu], [ZA3874; F, H, F, H, OPen], [ZA3875; F, H, F, H, OHex] , [ZA3876; F, H, F, H, O (i-Pr)], [ZA3877; F, H, F, H, O (i-Bu)], [ZA3878; F, H, F, H, O (c-Pr)], [ZA3879; F, H, F, H, O (c-Bu)], [ZA3880; F, H, F, H, O (c-Pen)], [ZA3881; F , H, F, H, O (c-Hex)], [ZA3882; F, H, F, H, OCH ₂ (c-Pr)], [ZA3883; F, H, F, H, OCH ₂ (c-Bu)], [ZA3884; F, H, F, H, OCH ₂ (c-Pen)], [ZA3885; F, H, F, H, OCH ₂ (c-Hex)], [ZA3886; F, H, F, H, OCH ₂ F], [ZA3887; F, H, F, H, OCHF ₂ ], [ZA3888; F, H, F, H, OCF ₃ ], [ZA3889; F, H, F, H, O (CH ₂ ) ₂ F], [ZA3890; F, H, F, H, OCH ₂ CHF ₂ ], [ZA3891; F, H, F, H, OCH ₂ CHF ₃ ], [ZA3892; F, H, F, H, O (CH ₂ ) ₃ F], [ZA3893; F, H, F, H, O (CH ₂ ) ₂ CHF ₂ ], [ZA3894; F, H, F, H, O (CH ₂ ) ₂ CF ₃ ], [ZA3895; F, H, F, H, OCH ₂ CH (CF ₃ ) ₂ ], [ZA3896; F, H, F, H, OCH ₂ Cl], [ZA3897; F , H, F, H, O (CH ₂ ) ₂ Cl], [ZA3898; F, H, F, H, O (CH ₂ ) ₃ Cl], [ZA3899; F, H, F, H, O (CH ₂ ) ₄ Cl], [ZA3900; F, H, F, H, O (CH ₂ ) ₅ Cl], [ZA3901; F, H, F, H, OCH ₂ OMe], [ZA3902; F, H, F , H, O (CH ₂ ) ₂ OMe], [ZA3903; F, H, F, H, O (CH ₂ ) ₃ OMe], [ZA3904; F, H, F, H, O (CH ₂ ) ₄ OMe ], [ZA3905; F, H, F, H, OCH ₂ OEt], [ZA3906; F, H, F, H, O (CH ₂ ) ₂ OEt], [ZA3907; F, H, F, H, O (CH ₂ ) ₃ OEt], [ZA3908; F, H, F, H, OCH ₂ OPr], [ZA3909; F, H, F, H, O (CH ₂ ) ₂ OPr], [ZA3910; F, H , F, H, O (CH ₂ ) ₃ OPr], [ZA3911; F, H, F, H, OCH ₂ CN], [ZA3912; F, H, F, H, O (CH ₂ ) ₂ CN], [ZA3913; F, H, F, H, O (CH ₂ ) ₃ CN], [ZA3914; F, H, F, H, O (CH ₂ ) ₄ CN], [ZA3915; F, H, F, H , O (CH ₂ ) ₅ CN], [ZA3916; F, H, F, H, OCH ₂ CH = CH ₂ ], [ZA3917; F, H, F, H, OCH ₂ C≡CH], [ZA3918; F, H, F, H, OCH ₂ C≡CCH ₃ ], [ZA3919; F, H, F, H, OCH ₂ Ph], [ZA3920; F, H, F, H, OCH ₂ (2-Py)], [ZA3921; F, H, F, H, OCH ₂ (3-Py)], [ZA3922; F, H, F, H, OCH ₂ (4-Py)], [ZA3923; F, H, F, H, O (CH ₂ ) ₂ Ph], [ZA3924; F, H, F, H, O ( CH ₂ ) ₂ (2-Py)], [ZA3925; F, H, F, H, O (CH ₂ ) ₂ (3-Py)], [ZA3926; F, H, F, H, O (CH ₂ ) ₂ (4-Py)], [ZA3927; F, H, F, H, OPh], [ZA3928; F, H, F, H, O (2-Py)], [ZA3929; F, H, F , H, O (3-Py)], [ZA3930; F, H, F, H, O (4-Py)], [ZA3931; F, H, F, H, Me], [ZA3932; F, H , F, H, Et], [ZA3933; F, H, F, H, Pr], [ZA3934; F, H, F, H, Bu], [ZA3935; F, H, F, H, Pen], [ZA3936; F, H, F, H, Hex], [ZA3937; F, H, F, H, (i-Pr)], [ZA3938; F, H, F, H, (i-Bu)], [ZA3939; F, H, F, H, (c-Pr)], [ZA3940; F, H, F, H, (c-Bu)], [ZA3941; F, H, F, H, (c- Pen)], [ZA3942; F, H, F, H, (c-Hex)], [ZA3943; F, H, F, H, CH ₂ (c-Pr)], [ZA3944; F, H, F , H, CH ₂ (c-Bu)], [ZA3945; F, H, F, H, CH ₂ (c-Pen)], [ZA3946; F, H, F, H, CH ₂ (c-Hex) ], [ZA3947; F, H, F, H, CH ₂ F], [ZA3948; F, H, F, H, CHF ₂ ], [ZA3949; F, H, F, H, CF ₃ ], [ZA3950 ; F, H, F, H, (CH ₂ ) ₂ F], [ZA3951; F, H, F, H, CH ₂ CHF ₂ ], [ZA3952; F, H, F, H, CH ₂ CHF ₃ ] , [ZA3953; F, H, F, H, (CH ₂ ) ₃ F], [ZA3954; F, H, F, H, (CH ₂ ) ₂ CHF ₂ ], [ZA3955; F, H, F, H, (CH ₂ ) ₂ CF ₃ ], [ZA3956; F, H, F, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA3957; F, H, F, H, CH ₂ Cl], [ZA3958; F, H, F, H, (CH ₂ ) ₂ Cl], [ZA3959; F, H, F, H, (CH ₂ ) ₃ Cl], [ZA3960; F, H, F, H, (CH ₂ ) ₄ Cl], [ZA3961; F, H, F, H, (CH ₂ ) ₅ Cl], [ZA3962; F, H, F, H, CH ₂ OMe], [ZA3963; F, H, F, H, (CH ₂ ) ₂ OMe], [ZA3964; F, H, F, H, (CH ₂ ) ₃ OMe], [ZA3965; F, H, F, H, (CH ₂ ) ₄ OMe], [ZA3966; F, H, F, H, CH ₂ OEt], [ZA3967; F, H, F, H, (CH ₂ ) ₂ OEt], [ZA3968; F, H, F, H, (CH ₂ ) ₃ OEt], [ZA3969; F, H, F, H, CH ₂ OPr], [ZA3970; F, H, F, H, (CH ₂ ) ₂ OPr], [ZA3971; F, H, F, H, (CH ₂ ) ₃ OPr], [ZA3972; F, H, F, H, CH ₂ CN], [ZA3973; F, H, F, H, (CH ₂ ) ₂ CN], [ZA3974; F, H, F, H, (CH ₂ ) ₃ CN], [ZA3975; F, H, F, H, (CH ₂ ) ₄ CN], [ZA3976; F, H, F, H, (CH ₂ ) ₅ CN], [ZA3977; F, H, F, H, CH ₂ CH = CH ₂ ], [ZA3978; F, H, F , H, CH ₂ C≡CH], [ZA3979; F, H, F, H, CH ₂ C≡CCH ₃ ], [ZA3980; F, H, F, H, CH ₂ Ph], [ZA3981; F, H, F, H, CH ₂ (2-Py)], [ZA3982; F, H, F, H, CH ₂ (3-Py)], [ZA3983; F, H, F, H, CH ₂ (4 -Py)], [ZA3984; F, H, F, H, (CH ₂ ) ₂ Ph], [ZA3985; F, H, F, H, (CH ₂ ) ₂ (2-Py)], [ZA3986; F, H, F, H, (CH ₂ ) ₂ (3-Py)], [ZA3987; F, H, F, H, (C H ₂ ) ₂ (4-Py)], [ZA3988; F, H, F, H, Ph], [ZA3989; F, H, F, H, 2-Py], [ZA3990; F, H, F, H, 3-Py], [ZA3991; F, H, F, H, 4-Py], [ZA3992; F, H, F, F, NHMe], [ZA3993; F, H, F, F, NHEt] , [ZA3994; F, H, F, F, NHPr], [ZA3995; F, H, F, F, NHBu], [ZA3996; F, H, F, F, NHPen], [ZA3997; F, H, F, F, NHHex], [ZA3998; F, H, F, F, NH (i-Pr)], [ZA3999; F, H, F, F, NH (i-Bu)], [ZA4000; F, H, F, F, NH (c-Pr)],

[ZA4001; F, H, F, F, NH (c-Bu)], [ZA4002; F, H, F, F, NH (c-Pen)], [ZA4003; F, H, F, F, NH (c-Hex)], [ZA4004; F, H, F, F, NHCH ₂ (c-Pr)], [ZA4005; F, H, F, F, NHCH ₂ (c-Bu)], [ZA4006; F, H, F, F, NHCH ₂ (c-Pen)], [ZA4007; F, H, F, F, NHCH ₂ (c-Hex)], [ZA4008; F, H, F, F, NHCH ₂ F], [ZA4009; F, H, F, F, NHCHF ₂ ], [ZA4010; F, H, F, F, NHCF ₃ ], [ZA4011; F, H, F, F, NH (CH ₂ ) ₂ F], [ZA4012; F, H, F, F, NHCH ₂ CHF ₂ ], [ZA4013; F, H, F, F, NHCH ₂ CHF ₃ ], [ZA4014; F, H, F, F, NH ( CH ₂ ) ₃ F], [ZA4015; F, H, F, F, NH (CH ₂ ) ₂ CHF ₂ ], [ZA4016; F, H, F, F, NH (CH ₂ ) ₂ CF ₃ ], [ ZA4017; F, H, F, F, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA4018; F, H, F, F, NHCH ₂ Cl], [ZA4019; F, H, F, F, NH (CH _{2) 2 Cl], [ZA4020} ; F, H, F, F, NH (CH 2) 3 Cl], [ZA4021; F, H, F, F, NH (CH 2) 4 Cl], [ZA4022; F , H, F, F, NH (CH ₂ ) ₅ Cl], [ZA4023; F, H, F, F, NHCH ₂ OMe], [ZA4024; F, H, F, F, NH (CH ₂ ) ₂ OMe ], [ZA4025; F, H, F, F, NH (CH ₂ ) ₃ OMe], [ZA4026; F, H, F, F, NH (CH ₂ ) ₄ OMe], [ZA4027; F, H, F , F, NHCH ₂ OEt], [ZA4028; F, H, F, F, NH (CH ₂ ) ₂ OEt], [ZA4029; F, H, F, F, NH (CH ₂ ) ₃ OEt], [ZA4030 ; F, H, F, F, NHCH ₂ OPr], [ZA4031; F, H, F, F, NH (CH ₂ ) ₂ OPr], [ZA4032; F, H, F, F, NH (CH ₂ ) ₃ OPr], [ZA4033; F, H, F, F , NHCH ₂ CN], [ZA4034; F, H, F, F, NH (CH ₂ ) ₂ CN], [ZA4035; F, H, F, F, NH (CH ₂ ) ₃ CN], [ZA4036; F , H, F, F, NH (CH ₂ ) ₄ CN], [ZA4037; F, H, F, F, NH (CH ₂ ) ₅ CN], [ZA4038; F, H, F, F, NHCH ₂ CH = CH ₂ ], [ZA4039; F, H, F, F, NHCH ₂ C≡CH], [ZA4040; F, H, F, F, NHCH ₂ C≡CCH ₃ ], [ZA4041; F, H, F , F, NHCH ₂ Ph], [ZA4042; F, H, F, F, NHCH ₂ (2-Py)], [ZA4043; F, H, F, F, NHCH ₂ (3-Py)], [ZA4044 ; F, H, F, F, NHCH ₂ (4-Py)], [ZA4045; F, H, F, F, NH (CH ₂ ) ₂ Ph], [ZA4046; F, H, F, F, NH (CH ₂ ) ₂ (2-Py)], [ZA4047; F, H, F, F, NH (CH ₂ ) ₂ (3-Py)], [ZA4048; F, H, F, F, NH (CH ₂ ) ₂ (4-Py)], [ZA4049; F, H, F, F, NHPh], [ZA4050; F, H, F, F, NH (2-Py)], [ZA4051; F, H, F, F, NH (3-Py)], [ZA4052; F, H, F, F, NH (4-Py)], [ZA4053; F, H, F, F, NMe ₂ ], [ZA4054; F , H, F, F, NMeEt], [ZA4055; F, H, F, F, NMePr], [ZA4056; F, H, F, F, NMeBu], [ZA4057; F, H, F, F, NMePen ], [ZA4058; F, H, F, F, NMeHex], [ZA4059; F, H, F, F, NMe (i-Pr)], [ZA4060; F, H, F, F, NMe (i- Bu)], [ZA4061; F, H, F, F, NMe (c-Pr)], [ZA4062; F, H, F, F, NMe (c-Bu)], [ZA4063; F, H, F , F, NMe (c-Pen)], [ZA4064; F, H, F, F, NMe (c-Hex)], [ZA4065; F, H, F, F, NMeCH ₂ (c-Pr)], [ZA4066; F, H, F, F, NMeCH ₂ (c-Bu)], [ZA4067; F, H, F, F, NMeCH ₂ (c-Pen)] , [ZA4068; F, H, F, F, NMeCH ₂ (c-Hex)], [ZA4069; F, H, F, F, NMeCH ₂ F], [ZA4070; F, H, F, F, NMeCHF ₂ ], [ZA4071; F, H, F, F, NMeCF ₃ ], [ZA4072; F, H, F, F, NMe (CH ₂ ) ₂ F], [ZA4073; F, H, F, F, NMeCH ₂ CHF ₂ ], [ZA4074; F, H, F, F, NMeCH ₂ CHF ₃ ], [ZA4075; F, H, F, F, NMe (CH ₂ ) ₃ F], [ZA4076; F, H, F, F, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA4077; F, H, F, F, NMe (CH ₂ ) ₂ CF ₃ ], [ZA4078; F, H, F, F, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA4079; F, H, F, F, NMeCH ₂ Cl], [ZA4080; F, H, F, F, NMe (CH ₂ ) ₂ Cl], [ZA4081; F, H, F, F , NMe (CH ₂ ) ₃ Cl], [ZA4082; F, H, F, F, NMe (CH ₂ ) ₄ Cl], [ZA4083; F, H, F, F, NMe (CH ₂ ) ₅ Cl], [ZA4084; F, H, F, F, NMeCH ₂ OMe], [ZA4085; F, H, F, F, NMe (CH ₂ ) ₂ OMe], [ZA4086; F, H, F, F, NMe (CH ₂ ) ₃ OMe], [ZA4087; F, H, F, F, NMe (CH ₂ ) ₄ OMe], [ZA4088; F, H, F, F, NMeCH ₂ OEt], [ZA4089; F, H, F , F, NMe (CH ₂ ) ₂ OEt], [ZA4090; F, H, F, F, NMe (CH ₂ ) ₃ OEt], [ZA4091; F, H, F, F, NMeCH ₂ OPr], [ZA4092 ; F, H, F, F, NMe (CH ₂ ) ₂ OPr], [ZA4093; F, H, F, F, NMe (CH ₂ ) ₃ OPr], [ZA4094; F, H, F, F, NMeCH ₂ CN], [ZA4095; F, H, F, F, NMe (CH ₂ ) ₂ CN], [ZA4096; F, H, F, F, NMe (CH ₂ ) ₃ CN], [ZA4097; F, H , F, F, NMe (CH ₂ ) ₄ CN], [ZA4098; F, H, F, F, NMe (CH ₂ ) ₅ CN], [Z A4099; F, H, F, F, NMeCH ₂ CH = CH ₂ ], [ZA4100; F, H, F, F, NMeCH ₂ C≡CH], [ZA4101; F, H, F, F, NMeCH ₂ C ≡CCH ₃ ], [ZA4102; F, H, F, F, NMeCH ₂ Ph], [ZA4103; F, H, F, F, NMeCH ₂ (2-Py)], [ZA4104; F, H, F, F, NMeCH ₂ (3-Py)], [ZA4105; F, H, F, F, NMeCH ₂ (4-Py)], [ZA4106; F, H, F, F, NMe (CH ₂ ) ₂ Ph] , [ZA4107; F, H, F, F, NMe (CH ₂ ) ₂ (2-Py)], [ZA4108; F, H, F, F, NMe (CH ₂ ) ₂ (3-Py)], [ ZA4109; F, H, F, F, NMe (CH ₂ ) ₂ (4-Py)], [ZA4110; F, H, F, F, NMePh], [ZA4111; F, H, F, F, NMe ( 2-Py)], [ZA4112; F, H, F, F, NMe (3-Py)], [ZA4113; F, H, F, F, NMe (4-Py)], [ZA4114; F, H , F, F, NEt ₂ ], [ZA4115; F, H, F, F, NEtPr], [ZA4116; F, H, F, F, NEtBu], [ZA4117; F, H, F, F, NEtPen] , [ZA4118; F, H, F, F, NEtHex], [ZA4119; F, H, F, F, NEt (i-Pr)], [ZA4120; F, H, F, F, NEt (i-Bu )], [ZA4121; F, H, F, F, NEt (c-Pr)], [ZA4122; F, H, F, F, NEt (c-Bu)], [ZA4123; F, H, F, F, NEt (c-Pen)], [ZA4124; F, H, F, F, NEt (c-Hex)], [ZA4125; F, H, F, F, NEtCH ₂ (c-Pr)], [ ZA4126; F, H, F, F, NEtCH ₂ (c-Bu)], [ZA4127; F, H, F, F, NEtCH ₂ (c-Pen)], [ZA4128; F, H, F, F, NEtCH ₂ (c-Hex)], [ZA4129; F, H, F, F, NEtCH ₂ F], [ZA4130; F, H, F, F, NEtCHF ₂ ], [ZA4131; F, H, F, F , NEtCF ₃ ], [ZA4132; F, H, F, F, NEt (CH ₂ ) ₂ F], [ZA4 133; F, H, F, F, NEtCH ₂ CHF ₂ ], [ZA4134; F, H, F, F, NEtCH ₂ CHF ₃ ], [ZA4135; F, H, F, F, NEt (CH ₂ ) ₃ F], [ZA4136; F, H, F, F, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA4137; F, H, F, F, NEt (CH ₂ ) ₂ CF ₃ ], [ZA4138; F, H, F, F, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA4139; F, H, F, F, NEtCH ₂ Cl], [ZA4140; F, H, F, F, NEt (CH ₂ ) ₂ Cl ], [ZA4141; F, H, F, F, NEt (CH ₂ ) ₃ Cl], [ZA4142; F, H, F, F, NEt (CH ₂ ) ₄ Cl], [ZA4143; F, H, F , F, NEt (CH ₂ ) ₅ Cl], [ZA4144; F, H, F, F, NEtCH ₂ OMe], [ZA4145; F, H, F, F, NEt (CH ₂ ) ₂ OMe], [ZA4146 ; F, H, F, F, NEt (CH ₂ ) ₃ OMe], [ZA4147; F, H, F, F, NEt (CH ₂ ) ₄ OMe], [ZA4148; F, H, F, F, NEtCH ₂ OEt], [ZA4149; F, H, F, F, NEt (CH ₂ ) ₂ OEt], [ZA4150; F, H, F, F, NEt (CH ₂ ) ₃ OEt], [ZA4151; F, H , F, F, NEtCH ₂ OPr], [ZA4152; F, H, F, F, NEt (CH ₂ ) ₂ OPr], [ZA4153; F, H, F, F, NEt (CH ₂ ) ₃ OPr], [ZA4154; F, H, F, F, NEtCH ₂ CN], [ZA4155; F, H, F, F, NEt (CH ₂ ) ₂ CN], [ZA4156; F, H, F, F, NEt (CH _{2) 3 CN], [ZA4157} ; F, H, F, F, NEt (CH 2) 4 CN], [ZA4158; F, H, F, F, NEt (CH 2) 5 CN], [ZA4159; F , H, F, F, NEtCH ₂ CH = CH ₂ ], [ZA4160; F, H, F, F, NEtCH ₂ C≡CH], [ZA4161; F, H, F, F, NEtCH ₂ C≡CCH ₃ ], [ZA4162; F, H, F, F, NEtCH ₂ Ph], [ZA4163; F, H, F, F, NEtCH ₂ (2-Py)], [ZA4164; F, H, F, F, NEtCH ₂ (3-Py)], [ZA4165; F, H, F, F, NEtCH ₂ (4-Py)], [ZA4166 ; F, H, F, F, NEt (CH ₂ ) ₂ Ph], [ZA4167; F, H, F, F, NEt (CH ₂ ) ₂ (2-Py)], [ZA4168; F, H, F , F, NEt (CH ₂ ) ₂ (3-Py)], [ZA4169; F, H, F, F, NEt (CH ₂ ) ₂ (4-Py)], [ZA4170; F, H, F, F , NEtPh], [ZA4171; F, H, F, F, NEt (2-Py)], [ZA4172; F, H, F, F, NEt (3-Py)], [ZA4173; F, H, F , F, NEt (4-Py)], [ZA4174; F, H, F, F, Pyr], [ZA4175; F, H, F, F, Pip], [ZA4176; F, H, F, F, Mor], [ZA4177; F, H, F, F, OMe], [ZA4178; F, H, F, F, OEt], [ZA4179; F, H, F, F, OPr], [ZA4180; F, H, F, F, OBu], [ZA4181; F, H, F, F, OPen], [ZA4182; F, H, F, F, OHex], [ZA4183; F, H, F, F, O ( i-Pr)], [ZA4184; F, H, F, F, O (i-Bu)], [ZA4185; F, H, F, F, O (c-Pr)], [ZA4186; F, H , F, F, O (c-Bu)], [ZA4187; F, H, F, F, O (c-Pen)], [ZA4188; F, H, F, F, O (c-Hex)] , [ZA4189; F, H, F, F, OCH ₂ (c-Pr)], [ZA4190; F, H, F, F, OCH ₂ (c-Bu)], [ZA4191; F, H, F, F, OCH ₂ (c-Pen)], [ZA4192; F, H, F, F, OCH ₂ (c-Hex)], [ZA4193; F, H, F, F, OCH ₂ F], [ZA4194; F, H, F, F, OCHF ₂ ], [ZA4195; F, H, F, F, OCF ₃ ], [ZA4196; F, H, F, F, O (CH ₂ ) ₂ F], [ZA4197; F, H, F, F, OCH ₂ CHF ₂ ], [ZA4198; F, H, F, F, OCH ₂ CHF ₃ ], [ZA4199; F, H, F, F, O (CH ₂ ) ₃ F] , [ZA4200; F, H, F, F, O (C H ₂ ) ₂ CHF ₂ ], [ZA4201; F, H, F, F, O (CH ₂ ) ₂ CF ₃ ], [ZA4202; F, H, F, F, OCH ₂ CH (CF ₃ ) ₂ ], [ZA4203; F, H, F, F, OCH ₂ Cl], [ZA4204; F, H, F, F, O (CH ₂ ) ₂ Cl], [ZA4205; F, H, F, F, O (CH _{2) 3 Cl], [ZA4206} ; F, H, F, F, O (CH 2) 4 Cl], [ZA4207; F, H, F, F, O (CH 2) 5 Cl], [ZA4208; F , H, F, F, OCH ₂ OMe], [ZA4209; F, H, F, F, O (CH ₂ ) ₂ OMe], [ZA4210; F, H, F, F, O (CH ₂ ) ₃ OMe ], [ZA4211; F, H, F, F, O (CH ₂ ) ₄ OMe], [ZA4212; F, H, F, F, OCH ₂ OEt], [ZA4213; F, H, F, F, O (CH ₂ ) ₂ OEt], [ZA4214; F, H, F, F, O (CH ₂ ) ₃ OEt], [ZA4215; F, H, F, F, OCH ₂ OPr], [ZA4216; F, H , F, F, O (CH ₂ ) ₂ OPr], [ZA4217; F, H, F, F, O (CH ₂ ) ₃ OPr], [ZA4218; F, H, F, F, OCH ₂ CN], [ZA4219; F, H, F, F, O (CH ₂ ) ₂ CN], [ZA4220; F, H, F, F, O (CH ₂ ) ₃ CN], [ZA4221; F, H, F, F , O (CH ₂ ) ₄ CN], [ZA4222; F, H, F, F, O (CH ₂ ) ₅ CN], [ZA4223; F, H, F, F, OCH ₂ CH = CH ₂ ], [ ZA4224; F, H, F, F, OCH ₂ C≡CH], [ZA4225; F, H, F, F, OCH ₂ C≡CCH ₃ ], [ZA4226; F, H, F, F, OCH ₂ Ph ], [ZA4227; F, H, F, F, OCH ₂ (2-Py)], [ZA4228; F, H, F, F, OCH ₂ (3-Py)], [ZA4229; F, H, F , F, OCH ₂ (4-Py)], [ZA4230; F, H, F, F, O (CH ₂ ) ₂ Ph], [ZA4231; F, H, F, F, O (CH ₂ ) ₂ ( 2-Py)], [ZA4232; F, H, F, F, O (CH ₂ ) ₂ (3-P y)], [ZA4233; F, H, F, F, O (CH ₂ ) ₂ (4-Py)], [ZA4234; F, H, F, F, OPh], [ZA4235; F, H, F , F, O (2-Py)], [ZA4236; F, H, F, F, O (3-Py)], [ZA4237; F, H, F, F, O (4-Py)], [ ZA4238; F, H, F, F, Me], [ZA4239; F, H, F, F, Et], [ZA4240; F, H, F, F, Pr], [ZA4241; F, H, F, F, Bu], [ZA4242; F, H, F, F, Pen], [ZA4243; F, H, F, F, Hex], [ZA4244; F, H, F, F, (i-Pr)] , [ZA4245; F, H, F, F, (i-Bu)], [ZA4246; F, H, F, F, (c-Pr)], [ZA4247; F, H, F, F, (c -Bu)], [ZA4248; F, H, F, F, (c-Pen)], [ZA4249; F, H, F, F, (c-Hex)], [ZA4250; F, H, F, F, CH ₂ (c-Pr)],

[ZA4251; F, H, F, F, CH ₂ (c-Bu)], [ZA4252; F, H, F, F, CH ₂ (c-Pen)], [ZA4253; F, H, F, F , CH ₂ (c-Hex)], [ZA4254; F, H, F, F, CH ₂ F], [ZA4255; F, H, F, F, CHF ₂ ], [ZA4256; F, H, F, F, CF ₃ ], [ZA4257; F, H, F, F, (CH ₂ ) ₂ F], [ZA4258; F, H, F, F, CH ₂ CHF ₂ ], [ZA4259; F, H, F , F, CH ₂ CHF ₃ ], [ZA4260; F, H, F, F, (CH ₂ ) ₃ F], [ZA4261; F, H, F, F, (CH ₂ ) ₂ CHF ₂ ], [ZA4262 ; F, H, F, F, (CH ₂ ) ₂ CF ₃ ], [ZA4263; F, H, F, F, CH ₂ CH (CF ₃ ) ₂ ], [ZA4264; F, H, F, F, CH ₂ Cl], [ZA4265; F, H, F, F, (CH ₂ ) ₂ Cl], [ZA4266; F, H, F, F, (CH ₂ ) ₃ Cl], [ZA4267; F, H, F, F, (CH ₂ ) ₄ Cl], [ZA4268; F, H, F, F, (CH ₂ ) ₅ Cl], [ZA4269; F, H, F, F, CH ₂ OMe], [ZA4270; F, H, F, F, (CH ₂ ) ₂ OMe], [ZA4271; F, H, F, F, (CH ₂ ) ₃ OMe], [ZA4272; F, H, F, F, (CH ₂ ) ₄ OMe], [ZA4273; F, H, F, F, CH ₂ OEt], [ZA4274; F, H, F, F, (CH ₂ ) ₂ OEt], [ZA4275; F, H, F, F, (CH ₂ ) ₃ OEt], [ZA4276; F, H, F, F, CH ₂ OPr], [ZA4277; F, H, F, F, (CH ₂ ) ₂ OPr], [ZA4278; F, H, F, F, (CH ₂ ) ₃ OPr], [ZA4279; F, H, F, F, CH ₂ CN], [ZA4280; F, H, F, F, (CH ₂ ) ₂ CN], [ZA4281; F, H, F, F, (CH ₂ ) ₃ CN], [ZA4282; F, H, F, F, (CH ₂ ) ₄ CN], [ZA4283; F, H, F, F, (CH ₂ ) ₅ CN], [ZA4284; F, H, F, F, CH ₂ CH = CH ₂ ], [ZA428 5; F, H, F, F, CH ₂ C≡CH], [ZA4286; F, H, F, F, CH ₂ C≡CCH ₃ ], [ZA4287; F, H, F, F, CH ₂ Ph ], [ZA4288; F, H, F, F, CH ₂ (2-Py)], [ZA4289; F, H, F, F, CH ₂ (3-Py)], [ZA4290; F, H, F , F, CH ₂ (4-Py)], [ZA4291; F, H, F, F, (CH ₂ ) ₂ Ph], [ZA4292; F, H, F, F, (CH ₂ ) ₂ (2- Py)], [ZA4293; F, H, F, F, (CH ₂ ) ₂ (3-Py)], [ZA4294; F, H, F, F, (CH ₂ ) ₂ (4-Py)], [ZA4295; F, H, F, F, Ph], [ZA4296; F, H, F, F, 2-Py], [ZA4297; F, H, F, F, 3-Py], [ZA4298; F , H, F, F, 4-Py], [ZA4299; F, H, Cl, H, NHMe], [ZA4300; F, H, Cl, H, NHEt], [ZA4301; F, H, Cl, H , NHPr], [ZA4302; F, H, Cl, H, NHBu], [ZA4303; F, H, Cl, H, NHPen], [ZA4304; F, H, Cl, H, NHHex], [ZA4305; F , H, Cl, H, NH (i-Pr)], [ZA4306; F, H, Cl, H, NH (i-Bu)], [ZA4307; F, H, Cl, H, NH (c-Pr )], [ZA4308; F, H, Cl, H, NH (c-Bu)], [ZA4309; F, H, Cl, H, NH (c-Pen)], [ZA4310; F, H, Cl, H, NH (c-Hex)], [ZA4311; F, H, Cl, H, NHCH ₂ (c-Pr)], [ZA4312; F, H, Cl, H, NHCH ₂ (c-Bu)], [ZA4313; F, H, Cl, H, NHCH ₂ (c-Pen)], [ZA4314; F, H, Cl, H, NHCH ₂ (c-Hex)], [ZA4315; F, H, Cl, H , NHCH ₂ F], [ZA4316; F, H, Cl, H, NHCHF ₂ ], [ZA4317; F, H, Cl, H, NHCF ₃ ], [ZA4318; F, H, Cl, H, NH (CH ₂ ) ₂ F], [ZA4319; F, H, Cl, H, NHCH ₂ CHF ₂ ], [ZA4320; F, H, Cl, H, NHCH ₂ CHF ₃ ], [ZA4 321; F, H, Cl, H, NH (CH ₂ ) ₃ F], [ZA4322; F, H, Cl, H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA4323; F, H, Cl, H , NH (CH ₂ ) ₂ CF ₃ ], [ZA4324; F, H, Cl, H, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA4325; F, H, Cl, H, NHCH ₂ Cl], [ZA4326 ; F, H, Cl, H, NH (CH ₂ ) ₂ Cl], [ZA4327; F, H, Cl, H, NH (CH ₂ ) ₃ Cl], [ZA4328; F, H, Cl, H, NH (CH ₂ ) ₄ Cl], [ZA4329; F, H, Cl, H, NH (CH ₂ ) ₅ Cl], [ZA4330; F, H, Cl, H, NHCH ₂ OMe], [ZA4331; F, H , Cl, H, NH (CH ₂ ) ₂ OMe], [ZA4332; F, H, Cl, H, NH (CH ₂ ) ₃ OMe], [ZA4333; F, H, Cl, H, NH (CH ₂ ) ₄ OMe], [ZA4334; F, H, Cl, H, NHCH ₂ OEt], [ZA4335; F, H, Cl, H, NH (CH ₂ ) ₂ OEt], [ZA4336; F, H, Cl, H , NH (CH ₂ ) ₃ OEt], [ZA4337; F, H, Cl, H, NHCH ₂ OPr], [ZA4338; F, H, Cl, H, NH (CH ₂ ) ₂ OPr], [ZA4339; F , H, Cl, H, NH (CH ₂ ) ₃ OPr], [ZA4340; F, H, Cl, H, NHCH ₂ CN], [ZA4341; F, H, Cl, H, NH (CH ₂ ) ₂ CN ], [ZA4342; F, H, Cl, H, NH (CH ₂ ) ₃ CN], [ZA4343; F, H, Cl, H, NH (CH ₂ ) ₄ CN], [ZA4344; F, H, Cl , H, NH (CH ₂ ) ₅ CN], [ZA4345; F, H, Cl, H, NHCH ₂ CH = CH ₂ ], [ZA4346; F, H, Cl, H, NHCH ₂ C≡CH], [ ZA4347; F, H, Cl, H, NHCH ₂ C≡CCH ₃ ], [ZA4348; F, H, Cl, H, NHCH ₂ Ph], [ZA4349; F, H, Cl, H, NHCH ₂ (2- Py)], [ZA4350; F, H, Cl, H, NHCH ₂ (3-Py)], [ZA4351; F, H, Cl, H, NHCH ₂ (4-Py)], [ZA4352; F, H, Cl, H, NH (CH ₂ ) ₂ Ph], [ZA4353; F, H, Cl, H, NH (CH ₂ ) ₂ (2-Py) ], [ZA4354; F, H, Cl, H, NH (CH ₂ ) ₂ (3-Py)], [ZA4355; F, H, Cl, H, NH (CH ₂ ) ₂ (4-Py)], [ZA4356; F, H, Cl, H, NHPh], [ZA4357; F, H, Cl, H, NH (2-Py)], [ZA4358; F, H, Cl, H, NH (3-Py) ], [ZA4359; F, H, Cl, H, NH (4-Py)], [ZA4360; F, H, Cl, H, NMe ₂ ], [ZA4361; F, H, Cl, H, NMeEt], [ZA4362; F, H, Cl, H, NMePr], [ZA4363; F, H, Cl, H, NMeBu], [ZA4364; F, H, Cl, H, NMePen], [ZA4365; F, H, Cl , H, NMeHex], [ZA4366; F, H, Cl, H, NMe (i-Pr)], [ZA4367; F, H, Cl, H, NMe (i-Bu)], [ZA4368; F, H , Cl, H, NMe (c-Pr)], [ZA4369; F, H, Cl, H, NMe (c-Bu)], [ZA4370; F, H, Cl, H, NMe (c-Pen)] , [ZA4371; F, H, Cl, H, NMe (c-Hex)], [ZA4372; F, H, Cl, H, NMeCH ₂ (c-Pr)], [ZA4373; F, H, Cl, H , NMeCH ₂ (c-Bu)], [ZA4374; F, H, Cl, H, NMeCH ₂ (c-Pen)], [ZA4375; F, H, Cl, H, NMeCH ₂ (c-Hex)], [ZA4376; F, H, Cl, H, NMeCH ₂ F], [ZA4377; F, H, Cl, H, NMeCHF ₂ ], [ZA4378; F, H, Cl, H, NMeCF ₃ ], [ZA4379; F , H, Cl, H, NMe (CH ₂ ) ₂ F], [ZA4380; F, H, Cl, H, NMeCH ₂ CHF ₂ ], [ZA4381; F, H, Cl, H, NMeCH ₂ CHF ₃ ], [ZA4382; F, H, Cl, H, NMe (CH ₂ ) ₃ F], [ZA4383; F, H, Cl, H, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA4384; F, H, Cl, H, NMe (CH ₂ ) ₂ CF ₃ ], [ ZA4385; F, H, Cl, H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA4386; F, H, Cl, H, NMeCH ₂ Cl], [ZA4387; F, H, Cl, H, NMe (CH _{2) 2 Cl], [ZA4388} ; F, H, Cl, H, NMe (CH 2) 3 Cl], [ZA4389; F, H, Cl, H, NMe (CH 2) 4 Cl], [ZA4390; F , H, Cl, H, NMe (CH ₂ ) ₅ Cl], [ZA4391; F, H, Cl, H, NMeCH ₂ OMe], [ZA4392; F, H, Cl, H, NMe (CH ₂ ) ₂ OMe ], [ZA4393; F, H, Cl, H, NMe (CH ₂ ) ₃ OMe], [ZA4394; F, H, Cl, H, NMe (CH ₂ ) ₄ OMe], [ZA4395; F, H, Cl , H, NMeCH ₂ OEt], [ZA4396; F, H, Cl, H, NMe (CH ₂ ) ₂ OEt], [ZA4397; F, H, Cl, H, NMe (CH ₂ ) ₃ OEt], [ZA4398 ; F, H, Cl, H, NMeCH ₂ OPr], [ZA4399; F, H, Cl, H, NMe (CH ₂ ) ₂ OPr], [ZA4400; F, H, Cl, H, NMe (CH ₂ ) ₃ OPr], [ZA4401; F, H, Cl, H, NMeCH ₂ CN], [ZA4402; F, H, Cl, H, NMe (CH ₂ ) ₂ CN], [ZA4403; F, H, Cl, H , NMe (CH ₂ ) ₃ CN], [ZA4404; F, H, Cl, H, NMe (CH ₂ ) ₄ CN], [ZA4405; F, H, Cl, H, NMe (CH ₂ ) ₅ CN], [ZA4406; F, H, Cl, H, NMeCH ₂ CH = CH ₂ ], [ZA4407; F, H, Cl, H, NMeCH ₂ C≡CH], [ZA4408; F, H, Cl, H, NMeCH ₂ C≡CCH ₃ ], [ZA4409; F, H, Cl, H, NMeCH ₂ Ph], [ZA4410; F, H, Cl, H, NMeCH ₂ (2-Py)], [ZA4411; F, H, Cl , H, NMeCH ₂ (3-Py)], [ZA4412; F, H, Cl, H, NMeCH ₂ (4-Py)], [ZA4413; F, H, Cl, H, NMe (CH ₂ ) ₂ Ph ], [ZA4414; F, H, Cl, H, NMe (CH ₂ ) ₂ (2-Py)], [ZA4415; F, H, Cl, H, NMe (CH ₂ ) ₂ (3-Py)], [ZA4416; F, H, Cl, H, NMe (CH ₂ ) ₂ (4 -Py)], [ZA4417; F, H, Cl, H, NMePh], [ZA4418; F, H, Cl, H, NMe (2-Py)], [ZA4419; F, H, Cl, H, NMe (3-Py)], [ZA4420; F, H, Cl, H, NMe (4-Py)], [ZA4421; F, H, Cl, H, NEt ₂ ], [ZA4422; F, H, Cl, H, NEtPr], [ZA4423; F, H, Cl, H, NEtBu], [ZA4424; F, H, Cl, H, NEtPen], [ZA4425; F, H, Cl, H, NEtHex], [ZA4426; F, H, Cl, H, NEt (i-Pr)], [ZA4427; F, H, Cl, H, NEt (i-Bu)], [ZA4428; F, H, Cl, H, NEt (c- Pr)], [ZA4429; F, H, Cl, H, NEt (c-Bu)], [ZA4430; F, H, Cl, H, NEt (c-Pen)], [ZA4431; F, H, Cl , H, NEt (c-Hex)], [ZA4432; F, H, Cl, H, NEtCH ₂ (c-Pr)], [ZA4433; F, H, Cl, H, NEtCH ₂ (c-Bu)] , [ZA4434; F, H, Cl, H, NEtCH ₂ (c-Pen)], [ZA4435; F, H, Cl, H, NEtCH ₂ (c-Hex)], [ZA4436; F, H, Cl, H, NEtCH ₂ F], [ZA4437; F, H, Cl, H, NEtCHF ₂ ], [ZA4438; F, H, Cl, H, NEtCF ₃ ], [ZA4439; F, H, Cl, H, NEt ( CH ₂ ) ₂ F], [ZA4440; F, H, Cl, H, NEtCH ₂ CHF ₂ ], [ZA4441; F, H, Cl, H, NEtCH ₂ CHF ₃ ], [ZA4442; F, H, Cl, H, NEt (CH ₂ ) ₃ F], [ZA4443; F, H, Cl, H, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA4444; F, H, Cl, H, NEt (CH ₂ ) ₂ CF ₃ ], [ZA4445; F, H, Cl, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA4446; F, H, Cl, H, NEtCH ₂ Cl], [ZA4447; F, H, Cl, H , NEt (CH _{2) 2 Cl], [ZA4448} ; F, H, Cl, H, NEt (CH 2) 3 Cl], [ZA4449; F, H, Cl, H, NEt (CH 2) 4 Cl], [ZA4450; F , H, Cl, H, NEt (CH ₂ ) ₅ Cl], [ZA4451; F, H, Cl, H, NEtCH ₂ OMe], [ZA4452; F, H, Cl, H, NEt (CH ₂ ) ₂ OMe ], [ZA4453; F, H, Cl, H, NEt (CH ₂ ) ₃ OMe], [ZA4454; F, H, Cl, H, NEt (CH ₂ ) ₄ OMe], [ZA4455; F, H, Cl , H, NEtCH ₂ OEt], [ZA4456; F, H, Cl, H, NEt (CH ₂ ) ₂ OEt], [ZA4457; F, H, Cl, H, NEt (CH ₂ ) ₃ OEt], [ZA4458 ; F, H, Cl, H, NEtCH ₂ OPr], [ZA4459; F, H, Cl, H, NEt (CH ₂ ) ₂ OPr], [ZA4460; F, H, Cl, H, NEt (CH ₂ ) ₃ OPr], [ZA4461; F, H, Cl, H, NEtCH ₂ CN], [ZA4462; F, H, Cl, H, NEt (CH ₂ ) ₂ CN], [ZA4463; F, H, Cl, H , NEt (CH ₂ ) ₃ CN], [ZA4464; F, H, Cl, H, NEt (CH ₂ ) ₄ CN], [ZA4465; F, H, Cl, H, NEt (CH ₂ ) ₅ CN], [ZA4466; F, H, Cl, H, NEtCH ₂ CH = CH ₂ ], [ZA4467; F, H, Cl, H, NEtCH ₂ C≡CH], [ZA4468; F, H, Cl, H, NEtCH ₂ C≡CCH ₃ ], [ZA4469; F, H, Cl, H, NEtCH ₂ Ph], [ZA4470; F, H, Cl, H, NEtCH ₂ (2-Py)], [ZA4471; F, H, Cl , H, NEtCH ₂ (3-Py)], [ZA4472; F, H, Cl, H, NEtCH ₂ (4-Py)], [ZA4473; F, H, Cl, H, NEt (CH ₂ ) ₂ Ph ], [ZA4474; F, H, Cl, H, NEt (CH ₂ ) ₂ (2-Py)], [ZA4475; F, H, Cl, H, NEt (CH ₂ ) ₂ (3-Py)], [ZA4476; F, H, Cl, H, NEt (CH ₂ ) ₂ (4-Py)], [ZA447 7; F, H, Cl, H, NEtPh], [ZA4478; F, H, Cl, H, NEt (2-Py)], [ZA4479; F, H, Cl, H, NEt (3-Py)] , [ZA4480; F, H, Cl, H, NEt (4-Py)], [ZA4481; F, H, Cl, H, Pyr], [ZA4482; F, H, Cl, H, Pip], [ZA4483 ; F, H, Cl, H, Mor], [ZA4484; F, H, Cl, H, OMe], [ZA4485; F, H, Cl, H, OEt], [ZA4486; F, H, Cl, H , OPr], [ZA4487; F, H, Cl, H, OBu], [ZA4488; F, H, Cl, H, OPen], [ZA4489; F, H, Cl, H, OHex], [ZA4490; F , H, Cl, H, O (i-Pr)], [ZA4491; F, H, Cl, H, O (i-Bu)], [ZA4492; F, H, Cl, H, O (c-Pr )], [ZA4493; F, H, Cl, H, O (c-Bu)], [ZA4494; F, H, Cl, H, O (c-Pen)], [ZA4495; F, H, Cl, H, O (c-Hex)], [ZA4496; F, H, Cl, H, OCH ₂ (c-Pr)], [ZA
4497; F, H, Cl, H, OCH ₂ (c-Bu)], [ZA4498; F, H, Cl, H, OCH ₂ (c-Pen)], [ZA4499; F, H, Cl, H, OCH ₂ (c-Hex)], [ZA4500; F, H, Cl, H, OCH ₂ F],

[ZA4501; F, H, Cl, H, OCHF ₂ ], [ZA4502; F, H, Cl, H, OCF ₃ ], [ZA4503; F, H, Cl, H, O (CH ₂ ) ₂ F], [ZA4504; F, H, Cl, H, OCH ₂ CHF ₂ ], [ZA4505; F, H, Cl, H, OCH ₂ CHF ₃ ], [ZA4506; F, H, Cl, H, O (CH ₂ ) ₃ F], [ZA4507; F, H, Cl, H, O (CH ₂ ) ₂ CHF ₂ ], [ZA4508; F, H, Cl, H, O (CH ₂ ) ₂ CF ₃ ], [ZA4509; F , H, Cl, H, OCH ₂ CH (CF ₃ ) ₂ ], [ZA4510; F, H, Cl, H, OCH ₂ Cl], [ZA4511; F, H, Cl, H, O (CH ₂ ) ₂ Cl], [ZA4512; F, H, Cl, H, O (CH ₂ ) ₃ Cl], [ZA4513; F, H, Cl, H, O (CH ₂ ) ₄ Cl], [ZA4514; F, H, Cl, H, O (CH ₂ ) ₅ Cl], [ZA4515; F, H, Cl, H, OCH ₂ OMe], [ZA4516; F, H, Cl, H, O (CH ₂ ) ₂ OMe], [ ZA4517; F, H, Cl, H, O (CH ₂ ) ₃ OMe], [ZA4518; F, H, Cl, H, O (CH ₂ ) ₄ OMe], [ZA4519; F, H, Cl, H, OCH ₂ OEt], [ZA4520; F, H, Cl, H, O (CH ₂ ) ₂ OEt], [ZA4521; F, H, Cl, H, O (CH ₂ ) ₃ OEt], [ZA4522; F, H, Cl, H, OCH ₂ OPr], [ZA4523; F, H, Cl, H, O (CH ₂ ) ₂ OPr], [ZA4524; F, H, Cl, H, O (CH ₂ ) ₃ OPr] , [ZA4525; F, H, Cl, H, OCH ₂ CN], [ZA4526; F, H, Cl, H, O (CH ₂ ) ₂ CN], [ZA4527; F, H, Cl, H, O ( _{CH 2) 3 CN], [} ZA4528; F, H, Cl, H, O (CH 2) 4 CN], [ZA4529; F, H, Cl, H, O (CH 2) 5 CN], [ZA4530; F, H, Cl, H, OCH ₂ CH = CH ₂ ], [ZA4531; F, H, Cl, H, OCH ₂ C≡CH], [ZA4532; F, H, Cl, H, OCH ₂ C≡C CH ₃ ], [ZA4533; F, H, Cl, H, OCH ₂ Ph], [ZA4534; F, H, Cl, H, OCH ₂ (2-Py)], [ZA4535; F, H, Cl, H , OCH ₂ (3-Py)], [ZA4536; F, H, Cl, H, OCH ₂ (4-Py)], [ZA4537; F, H, Cl, H, O (CH ₂ ) ₂ Ph], [ZA4538; F, H, Cl, H, O (CH ₂ ) ₂ (2-Py)], [ZA4539; F, H, Cl, H, O (CH ₂ ) ₂ (3-Py)], [ZA4540 ; F, H, Cl, H, O (CH ₂ ) ₂ (4-Py)], [ZA4541; F, H, Cl, H, OPh], [ZA4542; F, H, Cl, H, O (2 -Py)], [ZA4543; F, H, Cl, H, O (3-Py)], [ZA4544; F, H, Cl, H, O (4-Py)], [ZA4545; F, H, Cl, H, Me], [ZA4546; F, H, Cl, H, Et], [ZA4547; F, H, Cl, H, Pr], [ZA4548; F, H, Cl, H, Bu], [ ZA4549; F, H, Cl, H, Pen], [ZA4550; F, H, Cl, H, Hex], [ZA4551; F, H, Cl, H, (i-Pr)], [ZA4552; F, H, Cl, H, (i-Bu)], [ZA4553; F, H, Cl, H, (c-Pr)], [ZA4554; F, H, Cl, H, (c-Bu)], [ ZA4555; F, H, Cl, H, (c-Pen)], [ZA4556; F, H, Cl, H, (c-Hex)], [ZA4557; F, H, Cl, H, CH ₂ (c -Pr)], [ZA4558; F, H, Cl, H, CH ₂ (c-Bu)], [ZA4559; F, H, Cl, H, CH ₂ (c-Pen)], [ZA4560; F, H, Cl, H, CH ₂ (c-Hex)], [ZA4561; F, H, Cl, H, CH ₂ F], [ZA4562; F, H, Cl, H, CHF ₂ ], [ZA4563; F , H, Cl, H, CF ₃ ], [ZA4564; F, H, Cl, H, (CH ₂ ) ₂ F], [ZA4565; F, H, Cl, H, CH ₂ CHF ₂ ], [ZA4566; F, H, Cl, H, CH ₂ CHF ₃ ], [ZA4567; F, H, Cl, H, (CH ₂ ) ₃ F], [ZA4568; F, H, Cl, H, (CH ₂ ) ₂ CHF ₂ ], [Z A4569; F, H, Cl, H, (CH ₂ ) ₂ CF ₃ ], [ZA4570; F, H, Cl, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA4571; F, H, Cl, H , CH ₂ Cl], [ZA4572; F, H, Cl, H, (CH ₂ ) ₂ Cl], [ZA4573; F, H, Cl, H, (CH ₂ ) ₃ Cl], [ZA4574; F, H , Cl, H, (CH ₂ ) ₄ Cl], [ZA4575; F, H, Cl, H, (CH ₂ ) ₅ Cl], [ZA4576; F, H, Cl, H, CH ₂ OMe], [ZA4577 ; F, H, Cl, H, (CH ₂ ) ₂ OMe], [ZA4578; F, H, Cl, H, (CH ₂ ) ₃ OMe], [ZA4579; F, H, Cl, H, (CH ₂ ) ₄ OMe], [ZA4580; F, H, Cl, H, CH ₂ OEt], [ZA4581; F, H, Cl, H, (CH ₂ ) ₂ OEt], [ZA4582; F, H, Cl, H , (CH ₂ ) ₃ OEt], [ZA4583; F, H, Cl, H, CH ₂ OPr], [ZA4584; F, H, Cl, H, (CH ₂ ) ₂ OPr], [ZA4585; F, H , Cl, H, (CH ₂ ) ₃ OPr], [ZA4586; F, H, Cl, H, CH ₂ CN], [ZA4587; F, H, Cl, H, (CH ₂ ) ₂ CN], [ZA4588 ; F, H, Cl, H, (CH ₂ ) ₃ CN], [ZA4589; F, H, Cl, H, (CH ₂ ) ₄ CN], [ZA4590; F, H, Cl, H, (CH ₂ ) ₅ CN], [ZA4591; F, H, Cl, H, CH ₂ CH = CH ₂ ], [ZA4592; F, H, Cl, H, CH ₂ C≡CH], [ZA4593; F, H, Cl , H, CH ₂ C≡CCH ₃ ], [ZA4594; F, H, Cl, H, CH ₂ Ph], [ZA4595; F, H, Cl, H, CH ₂ (2-Py)], [ZA4596; F, H, Cl, H, CH ₂ (3-Py)], [ZA4597; F, H, Cl, H, CH ₂ (4-Py)], [ZA4598; F, H, Cl, H, (CH ₂ ) ₂ Ph], [ZA4599; F, H, Cl, H, (CH ₂ ) ₂ (2-Py)], [ZA4600; F, H, Cl, H, (CH ₂ ) ₂ (3-Py) ], [ZA4601; F, H, Cl , H, (CH ₂ ) ₂ (4-Py)], [ZA4602; F, H, Cl, H, Ph], [ZA4603; F, H, Cl, H, 2-Py], [ZA4604; F, H, Cl, H, 3-Py], [ZA4605; F, H, Cl, H, 4-Py], [ZA4606; F, H, Cl, Cl, NHMe], [ZA4607; F, H, Cl, Cl, NHEt], [ZA4608; F, H, Cl, Cl, NHPr], [ZA4609; F, H, Cl, Cl, NHBu], [ZA4610; F, H, Cl, Cl, NHPen], [ZA4611; F, H, Cl, Cl, NHHex], [ZA4612; F, H, Cl, Cl, NH (i-Pr)], [ZA4613; F, H, Cl, Cl, NH (i-Bu)], [ ZA4614; F, H, Cl, Cl, NH (c-Pr)], [ZA4615; F, H, Cl, Cl, NH (c-Bu)], [ZA4616; F, H, Cl, Cl, NH ( c-Pen)], [ZA4617; F, H, Cl, Cl, NH (c-Hex)], [ZA4618; F, H, Cl, Cl, NHCH ₂ (c-Pr)], [ZA4619; F, H, Cl, Cl, NHCH ₂ (c-Bu)], [ZA4620; F, H, Cl, Cl, NHCH ₂ (c-Pen)], [ZA4621; F, H, Cl, Cl, NHCH ₂ (c -Hex)], [ZA4622; F, H, Cl, Cl, NHCH ₂ F], [ZA4623; F, H, Cl, Cl, NHCHF ₂ ], [ZA4624; F, H, Cl, Cl, NHCF ₃ ] , [ZA4625; F, H, Cl, Cl, NH (CH ₂ ) ₂ F], [ZA4626; F, H, Cl, Cl, NHCH ₂ CHF ₂ ], [ZA4627; F, H, Cl, Cl, NHCH ₂ CHF ₃ ], [ZA4628; F, H, Cl, Cl, NH (CH ₂ ) ₃ F], [ZA4629; F, H, Cl, Cl, NH (CH ₂ ) ₂ CHF ₂ ], [ZA4630; F , H, Cl, Cl, NH (CH ₂ ) ₂ CF ₃ ], [ZA4631; F, H, Cl, Cl, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA4632; F, H, Cl, Cl, NHCH ₂ Cl], [ZA4633; F, H, Cl, Cl, NH (CH ₂ ) ₂ Cl], [ZA4634; F, H, Cl, Cl, NH (CH ₂ ) ₃ Cl], [ZA4635; F, H , C l, Cl, NH (CH ₂ ) ₄ Cl], [ZA4636; F, H, Cl, Cl, NH (CH ₂ ) ₅ Cl], [ZA4637; F, H, Cl, Cl, NHCH ₂ OMe], [ ZA4638; F, H, Cl, Cl, NH (CH ₂ ) ₂ OMe], [ZA4639; F, H, Cl, Cl, NH (CH ₂ ) ₃ OMe], [ZA4640; F, H, Cl, Cl, NH (CH ₂ ) ₄ OMe], [ZA4641; F, H, Cl, Cl, NHCH ₂ OEt], [ZA4642; F, H, Cl, Cl, NH (CH ₂ ) ₂ OEt], [ZA4643; F, H, Cl, Cl, NH (CH ₂ ) ₃ OEt], [ZA4644; F, H, Cl, Cl, NHCH ₂ OPr], [ZA4645; F, H, Cl, Cl, NH (CH ₂ ) ₂ OPr] , [ZA4646; F, H, Cl, Cl, NH (CH ₂ ) ₃ OPr], [ZA4647; F, H, Cl, Cl, NHCH ₂ CN], [ZA4648; F, H, Cl, Cl, NH ( _{CH 2) 2 CN], [} ZA4649; F, H, Cl, Cl, NH (CH 2) 3 CN], [ZA4650; F, H, Cl, Cl, NH (CH 2) 4 CN], [ZA4651; F, H, Cl, Cl, NH (CH ₂ ) ₅ CN], [ZA4652; F, H, Cl, Cl, NHCH ₂ CH = CH ₂ ], [ZA4653; F, H, Cl, Cl, NHCH ₂ C ≡CH], [ZA4654; F, H, Cl, Cl, NHCH ₂ C≡CCH ₃ ], [ZA4655; F, H, Cl, Cl, NHCH ₂ Ph], [ZA4656; F, H, Cl, Cl, NHCH ₂ (2-Py)], [ZA4657; F, H, Cl, Cl, NHCH ₂ (3-Py)], [ZA4658; F, H, Cl, Cl, NHCH ₂ (4-Py)], [ ZA4659; F, H, Cl, Cl, NH (CH ₂ ) ₂ Ph], [ZA4660; F, H, Cl, Cl, NH (CH ₂ ) ₂ (2-Py)], [ZA4661; F, H, Cl, Cl, NH (CH ₂ ) ₂ (3-Py)], [ZA4662; F, H, Cl, Cl, NH (CH ₂ ) ₂ (4-Py)], [ZA4663; F, H, Cl, Cl, NHPh], [ZA4664; F, H, Cl, Cl, NH (2-Py)], [ZA4665; F, H, Cl, Cl, NH (3-Py)], [ZA4666; F, H, Cl, Cl, NH (4-Py)], [ZA4667; F, H, Cl, Cl, NMe ₂ ], [ZA4668; F , H, Cl, Cl, NMeEt], [ZA4669; F, H, Cl, Cl, NMePr], [ZA4670; F, H, Cl, Cl, NMeBu], [ZA4671; F, H, Cl, Cl, NMePen ], [ZA4672; F, H, Cl, Cl, NMeHex], [ZA4673; F, H, Cl, Cl, NMe (i-Pr)], [ZA4674; F, H, Cl, Cl, NMe (i- Bu)], [ZA4675; F, H, Cl, Cl, NMe (c-Pr)], [ZA4676; F, H, Cl, Cl, NMe (c-Bu)], [ZA4677; F, H, Cl , Cl, NMe (c-Pen)], [ZA4678; F, H, Cl, Cl, NMe (c-Hex)], [ZA4679; F, H, Cl, Cl, NMeCH ₂ (c-Pr)], [ZA4680; F, H, Cl, Cl, NMeCH ₂ (c-Bu)], [ZA4681; F, H, Cl, Cl, NMeCH ₂ (c-Pen)], [ZA4682; F, H, Cl, Cl , NMeCH ₂ (c-Hex)], [ZA4683; F, H, Cl, Cl, NMeCH ₂ F], [ZA4684; F, H, Cl, Cl, NMeCHF ₂ ], [ZA4685; F, H, Cl, Cl, NMeCF ₃ ], [ZA4686; F, H, Cl, Cl, NMe (CH ₂ ) ₂ F], [ZA4687; F, H, Cl, Cl, NMeCH ₂ CHF ₂ ], [ZA4688; F, H, Cl, Cl, NMeCH ₂ CHF ₃ ], [ZA4689; F, H, Cl, Cl, NMe (CH ₂ ) ₃ F], [ZA4690; F, H, Cl, Cl, NMe (CH ₂ ) ₂ CHF ₂ ] , [ZA4691; F, H, Cl, Cl, NMe (CH ₂ ) ₂ CF ₃ ], [ZA4692; F, H, Cl, Cl, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA4693; F, H, Cl, Cl, NMeCH ₂ Cl], [ZA4694; F, H, Cl, Cl, NMe (CH ₂ ) ₂ Cl], [ZA4695; F, H, Cl, Cl, NMe (CH ₂ ) ₃ Cl], [ ZA4696; F, H, Cl, Cl, NMe (CH ₂ ) ₄ Cl], [ZA4697; F, H, Cl, Cl, NMe (CH ₂ ) ₅ Cl], [ZA4698; F, H, Cl, Cl, NMeCH ₂ OMe], [ZA4699; F, H, Cl, Cl, NMe (CH ₂ ) ₂ OMe], [ZA4700; F, H, Cl, Cl, NMe (CH ₂ ) ₃ OMe], [ZA4701; F, H, Cl, Cl, NMe (CH ₂ ) ₄ OMe], [ZA4702; F, H, Cl, Cl, NMeCH ₂ OEt], [ZA4703; F, H, Cl, Cl, NMe (CH ₂ ) ₂ OEt], [ZA4704; F, H, Cl, Cl, NMe (CH ₂ ) ₃ OEt], [ZA4705; F, H, Cl, Cl, NMeCH ₂ OPr], [ZA4706; F, H, Cl, Cl, NMe (CH ₂ ) ₂ OPr], [ZA4707; F, H, Cl, Cl, NMe (CH ₂ ) ₃ OPr], [ ZA4708; F, H, Cl, Cl, NMeCH ₂ CN], [ZA4709; F, H, Cl, Cl, NMe (CH ₂ ) ₂ CN], [ZA4710; F, H, Cl, Cl, NMe (CH ₂ ) ₃ CN], [ZA4711; F, H, Cl, Cl, NMe (CH ₂ ) ₄ CN], [ZA4712; F, H, Cl, Cl, NMe (CH ₂ ) ₅ CN], [ZA4713; F, H, Cl, Cl, NMeCH ₂ CH = CH ₂ ], [ZA4714; F, H, Cl, Cl, NMeCH ₂ C≡CH], [ZA4715; F, H, Cl, Cl, NMeCH ₂ C≡CCH ₃ ] , [ZA4716; F, H, Cl, Cl, NMeCH ₂ Ph], [ZA4717; F, H, Cl, Cl, NMeCH ₂ (2-Py)], [ZA4718; F, H, Cl, Cl, NMeCH ₂ (3-Py)], [ZA4719; F, H, Cl, Cl, NMeCH ₂ (4-Py)], [ZA4720; F, H, Cl, Cl, NMe (CH ₂ ) ₂ Ph], [ZA4721; F, H, Cl, Cl, NMe (CH ₂ ) ₂ (2-Py)], [ZA4722; F, H, Cl, Cl, NMe (CH ₂ ) ₂ (3-Py)], [ZA4723; F, H, Cl, Cl, NMe (CH ₂ ) ₂ (4-Py)], [ZA4724; F, H, Cl, Cl, NMePh], [ZA4725; F, H, Cl, Cl, NMe (2-Py) ], [ZA4726; F, H, Cl, Cl, N Me (3-Py)], [ZA4727; F, H, Cl, Cl, NMe (4-Py)], [ZA4728; F, H, Cl, Cl, NEt ₂ ], [ZA4729; F, H, Cl , Cl, NEtPr], [ZA4730; F, H, Cl, Cl, NEtBu], [ZA4731; F, H, Cl, Cl, NEtPen], [ZA4732; F, H, Cl, Cl, NEtHex], [ZA4733 ; F, H, Cl, Cl, NEt (i-Pr)], [ZA4734; F, H, Cl, Cl, NEt (i-Bu)], [ZA4735; F, H, Cl, Cl, NEt (c -Pr)], [ZA4736; F, H, Cl, Cl, NEt (c-Bu)], [ZA4737; F, H, Cl, Cl, NEt (c-Pen)], [ZA4738; F, H, Cl, Cl, NEt (c-Hex)], [ZA4739; F, H, Cl, Cl, NEtCH ₂ (c-Pr)], [ZA4740; F, H, Cl, Cl, NEtCH ₂ (c-Bu) ], [ZA4741; F, H, Cl, Cl, NEtCH ₂ (c-Pen)], [ZA4742; F, H, Cl, Cl, NEtCH ₂ (c-Hex)], [ZA4743; F, H, Cl , Cl, NEtC
H ₂ F], [ZA4744; F, H, Cl, Cl, NEtCHF ₂ ], [ZA4745; F, H, Cl, Cl, NEtCF ₃ ], [ZA4746; F, H, Cl, Cl, NEt (CH ₂ ) ₂ F], [ZA4747; F, H, Cl, Cl, NEtCH ₂ CHF ₂ ], [ZA4748; F, H, Cl, Cl, NEtCH ₂ CHF ₃ ], [ZA4749; F, H, Cl, Cl, NEt (CH ₂ ) ₃ F], [ZA4750; F, H, Cl, Cl, NEt (CH ₂ ) ₂ CHF ₂ ],

[ZA4751; F, H, Cl, Cl, NEt (CH ₂ ) ₂ CF ₃ ], [ZA4752; F, H, Cl, Cl, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA4753; F, H, Cl , Cl, NEtCH ₂ Cl], [ZA4754; F, H, Cl, Cl, NEt (CH ₂ ) ₂ Cl], [ZA4755; F, H, Cl, Cl, NEt (CH ₂ ) ₃ Cl], [ZA4756 ; F, H, Cl, Cl, NEt (CH ₂ ) ₄ Cl], [ZA4757; F, H, Cl, Cl, NEt (CH ₂ ) ₅ Cl], [ZA4758; F, H, Cl, Cl, NEtCH ₂ OMe], [ZA4759; F, H, Cl, Cl, NEt (CH ₂ ) ₂ OMe], [ZA4760; F, H, Cl, Cl, NEt (CH ₂ ) ₃ OMe], [ZA4761; F, H , Cl, Cl, NEt (CH ₂ ) ₄ OMe], [ZA4762; F, H, Cl, Cl, NEtCH ₂ OEt], [ZA4763; F, H, Cl, Cl, NEt (CH ₂ ) ₂ OEt], [ZA4764; F, H, Cl, Cl, NEt (CH ₂ ) ₃ OEt], [ZA4765; F, H, Cl, Cl, NEtCH ₂ OPr], [ZA4766; F, H, Cl, Cl, NEt (CH ₂ ) ₂ OPr], [ZA4767; F, H, Cl, Cl, NEt (CH ₂ ) ₃ OPr], [ZA4768; F, H, Cl, Cl, NEtCH ₂ CN], [ZA4769; F, H, Cl , Cl, NEt (CH ₂ ) ₂ CN], [ZA4770; F, H, Cl, Cl, NEt (CH ₂ ) ₃ CN], [ZA4771; F, H, Cl, Cl, NEt (CH ₂ ) ₄ CN ], [ZA4772; F, H, Cl, Cl, NEt (CH ₂ ) ₅ CN], [ZA4773; F, H, Cl, Cl, NEtCH ₂ CH = CH ₂ ], [ZA4774; F, H, Cl, Cl, NEtCH ₂ C≡CH], [ZA4775; F, H, Cl, Cl, NEtCH ₂ C≡CCH ₃ ], [ZA4776; F, H, Cl, Cl, NEtCH ₂ Ph], [ZA4777; F, H , Cl, Cl, NEtCH ₂ (2-Py)], [ZA4778; F, H, Cl, Cl, NEtCH ₂ (3-Py)], [ZA4779; F, H, Cl, Cl, NEtCH ₂ (4- Py )], [ZA4780; F, H, Cl, Cl, NEt (CH ₂ ) ₂ Ph], [ZA4781; F, H, Cl, Cl, NEt (CH ₂ ) ₂ (2-Py)], [ZA4782; F, H, Cl, Cl, NEt (CH ₂ ) ₂ (3-Py)], [ZA4783; F, H, Cl, Cl, NEt (CH ₂ ) ₂ (4-Py)], [ZA4784; F, H, Cl, Cl, NEtPh], [ZA4785; F, H, Cl, Cl, NEt (2-Py)], [ZA4786; F, H, Cl, Cl, NEt (3-Py)], [ZA4787; F, H, Cl, Cl, NEt (4-Py)], [ZA4788; F, H, Cl, Cl, Pyr], [ZA4789; F, H, Cl, Cl, Pip], [ZA4790; F, H , Cl, Cl, Mor], [ZA4791; F, H, Cl, Cl, OMe], [ZA4792; F, H, Cl, Cl, OEt], [ZA4793; F, H, Cl, Cl, OPr], [ZA4794; F, H, Cl, Cl, OBu], [ZA4795; F, H, Cl, Cl, OPen], [ZA4796; F, H, Cl, Cl, OHex], [ZA4797; F, H, Cl , Cl, O (i-Pr)], [ZA4798; F, H, Cl, Cl, O (i-Bu)], [ZA4799; F, H, Cl, Cl, O (c-Pr)], [ ZA4800; F, H, Cl, Cl, O (c-Bu)], [ZA4801; F, H, Cl, Cl, O (c-Pen)], [ZA4802; F, H, Cl, Cl, O ( c-Hex)], [ZA4803; F, H, Cl, Cl, OCH ₂ (c-Pr)], [ZA4804; F, H, Cl, Cl, OCH ₂ (c-Bu)], [ZA4805; F , H, Cl, Cl, OCH ₂ (c-Pen)], [ZA4806; F, H, Cl, Cl, OCH ₂ (c-Hex)], [ZA4807; F, H, Cl, Cl, OCH ₂ F ], [ZA4808; F, H, Cl, Cl, OCHF ₂ ], [ZA4809; F, H, Cl, Cl, OCF ₃ ], [ZA4810; F, H, Cl, Cl, O (CH ₂ ) ₂ F ], [ZA4811; F, H, Cl, Cl, OCH ₂ CHF ₂ ], [ZA4812; F, H, Cl, Cl, OCH ₂ CHF ₃ ], [ZA4813; F, H, Cl, Cl, O (CH ₂ ) ₃ F], [ZA4814; F, H, Cl, Cl, O (CH ₂ ) ₂ CHF ₂ ], [ZA4815; F, H, Cl, Cl, O (CH ₂ ) ₂ CF ₃ ], [ZA4816; F, H, Cl, Cl, OCH ₂ CH (CF ₃ ) ₂ ], [ ZA4817; F, H, Cl, Cl, OCH ₂ Cl], [ZA4818; F, H, Cl, Cl, O (CH ₂ ) ₂ Cl], [ZA4819; F, H, Cl, Cl, O (CH _{2 ) 3 Cl], [ZA4820;} F, H, Cl, Cl, O (CH 2) 4 Cl], [ZA4821; F, H, Cl, Cl, O (CH 2) 5 Cl], [ZA4822; F, H, Cl, Cl, OCH ₂ OMe], [ZA4823; F, H, Cl, Cl, O (CH ₂ ) ₂ OMe], [ZA4824; F, H, Cl, Cl, O (CH ₂ ) ₃ OMe] , [ZA4825; F, H, Cl, Cl, O (CH ₂ ) ₄ OMe], [ZA4826; F, H, Cl, Cl, OCH ₂ OEt], [ZA4827; F, H, Cl, Cl, O ( CH ₂ ) ₂ OEt], [ZA4828; F, H, Cl, Cl, O (CH ₂ ) ₃ OEt], [ZA4829; F, H, Cl, Cl, OCH ₂ OPr], [ZA4830; F, H, Cl, Cl, O (CH ₂ ) ₂ OPr], [ZA4831; F, H, Cl, Cl, O (CH ₂ ) ₃ OPr], [ZA4832; F, H, Cl, Cl, OCH ₂ CN], [ ZA4833; F, H, Cl, Cl, O (CH ₂ ) ₂ CN], [ZA4834; F, H, Cl, Cl, O (CH ₂ ) ₃ CN], [ZA4835; F, H, Cl, Cl, O (CH ₂ ) ₄ CN], [ZA4836; F, H, Cl, Cl, O (CH ₂ ) ₅ CN], [ZA4837; F, H, Cl, Cl, OCH ₂ CH = CH ₂ ], [ZA4838 ; F, H, Cl, Cl, OCH ₂ C≡CH], [ZA4839; F, H, Cl, Cl, OCH ₂ C≡CCH ₃ ], [ZA4840; F, H, Cl, Cl, OCH ₂ Ph] , [ZA4841; F, H, Cl, Cl, OCH ₂ (2-Py)], [ZA4842; F, H, Cl, Cl, OCH ₂ (3-Py)], [ZA4843; F, H, Cl, Cl, OCH ₂ (4-Py)], [ZA4844; F, H, Cl, Cl, O (CH ₂ ) ₂ Ph], [ZA4845 ; F, H, Cl, Cl, O (CH ₂ ) ₂ (2-Py)], [ZA4846; F, H, Cl, Cl, O (CH ₂ ) ₂ (3-Py)], [ZA4847; F , H, Cl, Cl, O (CH ₂ ) ₂ (4-Py)], [ZA4848; F, H, Cl, Cl, OPh], [ZA4849; F, H, Cl, Cl, O (2-Py )], [ZA4850; F, H, Cl, Cl, O (3-Py)], [ZA4851; F, H, Cl, Cl, O (4-Py)], [ZA4852; F, H, Cl, Cl, Me], [ZA4853; F, H, Cl, Cl, Et], [ZA4854; F, H, Cl, Cl, Pr], [ZA4855; F, H, Cl, Cl, Bu], [ZA4856; F, H, Cl, Cl, Pen], [ZA4857; F, H, Cl, Cl, Hex], [ZA4858; F, H, Cl, Cl, (i-Pr)], [ZA4859; F, H, Cl, Cl, (i-Bu)], [ZA4860; F, H, Cl, Cl, (c-Pr)], [ZA4861; F, H, Cl, Cl, (c-Bu)], [ZA4862; F, H, Cl, Cl, (c-Pen)], [ZA4863; F, H, Cl, Cl, (c-Hex)], [ZA4864; F, H, Cl, Cl, CH ₂ (c-Pr )], [ZA4865; F, H, Cl, Cl, CH ₂ (c-Bu)], [ZA4866; F, H, Cl, Cl, CH ₂ (c-Pen)], [ZA4867; F, H, Cl, Cl, CH ₂ (c-Hex)], [ZA4868; F, H, Cl, Cl, CH ₂ F], [ZA4869; F, H, Cl, Cl, CHF ₂ ], [ZA4870; F, H , Cl, Cl, CF ₃ ], [ZA4871; F, H, Cl, Cl, (CH ₂ ) ₂ F], [ZA4872; F, H, Cl, Cl, CH ₂ CHF ₂ ], [ZA4873; F, H, Cl, Cl, CH ₂ CHF ₃ ], [ZA4874; F, H, Cl, Cl, (CH ₂ ) ₃ F], [ZA4875; F, H, Cl, Cl, (CH ₂ ) ₂ CHF ₂ ] , [ZA4876; F, H, Cl, Cl, (CH ₂ ) ₂ CF ₃ ], [ZA4877; F, H, Cl, Cl, CH ₂ CH (CF ₃ ) ₂ ], [ZA4878; F, H, Cl , Cl, CH ₂ Cl], [ZA4879; F, H, Cl, Cl, (CH ₂ ) ₂ Cl], [ZA488 0; F, H, Cl, Cl, (CH ₂ ) ₃ Cl], [ZA4881; F, H, Cl, Cl, (CH ₂ ) ₄ Cl], [ZA4882; F, H, Cl, Cl, (CH ₂ ) ₅ Cl], [ZA4883; F, H, Cl, Cl, CH ₂ OMe], [ZA4884; F, H, Cl, Cl, (CH ₂ ) ₂ OMe], [ZA4885; F, H, Cl, Cl, (CH ₂ ) ₃ OMe], [ZA4886; F, H, Cl, Cl, (CH ₂ ) ₄ OMe], [ZA4887; F, H, Cl, Cl, CH ₂ OEt], [ZA4888; F, H, Cl, Cl, (CH ₂ ) ₂ OEt], [ZA4889; F, H, Cl, Cl, (CH ₂ ) ₃ OEt], [ZA4890; F, H, Cl, Cl, CH ₂ OPr], [ ZA4891; F, H, Cl, Cl, (CH ₂ ) ₂ OPr], [ZA4892; F, H, Cl, Cl, (CH ₂ ) ₃ OPr], [ZA4893; F, H, Cl, Cl, CH ₂ CN], [ZA4894; F, H, Cl, Cl, (CH ₂ ) ₂ CN], [ZA4895; F, H, Cl, Cl, (CH ₂ ) ₃ CN], [ZA4896; F, H, Cl, Cl, (CH ₂ ) ₄ CN], [ZA4897; F, H, Cl, Cl, (CH ₂ ) ₅ CN], [ZA4898; F, H, Cl, Cl, CH ₂ CH = CH ₂ ], [ZA4899 ; F, H, Cl, Cl, CH ₂ C≡CH], [ZA4900; F, H, Cl, Cl, CH ₂ C≡CCH ₃ ], [ZA4901; F, H, Cl, Cl, CH ₂ Ph] , [ZA4902; F, H, Cl, Cl, CH ₂ (2-Py)], [ZA4903; F, H, Cl, Cl, CH ₂ (3-Py)], [ZA4904; F, H, Cl, Cl, CH ₂ (4-Py)], [ZA4905; F, H, Cl, Cl, (CH ₂ ) ₂ Ph], [ZA4906; F, H, Cl, Cl, (CH ₂ ) ₂ (2-Py )], [ZA4907; F, H, Cl, Cl, (CH ₂ ) ₂ (3-Py)], [ZA4908; F, H, Cl, Cl, (CH ₂ ) ₂ (4-Py)], [ ZA4909; F, H, Cl, Cl, Ph], [ZA4910; F, H, Cl, Cl, 2-Py], [ZA4911; F, H, Cl, Cl, 3-Py], [ZA4912; F, H , Cl, Cl, 4-Py], [ZA4913; F, H, Et, H, NHMe], [ZA4914; F, H, Et, H, NHEt], [ZA4915; F, H, Et, H, NHPr ], [ZA4916; F, H, Et, H, NHBu], [ZA4917; F, H, Et, H, NHPen], [ZA4918; F, H, Et, H, NHHex], [ZA4919; F, H , Et, H, NH (i-Pr)], [ZA4920; F, H, Et, H, NH (i-Bu)], [ZA4921; F, H, Et, H, NH (c-Pr)] , [ZA4922; F, H, Et, H, NH (c-Bu)], [ZA4923; F, H, Et, H, NH (c-Pen)], [ZA4924; F, H, Et, H, NH (c-Hex)], [ZA4925; F, H, Et, H, NHCH ₂ (c-Pr)], [ZA4926; F, H, Et, H, NHCH ₂ (c-Bu)], [ZA4927 ; F, H, Et, H, NHCH ₂ (c-Pen)], [ZA4928; F, H, Et, H, NHCH ₂ (c-Hex)], [ZA4929; F, H, Et, H, NHCH ₂ F], [ZA4930; F, H, Et, H, NHCHF ₂ ], [ZA4931; F, H, Et, H, NHCF ₃ ], [ZA4932; F, H, Et, H, NH (CH ₂ ) ₂ F], [ZA4933; F, H, Et, H, NHCH ₂ CHF ₂ ], [ZA4934; F, H, Et, H, NHCH ₂ CHF ₃ ], [ZA4935; F, H, Et, H, NH (CH ₂ ) ₃ F], [ZA4936; F, H, Et, H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA4937; F, H, Et, H, NH (CH ₂ ) ₂ CF ₃ ], [ZA4938; F, H, Et, H, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA4939; F, H, Et, H, NHCH ₂ Cl], [ZA4940; F, H, Et, H, NH ( _{CH 2) 2 Cl], [} ZA4941; F, H, Et, H, NH (CH 2) 3 Cl], [ZA4942; F, H, Et, H, NH (CH 2) 4 Cl], [ZA4943; F, H, Et, H, NH (CH ₂ ) ₅ Cl], [ZA4944; F, H, Et, H, NHCH ₂ OMe], [ZA4945; F, H, Et, H, NH (CH ₂ ) ₂ OMe], [ZA4946; F, H , Et, H, NH (CH ₂ ) ₃ OMe], [ZA4947; F, H, Et, H, NH (CH ₂ ) ₄ OMe], [ZA4948; F, H, Et, H, NHCH ₂ OEt], [ZA4949; F, H, Et, H, NH (CH ₂ ) ₂ OEt], [ZA4950; F, H, Et, H, NH (CH ₂ ) ₃ OEt], [ZA4951; F, H, Et, H , NHCH ₂ OPr], [ZA4952; F, H, Et, H, NH (CH ₂ ) ₂ OPr], [ZA4953; F, H, Et, H, NH (CH ₂ ) ₃ OPr], [ZA4954; F , H, Et, H, NHCH ₂ CN], [ZA4955; F, H, Et, H, NH (CH ₂ ) ₂ CN], [ZA4956; F, H, Et, H, NH (CH ₂ ) ₃ CN ], [ZA4957; F, H, Et, H, NH (CH ₂ ) ₄ CN], [ZA4958; F, H, Et, H, NH (CH ₂ ) ₅ CN], [ZA4959; F, H, Et , H, NHCH ₂ CH = CH ₂ ], [ZA4960; F, H, Et, H, NHCH ₂ C≡CH], [ZA4961; F, H, Et, H, NHCH ₂ C≡CCH ₃ ], [ZA4962 ; F, H, Et, H, NHCH ₂ Ph], [ZA4963; F, H, Et, H, NHCH ₂ (2-Py)], [ZA4964; F, H, Et, H, NHCH ₂ (3- Py)], [ZA4965; F, H, Et, H, NHCH ₂ (4-Py)], [ZA4966; F, H, Et, H, NH (CH ₂ ) ₂ Ph], [ZA4967; F, H , Et, H, NH (CH ₂ ) ₂ (2-Py)], [ZA4968; F, H, Et, H, NH (CH ₂ ) ₂ (3-Py)], [ZA4969; F, H, Et , H, NH (CH ₂ ) ₂ (4-Py)], [ZA4970; F, H, Et, H, NHPh], [ZA4971; F, H, Et, H, NH (2-Py)], [ ZA4972; F, H, Et, H, NH (3-Py)], [ZA4973; F, H, Et, H, NH (4-Py)], [ZA4974; F, H, Et, H, NMe ₂ ], [ZA4975; F, H, Et, H, NMeEt], [ZA4976; F, H, Et, H, NMePr], [ZA4977; F, H, Et, H, NMeBu], [ZA4978; F, H , Et, H, N MePen], [ZA4979; F, H, Et, H, NMeHex], [ZA4980; F, H, Et, H, NMe (i-Pr)], [ZA4981; F, H, Et, H, NMe (i -Bu)], [ZA4982; F, H, Et, H, NMe (c-Pr)], [ZA4983; F, H, Et, H, NMe (c-Bu)], [ZA4984; F, H, Et, H, NMe (c-Pen)], [ZA4985; F, H, Et, H, NMe (c-Hex)], [ZA4986; F, H, Et, H, NMeCH ₂ (c-Pr)] , [ZA4987; F, H, Et, H, NMeCH ₂ (c-Bu)], [ZA4988; F, H, Et, H, NMeCH ₂ (c-Pen)], [ZA4989; F, H, Et, H, NMeCH ₂ (c-Hex)], [ZA4990; F, H, Et, H, NMeCH ₂ F], [ZA4991; F, H, Et, H, NMeCHF ₂ ], [ZA4992; F, H, Et , H, NMeCF ₃ ], [ZA4993; F, H, Et, H, NMe (CH ₂ ) ₂ F], [ZA4994; F, H, Et, H, NMeCH ₂ CHF ₂ ], [ZA4995; F, H , Et, H, NMeCH ₂ CHF ₃ ], [ZA4996; F, H, Et, H, NMe (CH ₂
) ₃ F], [ZA4997; F, H, Et, H, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA4998; F, H, Et, H, NMe (CH ₂ ) ₂ CF ₃ ], [ZA4999; F, H, Et, H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA5000; F, H, Et, H, NMeCH ₂ Cl],

[ZA5001; F, H, Et, H, NMe (CH ₂ ) ₂ Cl], [ZA5002; F, H, Et, H, NMe (CH ₂ ) ₃ Cl], [ZA5003; F, H, Et, H , NMe (CH ₂ ) ₄ Cl], [ZA5004; F, H, Et, H, NMe (CH ₂ ) ₅ Cl], [ZA5005; F, H, Et, H, NMeCH ₂ OMe], [ZA5006; F , H, Et, H, NMe (CH ₂ ) ₂ OMe], [ZA5007; F, H, Et, H, NMe (CH ₂ ) ₃ OMe], [ZA5008; F, H, Et, H, NMe (CH ₂ ) ₄ OMe], [ZA5009; F, H, Et, H, NMeCH ₂ OEt], [ZA5010; F, H, Et, H, NMe (CH ₂ ) ₂ OEt], [ZA5011; F, H, Et , H, NMe (CH ₂ ) ₃ OEt], [ZA5012; F, H, Et, H, NMeCH ₂ OPr], [ZA5013; F, H, Et, H, NMe (CH ₂ ) ₂ OPr], [ZA5014 ; F, H, Et, H, NMe (CH ₂ ) ₃ OPr], [ZA5015; F, H, Et, H, NMeCH ₂ CN], [ZA5016; F, H, Et, H, NMe (CH ₂ ) ₂ CN], [ZA5017; F, H, Et, H, NMe (CH ₂ ) ₃ CN], [ZA5018; F, H, Et, H, NMe (CH ₂ ) ₄ CN], [ZA5019; F, H , Et, H, NMe (CH ₂ ) ₅ CN], [ZA5020; F, H, Et, H, NMeCH ₂ CH = CH ₂ ], [ZA5021; F, H, Et, H, NMeCH ₂ C≡CH] , [ZA5022; F, H, Et, H, NMeCH ₂ C≡CCH ₃ ], [ZA5023; F, H, Et, H, NMeCH ₂ Ph], [ZA5024; F, H, Et, H, NMeCH ₂ ( 2-Py)], [ZA5025; F, H, Et, H, NMeCH ₂ (3-Py)], [ZA5026; F, H, Et, H, NMeCH ₂ (4-Py)], [ZA5027; F , H, Et, H, NMe (CH ₂ ) ₂ Ph], [ZA5028; F, H, Et, H, NMe (CH ₂ ) ₂ (2-Py)], [ZA5029; F, H, Et, H , NMe (CH ₂ ) ₂ (3-Py)], [ZA5030; F, H, Et, H, NMe ( CH ₂ ) ₂ (4-Py)], [ZA5031; F, H, Et, H, NMePh], [ZA5032; F, H, Et, H, NMe (2-Py)], [ZA5033; F, H , Et, H, NMe (3-Py)], [ZA5034; F, H, Et, H, NMe (4-Py)], [ZA5035; F, H, Et, H, NEt ₂ ], [ZA5036; F, H, Et, H, NEtPr], [ZA5037; F, H, Et, H, NEtBu], [ZA5038; F, H, Et, H, NEtPen], [ZA5039; F, H, Et, H, NEtHex], [ZA5040; F, H, Et, H, NEt (i-Pr)], [ZA5041; F, H, Et, H, NEt (i-Bu)], [ZA5042; F, H, Et, H, NEt (c-Pr)], [ZA5043; F, H, Et, H, NEt (c-Bu)], [ZA5044; F, H, Et, H, NEt (c-Pen)], [ZA5045 ; F, H, Et, H, NEt (c-Hex)], [ZA5046; F, H, Et, H, NEtCH ₂ (c-Pr)], [ZA5047; F, H, Et, H, NEtCH ₂ (c-Bu)], [ZA5048; F, H, Et, H, NEtCH ₂ (c-Pen)], [ZA5049; F, H, Et, H, NEtCH ₂ (c-Hex)], [ZA5050; F, H, Et, H, NEtCH ₂ F], [ZA5051; F, H, Et, H, NEtCHF ₂ ], [ZA5052; F, H, Et, H, NEtCF ₃ ], [ZA5053; F, H, Et, H, NEt (CH ₂ ) ₂ F], [ZA5054; F, H, Et, H, NEtCH ₂ CHF ₂ ], [ZA5055; F, H, Et, H, NEtCH ₂ CHF ₃ ], [ZA5056; F, H, Et, H, NEt (CH ₂ ) ₃ F], [ZA5057; F, H, Et, H, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA5058; F, H, Et, H, NEt (CH ₂ ) ₂ CF ₃ ], [ZA5059; F, H, Et, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA5060; F, H, Et, H, NEtCH ₂ Cl], [ZA5061; F , H, Et, H, NEt (CH ₂ ) ₂ Cl], [ZA5062; F, H, Et, H, NEt (CH ₂ ) ₃ Cl], [ZA5063; F, H, Et, H, NEt (C H ₂ ) ₄ Cl], [ZA5064; F, H, Et, H, NEt (CH ₂ ) ₅ Cl], [ZA5065; F, H, Et, H, NEtCH ₂ OMe], [ZA5066; F, H, Et, H, NEt (CH ₂ ) ₂ OMe], [ZA5067; F, H, Et, H, NEt (CH ₂ ) ₃ OMe], [ZA5068; F, H, Et, H, NEt (CH ₂ ) ₄ OMe], [ZA5069; F, H, Et, H, NEtCH ₂ OEt], [ZA5070; F, H, Et, H, NEt (CH ₂ ) ₂ OEt], [ZA5071; F, H, Et, H, NEt (CH ₂ ) ₃ OEt], [ZA5072; F, H, Et, H, NEtCH ₂ OPr], [ZA5073; F, H, Et, H, NEt (CH ₂ ) ₂ OPr], [ZA5074; F, H, Et, H, NEt (CH ₂ ) ₃ OPr], [ZA5075; F, H, Et, H, NEtCH ₂ CN], [ZA5076; F, H, Et, H, NEt (CH ₂ ) ₂ CN] , [ZA5077; F, H, Et, H, NEt (CH ₂ ) ₃ CN], [ZA5078; F, H, Et, H, NEt (CH ₂ ) ₄ CN], [ZA5079; F, H, Et, H, NEt (CH ₂ ) ₅ CN], [ZA5080; F, H, Et, H, NEtCH ₂ CH = CH ₂ ], [ZA5081; F, H, Et, H, NEtCH ₂ C≡CH], [ZA5082 ; F, H, Et, H, NEtCH ₂ C≡CCH ₃ ], [ZA5083; F, H, Et, H, NEtCH ₂ Ph], [ZA5084; F, H, Et, H, NEtCH ₂ (2-Py )], [ZA5085; F, H, Et, H, NEtCH ₂ (3-Py)], [ZA5086; F, H, Et, H, NEtCH ₂ (4-Py)], [ZA5087; F, H, Et, H, NEt (CH ₂ ) ₂ Ph], [ZA5088; F, H, Et, H, NEt (CH ₂ ) ₂ (2-Py)], [ZA5089; F, H, Et, H, NEt ( CH ₂ ) ₂ (3-Py)], [ZA5090; F, H, Et, H, NEt (CH ₂ ) ₂ (4-Py)], [ZA5091; F, H, Et, H, NEtPh], [ ZA5092; F, H, Et, H, NEt (2-Py)], [ZA5093; F, H, Et, H, NEt ( 3-Py)], [ZA5094; F, H, Et, H, NEt (4-Py)], [ZA5095; F, H, Et, H, Pyr], [ZA5096; F, H, Et, H, Pip], [ZA5097; F, H, Et, H, Mor], [ZA5098; F, H, Et, H, OMe], [ZA5099; F, H, Et, H, OEt], [ZA5100; F, H, Et, H, OPr], [ZA5101; F, H, Et, H, OBu], [ZA5102; F, H, Et, H, OPen], [ZA5103; F, H, Et, H, OHex] , [ZA5104; F, H, Et, H, O (i-Pr)], [ZA5105; F, H, Et, H, O (i-Bu)], [ZA5106; F, H, Et, H, O (c-Pr)], [ZA5107; F, H, Et, H, O (c-Bu)], [ZA5108; F, H, Et, H, O (c-Pen)], [ZA5109; F , H, Et, H, O (c-Hex)], [ZA5110; F, H, Et, H, OCH ₂ (c-Pr)], [ZA5111; F, H, Et, H, OCH ₂ (c -Bu)], [ZA5112; F, H, Et, H, OCH ₂ (c-Pen)], [ZA5113; F, H, Et, H, OCH ₂ (c-Hex)], [ZA5114; F, H, Et, H, OCH ₂ F], [ZA5115; F, H, Et, H, OCHF ₂ ], [ZA5116; F, H, Et, H, OCF ₃ ], [ZA5117; F, H, Et, H, O (CH ₂ ) ₂ F], [ZA5118; F, H, Et, H, OCH ₂ CHF ₂ ], [ZA5119; F, H, Et, H, OCH ₂ CHF ₃ ], [ZA5120; F, H, Et, H, O (CH ₂ ) ₃ F], [ZA5121; F, H, Et, H, O (CH ₂ ) ₂ CHF ₂ ], [ZA5122; F, H, Et, H, O (CH ₂ ) ₂ CF ₃ ], [ZA5123; F, H, Et, H, OCH ₂ CH (CF ₃ ) ₂ ], [ZA5124; F, H, Et, H, OCH ₂ Cl], [ZA5125; F, H , Et, H, O (CH ₂ ) ₂ Cl], [ZA5126; F, H, Et, H, O (CH ₂ ) ₃ Cl], [ZA5127; F, H, Et, H, O (CH ₂ ) ₄ Cl], [ZA5128; F, H, Et, H, O (CH ₂ ) ₅ Cl], [ZA5129; F, H, Et, H, OCH ₂ OMe], [ZA5130; F, H, Et, H, O (CH ₂ ) ₂ OMe], [ZA5131; F, H, Et, H, O (CH ₂ ) ₃ OMe], [ZA5132; F, H, Et, H, O (CH ₂ ) ₄ OMe], [ZA5133; F, H, Et, H, OCH ₂ OEt], [ZA5134; F, H, Et, H, O (CH ₂ ) ₂ OEt] , [ZA5135; F, H, Et, H, O (CH ₂ ) ₃ OEt], [ZA5136; F, H, Et, H, OCH ₂ OPr], [ZA5137; F, H, Et, H, O ( CH ₂ ) ₂ OPr], [ZA5138; F, H, Et, H, O (CH ₂ ) ₃ OPr], [ZA5139; F, H, Et, H, OCH ₂ CN], [ZA5140; F, H, Et, H, O (CH ₂ ) ₂ CN], [ZA5141; F, H, Et, H, O (CH ₂ ) ₃ CN], [ZA5142; F, H, Et, H, O (CH ₂ ) ₄ CN], [ZA5143; F, H, Et, H, O (CH ₂ ) ₅ CN], [ZA5144; F, H, Et, H, OCH ₂ CH = CH ₂ ], [ZA5145; F, H, Et , H, OCH ₂ C≡CH], [ZA5146; F, H, Et, H, OCH ₂ C≡CCH ₃ ], [ZA5147; F, H, Et, H, OCH ₂ Ph], [ZA5148; F, H, Et, H, OCH ₂ (2-Py)], [ZA5149; F, H, Et, H, OCH ₂ (3-Py)], [ZA5150; F, H, Et, H, OCH ₂ (4 -Py)], [ZA5151; F, H, Et, H, O (CH ₂ ) ₂ Ph], [ZA5152; F, H, Et, H, O (CH ₂ ) ₂ (2-Py)], [ ZA5153; F, H, Et, H, O (CH ₂ ) ₂ (3-Py)], [ZA5154; F, H, Et, H, O (CH ₂ ) ₂ (4-Py)], [ZA5155; F, H, Et, H, OPh], [ZA5156; F, H, Et, H, O (2-Py)], [ZA5157; F, H, Et, H, O (3-Py)], [ ZA5158; F, H, Et, H, O (4-Py)], [ZA5159; F, H, Et, H, Me], [ZA5160; F, H, Et, H, Et], [ZA5161; F , H, Et, H, Pr], [ZA5162; F, H, Et, H, Bu], [ZA5 163; F, H, Et, H, Pen], [ZA5164; F, H, Et, H, Hex], [ZA5165; F, H, Et, H, (i-Pr)], [ZA5166; F, H, Et, H, (i-Bu)], [ZA5167; F, H, Et, H, (c-Pr)], [ZA5168; F, H, Et, H, (c-Bu)], [ ZA5169; F, H, Et, H, (c-Pen)], [ZA5170; F, H, Et, H, (c-Hex)], [ZA5171; F, H, Et, H, CH ₂ (c -Pr)], [ZA5172; F, H, Et, H, CH ₂ (c-Bu)], [ZA5173; F, H, Et, H, CH ₂ (c-Pen)], [ZA5174; F, H, Et, H, CH ₂ (c-Hex)], [ZA5175; F, H, Et, H, CH ₂ F], [ZA5176; F, H, Et, H, CHF ₂ ], [ZA5177; F , H, Et, H, CF ₃ ], [ZA5178; F, H, Et, H, (CH ₂ ) ₂ F], [ZA5179; F, H, Et, H, CH ₂ CHF ₂ ], [ZA5180; F, H, Et, H, CH ₂ CHF ₃ ], [ZA5181; F, H, Et, H, (CH ₂ ) ₃ F], [ZA5182; F, H, Et, H, (CH ₂ ) ₂ CHF ₂ ], [ZA5183; F, H, Et, H, (CH ₂ ) ₂ CF ₃ ], [ZA5184; F, H, Et, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA5185; F, H , Et, H, CH ₂ Cl], [ZA5186; F, H, Et, H, (CH ₂ ) ₂ Cl], [ZA5187; F, H, Et, H, (CH ₂ ) ₃ Cl], [ZA5188 ; F, H, Et, H, (CH ₂ ) ₄ Cl], [ZA5189; F, H, Et, H, (CH ₂ ) ₅ Cl], [ZA5190; F, H, Et, H, CH ₂ OMe ], [ZA5191; F, H, Et, H, (CH ₂ ) ₂ OMe], [ZA5192; F, H, Et, H, (CH ₂ ) ₃ OMe], [ZA5193; F, H, Et, H , (CH ₂ ) ₄ OMe], [ZA5194; F, H, Et, H, CH ₂ OEt], [ZA5195; F, H, Et, H, (CH ₂ ) ₂ OEt], [ZA5196; F, H , Et, H, (CH ₂ ) ₃ OEt], [ZA5197; F, H, Et, H, CH ₂ O Pr], [ZA5198; F, H, Et, H, (CH ₂ ) ₂ OPr], [ZA5199; F, H, Et, H, (CH ₂ ) ₃ OPr], [ZA5200; F, H, Et, H, CH ₂ CN], [ZA5201; F, H, Et, H, (CH ₂ ) ₂ CN], [ZA5202; F, H, Et, H, (CH ₂ ) ₃ CN], [ZA5203; F, H, Et, H, (CH ₂ ) ₄ CN], [ZA5204; F, H, Et, H, (CH ₂ ) ₅ CN], [ZA5205; F, H, Et, H, CH ₂ CH = CH ₂ ], [ZA5206; F, H, Et, H, CH ₂ C≡CH], [ZA5207; F, H, Et, H, CH ₂ C≡CCH ₃ ], [ZA5208; F, H, Et, H, CH ₂ Ph], [ZA5209; F, H, Et, H, CH ₂ (2-Py)], [ZA5210; F, H, Et, H, CH ₂ (3-Py)], [ZA5211; F, H, Et, H, CH ₂ (4-Py)], [ZA5212; F, H, Et, H, (CH ₂ ) ₂ Ph], [ZA5213; F, H, Et, H, (CH ₂ ) ₂ (2-Py)], [ZA5214; F, H, Et, H, (CH ₂ ) ₂ (3-Py)], [ZA5215; F, H, Et, H, (CH ₂ ) ₂ (4-Py )], [ZA5216; F, H, Et, H, Ph], [ZA5217; F, H, Et, H, 2-Py], [ZA5218; F, H, Et, H, 3-Py], [ ZA5219; F, H, Et, H, 4-Py], [ZA5220; F, H, Me, Et, NHMe], [ZA5221; F, H, Me, Et, NHEt], [ZA5222; F, H, Me, Et, NHPr], [ZA5223; F, H, Me, Et, NHBu], [ZA5224; F, H, Me, Et, NHPen], [ZA5225; F, H, Me, Et, NHHex], [ ZA5226; F, H, Me, Et, NH (i-Pr)], [ZA5227; F, H, Me, Et, NH (i-Bu)], [ZA5228; F, H, Me, Et, NH ( c-Pr)], [ZA5229; F, H, Me, Et, NH (c-Bu)], [ZA5230; F, H, Me, Et, NH (c-Pen)], [ZA5231; F, H , Me, Et, NH (c-Hex)], [ZA5232; F, H, Me, Et, NHCH ₂ (c- Pr)], [ZA5233; F, H, Me, Et, NHCH ₂ (c-Bu)], [ZA5234; F, H, Me, Et, NHCH ₂ (c-Pen)], [ZA5235; F, H , Me, Et, NHCH ₂ (c-Hex)], [ZA5236; F, H, Me, Et, NHCH ₂ F], [ZA5237; F, H, Me, Et, NHCHF ₂ ], [ZA5238; F, H, Me, Et, NHCF ₃ ], [ZA5239; F, H, Me, Et, NH (CH ₂ ) ₂ F], [ZA5240; F, H, Me, Et, NHCH ₂ CHF ₂ ], [ZA5241; F, H, Me, Et, NHCH ₂ CHF ₃ ], [ZA5242; F, H, Me, Et, NH (CH ₂ ) ₃ F], [ZA5243; F, H, Me, Et, NH (CH ₂ ) ₂ CHF ₂ ], [ZA5244; F, H, Me, Et, NH (CH ₂ ) ₂ CF ₃ ], [ZA5245; F, H, Me, Et, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA5246; F, H, Me, Et, NHCH ₂ Cl], [ZA5247; F, H, Me, Et, NH (CH ₂ )
₂ Cl], [ZA5248; F, H, Me, Et, NH (CH ₂ ) ₃ Cl], [ZA5249; F, H, Me, Et, NH (CH ₂ ) ₄ Cl], [ZA5250; F, H , Me, Et, NH (CH ₂ ) ₅ Cl],

[ZA5251; F, H, Me, Et, NHCH ₂ OMe], [ZA5252; F, H, Me, Et, NH (CH ₂ ) ₂ OMe], [ZA5253; F, H, Me, Et, NH (CH ₂ ) ₃ OMe], [ZA5254; F, H, Me, Et, NH (CH ₂ ) ₄ OMe], [ZA5255; F, H, Me, Et, NHCH ₂ OEt], [ZA5256; F, H, Me , Et, NH (CH ₂ ) ₂ OEt], [ZA5257; F, H, Me, Et, NH (CH ₂ ) ₃ OEt], [ZA5258; F, H, Me, Et, NHCH ₂ OPr], [ZA5259 ; F, H, Me, Et, NH (CH ₂ ) ₂ OPr], [ZA5260; F, H, Me, Et, NH (CH ₂ ) ₃ OPr], [ZA5261; F, H, Me, Et, NHCH ₂ CN], [ZA5262; F, H, Me, Et, NH (CH ₂ ) ₂ CN], [ZA5263; F, H, Me, Et, NH (CH ₂ ) ₃ CN], [ZA5264; F, H , Me, Et, NH (CH ₂ ) ₄ CN], [ZA5265; F, H, Me, Et, NH (CH ₂ ) ₅ CN], [ZA5266; F, H, Me, Et, NHCH ₂ CH = CH ₂ ], [ZA5267; F, H, Me, Et, NHCH ₂ C≡CH], [ZA5268; F, H, Me, Et, NHCH ₂ C≡CCH ₃ ], [ZA5269; F, H, Me, Et , NHCH ₂ Ph], [ZA5270; F, H, Me, Et, NHCH ₂ (2-Py)], [ZA5271; F, H, Me, Et, NHCH ₂ (3-Py)], [ZA5272; F , H, Me, Et, NHCH ₂ (4-Py)], [ZA5273; F, H, Me, Et, NH (CH ₂ ) ₂ Ph], [ZA5274; F, H, Me, Et, NH (CH ₂ ) ₂ (2-Py)], [ZA5275; F, H, Me, Et, NH (CH ₂ ) ₂ (3-Py)], [ZA5276; F, H, Me, Et, NH (CH ₂ ) ₂ (4-Py)], [ZA5277; F, H, Me, Et, NHPh], [ZA5278; F, H, Me, Et, NH (2-Py)], [ZA5279; F, H, Me, Et, NH (3-Py)], [ZA5280; F, H, Me, Et, NH (4-Py)], [ZA5281; F, H , Me, Et, NMe ₂ ], [ZA5282; F, H, Me, Et, NMeEt], [ZA5283; F, H, Me, Et, NMePr], [ZA5284; F, H, Me, Et, NMeBu] , [ZA5285; F, H, Me, Et, NMePen], [ZA5286; F, H, Me, Et, NMeHex], [ZA5287; F, H, Me, Et, NMe (i-Pr)], [ZA5288 ; F, H, Me, Et, NMe (i-Bu)], [ZA5289; F, H, Me, Et, NMe (c-Pr)], [ZA5290; F, H, Me, Et, NMe (c -Bu)], [ZA5291; F, H, Me, Et, NMe (c-Pen)], [ZA5292; F, H, Me, Et, NMe (c-Hex)], [ZA5293; F, H, Me, Et, NMeCH ₂ (c-Pr)], [ZA5294; F, H, Me, Et, NMeCH ₂ (c-Bu)], [ZA5295; F, H, Me, Et, NMeCH ₂ (c-Pen )], [ZA5296; F, H, Me, Et, NMeCH ₂ (c-Hex)], [ZA5297; F, H, Me, Et, NMeCH ₂ F], [ZA5298; F, H, Me, Et, NMeCHF ₂ ], [ZA5299; F, H, Me, Et, NMeCF ₃ ], [ZA5300; F, H, Me, Et, NMe (CH ₂ ) ₂ F], [ZA5301; F, H, Me, Et, NMeCH ₂ CHF ₂ ], [ZA5302; F, H, Me, Et, NMeCH ₂ CHF ₃ ], [ZA5303; F, H, Me, Et, NMe (CH ₂ ) ₃ F], [ZA5304; F, H, Me, Et, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA5305; F, H, Me, Et, NMe (CH ₂ ) ₂ CF ₃ ], [ZA5306; F, H, Me, Et, NMeCH ₂ CH ( CF ₃ ) ₂ ], [ZA5307; F, H, Me, Et, NMeCH ₂ Cl], [ZA5308; F, H, Me, Et, NMe (CH ₂ ) ₂ Cl], [ZA5309; F, H, Me , Et, NMe (CH ₂ ) ₃ Cl], [ZA5310; F, H, Me, Et, NMe (CH ₂ ) ₄ Cl], [ZA5311; F, H, Me, Et, NMe (CH ₂ ) ₅ Cl ], [ZA5312; F, H, Me, Et, NMeCH ₂ OMe], [ZA5 313; F, H, Me, Et, NMe (CH ₂ ) ₂ OMe], [ZA5314; F, H, Me, Et, NMe (CH ₂ ) ₃ OMe], [ZA5315; F, H, Me, Et, NMe (CH ₂ ) ₄ OMe], [ZA5316; F, H, Me, Et, NMeCH ₂ OEt], [ZA5317; F, H, Me, Et, NMe (CH ₂ ) ₂ OEt], [ZA5318; F, H, Me, Et, NMe (CH ₂ ) ₃ OEt], [ZA5319; F, H, Me, Et, NMeCH ₂ OPr], [ZA5320; F, H, Me, Et, NMe (CH ₂ ) ₂ OPr] , [ZA5321; F, H, Me, Et, NMe (CH ₂ ) ₃ OPr], [ZA5322; F, H, Me, Et, NMeCH ₂ CN], [ZA5323; F, H, Me, Et, NMe ( _{CH 2) 2 CN], [} ZA5324; F, H, Me, Et, NMe (CH 2) 3 CN], [ZA5325; F, H, Me, Et, NMe (CH 2) 4 CN], [ZA5326; F, H, Me, Et, NMe (CH ₂ ) ₅ CN], [ZA5327; F, H, Me, Et, NMeCH ₂ CH = CH ₂ ], [ZA5328; F, H, Me, Et, NMeCH ₂ C ≡CH], [ZA5329; F, H, Me, Et, NMeCH ₂ C≡CCH ₃ ], [ZA5330; F, H, Me, Et, NMeCH ₂ Ph], [ZA5331; F, H, Me, Et, NMeCH ₂ (2-Py)], [ZA5332; F, H, Me, Et, NMeCH ₂ (3-Py)], [ZA5333; F, H, Me, Et, NMeCH ₂ (4-Py)], [ ZA5334; F, H, Me, Et, NMe (CH ₂ ) ₂ Ph], [ZA5335; F, H, Me, Et, NMe (CH ₂ ) ₂ (2-Py)], [ZA5336; F, H, Me, Et, NMe (CH ₂ ) ₂ (3-Py)], [ZA5337; F, H, Me, Et, NMe (CH ₂ ) ₂ (4-Py)], [ZA5338; F, H, Me, Et, NMePh], [ZA5339; F, H, Me, Et, NMe (2-Py)], [ZA5340; F, H, Me, Et, NMe (3-Py)], [ZA5341; F, H, Me, Et, NMe (4-Py)], [ZA5342; F, H, Me, E t, NEt ₂ ], [ZA5343; F, H, Me, Et, NEtPr], [ZA5344; F, H, Me, Et, NEtBu], [ZA5345; F, H, Me, Et, NEtPen], [ZA5346 ; F, H, Me, Et, NEtHex], [ZA5347; F, H, Me, Et, NEt (i-Pr)], [ZA5348; F, H, Me, Et, NEt (i-Bu)], [ZA5349; F, H, Me, Et, NEt (c-Pr)], [ZA5350; F, H, Me, Et, NEt (c-Bu)], [ZA5351; F, H, Me, Et, NEt (c-Pen)], [ZA5352; F, H, Me, Et, NEt (c-Hex)], [ZA5353; F, H, Me, Et, NEtCH ₂ (c-Pr)], [ZA5354; F , H, Me, Et, NEtCH ₂ (c-Bu)], [ZA5355; F, H, Me, Et, NEtCH ₂ (c-Pen)], [ZA5356; F, H, Me, Et, NEtCH ₂ ( c-Hex)], [ZA5357; F, H, Me, Et, NEtCH ₂ F], [ZA5358; F, H, Me, Et, NEtCHF ₂ ], [ZA5359; F, H, Me, Et, NEtCF ₃ ], [ZA5360; F, H, Me, Et, NEt (CH ₂ ) ₂ F], [ZA5361; F, H, Me, Et, NEtCH ₂ CHF ₂ ], [ZA5362; F, H, Me, Et, NEtCH ₂ CHF ₃ ], [ZA5363; F, H, Me, Et, NEt (CH ₂ ) ₃ F], [ZA5364; F, H, Me, Et, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA5365; F, H, Me, Et, NEt (CH ₂ ) ₂ CF ₃ ], [ZA5366; F, H, Me, Et, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA5367; F, H, Me, Et, NEtCH ₂ Cl], [ZA5368; F, H, Me, Et, NEt (CH ₂ ) ₂ Cl], [ZA5369; F, H, Me, Et, NEt (CH ₂ ) ₃ Cl], [ZA5370; F, H, Me, Et, NEt (CH ₂ ) ₄ Cl], [ZA5371; F, H, Me, Et, NEt (CH ₂ ) ₅ Cl], [ZA5372; F, H, Me, Et, NEtCH ₂ OMe] , [ZA5373; F, H, Me, Et, NEt (CH ₂ ) ₂ OMe ], [ZA5374; F, H, Me, Et, NEt (CH ₂ ) ₃ OMe], [ZA5375; F, H, Me, Et, NEt (CH ₂ ) ₄ OMe], [ZA5376; F, H, Me , Et, NEtCH ₂ OEt], [ZA5377; F, H, Me, Et, NEt (CH ₂ ) ₂ OEt], [ZA5378; F, H, Me, Et, NEt (CH ₂ ) ₃ OEt], [ZA5379 ; F, H, Me, Et, NEtCH ₂ OPr], [ZA5380; F, H, Me, Et, NEt (CH ₂ ) ₂ OPr], [ZA5381; F, H, Me, Et, NEt (CH ₂ ) ₃ OPr], [ZA5382; F, H, Me, Et, NEtCH ₂ CN], [ZA5383; F, H, Me, Et, NEt (CH ₂ ) ₂ CN], [ZA5384; F, H, Me, Et , NEt (CH ₂ ) ₃ CN], [ZA5385; F, H, Me, Et, NEt (CH ₂ ) ₄ CN], [ZA5386; F, H, Me, Et, NEt (CH ₂ ) ₅ CN], [ZA5387; F, H, Me, Et, NEtCH ₂ CH = CH ₂ ], [ZA5388; F, H, Me, Et, NEtCH ₂ C≡CH], [ZA5389; F, H, Me, Et, NEtCH ₂ C≡CCH ₃ ], [ZA5390; F, H, Me, Et, NEtCH ₂ Ph], [ZA5391; F, H, Me, Et, NEtCH ₂ (2-Py)], [ZA5392; F, H, Me , Et, NEtCH ₂ (3-Py)], [ZA5393; F, H, Me, Et, NEtCH ₂ (4-Py)], [ZA5394; F, H, Me, Et, NEt (CH ₂ ) ₂ Ph ], [ZA5395; F, H, Me, Et, NEt (CH ₂ ) ₂ (2-Py)], [ZA5396; F, H, Me, Et, NEt (CH ₂ ) ₂ (3-Py)], [ZA5397; F, H, Me, Et, NEt (CH ₂ ) ₂ (4-Py)], [ZA5398; F, H, Me, Et, NEtPh], [ZA5399; F, H, Me, Et, NEt (2-Py)], [ZA5400; F, H, Me, Et, NEt (3-Py)], [ZA5401; F, H, Me, Et, NEt (4-Py)], [ZA5402; F, H, Me, Et, Pyr], [ZA5403; F, H, Me, Et, Pip], [ZA5404; F, H, Me, Et, Mor], [ZA5405; F, H, Me, Et, OMe], [ZA5406; F, H, Me, Et, OEt], [ZA5407; F, H, Me , Et, OPr], [ZA5408; F, H, Me, Et, OBu], [ZA5409; F, H, Me, Et, OPen], [ZA5410; F, H, Me, Et, OHex], [ZA5411 ; F, H, Me, Et, O (i-Pr)], [ZA5412; F, H, Me, Et, O (i-Bu)], [ZA5413; F, H, Me, Et, O (c -Pr)], [ZA5414; F, H, Me, Et, O (c-Bu)], [ZA5415; F, H, Me, Et, O (c-Pen)], [ZA5416; F, H, Me, Et, O (c-Hex)], [ZA5417; F, H, Me, Et, OCH ₂ (c-Pr)], [ZA5418; F, H, Me, Et, OCH ₂ (c-Bu) ], [ZA5419; F, H, Me, Et, OCH ₂ (c-Pen)], [ZA5420; F, H, Me, Et, OCH ₂ (c-Hex)], [ZA5421; F, H, Me , Et, OCH ₂ F], [ZA5422; F, H, Me, Et, OCHF ₂ ], [ZA5423; F, H, Me, Et, OCF ₃ ], [ZA5424; F, H, Me, Et, O (CH ₂ ) ₂ F], [ZA5425; F, H, Me, Et, OCH ₂ CHF ₂ ], [ZA5426; F, H, Me, Et, OCH ₂ CHF ₃ ], [ZA5427; F, H, Me , Et, O (CH ₂ ) ₃ F], [ZA5428; F, H, Me, Et, O (CH ₂ ) ₂ CHF ₂ ], [ZA5429; F, H, Me, Et, O (CH ₂ ) ₂ CF ₃ ], [ZA5430; F, H, Me, Et, OCH ₂ CH (CF ₃ ) ₂ ], [ZA5431; F, H, Me, Et, OCH ₂ Cl], [ZA5432; F, H, Me, Et, O (CH ₂ ) ₂ Cl], [ZA5433; F, H, Me, Et, O (CH ₂ ) ₃ Cl], [ZA5434; F, H, Me, Et, O (CH ₂ ) ₄ Cl] , [ZA5435; F, H, Me, Et, O (CH ₂ ) ₅ Cl], [ZA5436; F, H, Me, Et, OCH ₂ OMe], [ZA5437; F, H, Me, Et, O ( CH ₂ ) ₂ OMe], [ ZA5438; F, H, Me, Et, O (CH ₂ ) ₃ OMe], [ZA5439; F, H, Me, Et, O (CH ₂ ) ₄ OMe], [ZA5440; F, H, Me, Et, OCH ₂ OEt], [ZA5441; F, H, Me, Et, O (CH ₂ ) ₂ OEt], [ZA5442; F, H, Me, Et, O (CH ₂ ) ₃ OEt], [ZA5443; F, H, Me, Et, OCH ₂ OPr], [ZA5444; F, H, Me, Et, O (CH ₂ ) ₂ OPr], [ZA5445; F, H, Me, Et, O (CH ₂ ) ₃ OPr] , [ZA5446; F, H, Me, Et, OCH ₂ CN], [ZA5447; F, H, Me, Et, O (CH ₂ ) ₂ CN], [ZA5448; F, H, Me, Et, O ( _{CH 2) 3 CN], [} ZA5449; F, H, Me, Et, O (CH 2) 4 CN], [ZA5450; F, H, Me, Et, O (CH 2) 5 CN], [ZA5451; F, H, Me, Et, OCH ₂ CH = CH ₂ ], [ZA5452; F, H, Me, Et, OCH ₂ C≡CH], [ZA5453; F, H, Me, Et, OCH ₂ C≡CCH ₃ ], [ZA5454; F, H, Me, Et, OCH ₂ Ph], [ZA5455; F, H, Me, Et, OCH ₂ (2-Py)], [ZA5456; F, H, Me, Et, OCH ₂ (3-Py)], [ZA5457; F, H, Me, Et, OCH ₂ (4-Py)], [ZA5458; F, H, Me, Et, O (CH ₂ ) ₂ Ph], [ ZA5459; F, H, Me, Et, O (CH ₂ ) ₂ (2-Py)], [ZA5460; F, H, Me, Et, O (CH ₂ ) ₂ (3-Py)], [ZA5461; F, H, Me, Et, O (CH ₂ ) ₂ (4-Py)], [ZA5462; F, H, Me, Et, OPh], [ZA5463; F, H, Me, Et, O (2- Py)], [ZA5464; F, H, Me, Et, O (3-Py)], [ZA5465; F, H, Me, Et, O (4-Py)], [ZA5466; F, H, Me , Et, Me], [ZA5467; F, H, Me, Et, Et], [ZA5468; F, H, Me, Et, Pr], [ZA5469; F, H, Me, Et, Bu], [ZA5470 ; F, H, Me, Et , Pen], [ZA5471; F, H, Me, Et, Hex], [ZA5472; F, H, Me, Et, (i-Pr)], [ZA5473; F, H, Me, Et, (i- Bu)], [ZA5474; F, H, Me, Et, (c-Pr)], [ZA5475; F, H, Me, Et, (c-Bu)], [ZA5476; F, H, Me, Et , (c-Pen)], [ZA5477; F, H, Me, Et, (c-Hex)], [ZA5478; F, H, Me, Et, CH ₂ (c-Pr)], [ZA5479; F , H, Me, Et, CH ₂ (c-Bu)], [ZA5480; F, H, Me, Et, CH ₂ (c-Pen)], [ZA5481; F, H, Me, Et, CH ₂ ( c-Hex)], [ZA5482; F, H, Me, Et, CH ₂ F], [ZA5483; F, H, Me, Et, CHF ₂ ], [ZA5484; F, H, Me, Et, CF ₃ ], [ZA5485; F, H, Me, Et, (CH ₂ ) ₂ F], [ZA5486; F, H, Me, Et, CH ₂ CHF ₂ ], [ZA5487; F, H, Me, Et, CH ₂ CHF ₃ ], [ZA5488; F, H, Me, Et, (CH ₂ ) ₃ F], [ZA5489; F, H, Me, Et, (CH ₂ ) ₂ CHF ₂ ], [ZA5490; F, H , Me, Et, (CH ₂ ) ₂ CF ₃ ], [ZA5491; F, H, Me, Et,
CH ₂ CH (CF ₃ ) ₂ ], [ZA5492; F, H, Me, Et, CH ₂ Cl], [ZA5493; F, H, Me, Et, (CH ₂ ) ₂ Cl], [ZA5494; F, H, Me, Et, (CH ₂ ) ₃ Cl], [ZA5495; F, H, Me, Et, (CH ₂ ) ₄ Cl], [ZA5496; F, H, Me, Et, (CH ₂ ) ₅ Cl ], [ZA5497; F, H, Me, Et, CH ₂ OMe], [ZA5498; F, H, Me, Et, (CH ₂ ) ₂ OMe], [ZA5499; F, H, Me, Et, (CH ₂ ) ₃ OMe], [ZA5500; F, H, Me, Et, (CH ₂ ) ₄ OMe],

[ZA5501; F, H, Me, Et, CH ₂ OEt], [ZA5502; F, H, Me, Et, (CH ₂ ) ₂ OEt], [ZA5503; F, H, Me, Et, (CH ₂ ) ₃ OEt], [ZA5504; F, H, Me, Et, CH ₂ OPr], [ZA5505; F, H, Me, Et, (CH ₂ ) ₂ OPr], [ZA5506; F, H, Me, Et, (CH ₂ ) ₃ OPr], [ZA5507; F, H, Me, Et, CH ₂ CN], [ZA5508; F, H, Me, Et, (CH ₂ ) ₂ CN], [ZA5509; F, H, Me, Et, (CH ₂ ) ₃ CN], [ZA5510; F, H, Me, Et, (CH ₂ ) ₄ CN], [ZA5511; F, H, Me, Et, (CH ₂ ) ₅ CN], [ZA5512; F, H, Me, Et, CH ₂ CH = CH ₂ ], [ZA5513; F, H, Me, Et, CH ₂ C≡CH], [ZA5514; F, H, Me, Et, CH ₂ C≡CCH ₃ ], [ZA5515; F, H, Me, Et, CH ₂ Ph], [ZA5516; F, H, Me, Et, CH ₂ (2-Py)], [ZA5517; F, H, Me , Et, CH ₂ (3-Py)], [ZA5518; F, H, Me, Et, CH ₂ (4-Py)], [ZA5519; F, H, Me, Et, (CH ₂ ) ₂ Ph] , [ZA5520; F, H, Me, Et, (CH ₂ ) ₂ (2-Py)], [ZA5521; F, H, Me, Et, (CH ₂ ) ₂ (3-Py)], [ZA5522; F, H, Me, Et, (CH ₂ ) ₂ (4-Py)], [ZA5523; F, H, Me, Et, Ph], [ZA5524; F, H, Me, Et, 2-Py], [ZA5525; F, H, Me, Et, 3-Py], [ZA5526; F, H, Me, Et, 4-Py], [ZA5527; H, F, H, H, NHMe], [ZA5528; H , F, H, H, NHEt], [ZA5529; H, F, H, H, NHPr], [ZA5530; H, F, H, H, NHBu], [ZA5531; H, F, H, H, NHPen ], [ZA5532; H, F, H, H, NHHex], [ZA5533; H, F, H, H, NH (i-Pr)], [ZA5534; H, F, H, H, NH (i- Bu)], [ZA5535; H, F, H, H, NH (c-Pr)], [ZA5536; H, F, H, H, NH (c-Bu)], [ZA5537; H, F, H, H, NH (c-Pen)], [ZA5538; H, F, H, H, NH (c-Hex)], [ZA5539; H, F, H, H, NHCH ₂ (c-Pr)], [ZA5540; H, F, H, H, NHCH ₂ (c- Bu)], [ZA5541; H, F, H, H, NHCH ₂ (c-Pen)], [ZA5542; H, F, H, H, NHCH ₂ (c-Hex)], [ZA5543; H, F , H, H, NHCH ₂ F], [ZA5544; H, F, H, H, NHCHF ₂ ], [ZA5545; H, F, H, H, NHCF ₃ ], [ZA5546; H, F, H, H , NH (CH ₂ ) ₂ F], [ZA5547; H, F, H, H, NHCH ₂ CHF ₂ ], [ZA5548; H, F, H, H, NHCH ₂ CHF ₃ ], [ZA5549; H, F , H, H, NH (CH ₂ ) ₃ F], [ZA5550; H, F, H, H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA5551; H, F, H, H, NH (CH ₂ ) ₂ CF ₃ ], [ZA5552; H, F, H, H, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA5553; H, F, H, H, NHCH ₂ Cl], [ZA5554; H, F, H, H, NH (CH ₂ ) ₂ Cl], [ZA5555; H, F, H, H, NH (CH ₂ ) ₃ Cl], [ZA5556; H, F, H, H, NH (CH ₂ ) ₄ Cl], [ZA5557; H, F, H, H, NH (CH ₂ ) ₅ Cl], [ZA5558; H, F, H, H, NHCH ₂ OMe], [ZA5559; H, F, H, H, NH (CH ₂ ) ₂ OMe], [ZA5560; H, F, H, H, NH (CH ₂ ) ₃ OMe], [ZA5561; H, F, H, H, NH (CH ₂ ) ₄ OMe], [ ZA5562; H, F, H, H, NHCH ₂ OEt], [ZA5563; H, F, H, H, NH (CH ₂ ) ₂ OEt], [ZA5564; H, F, H, H, NH (CH ₂ ) ₃ OEt], [ZA5565; H, F, H, H, NHCH ₂ OPr], [ZA5566; H, F, H, H, NH (CH ₂ ) ₂ OPr], [ZA5567; H, F, H, H, NH (CH ₂ ) ₃ OPr], [ZA5568 ; H, F, H, H, NHCH ₂ CN], [ZA5569; H, F, H, H, NH (CH ₂ ) ₂ CN], [ZA5570; H, F, H, H, NH (CH ₂ ) ₃ CN], [ZA5571; H, F, H, H, NH (CH ₂ ) ₄ CN], [ZA5572; H, F, H, H, NH (CH ₂ ) ₅ CN], [ZA5573; H, F , H, H, NHCH ₂ CH = CH ₂ ], [ZA5574; H, F, H, H, NHCH ₂ C≡CH], [ZA5575; H, F, H, H, NHCH ₂ C≡CCH ₃ ], [ZA5576; H, F, H, H, NHCH ₂ Ph], [ZA5577; H, F, H, H, NHCH ₂ (2-Py)], [ZA5578; H, F, H, H, NHCH ₂ ( 3-Py)], [ZA5579; H, F, H, H, NHCH ₂ (4-Py)], [ZA5580; H, F, H, H, NH (CH ₂ ) ₂ Ph], [ZA5581; H , F, H, H, NH (CH ₂ ) ₂ (2-Py)], [ZA5582; H, F, H, H, NH (CH ₂ ) ₂ (3-Py)], [ZA5583; H, F , H, H, NH (CH ₂ ) ₂ (4-Py)], [ZA5584; H, F, H, H, NHPh], [ZA5585; H, F, H, H, NH (2-Py)] , [ZA5586; H, F, H, H, NH (3-Py)], [ZA5587; H, F, H, H, NH (4-Py)], [ZA5588; H, F, H, H, NMe ₂ ], [ZA5589; H, F, H, H, NMeEt], [ZA5590; H, F, H, H, NMePr], [ZA5591; H, F, H, H, NMeBu], [ZA5592; H , F, H, H, NMePen], [ZA5593; H, F, H, H, NMeHex], [ZA5594; H, F, H, H, NMe (i-Pr)], [ZA5595; H, F, H, H, NMe (i-Bu)], [ZA5596; H, F, H, H, NMe (c-Pr)], [ZA5597; H, F, H, H, NMe (c-Bu)], [ZA5598; H, F, H, H, NMe (c-Pen)], [ZA5599; H, F, H, H, NMe (c-Hex)], [ZA5600; H, F, H, H, NMeCH ₂ (c-Pr)], [ZA5601; H, F, H, H, NMeCH ₂ (c-Bu)], [ZA5602; H, F, H, H, NMeCH ₂ (c-Pen)], [ZA5603; H, F, H, H, NMeCH ₂ (c-Hex)], [ZA5604; H, F, H, H, NMeCH ₂ F], [ZA5605; H, F, H, H, NMeCHF ₂ ], [ZA5606; H, F, H, H, NMeCF ₃ ], [ZA5607; H, F, H, H, NMe (CH ₂ ) ₂ F], [ZA5608; H, F, H, H, NMeCH ₂ CHF ₂ ], [ZA5609; H, F, H, H, NMeCH ₂ CHF ₃ ], [ZA5610; H, F, H, H, NMe (CH ₂ ) ₃ F], [ZA5611; H, F, H, H, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA5612; H, F, H, H, NMe (CH ₂ ) ₂ CF ₃ ], [ZA5613; H, F, H, H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA5614; H, F, H, H, NMeCH ₂ Cl], [ZA5615; H, F, H, H, NMe (CH ₂ ) ₂ Cl], [ZA5616; H , F, H, H, NMe (CH ₂ ) ₃ Cl], [ZA5617; H, F, H, H, NMe (CH ₂ ) ₄ Cl], [ZA5618; H, F, H, H, NMe (CH ₂ ) ₅ Cl], [ZA5619; H, F, H, H, NMeCH ₂ OMe], [ZA5620; H, F, H, H, NMe (CH ₂ ) ₂ OMe], [ZA5621; H, F, H , H, NMe (CH ₂ ) ₃ OMe], [ZA5622; H, F, H, H, NMe (CH ₂ ) ₄ OMe], [ZA5623; H, F, H, H, NMeCH ₂ OEt], [ZA5624 ; H, F, H, H, NMe (CH ₂ ) ₂ OEt], [ZA5625; H, F, H, H, NMe (CH ₂ ) ₃ OEt], [ZA5626; H, F, H, H, NMeCH ₂ OPr], [ZA5627; H, F, H, H, NMe (CH ₂ ) ₂ OPr], [ZA5628; H, F, H, H, NMe (CH ₂ ) ₃ OPr], [ZA5629; H, F , H, H, NMeCH ₂ CN], [ZA5630; H, F, H, H, NMe (CH ₂ ) ₂ CN], [ZA5631; H, F, H, H, NMe (CH ₂ ) ₃ CN], [ZA5632; H, F, H, H, NMe (CH ₂ ) ₄ CN], [ZA5633; H, F, H, H, NMe (CH ₂ ) ₅ CN], [ZA5634; H, F, H, H, NMeCH ₂ CH = CH ₂ ], [ZA5635; H, F, H, H, NMeCH ₂ C≡CH], [ZA5636; H, F, H, H, NMeCH ₂ C≡CCH ₃ ], [ZA5637; H, F, H, H, NMeCH ₂ Ph], [ZA5638; H, F, H, H, NMeCH ₂ (2-Py)], [ZA5639; H , F, H, H, NMeCH ₂ (3-Py)], [ZA5640; H, F, H, H, NMeCH ₂ (4-Py)], [ZA5641; H, F, H, H, NMe (CH ₂ ) ₂ Ph], [ZA5642; H, F, H, H, NMe (CH ₂ ) ₂ (2-Py)], [ZA5643; H, F, H, H, NMe (CH ₂ ) ₂ (3- Py)], [ZA5644; H, F, H, H, NMe (CH ₂ ) ₂ (4-Py)], [ZA5645; H, F, H, H, NMePh], [ZA5646; H, F, H , H, NMe (2-Py)], [ZA5647; H, F, H, H, NMe (3-Py)], [ZA5648; H, F, H, H, NMe (4-Py)], [ ZA5649; H, F, H, H, NEt ₂ ], [ZA5650; H, F, H, H, NEtPr], [ZA5651; H, F, H, H, NEtBu], [ZA5652; H, F, H , H, NEtPen], [ZA5653; H, F, H, H, NEtHex], [ZA5654; H, F, H, H, NEt (i-Pr)], [ZA5655; H, F, H, H, NEt (i-Bu)], [ZA5656; H, F, H, H, NEt (c-Pr)], [ZA5657; H, F, H, H, NEt (c-Bu)], [ZA5658; H , F, H, H, NEt (c-Pen)], [ZA5659; H, F, H, H, NEt (c-Hex)], [ZA5660; H, F, H, H, NEtCH ₂ (c- Pr)], [ZA5661; H, F, H, H, NEtCH ₂ (c-Bu)], [ZA5662; H, F, H, H, NEtCH ₂ (c-Pen)], [ZA5663; H, F , H, H, NEtCH ₂ (c-Hex)], [ZA5664; H, F, H, H, NEtCH ₂ F], [ZA5665; H, F, H, H, NEtCHF ₂ ], [ZA5666; H, F, H, H, NEtCF ₃ ], [ZA5667; H, F, H, H, NEt (CH ₂ ) ₂ F], [ZA5668; H, F, H, H, NEtCH ₂ CHF ₂ ], [ZA5669; H, F, H, H, NEtCH ₂ CHF ₃ ], [ZA5670; H, F, H, H, NEt ( CH ₂ ) ₃ F], [ZA5671; H, F, H, H, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA5672; H, F, H, H, NEt (CH ₂ ) ₂ CF ₃ ], [ ZA5673; H, F, H, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA5674; H, F, H, H, NEtCH ₂ Cl], [ZA5675; H, F, H, H, NEt (CH _{2) 2 Cl], [ZA5676} ; H, F, H, H, NEt (CH 2) 3 Cl], [ZA5677; H, F, H, H, NEt (CH 2) 4 Cl], [ZA5678; H , F, H, H, NEt (CH ₂ ) ₅ Cl], [ZA5679; H, F, H, H, NEtCH ₂ OMe], [ZA5680; H, F, H, H, NEt (CH ₂ ) ₂ OMe ], [ZA5681; H, F, H, H, NEt (CH ₂ ) ₃ OMe], [ZA5682; H, F, H, H, NEt (CH ₂ ) ₄ OMe], [ZA5683; H, F, H , H, NEtCH ₂ OEt], [ZA5684; H, F, H, H, NEt (CH ₂ ) ₂ OEt], [ZA5685; H, F, H, H, NEt (CH ₂ ) ₃ OEt], [ZA5686 ; H, F, H, H, NEtCH ₂ OPr], [ZA5687; H, F, H, H, NEt (CH ₂ ) ₂ OPr], [ZA5688; H, F, H, H, NEt (CH ₂ ) ₃ OPr], [ZA5689; H, F, H, H, NEtCH ₂ CN], [ZA5690; H, F, H, H, NEt (CH ₂ ) ₂ CN], [ZA5691; H, F, H, H , NEt (CH ₂ ) ₃ CN], [ZA5692; H, F, H, H, NEt (CH ₂ ) ₄ CN], [ZA5693; H, F, H, H, NEt (CH ₂ ) ₅ CN], [ZA5694; H, F, H, H, NEtCH ₂ CH = CH ₂ ], [ZA5695; H, F, H, H, NEtCH ₂ C≡CH], [ZA5696; H, F, H, H, NEtCH ₂ C≡CCH ₃ ], [ZA5697; H, F, H, H, NEtCH ₂ Ph], [ZA5698; H, F, H, H, NEtCH ₂ (2-Py)], [ZA5699; H, F, H, H, NEtCH ₂ (3-Py)], [ZA5700; H, F, H, H, NEtCH ₂ (4-Py)] , [ZA5701; H, F, H, H, NEt (CH ₂ ) ₂ Ph], [ZA5702; H, F, H, H, NEt (CH ₂ ) ₂ (2-Py)], [ZA5703; H, F, H, H, NEt (CH ₂ ) ₂ (3-Py)], [ZA5704; H, F, H, H, NEt (CH ₂ ) ₂ (4-Py)], [ZA5705; H, F, H, H, NEtPh], [ZA5706; H, F, H, H, NEt (2-Py)], [ZA5707; H, F, H, H, NEt (3-Py)], [ZA5708; H, F, H, H, NEt (4-Py)], [ZA5709; H, F, H, H, Pyr], [ZA5710; H, F, H, H, Pip], [ZA5711; H, F, H , H, Mor], [ZA5712; H, F, H, H, OMe], [ZA5713; H, F, H, H, OEt], [ZA5714; H, F, H, H, OPr], [ZA5715 ; H, F, H, H, OBu], [ZA5716; H, F, H, H, OPen], [ZA5717; H, F, H, H, OHex], [ZA5718; H, F, H, H , O (i-Pr)], [ZA5719; H, F, H, H, O (i-Bu)], [ZA5720; H, F, H, H, O (c-Pr)], [ZA5721; H, F, H, H, O (c-Bu)], [ZA5722; H, F, H, H, O (c-Pen)], [ZA5723; H, F, H, H, O (c- Hex)], [ZA5724; H, F, H, H, OCH ₂ (c-Pr)], [ZA5725; H, F, H, H, OCH ₂ (c-Bu)], [ZA5726; H, F , H, H, OCH ₂ (c-Pen)], [ZA5727; H, F, H, H, OCH ₂ (c-Hex)], [ZA5728; H, F, H, H, OCH ₂ F], [ZA5729; H, F, H, H, OCHF ₂ ], [ZA5730; H, F, H, H, OCF ₃ ], [ZA5731; H, F, H, H, O (CH ₂ ) ₂ F], [ZA5732; H, F, H, H, OCH ₂ CHF ₂ ], [ZA5733; H, F, H, H, OCH ₂ CHF ₃ ], [ZA5734; H, F, H, H, O (CH ₂ ) ₃ F], [ZA5735; H, F , H, H, O (CH ₂ ) ₂ CHF ₂ ], [ZA5736; H, F, H, H, O (CH ₂ ) ₂ CF ₃ ], [ZA5737; H, F, H, H, OCH ₂ CH (CF ₃ ) ₂ ], [ZA5738; H, F, H, H, OCH ₂ Cl], [ZA5739; H, F, H, H, O (CH ₂ ) ₂ Cl], [ZA5740; H, F, H, H, O (CH ₂ ) ₃ Cl], [ZA5741; H, F, H, H, O (CH ₂ ) ₄ Cl], [ZA5742; H, F, H, H, O (CH ₂ ) ₅ Cl], [ZA5743; H, F, H, H, OCH ₂ OMe], [ZA5744; H, F, H, H, O (CH ₂ ) ₂ OMe], [ZA5745; H, F, H, H, O (CH ₂ ) ₃ OMe], [ZA5746; H, F, H, H, O (CH ₂ ) ₄ OMe], [ZA5747; H, F, H, H, OCH ₂ OEt], [ZA5748; H, F, H, H, O (CH ₂ ) ₂ OEt], [ZA5749; H, F, H, H, O (CH ₂ ) ₃
OEt], [ZA5750; H, F, H, H, OCH ₂ OPr],

[ZA5751; H, F, H, H, O (CH ₂ ) ₂ OPr], [ZA5752; H, F, H, H, O (CH ₂ ) ₃ OPr], [ZA5753; H, F, H, H , OCH ₂ CN], [ZA5754; H, F, H, H, O (CH ₂ ) ₂ CN], [ZA5755; H, F, H, H, O (CH ₂ ) ₃ CN], [ZA5756; H , F, H, H, O (CH ₂ ) ₄ CN], [ZA5757; H, F, H, H, O (CH ₂ ) ₅ CN], [ZA5758; H, F, H, H, OCH ₂ CH = CH ₂ ], [ZA5759; H, F, H, H, OCH ₂ C≡CH], [ZA5760; H, F, H, H, OCH ₂ C≡CCH ₃ ], [ZA5761; H, F, H , H, OCH ₂ Ph], [ZA5762; H, F, H, H, OCH ₂ (2-Py)], [ZA5763; H, F, H, H, OCH ₂ (3-Py)], [ZA5764 ; H, F, H, H, OCH ₂ (4-Py)], [ZA5765; H, F, H, H, O (CH ₂ ) ₂ Ph], [ZA5766; H, F, H, H, O (CH ₂ ) ₂ (2-Py)], [ZA5767; H, F, H, H, O (CH ₂ ) ₂ (3-Py)], [ZA5768; H, F, H, H, O (CH ₂ ) ₂ (4-Py)], [ZA5769; H, F, H, H, OPh], [ZA5770; H, F, H, H, O (2-Py)], [ZA5771; H, F, H, H, O (3-Py)], [ZA5772; H, F, H, H, O (4-Py)], [ZA5773; H, F, H, H, Me], [ZA5774; H, F, H, H, Et], [ZA5775; H, F, H, H, Pr], [ZA5776; H, F, H, H, Bu], [ZA5777; H, F, H, H, Pen] , [ZA5778; H, F, H, H, Hex], [ZA5779; H, F, H, H, (i-Pr)], [ZA5780; H, F, H, H, (i-Bu)] , [ZA5781; H, F, H, H, (c-Pr)], [ZA5782; H, F, H, H, (c-Bu)], [ZA5783; H, F, H, H, (c -Pen)], [ZA5784; H, F, H, H, (c-Hex)], [ZA5785; H, F, H, H, CH ₂ (c-Pr)], [ZA5786; H, F, H, H, CH ₂ (c-Bu)], [ZA5787; H, F, H, H, CH ₂ (c-Pen)], [ZA5788; H, F, H, H, CH ₂ (c-Hex)], [ZA5789; H, F, H, H, CH ₂ F], [ZA5790; H, F, H, H, CHF ₂ ], [ZA5791; H, F, H, H, CF ₃ ], [ZA5792; H, F, H, H, (CH ₂ ) ₂ F], [ZA5793; H, F , H, H, CH ₂ CHF ₂ ], [ZA5794; H, F, H, H, CH ₂ CHF ₃ ], [ZA5795; H, F, H, H, (CH ₂ ) ₃ F], [ZA5796; H, F, H, H, (CH ₂ ) ₂ CHF ₂ ], [ZA5797; H, F, H, H, (CH ₂ ) ₂ CF ₃ ], [ZA5798; H, F, H, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA5799; H, F, H, H, CH ₂ Cl], [ZA5800; H, F, H, H, (CH ₂ ) ₂ Cl], [ZA5801; H, F, H, H, (CH ₂ ) ₃ Cl], [ZA5802; H, F, H, H, (CH ₂ ) ₄ Cl], [ZA5803; H, F, H, H, (CH ₂ ) ₅ Cl], [ZA5804; H, F, H, H, CH ₂ OMe], [ZA5805; H, F, H, H, (CH ₂ ) ₂ OMe], [ZA5806; H, F, H, H, (CH ₂ ) ₃ OMe], [ZA5807; H, F, H, H, (CH ₂ ) ₄ OMe], [ZA5808; H, F, H, H, CH ₂ OEt], [ZA5809; H, F, H, H, (CH ₂ ) ₂ OEt], [ZA5810; H, F, H, H, (CH ₂ ) ₃ OEt], [ZA5811; H, F, H, H, CH ₂ OPr], [ZA5812; H, F, H, H, (CH ₂ ) ₂ OPr], [ZA5813; H, F, H, H, (CH ₂ ) ₃ OPr], [ZA5814; H, F, H, H, CH ₂ CN], [ZA5815; H, F, H, H, (CH ₂ ) ₂ CN], [ZA5816; H, F, H, H, (CH ₂ ) ₃ CN], [ZA5817; H, F, H, H, (CH ₂ ) ₄ CN], [ZA5818; H, F, H, H, (CH ₂ ) ₅ CN], [ZA5819; H, F, H, H, CH ₂ CH = CH ₂ ], [ZA5820; H, F, H , H, CH ₂ C≡CH], [ZA5821; H, F, H, H, CH ₂ C ≡CCH ₃ ], [ZA5822; H, F, H, H, CH ₂ Ph], [ZA5823; H, F, H, H, CH ₂ (2-Py)], [ZA5824; H, F, H, H, CH ₂ (3-Py)], [ZA5825; H, F, H, H, CH ₂ (4-Py)], [ZA5826; H, F, H, H, (CH ₂ ) ₂ Ph], [ZA5827; H, F, H, H, (CH ₂ ) ₂ (2-Py)], [ZA5828; H, F, H, H, (CH ₂ ) ₂ (3-Py)], [ZA5829; H , F, H, H, (CH ₂ ) ₂ (4-Py)], [ZA5830; H, F, H, H, Ph], [ZA5831; H, F, H, H, 2-Py], [ ZA5832; H, F, H, H, 3-Py], [ZA5833; H, F, H, H, 4-Py], [ZA5834; H, F, Me, H, NHMe], [ZA5835; H, F, Me, H, NHEt], [ZA5836; H, F, Me, H, NHPr], [ZA5837; H, F, Me, H, NHBu], [ZA5838; H, F, Me, H, NHPen] , [ZA5839; H, F, Me, H, NHHex], [ZA5840; H, F, Me, H, NH (i-Pr)], [ZA5841; H, F, Me, H, NH (i-Bu )], [ZA5842; H, F, Me, H, NH (c-Pr)], [ZA5843; H, F, Me, H, NH (c-Bu)], [ZA5844; H, F, Me, H, NH (c-Pen)], [ZA5845; H, F, Me, H, NH (c-Hex)], [ZA5846; H, F, Me, H, NHCH ₂ (c-Pr)], [ ZA5847; H, F, Me, H, NHCH ₂ (c-Bu)], [ZA5848; H, F, Me, H, NHCH ₂ (c-Pen)], [ZA5849; H, F, Me, H, NHCH ₂ (c-Hex)], [ZA5850; H, F, Me, H, NHCH ₂ F], [ZA5851; H, F, Me, H, NHCHF ₂ ], [ZA5852; H, F, Me, H , NHCF ₃ ], [ZA5853; H, F, Me, H, NH (CH ₂ ) ₂ F], [ZA5854; H, F, Me, H, NHCH ₂ CHF ₂ ], [ZA5855; H, F, Me , H, NHCH ₂ CHF ₃ ], [ZA5856; H, F, Me, H, NH (CH ₂ ) ₃ F], [ZA5857; H, F, Me, H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA5858; H, F, Me, H, NH (CH ₂ ) ₂ CF ₃ ], [ZA5859; H, F, Me, H, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA5860; H, F, Me, H, NHCH ₂ Cl], [ZA5861; H, F, Me, H, NH (CH ₂ ) ₂ Cl], [ZA5862; H, F, Me, H, NH (CH ₂ ) ₃ Cl], [ZA5863; H, F, Me, H, NH (CH ₂ ) ₄ Cl], [ZA5864; H, F, Me, H, NH (CH ₂ ) ₅ Cl], [ZA5865 ; H, F, Me, H, NHCH ₂ OMe], [ZA5866; H, F, Me, H, NH (CH ₂ ) ₂ OMe], [ZA5867; H, F, Me, H, NH (CH ₂ ) ₃ OMe], [ZA5868; H, F, Me, H, NH (CH ₂ ) ₄ OMe], [ZA5869; H, F, Me, H, NHCH ₂ OEt], [ZA5870; H, F, Me, H , NH (CH ₂ ) ₂ OEt], [ZA5871; H, F, Me, H, NH (CH ₂ ) ₃ OEt], [ZA5872; H, F, Me, H, NHCH ₂ OPr], [ZA5873; H , F, Me, H, NH (CH ₂ ) ₂ OPr], [ZA5874; H, F, Me, H, NH (CH ₂ ) ₃ OPr], [ZA5875; H, F, Me, H, NHCH ₂ CN ], [ZA5876; H, F, Me, H, NH (CH ₂ ) ₂ CN], [ZA5877; H, F, Me, H, NH (CH ₂ ) ₃ CN], [ZA5878; H, F, Me , H, NH (CH ₂ ) ₄ CN], [ZA5879; H, F, Me, H, NH (CH ₂ ) ₅ CN], [ZA5880; H, F, Me, H, NHCH ₂ CH = CH ₂ ] , [ZA5881; H, F, Me, H, NHCH ₂ C≡CH], [ZA5882; H, F, Me, H, NHCH ₂ C≡CCH ₃ ], [ZA5883; H, F, Me, H, NHCH ₂ Ph], [ZA5884; H, F, Me, H, NHCH ₂ (2-Py)], [ZA5885; H, F, Me, H, NHCH ₂ (3-Py)], [ZA5886; H, F , Me, H, NHCH ₂ (4-Py)], [ZA5887; H, F, Me, H, NH (CH ₂ ) ₂ Ph], [Z A5888; H, F, Me, H, NH (CH ₂ ) ₂ (2-Py)], [ZA5889; H, F, Me, H, NH (CH ₂ ) ₂ (3-Py)], [ZA5890; H, F, Me, H, NH (CH ₂ ) ₂ (4-Py)], [ZA5891; H, F, Me, H, NHPh], [ZA5892; H, F, Me, H, NH (2- Py)], [ZA5893; H, F, Me, H, NH (3-Py)], [ZA5894; H, F, Me, H, NH (4-Py)], [ZA5895; H, F, Me , H, NMe ₂ ], [ZA5896; H, F, Me, H, NMeEt], [ZA5897; H, F, Me, H, NMePr], [ZA5898; H, F, Me, H, NMeBu], [ ZA5899; H, F, Me, H, NMePen], [ZA5900; H, F, Me, H, NMeHex], [ZA5901; H, F, Me, H, NMe (i-Pr)], [ZA5902; H , F, Me, H, NMe (i-Bu)], [ZA5903; H, F, Me, H, NMe (c-Pr)], [ZA5904; H, F, Me, H, NMe (c-Bu )], [ZA5905; H, F, Me, H, NMe (c-Pen)], [ZA5906; H, F, Me, H, NMe (c-Hex)], [ZA5907; H, F, Me, H, NMeCH ₂ (c-Pr)], [ZA5908; H, F, Me, H, NMeCH ₂ (c-Bu)], [ZA5909; H, F, Me, H, NMeCH ₂ (c-Pen)] , [ZA5910; H, F, Me, H, NMeCH ₂ (c-Hex)], [ZA5911; H, F, Me, H, NMeCH ₂ F], [ZA5912; H, F, Me, H, NMeCHF ₂ ], [ZA5913; H, F, Me, H, NMeCF ₃ ], [ZA5914; H, F, Me, H, NMe (CH ₂ ) ₂ F], [ZA5915; H, F, Me, H, NMeCH ₂ CHF ₂ ], [ZA5916; H, F, Me, H, NMeCH ₂ CHF ₃ ], [ZA5917; H, F, Me, H, NMe (CH ₂ ) ₃ F], [ZA5918; H, F, Me, H, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA5919; H, F, Me, H, NMe (CH ₂ ) ₂ CF ₃ ], [ZA5920; H, F, Me, H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA5921 ; H, F, Me, H, NMeCH ₂ Cl], [ZA5922; H, F, Me, H, NMe (CH ₂ ) ₂ Cl], [ZA5923; H, F, Me, H, NMe (CH ₂ ) ₃ Cl], [ZA5924; H, F, Me, H, NMe (CH ₂ ) ₄ Cl], [ZA5925; H, F, Me, H, NMe (CH ₂ ) ₅ Cl], [ZA5926; H, F , Me, H, NMeCH ₂ OMe], [ZA5927; H, F, Me, H, NMe (CH ₂ ) ₂ OMe], [ZA5928; H, F, Me, H, NMe (CH ₂ ) ₃ OMe], [ZA5929; H, F, Me, H, NMe (CH ₂ ) ₄ OMe], [ZA5930; H, F, Me, H, NMeCH ₂ OEt], [ZA5931; H, F, Me, H, NMe (CH ₂ ) ₂ OEt], [ZA5932; H, F, Me, H, NMe (CH ₂ ) ₃ OEt], [ZA5933; H, F, Me, H, NMeCH ₂ OPr], [ZA5934; H, F, Me , H, NMe (CH ₂ ) ₂ OPr], [ZA5935; H, F, Me, H, NMe (CH ₂ ) ₃ OPr], [ZA5936; H, F, Me, H, NMeCH ₂ CN], [ZA5937 ; H, F, Me, H, NMe (CH ₂ ) ₂ CN], [ZA5938; H, F, Me, H, NMe (CH ₂ ) ₃ CN], [ZA5939; H, F, Me, H, NMe (CH ₂ ) ₄ CN], [ZA5940; H, F, Me, H, NMe (CH ₂ ) ₅ CN], [ZA5941; H, F, Me, H, NMeCH ₂ CH = CH ₂ ], [ZA5942; H, F, Me, H, NMeCH ₂ C≡CH], [ZA5943; H, F, Me, H, NMeCH ₂ C≡CCH ₃ ], [ZA5944; H, F, Me, H, NMeCH ₂ Ph], [ZA5945; H, F, Me, H, NMeCH ₂ (2-Py)], [ZA5946; H, F, Me, H, NMeCH ₂ (3-Py)], [ZA5947; H, F, Me, H , NMeCH ₂ (4-Py)], [ZA5948; H, F, Me, H, NMe (CH ₂ ) ₂ Ph], [ZA5949; H, F, Me, H, NMe (CH ₂ ) ₂ (2- Py)], [ZA5950; H, F, Me, H, NMe (CH ₂ ) ₂ (3-Py)] , [ZA5951; H, F, Me, H, NMe (CH ₂ ) ₂ (4-Py)], [ZA5952; H, F, Me, H, NMePh], [ZA5953; H, F, Me, H, NMe (2-Py)], [ZA5954; H, F, Me, H, NMe (3-Py)], [ZA5955; H, F, Me, H, NMe (4-Py)], [ZA5956; H , F, Me, H, NEt ₂ ], [ZA5957; H, F, Me, H, NEtPr], [ZA5958; H, F, Me, H, NEtBu], [ZA5959; H, F, Me, H, NEtPen], [ZA5960; H, F, Me, H, NEtHex], [ZA5961; H, F, Me, H, NEt (i-Pr)], [ZA5962; H, F, Me, H, NEt (i -Bu)], [ZA5963; H, F, Me, H, NEt (c-Pr)], [ZA5964; H, F, Me, H, NEt (c-Bu)], [ZA5965; H, F, Me, H, NEt (c-Pen)], [ZA5966; H, F, Me, H, NEt (c-Hex)], [ZA5967; H, F, Me, H, NEtCH ₂ (c-Pr)] , [ZA5968; H, F, Me, H, NEtCH ₂ (c-Bu)], [ZA5969; H, F, Me, H, NEtCH ₂ (c-Pen)], [ZA5970; H, F, Me, H, NEtCH ₂ (c-Hex)], [ZA5971; H, F, Me, H, NEtCH ₂ F], [ZA5972; H, F, Me, H, NEtCHF ₂ ], [ZA5973; H, F, Me , H, NEtCF ₃ ], [ZA5974; H, F, Me, H, NEt (CH ₂ ) ₂ F], [ZA5975; H, F, Me, H, NEtCH ₂ CHF ₂ ], [ZA5976; H, F , Me, H, NEtCH ₂ CHF ₃ ], [ZA5977; H, F, Me, H, NEt (CH ₂ ) ₃ F], [ZA5978; H, F, Me, H, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA5979; H, F, Me, H, NEt (CH ₂ ) ₂ CF ₃ ], [ZA5980; H, F, Me, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA5981; H, F , Me, H, NEtCH ₂ Cl], [ZA5982; H, F, Me, H, NEt (CH ₂ ) ₂ Cl], [ZA5983; H, F, Me, H, NEt (CH ₂ ) ₃ Cl], [ZA5984; H, F, Me, H, NEt (CH ₂ ) ₄ Cl], [ZA5985; H, F, Me, H, NEt (CH ₂ ) ₅ Cl], [ZA5986; H, F, Me, H , NEtCH ₂ OMe], [ZA5987; H, F, Me, H, NEt (CH ₂ ) ₂ OMe], [ZA5988; H, F, Me, H, NEt (CH ₂ ) ₃ OMe], [ZA5989; H , F, Me, H, NEt (CH ₂ ) ₄ OMe], [ZA5990; H, F, Me, H, NEtCH ₂ OEt], [ZA5991; H, F, Me, H, NEt (CH ₂ ) ₂ OEt ], [ZA5992; H, F, Me, H, NEt (CH ₂ ) ₃ OEt], [ZA5993; H, F, Me, H, NEtCH ₂ OPr], [ZA5994; H, F, Me, H, NEt (CH ₂ ) ₂ OPr], [ZA5995; H, F, Me, H, NEt (CH ₂ ) ₃ OPr], [ZA5996; H, F, Me, H, NEtCH ₂ CN], [ZA5997; H, F , Me, H,
NEt (CH ₂ ) ₂ CN], [ZA5998; H, F, Me, H, NEt (CH ₂ ) ₃ CN], [ZA5999; H, F, Me, H, NEt (CH ₂ ) ₄ CN], [ ZA6000; H, F, Me, H, NEt (CH ₂ ) ₅ CN],

[ZA6001; H, F, Me, H, NEtCH ₂ CH = CH ₂ ], [ZA6002; H, F, Me, H, NEtCH ₂ C≡CH], [ZA6003; H, F, Me, H, NEtCH ₂ C≡CCH ₃ ], [ZA6004; H, F, Me, H, NEtCH ₂ Ph], [ZA6005; H, F, Me, H, NEtCH ₂ (2-Py)], [ZA6006; H, F, Me , H, NEtCH ₂ (3-Py)], [ZA6007; H, F, Me, H, NEtCH ₂ (4-Py)], [ZA6008; H, F, Me, H, NEt (CH ₂ ) ₂ Ph ], [ZA6009; H, F, Me, H, NEt (CH ₂ ) ₂ (2-Py)], [ZA6010; H, F, Me, H, NEt (CH ₂ ) ₂ (3-Py)], [ZA6011; H, F, Me, H, NEt (CH ₂ ) ₂ (4-Py)], [ZA6012; H, F, Me, H, NEtPh], [ZA6013; H, F, Me, H, NEt (2-Py)], [ZA6014; H, F, Me, H, NEt (3-Py)], [ZA6015; H, F, Me, H, NEt (4-Py)], [ZA6016; H, F, Me, H, Pyr], [ZA6017; H, F, Me, H, Pip], [ZA6018; H, F, Me, H, Mor], [ZA6019; H, F, Me, H, OMe] , [ZA6020; H, F, Me, H, OEt], [ZA6021; H, F, Me, H, OPr], [ZA6022; H, F, Me, H, OBu], [ZA6023; H, F, Me, H, OPen], [ZA6024; H, F, Me, H, OHex], [ZA6025; H, F, Me, H, O (i-Pr)], [ZA6026; H, F, Me, H , O (i-Bu)], [ZA6027; H, F, Me, H, O (c-Pr)], [ZA6028; H, F, Me, H, O (c-Bu)], [ZA6029; H, F, Me, H, O (c-Pen)], [ZA6030; H, F, Me, H, O (c-Hex)], [ZA6031; H, F, Me, H, OCH ₂ (c -Pr)], [ZA6032; H, F, Me, H, OCH ₂ (c-Bu)], [ZA6033; H, F, Me, H, OCH ₂ (c-Pen)], [ZA6034; H, F, Me, H, OCH ₂ (c-Hex)], [ZA6035; H, F, Me, H, OCH ₂ F], [ ZA6036; H, F, Me, H, OCHF ₂ ], [ZA6037; H, F, Me, H, OCF ₃ ], [ZA6038; H, F, Me, H, O (CH ₂ ) ₂ F], [ ZA6039; H, F, Me, H, OCH ₂ CHF ₂ ], [ZA6040; H, F, Me, H, OCH ₂ CHF ₃ ], [ZA6041; H, F, Me, H, O (CH ₂ ) ₃ F], [ZA6042; H, F, Me, H, O (CH ₂ ) ₂ CHF ₂ ], [ZA6043; H, F, Me, H, O (CH ₂ ) ₂ CF ₃ ], [ZA6044; H, F, Me, H, OCH ₂ CH (CF ₃ ) ₂ ], [ZA6045; H, F, Me, H, OCH ₂ Cl], [ZA6046; H, F, Me, H, O (CH ₂ ) ₂ Cl ], [ZA6047; H, F, Me, H, O (CH ₂ ) ₃ Cl], [ZA6048; H, F, Me, H, O (CH ₂ ) ₄ Cl], [ZA6049; H, F, Me , H, O (CH ₂ ) ₅ Cl], [ZA6050; H, F, Me, H, OCH ₂ OMe], [ZA6051; H, F, Me, H, O (CH ₂ ) ₂ OMe], [ZA6052 ; H, F, Me, H, O (CH ₂ ) ₃ OMe], [ZA6053; H, F, Me, H, O (CH ₂ ) ₄ OMe], [ZA6054; H, F, Me, H, OCH ₂ OEt], [ZA6055; H, F, Me, H, O (CH ₂ ) ₂ OEt], [ZA6056; H, F, Me, H, O (CH ₂ ) ₃ OEt], [ZA6057; H, F , Me, H, OCH ₂ OPr], [ZA6058; H, F, Me, H, O (CH ₂ ) ₂ OPr], [ZA6059; H, F, Me, H, O (CH ₂ ) ₃ OPr], [ZA6060; H, F, Me, H, OCH ₂ CN], [ZA6061; H, F, Me, H, O (CH ₂ ) ₂ CN], [ZA6062; H, F, Me, H, O (CH _{2) 3 CN], [ZA6063} ; H, F, Me, H, O (CH 2) 4 CN], [ZA6064; H, F, Me, H, O (CH 2) 5 CN], [ZA6065; H , F, Me, H, OCH ₂ CH = CH ₂ ], [ZA6066; H, F, Me, H, OCH ₂ C≡CH], [ZA6067; H, F, Me, H, OCH ₂ C≡CC H ₃ ], [ZA6068; H, F, Me, H, OCH ₂ Ph], [ZA6069; H, F, Me, H, OCH ₂ (2-Py)], [ZA6070; H, F, Me, H , OCH ₂ (3-Py)], [ZA6071; H, F, Me, H, OCH ₂ (4-Py)], [ZA6072; H, F, Me, H, O (CH ₂ ) ₂ Ph], [ZA6073; H, F, Me, H, O (CH ₂ ) ₂ (2-Py)], [ZA6074; H, F, Me, H, O (CH ₂ ) ₂ (3-Py)], [ZA6075 ; H, F, Me, H, O (CH ₂ ) ₂ (4-Py)], [ZA6076; H, F, Me, H, OPh], [ZA6077; H, F, Me, H, O (2 -Py)], [ZA6078; H, F, Me, H, O (3-Py)], [ZA6079; H, F, Me, H, O (4-Py)], [ZA6080; H, F, Me, H, Me], [ZA6081; H, F, Me, H, Et], [ZA6082; H, F, Me, H, Pr], [ZA6083; H, F, Me, H, Bu], [ ZA6084; H, F, Me, H, Pen], [ZA6085; H, F, Me, H, Hex], [ZA6086; H, F, Me, H, (i-Pr)], [ZA6087; H, F, Me, H, (i-Bu)], [ZA6088; H, F, Me, H, (c-Pr)], [ZA6089; H, F, Me, H, (c-Bu)], [ ZA6090; H, F, Me, H, (c-Pen)], [ZA6091; H, F, Me, H, (c-Hex)], [ZA6092; H, F, Me, H, CH ₂ (c -Pr)], [ZA6093; H, F, Me, H, CH ₂ (c-Bu)], [ZA6094; H, F, Me, H, CH ₂ (c-Pen)], [ZA6095; H, F, Me, H, CH ₂ (c-Hex)], [ZA6096; H, F, Me, H, CH ₂ F], [ZA6097; H, F, Me, H, CHF ₂ ], [ZA6098; H , F, Me, H, CF ₃ ], [ZA6099; H, F, Me, H, (CH ₂ ) ₂ F], [ZA6100; H, F, Me, H, CH ₂ CHF ₂ ], [ZA6101; H, F, Me, H, CH ₂ CHF ₃ ], [ZA6102; H, F, Me, H, (CH ₂ ) ₃ F], [ZA6103; H, F, Me, H, (CH ₂ ) ₂ CHF ₂ ], [ZA 6104; H, F, Me, H, (CH ₂ ) ₂ CF ₃ ], [ZA6105; H, F, Me, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA6106; H, F, Me, H , CH ₂ Cl], [ZA6107; H, F, Me, H, (CH ₂ ) ₂ Cl], [ZA6108; H, F, Me, H, (CH ₂ ) ₃ Cl], [ZA6109; H, F , Me, H, (CH ₂ ) ₄ Cl], [ZA6110; H, F, Me, H, (CH ₂ ) ₅ Cl], [ZA6111; H, F, Me, H, CH ₂ OMe], [ZA6112 ; H, F, Me, H, (CH ₂ ) ₂ OMe], [ZA6113; H, F, Me, H, (CH ₂ ) ₃ OMe], [ZA6114; H, F, Me, H, (CH ₂ ) ₄ OMe], [ZA6115; H, F, Me, H, CH ₂ OEt], [ZA6116; H, F, Me, H, (CH ₂ ) ₂ OEt], [ZA6117; H, F, Me, H , (CH ₂ ) ₃ OEt], [ZA6118; H, F, Me, H, CH ₂ OPr], [ZA6119; H, F, Me, H, (CH ₂ ) ₂ OPr], [ZA6120; H, F , Me, H, (CH ₂ ) ₃ OPr], [ZA6121; H, F, Me, H, CH ₂ CN], [ZA6122; H, F, Me, H, (CH ₂ ) ₂ CN], [ZA6123 ; H, F, Me, H, (CH ₂ ) ₃ CN], [ZA6124; H, F, Me, H, (CH ₂ ) ₄ CN], [ZA6125; H, F, Me, H, (CH ₂ ) ₅ CN], [ZA6126; H, F, Me, H, CH ₂ CH = CH ₂ ], [ZA6127; H, F, Me, H, CH ₂ C≡CH], [ZA6128; H, F, Me , H, CH ₂ C≡CCH ₃ ], [ZA6129; H, F, Me, H, CH ₂ Ph], [ZA6130; H, F, Me, H, CH ₂ (2-Py)], [ZA6131; H, F, Me, H, CH ₂ (3-Py)], [ZA6132; H, F, Me, H, CH ₂ (4-Py)], [ZA6133; H, F, Me, H, (CH ₂ ) ₂ Ph], [ZA6134; H, F, Me, H, (CH ₂ ) ₂ (2-Py)], [ZA6135; H, F, Me, H, (CH ₂ ) ₂ (3-Py) ], [ZA6136; H, F, Me, H, (CH ₂ ) ₂ (4-Py)], [ZA6137; H, F, Me, H, Ph], [ZA6138; H, F, Me, H, 2-Py], [ZA6139; H, F , Me, H, 3-Py], [ZA6140; H, F, Me, H, 4-Py], [ZA6141; H, F, Me, Me, NHMe], [ZA6142; H, F, Me, Me , NHEt], [ZA6143; H, F, Me, Me, NHPr], [ZA6144; H, F, Me, Me, NHBu], [ZA6145; H, F, Me, Me, NHPen], [ZA6146; H , F, Me, Me, NHHex], [ZA6147; H, F, Me, Me, NH (i-Pr)], [ZA6148; H, F, Me, Me, NH (i-Bu)], [ZA6149 ; H, F, Me, Me, NH (c-Pr)], [ZA6150; H, F, Me, Me, NH (c-Bu)], [ZA6151; H, F, Me, Me, NH (c -Pen)], [ZA6152; H, F, Me, Me, NH (c-Hex)], [ZA6153; H, F, Me, Me, NHCH ₂ (c-Pr)], [ZA6154; H, F , Me, Me, NHCH ₂ (c-Bu)], [ZA6155; H, F, Me, Me, NHCH ₂ (c-Pen)], [ZA6156; H, F, Me, Me, NHCH ₂ (c- Hex)], [ZA6157; H, F, Me, Me, NHCH ₂ F], [ZA6158; H, F, Me, Me, NHCHF ₂ ], [ZA6159; H, F, Me, Me, NHCF ₃ ], [ZA6160; H, F, Me, Me, NH (CH ₂ ) ₂ F], [ZA6161; H, F, Me, Me, NHCH ₂ CHF ₂ ], [ZA6162; H, F, Me, Me, NHCH ₂ CHF ₃ ], [ZA6163; H, F, Me, Me, NH (CH ₂ ) ₃ F], [ZA6164; H, F, Me, Me, NH (CH ₂ ) ₂ CHF ₂ ], [ZA6165; H, F, Me, Me, NH (CH ₂ ) ₂ CF ₃ ], [ZA6166; H, F, Me, Me, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA6167; H, F, Me, Me, NHCH ₂ Cl], [ZA6168; H, F, Me, Me, NH (CH ₂ ) ₂ Cl], [ZA6169; H, F, Me, Me, NH (CH ₂ ) ₃ Cl], [ZA6170; H, F, Me , Me, NH (CH ₂ ) ₄ Cl], [ZA6171; H, F, Me, Me, NH (CH ₂ ) ₅ Cl], [ZA6172; H, F, Me, Me, NHCH ₂ OMe], [ZA6173 ; H, F, Me, Me, NH (CH ₂ ) ₂ OMe], [ZA6174; H, F, Me, Me, NH (CH ₂ ) ₃ OMe], [ZA6175; H, F, Me, Me, NH (CH ₂ ) ₄ OMe], [ZA6176; H, F, Me, Me, NHCH ₂ OEt], [ZA6177; H, F, Me, Me, NH (CH ₂ ) ₂ OEt], [ZA6178; H, F , Me, Me, NH (CH ₂ ) ₃ OEt], [ZA6179; H, F, Me, Me, NHCH ₂ OPr], [ZA6180; H, F, Me, Me, NH (CH ₂ ) ₂ OPr], [ZA6181; H, F, Me, Me, NH (CH ₂ ) ₃ OPr], [ZA6182; H, F, Me, Me, NHCH ₂ CN], [ZA6183; H, F, Me, Me, NH (CH _{2) 2 CN], [ZA6184} ; H, F, Me, Me, NH (CH 2) 3 CN], [ZA6185; H, F, Me, Me, NH (CH 2) 4 CN], [ZA6186; H , F, Me, Me, NH (CH ₂ ) ₅ CN], [ZA6187; H, F, Me, Me, NHCH ₂ CH = CH ₂ ], [ZA6188; H, F, Me, Me, NHCH ₂ C≡ CH], [ZA6189; H, F, Me, Me, NHCH ₂ C≡CCH ₃ ], [ZA6190; H, F, Me, Me, NHCH ₂ Ph], [ZA6191; H, F, Me, Me, NHCH ₂ (2-Py)], [ZA6192; H, F, Me, Me, NHCH ₂ (3-Py)], [ZA6193; H, F, Me, Me, NHCH ₂ (4-Py)], [ZA6194 ; H, F, Me, Me, NH (CH ₂ ) ₂ Ph], [ZA6195; H, F, Me, Me, NH (CH ₂ ) ₂ (2-Py)], [ZA6196; H, F, Me , Me, NH (CH ₂ ) ₂ (3-Py)], [ZA6197; H, F, Me, Me, NH (CH ₂ ) ₂ (4-Py)], [ZA6198; H, F, Me, Me , NHPh], [ZA6199; H, F, Me, Me, NH (2-Py)], [ZA6200; H, F, M e, Me, NH (3-Py)], [ZA6201; H, F, Me, Me, NH (4-Py)], [ZA6202; H, F, Me, Me, NMe ₂ ], [ZA6203; H , F, Me, Me, NMeEt], [ZA6204; H, F, Me, Me, NMePr], [ZA6205; H, F, Me, Me, NMeBu], [ZA6206; H, F, Me, Me, NMePen ], [ZA6207; H, F, Me, Me, NMeHex], [ZA6208; H, F, Me, Me, NMe (i-Pr)], [ZA6209; H, F, Me, Me, NMe (i- Bu)], [ZA6210; H, F, Me, Me, NMe (c-Pr)], [ZA6211; H, F, Me, Me, NMe (c-Bu)], [ZA6212; H, F, Me , Me, NMe (c-Pen)], [ZA6213; H, F, Me, Me, NMe (c-Hex)], [ZA6214; H, F, Me, Me, NMeCH ₂ (c-Pr)], [ZA6215; H, F, Me, Me, NMeCH ₂ (c-Bu)], [ZA6216; H, F, Me, Me, NMeCH ₂ (c-Pen)], [ZA6217; H, F, Me, Me , NMeCH ₂ (c-Hex)], [ZA6218; H, F, Me, Me, NMeCH ₂ F], [ZA6219; H, F, Me, Me, NMeCHF ₂ ], [ZA6220; H, F, Me, Me, NMeCF ₃ ], [ZA6221; H, F, Me, Me, NMe (CH ₂ ) ₂ F], [ZA6222; H, F, Me, Me, NMeCH ₂ CHF ₂ ], [ZA6223; H, F, Me, Me, NMeCH ₂ CHF ₃ ], [ZA6224; H, F, Me, Me, NMe (CH ₂ ) ₃ F], [ZA6225; H, F, Me, Me, NMe (CH ₂ ) ₂ CHF ₂ ] , [ZA6226; H, F, Me, Me, NMe (CH ₂ ) ₂ CF ₃ ], [ZA6227; H, F, Me, Me, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA6228; H, F, Me, Me, NMeCH ₂ Cl], [ZA6229; H, F, Me, Me, NMe (CH ₂ ) ₂ Cl], [ZA6230; H, F, Me, Me, NMe (CH ₂ ) ₃ Cl], [ ZA6231; H, F, Me, Me, NMe (CH ₂ ) ₄ Cl], [ZA6232; H, F, Me, M e, NMe (CH ₂ ) ₅ Cl], [ZA6233; H, F, Me, Me, NMeCH ₂ OMe], [ZA6234; H, F, Me, Me, NMe (CH ₂ ) ₂ OMe], [ZA6235; H, F, Me, Me, NMe (CH ₂ ) ₃ OMe], [ZA6236; H, F, Me, Me, NMe (CH ₂ ) ₄ OMe], [ZA6237; H, F, Me, Me, NMeCH ₂ OEt], [ZA6238; H, F, Me, Me, NMe (CH ₂ ) ₂ OEt], [ZA6239; H, F, Me, Me, NMe (CH ₂ ) ₃ OEt], [ZA6240; H, F, Me, Me, NMeCH ₂ OPr], [ZA6241; H, F, Me, Me, NMe (CH ₂ ) ₂ OPr], [ZA6242; H, F, Me, Me, NMe (CH ₂ ) ₃ OPr], [ ZA6243; H, F, Me, Me, NMeCH ₂ CN], [ZA6244; H, F, Me, Me, NMe (CH ₂ ) ₂ CN], [ZA6245; H, F, Me, Me, NMe (CH ₂ ) ₃ CN], [ZA6246; H, F, Me, Me, NMe (CH ₂ ) ₄ CN], [ZA6247; H, F, Me, Me, NMe (
CH ₂ ) ₅ CN], [ZA6248; H, F, Me, Me, NMeCH ₂ CH = CH ₂ ], [ZA6249; H, F, Me, Me, NMeCH ₂ C≡CH], [ZA6250; H, F , Me, Me, NMeCH ₂ C≡CCH ₃ ],

[ZA6251; H, F, Me, Me, NMeCH ₂ Ph], [ZA6252; H, F, Me, Me, NMeCH ₂ (2-Py)], [ZA6253; H, F, Me, Me, NMeCH ₂ ( 3-Py)], [ZA6254; H, F, Me, Me, NMeCH ₂ (4-Py)], [ZA6255; H, F, Me, Me, NMe (CH ₂ ) ₂ Ph], [ZA6256; H , F, Me, Me, NMe (CH ₂ ) ₂ (2-Py)], [ZA6257; H, F, Me, Me, NMe (CH ₂ ) ₂ (3-Py)], [ZA6258; H, F , Me, Me, NMe (CH ₂ ) ₂ (4-Py)], [ZA6259; H, F, Me, Me, NMePh], [ZA6260; H, F, Me, Me, NMe (2-Py)] , [ZA6261; H, F, Me, Me, NMe (3-Py)], [ZA6262; H, F, Me, Me, NMe (4-Py)], [ZA6263; H, F, Me, Me, NEt ₂ ], [ZA6264; H, F, Me, Me, NEtPr], [ZA6265; H, F, Me, Me, NEtBu], [ZA6266; H, F, Me, Me, NEtPen], [ZA6267; H , F, Me, Me, NEtHex], [ZA6268; H, F, Me, Me, NEt (i-Pr)], [ZA6269; H, F, Me, Me, NEt (i-Bu)], [ZA6270 ; H, F, Me, Me, NEt (c-Pr)], [ZA6271; H, F, Me, Me, NEt (c-Bu)], [ZA6272; H, F, Me, Me, NEt (c -Pen)], [ZA6273; H, F, Me, Me, NEt (c-Hex)], [ZA6274; H, F, Me, Me, NEtCH ₂ (c-Pr)], [ZA6275; H, F , Me, Me, NEtCH ₂ (c-Bu)], [ZA6276; H, F, Me, Me, NEtCH ₂ (c-Pen)], [ZA6277; H, F, Me, Me, NEtCH ₂ (c- Hex)], [ZA6278; H, F, Me, Me, NEtCH ₂ F], [ZA6279; H, F, Me, Me, NEtCHF ₂ ], [ZA6280; H, F, Me, Me, NEtCF ₃ ], [ZA6281; H, F, Me, Me, NEt (CH ₂ ) ₂ F], [ZA6282; H, F, Me, Me, NEtCH ₂ CHF ₂ ], [ZA6283; H, F, Me, Me, NEtCH ₂ CHF ₃ ], [ZA6284; H, F, Me, Me, NEt (CH ₂ ) ₃ F], [ZA6285; H, F, Me, Me, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA6286; H, F, Me, Me, NEt (CH ₂ ) ₂ CF ₃ ], [ZA6287; H, F, Me, Me, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA6288; H, F, Me, Me, NEtCH ₂ Cl], [ZA6289; H, F, Me, Me, NEt (CH ₂ ) ₂ Cl], [ZA6290; H, F, Me, Me, NEt (CH ₂ ) ₃ Cl], [ZA6291; H, F, Me, Me, NEt (CH ₂ ) ₄ Cl], [ZA6292; H, F, Me, Me, NEt (CH ₂ ) ₅ Cl], [ZA6293; H, F, Me, Me, NEtCH ₂ OMe], [ZA6294; H, F, Me, Me, NEt (CH ₂ ) ₂ OMe], [ZA6295; H, F, Me, Me, NEt (CH ₂ ) ₃ OMe], [ ZA6296; H, F, Me, Me, NEt (CH ₂ ) ₄ OMe], [ZA6297; H, F, Me, Me, NEtCH ₂ OEt], [ZA6298; H, F, Me, Me, NEt (CH ₂ ) ₂ OEt], [ZA6299; H, F, Me, Me, NEt (CH ₂ ) ₃ OEt], [ZA6300; H, F, Me, Me, NEtCH ₂ OPr], [ZA6301; H, F, Me, Me, NEt (CH ₂ ) ₂ OPr], [ZA6302; H, F, Me, Me, NEt (CH ₂ ) ₃ OPr], [ZA6303; H, F, Me, Me, NEtCH ₂ CN], [ZA6304; H, F, Me, Me, NEt (CH ₂ ) ₂ CN], [ZA6305; H, F, Me, Me, NEt (CH ₂ ) ₃ CN], [ZA6306; H, F, Me, Me, NEt ( CH ₂ ) ₄ CN], [ZA6307; H, F, Me, Me, NEt (CH ₂ ) ₅ CN], [ZA6308; H, F, Me, Me, NEtCH ₂ CH = CH ₂ ], [ZA6309; H , F, Me, Me, NEtCH ₂ C≡CH], [ZA6310; H, F, Me, Me, NEtCH ₂ C≡CCH ₃ ], [ZA6311; H, F, Me, Me, NEtCH ₂ Ph], [ZA6312; H, F, Me, Me, NEtCH ₂ (2-Py)], [ZA6313; H, F, Me, Me, NEtCH ₂ (3-Py)], [ZA6314; H, F, Me, Me , NEtCH ₂ (4-Py)], [ZA6315; H, F, Me, Me, NEt (CH ₂ ) ₂ Ph], [ZA6316; H, F, Me, Me, NEt (CH ₂ ) ₂ (2- Py)], [ZA6317; H, F, Me, Me, NEt (CH ₂ ) ₂ (3-Py)], [ZA6318; H, F, Me, Me, NEt (CH ₂ ) ₂ (4-Py) ], [ZA6319; H, F, Me, Me, NEtPh], [ZA6320; H, F, Me, Me, NEt (2-Py)], [ZA6321; H, F, Me, Me, NEt (3- Py)], [ZA6322; H, F, Me, Me, NEt (4-Py)], [ZA6323; H, F, Me, Me, Pyr], [ZA6324; H, F, Me, Me, Pip] , [ZA6325; H, F, Me, Me, Mor], [ZA6326; H, F, Me, Me, OMe], [ZA6327; H, F, Me, Me, OEt], [ZA6328; H, F, Me, Me, OPr], [ZA6329; H, F, Me, Me, OBu], [ZA6330; H, F, Me, Me, OPen], [ZA6331; H, F, Me, Me, OHex], [ ZA6332; H, F, Me, Me, O (i-Pr)], [ZA6333; H, F, Me, Me, O (i-Bu)], [ZA6334; H, F, Me, Me, O ( c-Pr)], [ZA6335; H, F, Me, Me, O (c-Bu)], [ZA6336; H, F, Me, Me, O (c-Pen)], [ZA6337; H, F , Me, Me, O (c-Hex)], [ZA6338; H, F, Me, Me, OCH ₂ (c-Pr)], [ZA6339; H, F, Me, Me, OCH ₂ (c-Bu )], [ZA6340; H, F, Me, Me, OCH ₂ (c-Pen)], [ZA6341; H, F, Me, Me, OCH ₂ (c-Hex)], [ZA6342; H, F, Me, Me, OCH ₂ F], [ZA6343; H, F, Me, Me, OCHF ₂ ], [ZA6344; H, F, Me, Me, OCF ₃ ], [ZA6345; H, F, Me, Me, O (CH ₂ ) ₂ F], [ZA6346; H, F, Me, Me, O CH ₂ CHF ₂ ], [ZA6347; H, F, Me, Me, OCH ₂ CHF ₃ ], [ZA6348; H, F, Me, Me, O (CH ₂ ) ₃ F], [ZA6349; H, F, Me, Me, O (CH ₂ ) ₂ CHF ₂ ], [ZA6350; H, F, Me, Me, O (CH ₂ ) ₂ CF ₃ ], [ZA6351; H, F, Me, Me, OCH ₂ CH ( CF ₃ ) ₂ ], [ZA6352; H, F, Me, Me, OCH ₂ Cl], [ZA6353; H, F, Me, Me, O (CH ₂ ) ₂ Cl], [ZA6354; H, F, Me , Me, O (CH ₂ ) ₃ Cl], [ZA6355; H, F, Me, Me, O (CH ₂ ) ₄ Cl], [ZA6356; H, F, Me, Me, O (CH ₂ ) ₅ Cl ], [ZA6357; H, F, Me, Me, OCH ₂ OMe], [ZA6358; H, F, Me, Me, O (CH ₂ ) ₂ OMe], [ZA6359; H, F, Me, Me, O (CH ₂ ) ₃ OMe], [ZA6360; H, F, Me, Me, O (CH ₂ ) ₄ OMe], [ZA6361; H, F, Me, Me, OCH ₂ OEt], [ZA6362; H, F , Me, Me, O (CH ₂ ) ₂ OEt], [ZA6363; H, F, Me, Me, O (CH ₂ ) ₃ OEt], [ZA6364; H, F, Me, Me, OCH ₂ OPr], [ZA6365; H, F, Me, Me, O (CH ₂ ) ₂ OPr], [ZA6366; H, F, Me, Me, O (CH ₂ ) ₃ OPr], [ZA6367; H, F, Me, Me , OCH ₂ CN], [ZA6368; H, F, Me, Me, O (CH ₂ ) ₂ CN], [ZA6369; H, F, Me, Me, O (CH ₂ ) ₃ CN], [ZA6370; H , F, Me, Me, O (CH ₂ ) ₄ CN], [ZA6371; H, F, Me, Me, O (CH ₂ ) ₅ CN], [ZA6372; H, F, Me, Me, OCH ₂ CH = CH ₂ ], [ZA6373; H, F, Me, Me, OCH ₂ C≡CH], [ZA6374; H, F, Me, Me, OCH ₂ C≡CCH ₃ ], [ZA6375; H, F, Me , Me, OCH ₂ Ph], [ZA6376; H, F, Me, Me, OCH ₂ (2-Py)], [ZA63 77; H, F, Me, Me, OCH ₂ (3-Py)], [ZA6378; H, F, Me, Me, OCH ₂ (4-Py)], [ZA6379; H, F, Me, Me, O (CH ₂ ) ₂ Ph], [ZA6380; H, F, Me, Me, O (CH ₂ ) ₂ (2-Py)], [ZA6381; H, F, Me, Me, O (CH ₂ ) ₂ (3-Py)], [ZA6382; H, F, Me, Me, O (CH ₂ ) ₂ (4-Py)], [ZA6383; H, F, Me, Me, OPh], [ZA6384; H, F, Me, Me, O (2-Py)], [ZA6385; H, F, Me, Me, O (3-Py)], [ZA6386; H, F, Me, Me, O (4-Py) ], [ZA6387; H, F, Me, Me, Me], [ZA6388; H, F, Me, Me, Et], [ZA6389; H, F, Me, Me, Pr], [ZA6390; H, F , Me, Me, Bu], [ZA6391; H, F, Me, Me, Pen], [ZA6392; H, F, Me, Me, Hex], [ZA6393; H, F, Me, Me, (i- Pr)], [ZA6394; H, F, Me, Me, (i-Bu)], [ZA6395; H, F, Me, Me, (c-Pr)], [ZA6396; H, F, Me, Me , (c-Bu)], [ZA6397; H, F, Me, Me, (c-Pen)], [ZA6398; H, F, Me, Me, (c-Hex)], [ZA6399; H, F , Me, Me, CH ₂ (c-Pr)], [ZA6400; H, F, Me, Me, CH ₂ (c-Bu)], [ZA6401; H, F, Me, Me, CH ₂ (c- Pen)], [ZA6402; H, F, Me, Me, CH ₂ (c-Hex)], [ZA6403; H, F, Me, Me, CH ₂ F], [ZA6404; H, F, Me, Me , CHF ₂ ], [ZA6405; H, F, Me, Me, CF ₃ ], [ZA6406; H, F, Me, Me, (CH ₂ ) ₂ F], [ZA6407; H, F, Me, Me, CH ₂ CHF ₂ ], [ZA6408; H, F, Me, Me, CH ₂ CHF ₃ ], [ZA6409; H, F, Me, Me, (CH ₂ ) ₃ F], [ZA6410; H, F, Me , Me, (CH ₂ ) ₂ CHF ₂ ], [ZA6411; H, F, Me, Me, (CH ₂ ) ₂ CF ₃ ], [ZA 6412; H, F, Me, Me, CH ₂ CH (CF ₃ ) ₂ ], [ZA6413; H, F, Me, Me, CH ₂ Cl], [ZA6414; H, F, Me, Me, (CH ₂ ) ₂ Cl], [ZA6415; H, F, Me, Me, (CH ₂ ) ₃ Cl], [ZA6416; H, F, Me, Me, (CH ₂ ) ₄ Cl], [ZA6417; H, F, Me, Me, (CH ₂ ) ₅ Cl], [ZA6418; H, F, Me, Me, CH ₂ OMe], [ZA6419; H, F, Me, Me, (CH ₂ ) ₂ OMe], [ZA6420; H, F, Me, Me, (CH ₂ ) ₃ OMe], [ZA6421; H, F, Me, Me, (CH ₂ ) ₄ OMe], [ZA6422; H, F, Me, Me, CH ₂ OEt] , [ZA6423; H, F, Me, Me, (CH ₂ ) ₂ OEt], [ZA6424; H, F, Me, Me, (CH ₂ ) ₃ OEt], [ZA6425; H, F, Me, Me, CH ₂ OPr], [ZA6426; H, F, Me, Me, (CH ₂ ) ₂ OPr], [ZA6427; H, F, Me, Me, (CH ₂ ) ₃ OPr], [ZA6428; H, F, Me, Me, CH ₂ CN], [ZA6429; H, F, Me, Me, (CH ₂ ) ₂ CN], [ZA6430; H, F, Me, Me, (CH ₂ ) ₃ CN], [ZA6431; H, F, Me, Me, (CH ₂ ) ₄ CN], [ZA6432; H, F, Me, Me, (CH ₂ ) ₅ CN], [ZA6433; H, F, Me, Me, CH ₂ CH = CH ₂ ], [ZA6434; H, F, Me, Me, CH ₂ C≡CH], [ZA6435; H, F, Me, Me, CH ₂ C≡CCH ₃ ], [ZA6436; H, F, Me, Me, CH ₂ Ph], [ZA6437; H, F, Me, Me, CH ₂ (2-Py)], [ZA6438; H, F, Me, Me, CH ₂ (3-Py)], [ZA6439; H, F, Me, Me, CH ₂ (4-Py)], [ZA6440; H, F, Me, Me, (CH ₂ ) ₂ Ph], [ZA6441; H, F, Me, Me, (CH ₂ ) ₂ (2-Py)], [ZA6442; H, F, Me, Me, (CH ₂ ) ₂ (3-Py)], [ZA6443; H, F, Me, Me, (CH ₂ ) ₂ (4-Py)], [ZA6444; H, F, Me, Me, Ph], [ZA6445; H, F, Me, Me, 2-Py], [ZA6446; H, F, Me , Me, 3-Py], [ZA6447; H, F, Me, Me, 4-Py], [ZA6448; H, F, F, H, NHMe], [ZA6449; H, F, F, H, NHEt ], [ZA6450; H, F, F, H, NHPr], [ZA6451; H, F, F, H, NHBu], [ZA6452; H, F, F, H, NHPen], [ZA6453; H, F , F, H, NHHex], [ZA6454; H, F, F, H, NH (i-Pr)], [ZA6455; H, F, F, H, NH (i-Bu)], [ZA6456; H , F, F, H, NH (c-Pr)], [ZA6457; H, F, F, H, NH (c-Bu)], [ZA6458; H, F, F, H, NH (c-Pen )], [ZA6459; H, F, F, H, NH (c-Hex)], [ZA6460; H, F, F, H, NHCH ₂ (c-Pr)], [ZA6461; H, F, F , H, NHCH ₂ (c-Bu)], [ZA6462; H, F, F, H, NHCH ₂ (c-Pen)], [ZA6463; H, F, F, H, NHCH ₂ (c-Hex) ], [ZA6464; H, F, F, H, NHCH ₂ F], [ZA6465; H, F, F, H, NHCHF ₂ ], [ZA6466; H, F, F, H, NHCF ₃ ], [ZA6467 ; H, F, F, H, NH (CH ₂ ) ₂ F], [ZA6468; H, F, F, H, NHCH ₂ CHF ₂ ], [ZA6469; H, F, F, H, NHCH ₂ CHF ₃ ], [ZA6470; H, F, F, H, NH (CH ₂ ) ₃ F], [ZA6471; H, F, F, H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA6472; H, F, F, H, NH (CH ₂ ) ₂ CF ₃ ], [ZA6473; H, F, F, H, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA6474; H, F, F, H, NHCH ₂ Cl] , [ZA6475; H, F, F, H, NH (CH ₂ ) ₂ Cl], [ZA6476; H, F, F, H, NH (CH ₂ ) ₃ Cl], [ZA6477; H, F, F, H, NH (CH ₂ ) ₄ Cl], [ZA6478; H, F, F, H, NH (CH ₂ ) ₅ Cl], [ZA647 9; H, F, F, H, NHCH ₂ OMe], [ZA6480; H, F, F, H, NH (CH ₂ ) ₂ OMe], [ZA6481; H, F, F, H, NH (CH ₂ ) ₃ OMe], [ZA6482; H, F, F, H, NH (CH ₂ ) ₄ OMe], [ZA6483; H, F, F, H, NHCH ₂ OEt], [ZA6484; H, F, F, H, NH (CH ₂ ) ₂ OEt], [ZA6485; H, F, F, H, NH (CH ₂ ) ₃ OEt], [ZA6486; H, F, F, H, NHCH ₂ OPr], [ZA6487; H, F, F, H, NH (CH ₂ ) ₂ OPr], [ZA6488; H, F, F, H, NH (CH ₂ ) ₃ OPr], [ZA6489; H, F, F, H, NHCH ₂ CN], [ZA6490; H, F, F, H, NH (CH ₂ ) ₂ CN], [ZA6491; H, F, F, H, NH (CH ₂ ) ₃ CN], [ZA6492; H, F, F, H, NH (CH ₂ ) ₄ CN], [ZA6493; H, F, F, H, NH (CH ₂ ) ₅ CN], [ZA6494; H, F, F, H, NHCH ₂ CH = CH ₂ ], [ZA6495; H, F, F, H, NHCH ₂
C≡CH], [ZA6496; H, F, F, H, NHCH ₂ C≡CCH ₃ ], [ZA6497; H, F, F, H, NHCH ₂ Ph], [ZA6498; H, F, F, H , NHCH ₂ (2-Py)], [ZA6499; H, F, F, H, NHCH ₂ (3-Py)], [ZA6500; H, F, F, H, NHCH ₂ (4-Py)],

[ZA6501; H, F, F, H, NH (CH ₂ ) ₂ Ph], [ZA6502; H, F, F, H, NH (CH ₂ ) ₂ (2-Py)], [ZA6503; H, F , F, H, NH (CH ₂ ) ₂ (3-Py)], [ZA6504; H, F, F, H, NH (CH ₂ ) ₂ (4-Py)], [ZA6505; H, F, F , H, NHPh], [ZA6506; H, F, F, H, NH (2-Py)], [ZA6507; H, F, F, H, NH (3-Py)], [ZA6508; H, F , F, H, NH (4-Py)], [ZA6509; H, F, F, H, NMe ₂ ], [ZA6510; H, F, F, H, NMeEt], [ZA6511; H, F, F , H, NMePr], [ZA6512; H, F, F, H, NMeBu], [ZA6513; H, F, F, H, NMePen], [ZA6514; H, F, F, H, NMeHex], [ZA6515 ; H, F, F, H, NMe (i-Pr)], [ZA6516; H, F, F, H, NMe (i-Bu)], [ZA6517; H, F, F, H, NMe (c -Pr)], [ZA6518; H, F, F, H, NMe (c-Bu)], [ZA6519; H, F, F, H, NMe (c-Pen)], [ZA6520; H, F, F, H, NMe (c-Hex)], [ZA6521; H, F, F, H, NMeCH ₂ (c-Pr)], [ZA6522; H, F, F, H, NMeCH ₂ (c-Bu) ], [ZA6523; H, F, F, H, NMeCH ₂ (c-Pen)], [ZA6524; H, F, F, H, NMeCH ₂ (c-Hex)], [ZA6525; H, F, F , H, NMeCH ₂ F], [ZA6526; H, F, F, H, NMeCHF ₂ ], [ZA6527; H, F, F, H, NMeCF ₃ ], [ZA6528; H, F, F, H, NMe (CH ₂ ) ₂ F], [ZA6529; H, F, F, H, NMeCH ₂ CHF ₂ ], [ZA6530; H, F, F, H, NMeCH ₂ CHF ₃ ], [ZA6531; H, F, F , H, NMe (CH ₂ ) ₃ F], [ZA6532; H, F, F, H, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA6533; H, F, F, H, NMe (CH ₂ ) ₂ CF ₃ ], [ZA6534; H, F, F, H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA653 5; H, F, F, H, NMeCH ₂ Cl], [ZA6536; H, F, F, H, NMe (CH ₂ ) ₂ Cl], [ZA6537; H, F, F, H, NMe (CH ₂ ) ₃ Cl], [ZA6538; H, F, F, H, NMe (CH ₂ ) ₄ Cl], [ZA6539; H, F, F, H, NMe (CH ₂ ) ₅ Cl], [ZA6540; H, F, F, H, NMeCH ₂ OMe], [ZA6541; H, F, F, H, NMe (CH ₂ ) ₂ OMe], [ZA6542; H, F, F, H, NMe (CH ₂ ) ₃ OMe] , [ZA6543; H, F, F, H, NMe (CH ₂ ) ₄ OMe], [ZA6544; H, F, F, H, NMeCH ₂ OEt], [ZA6545; H, F, F, H, NMe ( CH ₂ ) ₂ OEt], [ZA6546; H, F, F, H, NMe (CH ₂ ) ₃ OEt], [ZA6547; H, F, F, H, NMeCH ₂ OPr], [ZA6548; H, F, F, H, NMe (CH ₂ ) ₂ OPr], [ZA6549; H, F, F, H, NMe (CH ₂ ) ₃ OPr], [ZA6550; H, F, F, H, NMeCH ₂ CN], [ ZA6551; H, F, F, H, NMe (CH ₂ ) ₂ CN], [ZA6552; H, F, F, H, NMe (CH ₂ ) ₃ CN], [ZA6553; H, F, F, H, NMe (CH ₂ ) ₄ CN], [ZA6554; H, F, F, H, NMe (CH ₂ ) ₅ CN], [ZA6555; H, F, F, H, NMeCH ₂ CH = CH ₂ ], [ZA6556 ; H, F, F, H, NMeCH ₂ C≡CH], [ZA6557; H, F, F, H, NMeCH ₂ C≡CCH ₃ ], [ZA6558; H, F, F, H, NMeCH ₂ Ph] , [ZA6559; H, F, F, H, NMeCH ₂ (2-Py)], [ZA6560; H, F, F, H, NMeCH ₂ (3-Py)], [ZA6561; H, F, F, H, NMeCH ₂ (4-Py)], [ZA6562; H, F, F, H, NMe (CH ₂ ) ₂ Ph], [ZA6563; H, F, F, H, NMe (CH ₂ ) ₂ (2 -Py)], [ZA6564; H, F, F, H, NMe (CH ₂ ) ₂ (3-Py)], [ZA6565; H, F, F, H, NMe (CH ₂ ) ₂ (4-Py)], [ZA6566; H, F, F, H, NMePh], [ZA6567; H, F, F, H, NMe (2-Py)], [ZA6568; H, F, F, H , NMe (3-Py)], [ZA6569; H, F, F, H, NMe (4-Py)], [ZA6570; H, F, F, H, NEt ₂ ], [ZA6571; H, F, F, H, NEtPr], [ZA6572; H, F, F, H, NEtBu], [ZA6573; H, F, F, H, NEtPen], [ZA6574; H, F, F, H, NEtHex], [ ZA6575; H, F, F, H, NEt (i-Pr)], [ZA6576; H, F, F, H, NEt (i-Bu)], [ZA6577; H, F, F, H, NEt ( c-Pr)], [ZA6578; H, F, F, H, NEt (c-Bu)], [ZA6579; H, F, F, H, NEt (c-Pen)], [ZA6580; H, F , F, H, NEt (c-Hex)], [ZA6581; H, F, F, H, NEtCH ₂ (c-Pr)], [ZA6582; H, F, F, H, NEtCH ₂ (c-Bu )], [ZA6583; H, F, F, H, NEtCH ₂ (c-Pen)], [ZA6584; H, F, F, H, NEtCH ₂ (c-Hex)], [ZA6585; H, F, F, H, NEtCH ₂ F], [ZA6586; H, F, F, H, NEtCHF ₂ ], [ZA6587; H, F, F, H, NEtCF ₃ ], [ZA6588; H, F, F, H, NEt (CH ₂ ) ₂ F], [ZA6589; H, F, F, H, NEtCH ₂ CHF ₂ ], [ZA6590; H, F, F, H, NEtCH ₂ CHF ₃ ], [ZA6591; H, F, F, H, NEt (CH ₂ ) ₃ F], [ZA6592; H, F, F, H, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA6593; H, F, F, H, NEt (CH ₂ ) ₂ CF ₃ ], [ZA6594; H, F, F, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA6595; H, F, F, H, NEtCH ₂ Cl], [ZA6596; H, F, F , H, NEt (CH ₂ ) ₂ Cl], [ZA6597; H, F, F, H, NEt (CH ₂ ) ₃ Cl], [ZA6598; H, F, F, H, NEt (CH ₂ ) ₄ Cl ], [ZA6599; H, F, F, H, NEt (CH ₂ ) ₅ Cl], [ZA6600; H, F, F, H, NEtCH ₂ OMe], [ZA6601; H, F, F, H, NEt (CH ₂ ) ₂ OMe], [ZA6602; H, F, F, H, NEt (CH ₂ ) ₃ OMe], [ZA6603; H, F, F, H, NEt (CH ₂ ) ₄ OMe], [ZA6604; H, F, F, H, NEtCH ₂ OEt], [ZA6605; H, F, F, H, NEt (CH ₂ ) ₂ OEt], [ZA6606; H, F, F, H, NEt (CH ₂ ) ₃ OEt], [ZA6607; H, F, F, H, NEtCH ₂ OPr] , [ZA6608; H, F, F, H, NEt (CH ₂ ) ₂ OPr], [ZA6609; H, F, F, H, NEt (CH ₂ ) ₃ OPr], [ZA6610; H, F, F, H, NEtCH ₂ CN], [ZA6611; H, F, F, H, NEt (CH ₂ ) ₂ CN], [ZA6612; H, F, F, H, NEt (CH ₂ ) ₃ CN], [ZA6613; H, F, F, H, NEt (CH ₂ ) ₄ CN], [ZA6614; H, F, F, H, NEt (CH ₂ ) ₅ CN], [ZA6615; H, F, F, H, NEtCH ₂ CH = CH ₂ ], [ZA6616; H, F, F, H, NEtCH ₂ C≡CH], [ZA6617; H, F, F, H, NEtCH ₂ C≡CCH ₃ ], [ZA6618; H, F, F, H, NEtCH ₂ Ph], [ZA6619; H, F, F, H, NEtCH ₂ (2-Py)], [ZA6620; H, F, F, H, NEtCH ₂ (3-Py)], [ ZA6621; H, F, F, H, NEtCH ₂ (4-Py)], [ZA6622; H, F, F, H, NEt (CH ₂ ) ₂ Ph], [ZA6623; H, F, F, H, NEt (CH ₂ ) ₂ (2-Py)], [ZA6624; H, F, F, H, NEt (CH ₂ ) ₂ (3-Py)], [ZA6625; H, F, F, H, NEt ( CH ₂ ) ₂ (4-Py)], [ZA6626; H, F, F, H, NEtPh], [ZA6627; H, F, F, H, NEt (2-Py)], [ZA6628; H, F , F, H, NEt (3-Py)], [ZA6629; H, F, F, H, NEt (4-Py)], [ZA6630; H, F, F, H, Pyr], [ZA6631; H , F, F, H, Pip], [ZA6632; H, F, F, H, Mor], [ZA6633; H, F, F, H, OMe], [ZA6634; H, F, F, H, OEt], [ZA6635; H, F, F, H, OPr], [ZA6636; H, F, F, H, OBu], [ZA6637; H, F, F, H, OPen], [ZA6638; H, F, F, H, OHex] , [ZA6639; H, F, F, H, O (i-Pr)], [ZA6640; H, F, F, H, O (i-Bu)], [ZA6641; H, F, F, H, O (c-Pr)], [ZA6642; H, F, F, H, O (c-Bu)], [ZA6643; H, F, F, H, O (c-Pen)], [ZA6644; H , F, F, H, O (c-Hex)], [ZA6645; H, F, F, H, OCH ₂ (c-Pr)], [ZA6646; H, F, F, H, OCH ₂ (c -Bu)], [ZA6647; H, F, F, H, OCH ₂ (c-Pen)], [ZA6648; H, F, F, H, OCH ₂ (c-Hex)], [ZA6649; H, F, F, H, OCH ₂ F], [ZA6650; H, F, F, H, OCHF ₂ ], [ZA6651; H, F, F, H, OCF ₃ ], [ZA6652; H, F, F, H, O (CH ₂ ) ₂ F], [ZA6653; H, F, F, H, OCH ₂ CHF ₂ ], [ZA6654; H, F, F, H, OCH ₂ CHF ₃ ], [ZA6655; H, F, F, H, O (CH ₂ ) ₃ F], [ZA6656; H, F, F, H, O (CH ₂ ) ₂ CHF ₂ ], [ZA6657; H, F, F, H, O (CH _{2) 2 CF 3], [} ZA6658; H, F, F, H, OCH 2 CH (CF 3) 2], [ZA6659; H, F, F, H, OCH 2 Cl], [ZA6660; H, F , F, H, O (CH ₂ ) ₂ Cl], [ZA6661; H, F, F, H, O (CH ₂ ) ₃ Cl], [ZA6662; H, F, F, H, O (CH ₂ ) ₄ Cl], [ZA6663; H, F, F, H, O (CH ₂ ) ₅ Cl], [ZA6664; H, F, F, H, OCH ₂ OMe], [ZA6665; H, F, F, H , O (CH ₂ ) ₂ OMe], [ZA6666; H, F, F, H, O (CH ₂ ) ₃ OMe], [ZA6667; H, F, F, H, O (CH ₂ ) ₄ OMe], [ZA6668; H, F, F, H, OCH ₂ OEt], [ZA6669; H, F, F, H, O (CH ₂ ) ₂ OEt], [ZA6670; H, F, F, H, O (CH ₂ ) ₃ OEt], [ZA6671; H, F, F, H, OCH ₂ OPr], [ZA6672; H, F, F, H, O (CH ₂ ) ₂ OPr], [ZA6673; H, F, F , H, O (CH ₂ ) ₃ OPr], [ZA6674; H, F, F, H, OCH ₂ CN], [ZA6675; H, F, F, H, O (CH ₂ ) ₂ CN], [ZA6676 ; H, F, F, H, O (CH ₂ ) ₃ CN], [ZA6677; H, F, F, H, O (CH ₂ ) ₄ CN], [ZA6678; H, F, F, H, O (CH ₂ ) ₅ CN], [ZA6679; H, F, F, H, OCH ₂ CH = CH ₂ ], [ZA6680; H, F, F, H, OCH ₂ C≡CH], [ZA6681; H, F, F, H, OCH ₂ C≡CCH ₃ ], [ZA6682; H, F, F, H, OCH ₂ Ph], [ZA6683; H, F, F, H, OCH ₂ (2-Py)], [ZA6684; H, F, F, H, OCH ₂ (3-Py)], [ZA6685; H, F, F, H, OCH ₂ (4-Py)], [ZA6686; H, F, F, H , O (CH ₂ ) ₂ Ph], [ZA6687; H, F, F, H, O (CH ₂ ) ₂ (2-Py)], [ZA6688; H, F, F, H, O (CH ₂ ) ₂ (3-Py)], [ZA6689; H, F, F, H, O (CH ₂ ) ₂ (4-Py)], [ZA6690; H, F, F, H, OPh], [ZA6691; H , F, F, H, O (2-Py)], [ZA6692; H, F, F, H, O (3-Py)], [ZA6693; H, F, F, H, O (4-Py )], [ZA6694; H, F, F, H, Me], [ZA6695; H, F, F, H, Et], [ZA6696; H, F, F, H, Pr], [ZA6697; H, F, F, H, Bu], [ZA6698; H, F, F, H, Pen], [ZA6699; H, F, F, H, Hex], [ZA6700; H, F, F, H, (i -Pr)], [ZA6701; H, F, F, H, (i-Bu)], [ZA6702; H, F, F, H, (c-Pr)], [ZA6703; H, F, F, H, (c-Bu)], [ZA670 4; H, F, F, H, (c-Pen)], [ZA6705; H, F, F, H, (c-Hex)], [ZA6706; H, F, F, H, CH ₂ (c -Pr)], [ZA6707; H, F, F, H, CH ₂ (c-Bu)], [ZA6708; H, F, F, H, CH ₂ (c-Pen)], [ZA6709; H, F, F, H, CH ₂ (c-Hex)], [ZA6710; H, F, F, H, CH ₂ F], [ZA6711; H, F, F, H, CHF ₂ ], [ZA6712; H , F, F, H, CF ₃ ], [ZA6713; H, F, F, H, (CH ₂ ) ₂ F], [ZA6714; H, F, F, H, CH ₂ CHF ₂ ], [ZA6715; H, F, F, H, CH ₂ CHF ₃ ], [ZA6716; H, F, F, H, (CH ₂ ) ₃ F], [ZA6717; H, F, F, H, (CH ₂ ) ₂ CHF ₂ ], [ZA6718; H, F, F, H, (CH ₂ ) ₂ CF ₃ ], [ZA6719; H, F, F, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA6720; H, F , F, H, CH ₂ Cl], [ZA6721; H, F, F, H, (CH ₂ ) ₂ Cl], [ZA6722; H, F, F, H, (CH ₂ ) ₃ Cl], [ZA6723 ; H, F, F, H, (CH ₂ ) ₄ Cl], [ZA6724; H, F, F, H, (CH ₂ ) ₅ Cl], [ZA6725; H, F, F, H, CH ₂ OMe ], [ZA6726; H, F, F, H, (CH ₂ ) ₂ OMe], [ZA6727; H, F, F, H, (CH ₂ ) ₃ OMe], [ZA6728; H, F, F, H , (CH ₂ ) ₄ OMe], [ZA6729; H, F, F, H, CH ₂ OEt], [ZA6730; H, F, F, H, (CH ₂ ) ₂ OEt], [ZA6731; H, F , F, H, (CH ₂ ) ₃ OEt], [ZA6732; H, F, F, H, CH ₂ OPr], [ZA6733; H, F, F, H, (CH ₂ ) ₂ OPr], [ZA6734 ; H, F, F, H, (CH ₂ ) ₃ OPr], [ZA6735; H, F, F, H, CH ₂ CN], [ZA6736; H, F, F, H, (CH ₂ ) ₂ CN ], [ZA6737; H, F, F, H, (CH ₂ ) ₃ CN], [ZA6738; H, F, F, H, (CH ₂ ) ₄ CN], [ZA6739; H, F, F, H, (CH ₂ ) ₅ CN], [ZA6740; H, F, F, H, CH ₂ CH = CH ₂ ], [ZA6741; H, F, F , H, CH ₂ C≡CH], [ZA6742; H, F, F, H, CH ₂ C≡CCH ₃ ], [ZA6743; H, F, F, H, CH ₂ Ph], [ZA6744; H, F, F, H, CH ₂ (2-Py)], [ZA6745; H, F, F, H, CH ₂ (3-Py)], [ZA6746; H, F, F, H, CH ₂ (4 -Py)], [ZA6747; H, F, F, H, (CH ₂ ) ₂ Ph], [ZA6748; H, F, F, H, (CH ₂ ) ₂ (2-Py)], [ZA6749; H, F, F, H, (CH ₂ ) ₂ (3-Py)], [ZA6750; H, F, F, H, (CH ₂ ) ₂ (4-Py)],

[ZA6751; H, F, F, H, Ph], [ZA6752; H, F, F, H, 2-Py], [ZA6753; H, F, F, H, 3-Py], [ZA6754; H , F, F, H, 4-Py], [ZA6755; H, F, F, F, NHMe], [ZA6756; H, F, F, F, NHEt], [ZA6757; H, F, F, F , NHPr], [ZA6758; H, F, F, F, NHBu], [ZA6759; H, F, F, F, NHPen], [ZA6760; H, F, F, F, NHHex], [ZA6761; H , F, F, F, NH (i-Pr)], [ZA6762; H, F, F, F, NH (i-Bu)], [ZA6763; H, F, F, F, NH (c-Pr )], [ZA6764; H, F, F, F, NH (c-Bu)], [ZA6765; H, F, F, F, NH (c-Pen)], [ZA6766; H, F, F, F, NH (c-Hex)], [ZA6767; H, F, F, F, NHCH ₂ (c-Pr)], [ZA6768; H, F, F, F, NHCH ₂ (c-Bu)], [ZA6769; H, F, F, F, NHCH ₂ (c-Pen)], [ZA6770; H, F, F, F, NHCH ₂ (c-Hex)], [ZA6771; H, F, F, F , NHCH ₂ F], [ZA6772; H, F, F, F, NHCHF ₂ ], [ZA6773; H, F, F, F, NHCF ₃ ], [ZA6774; H, F, F, F, NH (CH ₂ ) ₂ F], [ZA6775; H, F, F, F, NHCH ₂ CHF ₂ ], [ZA6776; H, F, F, F, NHCH ₂ CHF ₃ ], [ZA6777; H, F, F, F , NH (CH ₂ ) ₃ F], [ZA6778; H, F, F, F, NH (CH ₂ ) ₂ CHF ₂ ], [ZA6779; H, F, F, F, NH (CH ₂ ) ₂ CF ₃ ], [ZA6780; H, F, F, F, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA6781; H, F, F, F, NHCH ₂ Cl], [ZA6782; H, F, F, F, NH (CH ₂ ) ₂ Cl], [ZA6783; H, F, F, F, NH (CH ₂ ) ₃ Cl], [ZA6784; H, F, F, F, NH (CH ₂ ) ₄ Cl], [ ZA6785; H, F, F, F, NH (CH ₂ ) ₅ Cl], [ZA6786; H, F, F, F, NHCH ₂ OMe], [ZA6 787; H, F, F, F, NH (CH ₂ ) ₂ OMe], [ZA6788; H, F, F, F, NH (CH ₂ ) ₃ OMe], [ZA6789; H, F, F, F, NH (CH ₂ ) ₄ OMe], [ZA6790; H, F, F, F, NHCH ₂ OEt], [ZA6791; H, F, F, F, NH (CH ₂ ) ₂ OEt], [ZA6792; H, F, F, F, NH (CH ₂ ) ₃ OEt], [ZA6793; H, F, F, F, NHCH ₂ OPr], [ZA6794; H, F, F, F, NH (CH ₂ ) ₂ OPr] , [ZA6795; H, F, F, F, NH (CH ₂ ) ₃ OPr], [ZA6796; H, F, F, F, NHCH ₂ CN], [ZA6797; H, F, F, F, NH ( _{CH 2) 2 CN], [} ZA6798; H, F, F, F, NH (CH 2) 3 CN], [ZA6799; H, F, F, F, NH (CH 2) 4 CN], [ZA6800; H, F, F, F, NH (CH ₂ ) ₅ CN], [ZA6801; H, F, F, F, NHCH ₂ CH = CH ₂ ], [ZA6802; H, F, F, F, NHCH ₂ C ≡CH], [ZA6803; H, F, F, F, NHCH ₂ C≡CCH ₃ ], [ZA6804; H, F, F, F, NHCH ₂ Ph], [ZA6805; H, F, F, F, NHCH ₂ (2-Py)], [ZA6806; H, F, F, F, NHCH ₂ (3-Py)], [ZA6807; H, F, F, F, NHCH ₂ (4-Py)], [ ZA6808; H, F, F, F, NH (CH ₂ ) ₂ Ph], [ZA6809; H, F, F, F, NH (CH ₂ ) ₂ (2-Py)], [ZA6810; H, F, F, F, NH (CH ₂ ) ₂ (3-Py)], [ZA6811; H, F, F, F, NH (CH ₂ ) ₂ (4-Py)], [ZA6812; H, F, F, F, NHPh], [ZA6813; H, F, F, F, NH (2-Py)], [ZA6814; H, F, F, F, NH (3-Py)], [ZA6815; H, F, F, F, NH (4-Py)], [ZA6816; H, F, F, F, NMe ₂ ], [ZA6817; H, F, F, F, NMeEt], [ZA6818; H, F, F, F, NMePr], [ZA6819; H, F, F, F, NMeBu], [ZA6820; H, F, F, F, NMePen], [ZA6821; H, F, F, F, NMeHex], [ZA6822; H, F, F, F, NMe (i-Pr)], [ZA6823; H, F, F , F, NMe (i-Bu)], [ZA6824; H, F, F, F, NMe (c-Pr)], [ZA6825; H, F, F, F, NMe (c-Bu)], [ ZA6826; H, F, F, F, NMe (c-Pen)], [ZA6827; H, F, F, F, NMe (c-Hex)], [ZA6828; H, F, F, F, NMeCH ₂ (c-Pr)], [ZA6829; H, F, F, F, NMeCH ₂ (c-Bu)], [ZA6830; H, F, F, F, NMeCH ₂ (c-Pen)], [ZA6831; H, F, F, F, NMeCH ₂ (c-Hex)], [ZA6832; H, F, F, F, NMeCH ₂ F], [ZA6833; H, F, F, F, NMeCHF ₂ ], [ZA6834 ; H, F, F, F, NMeCF ₃ ], [ZA6835; H, F, F, F, NMe (CH ₂ ) ₂ F], [ZA6836; H, F, F, F, NMeCH ₂ CHF ₂ ], [ZA6837; H, F, F, F, NMeCH ₂ CHF ₃ ], [ZA6838; H, F, F, F, NMe (CH ₂ ) ₃ F], [ZA6839; H, F, F, F, NMe ( CH ₂ ) ₂ CHF ₂ ], [ZA6840; H, F, F, F, NMe (CH ₂ ) ₂ CF ₃ ], [ZA6841; H, F, F, F, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA6842; H, F, F, F, NMeCH ₂ Cl], [ZA6843; H, F, F, F, NMe (CH ₂ ) ₂ Cl], [ZA6844; H, F, F, F, NMe (CH _{2) 3 Cl], [ZA6845} ; H, F, F, F, NMe (CH 2) 4 Cl], [ZA6846; H, F, F, F, NMe (CH 2) 5 Cl], [ZA6847; H , F, F, F, NMeCH ₂ OMe], [ZA6848; H, F, F, F, NMe (CH ₂ ) ₂ OMe], [ZA6849; H, F, F, F, NMe (CH ₂ ) ₃ OMe ], [ZA6850; H, F, F, F, NMe (CH ₂ ) ₄ OMe], [ZA6851; H, F, F, F, NMeCH ₂ OEt], [ZA6852; H, F, F, F, NMe (CH ₂ ) ₂ OEt], [ZA6853; H, F, F, F, NMe (CH ₂ ) ₃ OEt], [ZA6854; H, F, F, F, NMeCH ₂ OPr], [ZA6855; H, F, F, F, NMe (CH ₂ ) ₂ OPr], [ZA6856; H, F, F, F, NMe (CH ₂ ) ₃ OPr], [ZA6857; H, F, F, F, NMeCH ₂ CN], [ZA6858; H, F, F, F, NMe (CH ₂ ) ₂ CN], [ZA6859; H, F, F, F, NMe (CH ₂ ) ₃ CN], [ZA6860; H, F, F, F, NMe (CH ₂ ) ₄ CN], [ZA6861; H, F, F, F, NMe (CH ₂ ) ₅ CN], [ZA6862; H, F, F, F, NMeCH ₂ CH = CH ₂ ], [ZA6863; H, F , F, F, NMeCH ₂ C≡CH], [ZA6864; H, F, F, F, NMeCH ₂ C≡CCH ₃ ], [ZA6865; H, F, F, F, NMeCH ₂ Ph], [ZA6866; H, F, F, F, NMeCH ₂ (2-Py)], [ZA6867; H, F, F, F, NMeCH ₂ (3-Py)], [ZA6868; H, F, F, F, NMeCH ₂ (4-Py)], [ZA6869; H, F, F, F, NMe (CH ₂ ) ₂ Ph], [ZA6870; H, F, F, F, NMe (CH ₂ ) ₂ (2-Py)] , [ZA6871; H, F, F, F, NMe (CH ₂ ) ₂ (3-Py)], [ZA6872; H, F, F, F, NMe (CH ₂ ) ₂ (4-Py)], [ ZA6873; H, F, F, F, NMePh], [ZA6874; H, F, F, F, NMe (2-Py)], [ZA6875; H, F, F, F, NMe (3-Py)] , [ZA6876; H, F, F, F, NMe (4-Py)], [ZA6877; H, F, F, F, NEt ₂ ], [ZA6878; H, F, F, F, NEtPr], [ ZA6879; H, F, F, F, NEtBu], [ZA6880; H, F, F, F, NEtPen], [ZA6881; H, F, F, F, NEtHex], [ZA6882; H, F, F, F, NEt (i-Pr)], [ZA6883; H, F, F, F, NEt (i-Bu)], [ZA6884; H, F, F, F, NEt (c-Pr)], [ZA6885 ; H, F, F, F, NEt (c-Bu)], [ZA6 886; H, F, F, F, NEt (c-Pen)], [ZA6887; H, F, F, F, NEt (c-Hex)], [ZA6888; H, F, F, F, NEtCH 2 (c-Pr)], [ZA6889; H, F, F, F, NEtCH ₂ (c-Bu)], [ZA6890; H, F, F, F, NEtCH ₂ (c-Pen)], [ZA6891; H, F, F, F, NEtCH ₂ (c-Hex)], [ZA6892; H, F, F, F, NEtCH ₂ F], [ZA6893; H, F, F, F, NEtCHF ₂ ], [ZA6894 ; H, F, F, F, NEtCF ₃ ], [ZA6895; H, F, F, F, NEt (CH ₂ ) ₂ F], [ZA6896; H, F, F, F, NEtCH ₂ CHF ₂ ], [ZA6897; H, F, F, F, NEtCH ₂ CHF ₃ ], [ZA6898; H, F, F, F, NEt (CH ₂ ) ₃ F], [ZA6899; H, F, F, F, NEt ( _{CH 2) 2 CHF 2],} [ZA6900; H, F, F, F, NEt (CH 2) 2 CF 3], [ZA6901; H, F, F, F, NEtCH 2 CH (CF 3) 2], [ZA6902; H, F, F, F, NEtCH ₂ Cl], [ZA6903; H, F, F, F, NEt (CH ₂ ) ₂ Cl], [ZA6904; H, F, F, F, NEt (CH _{2) 3 Cl], [ZA6905} ; H, F, F, F, NEt (CH 2) 4 Cl], [ZA6906; H, F, F, F, NEt (CH 2) 5 Cl], [ZA6907; H , F, F, F, NEtCH ₂ OMe], [ZA6908; H, F, F, F, NEt (CH ₂ ) ₂ OMe], [ZA6909; H, F, F, F, NEt (CH ₂ ) ₃ OMe ], [ZA6910; H, F, F, F, NEt (CH ₂ ) ₄ OMe], [ZA6911; H, F, F, F, NEtCH ₂ OEt], [ZA6912; H, F, F, F, NEt (CH ₂ ) ₂ OEt], [ZA6913; H, F, F, F, NEt (CH ₂ ) ₃ OEt], [ZA6914; H, F, F, F, NEtCH ₂ OPr], [ZA6915; H, F , F, F, NEt (CH 2) 2 OPr], [ZA6916; H, F, F, F, NEt (CH 2) 3 OPr], [ZA6917; H, F, F, F, NEtCH ₂ CN], [ZA6918; H, F, F, F, NEt (CH ₂ ) ₂ CN], [ZA6919; H, F, F, F, NEt (CH ₂ ) ₃ CN], [ZA6920; H, F, F, F, NEt (CH ₂ ) ₄ CN], [ZA6921; H, F, F, F, NEt (CH ₂ ) ₅ CN], [ZA6922; H, F, F, F, NEtCH ₂ CH = CH ₂ ], [ZA6923; H, F, F, F, NEtCH ₂ C≡CH], [ZA6924; H, F, F, F, NEtCH ₂ C≡CCH ₃ ], [ZA6925; H, F, F, F, NEtCH ₂ Ph], [ZA6926; H, F, F, F, NEtCH ₂ (2-Py)], [ZA6927; H, F, F, F, NEtCH ₂ (3-Py)], [ ZA6928; H, F, F, F, NEtCH ₂ (4-Py)], [ZA6929; H, F, F, F, NEt (CH ₂ ) ₂ Ph], [ZA6930; H, F, F, F, NEt (CH ₂ ) ₂ (2-Py)], [ZA6931; H, F, F, F, NEt (CH ₂ ) ₂ (3-Py)], [ZA6932; H, F, F, F, NEt ( CH ₂ ) ₂ (4-Py)], [ZA6933; H, F, F, F, NEtPh], [ZA6934; H, F, F, F, NEt (2-Py)], [ZA6935; H, F , F, F, NEt (3-Py)], [ZA6936; H, F, F, F, NEt (4-Py)], [ZA6937; H, F, F, F, Pyr], [ZA6938; H , F, F, F, Pip], [ZA6939; H, F, F, F, Mor], [ZA6940; H, F, F, F, OMe], [ZA6941; H, F, F, F, OEt ], [ZA6942; H, F, F, F, OPr], [ZA6943; H, F, F, F, OBu], [ZA6944; H, F, F, F, OPen], [ZA6945; H, F , F, F, OHex], [ZA6946; H, F, F, F, O (i-Pr)], [ZA6947; H, F, F, F, O (i-Bu)], [ZA6948; H , F, F, F, O (c-Pr)], [ZA6949; H, F, F, F, O (c-Bu)], [ZA6950; H, F, F, F, O (c-Pen )], [ZA6951; H, F, F, F, O (c-Hex)], [ZA6952; H, F, F, F, OCH ₂ (c-Pr)], [ZA6953 ; H, F, F, F, OCH ₂ (c-Bu)], [ZA6954; H, F, F, F, OCH ₂ (c-Pen)], [ZA6955; H, F, F, F, OCH _{2 (c-Hex)],} [ZA6956; H, F, F, F, OCH 2 F], [ZA6957; H, F, F, F, OCHF 2], [ZA6958; H, F, F, F, OCF ₃ ], [ZA6959; H, F, F, F, O (CH ₂ ) ₂ F], [ZA6960; H, F, F, F, OCH ₂ CHF ₂ ], [ZA6961; H, F, F, F, OCH ₂ CHF ₃ ], [ZA6962; H, F, F, F, O (CH ₂ ) ₃ F], [ZA6963; H, F, F, F, O (CH ₂ ) ₂ CHF ₂ ], [ ZA6964; H, F, F, F, O (CH ₂ ) ₂ CF ₃ ], [ZA6965; H, F, F, F, OCH ₂ CH (CF ₃ ) ₂ ], [ZA6966; H, F, F, F, OCH ₂ Cl], [ZA6967; H, F, F, F, O (CH ₂ ) ₂ Cl], [ZA6968; H, F, F, F, O (CH ₂ ) ₃ Cl], [ZA6969; H, F, F, F, O (CH ₂ ) ₄ Cl], [ZA6970; H, F, F, F, O (CH ₂ ) ₅ Cl], [ZA6971; H, F, F, F, OCH ₂ OMe], [ZA6972; H, F, F, F, O (CH ₂ ) ₂ OMe], [ZA6973; H, F, F, F, O (CH ₂ ) ₃ OMe], [ZA6974; H, F, F, F, O (CH ₂ ) ₄ OMe], [ZA6975; H, F, F, F, OCH ₂ OEt], [ZA6976; H, F, F, F, O (CH ₂ ) ₂ OEt], [ ZA6977; H, F, F, F, O (CH ₂ ) ₃ OEt], [ZA6978; H, F, F, F, OCH ₂ OPr], [ZA6979; H, F, F, F, O (CH ₂ ) ₂ OPr], [ZA6980; H, F, F, F, O (CH ₂ ) ₃ OPr], [ZA6981; H, F, F, F, OCH ₂ CN], [ZA6982; H, F, F, _{F, O (CH 2) 2} CN], [ZA6983; H, F, F, F, O (CH 2) 3 CN], [ZA6984; H, F, F, F, O (CH 2) 4 CN] , [ZA6985; H, F, F, F, O (CH ₂ ) ₅ CN], [ZA6986; H, F , F, F, OCH ₂ CH = CH ₂ ], [ZA6987; H, F, F, F, OCH ₂ C≡CH], [ZA6988; H, F, F, F, OCH ₂ C≡CCH ₃ ], [ZA6989; H, F, F, F, OCH ₂ Ph], [ZA6990; H, F, F, F, OCH ₂ (2-Py)], [ZA6991; H, F, F, F, OCH ₂ ( 3-Py)], [ZA6992; H, F, F, F, OCH ₂ (4-Py)], [ZA6993; H, F, F, F, O (CH ₂ ) ₂ Ph], [ZA6994; H , F, F, F, O (CH ₂ ) ₂ (2-Py)], [ZA6995; H, F, F, F, O (CH ₂ ) ₂ (3-Py)], [ZA6996; H, F , F, F, O (CH ₂ ) ₂ (4-Py)], [ZA6997; H, F, F, F, OPh], [ZA6998; H, F, F, F, O (2-Py)] , [ZA6999; H, F, F, F, O (3-Py)], [ZA7000; H, F, F, F, O (4-Py)],

[ZA7001; H, F, F, F, Me], [ZA7002; H, F, F, F, Et], [ZA7003; H, F, F, F, Pr], [ZA7004; H, F, F , F, Bu], [ZA7005; H, F, F, F, Pen], [ZA7006; H, F, F, F, Hex], [ZA7007; H, F, F, F, (i-Pr) ], [ZA7008; H, F, F, F, (i-Bu)], [ZA7009; H, F, F, F, (c-Pr)], [ZA7010; H, F, F, F, ( c-Bu)], [ZA7011; H, F, F, F, (c-Pen)], [ZA7012; H, F, F, F, (c-Hex)], [ZA7013; H, F, F , F, CH ₂ (c-Pr)], [ZA7014; H, F, F, F, CH ₂ (c-Bu)], [ZA7015; H, F, F, F, CH ₂ (c-Pen) ], [ZA7016; H, F, F, F, CH ₂ (c-Hex)], [ZA7017; H, F, F, F, CH ₂ F], [ZA7018; H, F, F, F, CHF ₂ ], [ZA7019; H, F, F, F, CF ₃ ], [ZA7020; H, F, F, F, (CH ₂ ) ₂ F], [ZA7021; H, F, F, F, CH ₂ CHF ₂ ], [ZA7022; H, F, F, F, CH ₂ CHF ₃ ], [ZA7023; H, F, F, F, (CH ₂ ) ₃ F], [ZA7024; H, F, F, F , (CH ₂ ) ₂ CHF ₂ ], [ZA7025; H, F, F, F, (CH ₂ ) ₂ CF ₃ ], [ZA7026; H, F, F, F, CH ₂ CH (CF ₃ ) ₂ ] , [ZA7027; H, F, F, F, CH ₂ Cl], [ZA7028; H, F, F, F, (CH ₂ ) ₂ Cl], [ZA7029; H, F, F, F, (CH ₂ ) ₃ Cl], [ZA7030; H, F, F, F, (CH ₂ ) ₄ Cl], [ZA7031; H, F, F, F, (CH ₂ ) ₅ Cl], [ZA7032; H, F, F, F, CH ₂ OMe], [ZA7033; H, F, F, F, (CH ₂ ) ₂ OMe], [ZA7034; H, F, F, F, (CH ₂ ) ₃ OMe], [ZA7035; H, F, F, F, (CH ₂ ) ₄ OMe], [ZA7036; H, F, F, F, CH ₂ OEt], [ZA7037; H, F, F, F, (CH ₂ ) ₂ OEt] , [ZA7 038; H, F, F, F, (CH ₂ ) ₃ OEt], [ZA7039; H, F, F, F, CH ₂ OPr], [ZA7040; H, F, F, F, (CH ₂ ) ₂ OPr], [ZA7041; H, F, F, F, (CH ₂ ) ₃ OPr], [ZA7042; H, F, F, F, CH ₂ CN], [ZA7043; H, F, F, F, ( _{CH 2) 2 CN], [} ZA7044; H, F, F, F, (CH 2) 3 CN], [ZA7045; H, F, F, F, (CH 2) 4 CN], [ZA7046; H, F, F, F, (CH ₂ ) ₅ CN], [ZA7047; H, F, F, F, CH ₂ CH = CH ₂ ], [ZA7048; H, F, F, F, CH ₂ C≡CH] , [ZA7049; H, F, F, F, CH ₂ C≡CCH ₃ ], [ZA7050; H, F, F, F, CH ₂ Ph], [ZA7051; H, F, F, F, CH ₂ ( 2-Py)], [ZA7052; H, F, F, F, CH ₂ (3-Py)], [ZA7053; H, F, F, F, CH ₂ (4-Py)], [ZA7054; H , F, F, F, (CH ₂ ) ₂ Ph], [ZA7055; H, F, F, F, (CH ₂ ) ₂ (2-Py)], [ZA7056; H, F, F, F, ( CH ₂ ) ₂ (3-Py)], [ZA7057; H, F, F, F, (CH ₂ ) ₂ (4-Py)], [ZA7058; H, F, F, F, Ph], [ZA7059 ; H, F, F, F, 2-Py], [ZA7060; H, F, F, F, 3-Py], [ZA7061; H, F, F, F, 4-Py], [ZA7062; H , F, Cl, H, NHMe], [ZA7063; H, F, Cl, H, NHEt], [ZA7064; H, F, Cl, H, NHPr], [ZA7065; H, F, Cl, H, NHBu ], [ZA7066; H, F, Cl, H, NHPen], [ZA7067; H, F, Cl, H, NHHex], [ZA7068; H, F, Cl, H, NH (i-Pr)], [ ZA7069; H, F, Cl, H, NH (i-Bu)], [ZA7070; H, F, Cl, H, NH (c-Pr)], [ZA7071; H, F, Cl, H, NH ( c-Bu)], [ZA7072; H, F, Cl, H, NH (c-Pen)], [ZA7073; H, F, Cl, H, NH (c-Hex)], [ZA7074; H, F , C l, H, NHCH ₂ (c-Pr)], [ZA7075; H, F, Cl, H, NHCH ₂ (c-Bu)], [ZA7076; H, F, Cl, H, NHCH ₂ (c-Pen )], [ZA7077; H, F, Cl, H, NHCH ₂ (c-Hex)], [ZA7078; H, F, Cl, H, NHCH ₂ F], [ZA7079; H, F, Cl, H, NHCHF ₂ ], [ZA7080; H, F, Cl, H, NHCF ₃ ], [ZA7081; H, F, Cl, H, NH (CH ₂ ) ₂ F], [ZA7082; H, F, Cl, H, NHCH ₂ CHF ₂ ], [ZA7083; H, F, Cl, H, NHCH ₂ CHF ₃ ], [ZA7084; H, F, Cl, H, NH (CH ₂ ) ₃ F], [ZA7085; H, F, Cl, H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA7086; H, F, Cl, H, NH (CH ₂ ) ₂ CF ₃ ], [ZA7087; H, F, Cl, H, NHCH ₂ CH ( CF ₃ ) ₂ ], [ZA7088; H, F, Cl, H, NHCH ₂ Cl], [ZA7089; H, F, Cl, H, NH (CH ₂ ) ₂ Cl], [ZA7090; H, F, Cl , H, NH (CH ₂ ) ₃ Cl], [ZA7091; H, F, Cl, H, NH (CH ₂ ) ₄ Cl], [ZA7092; H, F, Cl, H, NH (CH ₂ ) ₅ Cl ], [ZA7093; H, F, Cl, H, NHCH ₂ OMe], [ZA7094; H, F, Cl, H, NH (CH ₂ ) ₂ OMe], [ZA7095; H, F, Cl, H, NH (CH ₂ ) ₃ OMe], [ZA7096; H, F, Cl, H, NH (CH ₂ ) ₄ OMe], [ZA7097; H, F, Cl, H, NHCH ₂ OEt], [ZA7098; H, F , Cl, H, NH (CH ₂ ) ₂ OEt], [ZA7099; H, F, Cl, H, NH (CH ₂ ) ₃ OEt], [ZA7100; H, F, Cl, H, NHCH ₂ OPr], [ZA7101; H, F, Cl, H, NH (CH ₂ ) ₂ OPr], [ZA7102; H, F, Cl, H, NH (CH ₂ ) ₃ OPr], [ZA7103; H, F, Cl, H , NHCH ₂ CN], [ZA7104; H, F, Cl, H, NH (CH ₂ ) ₂ CN], [ZA7105; H, F, Cl, H, N H (CH ₂ ) ₃ CN], [ZA7106; H, F, Cl, H, NH (CH ₂ ) ₄ CN], [ZA7107; H, F, Cl, H, NH (CH ₂ ) ₅ CN], [ ZA7108; H, F, Cl, H, NHCH ₂ CH = CH ₂ ], [ZA7109; H, F, Cl, H, NHCH ₂ C≡CH], [ZA7110; H, F, Cl, H, NHCH ₂ C ≡CCH ₃ ], [ZA7111; H, F, Cl, H, NHCH ₂ Ph], [ZA7112; H, F, Cl, H, NHCH ₂ (2-Py)], [ZA7113; H, F, Cl, H, NHCH ₂ (3-Py)], [ZA7114; H, F, Cl, H, NHCH ₂ (4-Py)], [ZA7115; H, F, Cl, H, NH (CH ₂ ) ₂ Ph] , [ZA7116; H, F, Cl, H, NH (CH ₂ ) ₂ (2-Py)], [ZA7117; H, F, Cl, H, NH (CH ₂ ) ₂ (3-Py)], [ ZA7118; H, F, Cl, H, NH (CH ₂ ) ₂ (4-Py)], [ZA7119; H, F, Cl, H, NHPh], [ZA7120; H, F, Cl, H, NH ( 2-Py)], [ZA7121; H, F, Cl, H, NH (3-Py)], [ZA7122; H, F, Cl, H, NH (4-Py)], [ZA7123; H, F , Cl, H, NMe ₂ ], [ZA7124; H, F, Cl, H, NMeEt], [ZA7125; H, F, Cl, H, NMePr], [ZA7126; H, F, Cl, H, NMeBu] , [ZA7127; H, F, Cl, H, NMePen], [ZA7128; H, F, Cl, H, NMeHex], [ZA7129; H, F, Cl, H, NMe (i-Pr)], [ZA7130 ; H, F, Cl, H, NMe (i-Bu)], [ZA7131; H, F, Cl, H, NMe (c-Pr)], [ZA7132; H, F, Cl, H, NMe (c -Bu)], [ZA7133; H, F, Cl, H, NMe (c-Pen)], [ZA7134; H, F, Cl, H, NMe (c-Hex)], [ZA7135; H, F, Cl, H, NMeCH ₂ (c-Pr)], [ZA7136; H, F, Cl, H, NMeCH ₂ (c-Bu)], [ZA7137; H, F, Cl, H, NMeCH ₂ (c-Pen )], [ZA7138; H, F, Cl, H, NMeCH ₂ (c- Hex)], [ZA7139; H, F, Cl, H, NMeCH ₂ F], [ZA7140; H, F, Cl, H, NMeCHF ₂ ], [ZA7141; H, F, Cl, H, NMeCF ₃ ], [ZA7142; H, F, Cl, H, NMe (CH ₂ ) ₂ F], [ZA7143; H, F, Cl, H, NMeCH ₂ CHF ₂ ], [ZA7144; H, F, Cl, H, NMeCH ₂ CHF ₃ ], [ZA7145; H, F, Cl, H, NMe (CH ₂ ) ₃ F], [ZA7146; H, F, Cl, H, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA7147; H, F, Cl, H, NMe (CH ₂ ) ₂ CF ₃ ], [ZA7148; H, F, Cl, H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA7149; H, F, Cl, H, NMeCH ₂ Cl], [ZA7150; H, F, Cl, H, NMe (CH ₂ ) ₂ Cl], [ZA7151; H, F, Cl, H, NMe (CH ₂ ) ₃ Cl], [ZA7152; H, F, Cl, H, NMe (CH ₂ ) ₄ Cl], [ZA7153; H, F, Cl, H, NMe (CH ₂ ) ₅ Cl], [ZA7154; H, F, Cl, H, NMeCH ₂ OMe], [ ZA7155; H, F, Cl, H, NMe (CH ₂ ) ₂ OMe], [ZA7156; H, F, Cl, H, NMe (CH ₂ ) ₃ OMe], [ZA7157; H, F, Cl, H, NMe (CH ₂ ) ₄ OMe], [ZA7158; H, F, Cl, H, NMeCH ₂ OEt], [ZA7159; H, F, Cl, H, NMe (CH ₂ ) ₂ OEt], [ZA7160; H, F, Cl, H, NMe (CH ₂ ) ₃ OEt], [ZA7161; H, F, Cl, H, NMeCH ₂ OPr], [ZA7162; H, F, Cl, H, NMe (CH ₂ ) ₂ OPr] , [ZA7163; H, F, Cl, H, NMe (CH ₂ ) ₃ OPr], [ZA7164; H, F, Cl, H, NMeCH ₂ CN], [ZA7165; H, F, Cl, H, NMe ( _{CH 2) 2 CN], [} ZA7166; H, F, Cl, H, NMe (CH 2) 3 CN], [ZA7167; H, F, Cl, H, NMe (CH 2) 4 CN], [ZA7168; H, F, Cl, H, NMe (CH ₂ ) ₅ CN], [ZA7169; H, F, Cl, H, NMeCH ₂ CH = CH ₂ ], [ZA7170; H, F, Cl, H, NMeCH ₂ C≡CH], [ZA7171; H, F, Cl, H, NMeCH ₂ C≡CCH ₃ ], [ZA7172; H, F, Cl, H, NMeCH ₂ Ph], [ZA7173; H, F, Cl, H, NMeCH ₂ (2-Py)], [ZA7174; H, F, Cl , H, NMeCH ₂ (3-Py)], [ZA7175; H, F, Cl, H, NMeCH ₂ (4-Py)], [ZA7176; H, F, Cl, H, NMe (CH ₂ ) ₂ Ph ], [ZA7177; H, F, Cl, H, NMe (CH ₂ ) ₂ (2-Py)], [ZA7178; H, F, Cl, H, NMe (CH ₂ ) ₂ (3-Py)], [ZA7179; H, F, Cl, H, NMe (CH ₂ ) ₂ (4-Py)], [ZA7180; H, F, Cl, H, NMePh], [ZA7181; H, F, Cl, H, NMe (2-Py)], [ZA7182; H, F, Cl, H, NMe (3-Py)], [ZA7183; H, F, Cl, H, NMe (4-Py)], [ZA7184; H, F, Cl, H, NEt ₂ ], [ZA7185; H, F, Cl, H, NEtPr], [ZA7186; H, F, Cl, H, NEtBu], [ZA7187; H, F, Cl, H, NEtPen ], [ZA7188; H, F, Cl, H, NEtHex], [ZA7189; H, F, Cl, H, NEt (i-Pr)], [ZA7190; H, F, Cl, H, NEt (i- Bu)], [ZA7191; H, F, Cl, H, NEt (c-Pr)], [ZA7192; H, F, Cl, H, NEt (c-Bu)], [ZA7193; H, F, Cl , H, NEt (c-Pen)], [ZA7194; H, F, Cl, H, NEt (c-Hex)], [ZA7195; H, F, Cl, H, NEtCH ₂ (c-Pr)], [ZA7196; H, F, Cl, H, NEtCH ₂ (c-Bu)], [ZA7197; H, F, Cl, H, NEtCH ₂ (c-Pen)], [ZA7198; H, F, Cl, H , NEtCH ₂ (c-Hex)], [ZA7199; H, F, Cl, H, NEtCH ₂ F], [ZA7200; H, F, Cl, H, NEtCHF ₂ ], [ZA7201; H, F, Cl, H, NEtCF ₃ ], [ ZA7202; H, F, Cl, H, NEt (CH ₂ ) ₂ F], [ZA7203; H, F, Cl, H, NEtCH ₂ CHF ₂ ], [ZA7204; H, F, Cl, H, NEtCH ₂ CHF ₃ ], [ZA7205; H, F, Cl, H, NEt (CH ₂ ) ₃ F], [ZA7206; H, F, Cl, H, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA7207; H, F , Cl, H, NEt (CH ₂ ) ₂ CF ₃ ], [ZA7208; H, F, Cl, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA7209; H, F, Cl, H, NEtCH ₂ Cl ], [ZA7210; H, F, Cl, H, NEt (CH ₂ ) ₂ Cl], [ZA7211; H, F, Cl, H, NEt (CH ₂ ) ₃ Cl], [ZA7212; H, F, Cl , H, NEt (CH ₂ ) ₄ Cl], [ZA7213; H, F, Cl, H, NEt (CH ₂ ) ₅ Cl], [ZA7214; H, F, Cl, H, NEtCH ₂ OMe], [ZA7215 ; H, F, Cl, H, NEt (CH ₂ ) ₂ OMe], [ZA7216; H, F, Cl, H, NEt (CH ₂ ) ₃ OMe], [ZA7217; H, F, Cl, H, NEt (CH ₂ ) ₄ OMe], [ZA7218; H, F, Cl, H, NEtCH ₂ OEt], [ZA7219; H, F, Cl, H, NEt (CH ₂ ) ₂ OEt], [ZA7220; H, F , Cl, H, NEt (CH ₂ ) ₃ OEt], [ZA7221; H, F, Cl, H, NEtCH ₂ OPr], [ZA7222; H, F, Cl, H, NEt (CH ₂ ) ₂ OPr], [ZA7223; H, F, Cl, H, NEt (CH ₂ ) ₃ OPr], [ZA7224; H, F, Cl, H, NEtCH ₂ CN], [ZA7225; H, F, Cl, H, NEt (CH _{2) 2 CN], [ZA7226} ; H, F, Cl, H, NEt (CH 2) 3 CN], [ZA7227; H, F, Cl, H, NEt (CH 2) 4 CN], [ZA7228; H , F, Cl, H, NEt (CH ₂ ) ₅ CN], [ZA7229; H, F, Cl, H, NEtCH ₂ CH = CH ₂ ], [ZA7230; H, F, Cl, H, NEtCH ₂ C≡ CH], [ZA7231; H, F, Cl, H, NEtCH ₂ C≡CCH ₃ ], [ZA7232; H, F, Cl, H, NEtCH ₂ Ph], [ZA7233; H, F, Cl, H, NEtCH ₂ (2-Py)], [ZA7234; H, F, Cl, H, NEtCH ₂ (3-Py)], [ZA7235; H, F, Cl, H, NEtCH ₂ (4-Py)], [ZA7236; H, F, Cl, H, NEt (CH ₂ ) ₂ Ph], [ZA7237; H, F, Cl, H, NEt (CH ₂ ) ₂ (2-Py)], [ZA7238; H, F, Cl, H, NEt (CH ₂ ) ₂ (3-Py)] , [ZA7239; H, F, Cl, H, NEt (CH ₂ ) ₂ (4-Py)], [ZA7240; H, F, Cl, H, NEtPh], [ZA7241; H, F, Cl, H, NEt (2-Py)], [ZA7242; H, F, Cl, H, NEt (3-Py)], [ZA7243; H, F, Cl, H, NEt (4-Py)], [ZA7244; H , F, Cl, H, Pyr], [ZA7245; H, F, Cl, H, Pip], [ZA7246; H, F, Cl, H, Mor], [ZA7247; H, F, Cl, H, OMe ], [ZA7248
; H, F, Cl, H, OEt], [ZA7249; H, F, Cl, H, OPr], [ZA7250; H, F, Cl, H, OBu],

[ZA7251; H, F, Cl, H, OPen], [ZA7252; H, F, Cl, H, OHex], [ZA7253; H, F, Cl, H, O (i-Pr)], [ZA7254; H, F, Cl, H, O (i-Bu)], [ZA7255; H, F, Cl, H, O (c-Pr)], [ZA7256; H, F, Cl, H, O (c- Bu)], [ZA7257; H, F, Cl, H, O (c-Pen)], [ZA7258; H, F, Cl, H, O (c-Hex)], [ZA7259; H, F, Cl , H, OCH ₂ (c-Pr)], [ZA7260; H, F, Cl, H, OCH ₂ (c-Bu)], [ZA7261; H, F, Cl, H, OCH ₂ (c-Pen) ], [ZA7262; H, F, Cl, H, OCH ₂ (c-Hex)], [ZA7263; H, F, Cl, H, OCH ₂ F], [ZA7264; H, F, Cl, H, OCHF ₂ ], [ZA7265; H, F, Cl, H, OCF ₃ ], [ZA7266; H, F, Cl, H, O (CH ₂ ) ₂ F], [ZA7267; H, F, Cl, H, OCH ₂ CHF ₂ ], [ZA7268; H, F, Cl, H, OCH ₂ CHF ₃ ], [ZA7269; H, F, Cl, H, O (CH ₂ ) ₃ F], [ZA7270; H, F, Cl , H, O (CH ₂ ) ₂ CHF ₂ ], [ZA7271; H, F, Cl, H, O (CH ₂ ) ₂ CF ₃ ], [ZA7272; H, F, Cl, H, OCH ₂ CH (CF ₃ ) ₂ ], [ZA7273; H, F, Cl, H, OCH ₂ Cl], [ZA7274; H, F, Cl, H, O (CH ₂ ) ₂ Cl], [ZA7275; H, F, Cl, H, O (CH ₂ ) ₃ Cl], [ZA7276; H, F, Cl, H, O (CH ₂ ) ₄ Cl], [ZA7277; H, F, Cl, H, O (CH ₂ ) ₅ Cl] , [ZA7278; H, F, Cl, H, OCH ₂ OMe], [ZA7279; H, F, Cl, H, O (CH ₂ ) ₂ OMe], [ZA7280; H, F, Cl, H, O ( CH ₂ ) ₃ OMe], [ZA7281; H, F, Cl, H, O (CH ₂ ) ₄ OMe], [ZA7282; H, F, Cl, H, OCH ₂ OEt], [ZA7283; H, F, Cl, H, O (CH ₂ ) ₂ OEt], [ZA7284; H, F, Cl, H, O (CH ₂ ) ₃ OEt], [ZA7285; H, F, Cl, H, OCH ₂ OPr], [ZA7286; H, F, Cl, H, O (CH ₂ ) ₂ OPr], [ZA7287; H, F , Cl, H, O (CH ₂ ) ₃ OPr], [ZA7288; H, F, Cl, H, OCH ₂ CN], [ZA7289; H, F, Cl, H, O (CH ₂ ) ₂ CN], [ZA7290; H, F, Cl, H, O (CH ₂ ) ₃ CN], [ZA7291; H, F, Cl, H, O (CH ₂ ) ₄ CN], [ZA7292; H, F, Cl, H , O (CH ₂ ) ₅ CN], [ZA7293; H, F, Cl, H, OCH ₂ CH = CH ₂ ], [ZA7294; H, F, Cl, H, OCH ₂ C≡CH], [ZA7295; H, F, Cl, H, OCH ₂ C≡CCH ₃ ], [ZA7296; H, F, Cl, H, OCH ₂ Ph], [ZA7297; H, F, Cl, H, OCH ₂ (2-Py) ], [ZA7298; H, F, Cl, H, OCH ₂ (3-Py)], [ZA7299; H, F, Cl, H, OCH ₂ (4-Py)], [ZA7300; H, F, Cl , H, O (CH ₂ ) ₂ Ph], [ZA7301; H, F, Cl, H, O (CH ₂ ) ₂ (2-Py)], [ZA7302; H, F, Cl, H, O (CH ₂ ) ₂ (3-Py)], [ZA7303; H, F, Cl, H, O (CH ₂ ) ₂ (4-Py)], [ZA7304; H, F, Cl, H, OPh], [ZA7305 ; H, F, Cl, H, O (2-Py)], [ZA7306; H, F, Cl, H, O (3-Py)], [ZA7307; H, F, Cl, H, O (4 -Py)], [ZA7308; H, F, Cl, H, Me], [ZA7309; H, F, Cl, H, Et], [ZA7310; H, F, Cl, H, Pr], [ZA7311; H, F, Cl, H, Bu], [ZA7312; H, F, Cl, H, Pen], [ZA7313; H, F, Cl, H, Hex], [ZA7314; H, F, Cl, H, (i-Pr)], [ZA7315; H, F, Cl, H, (i-Bu)], [ZA7316; H, F, Cl, H, (c-Pr)], [ZA7317; H, F, Cl, H, (c-Bu)], [ZA7318; H, F, Cl, H, (c-Pen)], [ZA7319; H, F, Cl, H, (c-Hex )], [ZA7320; H, F, Cl, H, CH ₂ (c-Pr)], [ZA7321; H, F, Cl, H, CH ₂ (c-Bu)], [ZA7322; H, F, Cl, H, CH ₂ (c-Pen)], [ZA7323; H, F, Cl, H, CH ₂ (c-Hex)], [ZA7324; H, F, Cl, H, CH ₂ F], [ ZA7325; H, F, Cl, H, CHF ₂ ], [ZA7326; H, F, Cl, H, CF ₃ ], [ZA7327; H, F, Cl, H, (CH ₂ ) ₂ F], [ZA7328 ; H, F, Cl, H, CH ₂ CHF ₂ ], [ZA7329; H, F, Cl, H, CH ₂ CHF ₃ ], [ZA7330; H, F, Cl, H, (CH ₂ ) ₃ F] , [ZA7331; H, F, Cl, H, (CH ₂ ) ₂ CHF ₂ ], [ZA7332; H, F, Cl, H, (CH ₂ ) ₂ CF ₃ ], [ZA7333; H, F, Cl, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA7334; H, F, Cl, H, CH ₂ Cl], [ZA7335; H, F, Cl, H, (CH ₂ ) ₂ Cl], [ZA7336; H, F, Cl, H, (CH ₂ ) ₃ Cl], [ZA7337; H, F, Cl, H, (CH ₂ ) ₄ Cl], [ZA7338; H, F, Cl, H, (CH ₂ ) ₅ Cl], [ZA7339; H, F, Cl, H, CH ₂ OMe], [ZA7340; H, F, Cl, H, (CH ₂ ) ₂ OMe], [ZA7341; H, F, Cl, H, (CH ₂ ) ₃ OMe], [ZA7342; H, F, Cl, H, (CH ₂ ) ₄ OMe], [ZA7343; H, F, Cl, H, CH ₂ OEt], [ZA7344; H, F, Cl, H, (CH ₂ ) ₂ OEt], [ZA7345; H, F, Cl, H, (CH ₂ ) ₃ OEt], [ZA7346; H, F, Cl, H, CH ₂ OPr], [ZA7347; H, F, Cl, H, (CH ₂ ) ₂ OPr], [ZA7348; H, F, Cl, H, (CH ₂ ) ₃ OPr], [ZA7349; H, F, Cl, H, CH ₂ CN] , [ZA7350; H, F, Cl, H, (CH ₂ ) ₂ CN], [ZA7351; H, F, Cl, H, (CH ₂ ) ₃ CN], [ZA7352; H, F, Cl, H, (CH ₂ ) ₄ CN], [Z A7353; H, F, Cl, H, (CH ₂ ) ₅ CN], [ZA7354; H, F, Cl, H, CH ₂ CH = CH ₂ ], [ZA7355; H, F, Cl, H, CH ₂ C≡CH], [ZA7356; H, F, Cl, H, CH ₂ C≡CCH ₃ ], [ZA7357; H, F, Cl, H, CH ₂ Ph], [ZA7358; H, F, Cl, H , CH ₂ (2-Py)], [ZA7359; H, F, Cl, H, CH ₂ (3-Py)], [ZA7360; H, F, Cl, H, CH ₂ (4-Py)], [ZA7361; H, F, Cl, H, (CH ₂ ) ₂ Ph], [ZA7362; H, F, Cl, H, (CH ₂ ) ₂ (2-Py)], [ZA7363; H, F, Cl , H, (CH ₂ ) ₂ (3-Py)], [ZA7364; H, F, Cl, H, (CH ₂ ) ₂ (4-Py)], [ZA7365; H, F, Cl, H, Ph ], [ZA7366; H, F, Cl, H, 2-Py], [ZA7367; H, F, Cl, H, 3-Py], [ZA7368; H, F, Cl, H, 4-Py], [ZA7369; H, F, Cl, Cl, NHMe], [ZA7370; H, F, Cl, Cl, NHEt], [ZA7371; H, F, Cl, Cl, NHPr], [ZA7372; H, F, Cl , Cl, NHBu], [ZA7373; H, F, Cl, Cl, NHPen], [ZA7374; H, F, Cl, Cl, NHHex], [ZA7375; H, F, Cl, Cl, NH (i-Pr )], [ZA7376; H, F, Cl, Cl, NH (i-Bu)], [ZA7377; H, F, Cl, Cl, NH (c-Pr)], [ZA7378; H, F, Cl, Cl, NH (c-Bu)], [ZA7379; H, F, Cl, Cl, NH (c-Pen)], [ZA7380; H, F, Cl, Cl, NH (c-Hex)], [ZA7381 ; H, F, Cl, Cl, NHCH ₂ (c-Pr)], [ZA7382; H, F, Cl, Cl, NHCH ₂ (c-Bu)], [ZA7383; H, F, Cl, Cl, NHCH ₂ (c-Pen)], [ZA7384; H, F, Cl, Cl, NHCH ₂ (c-Hex)], [ZA7385; H, F, Cl, Cl, NHCH ₂ F], [ZA7386; H, F , Cl, Cl, NHCHF ₂ ], [ZA7387; H, F, Cl, Cl, NHCF ₃ ], [ZA7388; H, F, Cl, Cl, NH (CH ₂ ) ₂ F], [ZA7389; H, F, Cl, Cl, NHCH ₂ CHF ₂ ], [ZA7390; H, F, Cl, Cl, NHCH ₂ CHF ₃ ], [ZA7391; H, F, Cl, Cl, NH (CH ₂ ) ₃ F], [ZA7392; H, F, Cl, Cl, NH (CH ₂ ) ₂ CHF ₂ ], [ZA7393; H, F, Cl, Cl, NH (CH ₂ ) ₂ CF ₃ ], [ZA7394; H, F, Cl, Cl, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA7395; H, F, Cl, Cl, NHCH ₂ Cl], [ZA7396; H, F, Cl, Cl, NH (CH ₂ ) ₂ Cl], [ZA7397; H, F, Cl, Cl, NH (CH ₂ ) ₃ Cl], [ZA7398; H, F, Cl, Cl, NH (CH ₂ ) ₄ Cl], [ZA7399; H, F, Cl, Cl, NH (CH ₂ ) ₅ Cl], [ZA7400; H, F, Cl, Cl, NHCH ₂ OMe], [ ZA7401; H, F, Cl, Cl, NH (CH ₂ ) ₂ OMe], [ZA7402; H, F, Cl, Cl, NH (CH ₂ ) ₃ OMe], [ZA7403; H, F, Cl, Cl, NH (CH ₂ ) ₄ OMe], [ZA7404; H, F, Cl, Cl, NHCH ₂ OEt], [ZA7405; H, F, Cl, Cl, NH (CH ₂ ) ₂ OEt], [ZA7406; H, F, Cl, Cl, NH (CH ₂ ) ₃ OEt], [ZA7407; H, F, Cl, Cl, NHCH ₂ OPr], [ZA7408; H, F, Cl, Cl, NH (CH ₂ ) ₂ OPr] , [ZA7409; H, F, Cl, Cl, NH (CH ₂ ) ₃ OPr], [ZA7410; H, F, Cl, Cl, NHCH ₂ CN], [ZA7411; H, F, Cl, Cl, NH ( _{CH 2) 2 CN], [} ZA7412; H, F, Cl, Cl, NH (CH 2) 3 CN], [ZA7413; H, F, Cl, Cl, NH (CH 2) 4 CN], [ZA7414; H, F, Cl, Cl, NH (CH ₂ ) ₅ CN], [ZA7415; H, F, Cl, Cl, NHCH ₂ CH = CH ₂ ], [ZA7416; H, F, Cl, Cl, NHCH ₂ C ≡CH], [ZA7417; H, F, Cl, Cl, NHC H ₂ C≡CCH ₃ ], [ZA7418; H, F, Cl, Cl, NHCH ₂ Ph], [ZA7419; H, F, Cl, Cl, NHCH ₂ (2-Py)], [ZA7420; H, F , Cl, Cl, NHCH ₂ (3-Py)], [ZA7421; H, F, Cl, Cl, NHCH ₂ (4-Py)], [ZA7422; H, F, Cl, Cl, NH (CH ₂ ) ₂ Ph], [ZA7423; H, F, Cl, Cl, NH (CH ₂ ) ₂ (2-Py)], [ZA7424; H, F, Cl, Cl, NH (CH ₂ ) ₂ (3-Py) ], [ZA7425; H, F, Cl, Cl, NH (CH ₂ ) ₂ (4-Py)], [ZA7426; H, F, Cl, Cl, NHPh], [ZA7427; H, F, Cl, Cl , NH (2-Py)], [ZA7428; H, F, Cl, Cl, NH (3-Py)], [ZA7429; H, F, Cl, Cl, NH (4-Py)], [ZA7430; H, F, Cl, Cl, NMe ₂ ], [ZA7431; H, F, Cl, Cl, NMeEt], [ZA7432; H, F, Cl, Cl, NMePr], [ZA7433; H, F, Cl, Cl , NMeBu], [ZA7434; H, F, Cl, Cl, NMePen], [ZA7435; H, F, Cl, Cl, NMeHex], [ZA7436; H, F, Cl, Cl, NMe (i-Pr)] , [ZA7437; H, F, Cl, Cl, NMe (i-Bu)], [ZA7438; H, F, Cl, Cl, NMe (c-Pr)], [ZA7439; H, F, Cl, Cl, NMe (c-Bu)], [ZA7440; H, F, Cl, Cl, NMe (c-Pen)], [ZA7441; H, F, Cl, Cl, NMe (c-Hex)], [ZA7442; H , F, Cl, Cl, NMeCH ₂ (c-Pr)], [ZA7443; H, F, Cl, Cl, NMeCH ₂ (c-Bu)], [ZA7444; H, F, Cl, Cl, NMeCH ₂ ( c-Pen)], [ZA7445; H, F, Cl, Cl, NMeCH ₂ (c-Hex)], [ZA7446; H, F, Cl, Cl, NMeCH ₂ F], [ZA7447; H, F, Cl , Cl, NMeCHF ₂ ], [ZA7448; H, F, Cl, Cl, NMeCF ₃ ], [ZA7449; H, F, Cl, Cl, NMe (CH ₂ ) ₂ F], [ZA7450; H, F, C l, Cl, NMeCH ₂ CHF ₂ ], [ZA7451; H, F, Cl, Cl, NMeCH ₂ CHF ₃ ], [ZA7452; H, F, Cl, Cl, NMe (CH ₂ ) ₃ F], [ZA7453; H, F, Cl, Cl, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA7454; H, F, Cl, Cl, NMe (CH ₂ ) ₂ CF ₃ ], [ZA7455; H, F, Cl, Cl, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA7456; H, F, Cl, Cl, NMeCH ₂ Cl], [ZA7457; H, F, Cl, Cl, NMe (CH ₂ ) ₂ Cl], [ZA7458; H , F, Cl, Cl, NMe (CH ₂ ) ₃ Cl], [ZA7459; H, F, Cl, Cl, NMe (CH ₂ ) ₄ Cl], [ZA7460; H, F, Cl, Cl, NMe (CH ₂ ) ₅ Cl], [ZA7461; H, F, Cl, Cl, NMeCH ₂ OMe], [ZA7462; H, F, Cl, Cl, NMe (CH ₂ ) ₂ OMe], [ZA7463; H, F, Cl , Cl, NMe (CH ₂ ) ₃ OMe], [ZA7464; H, F, Cl, Cl, NMe (CH ₂ ) ₄ OMe], [ZA7465; H, F, Cl, Cl, NMeCH ₂ OEt], [ZA7466 ; H, F, Cl, Cl, NMe (CH ₂ ) ₂ OEt], [ZA7467; H, F, Cl, Cl, NMe (CH ₂ ) ₃ OEt], [ZA7468; H, F, Cl, Cl, NMeCH ₂ OPr], [ZA7469; H, F, Cl, Cl, NMe (CH ₂ ) ₂ OPr], [ZA7470; H, F, Cl, Cl, NMe (CH ₂ ) ₃ OPr], [ZA7471; H, F , Cl, Cl, NMeCH ₂ CN], [ZA7472; H, F, Cl, Cl, NMe (CH ₂ ) ₂ CN], [ZA7473; H, F, Cl, Cl, NMe (CH ₂ ) ₃ CN], [ZA7474; H, F, Cl, Cl, NMe (CH ₂ ) ₄ CN], [ZA7475; H, F, Cl, Cl, NMe (CH ₂ ) ₅ CN], [ZA7476; H, F, Cl, Cl , NMeCH ₂ CH = CH ₂ ], [ZA7477; H, F, Cl, Cl, NMeCH ₂ C≡CH], [ZA7478; H, F, Cl, Cl, NMeCH ₂ C≡CCH ₃ ], [ ZA7479; H, F, Cl, Cl, NMeCH ₂ Ph], [ZA7480; H, F, Cl, Cl, NMeCH ₂ (2-Py)], [ZA7481; H, F, Cl, Cl, NMeCH ₂ (3 -Py)], [ZA7482; H, F, Cl, Cl, NMeCH ₂ (4-Py)], [ZA7483; H, F, Cl, Cl, NMe (CH ₂ ) ₂ Ph], [ZA7484; H, F, Cl, Cl, NMe (CH ₂ ) ₂ (2-Py)], [ZA7485; H, F, Cl, Cl, NMe (CH ₂ ) ₂ (3-Py)], [ZA7486; H, F, Cl, Cl, NMe (CH ₂ ) ₂ (4-Py)], [ZA7487; H, F, Cl, Cl, NMePh], [ZA7488; H, F, Cl, Cl, NMe (2-Py)], [ZA7489; H, F, Cl, Cl, NMe (3-Py)], [ZA7490; H, F, Cl, Cl, NMe (4-Py)], [ZA7491; H, F, Cl, Cl, NEt ₂ ], [ZA7492; H, F, Cl, Cl, NEtPr], [ZA7493; H, F, Cl, Cl, NEtBu], [ZA7494; H, F, Cl, Cl, NEtPe
n], [ZA7495; H, F, Cl, Cl, NEtHex], [ZA7496; H, F, Cl, Cl, NEt (i-Pr)], [ZA7497; H, F, Cl, Cl, NEt (i -Bu)], [ZA7498; H, F, Cl, Cl, NEt (c-Pr)], [ZA7499; H, F, Cl, Cl, NEt (c-Bu)], [ZA7500; H, F, Cl, Cl, NEt (c-Pen)],

[ZA7501; H, F, Cl, Cl, NEt (c-Hex)], [ZA7502; H, F, Cl, Cl, NEtCH ₂ (c-Pr)], [ZA7503; H, F, Cl, Cl, NEtCH ₂ (c-Bu)], [ZA7504; H, F, Cl, Cl, NEtCH ₂ (c-Pen)], [ZA7505; H, F, Cl, Cl, NEtCH ₂ (c-Hex)], [ ZA7506; H, F, Cl, Cl, NEtCH ₂ F], [ZA7507; H, F, Cl, Cl, NEtCHF ₂ ], [ZA7508; H, F, Cl, Cl, NEtCF ₃ ], [ZA7509; H, F, Cl, Cl, NEt (CH ₂ ) ₂ F], [ZA7510; H, F, Cl, Cl, NEtCH ₂ CHF ₂ ], [ZA7511; H, F, Cl, Cl, NEtCH ₂ CHF ₃ ], [ ZA7512; H, F, Cl, Cl, NEt (CH ₂ ) ₃ F], [ZA7513; H, F, Cl, Cl, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA7514; H, F, Cl, Cl , NEt (CH ₂ ) ₂ CF ₃ ], [ZA7515; H, F, Cl, Cl, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA7516; H, F, Cl, Cl, NEtCH ₂ Cl], [ZA7517 ; H, F, Cl, Cl, NEt (CH ₂ ) ₂ Cl], [ZA7518; H, F, Cl, Cl, NEt (CH ₂ ) ₃ Cl], [ZA7519; H, F, Cl, Cl, NEt (CH ₂ ) ₄ Cl], [ZA7520; H, F, Cl, Cl, NEt (CH ₂ ) ₅ Cl], [ZA7521; H, F, Cl, Cl, NEtCH ₂ OMe], [ZA7522; H, F , Cl, Cl, NEt (CH ₂ ) ₂ OMe], [ZA7523; H, F, Cl, Cl, NEt (CH ₂ ) ₃ OMe], [ZA7524; H, F, Cl, Cl, NEt (CH ₂ ) ₄ OMe], [ZA7525; H, F, Cl, Cl, NEtCH ₂ OEt], [ZA7526; H, F, Cl, Cl, NEt (CH ₂ ) ₂ OEt], [ZA7527; H, F, Cl, Cl , NEt (CH ₂ ) ₃ OEt], [ZA7528; H, F, Cl, Cl, NEtCH ₂ OPr], [ZA7529; H, F, Cl, Cl, NEt (CH ₂ ) ₂ OPr], [ZA7530; H , F, Cl , Cl, NEt (CH ₂ ) ₃ OPr], [ZA7531; H, F, Cl, Cl, NEtCH ₂ CN], [ZA7532; H, F, Cl, Cl, NEt (CH ₂ ) ₂ CN], [ZA7533 ; H, F, Cl, Cl, NEt (CH ₂ ) ₃ CN], [ZA7534; H, F, Cl, Cl, NEt (CH ₂ ) ₄ CN], [ZA7535; H, F, Cl, Cl, NEt (CH ₂ ) ₅ CN], [ZA7536; H, F, Cl, Cl, NEtCH ₂ CH = CH ₂ ], [ZA7537; H, F, Cl, Cl, NEtCH ₂ C≡CH], [ZA7538; H, F, Cl, Cl, NEtCH ₂ C≡CCH ₃ ], [ZA7539; H, F, Cl, Cl, NEtCH ₂ Ph], [ZA7540; H, F, Cl, Cl, NEtCH ₂ (2-Py)], [ZA7541; H, F, Cl, Cl, NEtCH ₂ (3-Py)], [ZA7542; H, F, Cl, Cl, NEtCH ₂ (4-Py)], [ZA7543; H, F, Cl, Cl , NEt (CH ₂ ) ₂ Ph], [ZA7544; H, F, Cl, Cl, NEt (CH ₂ ) ₂ (2-Py)], [ZA7545; H, F, Cl, Cl, NEt (CH ₂ ) ₂ (3-Py)], [ZA7546; H, F, Cl, Cl, NEt (CH ₂ ) ₂ (4-Py)], [ZA7547; H, F, Cl, Cl, NEtPh], [ZA7548; H , F, Cl, Cl, NEt (2-Py)], [ZA7549; H, F, Cl, Cl, NEt (3-Py)], [ZA7550; H, F, Cl, Cl, NEt (4-Py )], [ZA7551; H, F, Cl, Cl, Pyr], [ZA7552; H, F, Cl, Cl, Pip], [ZA7553; H, F, Cl, Cl, Mor], [ZA7554; H, F, Cl, Cl, OMe], [ZA7555; H, F, Cl, Cl, OEt], [ZA7556; H, F, Cl, Cl, OPr], [ZA7557; H, F, Cl, Cl, OBu] , [ZA7558; H, F, Cl, Cl, OPen], [ZA7559; H, F, Cl, Cl, OHex], [ZA7560; H, F, Cl, Cl, O (i-Pr)], [ZA7561 ; H, F, Cl, Cl, O (i-Bu)], [ZA7562; H, F, Cl, Cl, O (c-Pr)], [ZA7563; H, F, Cl , Cl, O (c-Bu)], [ZA7564; H, F, Cl, Cl, O (c-Pen)], [ZA7565; H, F, Cl, Cl, O (c-Hex)], [ ZA7566; H, F, Cl, Cl, OCH ₂ (c-Pr)], [ZA7567; H, F, Cl, Cl, OCH ₂ (c-Bu)], [ZA7568; H, F, Cl, Cl, OCH ₂ (c-Pen)], [ZA7569; H, F, Cl, Cl, OCH ₂ (c-Hex)], [ZA7570; H, F, Cl, Cl, OCH ₂ F], [ZA7571; H, F, Cl, Cl, OCHF ₂ ], [ZA7572; H, F, Cl, Cl, OCF ₃ ], [ZA7573; H, F, Cl, Cl, O (CH ₂ ) ₂ F], [ZA7574; H, F, Cl, Cl, OCH ₂ CHF ₂ ], [ZA7575; H, F, Cl, Cl, OCH ₂ CHF ₃ ], [ZA7576; H, F, Cl, Cl, O (CH ₂ ) ₃ F], [ ZA7577; H, F, Cl, Cl, O (CH ₂ ) ₂ CHF ₂ ], [ZA7578; H, F, Cl, Cl, O (CH ₂ ) ₂ CF ₃ ], [ZA7579; H, F, Cl, Cl, OCH ₂ CH (CF ₃ ) ₂ ], [ZA7580; H, F, Cl, Cl, OCH ₂ Cl], [ZA7581; H, F, Cl, Cl, O (CH ₂ ) ₂ Cl], [ZA7582 ; H, F, Cl, Cl, O (CH ₂ ) ₃ Cl], [ZA7583; H, F, Cl, Cl, O (CH ₂ ) ₄ Cl], [ZA7584; H, F, Cl, Cl, O (CH ₂ ) ₅ Cl], [ZA7585; H, F, Cl, Cl, OCH ₂ OMe], [ZA7586; H, F, Cl, Cl, O (CH ₂ ) ₂ OMe], [ZA7587; H, F , Cl, Cl, O (CH ₂ ) ₃ OMe], [ZA7588; H, F, Cl, Cl, O (CH ₂ ) ₄ OMe], [ZA7589; H, F, Cl, Cl, OCH ₂ OEt], [ZA7590; H, F, Cl, Cl, O (CH ₂ ) ₂ OEt], [ZA7591; H, F, Cl, Cl, O (CH ₂ ) ₃ OEt], [ZA7592; H, F, Cl, Cl , OCH ₂ OPr], [ZA7593; H, F, Cl, Cl, O (CH ₂ ) ₂ OPr], [ZA7594; H, F, Cl, Cl, O (CH ₂ ) ₃ OP r], [ZA7595; H, F, Cl, Cl, OCH ₂ CN], [ZA7596; H, F, Cl, Cl, O (CH ₂ ) ₂ CN], [ZA7597; H, F, Cl, Cl, O (CH ₂ ) ₃ CN], [ZA7598; H, F, Cl, Cl, O (CH ₂ ) ₄ CN], [ZA7599; H, F, Cl, Cl, O (CH ₂ ) ₅ CN], [ ZA7600; H, F, Cl, Cl, OCH ₂ CH = CH ₂ ], [ZA7601; H, F, Cl, Cl, OCH ₂ C≡CH], [ZA7602; H, F, Cl, Cl, OCH ₂ C ≡CCH ₃ ], [ZA7603; H, F, Cl, Cl, OCH ₂ Ph], [ZA7604; H, F, Cl, Cl, OCH ₂ (2-Py)], [ZA7605; H, F, Cl, Cl, OCH ₂ (3-Py)], [ZA7606; H, F, Cl, Cl, OCH ₂ (4-Py)], [ZA7607; H, F, Cl, Cl, O (CH ₂ ) ₂ Ph] , [ZA7608; H, F, Cl, Cl, O (CH ₂ ) ₂ (2-Py)], [ZA7609; H, F, Cl, Cl, O (CH ₂ ) ₂ (3-Py)], [ ZA7610; H, F, Cl, Cl, O (CH ₂ ) ₂ (4-Py)], [ZA7611; H, F, Cl, Cl, OPh], [ZA7612; H, F, Cl, Cl, O ( 2-Py)], [ZA7613; H, F, Cl, Cl, O (3-Py)], [ZA7614; H, F, Cl, Cl, O (4-Py)], [ZA7615; H, F , Cl, Cl, Me], [ZA7616; H, F, Cl, Cl, Et], [ZA7617; H, F, Cl, Cl, Pr], [ZA7618; H, F, Cl, Cl, Bu], [ZA7619; H, F, Cl, Cl, Pen], [ZA7620; H, F, Cl, Cl, Hex], [ZA7621; H, F, Cl, Cl, (i-Pr)], [ZA7622; H , F, Cl, Cl, (i-Bu)], [ZA7623; H, F, Cl, Cl, (c-Pr)], [ZA7624; H, F, Cl, Cl, (c-Bu)], [ZA7625; H, F, Cl, Cl, (c-Pen)], [ZA7626; H, F, Cl, Cl, (c-Hex)], [ZA7627; H, F, Cl, Cl, CH ₂ ( c-Pr)], [ZA7628; H, F, Cl, Cl, CH ₂ (c-Bu)], [ZA7629; H , F, Cl, Cl, CH ₂ (c-Pen)], [ZA7630; H, F, Cl, Cl, CH ₂ (c-Hex)], [ZA7631; H, F, Cl, Cl, CH ₂ F ], [ZA7632; H, F, Cl, Cl, CHF ₂ ], [ZA7633; H, F, Cl, Cl, CF ₃ ], [ZA7634; H, F, Cl, Cl, (CH ₂ ) ₂ F] , [ZA7635; H, F, Cl, Cl, CH ₂ CHF ₂ ], [ZA7636; H, F, Cl, Cl, CH ₂ CHF ₃ ], [ZA7637; H, F, Cl, Cl, (CH ₂ ) ₃ F], [ZA7638; H, F, Cl, Cl, (CH ₂ ) ₂ CHF ₂ ], [ZA7639; H, F, Cl, Cl, (CH ₂ ) ₂ CF ₃ ], [ZA7640; H, F , Cl, Cl, CH ₂ CH (CF ₃ ) ₂ ], [ZA7641; H, F, Cl, Cl, CH ₂ Cl], [ZA7642; H, F, Cl, Cl, (CH ₂ ) ₂ Cl], [ZA7643; H, F, Cl, Cl, (CH ₂ ) ₃ Cl], [ZA7644; H, F, Cl, Cl, (CH ₂ ) ₄ Cl], [ZA7645; H, F, Cl, Cl, ( CH ₂ ) ₅ Cl], [ZA7646; H, F, Cl, Cl, CH ₂ OMe], [ZA7647; H, F, Cl, Cl, (CH ₂ ) ₂ OMe], [ZA7648; H, F, Cl , Cl, (CH ₂ ) ₃ OMe], [ZA7649; H, F, Cl, Cl, (CH ₂ ) ₄ OMe], [ZA7650; H, F, Cl, Cl, CH ₂ OEt], [ZA7651; H , F, Cl, Cl, (CH ₂ ) ₂ OEt], [ZA7652; H, F, Cl, Cl, (CH ₂ ) ₃ OEt], [ZA7653; H, F, Cl, Cl, CH ₂ OPr], [ZA7654; H, F, Cl, Cl, (CH ₂ ) ₂ OPr], [ZA7655; H, F, Cl, Cl, (CH ₂ ) ₃ OPr], [ZA7656; H, F, Cl, Cl, CH ₂ CN], [ZA7657; H, F, Cl, Cl, (CH ₂ ) ₂ CN], [ZA7658; H, F, Cl, Cl, (CH ₂ ) ₃ CN], [ZA7659; H, F, Cl , Cl, (CH ₂ ) ₄ CN], [ZA7660; H, F, Cl, Cl, (CH ₂ ) ₅ CN], [ZA7661; H, F , Cl, Cl, CH ₂ CH = CH ₂ ], [ZA7662; H, F, Cl, Cl, CH ₂ C≡CH], [ZA7663; H, F, Cl, Cl, CH ₂ C≡CCH ₃ ], [ZA7664; H, F, Cl, Cl, CH ₂ Ph], [ZA7665; H, F, Cl, Cl, CH ₂ (2-Py)], [ZA7666; H, F, Cl, Cl, CH ₂ ( 3-Py)], [ZA7667; H, F, Cl, Cl, CH ₂ (4-Py)], [ZA7668; H, F, Cl, Cl, (CH ₂ ) ₂ Ph], [ZA7669; H, F, Cl, Cl, (CH ₂ ) ₂ (2-Py)], [ZA7670; H, F, Cl, Cl, (CH ₂ ) ₂ (3-Py)], [ZA7671; H, F, Cl, Cl, (CH ₂ ) ₂ (4-Py)], [ZA7672; H, F, Cl, Cl, Ph], [ZA7673; H, F, Cl, Cl, 2-Py], [ZA7674; H, F , Cl, Cl, 3-Py], [ZA7675; H, F, Cl, Cl, 4-Py], [ZA7676; H, F, Et, H, NHMe], [ZA7677; H, F, Et, H , NHEt], [ZA7678; H, F, Et, H, NHPr], [ZA7679; H, F, Et, H, NHBu], [ZA7680; H, F, Et, H, NHPen], [ZA7681; H , F, Et, H, NHHex], [ZA7682; H, F, Et, H, NH (i-Pr)], [ZA7683; H, F, Et, H, NH (i-Bu)], [ZA7684 ; H, F, Et, H, NH (c-Pr)], [ZA7685; H, F, Et, H, NH (c-Bu)], [ZA7686; H, F, Et, H, NH (c -Pen)], [ZA7687; H, F, Et, H, NH (c-Hex)], [ZA7688; H, F, Et, H, NHCH ₂ (c-Pr)], [ZA7689; H, F , Et, H, NHCH ₂ (c-Bu)], [ZA7690; H, F, Et, H, NHCH ₂ (c-Pen)], [ZA7691; H, F, Et, H, NHCH ₂ (c- Hex)], [ZA7692; H, F, Et, H, NHCH ₂ F], [ZA7693; H, F, Et, H, NHCHF ₂ ], [ZA7694; H, F, Et, H, NHCF ₃ ], [ZA7695; H, F, Et, H, NH (CH ₂ ) ₂ F], [ZA7696; H, F, Et, H, NHCH ₂ CHF ₂ ], [ZA7697; H, F, Et, H, NHCH ₂ CHF ₃ ], [ZA7698; H, F, Et, H, NH (CH ₂ ) ₃ F], [ZA7699; H, F, Et, H, NH (CH ₂ ) ₂ CHF ₂ ], [ZA7700; H, F, Et, H, NH (CH ₂ ) ₂ CF ₃ ], [ZA7701; H, F, Et, H, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA7702; H, F, Et, H, NHCH ₂ Cl], [ZA7703; H, F, Et, H, NH (CH ₂ ) ₂ Cl], [ZA7704; H , F, Et, H, NH (CH ₂ ) ₃ Cl], [ZA7705; H, F, Et, H, NH (CH ₂ ) ₄ Cl], [ZA7706; H, F, Et, H, NH (CH ₂ ) ₅ Cl], [ZA7707; H, F, Et, H, NHCH ₂ OMe], [ZA7708; H, F, Et, H, NH (CH ₂ ) ₂ OMe], [ZA7709; H, F, Et , H, NH (CH ₂ ) ₃ OMe], [ZA7710; H, F, Et, H, NH (CH ₂ ) ₄ OMe], [ZA7711; H, F, Et, H, NHCH ₂ OEt], [ZA7712 ; H, F, Et, H, NH (CH ₂ ) ₂ OEt], [ZA7713; H, F, Et, H, NH (CH ₂ ) ₃ OEt], [ZA7714; H, F, Et, H, NHCH ₂ OPr], [ZA7715; H, F, Et, H, NH (CH ₂ ) ₂ OPr], [ZA7716; H, F, Et, H, NH (CH ₂ ) ₃ OPr], [ZA7717; H, F , Et, H, NHCH ₂ CN], [ZA7718; H, F, Et, H, NH (CH ₂ ) ₂ CN], [ZA7719; H, F, Et, H, NH (CH ₂ ) ₃ CN], [ZA7720; H, F, Et, H, NH (CH ₂ ) ₄ CN], [ZA7721; H, F, Et, H, NH (CH ₂ ) ₅ CN], [ZA7722; H, F, Et, H , NHCH ₂ CH = CH ₂ ], [ZA7723; H, F, Et, H, NHCH ₂ C≡CH], [ZA7724; H, F, Et, H, NHCH ₂ C≡CCH ₃ ], [ZA7725; H , F, Et, H, NHCH ₂ Ph], [ZA7726; H, F, Et, H, NHCH ₂ (2-Py) ], [ZA7727; H, F, Et, H, NHCH ₂ (3-Py)], [ZA7728; H, F, Et, H, NHCH ₂ (4-Py)], [ZA7729; H, F, Et , H, NH (CH ₂ ) ₂ Ph], [ZA7730; H, F, Et, H, NH (CH ₂ ) ₂ (2-Py)], [ZA7731; H, F, Et, H, NH (CH ₂ ) ₂ (3-Py)], [ZA7732; H, F, Et, H, NH (CH ₂ ) ₂ (4-Py)], [ZA7733; H, F, Et, H, NHPh], [ZA7734 ; H, F, Et, H, NH (2-Py)], [ZA7735; H, F, Et, H, NH (3-Py)], [ZA7736; H, F, Et, H, NH (4 -Py)], [ZA7737; H, F, Et, H, NMe ₂ ], [ZA7738; H, F, Et, H, NMeEt], [ZA7739; H, F, Et, H, NMePr], [ZA7740 ; H, F, Et, H, NMeBu], [ZA7741; H, F, Et, H, NMePen], [ZA7742; H, F, Et, H, NMeHex], [ZA7743; H, F, Et, H , NMe (i-Pr)], [ZA7744; H, F, Et
, H, NMe (i-Bu)], [ZA7745; H, F, Et, H, NMe (c-Pr)], [ZA7746; H, F, Et, H, NMe (c-Bu)], [ ZA7747; H, F, Et, H, NMe (c-Pen)], [ZA7748; H, F, Et, H, NMe (c-Hex)], [ZA7749; H, F, Et, H, NMeCH ₂ (c-Pr)], [ZA7750; H, F, Et, H, NMeCH ₂ (c-Bu)],

[ZA7751; H, F, Et, H, NMeCH ₂ (c-Pen)], [ZA7752; H, F, Et, H, NMeCH ₂ (c-Hex)], [ZA7753; H, F, Et, H , NMeCH ₂ F], [ZA7754; H, F, Et, H, NMeCHF ₂ ], [ZA7755; H, F, Et, H, NMeCF ₃ ], [ZA7756; H, F, Et, H, NMe (CH ₂ ) ₂ F], [ZA7757; H, F, Et, H, NMeCH ₂ CHF ₂ ], [ZA7758; H, F, Et, H, NMeCH ₂ CHF ₃ ], [ZA7759; H, F, Et, H , NMe (CH ₂ ) ₃ F], [ZA7760; H, F, Et, H, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA7761; H, F, Et, H, NMe (CH ₂ ) ₂ CF ₃ ], [ZA7762; H, F, Et, H, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA7763; H, F, Et, H, NMeCH ₂ Cl], [ZA7764; H, F, Et, H, NMe (CH ₂ ) ₂ Cl], [ZA7765; H, F, Et, H, NMe (CH ₂ ) ₃ Cl], [ZA7766; H, F, Et, H, NMe (CH ₂ ) ₄ Cl], [ ZA7767; H, F, Et, H, NMe (CH ₂ ) ₅ Cl], [ZA7768; H, F, Et, H, NMeCH ₂ OMe], [ZA7769; H, F, Et, H, NMe (CH ₂ ) ₂ OMe], [ZA7770; H, F, Et, H, NMe (CH ₂ ) ₃ OMe], [ZA7771; H, F, Et, H, NMe (CH ₂ ) ₄ OMe], [ZA7772; H, F, Et, H, NMeCH ₂ OEt], [ZA7773; H, F, Et, H, NMe (CH ₂ ) ₂ OEt], [ZA7774; H, F, Et, H, NMe (CH ₂ ) ₃ OEt] , [ZA7775; H, F, Et, H, NMeCH ₂ OPr], [ZA7776; H, F, Et, H, NMe (CH ₂ ) ₂ OPr], [ZA7777; H, F, Et, H, NMe ( CH ₂ ) ₃ OPr], [ZA7778; H, F, Et, H, NMeCH ₂ CN], [ZA7779; H, F, Et, H, NMe (CH ₂ ) ₂ CN], [ZA7780; H, F, Et, H, NMe (CH ₂ ) ₃ CN], [ZA778 1; H, F, Et, H, NMe (CH 2) 4 CN], [ZA7782; H, F, Et, H, NMe (CH 2) 5 CN], [ZA7783; H, F, Et, H, NMeCH ₂ CH = CH ₂ ], [ZA7784; H, F, Et, H, NMeCH ₂ C≡CH], [ZA7785; H, F, Et, H, NMeCH ₂ C≡CCH ₃ ], [ZA7786; H, F, Et, H, NMeCH ₂ Ph], [ZA7787; H, F, Et, H, NMeCH ₂ (2-Py)], [ZA7788; H, F, Et, H, NMeCH ₂ (3-Py)] , [ZA7789; H, F, Et, H, NMeCH ₂ (4-Py)], [ZA7790; H, F, Et, H, NMe (CH ₂ ) ₂ Ph], [ZA7791; H, F, Et, H, NMe (CH ₂ ) ₂ (2-Py)], [ZA7792; H, F, Et, H, NMe (CH ₂ ) ₂ (3-Py)], [ZA7793; H, F, Et, H, NMe (CH ₂ ) ₂ (4-Py)], [ZA7794; H, F, Et, H, NMePh], [ZA7795; H, F, Et, H, NMe (2-Py)], [ZA7796; H , F, Et, H, NMe (3-Py)], [ZA7797; H, F, Et, H, NMe (4-Py)], [ZA7798; H, F, Et, H, NEt ₂ ], [ ZA7799; H, F, Et, H, NEtPr], [ZA7800; H, F, Et, H, NEtBu], [ZA7801; H, F, Et, H, NEtPen], [ZA7802; H, F, Et, H, NEtHex], [ZA7803; H, F, Et, H, NEt (i-Pr)], [ZA7804; H, F, Et, H, NEt (i-Bu)], [ZA7805; H, F, Et, H, NEt (c-Pr)], [ZA7806; H, F, Et, H, NEt (c-Bu)], [ZA7807; H, F, Et, H, NEt (c-Pen)], [ZA7808; H, F, Et, H, NEt (c-Hex)], [ZA7809; H, F, Et, H, NEtCH ₂ (c-Pr)], [ZA7810; H, F, Et, H, NEtCH ₂ (c-Bu)], [ZA7811; H, F, Et, H, NEtCH ₂ (c-Pen)], [ZA7812; H, F, Et, H, NEtCH ₂ (c-Hex)], [ ZA7813; H, F, Et, H, NEtCH ₂ F], [ZA7814; H, F, Et, H, NEtCHF ₂ ], [ZA7815; H, F, Et, H, NEtCF ₃ ], [ZA7816; H, F, Et, H, NEt (CH ₂ ) ₂ F], [ZA7817; H, F, Et, H, NEtCH ₂ CHF ₂ ], [ZA7818; H, F, Et, H, NEtCH ₂ CHF ₃ ], [ZA7819; H, F, Et, H, NEt (CH ₂ ) ₃ F], [ZA7820; H, F, Et, H, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA7821; H, F, Et, H, NEt (CH ₂ ) ₂ CF ₃ ], [ZA7822; H, F, Et, H, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA7823; H, F, Et, H, NEtCH ₂ Cl], [ZA7824; H, F, Et, H, NEt ( CH ₂ ) ₂ Cl], [ZA7825; H, F, Et, H, NEt (CH ₂ ) ₃ Cl], [ZA7826; H, F, Et, H, NEt (CH ₂ ) ₄ Cl], [ZA7827; H, F, Et, H, NEt (CH ₂ ) ₅ Cl], [ZA7828; H, F, Et, H, NEtCH ₂ OMe], [ZA7829; H, F, Et, H, NEt (CH ₂ ) ₂ OMe], [ZA7830; H, F, Et, H, NEt (CH ₂ ) ₃ OMe], [ZA7831; H, F, Et, H, NEt (CH ₂ ) ₄ OMe], [ZA7832; H, F, Et, H, NEtCH ₂ OEt], [ZA7833; H, F, Et, H, NEt (CH ₂ ) ₂ OEt], [ZA7834; H, F, Et, H, NEt (CH ₂ ) ₃ OEt], [ ZA7835; H, F, Et, H, NEtCH ₂ OPr], [ZA7836; H, F, Et, H, NEt (CH ₂ ) ₂ OPr], [ZA7837; H, F, Et, H, NEt (CH ₂ ) ₃ OPr], [ZA7838; H, F, Et, H, NEtCH ₂ CN], [ZA7839; H, F, Et, H, NEt (CH ₂ ) ₂ CN], [ZA7840; H, F, Et, H, NEt (CH ₂ ) ₃ CN], [ZA7841; H, F, Et, H, NEt (CH ₂ ) ₄ CN], [ZA7842; H, F, Et, H, NEt (CH ₂ ) ₅ CN] , [ZA7843; H, F, Et, H, NEtCH ₂ CH = CH ₂ ], [ZA7844; H, F, Et, H, NEtCH ₂ C≡CH], [ZA7845; H, F, Et, H, NEtCH ₂ C≡CCH ₃ ], [ZA7846; H, F, Et, H, NEtCH ₂ Ph], [ZA7847; H, F, Et, H, NEtCH ₂ (2-Py)], [ZA7848; H, F, Et, H, NEtCH ₂ (3-Py)], [ZA7849; H, F, Et, H, NEtCH ₂ (4-Py)], [ZA7850; H, F, Et, H, NEt (CH ₂ ) ₂ Ph], [ZA7851; H, F, Et, H, NEt ( CH ₂ ) ₂ (2-Py)], [ZA7852; H, F, Et, H, NEt (CH ₂ ) ₂ (3-Py)], [ZA7853; H, F, Et, H, NEt (CH ₂ ) ₂ (4-Py)], [ZA7854; H, F, Et, H, NEtPh], [ZA7855; H, F, Et, H, NEt (2-Py)], [ZA7856; H, F, Et , H, NEt (3-Py)], [ZA7857; H, F, Et, H, NEt (4-Py)], [ZA7858; H, F, Et, H, Pyr], [ZA7859; H, F , Et, H, Pip], [ZA7860; H, F, Et, H, Mor], [ZA7861; H, F, Et, H, OMe], [ZA7862; H, F, Et, H, OEt], [ZA7863; H, F, Et, H, OPr], [ZA7864; H, F, Et, H, OBu], [ZA7865; H, F, Et, H, OPen], [ZA7866; H, F, Et , H, OHex], [ZA7867; H, F, Et, H, O (i-Pr)], [ZA7868; H, F, Et, H, O (i-Bu)], [ZA7869; H, F , Et, H, O (c-Pr)], [ZA7870; H, F, Et, H, O (c-Bu)], [ZA7871; H, F, Et, H, O (c-Pen)] , [ZA7872; H, F, Et, H, O (c-Hex)], [ZA7873; H, F, Et, H, OCH ₂ (c-Pr)], [ZA7874; H, F, Et, H , OCH ₂ (c-Bu)], [ZA7875; H, F, Et, H, OCH ₂ (c-Pen)], [ZA7876; H, F, Et, H, OCH ₂ (c-Hex)], [ZA7877; H, F, Et, H, OCH ₂ F], [ZA7878; H, F, Et, H, OCHF ₂ ], [ZA 7879; H, F, Et, H, OCF ₃ ], [ZA7880; H, F, Et, H, O (CH ₂ ) ₂ F], [ZA7881; H, F, Et, H, OCH ₂ CHF ₂ ] , [ZA7882; H, F, Et, H, OCH ₂ CHF ₃ ], [ZA7883; H, F, Et, H, O (CH ₂ ) ₃ F], [ZA7884; H, F, Et, H, O (CH ₂ ) ₂ CHF ₂ ], [ZA7885; H, F, Et, H, O (CH ₂ ) ₂ CF ₃ ], [ZA7886; H, F, Et, H, OCH ₂ CH (CF ₃ ) ₂ ] , [ZA7887; H, F, Et, H, OCH ₂ Cl], [ZA7888; H, F, Et, H, O (CH ₂ ) ₂ Cl], [ZA7889; H, F, Et, H, O ( CH ₂ ) ₃ Cl], [ZA7890; H, F, Et, H, O (CH ₂ ) ₄ Cl], [ZA7891; H, F, Et, H, O (CH ₂ ) ₅ Cl], [ZA7892; H, F, Et, H, OCH ₂ OMe], [ZA7893; H, F, Et, H, O (CH ₂ ) ₂ OMe], [ZA7894; H, F, Et, H, O (CH ₂ ) ₃ OMe], [ZA7895; H, F, Et, H, O (CH ₂ ) ₄ OMe], [ZA7896; H, F, Et, H, OCH ₂ OEt], [ZA7897; H, F, Et, H, O (CH ₂ ) ₂ OEt], [ZA7898; H, F, Et, H, O (CH ₂ ) ₃ OEt], [ZA7899; H, F, Et, H, OCH ₂ OPr], [ZA7900; H, F, Et, H, O (CH ₂ ) ₂ OPr], [ZA7901; H, F, Et, H, O (CH ₂ ) ₃ OPr], [ZA7902; H, F, Et, H, OCH ₂ CN] , [ZA7903; H, F, Et, H, O (CH ₂ ) ₂ CN], [ZA7904; H, F, Et, H, O (CH ₂ ) ₃ CN], [ZA7905; H, F, Et, H, O (CH ₂ ) ₄ CN], [ZA7906; H, F, Et, H, O (CH ₂ ) ₅ CN], [ZA7907; H, F, Et, H, OCH ₂ CH = CH ₂ ], [ZA7908; H, F, Et, H, OCH ₂ C≡CH], [ZA7909; H, F, Et, H, OCH ₂ C≡CCH ₃ ], [ZA7910; H, F, Et, H, OCH ₂ Ph], [ZA7911; H, F, Et, H, OCH ₂ (2-Py)], [ZA7912; H, F, Et, H, OCH ₂ (3-Py)], [ZA7913; H, F, Et, H, OCH ₂ (4-Py)], [ZA7914; H, F, Et, H, O (CH ₂ ) ₂ Ph], [ZA7915; H, F, Et, H, O (CH ₂ ) ₂ (2-Py)], [ZA7916; H, F, Et, H, O (CH ₂ ) ₂ (3-Py)], [ZA7917; H, F, Et, H, O (CH ₂ ) ₂ (4 -Py)], [ZA7918; H, F, Et, H, OPh], [ZA7919; H, F, Et, H, O (2-Py)], [ZA7920; H, F, Et, H, O (3-Py)], [ZA7921; H, F, Et, H, O (4-Py)], [ZA7922; H, F, Et, H, Me], [ZA7923; H, F, Et, H , Et], [ZA7924; H, F, Et, H, Pr], [ZA7925; H, F, Et, H, Bu], [ZA7926; H, F, Et, H, Pen], [ZA7927; H , F, Et, H, Hex], [ZA7928; H, F, Et, H, (i-Pr)], [ZA7929; H, F, Et, H, (i-Bu)], [ZA7930; H , F, Et, H, (c-Pr)], [ZA7931; H, F, Et, H, (c-Bu)], [ZA7932; H, F, Et, H, (c-Pen)], [ZA7933; H, F, Et, H, (c-Hex)], [ZA7934; H, F, Et, H, CH ₂ (c-Pr)], [ZA7935; H, F, Et, H, CH ₂ (c-Bu)], [ZA7936; H, F, Et, H, CH ₂ (c-Pen)], [ZA7937; H, F, Et, H, CH ₂ (c-Hex)], [ZA7938 ; H, F, Et, H, CH ₂ F], [ZA7939; H, F, Et, H, CHF ₂ ], [ZA7940; H, F, Et, H, CF ₃ ], [ZA7941; H, F , Et, H, (CH ₂ ) ₂ F], [ZA7942; H, F, Et, H, CH ₂ CHF ₂ ], [ZA7943; H, F, Et, H, CH ₂ CHF ₃ ], [ZA7944; H, F, Et, H, (CH 2) 3 F], [ZA7945; H, F, Et, H, (CH 2) 2 CHF 2], [ZA7946; H, F, Et, H, (CH 2 ) ₂ CF ₃ ], [ZA7947; H, F, Et, H, CH ₂ CH (CF ₃ ) ₂ ], [ZA7948; H, F, Et, H, CH ₂ Cl], [ZA7949; H, F, Et, H, (CH ₂ ) ₂ Cl], [ZA7950; H, F, Et, H, (CH ₂ ) ₃ Cl], [ZA7951; H, F, Et, H, (CH ₂ ) ₄ Cl], [ZA7952; H , F, Et, H, (CH ₂ ) ₅ Cl], [ZA7953; H, F, Et, H, CH ₂ OMe], [ZA7954; H, F, Et, H, (CH ₂ ) ₂ OMe], [ZA7955; H, F, Et, H, (CH ₂ ) ₃ OMe], [ZA7956; H, F, Et, H, (CH ₂ ) ₄ OMe], [ZA7957; H, F, Et, H, CH ₂ OEt], [ZA7958; H, F, Et, H, (CH ₂ ) ₂ OEt], [ZA7959; H, F, Et, H, (CH ₂ ) ₃ OEt], [ZA7960; H, F, Et , H, CH ₂ OPr], [ZA7961; H, F, Et, H, (CH ₂ ) ₂ OPr], [ZA7962; H, F, Et, H, (CH ₂ ) ₃ OPr], [ZA7963; H , F, Et, H, CH ₂ CN], [ZA7964; H, F, Et, H, (CH ₂ ) ₂ CN], [ZA7965; H, F, Et, H, (CH ₂ ) ₃ CN], [ZA7966; H, F, Et, H, (CH ₂ ) ₄ CN], [ZA7967; H, F, Et, H, (CH ₂ ) ₅ CN], [ZA7968; H, F, Et, H, CH _{2 CH = CH 2], [} ZA7969; H, F, Et, H, CH 2 C≡CH], [ZA7970; H, F, Et, H, CH 2 C≡CCH 3], [ZA7971; H, F , Et, H, CH ₂ Ph], [ZA7972; H, F, Et, H, CH ₂ (2-Py)], [ZA7973; H, F, Et, H, CH ₂ (3-Py)], [ZA7974; H, F, Et, H, CH ₂ (4-Py)], [ZA7975; H, F, Et, H, (CH ₂ ) ₂ Ph], [ZA7976; H, F, Et, H, (CH ₂ ) ₂ (2-Py)], [ZA7977; H, F, Et, H, (CH ₂ ) ₂ (3-Py)], [ZA7978; H, F, Et, H, (CH ₂ ) ₂ (4-Py)], [ZA7979; H, F, Et, H, Ph], [ZA7980; H, F, Et, H, 2-Py], [ZA7981; H, F, Et, H, 3-Py], [ZA7982; H, F, Et, H, 4-Py], [ZA7983; H, F, Me, Et, NHMe], [ZA7984; H, F, Me, Et, NHEt], [ZA7985; H, F, Me, Et, NHPr] , [ZA7986; H, F, Me, Et, NHBu], [ZA7987; H, F, Me, Et, NHPen], [ZA7988; H, F, Me, Et, NHHex], [ZA7989; H, F, Me, Et, NH (i-Pr)], [ZA7990; H, F, Me, Et, NH (i-Bu)], [ZA7991; H, F, Me, Et, NH (c-Pr)], [ZA7992; H, F, Me, Et, NH (c-Bu)], [ZA7993; H, F, Me, Et, NH (c-Pen)], [ZA7994; H, F, Me, Et, NH (c-Hex)], [ZA7995; H, F, Me, Et, NHCH ₂ (c-Pr)], [ZA7996; H, F, Me, Et, NHCH ₂ (c-Bu)], [ZA7997; H, F, Me, Et, NHCH ₂ (c-Pe
n)], [ZA7998; H, F, Me, Et, NHCH ₂ (c-Hex)], [ZA7999; H, F, Me, Et, NHCH ₂ F], [ZA8000; H, F, Me, Et , NHCHF ₂ ],

[ZA8001; H, F, Me, Et, NHCF ₃ ], [ZA8002; H, F, Me, Et, NH (CH ₂ ) ₂ F], [ZA8003; H, F, Me, Et, NHCH ₂ CHF ₂ ], [ZA8004; H, F, Me, Et, NHCH ₂ CHF ₃ ], [ZA8005; H, F, Me, Et, NH (CH ₂ ) ₃ F], [ZA8006; H, F, Me, Et, NH (CH ₂ ) ₂ CHF ₂ ], [ZA8007; H, F, Me, Et, NH (CH ₂ ) ₂ CF ₃ ], [ZA8008; H, F, Me, Et, NHCH ₂ CH (CF ₃ ) ₂ ], [ZA8009; H, F, Me, Et, NHCH ₂ Cl], [ZA8010; H, F, Me, Et, NH (CH ₂ ) ₂ Cl], [ZA8011; H, F, Me, Et, NH (CH ₂ ) ₃ Cl], [ZA8012; H, F, Me, Et, NH (CH ₂ ) ₄ Cl], [ZA8013; H, F, Me, Et, NH (CH ₂ ) ₅ Cl], [ZA8014 ; H, F, Me, Et, NHCH ₂ OMe], [ZA8015; H, F, Me, Et, NH (CH ₂ ) ₂ OMe], [ZA8016; H, F, Me, Et, NH (CH ₂ ) ₃ OMe], [ZA8017; H, F, Me, Et, NH (CH ₂ ) ₄ OMe], [ZA8018; H, F, Me, Et, NHCH ₂ OEt], [ZA8019; H, F, Me, Et , NH (CH ₂ ) ₂ OEt], [ZA8020; H, F, Me, Et, NH (CH ₂ ) ₃ OEt], [ZA8021; H, F, Me, Et, NHCH ₂ OPr], [ZA8022; H , F, Me, Et, NH (CH ₂ ) ₂ OPr], [ZA8023; H, F, Me, Et, NH (CH ₂ ) ₃ OPr], [ZA8024; H, F, Me, Et, NHCH ₂ CN ], [ZA8025; H, F, Me, Et, NH (CH ₂ ) ₂ CN], [ZA8026; H, F, Me, Et, NH (CH ₂ ) ₃ CN], [ZA8027; H, F, Me , Et, NH (CH ₂ ) ₄ CN], [ZA8028; H, F, Me, Et, NH (CH ₂ ) ₅ CN], [ZA8029; H, F, Me, Et, NHCH ₂ CH = CH ₂ ] , [ZA8030; H, F, Me, Et, NHCH 2 C CH], [ZA8031; H, F, Me, Et, NHCH 2 C≡CCH 3], [ZA8032; H, F, Me, Et, NHCH 2 Ph], [ZA8033; H, F, Me, Et, NHCH ₂ (2-Py)], [ZA8034; H, F, Me, Et, NHCH ₂ (3-Py)], [ZA8035; H, F, Me, Et, NHCH ₂ (4-Py)], [ZA8036 ; H, F, Me, Et, NH (CH ₂ ) ₂ Ph], [ZA8037; H, F, Me, Et, NH (CH ₂ ) ₂ (2-Py)], [ZA8038; H, F, Me , Et, NH (CH ₂ ) ₂ (3-Py)], [ZA8039; H, F, Me, Et, NH (CH ₂ ) ₂ (4-Py)], [ZA8040; H, F, Me, Et , NHPh], [ZA8041; H, F, Me, Et, NH (2-Py)], [ZA8042; H, F, Me, Et, NH (3-Py)], [ZA8043; H, F, Me , Et, NH (4-Py)], [ZA8044; H, F, Me, Et, NMe ₂ ], [ZA8045; H, F, Me, Et, NMeEt], [ZA8046; H, F, Me, Et , NMePr], [ZA8047; H, F, Me, Et, NMeBu], [ZA8048; H, F, Me, Et, NMePen], [ZA8049; H, F, Me, Et, NMeHex], [ZA8050; H , F, Me, Et, NMe (i-Pr)], [ZA8051; H, F, Me, Et, NMe (i-Bu)], [ZA8052; H, F, Me, Et, NMe (c-Pr )], [ZA8053; H, F, Me, Et, NMe (c-Bu)], [ZA8054; H, F, Me, Et, NMe (c-Pen)], [ZA8055; H, F, Me, Et, NMe (c-Hex)], [ZA8056; H, F, Me, Et, NMeCH ₂ (c-Pr)], [ZA8057; H, F, Me, Et, NMeCH ₂ (c-Bu)], [ZA8058; H, F, Me, Et, NMeCH ₂ (c-Pen)], [ZA8059; H, F, Me, Et, NMeCH ₂ (c-Hex)], [ZA8060; H, F, Me, Et , NMeCH ₂ F], [ZA8061; H, F, Me, Et, NMeCHF ₂ ], [ZA8062; H, F, Me, Et, NMeCF ₃ ], [ZA8063; H, F, Me, Et, NM e (CH ₂ ) ₂ F], [ZA8064; H, F, Me, Et, NMeCH ₂ CHF ₂ ], [ZA8065; H, F, Me, Et, NMeCH ₂ CHF ₃ ], [ZA8066; H, F, Me, Et, NMe (CH ₂ ) ₃ F], [ZA8067; H, F, Me, Et, NMe (CH ₂ ) ₂ CHF ₂ ], [ZA8068; H, F, Me, Et, NMe (CH ₂ ) ₂ CF ₃ ], [ZA8069; H, F, Me, Et, NMeCH ₂ CH (CF ₃ ) ₂ ], [ZA8070; H, F, Me, Et, NMeCH ₂ Cl], [ZA8071; H, F, Me , Et, NMe (CH ₂ ) ₂ Cl], [ZA8072; H, F, Me, Et, NMe (CH ₂ ) ₃ Cl], [ZA8073; H, F, Me, Et, NMe (CH ₂ ) ₄ Cl ], [ZA8074; H, F, Me, Et, NMe (CH ₂ ) ₅ Cl], [ZA8075; H, F, Me, Et, NMeCH ₂ OMe], [ZA8076; H, F, Me, Et, NMe (CH ₂ ) ₂ OMe], [ZA8077; H, F, Me, Et, NMe (CH ₂ ) ₃ OMe], [ZA8078; H, F, Me, Et, NMe (CH ₂ ) ₄ OMe], [ZA8079 ; H, F, Me, Et, NMeCH ₂ OEt], [ZA8080; H, F, Me, Et, NMe (CH ₂ ) ₂ OEt], [ZA8081; H, F, Me, Et, NMe (CH ₂ ) ₃ OEt], [ZA8082; H, F, Me, Et, NMeCH ₂ OPr], [ZA8083; H, F, Me, Et, NMe (CH ₂ ) ₂ OPr], [ZA8084; H, F, Me, Et , NMe (CH ₂ ) ₃ OPr], [ZA8085; H, F, Me, Et, NMeCH ₂ CN], [ZA8086; H, F, Me, Et, NMe (CH ₂ ) ₂ CN], [ZA8087; H , F, Me, Et, NMe (CH ₂ ) ₃ CN], [ZA8088; H, F, Me, Et, NMe (CH ₂ ) ₄ CN], [ZA8089; H, F, Me, Et, NMe (CH ₂ ) ₅ CN], [ZA8090; H, F, Me, Et, NMeCH ₂ CH = CH ₂ ], [ZA8091; H, F, Me, Et, NMeCH ₂ C≡CH], [ZA8092; H, F, Me, Et, NMeCH ₂ C≡CCH ₃ ], [ZA8093; H, F, Me, Et, NMeCH ₂ Ph], [ZA8094; H, F, Me, Et, NMeCH ₂ (2-Py)], [ZA8095 ; H, F, Me, Et, NMeCH ₂ (3-Py)], [ZA8096; H, F, Me, Et, NMeCH ₂ (4-Py)], [ZA8097; H, F, Me, Et, NMe (CH ₂ ) ₂ Ph], [ZA8098; H, F, Me, Et, NMe (CH ₂ ) ₂ (2-Py)], [ZA8099; H, F, Me, Et, NMe (CH ₂ ) ₂ ( 3-Py)], [ZA8100; H, F, Me, Et, NMe (CH ₂ ) ₂ (4-Py)], [ZA8101; H, F, Me, Et, NMePh], [ZA8102; H, F , Me, Et, NMe (2-Py)], [ZA8103; H, F, Me, Et, NMe (3-Py)], [ZA8104; H, F, Me, Et, NMe (4-Py)] , [ZA8105; H, F, Me, Et, NEt ₂ ], [ZA8106; H, F, Me, Et, NEtPr], [ZA8107; H, F, Me, Et, NEtBu], [ZA8108; H, F , Me, Et, NEtPen], [ZA8109; H, F, Me, Et, NEtHex], [ZA8110; H, F, Me, Et, NEt (i-Pr)], [ZA8111; H, F, Me, Et, NEt (i-Bu)], [ZA8112; H, F, Me, Et, NEt (c-Pr)], [ZA8113; H, F, Me, Et, NEt (c-Bu)], [ZA8114 ; H, F, Me, Et, NEt (c-Pen)], [ZA8115; H, F, Me, Et, NEt (c-Hex)], [ZA8116; H, F, Me, Et, NEtCH ₂ ( c-Pr)], [ZA8117; H, F, Me, Et, NEtCH ₂ (c-Bu)], [ZA8118; H, F, Me, Et, NEtCH ₂ (c-Pen)], [ZA8119; H , F, Me, Et, NEtCH ₂ (c-Hex)], [ZA8120; H, F, Me, Et, NEtCH ₂ F], [ZA8121; H, F, Me, Et, NEtCHF ₂ ], [ZA8122; H, F, Me, Et, NEtCF ₃ ], [ZA8123; H, F, Me, Et, NEt (CH ₂ ) ₂ F], [ZA8124; H, F, Me, E t, NEtCH ₂ CHF ₂ ], [ZA8125; H, F, Me, Et, NEtCH ₂ CHF ₃ ], [ZA8126; H, F, Me, Et, NEt (CH ₂ ) ₃ F], [ZA8127; H, F, Me, Et, NEt (CH ₂ ) ₂ CHF ₂ ], [ZA8128; H, F, Me, Et, NEt (CH ₂ ) ₂ CF ₃ ], [ZA8129; H, F, Me, Et, NEtCH ₂ CH (CF ₃ ) ₂ ], [ZA8130; H, F, Me, Et, NEtCH ₂ Cl], [ZA8131; H, F, Me, Et, NEt (CH ₂ ) ₂ Cl], [ZA8132; H, F , Me, Et, NEt (CH ₂ ) ₃ Cl], [ZA8133; H, F, Me, Et, NEt (CH ₂ ) ₄ Cl], [ZA8134; H, F, Me, Et, NEt (CH ₂ ) ₅ Cl], [ZA8135; H, F, Me, Et, NEtCH ₂ OMe], [ZA8136; H, F, Me, Et, NEt (CH ₂ ) ₂ OMe], [ZA8137; H, F, Me, Et , NEt (CH ₂ ) ₃ OMe], [ZA8138; H, F, Me, Et, NEt (CH ₂ ) ₄ OMe], [ZA8139; H, F, Me, Et, NEtCH ₂ OEt], [ZA8140; H , F, Me, Et, NEt (CH ₂ ) ₂ OEt], [ZA8141; H, F, Me, Et, NEt (CH ₂ ) ₃ OEt], [ZA8142; H, F, Me, Et, NEtCH ₂ OPr ], [ZA8143; H, F, Me, Et, NEt (CH ₂ ) ₂ OPr], [ZA8144; H, F, Me, Et, NEt (CH ₂ ) ₃ OPr], [ZA8145; H, F, Me , Et, NEtCH ₂ CN], [ZA8146; H, F, Me, Et, NEt (CH ₂ ) ₂ CN], [ZA8147; H, F, Me, Et, NEt (CH ₂ ) ₃ CN], [ZA8148 ; H, F, Me, Et, NEt (CH ₂ ) ₄ CN], [ZA8149; H, F, Me, Et, NEt (CH ₂ ) ₅ CN], [ZA8150; H, F, Me, Et, NEtCH ₂ CH = CH ₂ ], [ZA8151; H, F, Me, Et, NEtCH ₂ C≡CH], [ZA8152; H, F, Me, Et, NEtCH ₂ C≡CCH ₃ ], [ZA8 153; H, F, Me, Et, NEtCH ₂ Ph], [ZA8154; H, F, Me, Et, NEtCH ₂ (2-Py)], [ZA8155; H, F, Me, Et, NEtCH ₂ (3 -Py)], [ZA8156; H, F, Me, Et, NEtCH ₂ (4-Py)], [ZA8157; H, F, Me, Et, NEt (CH ₂ ) ₂ Ph], [ZA8158; H, F, Me, Et, NEt (CH ₂ ) ₂ (2-Py)], [ZA8159; H, F, Me, Et, NEt (CH ₂ ) ₂ (3-Py)], [ZA8160; H, F, Me, Et, NEt (CH ₂ ) ₂ (4-Py)], [ZA8161; H, F, Me, Et, NEtPh], [ZA8162; H, F, Me, Et, NEt (2-Py)], [ZA8163; H, F, Me, Et, NEt (3-Py)], [ZA8164; H, F, Me, Et, NEt (4-Py)], [ZA8165; H, F, Me, Et, Pyr ], [ZA8166; H, F, Me, Et, Pip], [ZA8167; H, F, Me, Et, Mor], [ZA8168; H, F, Me, Et, OMe], [ZA8169; H, F , Me, Et, OEt], [ZA8170; H, F, Me, Et, OPr], [ZA8171; H, F, Me, Et, OBu], [ZA8172; H, F, Me, Et, OPen], [ZA8173; H, F, Me, Et, OHex], [ZA8174; H, F, Me, Et, O (i-Pr)], [ZA8175; H, F, Me, Et, O (i-Bu) ], [ZA8176; H, F, Me, Et, O (c-Pr)], [ZA8177; H, F, Me, Et, O (c-Bu)], [ZA8178; H, F, Me, Et , O (c-Pen)], [ZA8179; H, F, Me, Et, O (c-Hex)], [ZA8180; H, F, Me, Et, OCH ₂ (c-Pr)], [ZA8181 ; H, F, Me, Et, OCH ₂ (c-Bu)], [ZA8182; H, F, Me, Et, OCH ₂ (c-Pen)], [ZA8183; H, F, Me, Et, OCH ₂ (c-Hex)], [ZA8184; H, F, Me, Et, OCH ₂ F], [ZA8185; H, F, Me, Et, OCHF ₂ ], [ZA8186; H, F, Me, Et, OCF ₃ ], [ZA8187; H, F, Me, Et, O (CH ₂ ) ₂ F], [ZA8188; H, F, Me, Et, OCH ₂ CHF ₂ ], [ZA8189; H, F, Me, Et, OCH ₂ CHF ₃ ], [ZA8190; H, F, Me, Et, O (CH ₂ ) ₃ F], [ZA8191; H, F, Me, Et, O (CH ₂ ) ₂ CHF ₂ ], [ZA8192; H, F, Me, Et, O (CH ₂ ) ₂ CF ₃ ] , [ZA8193; H, F, Me, Et, OCH ₂ CH (CF ₃ ) ₂ ], [ZA8194; H, F, Me, Et, OCH ₂ Cl], [ZA8195; H, F, Me, Et, O (CH ₂ ) ₂ Cl], [ZA8196; H, F, Me, Et, O (CH ₂ ) ₃ Cl], [ZA8197; H, F, Me, Et, O (CH ₂ ) ₄ Cl], [ZA8198 ; H, F, Me, Et, O (CH ₂ ) ₅ Cl], [ZA8199; H, F, Me, Et, OCH ₂ OMe], [ZA8200; H, F, Me, Et, O (CH ₂ ) ₂ OMe], [ZA8201; H, F, Me, Et, O (CH ₂ ) ₃ OMe], [ZA8202; H, F, Me, Et, O (CH ₂ ) ₄ OMe], [ZA8203; H, F , Me, Et, OCH ₂ OEt], [ZA8204; H, F, Me, Et, O (CH ₂ ) ₂ OEt], [ZA8205; H, F, Me, Et, O (CH ₂ ) ₃ OEt], [ZA8206; H, F, Me, Et, OCH ₂ OPr], [ZA8207; H, F, Me, Et, O (CH ₂ ) ₂ OPr], [ZA8208; H, F, Me, Et, O (CH ₂ ) ₃ OPr], [ZA8209; H, F, Me, Et, OCH ₂ CN], [ZA8210; H, F, Me, Et, O (CH ₂ ) ₂ CN], [ZA8211; H, F, Me , Et, O (CH ₂ ) ₃ CN], [ZA8212; H, F, Me, Et, O (CH ₂ ) ₄ CN], [ZA8213; H, F, Me, Et, O (CH ₂ ) ₅ CN ], [ZA8214; H, F, Me, Et, OCH ₂ CH = CH ₂ ], [ZA8215; H, F, Me, Et, OCH ₂ C≡CH], [ZA8216; H, F, Me, Et, OCH ₂ C≡CCH ₃ ], [ZA8217; H, F, Me, Et, OCH ₂ Ph], [ZA8218; H, F , Me, Et, OCH ₂ (2-Py)], [ZA8219; H, F, Me, Et, OCH ₂ (3-Py)], [ZA8220; H, F, Me, Et, OCH ₂ (4- Py)], [ZA8221; H, F, Me, Et, O (CH ₂ ) ₂ Ph], [ZA8222; H, F, Me, Et, O (CH ₂ ) ₂ (2-Py)], [ZA8223 ; H, F, Me, Et, O (CH ₂ ) ₂ (3-Py)], [ZA8224; H, F, Me, Et, O (CH ₂ ) ₂ (4-Py)], [ZA8225; H , F, Me, Et, OPh], [ZA8226; H, F, Me, Et, O (2-Py)], [ZA8227; H, F, Me, Et, O (3-Py)], [ZA8228 ; H, F, Me, Et, O (4-Py)], [ZA8229; H, F, Me, Et, Me], [ZA8230; H, F, Me, Et, Et], [ZA8231; H, F, Me, Et, Pr], [ZA8232; H, F, Me, Et, Bu], [ZA8233; H, F, Me, Et, Pen], [ZA8234; H, F, Me, Et, Hex] , [ZA8235; H, F, Me, Et, (i-Pr)], [ZA8236; H, F, Me, Et, (i-Bu)], [ZA8237; H, F, Me, Et, (c -Pr)], [ZA
8238; H, F, Me, Et, (c-Bu)], [ZA8239; H, F, Me, Et, (c-Pen)], [ZA8240; H, F, Me, Et, (c-Hex )], [ZA8241; H, F, Me, Et, CH ₂ (c-Pr)], [ZA8242; H, F, Me, Et, CH ₂ (c-Bu)], [ZA8243; H, F, Me, Et, CH ₂ (c-Pen)], [ZA8244; H, F, Me, Et, CH ₂ (c-Hex)], [ZA8245; H, F, Me, Et, CH ₂ F], [ ZA8246; H, F, Me, Et, CHF ₂ ], [ZA8247; H, F, Me, Et, CF ₃ ], [ZA8248; H, F, Me, Et, (CH ₂ ) ₂ F], [ZA8249 ; H, F, Me, Et, CH ₂ CHF ₂ ], [ZA8250; H, F, Me, Et, CH ₂ CHF ₃ ],

[ZA8251; H, F, Me, Et, (CH ₂ ) ₃ F], [ZA8252; H, F, Me, Et, (CH ₂ ) ₂ CHF ₂ ], [ZA8253; H, F, Me, Et, (CH ₂ ) ₂ CF ₃ ], [ZA8254; H, F, Me, Et, CH ₂ CH (CF ₃ ) ₂ ], [ZA8255; H, F, Me, Et, CH ₂ Cl], [ZA8256; H , F, Me, Et, (CH ₂ ) ₂ Cl], [ZA8257; H, F, Me, Et, (CH ₂ ) ₃ Cl], [ZA8258; H, F, Me, Et, (CH ₂ ) ₄ Cl], [ZA8259; H, F, Me, Et, (CH ₂ ) ₅ Cl], [ZA8260; H, F, Me, Et, CH ₂ OMe], [ZA8261; H, F, Me, Et, ( CH ₂ ) ₂ OMe], [ZA8262; H, F, Me, Et, (CH ₂ ) ₃ OMe], [ZA8263; H, F, Me, Et, (CH ₂ ) ₄ OMe], [ZA8264; H, F, Me, Et, CH ₂ OEt], [ZA8265; H, F, Me, Et, (CH ₂ ) ₂ OEt], [ZA8266; H, F, Me, Et, (CH ₂ ) ₃ OEt], [ ZA8267; H, F, Me, Et, CH ₂ OPr], [ZA8268; H, F, Me, Et, (CH ₂ ) ₂ OPr], [ZA8269; H, F, Me, Et, (CH ₂ ) ₃ OPr], [ZA8270; H, F, Me, Et, CH ₂ CN], [ZA8271; H, F, Me, Et, (CH ₂ ) ₂ CN], [ZA8272; H, F, Me, Et, ( CH ₂ ) ₃ CN], [ZA8273; H, F, Me, Et, (CH ₂ ) ₄ CN], [ZA8274; H, F, Me, Et, (CH ₂ ) ₅ CN], [ZA8275; H, F, Me, Et, CH ₂ CH = CH ₂ ], [ZA8276; H, F, Me, Et, CH ₂ C≡CH], [ZA8277; H, F, Me, Et, CH ₂ C≡CCH ₃ ] , [ZA8278; H, F, Me, Et, CH ₂ Ph], [ZA8279; H, F, Me, Et, CH ₂ (2-Py)], [ZA8280; H, F, Me, Et, CH ₂ (3-Py)], [ZA8281; H, F, Me, Et, CH ₂ (4-Py)], [ZA8282; H, F, Me, Et , (CH ₂ ) ₂ Ph], [ZA8283; H, F, Me, Et, (CH ₂ ) ₂ (2-Py)], [ZA8284; H, F, Me, Et, (CH ₂ ) ₂ (3 -Py)], [ZA8285; H, F, Me, Et, (CH ₂ ) ₂ (4-Py)], [ZA8286; H, F, Me, Et, Ph], [ZA8287; H, F, Me , Et, 2-Py], [ZA8288; H, F, Me, Et, 3-Py], [ZA8289; H, F, Me, Et, 4-Py].

Formula (V)

In which the combination of R ³¹ , R ³² , R ³³ , R ³⁴ and R ^{35 is} a combination described in any one of the substituent numbers ZA1 to ZA8289 (hereinafter represented by the formula (V)) In which the compounds having substituent numbers ZA1 to ZA8289 are represented as the present compounds RD1 to RD8289, and the present compounds RD1 to RD8289 are collectively referred to as the present compound RD). .

For example, the present compound RD2 means a compound having the substituent number ZA2 in the compound represented by the formula (V), and in the compound represented by the formula (V), R ³¹ , R ³² , R ³³ and R ³⁴ are It represents a compound represented by the following, which is a hydrogen atom and R ³⁵ is NHEt.

Formula (VI)

In which the combination of R ⁴¹ , R ⁴² , R ⁴³ , R ⁴⁴ , R ⁴⁵ and R ⁴⁶ is a combination described in any one of the substituent numbers RC1 to RC12096 shown below (Hereinafter, the compounds having the substituent numbers RC1 to RC12096 are represented as the present compounds RC1 to RC12096, and the present compounds RC1 to RC12096 are collectively represented as the present compound RC). it can.
The substituent numbers RC1 to RC12096 represent a combination of R ⁴¹ , R ⁴² , R ⁴³ , R ⁴⁴ , R ⁴⁵ and R ^{46 in} the compound represented by the formula (VI). [Substituent number: R ⁴¹ , R ⁴² , R ⁴³ , R ⁴⁴ , R ⁴⁵ , R ⁴⁶ ]
For example, the substituent number RC4 represents a combination in which R ⁴¹ , R ⁴² , R ⁴³ , R ⁴⁴ and R ⁴⁵ are hydrogen atoms and R ⁴⁶ is an isopropyl group.

For example, the present compound RC4 means a compound whose substituent number is RC4 in the compound represented by the formula (VI), and R ⁴¹ , R ⁴² , R ⁴³ , R in the compound represented by the formula (VI). ⁴⁴ and R ⁴⁵ represent a hydrogen atom and R ⁴⁶ represents an isopropyl group.

[Substituent number; R ⁴¹ , R ⁴² , R ⁴³ , R ⁴⁴ , R ⁴⁵ , R ⁴⁶ ]: [RC1; H, H, H, H, H, Me], [RC2; H, H, H, H , H, Et], [RC3; H, H, H, H, H, Pr], [RC4; H, H, H, H, H, i-Pr], [RC5; H, H, H, H , H, c-Pr], [RC6; H, H, H, H, H, Bu], [RC7; H, H, H, H, H, i-Bu], [RC8; H, H, H , H, H, t-Bu], [RC9; H, H, H, H, H, c-PrCH ₂ ], [RC10; H, H, H, H, H, Ph], [RC11; H, H, H, H, H, Bn], [RC12; H, H, H, H, H, CF ₃ ], [RC13; H, H, H, H, H, CF ₃ CH ₂ ], [RC14; H, H, H, H, H, CF ₃ CF ₂ ], [RC15; H, H, H, H, H, CF ₂ H], [RC16; H, H, H, H, H, CF ₂ HCF ₂ ], [RC17; H, H, H, Me, H, Me], [RC18; H, H, H, Me, H, Et], [RC19; H, H, H, Me, H, Pr] , [RC20; H, H, H, Me, H, i-Pr], [RC21; H, H, H, Me, H, c-Pr], [RC22; H, H, H, Me, H, Bu], [RC23; H, H, H, Me, H, i-Bu], [RC24; H, H, H, Me, H, t-Bu], [RC25; H, H, H, Me, H, c-PrCH ₂ ], [RC26; H, H, H, Me, H, Ph], [RC27; H, H, H, Me, H, Bn], [RC28; H, H, H, Me , H, CF ₃ ], [RC29; H, H, H, Me, H, CF ₃ CH ₂ ], [RC30; H, H, H, Me, H, CF ₃ CF ₂ ], [RC31; H, H, H, Me, H, CF ₂ H], [RC32; H, H, H, Me, H, CF ₂ HCF ₂ ], [RC33; H, H, Me, Me, H, Me], [RC34 ; H, H, Me, Me, H, Et], [RC35; H, H, Me, Me, H, Pr], [RC36; H, H, Me, Me, H, i-Pr], [RC37 ; H, H, Me, Me, H, c-Pr], [RC38; H, H, Me, Me, H, Bu], [RC39; H, H, Me, Me, H, i-Bu], [RC40; H, H, Me, Me, H, t-Bu], [RC41; H, H, Me, Me, H, cP rCH ₂ ], [RC42; H, H, Me, Me, H, Ph], [RC43; H, H, Me, Me, H, Bn], [RC44; H, H, Me, Me, H, CF ₃ ], [RC45; H, H, Me, Me, H, CF ₃ CH ₂ ], [RC46; H, H, Me, Me, H, CF ₃ CF ₂ ], [RC47; H, H, Me, Me, H, CF ₂ H], [RC48; H, H, Me, Me, H, CF ₂ HCF ₂ ], [RC49; H, H, Me, Et, H, Me], [RC50; H, H , Me, Et, H, Et], [RC51; H, H, Me, Et, H, Pr], [RC52; H, H, Me, Et, H, i-Pr], [RC53; H, H , Me, Et, H, c-Pr], [RC54; H, H, Me, Et, H, Bu], [RC55; H, H, Me, Et, H, i-Bu], [RC56; H , H, Me, Et, H, t-Bu], [RC57; H, H, Me, Et, H, c-PrCH ₂ ], [RC58; H, H, Me, Et, H, Ph], [ RC59; H, H, Me, Et, H, Bn], [RC60; H, H, Me, Et, H, CF ₃ ], [RC61; H, H, Me, Et, H, CF ₃ CH ₂ ] , [RC62; H, H, Me, Et, H, CF ₃ CF ₂ ], [RC63; H, H, Me, Et, H, CF ₂ H], [RC64; H, H, Me, Et, H , CF ₂ HCF ₂ ], [RC65; H, H, Me, F, H, Me], [RC66; H, H, Me, F, H, Et], [RC67; H, H, Me, F, H, Pr], [RC68; H, H, Me, F, H, i-Pr], [RC69; H, H, Me, F, H, c-Pr], [RC70; H, H, Me, F, H, Bu], [RC71; H, H, Me, F, H, i-Bu], [RC72; H, H, Me, F, H, t-Bu], [RC73; H, H, Me, F, H, c-PrCH ₂ ], [RC74; H, H, Me, F, H, Ph], [RC75; H, H, Me, F, H, Bn], [RC76; H, H , Me, F, H, CF ₃ ], [RC77; H, H, Me, F, H, CF ₃ CH ₂ ], [RC78; H, H, Me, F, H, CF ₃ CF ₂ ], [ RC79; H, H, Me, F, H, CF ₂ H], [RC80; H, H, Me, F, H, CF ₂ HCF ₂ ], [RC81; H, H, Me, Cl, H, Me ], [R C82; H, H, Me, Cl, H, Et], [RC83; H, H, Me, Cl, H, Pr], [RC84; H, H, Me, Cl, H, i-Pr], [ RC85; H, H, Me, Cl, H, c-Pr], [RC86; H, H, Me, Cl, H, Bu], [RC87; H, H, Me, Cl, H, i-Bu] , [RC88; H, H, Me, Cl, H, t-Bu], [RC89; H, H, Me, Cl, H, c-PrCH ₂ ], [RC90; H, H, Me, Cl, H , Ph], [RC91; H, H, Me, Cl, H, Bn], [RC92; H, H, Me, Cl, H, CF ₃ ], [RC93; H, H, Me, Cl, H, CF ₃ CH ₂ ], [RC94; H, H, Me, Cl, H, CF ₃ CF ₂ ], [RC95; H, H, Me, Cl, H, CF ₂ H], [RC96; H, H, Me, Cl, H, CF ₂ HCF ₂ ], [RC97; H, H, Et, H, H, Me], [RC98; H, H, Et, H, H, Et], [RC99; H, H , Et, H, H, Pr], [RC100; H, H, Et, H, H, i-Pr], [RC101; H, H, Et, H, H, c-Pr], [RC102; H , H, Et, H, H, Bu], [RC103; H, H, Et, H, H, i-Bu], [RC104; H, H, Et, H, H, t-Bu], [RC105 ; H, H, Et, H, H, c-PrCH ₂ ], [RC106; H, H, Et, H, H, Ph], [RC107; H, H, Et, H, H, Bn], [ RC108; H, H, Et, H, H, CF ₃ ], [RC109; H, H, Et, H, H, CF ₃ CH ₂ ], [RC110; H, H, Et, H, H, CF ₃ CF ₂ ], [RC111; H, H, Et, H, H, CF ₂ H], [RC112; H, H, Et, H, H, CF ₂ HCF ₂ ], [RC113; H, H, Et, F, H, Me], [RC114; H, H, Et, F, H, Et], [RC115; H, H, Et, F, H, Pr], [RC116; H, H, Et, F, H, i-Pr], [RC117; H, H, Et, F, H, c-Pr], [RC118; H, H, Et, F, H, Bu], [RC119; H, H, Et, F, H, i-Bu], [RC120; H, H, Et, F, H, t-Bu], [RC121; H, H, Et, F, H, c-PrCH ₂ ], [RC122; H , H, Et, F, H, Ph], [RC123; H, H, Et, F, H, Bn], [RC124; H, H, Et, F, H, CF ₃ ], [RC125; H, H, Et, F, H , CF ₃ CH ₂ ], [RC126; H, H, Et, F, H, CF ₃ CF ₂ ], [RC127; H, H, Et, F, H, CF ₂ H], [RC128; H, H , Et, F, H, CF ₂ HCF ₂ ], [RC129; H, H, Et, Cl, H, Me], [RC130; H, H, Et, Cl, H, Et], [RC131; H, H, Et, Cl, H, Pr], [RC132; H, H, Et, Cl, H, i-Pr], [RC133; H, H, Et, Cl, H, c-Pr], [RC134; H, H, Et, Cl, H, Bu], [RC135; H, H, Et, Cl, H, i-Bu], [RC136; H, H, Et, Cl, H, t-Bu], [ RC137; H, H, Et, Cl, H, c-PrCH ₂ ], [RC138; H, H, Et, Cl, H, Ph], [RC139; H, H, Et, Cl, H, Bn], [RC140; H, H, Et, Cl, H, CF ₃ ], [RC141; H, H, Et, Cl, H, CF ₃ CH ₂ ], [RC142; H, H, Et, Cl, H, CF ₃ CF ₂ ], [RC143; H, H, Et, Cl, H, CF ₂ H], [RC144; H, H, Et, Cl, H, CF ₂ HCF ₂ ], [RC145; H, H, F , H, H, Me], [RC146; H, H, F, H, H, Et], [RC147; H, H, F, H, H, Pr], [RC148; H, H, F, H , H, i-Pr], [RC149; H, H, F, H, H, c-Pr], [RC150; H, H, F, H, H, Bu], [RC151; H, H, F , H, H, i-Bu], [RC152; H, H, F, H, H, t-Bu], [RC153; H, H, F, H, H, c-PrCH ₂ ], [RC154; H, H, F, H, H, Ph], [RC155; H, H, F, H, H, Bn], [RC156; H, H, F, H, H, CF ₃ ], [RC157; H , H, F, H, H, CF ₃ CH ₂ ], [RC158; H, H, F, H, H, CF ₃ CF ₂ ], [RC159; H, H, F, H, H, CF ₂ H ], [RC160; H, H, F, H, H, CF ₂ HCF ₂ ], [RC161; H, H, F, F, H, Me], [RC162; H, H, F, F, H, Et], [RC163; H, H, F, F, H, Pr], [RC164; H, H, F, F, H, i-Pr], [RC165; H, H, F, F, H, c-Pr], [RC166; H, H, F, F, H, Bu], [RC167; H, H, F, F, H, i-Bu], [RC168; H, H, F, F, H, t-Bu], [RC169; H, H, F, F, H, c-PrCH ₂ ], [RC170; H, H, F, F, H, Ph], [RC171 ; H, H, F, F, H, Bn], [RC172; H, H, F, F, H, CF ₃ ], [RC173; H, H, F, F, H, CF ₃ CH ₂ ], [RC174; H, H, F, F, H, CF ₃ CF ₂ ], [RC175; H, H, F, F, H, CF ₂ H], [RC176; H, H, F, F, H, CF ₂ HCF ₂ ], [RC177; H, H, F, Cl, H, Me], [RC178; H, H, F, Cl, H, Et], [RC179; H, H, F, Cl, H , Pr], [RC180; H, H, F, Cl, H, i-Pr], [RC181; H, H, F, Cl, H, c-Pr], [RC182; H, H, F, Cl , H, Bu], [RC183; H, H, F, Cl, H, i-Bu], [RC184; H, H, F, Cl, H, t-Bu], [RC185; H, H, F , Cl, H, c-PrCH ₂ ], [RC186; H, H, F, Cl, H, Ph], [RC187; H, H, F, Cl, H, Bn], [RC188; H, H, F, Cl, H, CF ₃ ], [RC189; H, H, F, Cl, H, CF ₃ CH ₂ ], [RC190; H, H, F, Cl, H, CF ₃ CF ₂ ], [RC191 ; H, H, F, Cl, H, CF ₂ H], [RC192; H, H, F, Cl, H, CF ₂ HCF ₂ ], [RC193; H, H, Cl, H, H, Me] , [RC194; H, H, Cl, H, H, Et], [RC195; H, H, Cl, H, H, Pr], [RC196; H, H, Cl, H, H, i-Pr] , [RC197; H, H, Cl, H, H, c-Pr], [RC198; H, H, Cl, H, H, Bu], [RC199; H, H, Cl, H, H, i- Bu], [RC200; H, H, Cl, H, H, t-Bu],

[RC201; H, H, Cl, H, H, c-PrCH ₂ ], [RC202; H, H, Cl, H, H, Ph], [RC203; H, H, Cl, H, H, Bn] , [RC204; H, H, Cl, H, H, CF ₃ ], [RC205; H, H, Cl, H, H, CF ₃ CH ₂ ], [RC206; H, H, Cl, H, H, CF ₃ CF ₂ ], [RC207; H, H, Cl, H, H, CF ₂ H], [RC208; H, H, Cl, H, H, CF ₂ HCF ₂ ], [RC209; H, H, Cl, Cl, H, Me], [RC210; H, H, Cl, Cl, H, Et], [RC211; H, H, Cl, Cl, H, Pr], [RC212; H, H, Cl, Cl, H, i-Pr], [RC213; H, H, Cl, Cl, H, c-Pr], [RC214; H, H, Cl, Cl, H, Bu], [RC215; H, H, Cl, Cl, H, i-Bu], [RC216; H, H, Cl, Cl, H, t-Bu], [RC217; H, H, Cl, Cl, H, c-PrCH ₂ ], [RC218 ; H, H, Cl, Cl, H, Ph], [RC219; H, H, Cl, Cl, H, Bn], [RC220; H, H, Cl, Cl, H, CF ₃ ], [RC221; H, H, Cl, Cl, H, CF ₃ CH ₂ ], [RC222; H, H, Cl, Cl, H, CF ₃ CF ₂ ], [RC223; H, H, Cl, Cl, H, CF ₂ H], [RC224; H, H, Cl, Cl, H, CF ₂ HCF ₂ ], [RC225; H, H, H, H, Me, Me], [RC226; H, H, H, H, Me , Et], [RC227; H, H, H, H, Me, Pr], [RC228; H, H, H, H, Me, i-Pr], [RC229; H, H, H, H, Me , c-Pr], [RC230; H, H, H, H, Me, Bu], [RC231; H, H, H, H, Me, i-Bu], [RC232; H, H, H, H , Me, t-Bu], [RC233; H, H, H, H, Me, c-PrCH ₂ ], [RC234; H, H, H, H, Me, Ph], [RC235; H, H, H, H, Me, Bn], [RC236; H, H, H, H, Me, CF ₃ ], [RC237; H, H, H, H, Me, CF ₃ CH ₂ ], [RC238; H, H, H, H, Me, CF ₃ CF ₂ ], [RC239; H, H, H, H, Me, CF ₂ H], [R C240; H, H, H, H, Me, CF ₂ HCF ₂ ], [RC241; H, H, H, Me, Me, Me], [RC242; H, H, H, Me, Me, Et], [RC243; H, H, H, Me, Me, Pr], [RC244; H, H, H, Me, Me, i-Pr], [RC245; H, H, H, Me, Me, c-Pr ], [RC246; H, H, H, Me, Me, Bu], [RC247; H, H, H, Me, Me, i-Bu], [RC248; H, H, H, Me, Me, t -Bu], [RC249; H, H, H, Me, Me, c-PrCH ₂ ], [RC250; H, H, H, Me, Me, Ph], [RC251; H, H, H, Me, Me, Bn], [RC252; H, H, H, Me, Me, CF ₃ ], [RC253; H, H, H, Me, Me, CF ₃ CH ₂ ], [RC254; H, H, H, Me, Me, CF ₃ CF ₂ ], [RC255; H, H, H, Me, Me, CF ₂ H], [RC256; H, H, H, Me, Me, CF ₂ HCF ₂ ], [RC257; H, H, Me, Me, Me, Me], [RC258; H, H, Me, Me, Me, Et], [RC259; H, H, Me, Me, Me, Pr], [RC260; H, H, Me, Me, Me, i-Pr], [RC261; H, H, Me, Me, Me, c-Pr], [RC262; H, H, Me, Me, Me, Bu], [RC263; H, H, Me, Me, Me, i-Bu], [RC264; H, H, Me, Me, Me, t-Bu], [RC265; H, H, Me, Me, Me, c-PrCH ₂ ], [RC266; H, H, Me, Me, Me, Ph], [RC267; H, H, Me, Me, Me, Bn], [RC268; H, H, Me, Me, Me, CF ₃ ] , [RC269; H, H, Me, Me, Me, CF ₃ CH ₂ ], [RC270; H, H, Me, Me, Me, CF ₃ CF ₂ ], [RC271; H, H, Me, Me, Me, CF ₂ H], [RC272; H, H, Me, Me, Me, CF ₂ HCF ₂ ], [RC273; H, H, Me, Et, Me, Me], [RC274; H, H, Me , Et, Me, Et], [RC275; H, H, Me, Et, Me, Pr], [RC276; H, H, Me, Et, Me, i-Pr], [RC277; H, H, Me , Et, Me, c-Pr], [ RC278; H, H, Me, Et, Me, Bu], [RC279; H, H, Me, Et, Me, i-Bu], [RC280; H, H, Me, Et, Me, t-Bu] , [RC281; H, H, Me, Et, Me, c-PrCH ₂ ], [RC282; H, H, Me, Et, Me, Ph], [RC283; H, H, Me, Et, Me, Bn ], [RC284; H, H, Me, Et, Me, CF ₃ ], [RC285; H, H, Me, Et, Me, CF ₃ CH ₂ ], [RC286; H, H, Me, Et, Me , CF ₃ CF ₂ ], [RC287; H, H, Me, Et, Me, CF ₂ H], [RC288; H, H, Me, Et, Me, CF ₂ HCF ₂ ], [RC289; H, H , Me, F, Me, Me], [RC290; H, H, Me, F, Me, Et], [RC291; H, H, Me, F, Me, Pr], [RC292; H, H, Me , F, Me, i-Pr], [RC293; H, H, Me, F, Me, c-Pr], [RC294; H, H, Me, F, Me, Bu], [RC295; H, H , Me, F, Me, i-Bu], [RC296; H, H, Me, F, Me, t-Bu], [RC297; H, H, Me, F, Me, c-PrCH ₂ ], [ RC298; H, H, Me, F, Me, Ph], [RC299; H, H, Me, F, Me, Bn], [RC300; H, H, Me, F, Me, CF ₃ ], [RC301 ; H, H, Me, F, Me, CF ₃ CH ₂ ], [RC302; H, H, Me, F, Me, CF ₃ CF ₂ ], [RC303; H, H, Me, F, Me, CF ₂ H], [RC304; H, H, Me, F, Me, CF ₂ HCF ₂ ], [RC305; H, H, Me, Cl, Me, Me], [RC306; H, H, Me, Cl, Me, Et], [RC307; H, H, Me, Cl, Me, Pr], [RC308; H, H, Me, Cl, Me, i-Pr], [RC309; H, H, Me, Cl, Me, c-Pr], [RC310; H, H, Me, Cl, Me, Bu], [RC311; H, H, Me, Cl, Me, i-Bu], [RC312; H, H, Me, Cl, Me, t-Bu], [RC313; H, H, Me, Cl, Me, c-PrCH ₂ ], [RC314; H, H, Me, Cl, Me, Ph], [RC315; H, H , Me, Cl, Me, Bn], [RC316; H, H, Me, Cl, Me, CF ₃ ], [RC317; H, H, Me, Cl, Me, CF ₃ CH ₂ ], [RC318; H, H, Me, Cl, Me, CF ₃ CF ₂ ], [RC319; H, H, Me, Cl, Me, CF ₂ H], [RC320; H, H, Me, Cl, Me, CF ₂ HCF ₂ ], [RC321; H, H, Et , H, Me, Me], [RC322; H, H, Et, H, Me, Et], [RC323; H, H, Et, H, Me, Pr], [RC324; H, H, Et, H , Me, i-Pr], [RC325; H, H, Et, H, Me, c-Pr], [RC326; H, H, Et, H, Me, Bu], [RC327; H, H, Et , H, Me, i-Bu], [RC328; H, H, Et, H, Me, t-Bu], [RC329; H, H, Et, H, Me, c-PrCH ₂ ], [RC330; H, H, Et, H, Me, Ph], [RC331; H, H, Et, H, Me, Bn], [RC332; H, H, Et, H, Me, CF ₃ ], [RC333; H , H, Et, H, Me, CF ₃ CH ₂ ], [RC334; H, H, Et, H, Me, CF ₃ CF ₂ ], [RC335; H, H, Et, H, Me, CF ₂ H ], [RC336; H, H, Et, H, Me, CF ₂ HCF ₂ ], [RC337; H, H, Et, F, Me, Me], [RC338; H, H, Et, F, Me, Et], [RC339; H, H, Et, F, Me, Pr], [RC340; H, H, Et, F, Me, i-Pr], [RC341; H, H, Et, F, Me, c-Pr], [RC342; H, H, Et, F, Me, Bu], [RC343; H, H, Et, F, Me, i-Bu], [RC344; H, H, Et, F, Me, t-Bu], [RC345; H, H, Et, F, Me, c-PrCH ₂ ], [RC346; H, H, Et, F, Me, Ph], [RC347; H, H, Et , F, Me, Bn], [RC348; H, H, Et, F, Me, CF ₃ ], [RC349; H, H, Et, F, Me, CF ₃ CH ₂ ], [RC350; H, H , Et, F, Me, CF ₃ CF ₂ ], [RC351; H, H, Et, F, Me, CF ₂ H], [RC352; H, H, Et, F, Me, CF ₂ HCF ₂ ], [RC353; H, H, Et, Cl, M e, Me], [RC354; H, H, Et, Cl, Me, Et], [RC355; H, H, Et, Cl, Me, Pr], [RC356; H, H, Et, Cl, Me, i-Pr], [RC357; H, H, Et, Cl, Me, c-Pr], [RC358; H, H, Et, Cl, Me, Bu], [RC359; H, H, Et, Cl, Me, i-Bu], [RC360; H, H, Et, Cl, Me, t-Bu], [RC361; H, H, Et, Cl, Me, c-PrCH ₂ ], [RC362; H, H , Et, Cl, Me, Ph], [RC363; H, H, Et, Cl, Me, Bn], [RC364; H, H, Et, Cl, Me, CF ₃ ], [RC365; H, H, Et, Cl, Me, CF ₃ CH ₂ ], [RC366; H, H, Et, Cl, Me, CF ₃ CF ₂ ], [RC367; H, H, Et, Cl, Me, CF ₂ H], [ RC368; H, H, Et, Cl, Me, CF ₂ HCF ₂ ], [RC369; H, H, F, H, Me, Me], [RC370; H, H, F, H, Me, Et], [RC371; H, H, F, H, Me, Pr], [RC372; H, H, F, H, Me, i-Pr], [RC373; H, H, F, H, Me, c-Pr ], [RC374; H, H, F, H, Me, Bu], [RC375; H, H, F, H, Me, i-Bu], [RC376; H, H, F, H, Me, t -Bu], [RC377; H, H, F, H, Me, c-PrCH ₂ ], [RC378; H, H, F, H, Me, Ph], [RC379; H, H, F, H, Me, Bn], [RC380; H, H, F, H, Me, CF ₃ ], [RC381; H, H, F, H, Me, CF ₃ CH ₂ ], [RC382; H, H, F, H, Me, CF ₃ CF ₂ ], [RC383; H, H, F, H, Me, CF ₂ H], [RC384; H, H, F, H, Me, CF ₂ HCF ₂ ], [RC385; H, H, F, F, Me, Me], [RC386; H, H, F, F, Me, Et], [RC387; H, H, F, F, Me, Pr], [RC388; H, H, F, F, Me, i-Pr], [RC389; H, H, F, F, Me, c-Pr], [RC390; H, H, F, F, Me, Bu], [RC391; H, H, F, F, Me, i-Bu], [RC392; H, H, F, F, Me, t-Bu], [RC3 93; H, H, F, F, Me, c-PrCH ₂ ], [RC394; H, H, F, F, Me, Ph], [RC395; H, H, F, F, Me, Bn], [RC396; H, H, F, F, Me, CF ₃ ], [RC397; H, H, F, F, Me, CF ₃ CH ₂ ], [RC398; H, H, F, F, Me, CF ₃ CF ₂ ], [RC399; H, H, F, F, Me, CF ₂ H], [RC400; H, H, F, F, Me, CF ₂ HCF ₂ ],

[RC401; H, H, F, Cl, Me, Me], [RC402; H, H, F, Cl, Me, Et], [RC403; H, H, F, Cl, Me, Pr], [RC404 ; H, H, F, Cl, Me, i-Pr], [RC405; H, H, F, Cl, Me, c-Pr], [RC406; H, H, F, Cl, Me, Bu], [RC407; H, H, F, Cl, Me, i-Bu], [RC408; H, H, F, Cl, Me, t-Bu], [RC409; H, H, F, Cl, Me, c -PrCH ₂ ], [RC410; H, H, F, Cl, Me, Ph], [RC411; H, H, F, Cl, Me, Bn], [RC412; H, H, F, Cl, Me, CF ₃ ], [RC413; H, H, F, Cl, Me, CF ₃ CH ₂ ], [RC414; H, H, F, Cl, Me, CF ₃ CF ₂ ], [RC415; H, H, F , Cl, Me, CF ₂ H], [RC416; H, H, F, Cl, Me, CF ₂ HCF ₂ ], [RC417; H, H, Cl, H, Me, Me], [RC418; H, H, Cl, H, Me, Et], [RC419; H, H, Cl, H, Me, Pr], [RC420; H, H, Cl, H, Me, i-Pr], [RC421; H, H, Cl, H, Me, c-Pr], [RC422; H, H, Cl, H, Me, Bu], [RC423; H, H, Cl, H, Me, i-Bu], [RC424; H, H, Cl, H, Me, t-Bu], [RC425; H, H, Cl, H, Me, c-PrCH ₂ ], [RC426; H, H, Cl, H, Me, Ph], [RC427; H, H, Cl, H, Me, Bn], [RC428; H, H, Cl, H, Me, CF ₃ ], [RC429; H, H, Cl, H, Me, CF ₃ CH ₂ ], [RC430; H, H, Cl, H, Me, CF ₃ CF ₂ ], [RC431; H, H, Cl, H, Me, CF ₂ H], [RC432; H, H, Cl, H, Me, CF ₂ HCF ₂ ], [RC433; H, H, Cl, Cl, Me, Me], [RC434; H, H, Cl, Cl, Me, Et], [RC435; H, H, Cl, Cl , Me, Pr], [RC436; H, H, Cl, Cl, Me, i-Pr], [RC437; H, H, Cl, Cl, Me, c-Pr], [RC438; H, H, Cl , Cl, Me, Bu], [RC439; H, H, Cl, Cl, Me, i- Bu], [RC440; H, H, Cl, Cl, Me, t-Bu], [RC441; H, H, Cl, Cl, Me, c-PrCH ₂ ], [RC442; H, H, Cl, Cl , Me, Ph], [RC443; H, H, Cl, Cl, Me, Bn], [RC444; H, H, Cl, Cl, Me, CF ₃ ], [RC445; H, H, Cl, Cl, Me, CF ₃ CH ₂ ], [RC446; H, H, Cl, Cl, Me, CF ₃ CF ₂ ], [RC447; H, H, Cl, Cl, Me, CF ₂ H], [RC448; H, H, Cl, Cl, Me, CF ₂ HCF ₂ ], [RC449; H, H, H, H, Et, Me], [RC450; H, H, H, H, Et, Et], [RC451; H , H, H, H, Et, Pr], [RC452; H, H, H, H, Et, i-Pr], [RC453; H, H, H, H, Et, c-Pr], [RC454 ; H, H, H, H, Et, Bu], [RC455; H, H, H, H, Et, i-Bu], [RC456; H, H, H, H, Et, t-Bu], [RC457; H, H, H, H, Et, c-PrCH ₂ ], [RC458; H, H, H, H, Et, Ph], [RC459; H, H, H, H, Et, Bn] , [RC460; H, H, H, H, Et, CF ₃ ], [RC461; H, H, H, H, Et, CF ₃ CH ₂ ], [RC462; H, H, H, H, Et, CF ₃ CF ₂ ], [RC463; H, H, H, H, Et, CF ₂ H], [RC464; H, H, H, H, Et, CF ₂ HCF ₂ ], [RC465; H, H, H, Me, Et, Me], [RC466; H, H, H, Me, Et, Et], [RC467; H, H, H, Me, Et, Pr], [RC468; H, H, H, Me, Et, i-Pr], [RC469; H, H, H, Me, Et, c-Pr], [RC470; H, H, H, Me, Et, Bu], [RC471; H, H, H, Me, Et, i-Bu], [RC472; H, H, H, Me, Et, t-Bu], [RC473; H, H, H, Me, Et, c-PrCH ₂ ], [RC474 ; H, H, H, Me, Et, Ph], [RC475; H, H, H, Me, Et, Bn], [RC476; H, H, H, Me, Et, CF ₃ ], [RC477; H, H, H, Me, Et, CF ₃ CH ₂ ], [RC478; H, H, H, Me , Et, CF ₃ CF ₂ ], [RC479; H, H, H, Me, Et, CF ₂ H], [RC480; H, H, H, Me, Et, CF ₂ HCF ₂ ], [RC481; H , H, Me, Me, Et, Me], [RC482; H, H, Me, Me, Et, Et], [RC483; H, H, Me, Me, Et, Pr], [RC484; H, H , Me, Me, Et, i-Pr], [RC485; H, H, Me, Me, Et, c-Pr], [RC486; H, H, Me, Me, Et, Bu], [RC487; H , H, Me, Me, Et, i-Bu], [RC488; H, H, Me, Me, Et, t-Bu], [RC489; H, H, Me, Me, Et, c-PrCH ₂ ] , [RC490; H, H, Me, Me, Et, Ph], [RC491; H, H, Me, Me, Et, Bn], [RC492; H, H, Me, Me, Et, CF ₃ ], [RC493; H, H, Me, Me, Et, CF ₃ CH ₂ ], [RC494; H, H, Me, Me, Et, CF ₃ CF ₂ ], [RC495; H, H, Me, Me, Et , CF ₂ H], [RC496; H, H, Me, Me, Et, CF ₂ HCF ₂ ], [RC497; H, H, Me, Et, Et, Me], [RC498; H, H, Me, Et, Et, Et], [RC499; H, H, Me, Et, Et, Pr], [RC500; H, H, Me, Et, Et, i-Pr], [RC501; H, H, Me, Et, Et, c-Pr], [RC502; H, H, Me, Et, Et, Bu], [RC503; H, H, Me, Et, Et, i-Bu], [RC504; H, H, Me, Et, Et, t-Bu], [RC505; H, H, Me, Et, Et, c-PrCH ₂ ], [RC506; H, H, Me, Et, Et, Ph], [RC507; H , H, Me, Et, Et, Bn], [RC508; H, H, Me, Et, Et, CF ₃ ], [RC509; H, H, Me, Et, Et, CF ₃ CH ₂ ], [RC510 ; H, H, Me, Et, Et, CF ₃ CF ₂ ], [RC511; H, H, Me, Et, Et, CF ₂ H], [RC512; H, H, Me, Et, Et, CF ₂ HCF ₂ ], [RC513; H, H, Me, F, Et, Me], [RC514; H, H, Me, F, Et, Et], [RC515; H, H, Me, F, E t, Pr], [RC516; H, H, Me, F, Et, i-Pr], [RC517; H, H, Me, F, Et, c-Pr], [RC518; H, H, Me, F, Et, Bu], [RC519; H, H, Me, F, Et, i-Bu], [RC520; H, H, Me, F, Et, t-Bu], [RC521; H, H, Me, F, Et, c-PrCH ₂ ], [RC522; H, H, Me, F, Et, Ph], [RC523; H, H, Me, F, Et, Bn], [RC524; H, H , Me, F, Et, CF ₃ ], [RC525; H, H, Me, F, Et, CF ₃ CH ₂ ], [RC526; H, H, Me, F, Et, CF ₃ CF ₂ ], [ RC527; H, H, Me, F, Et, CF ₂ H], [RC528; H, H, Me, F, Et, CF ₂ HCF ₂ ], [RC529; H, H, Me, Cl, Et, Me ], [RC530; H, H, Me, Cl, Et, Et], [RC531; H, H, Me, Cl, Et, Pr], [RC532; H, H, Me, Cl, Et, i-Pr ], [RC533; H, H, Me, Cl, Et, c-Pr], [RC534; H, H, Me, Cl, Et, Bu], [RC535; H, H, Me, Cl, Et, i -Bu], [RC536; H, H, Me, Cl, Et, t-Bu], [RC537; H, H, Me, Cl, Et, c-PrCH ₂ ], [RC538; H, H, Me, Cl, Et, Ph], [RC539; H, H, Me, Cl, Et, Bn], [RC540; H, H, Me, Cl, Et, CF ₃ ], [RC541; H, H, Me, Cl , Et, CF ₃ CH ₂ ], [RC542; H, H, Me, Cl, Et, CF ₃ CF ₂ ], [RC543; H, H, Me, Cl, Et, CF ₂ H], [RC544; H , H, Me, Cl, Et, CF ₂ HCF ₂ ], [RC545; H, H, Et, H, Et, Me], [RC546; H, H, Et, H, Et, Et], [RC547; H, H, Et, H, Et, Pr], [RC548; H, H, Et, H, Et, i-Pr], [RC549; H, H, Et, H, Et, c-Pr], [ RC550; H, H, Et, H, Et, Bu], [RC551; H, H, Et, H, Et, i-Bu], [RC552; H, H, Et, H, Et, t-Bu] , [RC553; H, H, Et, H, Et, c-PrCH ₂ ], [RC554; H, H, Et, H, Et, Ph], [RC555; H, H, Et, H, Et, Bn], [RC556; H, H, Et, H, Et, CF ₃ ], [RC557; H, H, Et, H, Et, CF ₃ CH ₂ ], [RC558; H, H, Et, H, Et, CF ₃ CF ₂ ], [RC559; H, H, Et, H , Et, CF ₂ H], [RC560; H, H, Et, H, Et, CF ₂ HCF ₂ ], [RC561; H, H, Et, F, Et, Me], [RC562; H, H, Et, F, Et, Et], [RC563; H, H, Et, F, Et, Pr], [RC564; H, H, Et, F, Et, i-Pr], [RC565; H, H, Et, F, Et, c-Pr], [RC566; H, H, Et, F, Et, Bu], [RC567; H, H, Et, F, Et, i-Bu], [RC568; H, H, Et, F, Et, t-Bu], [RC569; H, H, Et, F, Et, c-PrCH ₂ ], [RC570; H, H, Et, F, Et, Ph], [RC571 ; H, H, Et, F, Et, Bn], [RC572; H, H, Et, F, Et, CF ₃ ], [RC573; H, H, Et, F, Et, CF ₃ CH ₂ ], [RC574; H, H, Et, F, Et, CF ₃ CF ₂ ], [RC575; H, H, Et, F, Et, CF ₂ H], [RC576; H, H, Et, F, Et, CF ₂ HCF ₂ ], [RC577; H, H, Et, Cl, Et, Me], [RC578; H, H, Et, Cl, Et, Et], [RC579; H, H, Et, Cl, Et , Pr], [RC580; H, H, Et, Cl, Et, i-Pr], [RC581; H, H, Et, Cl, Et, c-Pr], [RC582; H, H, Et, Cl , Et, Bu], [RC583; H, H, Et, Cl, Et, i-Bu], [RC584; H, H, Et, Cl, Et, t-Bu], [RC585; H, H, Et , Cl, Et, c-PrCH ₂ ], [RC586; H, H, Et, Cl, Et, Ph], [RC587; H, H, Et, Cl, Et, Bn], [RC588; H, H, Et, Cl, Et, CF ₃ ], [RC589; H, H, Et, Cl, Et, CF ₃ CH ₂ ], [RC590; H, H, Et, Cl, Et, CF ₃ CF ₂ ], [RC591 ; H, H, Et, Cl, Et, CF ₂ H], [RC592; H, H, Et, Cl, Et, CF ₂ HCF ₂ ], [RC593; H, H, F, H, Et, Me], [RC594; H, H, F , H, Et, Et], [RC595; H, H, F, H, Et, Pr], [RC596; H, H, F, H, Et, i-Pr], [RC597; H, H, F , H, Et, c-Pr], [RC598; H, H, F, H, Et, Bu], [RC599; H, H, F, H, Et, i-Bu], [RC600; H, H , F, H, Et, t-Bu],

[RC601; H, H, F, H, Et, c-PrCH ₂ ], [RC602; H, H, F, H, Et, Ph], [RC603; H, H, F, H, Et, Bn] , [RC604; H, H, F, H, Et, CF ₃ ], [RC605; H, H, F, H, Et, CF ₃ CH ₂ ], [RC606; H, H, F, H, Et, CF ₃ CF ₂ ], [RC607; H, H, F, H, Et, CF ₂ H], [RC608; H, H, F, H, Et, CF ₂ HCF ₂ ], [RC609; H, H, F, F, Et, Me], [RC610; H, H, F, F, Et, Et], [RC611; H, H, F, F, Et, Pr], [RC612; H, H, F, F, Et, i-Pr], [RC613; H, H, F, F, Et, c-Pr], [RC614; H, H, F, F, Et, Bu], [RC615; H, H, F, F, Et, i-Bu], [RC616; H, H, F, F, Et, t-Bu], [RC617; H, H, F, F, Et, c-PrCH ₂ ], [RC618 ; H, H, F, F, Et, Ph], [RC619; H, H, F, F, Et, Bn], [RC620; H, H, F, F, Et, CF ₃ ], [RC621; H, H, F, F, Et, CF ₃ CH ₂ ], [RC622; H, H, F, F, Et, CF ₃ CF ₂ ], [RC623; H, H, F, F, Et, CF ₂ H], [RC624; H, H, F, F, Et, CF ₂ HCF ₂ ], [RC625; H, H, F, Cl, Et, Me], [RC626; H, H, F, Cl, Et , Et], [RC627; H, H, F, Cl, Et, Pr], [RC628; H, H, F, Cl, Et, i-Pr], [RC629; H, H, F, Cl, Et , c-Pr], [RC630; H, H, F, Cl, Et, Bu], [RC631; H, H, F, Cl, Et, i-Bu], [RC632; H, H, F, Cl , Et, t-Bu], [RC633; H, H, F, Cl, Et, c-PrCH ₂ ], [RC634; H, H, F, Cl, Et, Ph], [RC635; H, H, F, Cl, Et, Bn], [RC636; H, H, F, Cl, Et, CF ₃ ], [RC637; H, H, F, Cl, Et, CF ₃ CH ₂ ], [RC638; H, H, F, Cl, Et, CF ₃ CF ₂ ], [RC639; H, H, F, Cl, Et, CF ₂ H], [RC 640; H, H, F, Cl, Et, CF ₂ HCF ₂ ], [RC641; H, H, Cl, H, Et, Me], [RC642; H, H, Cl, H, Et, Et], [RC643; H, H, Cl, H, Et, Pr], [RC644; H, H, Cl, H, Et, i-Pr], [RC645; H, H, Cl, H, Et, c-Pr ], [RC646; H, H, Cl, H, Et, Bu], [RC647; H, H, Cl, H, Et, i-Bu], [RC648; H, H, Cl, H, Et, t -Bu], [RC649; H, H, Cl, H, Et, c-PrCH ₂ ], [RC650; H, H, Cl, H, Et, Ph], [RC651; H, H, Cl, H, Et, Bn], [RC652; H, H, Cl, H, Et, CF ₃ ], [RC653; H, H, Cl, H, Et, CF ₃ CH ₂ ], [RC654; H, H, Cl, H, Et, CF ₃ CF ₂ ], [RC655; H, H, Cl, H, Et, CF ₂ H], [RC656; H, H, Cl, H, Et, CF ₂ HCF ₂ ], [RC657; H, H, Cl, Cl, Et, Me], [RC658; H, H, Cl, Cl, Et, Et], [RC659; H, H, Cl, Cl, Et, Pr], [RC660; H, H, Cl, Cl, Et, i-Pr], [RC661; H, H, Cl, Cl, Et, c-Pr], [RC662; H, H, Cl, Cl, Et, Bu], [RC663; H, H, Cl, Cl, Et, i-Bu], [RC664; H, H, Cl, Cl, Et, t-Bu], [RC665; H, H, Cl, Cl, Et, c-PrCH ₂ ], [RC666; H, H, Cl, Cl, Et, Ph], [RC667; H, H, Cl, Cl, Et, Bn], [RC668; H, H, Cl, Cl, Et, CF ₃ ] , [RC669; H, H, Cl, Cl, Et, CF ₃ CH ₂ ], [RC670; H, H, Cl, Cl, Et, CF ₃ CF ₂ ], [RC671; H, H, Cl, Cl, Et, CF ₂ H], [RC672; H, H, Cl, Cl, Et, CF ₂ HCF ₂ ], [RC673; H, H, H, H, Pr, Me], [RC674; H, H, H , H, Pr, Et], [RC675; H, H, H, H, Pr, Pr], [RC676; H, H, H, H, Pr, i-Pr], [RC677; H, H, H , H, Pr, c-Pr], [RC678; H, H, H, H, Pr, Bu], [RC679; H, H, H, H, Pr, i-Bu], [RC680; H, H, H, H, Pr, t-Bu], [RC681; H, H, H, H, Pr, c-PrCH ₂ ], [RC682; H, H, H, H, Pr, Ph], [RC683; H, H, H, H, Pr, Bn], [RC684; H , H, H, H, Pr, CF ₃ ], [RC685; H, H, H, H, Pr, CF ₃ CH ₂ ], [RC686; H, H, H, H, Pr, CF ₃ CF ₂ ] , [RC687; H, H, H, H, Pr, CF ₂ H], [RC688; H, H, H, H, Pr, CF ₂ HCF ₂ ], [RC689; H, H, H, Me, Pr , Me], [RC690; H, H, H, Me, Pr, Et], [RC691; H, H, H, Me, Pr, Pr], [RC692; H, H, H, Me, Pr, i -Pr], [RC693; H, H, H, Me, Pr, c-Pr], [RC694; H, H, H, Me, Pr, Bu], [RC695; H, H, H, Me, Pr , i-Bu], [RC696; H, H, H, Me, Pr, t-Bu], [RC697; H, H, H, Me, Pr, c-PrCH ₂ ], [RC698; H, H, H, Me, Pr, Ph], [RC699; H, H, H, Me, Pr, Bn], [RC700; H, H, H, Me, Pr, CF ₃ ], [RC701; H, H, H , Me, Pr, CF ₃ CH ₂ ], [RC702; H, H, H, Me, Pr, CF ₃ CF ₂ ], [RC703; H, H, H, Me, Pr, CF ₂ H], [RC704 ; H, H, H, Me, Pr, CF ₂ HCF ₂ ], [RC705; H, H, Me, Me, Pr, Me], [RC706; H, H, Me, Me, Pr, Et], [ RC707; H, H, Me, Me, Pr, Pr], [RC708; H, H, Me, Me, Pr, i-Pr], [RC709; H, H, Me, Me, Pr, c-Pr] , [RC710; H, H, Me, Me, Pr, Bu], [RC711; H, H, Me, Me, Pr, i-Bu], [RC712; H, H, Me, Me, Pr, t- Bu], [RC713; H, H, Me, Me, Pr, c-PrCH ₂ ], [RC714; H, H, Me, Me, Pr, Ph], [RC715; H, H, Me, Me, Pr , Bn], [RC716; H, H, Me, Me, Pr, CF ₃ ], [RC71 7; H, H, Me, Me, Pr, CF ₃ CH ₂ ], [RC718; H, H, Me, Me, Pr, CF ₃ CF ₂ ], [RC719; H, H, Me, Me, Pr, CF ₂ H], [RC720; H, H, Me, Me, Pr, CF ₂ HCF ₂ ], [RC721; H, H, Me, Et, Pr, Me], [RC722; H, H, Me, Et , Pr, Et], [RC723; H, H, Me, Et, Pr, Pr], [RC724; H, H, Me, Et, Pr, i-Pr], [RC725; H, H, Me, Et , Pr, c-Pr], [RC726; H, H, Me, Et, Pr, Bu], [RC727; H, H, Me, Et, Pr, i-Bu], [RC728; H, H, Me , Et, Pr, t-Bu], [RC729; H, H, Me, Et, Pr, c-PrCH ₂ ], [RC730; H, H, Me, Et, Pr, Ph], [RC731; H, H, Me, Et, Pr, Bn], [RC732; H, H, Me, Et, Pr, CF ₃ ], [RC733; H, H, Me, Et, Pr, CF ₃ CH ₂ ], [RC734; H, H, Me, Et, Pr, CF ₃ CF ₂ ], [RC735; H, H, Me, Et, Pr, CF ₂ H], [RC736; H, H, Me, Et, Pr, CF ₂ HCF ₂ ], [RC737; H, H, Me, F, Pr, Me], [RC738; H, H, Me, F, Pr, Et], [RC739; H, H, Me, F, Pr, Pr] , [RC740; H, H, Me, F, Pr, i-Pr], [RC741; H, H, Me, F, Pr, c-Pr], [RC742; H, H, Me, F, Pr, Bu], [RC743; H, H, Me, F, Pr, i-Bu], [RC744; H, H, Me, F, Pr, t-Bu], [RC745; H, H, Me, F, Pr, c-PrCH ₂ ], [RC746; H, H, Me, F, Pr, Ph], [RC747; H, H, Me, F, Pr, Bn], [RC748; H, H, Me, F , Pr, CF ₃ ], [RC749; H, H, Me, F, Pr, CF ₃ CH ₂ ], [RC750; H, H, Me, F, Pr, CF ₃ CF ₂ ], [RC751; H, H, Me, F, Pr, CF ₂ H], [RC752; H, H, Me, F, Pr, CF ₂ HCF ₂ ], [RC753; H, H, Me, Cl, Pr, Me], [RC754 ; H, H , Me, Cl, Pr, Et], [RC755; H, H, Me, Cl, Pr, Pr], [RC756; H, H, Me, Cl, Pr, i-Pr], [RC757; H, H , Me, Cl, Pr, c-Pr], [RC758; H, H, Me, Cl, Pr, Bu], [RC759; H, H, Me, Cl, Pr, i-Bu], [RC760; H , H, Me, Cl, Pr, t-Bu], [RC761; H, H, Me, Cl, Pr, c-PrCH ₂ ], [RC762; H, H, Me, Cl, Pr, Ph], [ RC763; H, H, Me, Cl, Pr, Bn], [RC764; H, H, Me, Cl, Pr, CF ₃ ], [RC765; H, H, Me, Cl, Pr, CF ₃ CH ₂ ] , [RC766; H, H, Me, Cl, Pr, CF ₃ CF ₂ ], [RC767; H, H, Me, Cl, Pr, CF ₂ H], [RC768; H, H, Me, Cl, Pr , CF ₂ HCF ₂ ], [RC769; H, H, Et, H, Pr, Me], [RC770; H, H, Et, H, Pr, Et], [RC771; H, H, Et, H, Pr, Pr], [RC772; H, H, Et, H, Pr, i-Pr], [RC773; H, H, Et, H, Pr, c-Pr], [RC774; H, H, Et, H, Pr, Bu], [RC775; H, H, Et, H, Pr, i-Bu], [RC776; H, H, Et, H, Pr, t-Bu], [RC777; H, H, Et, H, Pr, c-PrCH ₂ ], [RC778; H, H, Et, H, Pr, Ph], [RC779; H, H, Et, H, Pr, Bn], [RC780; H, H , Et, H, Pr, CF ₃ ], [RC781; H, H, Et, H, Pr, CF ₃ CH ₂ ], [RC782; H, H, Et, H, Pr, CF ₃ CF ₂ ], [ RC783; H, H, Et, H, Pr, CF ₂ H], [RC784; H, H, Et, H, Pr, CF ₂ HCF ₂ ], [RC785; H, H, Et, F, Pr, Me ], [RC786; H, H, Et, F, Pr, Et], [RC787; H, H, Et, F, Pr, Pr], [RC788; H, H, Et, F, Pr, i-Pr ], [RC789; H, H, Et, F, Pr, c-Pr], [RC790; H, H, Et, F, Pr, Bu], [RC791; H, H, Et, F, Pr, i -Bu], [RC792; H, H, Et, F, Pr, t- Bu], [RC793; H, H, Et, F, Pr, c-PrCH ₂ ], [RC794; H, H, Et, F, Pr, Ph], [RC795; H, H, Et, F, Pr , Bn], [RC796; H, H, Et, F, Pr, CF ₃ ], [RC797; H, H, Et, F, Pr, CF ₃ CH ₂ ], [RC798; H, H, Et, F , Pr, CF ₃ CF ₂ ], [RC799; H, H, Et, F, Pr, CF ₂ H], [RC800; H, H, Et, F, Pr, CF ₂ HCF ₂ ],

[RC801; H, H, Et, Cl, Pr, Me], [RC802; H, H, Et, Cl, Pr, Et], [RC803; H, H, Et, Cl, Pr, Pr], [RC804 ; H, H, Et, Cl, Pr, i-Pr], [RC805; H, H, Et, Cl, Pr, c-Pr], [RC806; H, H, Et, Cl, Pr, Bu], [RC807; H, H, Et, Cl, Pr, i-Bu], [RC808; H, H, Et, Cl, Pr, t-Bu], [RC809; H, H, Et, Cl, Pr, c -PrCH ₂ ], [RC810; H, H, Et, Cl, Pr, Ph], [RC811; H, H, Et, Cl, Pr, Bn], [RC812; H, H, Et, Cl, Pr, CF ₃ ], [RC813; H, H, Et, Cl, Pr, CF ₃ CH ₂ ], [RC814; H, H, Et, Cl, Pr, CF ₃ CF ₂ ], [RC815; H, H, Et , Cl, Pr, CF ₂ H], [RC816; H, H, Et, Cl, Pr, CF ₂ HCF ₂ ], [RC817; H, H, F, H, Pr, Me], [RC818; H, H, F, H, Pr, Et], [RC819; H, H, F, H, Pr, Pr], [RC820; H, H, F, H, Pr, i-Pr], [RC821; H, H, F, H, Pr, c-Pr], [RC822; H, H, F, H, Pr, Bu], [RC823; H, H, F, H, Pr, i-Bu], [RC824; H, H, F, H, Pr, t-Bu], [RC825; H, H, F, H, Pr, c-PrCH ₂ ], [RC826; H, H, F, H, Pr, Ph], [RC827; H, H, F, H, Pr, Bn], [RC828; H, H, F, H, Pr, CF ₃ ], [RC829; H, H, F, H, Pr, CF ₃ CH ₂ ], [RC830; H, H, F, H, Pr, CF ₃ CF ₂ ], [RC831; H, H, F, H, Pr, CF ₂ H], [RC832; H, H, F, H, Pr, CF ₂ HCF ₂ ], [RC833; H, H, F, F, Pr, Me], [RC834; H, H, F, F, Pr, Et], [RC835; H, H, F, F , Pr, Pr], [RC836; H, H, F, F, Pr, i-Pr], [RC837; H, H, F, F, Pr, c-Pr], [RC838; H, H, F , F, Pr, Bu], [RC839; H, H, F, F, Pr, i-Bu], [RC840; H, H , F, F, Pr, t-Bu], [RC841; H, H, F, F, Pr, c-PrCH ₂ ], [RC842; H, H, F, F, Pr, Ph], [RC843; H, H, F, F, Pr, Bn], [RC844; H, H, F, F, Pr, CF ₃ ], [RC845; H, H, F, F, Pr, CF ₃ CH ₂ ], [ RC846; H, H, F, F, Pr, CF ₃ CF ₂ ], [RC847; H, H, F, F, Pr, CF ₂ H], [RC848; H, H, F, F, Pr, CF ₂ HCF ₂ ], [RC849; H, H, F, Cl, Pr, Me], [RC850; H, H, F, Cl, Pr, Et], [RC851; H, H, F, Cl, Pr, Pr], [RC852; H, H, F, Cl, Pr, i-Pr], [RC853; H, H, F, Cl, Pr, c-Pr], [RC854; H, H, F, Cl, Pr, Bu], [RC855; H, H, F, Cl, Pr, i-Bu], [RC856; H, H, F, Cl, Pr, t-Bu], [RC857; H, H, F, Cl, Pr, c-PrCH ₂ ], [RC858; H, H, F, Cl, Pr, Ph], [RC859; H, H, F, Cl, Pr, Bn], [RC860; H, H, F , Cl, Pr, CF ₃ ], [RC861; H, H, F, Cl, Pr, CF ₃ CH ₂ ], [RC862; H, H, F, Cl, Pr, CF ₃ CF ₂ ], [RC863; H, H, F, Cl, Pr, CF ₂ H], [RC864; H, H, F, Cl, Pr, CF ₂ HCF ₂ ], [RC865; H, H, Cl, H, Pr, Me], [RC866; H, H, Cl, H, Pr, Et], [RC867; H, H, Cl, H, Pr, Pr], [RC868; H, H, Cl, H, Pr, i-Pr], [RC869; H, H, Cl, H, Pr, c-Pr], [RC870; H, H, Cl, H, Pr, Bu], [RC871; H, H, Cl, H, Pr, i-Bu ], [RC872; H, H, Cl, H, Pr, t-Bu], [RC873; H, H, Cl, H, Pr, c-PrCH ₂ ], [RC874; H, H, Cl, H, Pr, Ph], [RC875; H, H, Cl, H, Pr, Bn], [RC876; H, H, Cl, H, Pr, CF ₃ ], [RC877; H, H, Cl, H, Pr , CF ₃ CH ₂ ], [RC878; H, H, Cl, H, Pr, CF ₃ CF ₂ ], [RC879; H, H, Cl, H, Pr, CF ₂ H], [RC880; H, H, Cl, H, Pr, CF ₂ HCF ₂ ], [RC881; H, H, Cl, Cl, Pr, Me], [RC882; H, H, Cl, Cl, Pr, Et], [RC883; H, H, Cl, Cl, Pr, Pr], [RC884; H, H, Cl, Cl, Pr, i- Pr], [RC885; H, H, Cl, Cl, Pr, c-Pr], [RC886; H, H, Cl, Cl, Pr, Bu], [RC887; H, H, Cl, Cl, Pr, i-Bu], [RC888; H, H, Cl, Cl, Pr, t-Bu], [RC889; H, H, Cl, Cl, Pr, c-PrCH ₂ ], [RC890; H, H, Cl , Cl, Pr, Ph], [RC891; H, H, Cl, Cl, Pr, Bn], [RC892; H, H, Cl, Cl, Pr, CF ₃ ], [RC893; H, H, Cl, Cl, Pr, CF ₃ CH ₂ ], [RC894; H, H, Cl, Cl, Pr, CF ₃ CF ₂ ], [RC895; H, H, Cl, Cl, Pr, CF ₂ H], [RC896; H, H, Cl, Cl, Pr, CF ₂ HCF ₂ ], [RC897; H, H, H, H, Bu, Me], [RC898; H, H, H, H, Bu, Et], [RC899 ; H, H, H, H, Bu, Pr], [RC900; H, H, H, H, Bu, i-Pr], [RC901; H, H, H, H, Bu, c-Pr], [RC902; H, H, H, H, Bu, Bu], [RC903; H, H, H, H, Bu, i-Bu], [RC904; H, H, H, H, Bu, t-Bu ], [RC905; H, H, H, H, Bu, c-PrCH ₂ ], [RC906; H, H, H, H, Bu, Ph], [RC907; H, H, H, H, Bu, Bn], [RC908; H, H, H, H, Bu, CF ₃ ], [RC909; H, H, H, H, Bu, CF ₃ CH ₂ ], [RC910; H, H, H, H, Bu, CF ₃ CF ₂ ], [RC911; H, H, H, H, Bu, CF ₂ H], [RC912; H, H, H, H, Bu, CF ₂ HCF ₂ ], [RC913; H, H, H, Me, Bu, Me], [RC914; H, H, H, Me, Bu, Et], [RC915; H, H, H, Me, Bu, Pr], [RC916; H, H, H, Me, Bu, i-Pr], [RC917; H, H, H, Me, B u, c-Pr], [RC918; H, H, H, Me, Bu, Bu], [RC919; H, H, H, Me, Bu, i-Bu], [RC920; H, H, H, Me, Bu, t-Bu], [RC921; H, H, H, Me, Bu, c-PrCH ₂ ], [RC922; H, H, H, Me, Bu, Ph], [RC923; H, H , H, Me, Bu, Bn], [RC924; H, H, H, Me, Bu, CF ₃ ], [RC925; H, H, H, Me, Bu, CF ₃ CH ₂ ], [RC926; H , H, H, Me, Bu, CF ₃ CF ₂ ], [RC927; H, H, H, Me, Bu, CF ₂ H], [RC928; H, H, H, Me, Bu, CF ₂ HCF ₂ ], [RC929; H, H, Me, Me, Bu, Me], [RC930; H, H, Me, Me, Bu, Et], [RC931; H, H, Me, Me, Bu, Pr], [RC932; H, H, Me, Me, Bu, i-Pr], [RC933; H, H, Me, Me, Bu, c-Pr], [RC934; H, H, Me, Me, Bu, Bu ], [RC935; H, H, Me, Me, Bu, i-Bu], [RC936; H, H, Me, Me, Bu, t-Bu], [RC937; H, H, Me, Me, Bu , c-PrCH ₂ ], [RC938; H, H, Me, Me, Bu, Ph], [RC939; H, H, Me, Me, Bu, Bn], [RC940; H, H, Me, Me, Bu, CF ₃ ], [RC941; H, H, Me, Me, Bu, CF ₃ CH ₂ ], [RC942; H, H, Me, Me, Bu, CF ₃ CF ₂ ], [RC943; H, H , Me, Me, Bu, CF ₂ H], [RC944; H, H, Me, Me, Bu, CF ₂ HCF ₂ ], [RC945; H, H, Me, Et, Bu, Me], [RC946; H, H, Me, Et, Bu, Et], [RC947; H, H, Me, Et, Bu, Pr], [RC948; H, H, Me, Et, Bu, i-Pr], [RC949; H, H, Me, Et, Bu, c-Pr], [RC950; H, H, Me, Et, Bu, Bu], [RC951; H, H, Me, Et, Bu, i-Bu], [ RC952; H, H, Me, Et, Bu, t-Bu], [RC953; H, H, Me, Et, Bu, c-PrCH ₂ ], [RC954; H, H, Me, Et, Bu, Ph ], [RC955; H, H , Me, Et, Bu, Bn], [RC956; H, H, Me, Et, Bu, CF ₃ ], [RC957; H, H, Me, Et, Bu, CF ₃ CH ₂ ], [RC958; H , H, Me, Et, Bu, CF ₃ CF ₂ ], [RC959; H, H, Me, Et, Bu, CF ₂ H], [RC960; H, H, Me, Et, Bu, CF ₂ HCF ₂ ], [RC961; H, H, Me, F, Bu, Me], [RC962; H, H, Me, F, Bu, Et], [RC963; H, H, Me, F, Bu, Pr], [RC964; H, H, Me, F, Bu, i-Pr], [RC965; H, H, Me, F, Bu, c-Pr], [RC966; H, H, Me, F, Bu, Bu ], [RC967; H, H, Me, F, Bu, i-Bu], [RC968; H, H, Me, F, Bu, t-Bu], [RC969; H, H, Me, F, Bu , c-PrCH ₂ ], [RC970; H, H, Me, F, Bu, Ph], [RC971; H, H, Me, F, Bu, Bn], [RC972; H, H, Me, F, Bu, CF ₃ ], [RC973; H, H, Me, F, Bu, CF ₃ CH ₂ ], [RC974; H, H, Me, F, Bu, CF ₃ CF ₂ ], [RC975; H, H , Me, F, Bu, CF ₂ H], [RC976; H, H, Me, F, Bu, CF ₂ HCF ₂ ], [RC977; H, H, Me, Cl, Bu, Me], [RC978; H, H, Me, Cl, Bu, Et], [RC979; H, H, Me, Cl, Bu, Pr], [RC980; H, H, Me, Cl, Bu, i-Pr], [RC981; H, H, Me, Cl, Bu, c-Pr], [RC982; H, H, Me, Cl, Bu, Bu], [RC983; H, H, Me, Cl, Bu, i-Bu], [ RC984; H, H, Me, Cl, Bu, t-Bu], [RC985; H, H, Me, Cl, Bu, c-PrCH ₂ ], [RC986; H, H, Me, Cl, Bu, Ph ], [RC987; H, H, Me, Cl, Bu, Bn], [RC988; H, H, Me, Cl, Bu, CF ₃ ], [RC989; H, H, Me, Cl, Bu, CF ₃ CH ₂ ], [RC990; H, H, Me, Cl, Bu, CF ₃ CF ₂ ], [RC991; H, H, Me, Cl, Bu, CF ₂ H], [RC992; H, H, Me, Cl, Bu, C F ₂ HCF ₂ ], [RC993; H, H, Et, H, Bu, Me], [RC994; H, H, Et, H, Bu, Et], [RC995; H, H, Et, H, Bu , Pr], [RC996; H, H, Et, H, Bu, i-Pr], [RC997; H, H, Et, H, Bu, c-Pr], [RC998; H, H, Et, H , Bu, Bu], [RC999; H, H, Et, H, Bu, i-Bu], [RC1000; H, H, Et, H, Bu, t-Bu],

[RC1001; H, H, Et, H, Bu, c-PrCH ₂ ], [RC1002; H, H, Et, H, Bu, Ph], [RC1003; H, H, Et, H, Bu, Bn] , [RC1004; H, H, Et, H, Bu, CF ₃ ], [RC1005; H, H, Et, H, Bu, CF ₃ CH ₂ ], [RC1006; H, H, Et, H, Bu, CF ₃ CF ₂ ], [RC1007; H, H, Et, H, Bu, CF ₂ H], [RC1008; H, H, Et, H, Bu, CF ₂ HCF ₂ ], [RC1009; H, H, Et, F, Bu, Me], [RC1010; H, H, Et, F, Bu, Et], [RC1011; H, H, Et, F, Bu, Pr], [RC1012; H, H, Et, F, Bu, i-Pr], [RC1013; H, H, Et, F, Bu, c-Pr], [RC1014; H, H, Et, F, Bu, Bu], [RC1015; H, H, Et, F, Bu, i-Bu], [RC1016; H, H, Et, F, Bu, t-Bu], [RC1017; H, H, Et, F, Bu, c-PrCH ₂ ], [RC1018 ; H, H, Et, F, Bu, Ph], [RC1019; H, H, Et, F, Bu, Bn], [RC1020; H, H, Et, F, Bu, CF ₃ ], [RC1021; H, H, Et, F, Bu, CF ₃ CH ₂ ], [RC1022; H, H, Et, F, Bu, CF ₃ CF ₂ ], [RC1023; H, H, Et, F, Bu, CF ₂ H], [RC1024; H, H, Et, F, Bu, CF ₂ HCF ₂ ], [RC1025; H, H, Et, Cl, Bu, Me], [RC1026; H, H, Et, Cl, Bu , Et], [RC1027; H, H, Et, Cl, Bu, Pr], [RC1028; H, H, Et, Cl, Bu, i-Pr], [RC1029; H, H, Et, Cl, Bu , c-Pr], [RC1030; H, H, Et, Cl, Bu, Bu], [RC1031; H, H, Et, Cl, Bu, i-Bu], [RC1032; H, H, Et, Cl , Bu, t-Bu], [RC1033; H, H, Et, Cl, Bu, c-PrCH ₂ ], [RC1034; H, H, Et, Cl, Bu, Ph], [RC1035; H, H, Et, Cl, Bu, Bn], [RC1036; H, H, Et, Cl, Bu, CF ₃ ], [RC1037; H, H, Et, Cl, Bu , CF ₃ CH ₂ ], [RC1038; H, H, Et, Cl, Bu, CF ₃ CF ₂ ], [RC1039; H, H, Et, Cl, Bu, CF ₂ H], [RC1040; H, H , Et, Cl, Bu, CF ₂ HCF ₂ ], [RC1041; H, H, F, H, Bu, Me], [RC1042; H, H, F, H, Bu, Et], [RC1043; H, H, F, H, Bu, Pr], [RC1044; H, H, F, H, Bu, i-Pr], [RC1045; H, H, F, H, Bu, c-Pr], [RC1046; H, H, F, H, Bu, Bu], [RC1047; H, H, F, H, Bu, i-Bu], [RC1048; H, H, F, H, Bu, t-Bu], [ RC1049; H, H, F, H, Bu, c-PrCH ₂ ], [RC1050; H, H, F, H, Bu, Ph], [RC1051; H, H, F, H, Bu, Bn], [RC1052; H, H, F, H, Bu, CF ₃ ], [RC1053; H, H, F, H, Bu, CF ₃ CH ₂ ], [RC1054; H, H, F, H, Bu, CF ₃ CF ₂ ], [RC1055; H, H, F, H, Bu, CF ₂ H], [RC1056; H, H, F, H, Bu, CF ₂ HCF ₂ ], [RC1057; H, H, F , F, Bu, Me], [RC1058; H, H, F, F, Bu, Et], [RC1059; H, H, F, F, Bu, Pr], [RC1060; H, H, F, F , Bu, i-Pr], [RC1061; H, H, F, F, Bu, c-Pr], [RC1062; H, H, F, F, Bu, Bu], [RC1063; H, H, F , F, Bu, i-Bu], [RC1064; H, H, F, F, Bu, t-Bu], [RC1065; H, H, F, F, Bu, c-PrCH ₂ ], [RC1066; H, H, F, F, Bu, Ph], [RC1067; H, H, F, F, Bu, Bn], [RC1068; H, H, F, F, Bu, CF ₃ ], [RC1069; H , H, F, F, Bu, CF ₃ CH ₂ ], [RC1070; H, H, F, F, Bu, CF ₃ CF ₂ ], [RC1071; H, H, F, F, Bu, CF ₂ H ], [RC1072; H, H, F, F, Bu, CF ₂ HCF ₂ ], [RC1073; H, H, F, Cl, Bu, Me], [RC1074; H, H, F, Cl, Bu, Et], [RC1075; H, H, F , Cl, Bu, Pr], [RC1076; H, H, F, Cl, Bu, i-Pr], [RC1077; H, H, F, Cl, Bu, c-Pr], [RC1078; H, H , F, Cl, Bu, Bu], [RC1079; H, H, F, Cl, Bu, i-Bu], [RC1080; H, H, F, Cl, Bu, t-Bu], [RC1081; H , H, F, Cl, Bu, c-PrCH ₂ ], [RC1082; H, H, F, Cl, Bu, Ph], [RC1083; H, H, F, Cl, Bu, Bn], [RC1084; H, H, F, Cl, Bu, CF ₃ ], [RC1085; H, H, F, Cl, Bu, CF ₃ CH ₂ ], [RC1086; H, H, F, Cl, Bu, CF ₃ CF ₂ ], [RC1087; H, H, F, Cl, Bu, CF ₂ H], [RC1088; H, H, F, Cl, Bu, CF ₂ HCF ₂ ], [RC1089; H, H, Cl, H, Bu, Me], [RC1090; H, H, Cl, H, Bu, Et], [RC1091; H, H, Cl, H, Bu, Pr], [RC1092; H, H, Cl, H, Bu, i-Pr], [RC1093; H, H, Cl, H, Bu, c-Pr], [RC1094; H, H, Cl, H, Bu, Bu], [RC1095; H, H, Cl, H, Bu, i-Bu], [RC1096; H, H, Cl, H, Bu, t-Bu], [RC1097; H, H, Cl, H, Bu, c-PrCH ₂ ], [RC1098; H, H , Cl, H, Bu, Ph], [RC1099; H, H, Cl, H, Bu, Bn], [RC1100; H, H, Cl, H, Bu, CF ₃ ], [RC1101; H, H, Cl, H, Bu, CF ₃ CH ₂ ], [RC1102; H, H, Cl, H, Bu, CF ₃ CF ₂ ], [RC1103; H, H, Cl, H, Bu, CF ₂ H], [ RC1104; H, H, Cl, H, Bu, CF ₂ HCF ₂ ], [RC1105; H, H, Cl, Cl, Bu, Me], [RC1106; H, H, Cl, Cl, Bu, Et], [RC1107; H, H, Cl, Cl, Bu, Pr], [RC1108; H, H, Cl, Cl, Bu, i-Pr], [RC1109; H, H, Cl, Cl, Bu, c-Pr ], [RC1110; H, H, Cl, Cl, Bu, Bu], [RC1111; H, H, Cl, Cl, Bu, i-Bu], [RC1112; H, H, Cl, Cl, Bu, t-Bu], [RC1113; H, H, Cl, Cl, Bu, c-PrCH ₂ ], [RC1114; H, H, Cl, Cl, Bu, Ph], [RC1115; H, H, Cl , Cl, Bu, Bn], [RC1116; H, H, Cl, Cl, Bu, CF ₃ ], [RC1117; H, H, Cl, Cl, Bu, CF ₃ CH ₂ ], [RC1118; H, H , Cl, Cl, Bu, CF ₃ CF ₂ ], [RC1119; H, H, Cl, Cl, Bu, CF ₂ H], [RC1120; H, H, Cl, Cl, Bu, CF ₂ HCF ₂ ], [RC1121; H, H, H, H, i-Pr, Me], [RC1122; H, H, H, H, i-Pr, Et], [RC1123; H, H, H, H, i-Pr , Pr], [RC1124; H, H, H, H, i-Pr, i-Pr], [RC1125; H, H, H, H, i-Pr, c-Pr], [RC1126; H, H , H, H, i-Pr, Bu], [RC1127; H, H, H, H, i-Pr, i-Bu], [RC1128; H, H, H, H, i-Pr, t-Bu ], [RC1129; H, H, H, H, i-Pr, c-PrCH ₂ ], [RC1130; H, H, H, H, i-Pr, Ph], [RC1131; H, H, H, H, i-Pr, Bn], [RC1132; H, H, H, H, i-Pr, CF ₃ ], [RC1133; H, H, H, H, i-Pr, CF ₃ CH ₂ ], [ RC1134; H, H, H, H, i-Pr, CF ₃ CF ₂ ], [RC1135; H, H, H, H, i-Pr, CF ₂ H], [RC1136; H, H, H, H , i-Pr, CF ₂ HCF ₂ ], [RC1137; H, H, H, Me, i-Pr, Me], [RC1138; H, H, H, Me, i-Pr, Et], [RC1139; H, H, H, Me, i-Pr, Pr], [RC1140; H, H, H, Me, i-Pr, i-Pr], [RC1141; H, H, H, Me, i-Pr, c-Pr], [RC1142; H, H, H, Me, i-Pr, Bu], [RC1143; H, H, H, Me, i-Pr, i-Bu], [RC1144; H, H, H, Me, i-Pr, t-Bu], [RC1145; H, H, H, Me, i-Pr, c-PrCH ₂ ], [RC1146; H, H, H, Me, i-Pr, Ph ], [RC1147; H, H, H, Me, i-Pr, Bn], [RC1 148; H, H, H, Me, i-Pr, CF ₃ ], [RC1149; H, H, H, Me, i-Pr, CF ₃ CH ₂ ], [RC1150; H, H, H, Me, i-Pr, CF ₃ CF ₂ ], [RC1151; H, H, H, Me, i-Pr, CF ₂ H], [RC1152; H, H, H, Me, i-Pr, CF ₂ HCF ₂ ] , [RC1153; H, H, Me, Me, i-Pr, Me], [RC1154; H, H, Me, Me, i-Pr, Et], [RC1155; H, H, Me, Me, i- Pr, Pr], [RC1156; H, H, Me, Me, i-Pr, i-Pr], [RC1157; H, H, Me, Me, i-Pr, c-Pr], [RC1158; H, H, Me, Me, i-Pr, Bu], [RC1159; H, H, Me, Me, i-Pr, i-Bu], [RC1160; H, H, Me, Me, i-Pr, t- Bu], [RC1161; H, H, Me, Me, i-Pr, c-PrCH ₂ ], [RC1162; H, H, Me, Me, i-Pr, Ph], [RC1163; H, H, Me , Me, i-Pr, Bn], [RC1164; H, H, Me, Me, i-Pr, CF ₃ ], [RC1165; H, H, Me, Me, i-Pr, CF ₃ CH ₂ ], [RC1166; H, H, Me, Me, i-Pr, CF ₃ CF ₂ ], [RC1167; H, H, Me, Me, i-Pr, CF ₂ H], [RC1168; H, H, Me, Me, i-Pr, CF ₂ HCF ₂ ], [RC1169; H, H, Me, Et, i-Pr, Me], [RC1170; H, H, Me, Et, i-Pr, Et], [RC1171 ; H, H, Me, Et, i-Pr, Pr], [RC1172; H, H, Me, Et, i-Pr, i-Pr], [RC1173; H, H, Me, Et, i-Pr , c-Pr], [RC1174; H, H, Me, Et, i-Pr, Bu], [RC1175; H, H, Me, Et, i-Pr, i-Bu], [RC1176; H, H , Me, Et, i-Pr, t-Bu], [RC1177; H, H, Me, Et, i-Pr, c-PrCH ₂ ], [RC1178; H, H, Me, Et, i-Pr, Ph], [RC1179; H, H, Me, Et, i-Pr, Bn], [RC1180; H, H, Me, Et, i-Pr, CF ₃ ], [RC1181; H, H, Me, Et , iP r, CF ₃ CH ₂ ], [RC1182; H, H, Me, Et, i-Pr, CF ₃ CF ₂ ], [RC1183; H, H, Me, Et, i-Pr, CF ₂ H], [ RC1184; H, H, Me, Et, i-Pr, CF ₂ HCF ₂ ], [RC1185; H, H, Me, F, i-Pr, Me], [RC1186; H, H, Me, F, i -Pr, Et], [RC1187; H, H, Me, F, i-Pr, Pr], [RC1188; H, H, Me, F, i-Pr, i-Pr], [RC1189; H, H , Me, F, i-Pr, c-Pr], [RC1190; H, H, Me, F, i-Pr, Bu], [RC1191; H, H, Me, F, i-Pr, i-Bu ], [RC1192; H, H, Me, F, i-Pr, t-Bu], [RC1193; H, H, Me, F, i-Pr, c-PrCH ₂ ], [RC1194; H, H, Me, F, i-Pr, Ph], [RC1195; H, H, Me, F, i-Pr, Bn], [RC1196; H, H, Me, F, i-Pr, CF ₃ ], [RC1197 ; H, H, Me, F, i-Pr, CF ₃ CH ₂ ], [RC1198; H, H, Me, F, i-Pr, CF ₃ CF ₂ ], [RC1199; H, H, Me, F , i-Pr, CF ₂ H], [RC1200; H, H, Me, F, i-Pr, CF ₂ HCF ₂ ],

[RC1201; H, H, Me, Cl, i-Pr, Me], [RC1202; H, H, Me, Cl, i-Pr, Et], [RC1203; H, H, Me, Cl, i-Pr , Pr], [RC1204; H, H, Me, Cl, i-Pr, i-Pr], [RC1205; H, H, Me, Cl, i-Pr, c-Pr], [RC1206; H, H , Me, Cl, i-Pr, Bu], [RC1207; H, H, Me, Cl, i-Pr, i-Bu], [RC1208; H, H, Me, Cl, i-Pr, t-Bu ], [RC1209; H, H, Me, Cl, i-Pr, c-PrCH ₂ ], [RC1210; H, H, Me, Cl, i-Pr, Ph], [RC1211; H, H, Me, Cl, i-Pr, Bn], [RC1212; H, H, Me, Cl, i-Pr, CF ₃ ], [RC1213; H, H, Me, Cl, i-Pr, CF ₃ CH ₂ ], [ RC1214; H, H, Me, Cl, i-Pr, CF ₃ CF ₂ ], [RC1215; H, H, Me, Cl, i-Pr, CF ₂ H], [RC1216; H, H, Me, Cl , i-Pr, CF ₂ HCF ₂ ], [RC1217; H, H, Et, H, i-Pr, Me], [RC1218; H, H, Et, H, i-Pr, Et], [RC1219; H, H, Et, H, i-Pr, Pr], [RC1220; H, H, Et, H, i-Pr, i-Pr], [RC1221; H, H, Et, H, i-Pr, c-Pr], [RC1222; H, H, Et, H, i-Pr, Bu], [RC1223; H, H, Et, H, i-Pr, i-Bu], [RC1224; H, H, Et, H, i-Pr, t-Bu], [RC1225; H, H, Et, H, i-Pr, c-PrCH ₂ ], [RC1226; H, H, Et, H, i-Pr, Ph ], [RC1227; H, H, Et, H, i-Pr, Bn], [RC1228; H, H, Et, H, i-Pr, CF ₃ ], [RC1229; H, H, Et, H, i-Pr, CF ₃ CH ₂ ], [RC1230; H, H, Et, H, i-Pr, CF ₃ CF ₂ ], [RC1231; H, H, Et, H, i-Pr, CF ₂ H] , [RC1232; H, H, Et, H, i-Pr, CF ₂ HCF ₂ ], [RC1233; H, H, Et, F, i-Pr, Me], [RC1234; H, H, Et, F , i-Pr, Et], [RC123 5; H, H, Et, F, i-Pr, Pr], [RC1236; H, H, Et, F, i-Pr, i-Pr], [RC1237; H, H, Et, F, i- Pr, c-Pr], [RC1238; H, H, Et, F, i-Pr, Bu], [RC1239; H, H, Et, F, i-Pr, i-Bu], [RC1240; H, H, Et, F, i-Pr, t-Bu], [RC1241; H, H, Et, F, i-Pr, c-PrCH ₂ ], [RC1242; H, H, Et, F, i-Pr , Ph], [RC1243; H, H, Et, F, i-Pr, Bn], [RC1244; H, H, Et, F, i-Pr, CF ₃ ], [RC1245; H, H, Et, F, i-Pr, CF ₃ CH ₂ ], [RC1246; H, H, Et, F, i-Pr, CF ₃ CF ₂ ], [RC1247; H, H, Et, F, i-Pr, CF ₂ H], [RC1248; H, H, Et, F, i-Pr, CF ₂ HCF ₂ ], [RC1249; H, H, Et, Cl, i-Pr, Me], [RC1250; H, H, Et , Cl, i-Pr, Et], [RC1251; H, H, Et, Cl, i-Pr, Pr], [RC1252; H, H, Et, Cl, i-Pr, i-Pr], [RC1253 ; H, H, Et, Cl, i-Pr, c-Pr], [RC1254; H, H, Et, Cl, i-Pr, Bu], [RC1255; H, H, Et, Cl, i-Pr , i-Bu], [RC1256 ; H, H, Et, Cl, i-Pr, t-Bu], [RC1257; H, H, Et, Cl, i-Pr, c-PrCH 2], [RC1258; H, H, Et, Cl, i-Pr, Ph], [RC1259; H, H, Et, Cl, i-Pr, Bn], [RC1260; H, H, Et, Cl, i-Pr, CF ₃ ], [RC1261; H, H, Et, Cl, i-Pr, CF ₃ CH ₂ ], [RC1262; H, H, Et, Cl, i-Pr, CF ₃ CF ₂ ], [RC1263; H, H , Et, Cl, i-Pr, CF ₂ H], [RC1264; H, H, Et, Cl, i-Pr, CF ₂ HCF ₂ ], [RC1265; H, H, F, H, i-Pr, Me], [RC1266; H, H, F, H, i-Pr, Et], [RC1267; H, H, F, H, i-Pr, Pr], [RC1268; H, H, F, H, i-Pr, i-Pr], [RC1269; H, H, F, H, i-Pr, c-Pr], [RC1270; H, H, F, H, i-Pr, Bu], [RC1271; H, H, F, H, i-Pr, i-Bu], [ RC1272; H, H, F, H, i-Pr, t-Bu], [RC1273; H, H, F, H, i-Pr, c-PrCH ₂ ], [RC1274; H, H, F, H , i-Pr, Ph], [RC1275; H, H, F, H, i-Pr, Bn], [RC1276; H, H, F, H, i-Pr, CF ₃ ], [RC1277; H, H, F, H, i-Pr, CF ₃ CH ₂ ], [RC1278; H, H, F, H, i-Pr, CF ₃ CF ₂ ], [RC1279; H, H, F, H, i- Pr, CF ₂ H], [RC1280; H, H, F, H, i-Pr, CF ₂ HCF ₂ ], [RC1281; H, H, F, F, i-Pr, Me], [RC1282; H , H, F, F, i-Pr, Et], [RC1283; H, H, F, F, i-Pr, Pr], [RC1284; H, H, F, F, i-Pr, i-Pr ], [RC1285; H, H, F, F, i-Pr, c-Pr], [RC1286; H, H, F, F, i-Pr, Bu], [RC1287; H, H, F, F , i-Pr, i-Bu], [RC1288; H, H, F, F, i-Pr, t-Bu], [RC1289; H, H, F, F, i-Pr, c-PrCH ₂ ] , [RC1290; H, H, F, F, i-Pr, Ph], [RC1291; H, H, F, F, i-Pr, Bn], [RC1292; H, H, F, F, i- Pr, CF ₃ ], [RC1293; H, H, F, F, i-Pr, CF ₃ CH ₂ ], [RC1294; H, H, F, F, i-Pr, CF ₃ CF ₂ ], [RC1295 ; H, H, F, F, i-Pr, CF ₂ H], [RC1296; H, H, F, F, i-Pr, CF ₂ HCF ₂ ], [RC1297; H, H, F, Cl, i-Pr, Me], [RC1298; H, H, F, Cl, i-Pr, Et], [RC1299; H, H, F, Cl, i-Pr, Pr], [RC1300; H, H, F, Cl, i-Pr, i-Pr], [RC1301; H, H, F, Cl, i-Pr, c-Pr], [RC1302; H, H, F, Cl, i-Pr, Bu] , [RC1303; H, H, F, Cl, i-Pr, i-Bu], [RC1304; H, H, F, Cl, i-Pr, t-Bu], [RC130 5; H, H, F, Cl, i-Pr, c-PrCH ₂ ], [RC1306; H, H, F, Cl, i-Pr, Ph], [RC1307; H, H, F, Cl, i -Pr, Bn], [RC1308; H, H, F, Cl, i-Pr, CF ₃ ], [RC1309; H, H, F, Cl, i-Pr, CF ₃ CH ₂ ], [RC1310; H , H, F, Cl, i-Pr, CF ₃ CF ₂ ], [RC1311; H, H, F, Cl, i-Pr, CF ₂ H], [RC1312; H, H, F, Cl, i- Pr, CF ₂ HCF ₂ ], [RC1313; H, H, Cl, H, i-Pr, Me], [RC1314; H, H, Cl, H, i-Pr, Et], [RC1315; H, H , Cl, H, i-Pr, Pr], [RC1316; H, H, Cl, H, i-Pr, i-Pr], [RC1317; H, H, Cl, H, i-Pr, c-Pr ], [RC1318; H, H, Cl, H, i-Pr, Bu], [RC1319; H, H, Cl, H, i-Pr, i-Bu], [RC1320; H, H, Cl, H , i-Pr, t-Bu], [RC1321; H, H, Cl, H, i-Pr, c-PrCH ₂ ], [RC1322; H, H, Cl, H, i-Pr, Ph], [ RC1323; H, H, Cl, H, i-Pr, Bn], [RC1324; H, H, Cl, H, i-Pr, CF ₃ ], [RC1325; H, H, Cl, H, i-Pr , CF ₃ CH ₂ ], [RC1326; H, H, Cl, H, i-Pr, CF ₃ CF ₂ ], [RC1327; H, H, Cl, H, i-Pr, CF ₂ H], [RC1328 ; H, H, Cl, H, i-Pr, CF ₂ HCF ₂ ], [RC1329; H, H, Cl, Cl, i-Pr, Me], [RC1330; H, H, Cl, Cl, i- Pr, Et], [RC1331; H, H, Cl, Cl, i-Pr, Pr], [RC1332; H, H, Cl, Cl, i-Pr, i-Pr], [RC1333; H, H, Cl, Cl, i-Pr, c-Pr], [RC1334; H, H, Cl, Cl, i-Pr, Bu], [RC1335; H, H, Cl, Cl, i-Pr, i-Bu] , [RC1336; H, H, Cl, Cl, i-Pr, t-Bu], [RC1337; H, H, Cl, Cl, i-Pr, c-PrCH ₂ ], [RC1338; H, H, Cl , Cl, i-Pr, Ph], [RC1339; H, H , Cl, Cl, i-Pr, Bn], [RC1340; H, H, Cl, Cl, i-Pr, CF ₃ ], [RC1341; H, H, Cl, Cl, i-Pr, CF ₃ CH ₂ ], [RC1342; H, H, Cl, Cl, i-Pr, CF ₃ CF ₂ ], [RC1343; H, H, Cl, Cl, i-Pr, CF ₂ H], [RC1344; H, H, Cl, Cl, i-Pr, CF ₂ HCF ₂ ], [RC1345; H, H, H, H, c-Pr, Me], [RC1346; H, H, H, H, c-Pr, Et], [RC1347; H, H, H, H, c-Pr, Pr], [RC1348; H, H, H, H, c-Pr, i-Pr], [RC1349; H, H, H, H, c -Pr, c-Pr], [RC1350; H, H, H, H, c-Pr, Bu], [RC1351; H, H, H, H, c-Pr, i-Bu], [RC1352; H , H, H, H, c-Pr, t-Bu], [RC1353; H, H, H, H, c-Pr, c-PrCH ₂ ], [RC1354; H, H, H, H, c- Pr, Ph], [RC1355; H, H, H, H, c-Pr, Bn], [RC1356; H, H, H, H, c-Pr, CF ₃ ], [RC1357; H, H, H , H, c-Pr, CF ₃ CH ₂ ], [RC1358; H, H, H, H, c-Pr, CF ₃ CF ₂ ], [RC1359; H, H, H, H, c-Pr, CF ₂ H], [RC1360; H, H, H, H, c-Pr, CF ₂ HCF ₂ ], [RC1361; H, H, H, Me, c-Pr, Me], [RC1362; H, H, H, Me, c-Pr, Et], [RC1363; H, H, H, Me, c-Pr, Pr], [RC1364; H, H, H, Me, c-Pr, i-Pr], [ RC1365; H, H, H, Me, c-Pr, c-Pr], [RC1366; H, H, H, Me, c-Pr, Bu], [RC1367; H, H, H, Me, c- Pr, i-Bu], [RC1368; H, H, H, Me, c-Pr, t-Bu], [RC1369; H, H, H, Me, c-Pr, c-PrCH ₂ ], [RC1370 ; H, H, H, Me, c-Pr, Ph], [RC1371; H, H, H, Me, c-Pr, Bn], [RC1372; H, H, H, Me, c-Pr, CF ₃ ], [RC1373; H, H, H, Me, c-Pr, CF ₃ CH ₂ ], [RC137 4; H, H, H, Me, c-Pr, CF ₃ CF ₂ ], [RC1375; H, H, H, Me, c-Pr, CF ₂ H], [RC1376; H, H, H, Me , c-Pr, CF ₂ HCF ₂ ], [RC1377; H, H, Me, Me, c-Pr, Me], [RC1378; H, H, Me, Me, c-Pr, Et], [RC1379; H, H, Me, Me, c-Pr, Pr], [RC1380; H, H, Me, Me, c-Pr, i-Pr], [RC1381; H, H, Me, Me, c-Pr, c-Pr], [RC1382; H, H, Me, Me, c-Pr, Bu], [RC1383; H, H, Me, Me, c-Pr, i-Bu], [RC1384; H, H, Me, Me, c-Pr, t-Bu], [RC1385; H, H, Me, Me, c-Pr, c-PrCH ₂ ], [RC1386; H, H, Me, Me, c-Pr, Ph ], [RC1387; H, H, Me, Me, c-Pr, Bn], [RC1388; H, H, Me, Me, c-Pr, CF ₃ ], [RC1389; H, H, Me, Me, c-Pr, CF ₃ CH ₂ ], [RC1390; H, H, Me, Me, c-Pr, CF ₃ CF ₂ ], [RC1391; H, H, Me, Me, c-Pr, CF ₂ H] , [RC1392; H, H, Me, Me, c-Pr, CF ₂ HCF ₂ ], [RC1393; H, H, Me, Et, c-Pr, Me], [RC1394; H, H, Me, Et , c-Pr, Et], [RC1395; H, H, Me, Et, c-Pr, Pr], [RC1396; H, H, Me, Et, c-Pr, i-Pr], [RC1397; H , H, Me, Et, c-Pr, c-Pr], [RC1398; H, H, Me, Et, c-Pr, Bu], [RC1399; H, H, Me, Et, c-Pr, i -Bu], [RC1400; H, H, Me, Et, c-Pr, t-Bu],

[RC1401; H, H, Me, Et, c-Pr, c-PrCH ₂ ], [RC1402; H, H, Me, Et, c-Pr, Ph], [RC1403; H, H, Me, Et, c-Pr, Bn], [RC1404; H, H, Me, Et, c-Pr, CF ₃ ], [RC1405; H, H, Me, Et, c-Pr, CF ₃ CH ₂ ], [RC1406; H, H, Me, Et, c-Pr, CF ₃ CF ₂ ], [RC1407; H, H, Me, Et, c-Pr, CF ₂ H], [RC1408; H, H, Me, Et, c -Pr, CF ₂ HCF ₂ ], [RC1409; H, H, Me, F, c-Pr, Me], [RC1410; H, H, Me, F, c-Pr, Et], [RC1411; H, H, Me, F, c-Pr, Pr], [RC1412; H, H, Me, F, c-Pr, i-Pr], [RC1413; H, H, Me, F, c-Pr, c- Pr], [RC1414; H, H, Me, F, c-Pr, Bu], [RC1415; H, H, Me, F, c-Pr, i-Bu], [RC1416; H, H, Me, F, c-Pr, t-Bu], [RC1417; H, H, Me, F, c-Pr, c-PrCH ₂ ], [RC1418; H, H, Me, F, c-Pr, Ph], [RC1419; H, H, Me, F, c-Pr, Bn], [RC1420; H, H, Me, F, c-Pr, CF ₃ ], [RC1421; H, H, Me, F, c- Pr, CF ₃ CH ₂ ], [RC1422; H, H, Me, F, c-Pr, CF ₃ CF ₂ ], [RC1423; H, H, Me, F, c-Pr, CF ₂ H], [ RC1424; H, H, Me, F, c-Pr, CF ₂ HCF ₂ ], [RC1425; H, H, Me, Cl, c-Pr, Me], [RC1426; H, H, Me, Cl, c -Pr, Et], [RC1427; H, H, Me, Cl, c-Pr, Pr], [RC1428; H, H, Me, Cl, c-Pr, i-Pr], [RC1429; H, H , Me, Cl, c-Pr, c-Pr], [RC1430; H, H, Me, Cl, c-Pr, Bu], [RC1431; H, H, Me, Cl, c-Pr, i-Bu ], [RC1432; H, H, Me, Cl, c-Pr, t-Bu], [RC1433; H, H, Me, Cl, c-Pr, c-PrCH ₂ ], [RC1434; H, H, Me, Cl, c-Pr, P h], [RC1435; H, H, Me, Cl, c-Pr, Bn], [RC1436; H, H, Me, Cl, c-Pr, CF ₃ ], [RC1437; H, H, Me, Cl , c-Pr, CF ₃ CH ₂ ], [RC1438; H, H, Me, Cl, c-Pr, CF ₃ CF ₂ ], [RC1439; H, H, Me, Cl, c-Pr, CF ₂ H ], [RC1440; H, H, Me, Cl, c-Pr, CF ₂ HCF ₂ ], [RC1441; H, H, Et, H, c-Pr, Me], [RC1442; H, H, Et, H, c-Pr, Et], [RC1443; H, H, Et, H, c-Pr, Pr], [RC1444; H, H, Et, H, c-Pr, i-Pr], [RC1445; H, H, Et, H, c-Pr, c-Pr], [RC1446; H, H, Et, H, c-Pr, Bu], [RC1447; H, H, Et, H, c-Pr, i-Bu], [RC1448; H, H, Et, H, c-Pr, t-Bu], [RC1449; H, H, Et, H, c-Pr, c-PrCH ₂ ], [RC1450; H , H, Et, H, c-Pr, Ph], [RC1451; H, H, Et, H, c-Pr, Bn], [RC1452; H, H, Et, H, c-Pr, CF ₃ ] , [RC1453; H, H, Et, H, c-Pr, CF ₃ CH ₂ ], [RC1454; H, H, Et, H, c-Pr, CF ₃ CF ₂ ], [RC1455; H, H, Et, H, c-Pr, CF ₂ H], [RC1456; H, H, Et, H, c-Pr, CF ₂ HCF ₂ ], [RC1457; H, H, Et, F, c-Pr, Me ], [RC1458; H, H, Et, F, c-Pr, Et], [RC1459; H, H, Et, F, c-Pr, Pr], [RC1460; H, H, Et, F, c -Pr, i-Pr], [RC1461; H, H, Et, F, c-Pr, c-Pr], [RC1462; H, H, Et, F, c-Pr, Bu], [RC1463; H , H, Et, F, c-Pr, i-Bu], [RC1464; H, H, Et, F, c-Pr, t-Bu], [RC1465; H, H, Et, F, c-Pr , c-PrCH ₂ ], [RC1466; H, H, Et, F, c-Pr, Ph], [RC1467; H, H, Et, F, c-Pr, Bn], [RC1468; H, H, Et, F, c-Pr, CF ₃ ], [RC1469; H, H, Et, F, c-Pr, CF ₃ CH ₂ ], [RC1470; H, H, Et, F, c-Pr, CF ₃ CF ₂ ], [RC1471; H, H, Et, F, c- Pr, CF ₂ H], [RC1472; H, H, Et, F, c-Pr, CF ₂ HCF ₂ ], [RC1473; H, H, Et, Cl, c-Pr, Me], [RC1474; H , H, Et, Cl, c-Pr, Et], [RC1475; H, H, Et, Cl, c-Pr, Pr], [RC1476; H, H, Et, Cl, c-Pr, i-Pr ], [RC1477; H, H, Et, Cl, c-Pr, c-Pr], [RC1478; H, H, Et, Cl, c-Pr, Bu], [RC1479; H, H, Et, Cl , c-Pr, i-Bu], [RC1480; H, H, Et, Cl, c-Pr, t-Bu], [RC1481; H, H, Et, Cl, c-Pr, c-PrCH ₂ ] , [RC1482; H, H, Et, Cl, c-Pr, Ph], [RC1483; H, H, Et, Cl, c-Pr, Bn], [RC1484; H, H, Et, Cl, c- Pr, CF ₃ ], [RC1485; H, H, Et, Cl, c-Pr, CF ₃ CH ₂ ], [RC1486; H, H, Et, Cl, c-Pr, CF ₃ CF ₂ ], [RC1487 ; H, H, Et, Cl, c-Pr, CF ₂ H], [RC1488; H, H, Et, Cl, c-Pr, CF ₂ HCF ₂ ], [RC1489; H, H, F, H, c-Pr, Me], [RC1490; H, H, F, H, c-Pr, Et], [RC1491; H, H, F, H, c-Pr, Pr], [RC1492; H, H, F, H, c-Pr, i-Pr], [RC1493; H, H, F, H, c-Pr, c-Pr], [RC1494; H, H, F, H, c-Pr, Bu] , [RC1495; H, H, F, H, c-Pr, i-Bu], [RC1496; H, H, F, H, c-Pr, t-Bu], [RC1497; H, H, F, H, c-Pr, c-PrCH ₂ ], [RC1498; H, H, F, H, c-Pr, Ph], [RC1499; H, H, F, H, c-Pr, Bn], [RC1500 ; H, H, F, H, c-Pr, CF ₃ ], [RC1501; H, H, F, H, c-Pr, CF ₃ CH ₂ ], [RC1502; H, H, F, H, c -Pr, CF ₃ CF ₂ ], [RC1503; H, H, F, H, c-Pr, CF ₂ H], [RC1504; H, H, F, H, c-Pr, CF ₂ HCF ₂ ], [RC1505; H, H, F, F, c-Pr, Me], [RC1506; H, H, F, F, c-Pr, Et], [RC1507; H, H, F, F, c-Pr, Pr], [RC1508; H, H, F, F, c-Pr , i-Pr], [RC1509; H, H, F, F, c-Pr, c-Pr], [RC1510; H, H, F, F, c-Pr, Bu], [RC1511; H, H , F, F, c-Pr, i-Bu], [RC1512; H, H, F, F, c-Pr, t-Bu], [RC1513; H, H, F, F, c-Pr, c -PrCH ₂ ], [RC1514; H, H, F, F, c-Pr, Ph], [RC1515; H, H, F, F, c-Pr, Bn], [RC1516; H, H, F, F, c-Pr, CF ₃ ], [RC1517; H, H, F, F, c-Pr, CF ₃ CH ₂ ], [RC1518; H, H, F, F, c-Pr, CF ₃ CF ₂ ], [RC1519; H, H, F, F, c-Pr, CF ₂ H], [RC1520; H, H, F, F, c-Pr, CF ₂ HCF ₂ ], [RC1521; H, H, F, Cl, c-Pr, Me], [RC1522; H, H, F, Cl, c-Pr, Et], [RC1523; H, H, F, Cl, c-Pr, Pr], [RC1524; H, H, F, Cl, c-Pr, i-Pr], [RC1525; H, H, F, Cl, c-Pr, c-Pr], [RC1526; H, H, F, Cl, c- Pr, Bu], [RC1527; H, H, F, Cl, c-Pr, i-Bu], [RC1528; H, H, F, Cl, c-Pr, t-Bu], [RC1529; H, H, F, Cl, c-Pr, c-PrCH ₂ ], [RC1530; H, H, F, Cl, c-Pr, Ph], [RC1531; H, H, F, Cl, c-Pr, Bn ], [RC1532; H, H, F, Cl, c-Pr, CF ₃ ], [RC1533; H, H, F, Cl, c-Pr, CF ₃ CH ₂ ], [RC1534; H, H, F , Cl, c-Pr, CF ₃ CF ₂ ], [RC1535; H, H, F, Cl, c-Pr, CF ₂ H], [RC1536; H, H, F, Cl, c-Pr, CF ₂ HCF ₂ ], [RC1537; H, H, Cl, H, c-Pr, Me], [RC1538; H, H, Cl, H, c-Pr, Et], [RC1539; H, H, Cl, H, c-Pr, Pr], [RC1540; H, H, Cl, H, c-Pr, i-Pr], [RC1541; H, H, Cl, H, c-Pr, c-Pr], [RC1542; H, H, Cl, H, c-Pr, Bu], [RC1543; H, H, Cl, H, c-Pr, i-Bu], [RC1544; H, H, Cl, H, c-Pr, t-Bu], [RC1545; H, H, Cl, H, c-Pr, c-PrCH ₂ ], [RC1546; H , H, Cl, H, c-Pr, Ph], [RC1547; H, H, Cl, H, c-Pr, Bn], [RC1548; H, H, Cl, H, c-Pr, CF ₃ ] , [RC1549; H, H, Cl, H, c-Pr, CF ₃ CH ₂ ], [RC1550; H, H, Cl, H, c-Pr, CF ₃ CF ₂ ], [RC1551; H, H, Cl, H, c-Pr, CF ₂ H], [RC1552; H, H, Cl, H, c-Pr, CF ₂ HCF ₂ ], [RC1553; H, H, Cl, Cl, c-Pr, Me ], [RC1554; H, H, Cl, Cl, c-Pr, Et], [RC1555; H, H, Cl, Cl, c-Pr, Pr], [RC1556; H, H, Cl, Cl, c -Pr, i-Pr], [RC1557; H, H, Cl, Cl, c-Pr, c-Pr], [RC1558; H, H, Cl, Cl, c-Pr, Bu], [RC1559; H , H, Cl, Cl, c-Pr, i-Bu], [RC1560; H, H, Cl, Cl, c-Pr, t-Bu], [RC1561; H, H, Cl, Cl, c-Pr , c-PrCH ₂ ], [RC1562; H, H, Cl, Cl, c-Pr, Ph], [RC1563; H, H, Cl, Cl, c-Pr, Bn], [RC1564; H, H, Cl, Cl, c-Pr, CF ₃ ], [RC1565; H, H, Cl, Cl, c-Pr, CF ₃ CH ₂ ], [RC1566; H, H, Cl, Cl, c-Pr, CF ₃ CF ₂ ], [RC1567; H, H, Cl, Cl, c-Pr, CF ₂ H], [RC1568; H, H, Cl, Cl, c-Pr, CF ₂ HCF ₂ ], [RC1569; H, H, H, H, i-Bu, Me], [RC1570; H, H, H, H, i-Bu, Et], [RC1571; H, H, H, H, i-Bu, Pr], [ RC1572; H, H, H, H, i-Bu, iP r], [RC1573; H, H, H, H, i-Bu, c-Pr], [RC1574; H, H, H, H, i-Bu, Bu], [RC1575; H, H, H, H, i-Bu, i-Bu], [RC1576; H, H, H, H, i-Bu, t-Bu], [RC1577; H, H, H, H, i-Bu, c-PrCH ₂ ], [RC1578; H, H, H, H, i-Bu, Ph], [RC1579; H, H, H, H, i-Bu, Bn], [RC1580; H, H, H, H, i -Bu, CF ₃ ], [RC1581; H, H, H, H, i-Bu, CF ₃ CH ₂ ], [RC1582; H, H, H, H, i-Bu, CF ₃ CF ₂ ], [ RC1583; H, H, H, H, i-Bu, CF ₂ H], [RC1584; H, H, H, H, i-Bu, CF ₂ HCF ₂ ], [RC1585; H, H, H, Me , i-Bu, Me], [RC1586; H, H, H, Me, i-Bu, Et], [RC1587; H, H, H, Me, i-Bu, Pr], [RC1588; H, H , H, Me, i-Bu, i-Pr], [RC1589; H, H, H, Me, i-Bu, c-Pr], [RC1590; H, H, H, Me, i-Bu, Bu ], [RC1591; H, H, H, Me, i-Bu, i-Bu], [RC1592; H, H, H, Me, i-Bu, t-Bu], [RC1593; H, H, H , Me, i-Bu, c-PrCH ₂ ], [RC1594; H, H, H, Me, i-Bu, Ph], [RC1595; H, H, H, Me, i-Bu, Bn], [ RC1596; H, H, H, Me, i-Bu, CF ₃ ], [RC1597; H, H, H, Me, i-Bu, CF ₃ CH ₂ ], [RC1598; H, H, H, Me, i-Bu, CF ₃ CF ₂ ], [RC1599; H, H, H, Me, i-Bu, CF ₂ H], [RC1600; H, H, H, Me, i-Bu, CF ₂ HCF ₂ ] ,

[RC1601; H, H, Me, Me, i-Bu, Me], [RC1602; H, H, Me, Me, i-Bu, Et], [RC1603; H, H, Me, Me, i-Bu , Pr], [RC1604; H, H, Me, Me, i-Bu, i-Pr], [RC1605; H, H, Me, Me, i-Bu, c-Pr], [RC1606; H, H , Me, Me, i-Bu, Bu], [RC1607; H, H, Me, Me, i-Bu, i-Bu], [RC1608; H, H, Me, Me, i-Bu, t-Bu ], [RC1609; H, H, Me, Me, i-Bu, c-PrCH ₂ ], [RC1610; H, H, Me, Me, i-Bu, Ph], [RC1611; H, H, Me, Me, i-Bu, Bn], [RC1612; H, H, Me, Me, i-Bu, CF ₃ ], [RC1613; H, H, Me, Me, i-Bu, CF ₃ CH ₂ ], [ RC1614; H, H, Me, Me, i-Bu, CF ₃ CF ₂ ], [RC1615; H, H, Me, Me, i-Bu, CF ₂ H], [RC1616; H, H, Me, Me , i-Bu, CF ₂ HCF ₂ ], [RC1617; H, H, Me, Et, i-Bu, Me], [RC1618; H, H, Me, Et, i-Bu, Et], [RC1619; H, H, Me, Et, i-Bu, Pr], [RC1620; H, H, Me, Et, i-Bu, i-Pr], [RC1621; H, H, Me, Et, i-Bu, c-Pr], [RC1622; H, H, Me, Et, i-Bu, Bu], [RC1623; H, H, Me, Et, i-Bu, i-Bu], [RC1624; H, H, Me, Et, i-Bu, t-Bu], [RC1625; H, H, Me, Et, i-Bu, c-PrCH ₂ ], [RC1626; H, H, Me, Et, i-Bu, Ph ], [RC1627; H, H, Me, Et, i-Bu, Bn], [RC1628; H, H, Me, Et, i-Bu, CF ₃ ], [RC1629; H, H, Me, Et, i-Bu, CF ₃ CH ₂ ], [RC1630; H, H, Me, Et, i-Bu, CF ₃ CF ₂ ], [RC1631; H, H, Me, Et, i-Bu, CF ₂ H] , [RC1632; H, H, Me, Et, i-Bu, CF ₂ HCF ₂ ], [RC1633; H, H, Me, F, i-Bu, Me], [RC1634; H, H, Me, F , i-Bu, Et], [RC1635; H, H, Me, F, i-Bu, Pr], [RC1636; H, H, Me, F, i-Bu, i-Pr], [RC1637; H , H, Me, F, i-Bu, c-Pr], [RC1638; H, H, Me, F, i-Bu, Bu], [RC1639; H, H, Me, F, i-Bu, i -Bu], [RC1640; H, H, Me, F, i-Bu, t-Bu], [RC1641; H, H, Me, F, i-Bu, c-PrCH ₂ ], [RC1642; H, H, Me, F, i-Bu, Ph], [RC1643; H, H, Me, F, i-Bu, Bn], [RC1644; H, H, Me, F, i-Bu, CF ₃ ], [RC1645; H, H, Me, F, i-Bu, CF ₃ CH ₂ ], [RC1646; H, H, Me, F, i-Bu, CF ₃ CF ₂ ], [RC1647; H, H, Me , F, i-Bu, CF ₂ H], [RC1648; H, H, Me, F, i-Bu, CF ₂ HCF ₂ ], [RC1649; H, H, Me, Cl, i-Bu, Me] , [RC1650; H, H, Me, Cl, i-Bu, Et], [RC1651; H, H, Me, Cl, i-Bu, Pr], [RC1652; H, H, Me, Cl, i- Bu, i-Pr], [RC1653; H, H, Me, Cl, i-Bu, c-Pr], [RC1654; H, H, Me, Cl, i-Bu, Bu], [RC1655; H, H, Me, Cl, i-Bu, i-Bu], [RC1656; H, H, Me, Cl, i-Bu, t-Bu], [RC1657; H, H, Me, Cl, i-Bu, c-PrCH ₂ ], [RC1658; H, H, Me, Cl, i-Bu, Ph], [RC1659; H, H, Me, Cl, i-Bu, Bn], [RC1660; H, H, Me , Cl, i-Bu, CF ₃ ], [RC1661; H, H, Me, Cl, i-Bu, CF ₃ CH ₂ ], [RC1662; H, H, Me, Cl, i-Bu, CF ₃ CF ₂ ], [RC1663; H, H, Me, Cl, i-Bu, CF ₂ H], [RC1664; H, H, Me, Cl, i-Bu, CF ₂ HCF ₂ ], [RC1665; H, H , Et, H, i-Bu, Me], [RC1666; H, H, Et, H, i-Bu, Et], [RC1667; H, H, Et, H, i-Bu, Pr], [RC1668 ; H, H, Et, H, i-Bu, i-Pr], [RC1669; H, H, Et, H, i-Bu, c-Pr], [RC1670; H, H, Et, H, i-Bu, Bu], [RC1671; H, H, Et, H, i-Bu, i-Bu], [RC1672; H, H, Et, H, i-Bu, t-Bu], [RC1673; H, H, Et, H, i-Bu, c- PrCH ₂ ], [RC1674; H, H, Et, H, i-Bu, Ph], [RC1675; H, H, Et, H, i-Bu, Bn], [RC1676; H, H, Et, H , i-Bu, CF ₃ ], [RC1677; H, H, Et, H, i-Bu, CF ₃ CH ₂ ], [RC1678; H, H, Et, H, i-Bu, CF ₃ CF ₂ ] , [RC1679; H, H, Et, H, i-Bu, CF ₂ H], [RC1680; H, H, Et, H, i-Bu, CF ₂ HCF ₂ ], [RC1681; H, H, Et , F, i-Bu, Me], [RC1682; H, H, Et, F, i-Bu, Et], [RC1683; H, H, Et, F, i-Bu, Pr], [RC1684; H , H, Et, F, i-Bu, i-Pr], [RC1685; H, H, Et, F, i-Bu, c-Pr], [RC1686; H, H, Et, F, i-Bu , Bu], [RC1687; H, H, Et, F, i-Bu, i-Bu], [RC1688; H, H, Et, F, i-Bu, t-Bu], [RC1689; H, H , Et, F, i-Bu, c-PrCH ₂ ], [RC1690; H, H, Et, F, i-Bu, Ph], [RC1691; H, H, Et, F, i-Bu, Bn] , [RC1692; H, H, Et, F, i-Bu, CF ₃ ], [RC1693; H, H, Et, F, i-Bu, CF ₃ CH ₂ ], [RC1694; H, H, Et, F, i-Bu, CF ₃ CF ₂ ], [RC1695; H, H, Et, F, i-Bu, CF ₂ H], [RC1696; H, H, Et, F, i-Bu, CF ₂ HCF ₂ ], [RC1697; H, H, Et, Cl, i-Bu, Me], [RC1698; H, H, Et, Cl, i-Bu, Et], [RC1699; H, H, Et, Cl, i-Bu, Pr], [RC1700; H, H, Et, Cl, i-Bu, i-Pr], [RC1701; H, H, Et, Cl, i-Bu, c-Pr], [RC1702; H, H, Et, Cl, i-Bu, Bu], [RC1703; H, H, Et, Cl, i-Bu, i-Bu], [RC1704; H, H, Et, Cl, i-Bu, t-Bu], [RC1705; H, H, Et, Cl, i- Bu, c-PrCH ₂ ], [RC1706; H, H, Et, Cl, i-Bu, Ph], [RC1707; H, H, Et, Cl, i-Bu, Bn], [RC1708; H, H , Et, Cl, i-Bu, CF ₃ ], [RC1709; H, H, Et, Cl, i-Bu, CF ₃ CH ₂ ], [RC1710; H, H, Et, Cl, i-Bu, CF ₃ CF ₂ ], [RC1711; H, H, Et, Cl, i-Bu, CF ₂ H], [RC1712; H, H, Et, Cl, i-Bu, CF ₂ HCF ₂ ], [RC1713; H , H, F, H, i-Bu, Me], [RC1714; H, H, F, H, i-Bu, Et], [RC1715; H, H, F, H, i-Bu, Pr], [RC1716; H, H, F, H, i-Bu, i-Pr], [RC1717; H, H, F, H, i-Bu, c-Pr], [RC1718; H, H, F, H , i-Bu, Bu], [RC1719; H, H, F, H, i-Bu, i-Bu], [RC1720; H, H, F, H, i-Bu, t-Bu], [RC1721 ; H, H, F, H, i-Bu, c-PrCH ₂ ], [RC1722; H, H, F, H, i-Bu, Ph], [RC1723; H, H, F, H, i- Bu, Bn], [RC1724; H, H, F, H, i-Bu, CF ₃ ], [RC1725; H, H, F, H, i-Bu, CF ₃ CH ₂ ], [RC1726; H, H, F, H, i-Bu, CF ₃ CF ₂ ], [RC1727; H, H, F, H, i-Bu, CF ₂ H], [RC1728; H, H, F, H, i-Bu , CF ₂ HCF ₂ ], [RC1729; H, H, F, F, i-Bu, Me], [RC1730; H, H, F, F, i-Bu, Et], [RC1731; H, H, F, F, i-Bu, Pr], [RC1732; H, H, F, F, i-Bu, i-Pr], [RC1733; H, H, F, F, i-Bu, c-Pr] , [RC1734; H, H, F, F, i-Bu, Bu], [RC1735; H, H, F, F, i-Bu, i-Bu], [RC1736; H, H, F, F, i-Bu, t-Bu], [RC1737; H, H, F, F, i-Bu, c-PrCH ₂ ], [RC1738; H, H, F, F, i-Bu, Ph], [RC1739; H, H, F, F, i-Bu, Bn], [RC1740; H, H, F, F, i-Bu, CF ₃ ], [RC1741; H, H, F, F, i-Bu, CF ₃ CH ₂ ], [RC1742; H, H, F, F, i-Bu, CF ₃ CF ₂ ], [RC1743; H, H , F, F, i-Bu, CF ₂ H], [RC1744; H, H, F, F, i-Bu, CF ₂ HCF ₂ ], [RC1745; H, H, F, Cl, i-Bu, Me], [RC1746; H, H, F, Cl, i-Bu, Et], [RC1747; H, H, F, Cl, i-Bu, Pr], [RC1748; H, H, F, Cl, i-Bu, i-Pr], [RC1749; H, H, F, Cl, i-Bu, c-Pr], [RC1750; H, H, F, Cl, i-Bu, Bu], [RC1751; H, H, F, Cl, i-Bu, i-Bu], [RC1752; H, H, F, Cl, i-Bu, t-Bu], [RC1753; H, H, F, Cl, i- Bu, c-PrCH ₂ ], [RC1754; H, H, F, Cl, i-Bu, Ph], [RC1755; H, H, F, Cl, i-Bu, Bn], [RC1756; H, H , F, Cl, i-Bu, CF ₃ ], [RC1757; H, H, F, Cl, i-Bu, CF ₃ CH ₂ ], [RC1758; H, H, F, Cl, i-Bu, CF ₃ CF ₂ ], [RC1759; H, H, F, Cl, i-Bu, CF ₂ H], [RC1760; H, H, F, Cl, i-Bu, CF ₂ HCF ₂ ], [RC1761; H , H, Cl, H, i-Bu, Me], [RC1762; H, H, Cl, H, i-Bu, Et], [RC1763; H, H, Cl, H, i-Bu, Pr], [RC1764; H, H, Cl, H, i-Bu, i-Pr], [RC1765; H, H, Cl, H, i-Bu, c-Pr], [RC1766; H, H, Cl, H , i-Bu, Bu], [RC1767; H, H, Cl, H, i-Bu, i-Bu], [RC1768; H, H, Cl, H, i-Bu, t-Bu], [RC1769 ; H, H, Cl, H, i-Bu, c-PrCH ₂ ], [RC1770; H, H, Cl, H, i-Bu, Ph], [RC1771; H, H, Cl, H, i- Bu, Bn], [RC1772; H, H, Cl, H, i-Bu, CF ₃ ], [RC1773; H, H, Cl, H, i-Bu, CF ₃ CH ₂ ], [RC1774; H, H, Cl, H, i-Bu, CF ₃ CF ₂ ], [RC1775; H, H, Cl, H, i-Bu, CF ₂ H], [RC1776; H, H, Cl, H, i-Bu, CF ₂ HCF ₂ ], [RC1777; H, H, Cl, Cl, i-Bu, Me], [RC1778 ; H, H, Cl, Cl, i-Bu, Et], [RC1779; H, H, Cl, Cl, i-Bu, Pr], [RC1780; H, H, Cl, Cl, i-Bu, i -Pr], [RC1781; H, H, Cl, Cl, i-Bu, c-Pr], [RC1782; H, H, Cl, Cl, i-Bu, Bu], [RC1783; H, H, Cl , Cl, i-Bu, i-Bu], [RC1784; H, H, Cl, Cl, i-Bu, t-Bu], [RC1785; H, H, Cl, Cl, i-Bu, c-PrCH ₂ ], [RC1786; H, H, Cl, Cl, i-Bu, Ph], [RC1787; H, H, Cl, Cl, i-Bu, Bn], [RC1788; H, H, Cl, Cl, i-Bu, CF ₃ ], [RC1789; H, H, Cl, Cl, i-Bu, CF ₃ CH ₂ ], [RC1790; H, H, Cl, Cl, i-Bu, CF ₃ CF ₂ ], [RC1791; H, H, Cl, Cl, i-Bu, CF ₂ H], [RC1792; H, H, Cl, Cl, i-Bu, CF ₂ HCF ₂ ], [RC1793; H, H, H, H, t-Bu, Me], [RC1794; H, H, H, H, t-Bu, Et], [RC1795; H, H, H, H, t-Bu, Pr], [RC1796; H, H, H, H, t-Bu, i-Pr], [RC1797; H, H, H, H, t-Bu, c-Pr], [RC1798; H, H, H, H, t-Bu, Bu], [RC1799; H, H, H, H, t-Bu, i-Bu], [RC1800; H, H, H, H, t-Bu, t-Bu],

[RC1801; H, H, H, H, t-Bu, c-PrCH ₂ ], [RC1802; H, H, H, H, t-Bu, Ph], [RC1803; H, H, H, H, t-Bu, Bn], [RC1804; H, H, H, H, t-Bu, CF ₃ ], [RC1805; H, H, H, H, t-Bu, CF ₃ CH ₂ ], [RC1806; H, H, H, H, t-Bu, CF ₃ CF ₂ ], [RC1807; H, H, H, H, t-Bu, CF ₂ H], [RC1808; H, H, H, H, t -Bu, CF ₂ HCF ₂ ], [RC1809; H, H, H, Me, t-Bu, Me], [RC1810; H, H, H, Me, t-Bu, Et], [RC1811; H, H, H, Me, t-Bu, Pr], [RC1812; H, H, H, Me, t-Bu, i-Pr], [RC1813; H, H, H, Me, t-Bu, c- Pr], [RC1814; H, H, H, Me, t-Bu, Bu], [RC1815; H, H, H, Me, t-Bu, i-Bu], [RC1816; H, H, H, Me, t-Bu, t-Bu], [RC1817; H, H, H, Me, t-Bu, c-PrCH ₂ ], [RC1818; H, H, H, Me, t-Bu, Ph], [RC1819; H, H, H, Me, t-Bu, Bn], [RC1820; H, H, H, Me, t-Bu, CF ₃ ], [RC1821; H, H, H, Me, t- Bu, CF ₃ CH ₂ ], [RC1822; H, H, H, Me, t-Bu, CF ₃ CF ₂ ], [RC1823; H, H, H, Me, t-Bu, CF ₂ H], [ RC1824; H, H, H, Me, t-Bu, CF ₂ HCF ₂ ], [RC1825; H, H, Me, Me, t-Bu, Me], [RC1826; H, H, Me, Me, t -Bu, Et], [RC1827; H, H, Me, Me, t-Bu, Pr], [RC1828; H, H, Me, Me, t-Bu, i-Pr], [RC1829; H, H , Me, Me, t-Bu, c-Pr], [RC1830; H, H, Me, Me, t-Bu, Bu], [RC1831; H, H, Me, Me, t-Bu, i-Bu ], [RC1832; H, H, Me, Me, t-Bu, t-Bu], [RC1833; H, H, Me, Me, t-Bu, c-PrCH ₂ ], [RC1834; H, H, Me, Me, t-Bu, Ph], [RC1835; H, H, M e, Me, t-Bu, Bn], [RC1836; H, H, Me, Me, t-Bu, CF ₃ ], [RC1837; H, H, Me, Me, t-Bu, CF ₃ CH ₂ ] , [RC1838; H, H, Me, Me, t-Bu, CF ₃ CF ₂ ], [RC1839; H, H, Me, Me, t-Bu, CF ₂ H], [RC1840; H, H, Me , Me, t-Bu, CF ₂ HCF ₂ ], [RC1841; H, H, Me, Et, t-Bu, Me], [RC1842; H, H, Me, Et, t-Bu, Et], [ RC1843; H, H, Me, Et, t-Bu, Pr], [RC1844; H, H, Me, Et, t-Bu, i-Pr], [RC1845; H, H, Me, Et, t- Bu, c-Pr], [RC1846; H, H, Me, Et, t-Bu, Bu], [RC1847; H, H, Me, Et, t-Bu, i-Bu], [RC1848; H, H, Me, Et, t-Bu, t-Bu], [RC1849; H, H, Me, Et, t-Bu, c-PrCH ₂ ], [RC1850; H, H, Me, Et, t-Bu , Ph], [RC1851; H, H, Me, Et, t-Bu, Bn], [RC1852; H, H, Me, Et, t-Bu, CF ₃ ], [RC1853; H, H, Me, Et, t-Bu, CF ₃ CH ₂ ], [RC1854; H, H, Me, Et, t-Bu, CF ₃ CF ₂ ], [RC1855; H, H, Me, Et, t-Bu, CF ₂ H], [RC1856; H, H, Me, Et, t-Bu, CF ₂ HCF ₂ ], [RC1857; H, H, Me, F, t-Bu, Me], [RC1858; H, H, Me , F, t-Bu, Et], [RC1859; H, H, Me, F, t-Bu, Pr], [RC1860; H, H, Me, F, t-Bu, i-Pr], [RC1861 ; H, H, Me, F, t-Bu, c-Pr], [RC1862; H, H, Me, F, t-Bu, Bu], [RC1863; H, H, Me, F, t-Bu , i-Bu], [RC1864; H, H, Me, F, t-Bu, t-Bu], [RC1865; H, H, Me, F, t-Bu, c-PrCH ₂ ], [RC1866; H, H, Me, F, t-Bu, Ph], [RC1867; H, H, Me, F, t-Bu, Bn], [RC1868; H, H, Me, F, t-Bu, CF ₃ ], [RC1869; H, H, Me, F, t-Bu, CF ₃ CH ₂ ], [RC1870; H, H, Me, F, t-Bu, CF ₃ CF ₂ ], [RC1871; H, H, Me, F, t- Bu, CF ₂ H], [RC1872; H, H, Me, F, t-Bu, CF ₂ HCF ₂ ], [RC1873; H, H, Me, Cl, t-Bu, Me], [RC1874; H , H, Me, Cl, t-Bu, Et], [RC1875; H, H, Me, Cl, t-Bu, Pr], [RC1876; H, H, Me, Cl, t-Bu, i-Pr ], [RC1877; H, H, Me, Cl, t-Bu, c-Pr], [RC1878; H, H, Me, Cl, t-Bu, Bu], [RC1879; H, H, Me, Cl , t-Bu, i-Bu], [RC1880; H, H, Me, Cl, t-Bu, t-Bu], [RC1881; H, H, Me, Cl, t-Bu, c-PrCH ₂ ] , [RC1882; H, H, Me, Cl, t-Bu, Ph], [RC1883; H, H, Me, Cl, t-Bu, Bn], [RC1884; H, H, Me, Cl, t- Bu, CF ₃ ], [RC1885; H, H, Me, Cl, t-Bu, CF ₃ CH ₂ ], [RC1886; H, H, Me, Cl, t-Bu, CF ₃ CF ₂ ], [RC1887 ; H, H, Me, Cl, t-Bu, CF ₂ H], [RC1888; H, H, Me, Cl, t-Bu, CF ₂ HCF ₂ ], [RC1889; H, H, Et, H, t-Bu, Me], [RC1890; H, H, Et, H, t-Bu, Et], [RC1891; H, H, Et, H, t-Bu, Pr], [RC1892; H, H, Et, H, t-Bu, i-Pr], [RC1893; H, H, Et, H, t-Bu, c-Pr], [RC1894; H, H, Et, H, t-Bu, Bu] , [RC1895; H, H, Et, H, t-Bu, i-Bu], [RC1896; H, H, Et, H, t-Bu, t-Bu], [RC1897; H, H, Et, H, t-Bu, c-PrCH ₂ ], [RC1898; H, H, Et, H, t-Bu, Ph], [RC1899; H, H, Et, H, t-Bu, Bn], [RC1900 ; H, H, Et, H, t-Bu, CF ₃ ], [RC1901; H, H, Et, H, t-Bu, CF ₃ CH ₂ ], [RC1902; H, H, Et, H, t -Bu, CF ₃ CF ₂ ], [RC1903; H, H, Et, H, t-Bu, CF ₂ H], [RC1904; H, H, Et, H, t-Bu, CF ₂ HCF ₂ ], [RC1905; H, H, Et, F, t-Bu, Me], [RC1906; H, H, Et, F, t-Bu, Et], [RC1907; H, H, Et, F, t-Bu, Pr], [RC1908; H, H, Et, F, t-Bu, i-Pr], [RC1909; H, H, Et, F, t-Bu, c-Pr], [RC1910; H, H, Et, F, t-Bu, Bu], [RC1911; H, H, Et, F, t-Bu, i-Bu], [RC1912; H, H, Et, F, t-Bu, t-Bu], [RC1913; H, H, Et, F, t-Bu, c-PrCH ₂ ], [RC1914; H, H, Et, F, t-Bu, Ph], [RC1915; H, H, Et, F, t-Bu, Bn], [RC1916; H, H, Et, F, t-Bu, CF ₃ ], [RC1917; H, H, Et, F, t-Bu, CF ₃ CH ₂ ], [RC1918; H, H, Et, F , t-Bu, CF ₃ CF ₂ ], [RC1919; H, H, Et, F, t-Bu, CF ₂ H], [RC1920; H, H, Et, F, t-Bu, CF ₂ HCF ₂ ], [RC1921; H, H, Et, Cl, t-Bu, Me], [RC1922; H, H, Et, Cl, t-Bu, Et], [RC1923; H, H, Et, Cl, t -Bu, Pr], [RC1924; H, H, Et, Cl, t-Bu, i-Pr], [RC1925; H, H, Et, Cl, t-Bu, c-Pr], [RC1926; H , H, Et, Cl, t-Bu, Bu], [RC1927; H, H, Et, Cl, t-Bu, i-Bu], [RC1928; H, H, Et, Cl, t-Bu, t -Bu], [RC1929; H, H, Et, Cl, t-Bu, c-PrCH ₂ ], [RC1930; H, H, Et, Cl, t-Bu, Ph], [RC1931; H, H, Et, Cl, t-Bu, Bn], [RC1932; H, H, Et, Cl, t-Bu, CF ₃ ], [RC1933; H, H, Et, Cl, t-Bu, CF ₃ CH ₂ ] , [RC1934; H, H, Et, Cl, t-Bu, CF ₃ CF ₂ ], [RC1935; H, H, Et, Cl, t-Bu, CF ₂ H], [RC1936; H, H, Et , Cl, t-Bu, CF ₂ H CF ₂ ], [RC1937; H, H, F, H, t-Bu, Me], [RC1938; H, H, F, H, t-Bu, Et], [RC1939; H, H, F, H , t-Bu, Pr], [RC1940; H, H, F, H, t-Bu, i-Pr], [RC1941; H, H, F, H, t-Bu, c-Pr], [RC1942 ; H, H, F, H, t-Bu, Bu], [RC1943; H, H, F, H, t-Bu, i-Bu], [RC1944; H, H, F, H, t-Bu , t-Bu], [RC1945; H, H, F, H, t-Bu, c-PrCH ₂ ], [RC1946; H, H, F, H, t-Bu, Ph], [RC1947; H, H, F, H, t-Bu, Bn], [RC1948; H, H, F, H, t-Bu, CF ₃ ], [RC1949; H, H, F, H, t-Bu, CF ₃ CH ₂ ], [RC1950; H, H, F, H, t-Bu, CF ₃ CF ₂ ], [RC1951; H, H, F, H, t-Bu, CF ₂ H], [RC1952; H, H , F, H, t-Bu, CF ₂ HCF ₂ ], [RC1953; H, H, F, F, t-Bu, Me], [RC1954; H, H, F, F, t-Bu, Et] , [RC1955; H, H, F, F, t-Bu, Pr], [RC1956; H, H, F, F, t-Bu, i-Pr], [RC1957; H, H, F, F, t-Bu, c-Pr], [RC1958; H, H, F, F, t-Bu, Bu], [RC1959; H, H, F, F, t-Bu, i-Bu], [RC1960; H, H, F, F, t-Bu, t-Bu], [RC1961; H, H, F, F, t-Bu, c-PrCH ₂ ], [RC1962; H, H, F, F, t -Bu, Ph], [RC1963; H, H, F, F, t-Bu, Bn], [RC1964; H, H, F, F, t-Bu, CF ₃ ], [RC1965; H, H, F, F, t-Bu, CF ₃ CH ₂ ], [RC1966; H, H, F, F, t-Bu, CF ₃ CF ₂ ], [RC1967; H, H, F, F, t-Bu, CF ₂ H], [RC1968; H, H, F, F, t-Bu, CF ₂ HCF ₂ ], [RC1969; H, H, F, Cl, t-Bu, Me], [RC1970; H, H , F, Cl, t-Bu, Et], [RC1971; H, H, F, Cl, t-Bu, Pr], [RC1972; H, H, F, Cl, t-Bu , i-Pr], [RC1973; H, H, F, Cl, t-Bu, c-Pr], [RC1974; H, H, F, Cl, t-Bu, Bu], [RC1975; H, H , F, Cl, t-Bu, i-Bu], [RC1976; H, H, F, Cl, t-Bu, t-Bu], [RC1977; H, H, F, Cl, t-Bu, c -PrCH ₂ ], [RC1978; H, H, F, Cl, t-Bu, Ph], [RC1979; H, H, F, Cl, t-Bu, Bn], [RC1980; H, H, F, Cl, t-Bu, CF ₃ ], [RC1981; H, H, F, Cl, t-Bu, CF ₃ CH ₂ ], [RC1982; H, H, F, Cl, t-Bu, CF ₃ CF ₂ ], [RC1983; H, H, F, Cl, t-Bu, CF ₂ H], [RC1984; H, H, F, Cl, t-Bu, CF ₂ HCF ₂ ], [RC1985; H, H, Cl, H, t-Bu, Me], [RC1986; H, H, Cl, H, t-Bu, Et], [RC1987; H, H, Cl, H, t-Bu, Pr], [RC1988; H, H, Cl, H, t-Bu, i-Pr], [RC1989; H, H, Cl, H, t-Bu, c-Pr], [RC1990; H, H, Cl, H, t- Bu, Bu], [RC1991; H, H, Cl, H, t-Bu, i-Bu], [RC1992; H, H, Cl, H, t-Bu, t-Bu], [RC1993; H, H, Cl, H, t-Bu, c-PrCH ₂ ], [RC1994; H, H, Cl, H, t-Bu, Ph], [RC1995; H, H, Cl, H, t-Bu, Bn ], [RC1996; H, H, Cl, H, t-Bu, CF ₃ ], [RC1997; H, H, Cl, H, t-Bu, CF ₃ CH ₂ ], [RC1998; H, H, Cl , H, t-Bu, CF ₃ CF ₂ ], [RC1999; H, H, Cl, H, t-Bu, CF ₂ H], [RC2000; H, H, Cl, H, t-Bu, CF ₂ HCF ₂ ],

[RC2001; H, H, Cl, Cl, t-Bu, Me], [RC2002; H, H, Cl, Cl, t-Bu, Et], [RC2003; H, H, Cl, Cl, t-Bu , Pr], [RC2004; H, H, Cl, Cl, t-Bu, i-Pr], [RC2005; H, H, Cl, Cl, t-Bu, c-Pr], [RC2006; H, H , Cl, Cl, t-Bu, Bu], [RC2007; H, H, Cl, Cl, t-Bu, i-Bu], [RC2008; H, H, Cl, Cl, t-Bu, t-Bu ], [RC2009; H, H, Cl, Cl, t-Bu, c-PrCH ₂ ], [RC2010; H, H, Cl, Cl, t-Bu, Ph], [RC2011; H, H, Cl, Cl, t-Bu, Bn], [RC2012; H, H, Cl, Cl, t-Bu, CF ₃ ], [RC2013; H, H, Cl, Cl, t-Bu, CF ₃ CH ₂ ], [ RC2014; H, H, Cl, Cl, t-Bu, CF ₃ CF ₂ ], [RC2015; H, H, Cl, Cl, t-Bu, CF ₂ H], [RC2016; H, H, Cl, Cl , t-Bu, CF ₂ HCF ₂ ], [RC2017; H, H, H, H, CF ₂ H, Me], [RC2018; H, H, H, H, CF ₂ H, Et], [RC2019; H, H, H, H, CF ₂ H, Pr], [RC2020; H, H, H, H, CF ₂ H, i-Pr], [RC2021; H, H, H, H, CF ₂ H, c-Pr], [RC2022; H, H, H, H, CF ₂ H, Bu], [RC2023; H, H, H, H, CF ₂ H, i-Bu], [RC2024; H, H, H, H, CF ₂ H, t-Bu], [RC2025; H, H, H, H, CF ₂ H, c-PrCH ₂ ], [RC2026; H, H, H, H, CF ₂ H, Ph ], [RC2027; H, H, H, H, CF ₂ H, Bn], [RC2028; H, H, H, H, CF ₂ H, CF ₃ ], [RC2029; H, H, H, H, CF ₂ H, CF ₃ CH ₂ ], [RC2030; H, H, H, H, CF ₂ H, CF ₃ CF ₂ ], [RC2031; H, H, H, H, CF ₂ H, CF ₂ H] , [RC2032; H, H, H, H, CF ₂ H, CF ₂ HCF ₂ ], [RC2033; H, H, H, Me, CF ₂ H, Me], [RC2034; H, H, H, Me, CF ₂ H, Et], [RC2035; H, H, H, Me, CF ₂ H, Pr], [RC2036; H, H, H, Me, CF ₂ H, i-Pr], [RC2037; H, H, H, Me, CF ₂ H, c-Pr], [RC2038; H, H, H, Me, CF ₂ H, Bu], [RC2039; H, H, H, Me, CF ₂ H, i-Bu], [RC2040; H, H, H, Me, CF ₂ H, t-Bu], [RC2041; H, H, H, Me, CF ₂ H, c-PrCH ₂ ], [RC2042; H , H, H, Me, CF ₂ H, Ph], [RC2043; H, H, H, Me, CF ₂ H, Bn], [RC2044; H, H, H, Me, CF ₂ H, CF ₃ ] , [RC2045; H, H, H, Me, CF ₂ H, CF ₃ CH ₂ ], [RC2046; H, H, H, Me, CF ₂ H, CF ₃ CF ₂ ], [RC2047; H, H, H, Me, CF ₂ H, CF ₂ H], [RC2048; H, H, H, Me, CF ₂ H, CF ₂ HCF ₂ ], [RC2049; H, H, Me, Me, CF ₂ H, Me ], [RC2050; H, H, Me, Me, CF ₂ H, Et], [RC2051; H, H, Me, Me, CF ₂ H, Pr], [RC2052; H, H, Me, Me, CF ₂ H, i-Pr], [RC2053; H, H, Me, Me, CF ₂ H, c-Pr], [RC2054; H, H, Me, Me, CF ₂ H, Bu], [RC2055; H , H, Me, Me, CF ₂ H, i-Bu], [RC2056; H, H, Me, Me, CF ₂ H, t-Bu], [RC2057; H, H, Me, Me, CF ₂ H , c-PrCH ₂ ], [RC2058; H, H, Me, Me, CF ₂ H, Ph], [RC2059; H, H, Me, Me, CF ₂ H, Bn], [RC2060; H, H, Me, Me, CF ₂ H, CF ₃ ], [RC2061; H, H, Me, Me, CF ₂ H, CF ₃ CH ₂ ], [RC2062; H, H, Me, Me, CF ₂ H, CF ₃ CF ₂ ], [RC2063; H, H, Me, Me, CF ₂ H, CF ₂ H], [RC2064; H, H, Me, Me, CF ₂ H, CF ₂ HCF ₂ ], [RC2065; H, H, Me, Et, CF ₂ H, Me], [RC2066 ; H, H, Me, Et, CF ₂ H, Et], [RC2067; H, H, Me, Et, CF ₂ H, Pr], [RC2068; H, H, Me, Et, CF ₂ H, i -Pr], [RC2069; H, H, Me, Et, CF ₂ H, c-Pr], [RC2070; H, H, Me, Et, CF ₂ H, Bu], [RC2071; H, H, Me , Et, CF ₂ H, i-Bu], [RC2072; H, H, Me, Et, CF ₂ H, t-Bu], [RC2073; H, H, Me, Et, CF ₂ H, c-PrCH ₂ ], [RC2074; H, H, Me, Et, CF ₂ H, Ph], [RC2075; H, H, Me, Et, CF ₂ H, Bn], [RC2076; H, H, Me, Et, CF ₂ H, CF ₃ ], [RC2077; H, H, Me, Et, CF ₂ H, CF ₃ CH ₂ ], [RC2078; H, H, Me, Et, CF ₂ H, CF ₃ CF ₂ ], [RC2079; H, H, Me, Et, CF ₂ H, CF ₂ H], [RC2080; H, H, Me, Et, CF ₂ H, CF ₂ HCF ₂ ], [RC2081; H, H, Me, F, CF ₂ H, Me], [RC2082; H, H, Me, F, CF ₂ H, Et], [RC2083; H, H, Me, F, CF ₂ H, Pr], [RC2084; H, H, Me, F, CF ₂ H, i-Pr], [RC2085; H, H, Me, F, CF ₂ H, c-Pr], [RC2086; H, H, Me, F, CF ₂ H, Bu], [RC2087; H, H, Me, F, CF ₂ H, i-Bu], [RC2088; H, H, Me, F, CF ₂ H, t-Bu], [RC2089; H, H, Me, F, CF ₂ H, c-PrCH ₂ ], [RC2090; H, H, Me, F, CF ₂ H, Ph], [RC2091; H, H, Me, F, CF ₂ H, Bn], [RC2092; H, H, Me, F, CF ₂ H, CF ₃ ], [RC2093; H, H, Me, F, CF ₂ H, CF ₃ CH ₂ ], [RC2094; H, H, Me, F , CF ₂ H, CF ₃ CF ₂ ], [RC2095; H, H, Me, F, CF ₂ H, CF ₂ H], [RC2096; H, H, Me, F, CF ₂ H, CF ₂ HCF ₂ ], [RC2097; H, H, Me, Cl, CF ₂ H, Me], [ RC2098; H, H, Me, Cl, CF ₂ H, Et], [RC2099; H, H, Me, Cl, CF ₂ H, Pr], [RC2100; H, H, Me, Cl, CF ₂ H, i-Pr], [RC2101; H, H, Me, Cl, CF ₂ H, c-Pr], [RC2102; H, H, Me, Cl, CF ₂ H, Bu], [RC2103; H, H, Me, Cl, CF ₂ H, i-Bu], [RC2104; H, H, Me, Cl, CF ₂ H, t-Bu], [RC2105; H, H, Me, Cl, CF ₂ H, c- PrCH ₂ ], [RC2106; H, H, Me, Cl, CF ₂ H, Ph], [RC2107; H, H, Me, Cl, CF ₂ H, Bn], [RC2108; H, H, Me, Cl , CF ₂ H, CF ₃ ], [RC2109; H, H, Me, Cl, CF ₂ H, CF ₃ CH ₂ ], [RC2110; H, H, Me, Cl, CF ₂ H, CF ₃ CF ₂ ] , [RC2111; H, H, Me, Cl, CF ₂ H, CF ₂ H], [RC2112; H, H, Me, Cl, CF ₂ H, CF ₂ HCF ₂ ], [RC2113; H, H, Et , H, CF ₂ H, Me], [RC2114; H, H, Et, H, CF ₂ H, Et], [RC2115; H, H, Et, H, CF ₂ H, Pr], [RC2116; H , H, Et, H, CF ₂ H, i-Pr], [RC2117; H, H, Et, H, CF ₂ H, c-Pr], [RC2118; H, H, Et, H, CF ₂ H , Bu], [RC2119; H, H, Et, H, CF ₂ H, i-Bu], [RC2120; H, H, Et, H, CF ₂ H, t-Bu], [RC2121; H, H , Et, H, CF ₂ H, c-PrCH ₂ ], [RC2122; H, H, Et, H, CF ₂ H, Ph], [RC2123; H, H, Et, H, CF ₂ H, Bn] , [RC2124; H, H, Et, H, CF ₂ H, CF ₃ ], [RC2125; H, H, Et, H, CF ₂ H, CF ₃ CH ₂ ], [RC2126; H, H, Et, H, CF ₂ H, CF ₃ CF ₂ ], [RC2127; H, H, Et, H, CF ₂ H, CF ₂ H], [RC2128; H, H, Et, H, CF ₂ H, CF ₂ HCF ₂ ], [RC2129; H, H, Et, F, CF ₂ H, Me], [RC2130; H, H, Et, F, CF ₂ H, Et], [RC2131; H, H, Et, F, CF ₂ H, Pr], [RC2132; H, H, Et, F, CF ₂ H, i-Pr], [RC2133; H, H, Et, F, CF ₂ H, c-Pr], [RC2134; H, H, Et, F, CF ₂ H, Bu], [RC2135; H, H, Et, F, CF ₂ H, i-Bu], [RC2136; H, H, Et, F, CF ₂ H, t-Bu], [RC2137; H, H, Et, F, CF ₂ H, c-PrCH ₂ ], [RC2138; H, H, Et, F, CF ₂ H, Ph], [RC2139; H, H, Et, F, CF ₂ H, Bn], [RC2140; H, H , Et, F, CF ₂ H, CF ₃ ], [RC2141; H, H, Et, F, CF ₂ H, CF ₃ CH ₂ ], [RC2142; H, H, Et, F, CF ₂ H, CF ₃ CF ₂ ], [RC2143; H, H, Et, F, CF ₂ H, CF ₂ H], [RC2144; H, H, Et, F, CF ₂ H, CF ₂ HCF ₂ ], [RC2145; H , H, Et, Cl, CF ₂ H, Me], [RC2146; H, H, Et, Cl, CF ₂ H, Et], [RC2147; H, H, Et, Cl, CF ₂ H, Pr], [RC2148; H, H, Et, Cl, CF ₂ H, i-Pr], [RC2149; H, H, Et, Cl, CF ₂ H, c-Pr], [RC2150; H, H, Et, Cl , CF ₂ H, Bu], [RC2151; H, H, Et, Cl, CF ₂ H, i-Bu], [RC2152; H, H, Et, Cl, CF ₂ H, t-Bu], [RC2153 ; H, H, Et, Cl, CF ₂ H, c-PrCH ₂ ], [RC2154; H, H, Et, Cl, CF ₂ H, Ph], [RC2155; H, H, Et, Cl, CF ₂ H, Bn], [RC2156; H, H, Et, Cl, CF ₂ H, CF ₃ ], [RC2157; H, H, Et, Cl, CF ₂ H, CF ₃ CH ₂ ], [RC2158; H, H, Et, Cl, CF ₂ H, CF ₃ CF ₂ ], [RC2159; H, H, Et, Cl, CF ₂ H, CF ₂ H], [RC2160; H, H, Et, Cl, CF ₂ H , CF ₂ HCF ₂ ], [RC2161; H, H, F, H, CF ₂ H, Me], [RC2162; H, H, F, H, CF ₂ H, Et], [RC2163; H, H, F, H, CF ₂ H, Pr], [RC2164; H, H, F , H, CF ₂ H, i-Pr], [RC2165; H, H, F, H, CF ₂ H, c-Pr], [RC2166; H, H, F, H, CF ₂ H, Bu], [RC2167; H, H, F, H, CF ₂ H, i-Bu], [RC2168; H, H, F, H, CF ₂ H, t-Bu], [RC2169; H, H, F, H , CF ₂ H, c-PrCH ₂ ], [RC2170; H, H, F, H, CF ₂ H, Ph], [RC2171; H, H, F, H, CF ₂ H, Bn], [RC2172; H, H, F, H, CF ₂ H, CF ₃ ], [RC2173; H, H, F, H, CF ₂ H, CF ₃ CH ₂ ], [RC2174; H, H, F, H, CF ₂ H, CF ₃ CF ₂ ], [RC2175; H, H, F, H, CF ₂ H, CF ₂ H], [RC2176; H, H, F, H, CF ₂ H, CF ₂ HCF ₂ ], [ RC2177; H, H, F, F, CF ₂ H, Me], [RC2178; H, H, F, F, CF ₂ H, Et], [RC2179; H, H, F, F, CF ₂ H, Pr], [RC2180; H, H, F, F, CF ₂ H, i-Pr], [RC2181; H, H, F, F, CF ₂ H, c-Pr], [RC2182; H, H, F, F, CF ₂ H, Bu], [RC2183; H, H, F, F, CF ₂ H, i-Bu], [RC2184; H, H, F, F, CF ₂ H, t-Bu] , [RC2185; H, H, F, F, CF ₂ H, c-PrCH ₂ ], [RC2186; H, H, F, F, CF ₂ H, Ph], [RC2187; H, H, F, F , CF ₂ H, Bn], [RC2188; H, H, F, F, CF ₂ H, CF ₃ ], [RC2189; H, H, F, F, CF ₂ H, CF ₃ CH ₂ ], [RC2190 ; H, H, F, F, CF ₂ H, CF ₃ CF ₂ ], [RC2191; H, H, F, F, CF ₂ H, CF ₂ H], [RC2192; H, H, F, F, CF ₂ H, CF ₂ HCF ₂ ], [RC2193; H, H, F, Cl, CF ₂ H, Me], [RC2194; H, H, F, Cl, CF ₂ H, Et], [RC2 195; H, H, F, Cl, CF ₂ H, Pr], [RC2196; H, H, F, Cl, CF ₂ H, i-Pr], [RC2197; H, H, F, Cl, CF ₂ H, c-Pr], [RC2198; H, H, F, Cl, CF ₂ H, Bu], [RC2199; H, H, F, Cl, CF ₂ H, i-Bu], [RC2200; H, H, F, Cl, CF ₂ H, t-Bu],

[RC2201; H, H, F, Cl, CF ₂ H, c-PrCH ₂ ], [RC2202; H, H, F, Cl, CF ₂ H, Ph], [RC2203; H, H, F, Cl, CF ₂ H, Bn], [RC2204; H, H, F, Cl, CF ₂ H, CF ₃ ], [RC2205; H, H, F, Cl, CF ₂ H, CF ₃ CH ₂ ], [RC2206; H, H, F, Cl, CF ₂ H, CF ₃ CF ₂ ], [RC2207; H, H, F, Cl, CF ₂ H, CF ₂ H], [RC2208; H, H, F, Cl, CF ₂ H, CF ₂ HCF ₂ ], [RC2209; H, H, Cl, H, CF ₂ H, Me], [RC2210; H, H, Cl, H, CF ₂ H, Et], [RC2211; H, H, Cl, H, CF ₂ H, Pr], [RC2212; H, H, Cl, H, CF ₂ H, i-Pr], [RC2213; H, H, Cl, H, CF ₂ H, c- Pr], [RC2214; H, H, Cl, H, CF ₂ H, Bu], [RC2215; H, H, Cl, H, CF ₂ H, i-Bu], [RC2216; H, H, Cl, H, CF ₂ H, t-Bu], [RC2217; H, H, Cl, H, CF ₂ H, c-PrCH ₂ ], [RC2218; H, H, Cl, H, CF ₂ H, Ph], [RC2219; H, H, Cl, H, CF ₂ H, Bn], [RC2220; H, H, Cl, H, CF ₂ H, CF ₃ ], [RC2221; H, H, Cl, H, CF ₂ H, CF ₃ CH ₂ ], [RC2222; H, H, Cl, H, CF ₂ H, CF ₃ CF ₂ ], [RC2223; H, H, Cl, H, CF ₂ H, CF ₂ H], [ RC2224; H, H, Cl, H, CF ₂ H, CF ₂ HCF ₂ ], [RC2225; H, H, Cl, Cl, CF ₂ H, Me], [RC2226; H, H, Cl, Cl, CF ₂ H, Et], [RC2227; H, H, Cl, Cl, CF ₂ H, Pr], [RC2228; H, H, Cl, Cl, CF ₂ H, i-Pr], [RC2229; H, H , Cl, Cl, CF ₂ H, c-Pr], [RC2230; H, H, Cl, Cl, CF ₂ H, Bu], [RC2231; H, H, Cl, Cl, CF ₂ H, i-Bu ], [RC2232; H, H, Cl, Cl, CF ₂ H, t-Bu], [R C2233; H, H, Cl, Cl, CF ₂ H, c-PrCH ₂ ], [RC2234; H, H, Cl, Cl, CF ₂ H, Ph], [RC2235; H, H, Cl, Cl, CF ₂ H, Bn], [RC2236; H, H, Cl, Cl, CF ₂ H, CF ₃ ], [RC2237; H, H, Cl, Cl, CF ₂ H, CF ₃ CH ₂ ], [RC2238; H , H, Cl, Cl, CF ₂ H, CF ₃ CF ₂ ], [RC2239; H, H, Cl, Cl, CF ₂ H, CF ₂ H], [RC2240; H, H, Cl, Cl, CF ₂ H, CF ₂ HCF ₂ ], [RC2241; H, H, H, H, CF ₃ , Me], [RC2242; H, H, H, H, CF ₃ , Et], [RC2243; H, H, H , H, CF ₃ , Pr], [RC2244; H, H, H, H, CF ₃ , i-Pr], [RC2245; H, H, H, H, CF ₃ , c-Pr], [RC2246; H, H, H, H, CF ₃ , Bu], [RC2247; H, H, H, H, CF ₃ , i-Bu], [RC2248; H, H, H, H, CF ₃ , t-Bu ], [RC2249; H, H, H, H, CF ₃ , c-PrCH ₂ ], [RC2250; H, H, H, H, CF ₃ , Ph], [RC2251; H, H, H, H, CF ₃ , Bn], [RC2252; H, H, H, H, CF ₃ , CF ₃ ], [RC2253; H, H, H, H, CF ₃ , CF ₃ CH ₂ ], [RC2254; H, H , H, H, CF ₃ , CF ₃ CF ₂ ], [RC2255; H, H, H, H, CF ₃ , CF ₂ H], [RC2256; H, H, H, H, CF ₃ , CF ₂ HCF ₂ ], [RC2257; H, H, H, Me, CF ₃ , Me], [RC2258; H, H, H, Me, CF ₃ , Et], [RC2259; H, H, H, Me, CF ₃ , Pr], [RC2260; H, H, H, Me, CF ₃ , i-Pr], [RC2261; H, H, H, Me, CF ₃ , c-Pr], [RC2262; H, H, H , Me, CF ₃ , Bu], [RC2263; H, H, H, Me, CF ₃ , i-Bu], [RC2264; H, H, H, Me, CF ₃ , t-Bu], [RC2265; H, H, H, Me, CF ₃ , c-PrCH ₂ ], [RC2266; H, H, H, Me, CF ₃ , Ph], [RC2267; H, H, H, Me, CF ₃ , Bn], [RC2268; H, H, H, Me, CF ₃ , CF ₃ ], [RC2269; H, H, H, Me, CF ₃ , CF ₃ CH ₂ ], [RC2270; H, H, H, Me, CF ₃ , CF ₃ CF ₂ ], [RC2271; H, H, H, Me, CF ₃ , CF ₂ H], [RC2272; H, H, H, Me, CF ₃ , CF ₂ HCF ₂ ], [RC2273; H, H, Me, Me, CF ₃ , Me], [RC2274; H, H, Me, Me, CF ₃ , Et], [RC2275; H, H, Me, Me, CF ₃ , Pr], [RC2276; H, H, Me, Me, CF ₃ , i-Pr], [RC2277; H , H, Me, Me, CF ₃ , c-Pr], [RC2278; H, H, Me, Me, CF ₃ , Bu], [RC2279; H, H, Me, Me, CF ₃ , i-Bu] , [RC2280; H, H, Me, Me, CF ₃ , t-Bu], [RC2281; H, H, Me, Me, CF ₃ , c-PrCH ₂ ], [RC2282; H, H, Me, Me , CF ₃ , Ph], [RC2283; H, H, Me, Me, CF ₃ , Bn], [RC2284; H, H, Me, Me, CF ₃ , CF ₃ ], [RC2285; H, H, Me , Me, CF ₃ , CF ₃ CH ₂ ], [RC2286; H, H, Me, Me, CF ₃ , CF ₃ CF ₂ ], [RC2287; H, H, Me, Me, CF ₃ , CF ₂ H] , [RC2288; H, H, Me, Me, CF ₃ , CF ₂ HCF ₂ ], [RC2289; H, H, Me, Et, CF ₃ , Me], [RC2290; H, H, Me, Et, CF ₃ , Et], [RC2291; H, H, Me, Et, CF ₃ , Pr], [RC2292; H, H, Me, Et, CF ₃ , i-Pr], [RC2293; H, H, Me, Et, CF ₃ , c-Pr], [RC2294; H, H, Me, Et, CF ₃ , Bu], [RC2295; H, H, Me, Et, CF ₃ , i-Bu], [RC2296; H , H, Me, Et, CF ₃ , t-Bu], [RC2297; H, H, Me, Et, CF ₃ , c-PrCH ₂ ], [RC2298; H, H, Me, Et, CF ₃ , Ph ] , [RC2299; H, H, Me, Et, CF ₃ , Bn], [RC2300; H, H, Me, Et, CF ₃ , CF ₃ ], [RC2301; H, H, Me, Et, CF ₃ , CF ₃ CH ₂ ], [RC2302; H, H, Me, Et, CF ₃ , CF ₃ CF ₂ ], [RC2303; H, H, Me, Et, CF ₃ , CF ₂ H], [RC2304; H, H, Me, Et, CF ₃ , CF ₂ HCF ₂ ], [RC2305; H, H, Me, F, CF ₃ , Me], [RC2306; H, H, Me, F, CF ₃ , Et], [ RC2307; H, H, Me, F, CF ₃ , Pr], [RC2308; H, H, Me, F, CF ₃ , i-Pr], [RC2309; H, H, Me, F, CF ₃ , c -Pr], [RC2310; H, H, Me, F, CF ₃ , Bu], [RC2311; H, H, Me, F, CF ₃ , i-Bu], [RC2312; H, H, Me, F , CF ₃ , t-Bu], [RC2313; H, H, Me, F, CF ₃ , c-PrCH ₂ ], [RC2314; H, H, Me, F, CF ₃ , Ph], [RC2315; H , H, Me, F, CF ₃ , Bn], [RC2316; H, H, Me, F, CF ₃ , CF ₃ ], [RC2317; H, H, Me, F, CF ₃ , CF ₃ CH ₂ ] , [RC2318; H, H, Me, F, CF ₃ , CF ₃ CF ₂ ], [RC2319; H, H, Me, F, CF ₃ , CF ₂ H], [RC2320; H, H, Me, F , CF ₃ , CF ₂ HCF ₂ ], [RC2321; H, H, Me, Cl, CF ₃ , Me], [RC2322; H, H, Me, Cl, CF ₃ , Et], [RC2323; H, H , Me, Cl, CF ₃ , Pr], [RC2324; H, H, Me, Cl, CF ₃ , i-Pr], [RC2325; H, H, Me, Cl, CF ₃ , c-Pr], [ RC2326; H, H, Me, Cl, CF ₃ , Bu], [RC2327; H, H, Me, Cl, CF ₃ , i-Bu], [RC2328; H, H, Me, Cl, CF ₃ , t -Bu], [RC2329; H, H, Me, Cl, CF ₃ , c-PrCH ₂ ], [RC2330; H, H, Me, Cl, CF ₃ , Ph], [RC2331; H, H, Me, Cl, CF ₃ , B n], [RC2332; H, H, Me, Cl, CF ₃ , CF ₃ ], [RC2333; H, H, Me, Cl, CF ₃ , CF ₃ CH ₂ ], [RC2334; H, H, Me, Cl, CF ₃ , CF ₃ CF ₂ ], [RC2335; H, H, Me, Cl, CF ₃ , CF ₂ H], [RC2336; H, H, Me, Cl, CF ₃ , CF ₂ HCF ₂ ], [RC2337; H, H, Et, H, CF ₃ , Me], [RC2338; H, H, Et, H, CF ₃ , Et], [RC2339; H, H, Et, H, CF ₃ , Pr] , [RC2340; H, H, Et, H, CF ₃ , i-Pr], [RC2341; H, H, Et, H, CF ₃ , c-Pr], [RC2342; H, H, Et, H, CF ₃ , Bu], [RC2343; H, H, Et, H, CF ₃ , i-Bu], [RC2344; H, H, Et, H, CF ₃ , t-Bu], [RC2345; H, H , Et, H, CF ₃ , c-PrCH ₂ ], [RC2346; H, H, Et, H, CF ₃ , Ph], [RC2347; H, H, Et, H, CF ₃ , Bn], [RC2348 ; H, H, Et, H, CF ₃ , CF ₃ ], [RC2349; H, H, Et, H, CF ₃ , CF ₃ CH ₂ ], [RC2350; H, H, Et, H, CF ₃ , CF ₃ CF ₂ ], [RC2351; H, H, Et, H, CF ₃ , CF ₂ H], [RC2352; H, H, Et, H, CF ₃ , CF ₂ HCF ₂ ], [RC2353; H, H, Et, F, CF ₃ , Me], [RC2354; H, H, Et, F, CF ₃ , Et], [RC2355; H, H, Et, F, CF ₃ , Pr], [RC2356; H , H, Et, F, CF ₃ , i-Pr], [RC2357; H, H, Et, F, CF ₃ , c-Pr], [RC2358; H, H, Et, F, CF ₃ , Bu] , [RC2359; H, H, Et, F, CF ₃ , i-Bu], [RC2360; H, H, Et, F, CF ₃ , t-Bu], [RC2361; H, H, Et, F, CF ₃ , c-PrCH ₂ ], [RC2362; H, H, Et, F, CF ₃ , Ph], [RC2363; H, H, Et, F, CF ₃ , Bn], [RC2364; H, H, Et, F, CF ₃ , CF ₃ ], [RC2 365; H, H, Et, F, CF ₃ , CF ₃ CH ₂ ], [RC2366; H, H, Et, F, CF ₃ , CF ₃ CF ₂ ], [RC2367; H, H, Et, F, CF ₃ , CF ₂ H], [RC2368; H, H, Et, F, CF ₃ , CF ₂ HCF ₂ ], [RC2369; H, H, Et, Cl, CF ₃ , Me], [RC2370; H, H, Et, Cl, CF ₃ , Et], [RC2371; H, H, Et, Cl, CF ₃ , Pr], [RC2372; H, H, Et, Cl, CF ₃ , i-Pr], [RC2373 ; H, H, Et, Cl, CF ₃ , c-Pr], [RC2374; H, H, Et, Cl, CF ₃ , Bu], [RC2375; H, H, Et, Cl, CF ₃ , i- Bu], [RC2376; H, H, Et, Cl, CF ₃ , t-Bu], [RC2377; H, H, Et, Cl, CF ₃ , c-PrCH ₂ ], [RC2378; H, H, Et , Cl, CF ₃ , Ph], [RC2379; H, H, Et, Cl, CF ₃ , Bn], [RC2380; H, H, Et, Cl, CF ₃ , CF ₃ ], [RC2381; H, H , Et, Cl, CF ₃ , CF ₃ CH ₂ ], [RC2382; H, H, Et, Cl, CF ₃ , CF ₃ CF ₂ ], [RC2383; H, H, Et, Cl, CF ₃ , CF ₂ H], [RC2384; H, H, Et, Cl, CF ₃ , CF ₂ HCF ₂ ], [RC2385; H, H, F, H, CF ₃ , Me], [RC2386; H, H, F, H , CF ₃ , Et], [RC2387; H, H, F, H, CF ₃ , Pr], [RC2388; H, H, F, H, CF ₃ , i-Pr], [RC2389; H, H, F, H, CF ₃ , c-Pr], [RC2390; H, H, F, H, CF ₃ , Bu], [RC2391; H, H, F, H, CF ₃ , i-Bu], [RC2392 ; H, H, F, H, CF ₃ , t-Bu], [RC2393; H, H, F, H, CF ₃ , c-PrCH ₂ ], [RC2394; H, H, F, H, CF ₃ , Ph], [RC2395; H, H, F, H, CF ₃ , Bn], [RC2396; H, H, F, H, CF ₃ , CF ₃ ], [RC2397; H, H, F, H, CF ₃ , CF ₃ CH ₂ ], [RC2398; H, H, F, H, CF ₃ , CF ₃ CF ₂ ], [RC2399; H, H, F, H, CF ₃ , CF ₂ H], [RC2400; H, H, F, H, CF ₃ , CF ₂ HCF ₂ ],

[RC2401; H, H, F, F, CF ₃ , Me], [RC2402; H, H, F, F, CF ₃ , Et], [RC2403; H, H, F, F, CF ₃ , Pr] , [RC2404; H, H, F, F, CF ₃ , i-Pr], [RC2405; H, H, F, F, CF ₃ , c-Pr], [RC2406; H, H, F, F, CF ₃ , Bu], [RC2407; H, H, F, F, CF ₃ , i-Bu], [RC2408; H, H, F, F, CF ₃ , t-Bu], [RC2409; H, H , F, F, CF ₃ , c-PrCH ₂ ], [RC2410; H, H, F, F, CF ₃ , Ph], [RC2411; H, H, F, F, CF ₃ , Bn], [RC2412 ; H, H, F, F, CF ₃ , CF ₃ ], [RC2413; H, H, F, F, CF ₃ , CF ₃ CH ₂ ], [RC2414; H, H, F, F, CF ₃ , CF ₃ CF ₂ ], [RC2415; H, H, F, F, CF ₃ , CF ₂ H], [RC2416; H, H, F, F, CF ₃ , CF ₂ HCF ₂ ], [RC2417; H, H, F, Cl, CF ₃ , Me], [RC2418; H, H, F, Cl, CF ₃ , Et], [RC2419; H, H, F, Cl, CF ₃ , Pr], [RC2420; H , H, F, Cl, CF ₃ , i-Pr], [RC2421; H, H, F, Cl, CF ₃ , c-Pr], [RC2422; H, H, F, Cl, CF ₃ , Bu] , [RC2423; H, H, F, Cl, CF ₃ , i-Bu], [RC2424; H, H, F, Cl, CF ₃ , t-Bu], [RC2425; H, H, F, Cl, CF ₃ , c-PrCH ₂ ], [RC2426; H, H, F, Cl, CF ₃ , Ph], [RC2427; H, H, F, Cl, CF ₃ , Bn], [RC2428; H, H, F, Cl, CF ₃ , CF ₃ ], [RC2429; H, H, F, Cl, CF ₃ , CF ₃ CH ₂ ], [RC2430; H, H, F, Cl, CF ₃ , CF ₃ CF ₂ ] , [RC2431; H, H, F, Cl, CF ₃ , CF ₂ H], [RC2432; H, H, F, Cl, CF ₃ , CF ₂ HCF ₂ ], [RC2433; H, H, Cl, H , CF ₃ , Me], [RC2434; H, H, Cl, H, CF ₃ , Et], [RC2 435; H, H, Cl, H, CF ₃ , Pr], [RC2436; H, H, Cl, H, CF ₃ , i-Pr], [RC2437; H, H, Cl, H, CF ₃ , c -Pr], [RC2438; H, H, Cl, H, CF ₃ , Bu], [RC2439; H, H, Cl, H, CF ₃ , i-Bu], [RC2440; H, H, Cl, H , CF ₃ , t-Bu], [RC2441; H, H, Cl, H, CF ₃ , c-PrCH ₂ ], [RC2442; H, H, Cl, H, CF ₃ , Ph], [RC2443; H , H, Cl, H, CF ₃ , Bn], [RC2444; H, H, Cl, H, CF ₃ , CF ₃ ], [RC2445; H, H, Cl, H, CF ₃ , CF ₃ CH ₂ ] , [RC2446; H, H, Cl, H, CF ₃ , CF ₃ CF ₂ ], [RC2447; H, H, Cl, H, CF ₃ , CF ₂ H], [RC2448; H, H, Cl, H , CF ₃ , CF ₂ HCF ₂ ], [RC2449; H, H, Cl, Cl, CF ₃ , Me], [RC2450; H, H, Cl, Cl, CF ₃ , Et], [RC2451; H, H , Cl, Cl, CF ₃ , Pr], [RC2452; H, H, Cl, Cl, CF ₃ , i-Pr], [RC2453; H, H, Cl, Cl, CF ₃ , c-Pr], [ RC2454; H, H, Cl, Cl, CF ₃ , Bu], [RC2455; H, H, Cl, Cl, CF ₃ , i-Bu], [RC2456; H, H, Cl, Cl, CF ₃ , t -Bu], [RC2457; H, H, Cl, Cl, CF ₃ , c-PrCH ₂ ], [RC2458; H, H, Cl, Cl, CF ₃ , Ph], [RC2459; H, H, Cl, Cl, CF ₃ , Bn], [RC2460; H, H, Cl, Cl, CF ₃ , CF ₃ ], [RC2461; H, H, Cl, Cl, CF ₃ , CF ₃ CH ₂ ], [RC2462; H , H, Cl, Cl, CF ₃ , CF ₃ CF ₂ ], [RC2463; H, H, Cl, Cl, CF ₃ , CF ₂ H], [RC2464; H, H, Cl, Cl, CF ₃ , CF ₂ HCF ₂ ], [RC2465; H, H, H, H, CF ₂ HCH ₂ , Me], [RC2466; H, H, H, H, CF ₂ HCH ₂ , Et], [RC2467; H, H, H, H, CF ₂ HCH ₂ , Pr], [RC2468; H, H, H, H, CF ₂ HCH ₂ , i-Pr], [RC2469; H, H, H, H, CF ₂ HCH ₂ , c-Pr], [RC2470 ; H, H, H, H, CF ₂ HCH ₂ , Bu], [RC2471; H, H, H, H, CF ₂ HCH ₂ , i-Bu], [RC2472; H, H, H, H, CF ₂ HCH ₂ , t-Bu], [RC2473; H, H, H, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC2474; H, H, H, H, CF ₂ HCH ₂ , Ph], [RC2475; H, H, H, H, CF ₂ HCH ₂ , Bn], [RC2476; H, H, H, H, CF ₂ HCH ₂ , CF ₃ ], [RC2477; H, H, H, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC2478; H, H, H, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC2479; H, H, H, H, CF ₂ HCH ₂ , CF ₂ H], [RC2480; H, H, H, H, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC2481; H, H, H, Me, CF ₂ HCH ₂ , Me], [RC2482; H, H, H, Me, CF ₂ HCH ₂ , Et], [RC2483; H, H, H, Me, CF ₂ HCH ₂ , Pr], [RC2484; H, H, H, Me, CF ₂ HCH ₂ , i -Pr], [RC2485; H, H, H, Me, CF ₂ HCH ₂ , c-Pr], [RC2486; H, H, H, Me, CF ₂ HCH ₂ , Bu], [RC2487; H, H , H, Me, CF ₂ HCH ₂ , i-Bu], [RC2488; H, H, H, Me, CF ₂ HCH ₂ , t-Bu], [RC2489; H, H, H, Me, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC2490; H, H, H, Me, CF ₂ HCH ₂ , Ph], [RC2491; H, H, H, Me, CF ₂ HCH ₂ , Bn], [RC2492; H , H, H, Me, CF ₂ HCH ₂ , CF ₃ ], [RC2493; H, H, H, Me, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC2494; H, H, H, Me, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC2495; H, H, H, Me, CF ₂ HCH ₂ , CF ₂ H], [RC2496; H, H, H, Me, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC2497; H, H, Me, Me, CF ₂ HCH ₂ , Me], [RC2498; H , H, Me, Me, CF ₂ HCH ₂ , Et], [RC2499; H, H, Me, Me, CF ₂ HCH ₂ , Pr], [RC2500; H, H, Me, Me, CF ₂ HCH ₂ , i-Pr], [RC2501; H, H, Me, Me, CF ₂ HCH ₂ , c-Pr], [RC2502; H, H, Me, Me, CF ₂ HCH ₂ , Bu], [RC2503; H, H, Me, Me, CF ₂ HCH ₂ , i-Bu], [RC2504; H, H, Me, Me, CF ₂ HCH ₂ , t-Bu], [RC2505; H, H, Me, Me, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC2506; H, H, Me, Me, CF ₂ HCH ₂ , Ph], [RC2507; H, H, Me, Me, CF ₂ HCH ₂ , Bn], [RC2508; H, H, Me, Me, CF ₂ HCH ₂ , CF ₃ ], [RC2509; H, H, Me, Me, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC2510; H, H, Me, Me, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC2511; H, H, Me, Me, CF ₂ HCH ₂ , CF ₂ H], [RC2512; H, H, Me, Me, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC2513; H, H, Me, Et, CF ₂ HCH ₂ , Me], [RC2514; H, H, Me, Et, CF ₂ HCH ₂ , Et], [RC2515; H, H, Me , Et, CF ₂ HCH ₂ , Pr], [RC2516; H, H, Me, Et, CF ₂ HCH ₂ , i-Pr], [RC2517; H, H, Me, Et, CF ₂ HCH ₂ , c- Pr], [RC2518; H, H, Me, Et, CF ₂ HCH ₂ , Bu], [RC2519; H, H, Me, Et, CF ₂ HCH ₂ , i-Bu], [RC2520; H, H, Me, Et, CF ₂ HCH ₂ , t-Bu], [RC2521; H, H, Me, Et, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC2522; H, H, Me, Et, CF ₂ HCH ₂ , Ph], [RC2 523; H, H, Me, Et, CF ₂ HCH ₂ , Bn], [RC2524; H, H, Me, Et, CF ₂ HCH ₂ , CF ₃ ], [RC2525; H, H, Me, Et, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC2526; H, H, Me, Et, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC2527; H, H, Me, Et, CF ₂ HCH ₂ , CF ₂ H], [RC2528; H, H, Me, Et, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC2529; H, H, Me, F, CF ₂ HCH ₂ , Me], [RC2530; H, H , Me, F, CF ₂ HCH ₂ , Et], [RC2531; H, H, Me, F, CF ₂ HCH ₂ , Pr], [RC2532; H, H, Me, F, CF ₂ HCH ₂ , i- Pr], [RC2533; H, H, Me, F, CF ₂ HCH ₂ , c-Pr], [RC2534; H, H, Me, F, CF ₂ HCH ₂ , Bu], [RC2535; H, H, Me, F, CF ₂ HCH ₂ , i-Bu], [RC2536; H, H, Me, F, CF ₂ HCH ₂ , t-Bu], [RC2537; H, H, Me, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC2538; H, H, Me, F, CF ₂ HCH ₂ , Ph], [RC2539; H, H, Me, F, CF ₂ HCH ₂ , Bn], [RC2540; H, H, Me, F, CF ₂ HCH ₂ , CF ₃ ], [RC2541; H, H, Me, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC2542; H, H, Me, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC2543; H, H, Me, F, CF ₂ HCH ₂ , CF ₂ H], [RC2544; H, H, Me, F, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC2545; H, H, Me, Cl, CF ₂ HCH ₂ , Me], [RC2546; H, H, Me, Cl, CF ₂ HCH ₂ , Et], [RC2547; H, H, Me, Cl , CF ₂ HCH ₂ , Pr], [RC2548; H, H, Me, Cl, CF ₂ HCH ₂ , i-Pr], [RC2549; H, H, Me, Cl, CF ₂ HCH ₂ , c-Pr] , [RC2550; H, H, Me, Cl, C F ₂ HCH ₂ , Bu], [RC2551; H, H, Me, Cl, CF ₂ HCH ₂ , i-Bu], [RC2552; H, H, Me, Cl, CF ₂ HCH ₂ , t-Bu], [RC2553; H, H, Me, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC2554; H, H, Me, Cl, CF ₂ HCH ₂ , Ph], [RC2555; H, H, Me, Cl, CF ₂ HCH ₂ , Bn], [RC2556; H, H, Me, Cl, CF ₂ HCH ₂ , CF ₃ ], [RC2557; H, H, Me, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC2558; H, H, Me, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC2559; H, H, Me, Cl, CF ₂ HCH ₂ , CF ₂ H], [RC2560; H, H, Me, Cl, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC2561; H, H, Et, H, CF ₂ HCH ₂ , Me], [RC2562; H, H, Et, H, CF ₂ HCH ₂ , Et], [RC2563; H, H, Et, H, CF ₂ HCH ₂ , Pr], [RC2564; H, H, Et, H, CF ₂ HCH ₂ , i-Pr], [RC2565; H, H, Et, H, CF ₂ HCH ₂ , c-Pr], [RC2566; H, H, Et, H, CF ₂ HCH ₂ , Bu], [RC2567; H, H, Et, H, CF ₂ HCH ₂ , i-Bu], [RC2568; H, H, Et, H, CF ₂ HCH ₂ , t-Bu], [RC2569; H, H, Et, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [ RC2570; H, H, Et, H, CF ₂ HCH ₂ , Ph], [RC2571; H, H, Et, H, CF ₂ HCH ₂ , Bn], [RC2572; H, H, Et, H, CF ₂ HCH ₂ , CF ₃ ], [RC2573; H, H, Et, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC2574; H, H, Et, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ] , [RC2575; H, H, Et, H, CF ₂ HCH ₂ , CF ₂ H], [RC2576; H, H, Et, H, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC2577; H, H , Et, F, CF ₂ HCH ₂ , Me], [RC2578; H, H, Et, F, CF ₂ HCH ₂ , Et], [RC2579; H, H, Et, F, CF ₂ HCH ₂ , Pr], [RC2580; H, H, Et , F, CF ₂ HCH ₂ , i-Pr], [RC2581; H, H, Et, F, CF ₂ HCH ₂ , c-Pr], [RC2582; H, H, Et, F, CF ₂ HCH ₂ , Bu], [RC2583; H, H, Et, F, CF ₂ HCH ₂ , i-Bu], [RC2584; H, H, Et, F, CF ₂ HCH ₂ , t-Bu], [RC2585; H, H, Et, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC2586; H, H, Et, F, CF ₂ HCH ₂ , Ph], [RC2587; H, H, Et, F, CF ₂ HCH ₂ , Bn], [RC2588; H, H, Et, F, CF ₂ HCH ₂ , CF ₃ ], [RC2589; H, H, Et, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC2590; H, H, Et, F, CF ₂ HCH ₂ , CF ₃
CF ₂ ], [RC2591; H, H, Et, F, CF ₂ HCH ₂ , CF ₂ H], [RC2592; H, H, Et, F, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC2593; H, H, Et, Cl, CF ₂ HCH ₂ , Me], [RC2594; H, H, Et, Cl, CF ₂ HCH ₂ , Et], [RC2595; H, H, Et, Cl, CF ₂ HCH ₂ , Pr], [RC2596; H, H, Et, Cl, CF ₂ HCH ₂ , i-Pr], [RC2597; H, H, Et, Cl, CF ₂ HCH ₂ , c-Pr], [RC2598; H , H, Et, Cl, CF ₂ HCH ₂ , Bu], [RC2599; H, H, Et, Cl, CF ₂ HCH ₂ , i-Bu], [RC2600; H, H, Et, Cl, CF ₂ HCH ₂ , t-Bu],

[RC2601; H, H, Et, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC2602; H, H, Et, Cl, CF ₂ HCH ₂ , Ph], [RC2603; H, H, Et, Cl, CF ₂ HCH ₂ , Bn], [RC2604; H, H, Et, Cl, CF ₂ HCH ₂ , CF ₃ ], [RC2605; H, H, Et, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC2606; H, H, Et, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC2607; H, H, Et, Cl, CF ₂ HCH ₂ , CF ₂ H], [RC2608; H, H, Et, Cl, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC2609; H, H, F, H, CF ₂ HCH ₂ , Me], [RC2610; H, H, F, H, CF ₂ HCH ₂ , Et], [RC2611; H, H, F, H, CF ₂ HCH ₂ , Pr], [RC2612; H, H, F, H, CF ₂ HCH ₂ , i-Pr], [RC2613; H, H, F, H, CF ₂ HCH ₂ , c-Pr], [RC2614; H, H, F, H, CF ₂ HCH ₂ , Bu], [RC2615; H, H, F, H, CF ₂ HCH ₂ , i-Bu], [RC2616; H, H, F, H, CF ₂ HCH ₂ , t-Bu], [RC2617; H, H, F, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [ RC2618; H, H, F, H, CF ₂ HCH ₂ , Ph], [RC2619; H, H, F, H, CF ₂ HCH ₂ , Bn], [RC2620; H, H, F, H, CF ₂ HCH ₂ , CF ₃ ], [RC2621; H, H, F, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC2622; H, H, F, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ] , [RC2623; H, H, F, H, CF ₂ HCH ₂ , CF ₂ H], [RC2624; H, H, F, H, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC2625; H, H , F, F, CF ₂ HCH ₂ , Me], [RC2626; H, H, F, F, CF ₂ HCH ₂ , Et], [RC2627; H, H, F, F, CF ₂ HCH ₂ , Pr] , [RC2628; H, H, F, F, CF ₂ HCH ₂ , i-Pr], [RC2629; H, H, F, F, CF ₂ HCH ₂ , c-Pr], [RC2630; H, H, F, F, CF ₂ HCH ₂ , Bu], [RC2631; H, H, F, F , CF ₂ HCH ₂ , i-Bu], [RC2632; H, H, F, F, CF ₂ HCH ₂ , t-Bu], [RC2633; H, H, F, F, CF ₂ HCH ₂ , c- PrCH ₂ ], [RC2634; H, H, F, F, CF ₂ HCH ₂ , Ph], [RC2635; H, H, F, F, CF ₂ HCH ₂ , Bn], [RC2636; H, H, F , F, CF ₂ HCH ₂ , CF ₃ ], [RC2637; H, H, F, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC2638; H, H, F, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC2639; H, H, F, F, CF ₂ HCH ₂ , CF ₂ H], [RC2640; H, H, F, F, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [ RC2641; H, H, F, Cl, CF ₂ HCH ₂ , Me], [RC2642; H, H, F, Cl, CF ₂ HCH ₂ , Et], [RC2643; H, H, F, Cl, CF ₂ HCH ₂ , Pr], [RC2644; H, H, F, Cl, CF ₂ HCH ₂ , i-Pr], [RC2645; H, H, F, Cl, CF ₂ HCH ₂ , c-Pr], [RC2646 ; H, H, F, Cl, CF ₂ HCH ₂ , Bu], [RC2647; H, H, F, Cl, CF ₂ HCH ₂ , i-Bu], [RC2648; H, H, F, Cl, CF ₂ HCH ₂ , t-Bu], [RC2649; H, H, F, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC2650; H, H, F, Cl, CF ₂ HCH ₂ , Ph], [RC2651; H, H, F, Cl, CF ₂ HCH ₂ , Bn], [RC2652; H, H, F, Cl, CF ₂ HCH ₂ , CF ₃ ], [RC2653; H, H, F, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC2654; H, H, F, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC2655; H, H, F, Cl, CF ₂ HCH ₂ , CF ₂ H], [RC2656; H, H, F, Cl, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC2657; H, H, Cl, H, CF ₂ HCH ₂ , Me], [RC2658; H, H, Cl, H, CF ₂ HCH ₂ , Et], [RC2659; H, H, Cl, H, CF ₂ HCH ₂ , Pr], [RC2660; H, H, Cl, H, CF ₂ HCH ₂ , i-Pr], [RC2661; H, H, Cl, H, CF ₂ HCH ₂ , c-Pr ], [RC2662; H, H, Cl, H, CF ₂ HCH ₂ , Bu], [RC2663; H, H, Cl, H, CF ₂ HCH ₂ , i-Bu], [RC2664; H, H, Cl , H, CF ₂ HCH ₂ , t-Bu], [RC2665; H, H, Cl, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC2666; H, H, Cl, H, CF ₂ HCH ₂ , Ph], [RC2667; H, H, Cl, H, CF ₂ HCH ₂ , Bn], [RC2668; H, H, Cl, H, CF ₂ HCH ₂ , CF ₃ ], [RC2669; H, H, Cl, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC2670; H, H, Cl, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC2671; H, H, Cl, H, CF ₂ HCH ₂ , CF ₂ H], [RC2672; H, H, Cl, H, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC2673; H, H, Cl, Cl, CF ₂ HCH ₂ , Me], [ RC2674; H, H, Cl, Cl, CF ₂ HCH ₂ , Et], [RC2675; H, H, Cl, Cl, CF ₂ HCH ₂ , Pr], [RC2676; H, H, Cl, Cl, CF ₂ HCH ₂ , i-Pr], [RC2677; H, H, Cl, Cl, CF ₂ HCH ₂ , c-Pr], [RC2678; H, H, Cl, Cl, CF ₂ HCH ₂ , Bu], [RC2679 ; H, H, Cl, Cl, CF ₂ HCH ₂ , i-Bu], [RC2680; H, H, Cl, Cl, CF ₂ HCH ₂ , t-Bu], [RC2681; H, H, Cl, Cl , CF ₂ HCH ₂ , c-PrCH ₂ ], [RC2682; H, H, Cl, Cl, CF ₂ HCH ₂ , Ph], [RC2683; H, H, Cl, Cl, CF ₂ HCH ₂ , Bn], [RC2684; H, H, Cl, Cl, CF ₂ HCH ₂ , CF ₃ ], [RC2685; H, H, Cl, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC2686; H, H, Cl, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC2687; H, H, Cl, Cl, CF ₂ HCH ₂ , CF ₂ H], [RC2688; H, H, Cl, Cl, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC2689; H, H, H, H , CF ₃ CH ₂ , Me], [RC2690; H, H, H, H, CF ₃ CH ₂ , Et], [RC2691; H, H, H, H, CF ₃ CH ₂ , Pr], [RC2692; H, H, H, H, CF ₃ CH ₂ , i-Pr], [RC2693; H, H, H, H, CF ₃ CH ₂ , c-Pr], [RC2694; H, H, H, H, CF ₃ CH ₂ , Bu], [RC2695; H, H, H, H, CF ₃ CH ₂ , i-Bu], [RC2696; H, H, H, H, CF ₃ CH ₂ , t-Bu], [RC2697; H, H, H, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RC2698; H, H, H, H, CF ₃ CH ₂ , Ph], [RC2699; H, H, H, H, CF ₃ CH ₂ , Bn], [RC2700; H, H, H, H, CF ₃ CH ₂ , CF ₃ ], [RC2701; H, H, H, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC2702; H, H, H, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC2703; H, H, H, H, CF ₃ CH ₂ , CF ₂ H], [RC2704; H, H, H, H, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC2705; H, H, H, Me, CF ₃ CH ₂ , Me], [RC2706; H, H, H, Me, CF ₃ CH ₂ , Et], [RC2707; H, H, H, Me, CF ₃ CH ₂ , Pr], [RC2708; H, H, H, Me, CF ₃ CH ₂ , i-Pr], [RC2709; H, H, H, Me, CF ₃ CH ₂ , c-Pr], [RC2710; H, H, H, Me, CF ₃ CH ₂ , Bu], [RC2711; H, H, H, Me, CF ₃ CH ₂ , i-Bu], [RC2712; H, H, H, Me, CF ₃ CH ₂ , t-Bu], [RC2713; H, H, H, Me, CF ₃ C H ₂ , c-PrCH ₂ ], [RC2714; H, H, H, Me, CF ₃ CH ₂ , Ph], [RC2715; H, H, H, Me, CF ₃ CH ₂ , Bn], [RC2716; H, H, H, Me, CF ₃ CH ₂ , CF ₃ ], [RC2717; H, H, H, Me, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC2718; H, H, H, Me, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC2719; H, H, H, Me, CF ₃ CH ₂ , CF ₂ H], [RC2720; H, H, H, Me, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC2721; H, H, Me, Me, CF ₃ CH ₂ , Me], [RC2722; H, H, Me, Me, CF ₃ CH ₂ , Et], [RC2723; H, H, Me , Me, CF ₃ CH ₂ , Pr], [RC2724; H, H, Me, Me, CF ₃ CH ₂ , i-Pr], [RC2725; H, H, Me, Me, CF ₃ CH ₂ , c- Pr], [RC2726; H, H, Me, Me, CF ₃ CH ₂ , Bu], [RC2727; H, H, Me, Me, CF ₃ CH ₂ , i-Bu], [RC2728; H, H, Me, Me, CF ₃ CH ₂ , t-Bu], [RC2729; H, H, Me, Me, CF ₃ CH ₂ , c-PrCH ₂ ], [RC2730; H, H, Me, Me, CF ₃ CH ₂ , Ph], [RC2731; H, H, Me, Me, CF ₃ CH ₂ , Bn], [RC2732; H, H, Me, Me, CF ₃ CH ₂ , CF ₃ ], [RC2733; H, H , Me, Me, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC2734; H, H, Me, Me, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC2735; H, H, Me, Me, CF ₃ CH ₂ , CF ₂ H], [RC2736; H, H, Me, Me, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC2737; H, H, Me, Et, CF ₃ CH ₂ , Me], [RC2738; H, H, Me, Et, CF ₃ CH ₂ , Et], [RC2739; H, H, Me, Et, CF ₃ CH ₂ , Pr], [RC2740; H, H, Me, Et, CF ₃ CH ₂ , i-Pr], [RC2741; H, H, Me, Et, C F ₃ CH ₂ , c-Pr], [RC2742; H, H, Me, Et, CF ₃ CH ₂ , Bu], [RC2743; H, H, Me, Et, CF ₃ CH ₂ , i-Bu], [RC2744; H, H, Me, Et, CF ₃ CH ₂ , t-Bu], [RC2745; H, H, Me, Et, CF ₃ CH ₂ , c-PrCH ₂ ], [RC2746; H, H, Me, Et, CF ₃ CH ₂ , Ph], [RC2747; H, H, Me, Et, CF ₃ CH ₂ , Bn], [RC2748; H, H, Me, Et, CF ₃ CH ₂ , CF ₃ ] , [RC2749; H, H, Me, Et, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC2750; H, H, Me, Et, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC2751; H, H, Me, Et, CF ₃ CH ₂ , CF ₂ H], [RC2752; H, H, Me, Et, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC2753; H, H, Me, F, CF ₃ CH ₂ , Me], [RC2754; H, H, Me, F, CF ₃ CH ₂ , Et], [RC2755; H, H, Me, F, CF ₃ CH ₂ , Pr], [RC2756; H, H, Me, F, CF ₃ CH ₂ , i-Pr], [RC2757; H, H, Me, F, CF ₃ CH ₂ , c-Pr], [RC2758; H, H, Me, F, CF ₃ CH ₂ , Bu], [RC2759; H, H, Me, F, CF ₃ CH ₂ , i-Bu], [RC2760; H, H, Me, F, CF ₃ CH ₂ , t-Bu], [RC2761 ; H, H, Me, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RC2762; H, H, Me, F, CF ₃ CH ₂ , Ph], [RC2763; H, H, Me, F, CF ₃ CH ₂ , Bn], [RC2764; H, H, Me, F, CF ₃ CH ₂ , CF ₃ ], [RC2765; H, H, Me, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC2766; H, H, Me, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC2767; H, H, Me, F, CF ₃ CH ₂ , CF ₂ H], [RC2768; H, H, Me, F, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC2769; H, H, Me, Cl, C F ₃ CH ₂ , Me], [RC2770; H, H, Me, Cl, CF ₃ CH ₂ , Et], [RC2771; H, H, Me, Cl, CF ₃ CH ₂ , Pr], [RC2772; H , H, Me, Cl, CF ₃ CH ₂ , i-Pr], [RC2773; H, H, Me, Cl, CF ₃ CH ₂ , c-Pr], [RC2774; H, H, Me, Cl, CF ₃ CH ₂ , Bu], [RC2775; H, H, Me, Cl, CF ₃ CH
₂ , i-Bu], [RC2776; H, H, Me, Cl, CF ₃ CH ₂ , t-Bu], [RC2777; H, H, Me, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RC2778; H, H, Me, Cl, CF ₃ CH ₂ , Ph], [RC2779; H, H, Me, Cl, CF ₃ CH ₂ , Bn], [RC2780; H, H, Me, Cl, CF ₃ CH ₂ , CF ₃ ], [RC2781; H, H, Me, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC2782; H, H, Me, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC2783; H, H, Me, Cl, CF ₃ CH ₂ , CF ₂ H], [RC2784; H, H, Me, Cl, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC2785; H, H, Et, H, CF ₃ CH ₂ , Me], [RC2786; H, H, Et, H, CF ₃ CH ₂ , Et], [RC2787; H, H, Et, H, CF ₃ CH ₂ , Pr ], [RC2788; H, H, Et, H, CF ₃ CH ₂ , i-Pr], [RC2789; H, H, Et, H, CF ₃ CH ₂ , c-Pr], [RC2790; H, H , Et, H, CF ₃ CH ₂ , Bu], [RC2791; H, H, Et, H, CF ₃ CH ₂ , i-Bu], [RC2792; H, H, Et, H, CF ₃ CH ₂ , t-Bu], [RC2793; H, H, Et, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RC2794; H, H, Et, H, CF ₃ CH ₂ , Ph], [RC2795; H , H, Et, H, CF ₃ CH ₂ , Bn], [RC2796; H, H, Et, H, CF ₃ CH ₂ , CF ₃ ], [RC2797; H, H, Et, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC2798; H, H, Et, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC2799; H, H, Et, H, CF ₃ CH ₂ , CF ₂ H], [RC2800; H, H, Et, H, CF ₃ CH ₂ , CF ₂ HCF ₂ ],

[RC2801; H, H, Et, F, CF ₃ CH ₂ , Me], [RC2802; H, H, Et, F, CF ₃ CH ₂ , Et], [RC2803; H, H, Et, F, CF ₃ CH ₂ , Pr], [RC2804; H, H, Et, F, CF ₃ CH ₂ , i-Pr], [RC2805; H, H, Et, F, CF ₃ CH ₂ , c-Pr], [ RC2806; H, H, Et, F, CF ₃ CH ₂ , Bu], [RC2807; H, H, Et, F, CF ₃ CH ₂ , i-Bu], [RC2808; H, H, Et, F, CF ₃ CH ₂ , t-Bu], [RC2809; H, H, Et, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RC2810; H, H, Et, F, CF ₃ CH ₂ , Ph] , [RC2811; H, H, Et, F, CF ₃ CH ₂ , Bn], [RC2812; H, H, Et, F, CF ₃ CH ₂ , CF ₃ ], [RC2813; H, H, Et, F , CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC2814; H, H, Et, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC2815; H, H, Et, F, CF ₃ CH ₂ , CF ₂ H], [RC2816; H, H, Et, F, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC2817; H, H, Et, Cl, CF ₃ CH ₂ , Me], [RC2818; H , H, Et, Cl, CF ₃ CH ₂ , Et], [RC2819; H, H, Et, Cl, CF ₃ CH ₂ , Pr], [RC2820; H, H, Et, Cl, CF ₃ CH ₂ , i-Pr], [RC2821; H, H, Et, Cl, CF ₃ CH ₂ , c-Pr], [RC2822; H, H, Et, Cl, CF ₃ CH ₂ , Bu], [RC2823; H, H, Et, Cl, CF ₃ CH ₂ , i-Bu], [RC2824; H, H, Et, Cl, CF ₃ CH ₂ , t-Bu], [RC2825; H, H, Et, Cl, CF _{3 CH 2, c-PrCH 2]} , [RC2826; H, H, Et, Cl, CF 3 CH 2, Ph], [RC2827; H, H, Et, Cl, CF 3 CH 2, Bn], [RC2828; H, H, Et, Cl, CF ₃ CH ₂ , CF ₃ ], [RC2829; H, H, Et, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC2830; H, H, Et, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC2831; H, H, Et, Cl, CF ₃ CH ₂ , CF ₂ H], [RC2832; H, H, Et, Cl, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC2833; H, H, F, H, CF ₃ CH ₂ , Me], [RC2834; H, H, F, H, CF ₃ CH ₂ , Et], [RC2835; H, H, F, H, CF ₃ CH ₂ , Pr], [RC2836; H, H, F, H, CF ₃ CH ₂ , i-Pr], [RC2837; H, H, F, H, CF ₃ CH ₂ , c-Pr], [RC2838; H, H, F, H, CF ₃ CH ₂ , Bu], [RC2839; H, H, F, H , CF ₃ CH ₂ , i-Bu], [RC2840; H, H, F, H, CF ₃ CH ₂ , t-Bu], [RC2841; H, H, F, H, CF ₃ CH ₂ , c- PrCH ₂ ], [RC2842; H, H, F, H, CF ₃ CH ₂ , Ph], [RC2843; H, H, F, H, CF ₃ CH ₂ , Bn], [RC2844; H, H, F , H, CF ₃ CH ₂ , CF ₃ ], [RC2845; H, H, F, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC2846; H, H, F, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC2847; H, H, F, H, CF ₃ CH ₂ , CF ₂ H], [RC2848; H, H, F, H, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [ RC2849; H, H, F, F, CF ₃ CH ₂ , Me], [RC2850; H, H, F, F, CF ₃ CH ₂ , Et], [RC2851; H, H, F, F, CF ₃ CH ₂ , Pr], [RC2852; H, H, F, F, CF ₃ CH ₂ , i-Pr], [RC2853; H, H, F, F, CF ₃ CH ₂ , c-Pr], [RC2854 ; H, H, F, F, CF ₃ CH ₂ , Bu], [RC2855; H, H, F, F, CF ₃ CH ₂ , i-Bu], [RC2856; H, H, F, F, CF ₃ CH ₂ , t-Bu], [RC2857; H, H, F, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RC2858; H, H, F, F, CF ₃ CH ₂ , Ph ], [RC2859; H, H, F, F, CF ₃ CH ₂ , Bn], [RC2860; H, H, F, F, CF ₃ CH ₂ , CF ₃ ], [RC2861; H, H, F, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC2862; H, H, F, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC2863; H, H, F, F, CF ₃ CH ₂ , CF ₂ H], [RC2864; H, H, F, F, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC2865; H, H, F, Cl, CF ₃ CH ₂ , Me], [RC2866; H, H, F, Cl, CF ₃ CH ₂ , Et], [RC2867; H, H, F, Cl, CF ₃ CH ₂ , Pr], [RC2868; H, H, F, Cl, CF ₃ CH ₂ , i-Pr], [RC2869; H, H, F, Cl, CF ₃ CH ₂ , c-Pr], [RC2870; H, H, F, Cl, CF ₃ CH ₂ , Bu], [RC2871; H , H, F, Cl, CF ₃ CH ₂ , i-Bu], [RC2872; H, H, F, Cl, CF ₃ CH ₂ , t-Bu], [RC2873; H, H, F, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RC2874; H, H, F, Cl, CF ₃ CH ₂ , Ph], [RC2875; H, H, F, Cl, CF ₃ CH ₂ , Bn], [RC2876 ; H, H, F, Cl, CF ₃ CH ₂ , CF ₃ ], [RC2877; H, H, F, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC2878; H, H, F, Cl , CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC2879; H, H, F, Cl, CF ₃ CH ₂ , CF ₂ H], [RC2880; H, H, F, Cl, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC2881; H, H, Cl, H, CF ₃ CH ₂ , Me], [RC2882; H, H, Cl, H, CF ₃ CH ₂ , Et], [RC2883; H, H, Cl, H, CF ₃ CH ₂ , Pr], [RC2884; H, H, Cl, H, CF ₃ CH ₂ , i-Pr], [RC2885; H, H, Cl, H, CF ₃ CH ₂ , c -Pr], [RC2886; H, H, Cl, H, CF ₃ CH ₂ , Bu], [RC2887; H, H, Cl, H, CF ₃ CH ₂ , i-Bu], [RC2888; H, H, Cl, H, CF ₃ CH ₂ , t-Bu], [RC2889; H, H, Cl, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RC2890; H, H, Cl, H, CF ₃ CH ₂ , Ph], [RC2891; H, H, Cl, H, CF ₃ CH ₂ , Bn], [RC2892; H, H, Cl, H, CF ₃ CH ₂ , CF ₃ ], [RC2893; H, H, Cl, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC2894; H, H, Cl, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC2895; H, H, Cl, H, CF ₃ CH ₂ , CF ₂ H], [RC2896; H, H, Cl, H, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC2897; H, H, Cl, Cl, CF ₃ CH ₂ , Me], [RC2898; H, H, Cl, Cl, CF ₃ CH ₂ , Et], [RC2899; H, H, Cl, Cl, CF ₃ CH ₂ , Pr ], [RC2900; H, H, Cl, Cl, CF ₃ CH ₂ , i-Pr], [RC2901; H, H, Cl, Cl, CF ₃ CH ₂ , c-Pr], [RC2902; H, H , Cl, Cl, CF ₃ CH ₂ , Bu], [RC2903; H, H, Cl, Cl, CF ₃ CH ₂ , i-Bu], [RC2904; H, H, Cl, Cl, CF ₃ CH ₂ , t-Bu], [RC2905; H, H, Cl, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RC2906; H, H, Cl, Cl, CF ₃ CH ₂ , Ph], [RC2907; H , H, Cl, Cl, CF ₃ CH ₂ , Bn], [RC2908; H, H, Cl, Cl, CF ₃ CH ₂ , CF ₃ ], [RC2909; H, H, Cl, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC2910; H, H, Cl, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC2911; H, H, Cl, Cl, CF ₃ CH ₂ , CF ₂ H], [RC2912; H, H, Cl, Cl, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC2913; H, H, H, H, HCCCH ₂ , Me], [RC2914; H, H, H, H, HCCCH ₂ , Et], [RC2915; H, H, H, H, HCCCH ₂ , Pr], [RC2916; H, H, H, H, HCCCH ₂ , i-Pr], [RC2917; H, H, H, H, HCCCH ₂ , c-Pr], [RC2918; H, H, H, H, HCCCH ₂ , Bu], [RC2919; H, H, H, H, HCCCH ₂ , i-Bu], [RC2920; H, H, H, H, HCCCH ₂ , t-Bu], [RC2921; H, H, H, H, HCCCH ₂ , c-PrCH ₂ ], [RC2922; H, H, H, H, HCCCH ₂ , Ph], [RC2923; H, H, H, H, HCCCH ₂ , Bn], [RC2924; H, H, H, H, HCCCH ₂ , CF ₃ ], [RC2925; H, H, H, H, HCCCH ₂ , CF ₃ CH ₂ ], [RC2926; H, H, H, H, HCCCH ₂ , CF ₃ CF ₂ ], [RC2927; H, H, H, H, HCCCH ₂ , CF ₂ H], [RC2928; H, H, H, H, HCCCH ₂ , CF ₂ HCF ₂ ], [RC2929; H, H , H, Me, HCCCH ₂ , Me], [RC2930; H, H, H, Me, HCCCH ₂ , Et], [RC2931; H, H, H, Me, HCCCH ₂ , Pr], [RC2932; H, H, H, Me, HCCCH ₂ , i-Pr], [RC2933; H, H, H, Me, HCCCH ₂ , c-Pr], [RC2934; H, H, H, Me, HCCCH ₂ , Bu], [RC2935; H, H, H, Me, HCCCH ₂ , i-Bu], [RC2936; H, H, H, Me, HCCCH ₂ , t-Bu], [RC2937; H, H, H, Me, HCCCH ₂ , c-PrCH ₂ ], [RC2938; H, H, H, Me, HCCCH ₂ , Ph], [RC2939; H, H, H, Me, HCCCH ₂ , Bn], [RC2940; H, H, H , Me, HCCCH ₂ , CF ₃ ], [RC2941; H, H, H, Me, HCCCH ₂ , CF ₃ CH ₂ ], [RC2942; H, H, H, Me, HCCCH ₂ , CF ₃ CF ₂ ], [RC2943; H, H, H, Me, HCCCH ₂ , CF ₂ H], [RC2944; H, H, H, Me, HCCCH ₂ , CF ₂ HCF ₂ ], [RC2945; H, H, Me, Me, HCCCH ₂ , Me], [RC2946; H, H, Me, Me, HCCCH ₂ , Et], [RC2947; H, H, Me, Me, HCCCH ₂ , Pr], [RC2948; H, H, Me, Me, HCCCH ₂ , i-Pr], [RC2949; H, H, Me , Me, HCCCH ₂ , c-Pr], [RC2950; H, H, Me, Me, HCCCH ₂ , Bu], [RC2951; H, H, Me, Me, HCCCH ₂ , i-Bu], [RC2952; H, H, Me, Me, HCCCH ₂ , t-Bu], [RC2953; H, H, Me, Me, HCCCH ₂ , c-PrCH ₂ ], [RC2954; H, H, Me, Me, HCCCH ₂ , Ph], [RC2955; H, H, Me, Me, HCCCH ₂ , Bn], [RC2956; H, H, Me, Me, HCCCH ₂ , CF ₃ ], [RC2957; H, H, Me, Me, HCCCH ₂ , CF ₃ CH ₂ ], [RC2958; H, H, Me, Me, HCCCH ₂ , CF ₃ CF ₂ ], [RC2959; H, H, Me, Me, HCCCH ₂ , CF ₂ H], [RC2960; H, H, Me, Me, HCCCH ₂ , CF ₂ HCF ₂ ], [RC2961; H, H, Me, Et, HCCCH ₂ , Me], [RC2962; H, H, Me, Et, HCCCH ₂ , Et] , [RC2963; H, H, Me, Et, HCCCH ₂ , Pr], [RC2964; H, H, Me, Et, HCCCH ₂ , i-Pr], [RC2965; H, H, Me, Et, HCCCH ₂ , c-Pr], [RC2966; H, H, Me, Et, HCCCH ₂ , Bu], [RC2967; H, H, Me, Et, HCCCH ₂ , i-Bu], [RC2968; H, H, Me , Et, HCCCH ₂ , t-Bu], [RC2969; H, H, Me, Et, HCCCH ₂ , c-PrCH ₂ ], [RC2970; H, H, Me, Et, HCCCH ₂ , Ph], [RC2971 ; H, H, Me, Et, HCCCH ₂ , Bn], [RC2972; H, H, Me, Et, HCCCH ₂ , CF ₃ ], [RC2973; H, H, Me, Et, HCCCH ₂ , CF ₃ CH ₂ ], [RC2974; H, H, Me, Et, HCCCH ₂ , CF ₃ CF ₂ ], [RC2975; H, H, Me, Et, HCCCH ₂ , CF ₂ H], [RC 2976; H, H, Me, Et, HCCCH ₂ , CF ₂ HCF ₂ ], [RC2977; H, H, Me, F, HCCCH ₂ , Me], [RC2978; H, H, Me, F, HCCCH ₂ , Et], [RC2979; H, H, Me, F, HCCCH ₂ , Pr], [RC2980; H, H, Me, F, HCCCH ₂ , i-Pr], [RC2981; H, H, Me, F, HCCCH ₂ , c-Pr], [RC2982; H, H, Me, F, HCCCH ₂ , Bu], [RC2983; H, H, Me, F, HCCCH ₂ , i-Bu], [RC2984; H, H , Me, F, HCCCH ₂ , t-Bu], [RC2985; H, H, Me, F, HCCCH ₂ , c-PrCH ₂ ], [RC2986; H, H, Me, F, HCCCH ₂ , Ph], [RC2987; H, H, Me, F, HCCCH ₂ , Bn], [RC2988; H, H, Me, F, HCCCH ₂ , CF ₃ ], [RC2989; H, H, Me, F, HCCCH ₂ , CF ₃ CH ₂ ], [RC2990; H, H, Me, F, HCCCH ₂ , CF ₃ CF ₂ ], [RC2991; H, H, Me, F, HCCCH ₂ , CF ₂ H], [RC2992; H, H , Me, F, HCCCH ₂ ,
CF ₂ HCF ₂ ], [RC2993; H, H, Me, Cl, HCCCH ₂ , Me], [RC2994; H, H, Me, Cl, HCCCH ₂ , Et], [RC2995; H, H, Me, Cl , HCCCH ₂ , Pr], [RC2996; H, H, Me, Cl, HCCCH ₂ , i-Pr], [RC2997; H, H, Me, Cl, HCCCH ₂ , c-Pr], [RC2998; H, H, Me, Cl, HCCCH ₂ , Bu], [RC2999; H, H, Me, Cl, HCCCH ₂ , i-Bu], [RC3000; H, H, Me, Cl, HCCCH ₂ , t-Bu],

[RC3001; H, H, Me, Cl, HCCCH ₂ , c-PrCH ₂ ], [RC3002; H, H, Me, Cl, HCCCH ₂ , Ph], [RC3003; H, H, Me, Cl, HCCCH ₂ , Bn], [RC3004; H, H, Me, Cl, HCCCH ₂ , CF ₃ ], [RC3005; H, H, Me, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RC3006; H, H, Me , Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RC3007; H, H, Me, Cl, HCCCH ₂ , CF ₂ H], [RC3008; H, H, Me, Cl, HCCCH ₂ , CF ₂ HCF ₂ ] , [RC3009; H, H, Et, H, HCCCH ₂ , Me], [RC3010; H, H, Et, H, HCCCH ₂ , Et], [RC3011; H, H, Et, H, HCCCH ₂ , Pr ], [RC3012; H, H, Et, H, HCCCH ₂ , i-Pr], [RC3013; H, H, Et, H, HCCCH ₂ , c-Pr], [RC3014; H, H, Et, H _{, HCCCH 2, Bu], [} RC3015; H, H, Et, H, HCCCH 2, i-Bu], [RC3016; H, H, Et, H, HCCCH 2, t-Bu], [RC3017; H, H, Et, H, HCCCH ₂ , c-PrCH ₂ ], [RC3018; H, H, Et, H, HCCCH ₂ , Ph], [RC3019; H, H, Et, H, HCCCH ₂ , Bn], [ RC3020; H, H, Et, H, HCCCH ₂ , CF ₃ ], [RC3021; H, H, Et, H, HCCCH ₂ , CF ₃ CH ₂ ], [RC3022; H, H, Et, H, HCCCH ₂ , CF ₃ CF ₂ ], [RC3023; H, H, Et, H, HCCCH ₂ , CF ₂ H], [RC3024; H, H, Et, H, HCCCH ₂ , CF ₂ HCF ₂ ], [RC3025; H , H, Et, F, HCCCH ₂ , Me], [RC3026; H, H, Et, F, HCCCH ₂ , Et], [RC3027; H, H, Et, F, HCCCH ₂ , Pr], [RC3028; H, H, Et, F, HCCCH ₂ , i-Pr], [RC3029; H, H, Et, F, HCCCH ₂ , c-Pr], [RC3030; H, H, Et, F, HCCCH ₂ , Bu ], [R C3031; H, H, Et, F, HCCCH ₂ , i-Bu], [RC3032; H, H, Et, F, HCCCH ₂ , t-Bu], [RC3033; H, H, Et, F, HCCCH ₂ , c-PrCH ₂ ], [RC3034; H, H, Et, F, HCCCH ₂ , Ph], [RC3035; H, H, Et, F, HCCCH ₂ , Bn], [RC3036; H, H, Et, F, HCCCH ₂ , CF ₃ ], [RC3037; H, H, Et, F, HCCCH ₂ , CF ₃ CH ₂ ], [RC3038; H, H, Et, F, HCCCH ₂ , CF ₃ CF ₂ ], [ RC3039; H, H, Et, F, HCCCH ₂ , CF ₂ H], [RC3040; H, H, Et, F, HCCCH ₂ , CF ₂ HCF ₂ ], [RC3041; H, H, Et, Cl, HCCCH _{2, Me], [RC3042;} H, H, Et, Cl, HCCCH 2, Et], [RC3043; H, H, Et, Cl, HCCCH 2, Pr], [RC3044; H, H, Et, Cl, HCCCH ₂ , i-Pr], [RC3045; H, H, Et, Cl, HCCCH ₂ , c-Pr], [RC3046; H, H, Et, Cl, HCCCH ₂ , Bu], [RC3047; H, H , Et, Cl, HCCCH ₂ , i-Bu], [RC3048; H, H, Et, Cl, HCCCH ₂ , t-Bu], [RC3049; H, H, Et, Cl, HCCCH ₂ , c-PrCH ₂ ], [RC3050; H, H, Et, Cl, HCCCH ₂ , Ph], [RC3051; H, H, Et, Cl, HCCCH ₂ , Bn], [RC3052; H, H, Et, Cl, HCCCH ₂ , CF ₃ ], [RC3053; H, H, Et, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RC3054; H, H, Et, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RC3055; H, H , Et, Cl, HCCCH ₂ , CF ₂ H], [RC3056; H, H, Et, Cl, HCCCH ₂ , CF ₂ HCF ₂ ], [RC3057; H, H, F, H, HCCCH ₂ , Me], [RC3058; H, H, F, H, HCCCH ₂ , Et], [RC3059; H, H, F, H, HCCCH ₂ , Pr], [RC3060; H, H, F, H, HCCCH ₂ , i- Pr ], [RC3061; H, H, F, H, HCCCH ₂ , c-Pr], [RC3062; H, H, F, H, HCCCH ₂ , Bu], [RC3063; H, H, F, H, HCCCH ₂ , i-Bu], [RC3064; H, H, F, H, HCCCH ₂ , t-Bu], [RC3065; H, H, F, H, HCCCH ₂ , c-PrCH ₂ ], [RC3066; H , H, F, H, HCCCH ₂ , Ph], [RC3067; H, H, F, H, HCCCH ₂ , Bn], [RC3068; H, H, F, H, HCCCH ₂ , CF ₃ ], [RC3069 ; H, H, F, H, HCCCH ₂ , CF ₃ CH ₂ ], [RC3070; H, H, F, H, HCCCH ₂ , CF ₃ CF ₂ ], [RC3071; H, H, F, H, HCCCH ₂ , CF ₂ H], [RC3072; H, H, F, H, HCCCH ₂ , CF ₂ HCF ₂ ], [RC3073; H, H, F, F, HCCCH ₂ , Me], [RC3074; H, H , F, F, HCCCH ₂ , Et], [RC3075; H, H, F, F, HCCCH ₂ , Pr], [RC3076; H, H, F, F, HCCCH ₂ , i-Pr], [RC3077; H, H, F, F, HCCCH ₂ , c-Pr], [RC3078; H, H, F, F, HCCCH ₂ , Bu], [RC3079; H, H, F, F, HCCCH ₂ , i-Bu ], [RC3080; H, H, F, F, HCCCH ₂ , t-Bu], [RC3081; H, H, F, F, HCCCH ₂ , c-PrCH ₂ ], [RC3082; H, H, F, F, HCCCH ₂ , Ph], [RC3083; H, H, F, F, HCCCH ₂ , Bn], [RC3084; H, H, F, F, HCCCH ₂ , CF ₃ ], [RC3085; H, H, F, F, HCCCH ₂ , CF ₃ CH ₂ ], [RC3086; H, H, F, F, HCCCH ₂ , CF ₃ CF ₂ ], [RC3087; H, H, F, F, HCCCH ₂ , CF ₂ H ], [RC3088; H, H, F, F, HCCCH ₂ , CF ₂ HCF ₂ ], [RC3089; H, H, F, Cl, HCCCH ₂ , Me], [RC3090; H, H, F, Cl, HCCCH ₂ , Et], [RC3091; H, H, F, Cl, HCCCH ₂ , Pr], [RC3 092; H, H, F, Cl, HCCCH ₂ , i-Pr], [RC3093; H, H, F, Cl, HCCCH ₂ , c-Pr], [RC3094; H, H, F, Cl, HCCCH ₂ , Bu], [RC3095; H, H, F, Cl, HCCCH ₂ , i-Bu], [RC3096; H, H, F, Cl, HCCCH ₂ , t-Bu], [RC3097; H, H, F , Cl, HCCCH ₂ , c-PrCH ₂ ], [RC3098; H, H, F, Cl, HCCCH ₂ , Ph], [RC3099; H, H, F, Cl, HCCCH ₂ , Bn], [RC3100; H , H, F, Cl, HCCCH ₂ , CF ₃ ], [RC3101; H, H, F, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RC3102; H, H, F, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RC3103; H, H, F, Cl, HCCCH ₂ , CF ₂ H], [RC3104; H, H, F, Cl, HCCCH ₂ , CF ₂ HCF ₂ ], [RC3105; H, H, Cl, H, HCCCH ₂ , Me], [RC3106; H, H, Cl, H, HCCCH ₂ , Et], [RC3107; H, H, Cl, H, HCCCH ₂ , Pr], [RC3108; H, H , Cl, H, HCCCH ₂ , i-Pr], [RC3109; H, H, Cl, H, HCCCH ₂ , c-Pr], [RC3110; H, H, Cl, H, HCCCH ₂ , Bu], [ RC3111; H, H, Cl, H, HCCCH ₂ , i-Bu], [RC3112; H, H, Cl, H, HCCCH ₂ , t-Bu], [RC3113; H, H, Cl, H, HCCCH ₂ , c-PrCH ₂ ], [RC3114; H, H, Cl, H, HCCCH ₂ , Ph], [RC3115; H, H, Cl, H, HCCCH ₂ , Bn], [RC3116; H, H, Cl, H, HCCCH ₂ , CF ₃ ], [RC3117; H, H, Cl, H, HCCCH ₂ , CF ₃ CH ₂ ], [RC3118; H, H, Cl, H, HCCCH ₂ , CF ₃ CF ₂ ], [ RC3119; H, H, Cl, H, HCCCH ₂ , CF ₂ H], [RC3120; H, H, Cl, H, HCCCH ₂ , CF ₂ HCF ₂ ], [RC3121; H, H, Cl, Cl, HCCCH ₂ , Me], [RC3122; H , H, Cl, Cl, HCCCH ₂ , Et], [RC3123; H, H, Cl, Cl, HCCCH ₂ , Pr], [RC3124; H, H, Cl, Cl, HCCCH ₂ , i-Pr], [ RC3125; H, H, Cl, Cl, HCCCH ₂ , c-Pr], [RC3126; H, H, Cl, Cl, HCCCH ₂ , Bu], [RC3127; H, H, Cl, Cl, HCCCH ₂ , i -Bu], [RC3128; H, H, Cl, Cl, HCCCH ₂ , t-Bu], [RC3129; H, H, Cl, Cl, HCCCH ₂ , c-PrCH ₂ ], [RC3130; H, H, Cl, Cl, HCCCH ₂ , Ph], [RC3131; H, H, Cl, Cl, HCCCH ₂ , Bn], [RC3132; H, H, Cl, Cl, HCCCH ₂ , CF ₃ ], [RC3133; H, H, Cl, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RC3134; H, H, Cl, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RC3135; H, H, Cl, Cl, HCCCH ₂ , CF ₂ H], [RC3136; H, H, Cl, Cl, HCCCH ₂ , CF ₂ HCF ₂ ], [RC3137; H, H, H, H, CH ₃ CCCH ₂ , Me], [RC3138; H, H, H, H, CH ₃ CCCH ₂ , Et], [RC3139; H, H, H, H, CH ₃ CCCH ₂ , Pr], [RC3140; H, H, H, H, CH ₃ CCCH ₂ , i-Pr ], [RC3141; H, H, H, H, CH ₃ CCCH ₂ , c-Pr], [RC3142; H, H, H, H, CH ₃ CCCH ₂ , Bu], [RC3143; H, H, H , H, CH ₃ CCCH ₂ , i-Bu], [RC3144; H, H, H, H, CH ₃ CCCH ₂ , t-Bu], [RC3145; H, H, H, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC3146; H, H, H, H, CH ₃ CCCH ₂ , Ph], [RC3147; H, H, H, H, CH ₃ CCCH ₂ , Bn], [RC3148; H, H , H, H, CH ₃ CCCH ₂ , CF ₃ ], [RC3149; H, H, H, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC3150; H, H, H, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [ RC3151; H, H, H, H, CH ₃ CCCH ₂ , CF ₂ H], [RC3152; H, H, H, H, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC3153; H, H, H , Me, CH ₃ CCCH ₂ , Me], [RC3154; H, H, H, Me, CH ₃ CCCH ₂ , Et], [RC3155; H, H, H, Me, CH ₃ CCCH ₂ , Pr], [ RC3156; H, H, H, Me, CH ₃ CCCH ₂ , i-Pr], [RC3157; H, H, H, Me, CH ₃ CCCH ₂ , c-Pr], [RC3158; H, H, H, Me, CH ₃ CCCH ₂ , Bu], [RC3159; H, H, H, Me, CH ₃ CCCH ₂ , i-Bu], [RC3160; H, H, H, Me, CH ₃ CCCH ₂ , t-Bu ], [RC3161; H, H, H, Me, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC3162; H, H, H, Me, CH ₃ CCCH ₂ , Ph], [RC3163; H, H, H, Me, CH ₃ CCCH ₂ , Bn], [RC3164; H, H, H, Me, CH ₃ CCCH ₂ , CF ₃ ], [RC3165; H, H, H, Me, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC3166; H, H, H, Me, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC3167; H, H, H, Me, CH ₃ CCCH ₂ , CF ₂ H], [RC3168; H, H, H, Me, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC3169; H, H, Me, Me, CH ₃ CCCH ₂ , Me], [RC3170; H, H, Me, Me, CH ₃ CCCH ₂ , Et], [RC3171; H, H, Me, Me, CH ₃ CCCH ₂ , Pr], [RC3172; H, H, Me, Me, CH ₃ CCCH ₂ , i-Pr], [RC3173; H, H, Me, Me, CH ₃ CCCH ₂ , c-Pr], [RC3174; H, H, Me, Me, CH ₃ CCCH ₂ , Bu], [RC3175; H, H, Me, Me, CH ₃ CCCH ₂ , i-Bu], [RC3176; H, H, Me, Me, CH ₃ CCCH ₂ , t-Bu], [RC3177; H, H, Me, Me, CH ₃ CCCH ₂ , c-PrCH ₂ ] , [ RC3178; H, H, Me, Me, CH ₃ CCCH ₂ , Ph], [RC3179; H, H, Me, Me, CH ₃ CCCH ₂ , Bn], [RC3180; H, H, Me, Me, CH ₃ CCCH ₂ , CF ₃ ], [RC3181; H, H, Me, Me, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC3182; H, H, Me, Me, CH ₃ CCCH ₂ , CF ₃ CF ₂ ] , [RC3183; H, H, Me, Me, CH ₃ CCCH ₂ , CF ₂ H], [RC3184; H, H, Me, Me, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC3185; H, H , Me, Et, CH ₃ CCCH ₂ , Me], [RC3186; H, H, Me, Et, CH ₃ CCCH ₂ , Et], [RC3187; H, H, Me, Et, CH ₃ CCCH ₂ , Pr] , [RC3188; H, H, Me, Et, CH ₃ CCCH ₂ , i-Pr], [RC3189; H, H, Me, Et, CH ₃ CCCH ₂ , c-Pr], [RC3190; H, H, Me, Et, CH ₃ CCCH ₂ , Bu], [RC3191; H, H, Me, Et, CH ₃ CCCH ₂ , i-Bu], [RC3192; H, H, Me, Et, CH ₃ CCCH ₂ , t -Bu], [RC3193; H, H, Me, Et, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC3194; H, H, Me, Et, CH ₃ CCCH ₂ , Ph], [RC3195; H, H, Me, Et, CH ₃ CCCH ₂ , Bn], [RC3196; H, H, Me, Et, CH ₃ CCCH ₂ , CF ₃ ], [RC3197; H, H, Me, Et, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC3198; H, H, Me, Et, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC3199; H, H, Me, Et, CH ₃ CCCH ₂ , CF ₂ H], [ RC3200; H
, H, Me, Et, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ],

[RC3201; H, H, Me, F, CH ₃ CCCH ₂ , Me], [RC3202; H, H, Me, F, CH ₃ CCCH ₂ , Et], [RC3203; H, H, Me, F, CH ₃ CCCH ₂ , Pr], [RC3204; H, H, Me, F, CH ₃ CCCH ₂ , i-Pr], [RC3205; H, H, Me, F, CH ₃ CCCH ₂ , c-Pr], [ RC3206; H, H, Me, F, CH ₃ CCCH ₂ , Bu], [RC3207; H, H, Me, F, CH ₃ CCCH ₂ , i-Bu], [RC3208; H, H, Me, F, CH ₃ CCCH ₂ , t-Bu], [RC3209; H, H, Me, F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC3210; H, H, Me, F, CH ₃ CCCH ₂ , Ph] , [RC3211; H, H, Me, F, CH ₃ CCCH ₂ , Bn], [RC3212; H, H, Me, F, CH ₃ CCCH ₂ , CF ₃ ], [RC3213; H, H, Me, F , CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC3214; H, H, Me, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC3215; H, H, Me, F, CH ₃ CCCH ₂ , CF ₂ H], [RC3216; H, H, Me, F, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC3217; H, H, Me, Cl, CH ₃ CCCH ₂ , Me], [RC3218; H , H, Me, Cl, CH ₃ CCCH ₂ , Et], [RC3219; H, H, Me, Cl, CH ₃ CCCH ₂ , Pr], [RC3220; H, H, Me, Cl, CH ₃ CCCH ₂ , i-Pr], [RC3221; H, H, Me, Cl, CH ₃ CCCH ₂ , c-Pr], [RC3222; H, H, Me, Cl, CH ₃ CCCH ₂ , Bu], [RC3223; H, H, Me, Cl, CH ₃ CCCH ₂ , i-Bu], [RC3224; H, H, Me, Cl, CH ₃ CCCH ₂ , t-Bu], [RC3225; H, H, Me, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC3226; H, H, Me, Cl, CH ₃ CCCH ₂ , Ph], [RC3227; H, H, Me, Cl, CH ₃ CCCH ₂ , Bn], [RC3228; H , H, Me, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RC3229; H, H, Me, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC3230; H, H, Me, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC3231; H, H, Me, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RC3232; H, H, Me, Cl, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC3233; H, H, Et, H, CH ₃ CCCH ₂ , Me], [RC3234; H, H, Et, H, CH ₃ CCCH ₂ , Et], [RC3235; H, H, Et, H, CH ₃ CCCH ₂ , Pr], [RC3236; H, H, Et, H, CH ₃ CCCH ₂ , i-Pr], [RC3237; H, H, Et, H, CH ₃ CCCH ₂ , c-Pr ], [RC3238; H, H, Et, H, CH ₃ CCCH ₂ , Bu], [RC3239; H, H, Et, H, CH ₃ CCCH ₂ , i-Bu], [RC3240; H, H, Et , H, CH ₃ CCCH ₂ , t-Bu], [RC3241; H, H, Et, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC3242; H, H, Et, H, CH ₃ CCCH ₂ , Ph], [RC3243; H, H, Et, H, CH ₃ CCCH ₂ , Bn], [RC3244; H, H, Et, H, CH ₃ CCCH ₂ , CF ₃ ], [RC3245; H, H, Et, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC3246; H, H, Et, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC3247; H, H, Et, H, CH ₃ CCCH ₂ , CF ₂ H], [RC3248; H, H, Et, H, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC3249; H, H, Et, F, CH ₃ CCCH ₂ , Me], [ RC3250; H, H, Et, F, CH ₃ CCCH ₂ , Et], [RC3251; H, H, Et, F, CH ₃ CCCH ₂ , Pr], [RC3252; H, H, Et, F, CH ₃ CCCH ₂ , i-Pr], [RC3253; H, H, Et, F, CH ₃ CCCH ₂ , c-Pr], [RC3254; H, H, Et, F, CH ₃ CCCH ₂ , Bu], [RC 3255; H, H, Et, F, CH ₃ CCCH ₂ , i-Bu], [RC3256; H, H, Et, F, CH ₃ CCCH ₂ , t-Bu], [RC3257; H, H, Et, F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC3258; H, H, Et, F, CH ₃ CCCH ₂ , Ph], [RC3259; H, H, Et, F, CH ₃ CCCH ₂ , Bn] , [RC3260; H, H, Et, F, CH ₃ CCCH ₂ , CF ₃ ], [RC3261; H, H, Et, F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC3262; H, H, Et, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC3263; H, H, Et, F, CH ₃ CCCH ₂ , CF ₂ H], [RC3264; H, H, Et, F, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC3265; H, H, Et, Cl, CH ₃ CCCH ₂ , Me], [RC3266; H, H, Et, Cl, CH ₃ CCCH ₂ , Et], [RC3267; H , H, Et, Cl, CH ₃ CCCH ₂ , Pr], [RC3268; H, H, Et, Cl, CH ₃ CCCH ₂ , i-Pr], [RC3269; H, H, Et, Cl, CH ₃ CCCH ₂ , c-Pr], [RC3270; H, H, Et, Cl, CH ₃ CCCH ₂ , Bu], [RC3271; H, H, Et, Cl, CH ₃ CCCH ₂ , i-Bu], [RC3272; H, H, Et, Cl, CH ₃ CCCH ₂ , t-Bu], [RC3273; H, H, Et, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC3274; H, H, Et, Cl , CH ₃ CCCH ₂ , Ph], [RC3275; H, H, Et, Cl, CH ₃ CCCH ₂ , Bn], [RC3276; H, H, Et, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RC3277 ; H, H, Et, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC3278; H, H, Et, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC3279; H, H, Et , Cl, CH ₃ CCCH ₂ , CF ₂ H], [RC3280; H, H, Et, Cl, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC3281; H, H, F , H, CH ₃ CCCH ₂ , Me], [RC3282; H, H, F, H, CH ₃ CCCH ₂ , Et], [RC3283; H, H, F, H, CH ₃ CCCH ₂ , Pr], [ RC3284; H, H, F, H, CH ₃ CCCH ₂ , i-Pr], [RC3285; H, H, F, H, CH ₃ CCCH ₂ , c-Pr], [RC3286; H, H, F, H, CH ₃ CCCH ₂ , Bu], [RC3287; H, H, F, H, CH ₃ CCCH ₂ , i-Bu], [RC3288; H, H, F, H, CH ₃ CCCH ₂ , t-Bu ], [RC3289; H, H, F, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC3290; H, H, F, H, CH ₃ CCCH ₂ , Ph], [RC3291; H, H, F, H, CH ₃ CCCH ₂ , Bn], [RC3292; H, H, F, H, CH ₃ CCCH ₂ , CF ₃ ], [RC3293; H, H, F, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC3294; H, H, F, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC3295; H, H, F, H, CH ₃ CCCH ₂ , CF ₂ H], [RC3296; H, H, F, H, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC3297; H, H, F, F, CH ₃ CCCH ₂ , Me], [RC3298; H, H, F, F, CH ₃ CCCH ₂ , Et], [RC3299; H, H, F, F, CH ₃ CCCH ₂ , Pr], [RC3300; H, H, F, F, CH ₃ CCCH ₂ , i-Pr], [RC3301; H, H, F, F, CH ₃ CCCH ₂ , c-Pr], [RC3302; H, H, F, F, CH ₃ CCCH ₂ , Bu], [RC3303; H, H, F, F, CH ₃ CCCH ₂ , i-Bu], [RC3304; H, H, F, F, CH ₃ CCCH ₂ , t-Bu], [RC3305; H, H, F, F, CH ₃ CCCH ₂ , c-PrCH ₂ ] , [RC3306; H, H, F, F, CH ₃ CCCH ₂ , Ph], [RC3307; H, H, F, F, CH ₃ CCCH ₂ , Bn], [RC3308; H, H, F, F, CH ₃ CCCH ₂ , CF ₃ ], [RC3309; H, H, F, F, CH ₃ CCC H ₂ , CF ₃ CH ₂ ], [RC3310; H, H, F, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC3311; H, H, F, F, CH ₃ CCCH ₂ , CF ₂ H ], [RC3312; H, H, F, F, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC3313; H, H, F, Cl, CH ₃ CCCH ₂ , Me], [RC3314; H, H, F, Cl, CH ₃ CCCH ₂ , Et], [RC3315; H, H, F, Cl, CH ₃ CCCH ₂ , Pr], [RC3316; H, H, F, Cl, CH ₃ CCCH ₂ , i-Pr ], [RC3317; H, H, F, Cl, CH ₃ CCCH ₂ , c-Pr], [RC3318; H, H, F, Cl, CH ₃ CCCH ₂ , Bu], [RC3319; H, H, F , Cl, CH ₃ CCCH ₂ , i-Bu], [RC3320; H, H, F, Cl, CH ₃ CCCH ₂ , t-Bu], [RC3321; H, H, F, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC3322; H, H, F, Cl, CH ₃ CCCH ₂ , Ph], [RC3323; H, H, F, Cl, CH ₃ CCCH ₂ , Bn], [RC3324; H, H , F, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RC3325; H, H, F, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC3326; H, H, F, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC3327; H, H, F, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RC3328; H, H, F, Cl, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ] , [RC3329; H, H, Cl, H, CH ₃ CCCH ₂ , Me], [RC3330; H, H, Cl, H, CH ₃ CCCH ₂ , Et], [RC3331; H, H, Cl, H, CH ₃ CCCH ₂ , Pr], [RC3332; H, H, Cl, H, CH ₃ CCCH ₂ , i-Pr], [RC3333; H, H, Cl, H, CH ₃ CCCH ₂ , c-Pr], [RC3334; H, H, Cl, H, CH ₃ CCCH ₂ , Bu], [RC3335; H, H, Cl, H, CH ₃ CCCH ₂ , i-Bu], [RC3336; H, H, Cl, H , CH ₃ CCCH ₂ , t-Bu], [RC3337; H, H, Cl, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC3338; H, H, Cl, H, CH ₃ CCCH ₂ , Ph], [RC3339; H, H, Cl, H, CH ₃ CCCH ₂ , Bn], [RC3340; H, H, Cl, H, CH ₃ CCCH ₂ , CF ₃ ], [RC3341; H, H, Cl, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC3342; H, H, Cl, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC3343; H, H, Cl, H, CH ₃ CCCH ₂ , CF ₂ H] , [RC3344; H, H, Cl, H, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC3345; H, H, Cl, Cl, CH ₃ CCCH ₂ , Me], [RC3346; H, H, Cl , Cl, CH ₃ CCCH ₂ , Et], [RC3347; H, H, Cl, Cl, CH ₃ CCCH ₂ , Pr], [RC3348; H, H, Cl, Cl, CH ₃ CCCH ₂ , i-Pr] , [RC3349; H, H, Cl, Cl, CH ₃ CCCH ₂ , c-Pr], [RC3350; H, H, Cl, Cl, CH ₃ CCCH ₂ , Bu], [RC3351; H, H, Cl, Cl, CH ₃ CCCH ₂ , i-Bu], [RC3352; H, H, Cl, Cl, CH ₃ CCCH ₂ , t-Bu], [RC3353; H, H, Cl, Cl, CH ₃ CCCH ₂ , c -PrCH ₂ ], [RC3354; H, H, Cl, Cl, CH ₃ CCCH ₂ , Ph], [RC3355; H, H, Cl, Cl, CH ₃ CCCH ₂ , Bn], [RC3356; H, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RC3357; H, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC3358; H, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC3359; H, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RC3360; H, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC3361; H, H, H, H, c-Pr, Me], [RC3362; H, H, H, H, c-Pr, Et], [RC3363; H, H, H, H, c-Pr , Pr] , [RC3364; H, H, H, H, c-Pr, i-Pr], [RC3365; H, H, H, H, c-Pr, c-Pr], [RC3366; H, H, H, H, c-Pr, Bu], [RC3367; H, H, H, H, c-Pr, i-Bu], [RC3368; H, H, H, H, c-Pr, t-Bu], [ RC3369; H, H, H, H, c-Pr, c-PrCH ₂ ], [RC3370; H, H, H, H, c-Pr, Ph], [RC3371; H, H, H, H, c -Pr, Bn], [RC3372; H, H, H, H, c-Pr, CF ₃ ], [RC3373; H, H, H, H, c-Pr, CF ₃ CH ₂ ], [RC3374; H , H, H, H, c-Pr, CF ₃ CF ₂ ], [RC3375; H, H, H, H, c-Pr, CF ₂ H], [RC3376; H, H, H, H, c- Pr, CF ₂ HCF ₂ ], [RC3377; H, H, H, Me, c-Pr, Me], [RC3378; H, H, H, Me, c-Pr, Et], [RC3379; H, H , H, Me, c-Pr, Pr], [RC3380; H, H, H, Me, c-
Pr, i-Pr], [RC3381; H, H, H, Me, c-Pr, c-Pr], [RC3382; H, H, H, Me, c-Pr, Bu], [RC3383; H, H, H, Me, c-Pr, i-Bu], [RC3384; H, H, H, Me, c-Pr, t-Bu], [RC3385; H, H, H, Me, c-Pr, c-PrCH ₂ ], [RC3386; H, H, H, Me, c-Pr, Ph], [RC3387; H, H, H, Me, c-Pr, Bn], [RC3388; H, H, H , Me, c-Pr, CF ₃ ], [RC3389; H, H, H, Me, c-Pr, CF ₃ CH ₂ ], [RC3390; H, H, H, Me, c-Pr, CF ₃ CF ₂ ], [RC3391; H, H, H, Me, c-Pr, CF ₂ H], [RC3392; H, H, H, Me, c-Pr, CF ₂ HCF ₂ ], [RC3393; H, H , Me, Me, c-Pr, Me], [RC3394; H, H, Me, Me, c-Pr, Et], [RC3395; H, H, Me, Me, c-Pr, Pr], [RC3396 ; H, H, Me, Me, c-Pr, i-Pr], [RC3397; H, H, Me, Me, c-Pr, c-Pr], [RC3398; H, H, Me, Me, c -Pr, Bu], [RC3399; H, H, Me, Me, c-Pr, i-Bu], [RC3400; H, H, Me, Me, c-Pr, t-Bu],

[RC3401; H, H, Me, Me, c-Pr, c-PrCH ₂ ], [RC3402; H, H, Me, Me, c-Pr, Ph], [RC3403; H, H, Me, Me, c-Pr, Bn], [RC3404; H, H, Me, Me, c-Pr, CF ₃ ], [RC3405; H, H, Me, Me, c-Pr, CF ₃ CH ₂ ], [RC3406; H, H, Me, Me, c-Pr, CF ₃ CF ₂ ], [RC3407; H, H, Me, Me, c-Pr, CF ₂ H], [RC3408; H, H, Me, Me, c -Pr, CF ₂ HCF ₂ ], [RC3409; H, H, Me, Et, c-Pr, Me], [RC3410; H, H, Me, Et, c-Pr, Et], [RC3411; H, H, Me, Et, c-Pr, Pr], [RC3412; H, H, Me, Et, c-Pr, i-Pr], [RC3413; H, H, Me, Et, c-Pr, c- Pr], [RC3414; H, H, Me, Et, c-Pr, Bu], [RC3415; H, H, Me, Et, c-Pr, i-Bu], [RC3416; H, H, Me, Et, c-Pr, t-Bu], [RC3417; H, H, Me, Et, c-Pr, c-PrCH ₂ ], [RC3418; H, H, Me, Et, c-Pr, Ph], [RC3419; H, H, Me, Et, c-Pr, Bn], [RC3420; H, H, Me, Et, c-Pr, CF ₃ ], [RC3421; H, H, Me, Et, c- Pr, CF ₃ CH ₂ ], [RC3422; H, H, Me, Et, c-Pr, CF ₃ CF ₂ ], [RC3423; H, H, Me, Et, c-Pr, CF ₂ H], [ RC3424; H, H, Me, Et, c-Pr, CF ₂ HCF ₂ ], [RC3425; H, H, Me, F, c-Pr, Me], [RC3426; H, H, Me, F, c -Pr, Et], [RC3427; H, H, Me, F, c-Pr, Pr], [RC3428; H, H, Me, F, c-Pr, i-Pr], [RC3429; H, H , Me, F, c-Pr, c-Pr], [RC3430; H, H, Me, F, c-Pr, Bu], [RC3431; H, H, Me, F, c-Pr, i-Bu ], [RC3432; H, H, Me, F, c-Pr, t-Bu], [RC3433; H, H, Me, F, c-Pr, c-PrCH ₂ ], [RC3434; H, H, Me, F, c-Pr, Ph], [RC3435; H, H, Me, F, c-Pr, Bn], [RC3436; H, H, Me, F, c-Pr, CF ₃ ], [RC3437; H, H , Me, F, c-Pr, CF ₃ CH ₂ ], [RC3438; H, H, Me, F, c-Pr, CF ₃ CF ₂ ], [RC3439; H, H, Me, F, c-Pr , CF ₂ H], [RC3440; H, H, Me, F, c-Pr, CF ₂ HCF ₂ ], [RC3441; H, H, Me, Cl, c-Pr, Me], [RC3442; H, H, Me, Cl, c-Pr, Et], [RC3443; H, H, Me, Cl, c-Pr, Pr], [RC3444; H, H, Me, Cl, c-Pr, i-Pr] , [RC3445; H, H, Me, Cl, c-Pr, c-Pr], [RC3446; H, H, Me, Cl, c-Pr, Bu], [RC3447; H, H, Me, Cl, c-Pr, i-Bu], [RC3448; H, H, Me, Cl, c-Pr, t-Bu], [RC3449; H, H, Me, Cl, c-Pr, c-PrCH ₂ ], [RC3450; H, H, Me, Cl, c-Pr, Ph], [RC3451; H, H, Me, Cl, c-Pr, Bn], [RC3452; H, H, Me, Cl, c-Pr , CF ₃ ], [RC3453; H, H, Me, Cl, c-Pr, CF ₃ CH ₂ ], [RC3454; H, H, Me, Cl, c-Pr, CF ₃ CF ₂ ], [RC3455; H, H, Me, Cl, c-Pr, CF ₂ H], [RC3456; H, H, Me, Cl, c-Pr, CF ₂ HCF ₂ ], [RC3457; H, H, Et, H, c -Pr, Me], [RC3458; H, H, Et, H, c-Pr, Et], [RC3459; H, H, Et, H, c-Pr, Pr], [RC3460; H, H, Et , H, c-Pr, i-Pr], [RC3461; H, H, Et, H, c-Pr, c-Pr], [RC3462; H, H, Et, H, c-Pr, Bu], [RC3463; H, H, Et, H, c-Pr, i-Bu], [RC3464; H, H, Et, H, c-Pr, t-Bu], [RC3465; H, H, Et, H , c-Pr, c-PrCH ₂ ], [RC3466; H, H, Et, H, c-Pr, Ph], [RC3467; H, H, Et, H, c-Pr, Bn], [RC3468; H, H, Et, H, c-Pr, C F ₃ ], [RC3469; H, H, Et, H, c-Pr, CF ₃ CH ₂ ], [RC3470; H, H, Et, H, c-Pr, CF ₃ CF ₂ ], [RC3471; H , H, Et, H, c-Pr, CF ₂ H], [RC3472; H, H, Et, H, c-Pr, CF ₂ HCF ₂ ], [RC3473; H, H, Et, F, c- Pr, Me], [RC3474; H, H, Et, F, c-Pr, Et], [RC3475; H, H, Et, F, c-Pr, Pr], [RC3476; H, H, Et, F, c-Pr, i-Pr], [RC3477; H, H, Et, F, c-Pr, c-Pr], [RC3478; H, H, Et, F, c-Pr, Bu], [ RC3479; H, H, Et, F, c-Pr, i-Bu], [RC3480; H, H, Et, F, c-Pr, t-Bu], [RC3481; H, H, Et, F, c-Pr, c-PrCH ₂ ], [RC3482; H, H, Et, F, c-Pr, Ph], [RC3483; H, H, Et, F, c-Pr, Bn], [RC3484; H , H, Et, F, c-Pr, CF ₃ ], [RC3485; H, H, Et, F, c-Pr, CF ₃ CH ₂ ], [RC3486; H, H, Et, F, c-Pr , CF ₃ CF ₂ ], [RC3487; H, H, Et, F, c-Pr, CF ₂ H], [RC3488; H, H, Et, F, c-Pr, CF ₂ HCF ₂ ], [RC3489 ; H, H, Et, Cl, c-Pr, Me], [RC3490; H, H, Et, Cl, c-Pr, Et], [RC3491; H, H, Et, Cl, c-Pr, Pr ], [RC3492; H, H, Et, Cl, c-Pr, i-Pr], [RC3493; H, H, Et, Cl, c-Pr, c-Pr], [RC3494; H, H, Et , Cl, c-Pr, Bu], [RC3495; H, H, Et, Cl, c-Pr, i-Bu], [RC3496; H, H, Et, Cl, c-Pr, t-Bu], [RC3497; H, H, Et, Cl, c-Pr, c-PrCH ₂ ], [RC3498; H, H, Et, Cl, c-Pr, Ph], [RC3499; H, H, Et, Cl, c-Pr, Bn], [RC3500; H, H, Et, Cl, c-Pr, CF ₃ ], [RC3501; H, H, Et, Cl, c-Pr, CF ₃ CH ₂ ], [RC3502; H, H, Et, Cl, cP r, CF ₃ CF ₂ ], [RC3503; H, H, Et, Cl, c-Pr, CF ₂ H], [RC3504; H, H, Et, Cl, c-Pr, CF ₂ HCF ₂ ], [ RC3505; H, H, F, H, c-Pr, Me], [RC3506; H, H, F, H, c-Pr, Et], [RC3507; H, H, F, H, c-Pr, Pr], [RC3508; H, H, F, H, c-Pr, i-Pr], [RC3509; H, H, F, H, c-Pr, c-Pr], [RC3510; H, H, F, H, c-Pr, Bu], [RC3511; H, H, F, H, c-Pr, i-Bu], [RC3512; H, H, F, H, c-Pr, t-Bu] , [RC3513; H, H, F, H, c-Pr, c-PrCH ₂ ], [RC3514; H, H, F, H, c-Pr, Ph], [RC3515; H, H, F, H , c-Pr, Bn], [RC3516; H, H, F, H, c-Pr, CF ₃ ], [RC3517; H, H, F, H, c-Pr, CF ₃ CH ₂ ], [RC3518 ; H, H, F, H, c-Pr, CF ₃ CF ₂ ], [RC3519; H, H, F, H, c-Pr, CF ₂ H], [RC3520; H, H, F, H, c-Pr, CF ₂ HCF ₂ ], [RC3521; H, H, F, F, c-Pr, Me], [RC3522; H, H, F, F, c-Pr, Et], [RC3523; H , H, F, F, c-Pr, Pr], [RC3524; H, H, F, F, c-Pr, i-Pr], [RC3525; H, H, F, F, c-Pr, c -Pr], [RC3526; H, H, F, F, c-Pr, Bu], [RC3527; H, H, F, F, c-Pr, i-Bu], [RC3528; H, H, F , F, c-Pr, t-Bu], [RC3529; H, H, F, F, c-Pr, c-PrCH ₂ ], [RC3530; H, H, F, F, c-Pr, Ph] , [RC3531; H, H, F, F, c-Pr, Bn], [RC3532; H, H, F, F, c-Pr, CF ₃ ], [RC3533; H, H, F, F, c -Pr, CF ₃ CH ₂ ], [RC3534; H, H, F, F, c-Pr, CF ₃ CF ₂ ], [RC3535; H, H, F, F, c-Pr, CF ₂ H], [RC3536; H, H, F, F, c-Pr, CF ₂ HCF ₂ ], [RC3537; H, H, F, Cl, c-Pr, Me] , [RC3538; H, H, F, Cl, c-Pr, Et], [RC3539; H, H, F, Cl, c-Pr, Pr], [RC3540; H, H, F, Cl, c- Pr, i-Pr], [RC3541; H, H, F, Cl, c-Pr, c-Pr], [RC3542; H, H, F, Cl, c-Pr, Bu], [RC3543; H, H, F, Cl, c-Pr, i-Bu], [RC3544; H, H, F, Cl, c-Pr, t-Bu], [RC3545; H, H, F, Cl, c-Pr, c-PrCH ₂ ], [RC3546; H, H, F, Cl, c-Pr, Ph], [RC3547; H, H, F, Cl, c-Pr, Bn], [RC3548; H, H, F , Cl, c-Pr, CF ₃ ], [RC3549; H, H, F, Cl, c-Pr, CF ₃ CH ₂ ], [RC3550; H, H, F, Cl, c-Pr, CF ₃ CF ₂ ], [RC3551; H, H, F, Cl, c-Pr, CF ₂ H], [RC3552; H, H, F, Cl, c-Pr, CF ₂ HCF ₂ ], [RC3553; H, H , Cl, H, c-Pr, Me], [RC3554; H, H, Cl, H, c-Pr, Et], [RC3555; H, H, Cl, H, c-Pr, Pr], [RC3556 ; H, H, Cl, H, c-Pr, i-Pr], [RC3557; H, H, Cl, H, c-Pr, c-Pr], [RC3558; H, H, Cl, H, c -Pr, Bu], [RC3559; H, H, Cl, H, c-Pr, i-Bu], [RC3560; H, H, Cl, H, c-Pr, t-Bu], [RC3561; H , H, Cl, H, c-Pr, c-PrCH ₂ ], [RC3562; H, H, Cl, H, c-Pr, Ph], [RC3563; H, H, Cl, H, c-Pr, Bn], [RC3564; H, H, Cl, H, c-Pr, CF ₃ ], [RC3565; H, H, Cl, H, c-Pr, CF ₃ CH ₂ ], [RC3566; H, H, Cl, H, c-Pr, CF ₃ CF ₂ ], [RC3567; H, H, Cl, H, c-Pr, CF ₂ H], [RC3568; H, H, Cl, H, c-Pr, CF ₂ HCF ₂ ], [RC3569; H, H, Cl, Cl, c-Pr, Me], [RC3570; H, H, Cl, Cl, c-Pr, Et], [RC3571; H, H, Cl, Cl, c-Pr, Pr], [RC3572; H, H, Cl, Cl, c-Pr, i-Pr], [RC3573; H, H, Cl, Cl, c-Pr, c-Pr], [RC3574; H, H, Cl, Cl, c-Pr, Bu], [RC3575; H, H, Cl, Cl, c-Pr, i-Bu], [RC3576; H, H, Cl, Cl, c-Pr, t-Bu], [RC3577; H, H, Cl, Cl, c- Pr, c-PrCH ₂ ], [RC3578; H, H, Cl, Cl, c-Pr, Ph], [RC3579; H, H, Cl, Cl, c-Pr, Bn], [RC3580; H, H , Cl, Cl, c-Pr, CF ₃ ], [RC3581; H, H, Cl, Cl, c-Pr, CF ₃ CH ₂ ], [RC3582; H, H, Cl, Cl, c-Pr, CF ₃ CF ₂ ], [RC3583; H, H, Cl, Cl, c-Pr, CF ₂ H], [RC3584; H, H, Cl, Cl, c-Pr, CF ₂ HCF ₂ ], [RC3585; H , H, H, H, Bn, Me], [RC3586; H, H, H, H, Bn, Et], [RC3587; H, H, H, H, Bn, Pr], [RC3588; H, H , H, H, Bn, i-Pr], [RC3589; H, H, H, H, Bn, c-Pr], [RC3590; H, H, H, H, Bn, Bu], [RC3591; H , H, H, H, Bn, i-Bu], [RC3592; H, H, H, H, Bn, t-Bu], [RC3593; H, H, H, H, Bn, c-PrCH ₂ ] , [RC3594; H, H, H, H, Bn, Ph], [RC3595; H, H, H, H, Bn, Bn], [RC3596; H, H, H, H, Bn, CF ₃ ], [RC3597; H, H, H, H, Bn, CF ₃ CH ₂ ], [RC3598; H, H, H, H, Bn, CF ₃ CF ₂ ], [RC3599; H, H, H, H, Bn , CF ₂ H], [RC3600; H, H, H, H, Bn, CF ₂ HCF ₂ ],

[RC3601; H, H, H, Me, Bn, Me], [RC3602; H, H, H, Me, Bn, Et], [RC3603; H, H, H, Me, Bn, Pr], [RC3604 ; H, H, H, Me, Bn, i-Pr], [RC3605; H, H, H, Me, Bn, c-Pr], [RC3606; H, H, H, Me, Bn, Bu], [RC3607; H, H, H, Me, Bn, i-Bu], [RC3608; H, H, H, Me, Bn, t-Bu], [RC3609; H, H, H, Me, Bn, c -PrCH ₂ ], [RC3610; H, H, H, Me, Bn, Ph], [RC3611; H, H, H, Me, Bn, Bn], [RC3612; H, H, H, Me, Bn, CF ₃ ], [RC3613; H, H, H, Me, Bn, CF ₃ CH ₂ ], [RC3614; H, H, H, Me, Bn, CF ₃ CF ₂ ], [RC3615; H, H, H , Me, Bn, CF ₂ H], [RC3616; H, H, H, Me, Bn, CF ₂ HCF ₂ ], [RC3617; H, H, Me, Me, Bn, Me], [RC3618; H, H, Me, Me, Bn, Et], [RC3619; H, H, Me, Me, Bn, Pr], [RC3620; H, H, Me, Me, Bn, i-Pr], [RC3621; H, H, Me, Me, Bn, c-Pr], [RC3622; H, H, Me, Me, Bn, Bu], [RC3623; H, H, Me, Me, Bn, i-Bu], [RC3624; H, H, Me, Me, Bn, t-Bu], [RC3625; H, H, Me, Me, Bn, c-PrCH ₂ ], [RC3626; H, H, Me, Me, Bn, Ph], [RC3627; H, H, Me, Me, Bn, Bn], [RC3628; H, H, Me, Me, Bn, CF ₃ ], [RC3629; H, H, Me, Me, Bn, CF ₃ CH ₂ ], [RC3630; H, H, Me, Me, Bn, CF ₃ CF ₂ ], [RC3631; H, H, Me, Me, Bn, CF ₂ H], [RC3632; H, H, Me, Me, Bn, CF ₂ HCF ₂ ], [RC3633; H, H, Me, Et, Bn, Me], [RC3634; H, H, Me, Et, Bn, Et], [RC3635; H, H, Me, Et , Bn, Pr], [RC3636; H, H, Me, Et, Bn, i-Pr], [RC3637; H, H, Me, Et, Bn , c-Pr], [RC3638; H, H, Me, Et, Bn, Bu], [RC3639; H, H, Me, Et, Bn, i-Bu], [RC3640; H, H, Me, Et , Bn, t-Bu], [RC3641; H, H, Me, Et, Bn, c-PrCH ₂ ], [RC3642; H, H, Me, Et, Bn, Ph], [RC3643; H, H, Me, Et, Bn, Bn], [RC3644; H, H, Me, Et, Bn, CF ₃ ], [RC3645; H, H, Me, Et, Bn, CF ₃ CH ₂ ], [RC3646; H, H, Me, Et, Bn, CF ₃ CF ₂ ], [RC3647; H, H, Me, Et, Bn, CF ₂ H], [RC3648; H, H, Me, Et, Bn, CF ₂ HCF ₂ ] , [RC3649; H, H, Me, F, Bn, Me], [RC3650; H, H, Me, F, Bn, Et], [RC3651; H, H, Me, F, Bn, Pr], [ RC3652; H, H, Me, F, Bn, i-Pr], [RC3653; H, H, Me, F, Bn, c-Pr], [RC3654; H, H, Me, F, Bn, Bu] , [RC3655; H, H, Me, F, Bn, i-Bu], [RC3656; H, H, Me, F, Bn, t-Bu], [RC3657; H, H, Me, F, Bn, c-PrCH ₂ ], [RC3658; H, H, Me, F, Bn, Ph], [RC3659; H, H, Me, F, Bn, Bn], [RC3660; H, H, Me, F, Bn , CF ₃ ], [RC3661; H, H, Me, F, Bn, CF ₃ CH ₂ ], [RC3662; H, H, Me, F, Bn, CF ₃ CF ₂ ], [RC3663; H, H, Me, F, Bn, CF ₂ H], [RC3664; H, H, Me, F, Bn, CF ₂ HCF ₂ ], [RC3665; H, H, Me, Cl, Bn, Me], [RC3666; H , H, Me, Cl, Bn, Et], [RC3667; H, H, Me, Cl, Bn, Pr], [RC3668; H, H, Me, Cl, Bn, i-Pr], [RC3669; H , H, Me, Cl, Bn, c-Pr], [RC3670; H, H, Me, Cl, Bn, Bu], [RC3671; H, H, Me, Cl, Bn, i-Bu], [RC3672 ; H, H, Me, Cl, Bn, t-Bu], [RC3673; H, H, Me, Cl, Bn, c-PrCH ₂ ], [RC3 674; H, H, Me, Cl, Bn, Ph], [RC3675; H, H, Me, Cl, Bn, Bn], [RC3676; H, H, Me, Cl, Bn, CF ₃ ], [RC3677 ; H, H, Me, Cl, Bn, CF ₃ CH ₂ ], [RC3678; H, H, Me, Cl, Bn, CF ₃ CF ₂ ], [RC3679; H, H, Me, Cl, Bn, CF ₂ H], [RC3680; H, H, Me, Cl, Bn, CF ₂ HCF ₂ ], [RC3681; H, H, Et, H, Bn, Me], [RC3682; H, H, Et, H, Bn, Et], [RC3683; H, H, Et, H, Bn, Pr], [RC3684; H, H, Et, H, Bn, i-Pr], [RC3685; H, H, Et, H, Bn, c-Pr], [RC3686; H, H, Et, H, Bn, Bu], [RC3687; H, H, Et, H, Bn, i-Bu], [RC3688; H, H, Et, H, Bn, t-Bu], [RC3689; H, H, Et, H, Bn, c-PrCH ₂ ], [RC3690; H, H, Et, H, Bn, Ph], [RC3691; H, H , Et, H, Bn, Bn], [RC3692; H, H, Et, H, Bn, CF ₃ ], [RC3693; H, H, Et, H, Bn, CF ₃ CH ₂ ], [RC3694; H , H, Et, H, Bn, CF ₃ CF ₂ ], [RC3695; H, H, Et, H, Bn, CF ₂ H], [RC3696; H, H, Et, H, Bn, CF ₂ HCF ₂ ], [RC3697; H, H, Et, F, Bn, Me], [RC3698; H, H, Et, F, Bn, Et], [RC3699; H, H, Et, F, Bn, Pr], [RC3700; H, H, Et, F, Bn, i-Pr], [RC3701; H, H, Et, F, Bn, c-Pr], [RC3702; H, H, Et, F, Bn, Bu ], [RC3703; H, H, Et, F, Bn, i-Bu], [RC3704; H, H, Et, F, Bn, t-Bu], [RC3705; H, H, Et, F, Bn , c-PrCH ₂ ], [RC3706; H, H, Et, F, Bn, Ph], [RC3707; H, H, Et, F, Bn, Bn], [RC3708; H, H, Et, F, Bn, CF ₃ ], [RC3709; H, H, Et, F, Bn, CF ₃ CH ₂ ], [RC3710; H, H, Et, F, Bn, CF ₃ CF ₂ ], [RC3711; H, H, Et, F, Bn, CF ₂ H], [RC3712; H, H, Et, F, Bn, CF ₂ HCF ₂ ], [RC3713; H, H, Et, Cl , Bn, Me], [RC3714; H, H, Et, Cl, Bn, Et], [RC3715; H, H, Et, Cl, Bn, Pr], [RC3716; H, H, Et, Cl, Bn , i-Pr], [RC3717; H, H, Et, Cl, Bn, c-Pr], [RC3718; H, H, Et, Cl, Bn, Bu], [RC3719; H, H, Et, Cl , Bn, i-Bu], [RC3720; H, H, Et, Cl, Bn, t-Bu], [RC3721; H, H, Et, Cl, Bn, c-PrCH ₂ ], [RC3722; H, H, Et, Cl, Bn, Ph], [RC3723; H, H, Et, Cl, Bn, Bn], [RC3724; H, H, Et, Cl, Bn, CF ₃ ], [RC3725; H, H , Et, Cl, Bn, CF ₃ CH ₂ ], [RC3726; H, H, Et, Cl, Bn, CF ₃ CF ₂ ], [RC3727; H, H, Et, Cl, Bn, CF ₂ H], [RC3728; H, H, Et, Cl, Bn, CF ₂ HCF ₂ ], [RC3729; H, H, F, H, Bn, Me], [RC3730; H, H, F, H, Bn, Et] , [RC3731; H, H, F, H, Bn, Pr], [RC3732; H, H, F, H, Bn, i-Pr], [RC3733; H, H, F, H, Bn, c- Pr], [RC3734; H, H, F, H, Bn, Bu], [RC3735; H, H, F, H, Bn, i-Bu], [RC3736; H, H, F, H, Bn, t-Bu], [RC3737; H, H, F, H, Bn, c-PrCH ₂ ], [RC3738; H, H, F, H, Bn, Ph], [RC3739; H, H, F, H , Bn, Bn], [RC3740; H, H, F, H, Bn, CF ₃ ], [RC3741; H, H, F, H, Bn, CF ₃ CH ₂ ], [RC3742; H, H, F , H, Bn, CF ₃ CF ₂ ], [RC3743; H, H, F, H, Bn, CF ₂ H], [RC3744; H, H, F, H, Bn, CF ₂ HCF ₂ ], [RC3745 ; H, H, F, F, Bn, Me], [RC3746; H, H, F, F, Bn, Et], [RC3747; H, H, F, F, Bn, Pr], [RC3 748; H, H, F, F, Bn, i-Pr], [RC3749; H, H, F, F, Bn, c-Pr], [RC3750; H, H, F, F, Bn, Bu] , [RC3751; H, H, F, F, Bn, i-Bu], [RC3752; H, H, F, F, Bn, t-Bu], [RC3753; H, H, F, F, Bn, c-PrCH ₂ ], [RC3754; H, H, F, F, Bn, Ph], [RC3755; H, H, F, F, Bn, Bn], [RC3756; H, H, F, F, Bn , CF ₃ ], [RC3757; H, H, F, F, Bn, CF ₃ CH ₂ ], [RC3758; H, H, F, F, Bn, CF ₃ CF ₂ ], [RC3759; H, H, F, F, Bn, CF ₂ H], [RC3760; H, H, F, F, Bn, CF ₂ HCF ₂ ], [RC3761; H, H, F, Cl, Bn, Me], [RC3762; H , H, F, Cl, Bn, Et], [RC3763; H, H, F, Cl, Bn, Pr], [RC3764; H, H, F, Cl, Bn, i-Pr], [RC3765; H , H, F, Cl, Bn, c-Pr], [RC3766; H, H, F, Cl, Bn, Bu], [RC3767; H, H, F, Cl, Bn, i-Bu], [RC3768 ; H, H, F, Cl, Bn, t-Bu], [RC3769; H, H, F, Cl, Bn, c-PrCH ₂ ], [RC3770; H, H, F, Cl, Bn, Ph] , [RC3771; H, H, F, Cl, Bn, Bn], [RC3772; H, H, F, Cl, Bn, CF ₃ ], [RC3773; H, H, F, Cl, Bn, CF ₃ CH ₂ ], [RC3774; H, H, F, Cl, Bn, CF ₃ CF ₂ ], [RC3775; H, H, F, Cl, Bn, CF ₂ H], [RC3776; H, H, F, Cl , Bn, CF ₂ HCF ₂ ], [RC3777; H, H, Cl, H, Bn, Me], [RC3778; H, H, Cl, H, Bn, Et], [RC3779; H, H, Cl, H, Bn, Pr], [RC3780; H, H, Cl, H, Bn, i-Pr], [RC3781; H, H, Cl, H, Bn, c-Pr], [RC3782; H, H, Cl, H, Bn, Bu], [RC3783; H, H, Cl, H, Bn, i-Bu], [RC3784; H, H, Cl, H, Bn, t-Bu], [RC3785; H, H, Cl, H, Bn, c-PrCH ₂ ], [RC3786; H, H, Cl, H, Bn, Ph], [RC3787; H, H, Cl, H, Bn, Bn], [RC3788; H, H, Cl, H, Bn, CF ₃ ], [RC3789; H, H, Cl, H, Bn, CF ₃ CH ₂ ], [RC3790; H, H, Cl, H, Bn, CF ₃ CF ₂ ], [RC3791; H, H, Cl, H , Bn, CF ₂ H], [RC3792; H, H, Cl, H, Bn, CF ₂ HCF ₂ ], [RC3793; H, H, Cl, Cl, Bn, Me], [RC3794; H, H, Cl, Cl, Bn, Et], [RC3795; H, H, Cl, Cl, Bn, Pr], [RC3796; H, H, Cl, Cl, Bn, i-Pr], [RC3797; H, H, Cl, Cl, Bn, c-Pr], [RC3798; H, H, Cl, Cl, Bn, Bu], [RC3799; H, H, Cl, Cl, Bn, i-Bu], [RC3800; H, H, Cl, Cl, Bn, t-Bu],

[RC3801; H, H, Cl, Cl, Bn, c-PrCH ₂ ], [RC3802; H, H, Cl, Cl, Bn, Ph], [RC3803; H, H, Cl, Cl, Bn, Bn] , [RC3804; H, H, Cl, Cl, Bn, CF ₃ ], [RC3805; H, H, Cl, Cl, Bn, CF ₃ CH ₂ ], [RC3806; H, H, Cl, Cl, Bn, CF ₃ CF ₂ ], [RC3807; H, H, Cl, Cl, Bn, CF ₂ H], [RC3808; H, H, Cl, Cl, Bn, CF ₂ HCF ₂ ], [RC3809; H, H, H, H, Ph, Me], [RC3810; H, H, H, H, Ph, Et], [RC3811; H, H, H, H, Ph, Pr], [RC3812; H, H, H, H, Ph, i-Pr], [RC3813; H, H, H, H, Ph, c-Pr], [RC3814; H, H, H, H, Ph, Bu], [RC3815; H, H, H, H, Ph, i-Bu], [RC3816; H, H, H, H, Ph, t-Bu], [RC3817; H, H, H, H, Ph, c-PrCH ₂ ], [RC3818 ; H, H, H, H, Ph, Ph], [RC3819; H, H, H, H, Ph, Bn], [RC3820; H, H, H, H, Ph, CF ₃ ], [RC3821; H, H, H, H, Ph, CF ₃ CH ₂ ], [RC3822; H, H, H, H, Ph, CF ₃ CF ₂ ], [RC3823; H, H, H, H, Ph, CF ₂ H], [RC3824; H, H, H, H, Ph, CF ₂ HCF ₂ ], [RC3825; H, H, H, Me, Ph, Me], [RC3826; H, H, H, Me, Ph , Et], [RC3827; H, H, H, Me, Ph, Pr], [RC3828; H, H, H, Me, Ph, i-Pr], [RC3829; H, H, H, Me, Ph , c-Pr], [RC3830; H, H, H, Me, Ph, Bu], [RC3831; H, H, H, Me, Ph, i-Bu], [RC3832; H, H, H, Me , Ph, t-Bu], [RC3833; H, H, H, Me, Ph, c-PrCH ₂ ], [RC3834; H, H, H, Me, Ph, Ph], [RC3835; H, H, H, Me, Ph, Bn], [RC3836; H, H, H, Me, Ph, CF ₃ ], [RC3837; H, H, H, Me, Ph, CF ₃ CH ₂ ], [RC3838; H, H, H, Me, Ph, CF ₃ CF ₂ ], [RC3839; H, H, H, Me, Ph, CF ₂ H], [RC3840; H, H, H, Me, Ph, CF ₂ HCF ₂ ], [RC3841; H, H, Me, Me, Ph, Me], [RC3842; H, H, Me, Me, Ph, Et], [RC3843; H, H, Me, Me, Ph, Pr] , [RC3844; H, H, Me, Me, Ph, i-Pr], [RC3845; H, H, Me, Me, Ph, c-Pr], [RC3846; H, H, Me, Me, Ph, Bu], [RC3847; H, H, Me, Me, Ph, i-Bu], [RC3848; H, H, Me, Me, Ph, t-Bu], [RC3849; H, H, Me, Me, Ph, c-PrCH ₂ ], [RC3850; H, H, Me, Me, Ph, Ph], [RC3851; H, H, Me, Me, Ph, Bn], [RC3852; H, H, Me, Me , Ph, CF ₃ ], [RC3853; H, H, Me, Me, Ph, CF ₃ CH ₂ ], [RC3854; H, H, Me, Me, Ph, CF ₃ CF ₂ ], [RC3855; H, H, Me, Me, Ph, CF ₂ H], [RC3856; H, H, Me, Me, Ph, CF ₂ HCF ₂ ], [RC3857; H, H, Me, Et, Ph, Me], [RC3858 ; H, H, Me, Et, Ph, Et], [RC3859; H, H, Me, Et, Ph, Pr], [RC3860; H, H, Me, Et, Ph, i-Pr], [RC3861 ; H, H, Me, Et, Ph, c-Pr], [RC3862; H, H, Me, Et, Ph, Bu], [RC3863; H, H, Me, Et, Ph, i-Bu], [RC3864; H, H, Me, Et, Ph, t-Bu], [RC3865; H, H, Me, Et, Ph, c-PrCH ₂ ], [RC3866; H, H, Me, Et, Ph, Ph], [RC3867; H, H, Me, Et, Ph, Bn], [RC3868; H, H, Me, Et, Ph, CF ₃ ], [RC3869; H, H, Me, Et, Ph, CF ₃ CH ₂ ], [RC3870; H, H, Me, Et, Ph, CF ₃ CF ₂ ], [RC3871; H, H, Me, Et, Ph, CF ₂ H], [RC3872; H, H, Me , Et, Ph, CF ₂ HCF ₂ ], [RC3873; H, H, Me, F, Ph, M e], [RC3874; H, H, Me, F, Ph, Et], [RC3875; H, H, Me, F, Ph, Pr], [RC3876; H, H, Me, F, Ph, i- Pr], [RC3877; H, H, Me, F, Ph, c-Pr], [RC3878; H, H, Me, F, Ph, Bu], [RC3879; H, H, Me, F, Ph, i-Bu], [RC3880; H, H, Me, F, Ph, t-Bu], [RC3881; H, H, Me, F, Ph, c-PrCH ₂ ], [RC3882; H, H, Me , F, Ph, Ph], [RC3883; H, H, Me, F, Ph, Bn], [RC3884; H, H, Me, F, Ph, CF ₃ ], [RC3885; H, H, Me, F, Ph, CF ₃ CH ₂ ], [RC3886; H, H, Me, F, Ph, CF ₃ CF ₂ ], [RC3887; H, H, Me, F, Ph, CF ₂ H], [RC3888; H, H, Me, F, Ph, CF ₂ HCF ₂ ], [RC3889; H, H, Me, Cl, Ph, Me], [RC3890; H, H, Me, Cl, Ph, Et], [RC3891 ; H, H, Me, Cl, Ph, Pr], [RC3892; H, H, Me, Cl, Ph, i-Pr], [RC3893; H, H, Me, Cl, Ph, c-Pr], [RC3894; H, H, Me, Cl, Ph, Bu], [RC3895; H, H, Me, Cl, Ph, i-Bu], [RC3896; H, H, Me, Cl, Ph, t-Bu ], [RC3897; H, H, Me, Cl, Ph, c-PrCH ₂ ], [RC3898; H, H, Me, Cl, Ph, Ph], [RC3899; H, H, Me, Cl, Ph, Bn], [RC3900; H, H, Me, Cl, Ph, CF ₃ ], [RC3901; H, H, Me, Cl, Ph, CF ₃ CH ₂ ], [RC3902; H, H, Me, Cl, Ph, CF ₃ CF ₂ ], [RC3903; H, H, Me, Cl, Ph, CF ₂ H], [RC3904; H, H, Me, Cl, Ph, CF ₂ HCF ₂ ], [RC3905; H, H, Et, H, Ph, Me], [RC3906; H, H, Et, H, Ph, Et], [RC3907; H, H, Et, H, Ph, Pr], [RC3908; H, H, Et, H, Ph, i-Pr], [RC3909; H, H, Et, H, Ph, c-Pr], [RC3910; H, H, Et, H, Ph , Bu], [RC3911; H, H, Et, H, Ph, i-Bu], [RC3912; H, H, Et, H, Ph, t-Bu], [RC3913; H, H, Et, H , Ph, c-PrCH ₂ ], [RC3914; H, H, Et, H, Ph, Ph], [RC3915; H, H, Et, H, Ph, Bn], [RC3916; H, H, Et, H, Ph, CF ₃ ], [RC3917; H, H, Et, H, Ph, CF ₃ CH ₂ ], [RC3918; H, H, Et, H, Ph, CF ₃ CF ₂ ], [RC3919; H , H, Et, H, Ph, CF ₂ H], [RC3920; H, H, Et, H, Ph, CF ₂ HCF ₂ ], [RC3921; H, H, Et, F, Ph, Me], [ RC3922; H, H, Et, F, Ph, Et], [RC3923; H, H, Et, F, Ph, Pr], [RC3924; H, H, Et, F, Ph, i-Pr], [ RC3925; H, H, Et, F, Ph, c-Pr], [RC3926; H, H, Et, F, Ph, Bu], [RC3927; H, H, Et, F, Ph, i-Bu] , [RC3928; H, H, Et, F, Ph, t-Bu], [RC3929; H, H, Et, F, Ph, c-PrCH ₂ ], [RC3930; H, H, Et, F, Ph , Ph], [RC3931; H, H, Et, F, Ph, Bn], [RC3932; H, H, Et, F, Ph, CF ₃ ], [RC3933; H, H, Et, F, Ph, CF ₃ CH ₂ ], [RC3934; H, H, Et, F, Ph, CF ₃ CF ₂ ], [RC3935; H, H, Et, F, Ph, CF ₂ H], [RC3936; H, H, Et, F, Ph, CF ₂ HCF ₂ ], [RC3937; H, H, Et, Cl, Ph, Me], [RC3938; H, H, Et, Cl, Ph, Et], [RC3939; H, H , Et, Cl, Ph, Pr], [RC3940; H, H, Et, Cl, Ph, i-Pr], [RC3941; H, H, Et, Cl, Ph, c-Pr], [RC3942; H , H, Et, Cl, Ph, Bu], [RC3943; H, H, Et, Cl, Ph, i-Bu], [RC3944; H, H, Et, Cl, Ph, t-Bu], [RC3945 ; H, H, Et, Cl, Ph, c-PrCH ₂ ], [RC3946; H, H, Et, Cl, Ph, Ph], [RC3947; H, H, Et, C l, Ph, Bn], [RC3948; H, H, Et, Cl, Ph, CF ₃ ], [RC3949; H, H, Et, Cl, Ph, CF ₃ CH ₂ ], [RC3950; H, H, Et, Cl, Ph, CF ₃ CF ₂ ], [RC3951; H, H, Et, Cl, Ph, CF ₂ H], [RC3952; H, H, Et, Cl, Ph, CF ₂ HCF ₂ ], [ RC3953; H, H, F, H, Ph, Me], [RC3954; H, H, F, H, Ph, Et], [RC3955; H, H, F, H, Ph, Pr], [RC3956; H, H, F, H, Ph, i-Pr], [RC3957; H, H, F, H, Ph, c-Pr], [RC3958; H, H, F, H, Ph, Bu], [ RC3959; H, H, F, H, Ph, i-Bu], [RC3960; H, H, F, H, Ph, t-Bu], [RC3961; H, H, F, H, Ph, c- PrCH ₂ ], [RC3962; H, H, F, H, Ph, Ph], [RC3963; H, H, F, H, Ph, Bn], [RC3964; H, H, F, H, Ph, CF ₃ ], [RC3965; H, H, F, H, Ph, CF ₃ CH ₂ ], [RC3966; H, H, F, H, Ph, CF ₃ CF ₂ ], [RC3967; H, H, F, H, Ph, CF ₂ H], [RC3968; H, H, F, H, Ph, CF ₂ HCF ₂ ], [RC3969; H, H, F, F, Ph, Me], [RC3970; H, H , F, F, Ph, Et], [RC3971; H, H, F, F, Ph, Pr], [RC3972; H, H, F, F, Ph, i-Pr], [RC3973; H, H , F, F, Ph, c-Pr], [RC3974; H, H, F, F, Ph, Bu], [RC3975; H, H, F, F, Ph, i-Bu], [RC3976; H , H, F, F, Ph, t-Bu], [RC3977; H, H, F, F, Ph, c-PrCH ₂ ], [RC3978; H, H, F, F, Ph, Ph], [ RC3979; H, H, F, F, Ph, Bn], [RC3980; H, H, F, F, Ph, CF ₃ ], [RC3981; H, H, F, F, Ph, CF ₃ CH ₂ ] , [RC3982; H, H, F, F, Ph, CF ₃ CF ₂ ], [RC3983; H, H, F, F, Ph, CF ₂ H], [RC3984; H, H, F, F, Ph , CF ₂ HCF ₂ ], [RC3 985; H, H, F, Cl, Ph, Me], [RC3986; H, H, F, Cl, Ph, Et], [RC3987; H, H, F, Cl, Ph, Pr], [RC3988; H, H, F, Cl, Ph, i-Pr], [RC3989; H, H, F, Cl, Ph, c-Pr], [RC3990; H, H, F, Cl, Ph, Bu], [ RC3991; H, H, F, Cl, Ph, i-Bu], [RC3992; H, H, F, Cl, Ph, t-Bu], [RC3993; H, H, F, Cl, Ph, c- PrCH ₂ ], [RC3994; H, H, F, Cl, Ph, Ph], [RC3995; H, H, F, Cl, Ph, Bn], [RC3996; H, H, F, Cl, Ph, CF ₃ ], [RC3997; H, H, F, Cl, Ph, CF ₃ CH ₂ ], [RC3998; H, H, F, Cl, Ph, CF ₃ CF ₂ ], [RC3999; H, H, F, Cl, Ph, CF ₂ H], [RC4000; H, H, F, Cl, Ph, CF ₂ HCF ₂ ],

[RC4001; H, H, Cl, H, Ph, Me], [RC4002; H, H, Cl, H, Ph, Et], [RC4003; H, H, Cl, H, Ph, Pr], [RC4004 ; H, H, Cl, H, Ph, i-Pr], [RC4005; H, H, Cl, H, Ph, c-Pr], [RC4006; H, H, Cl, H, Ph, Bu], [RC4007; H, H, Cl, H, Ph, i-Bu], [RC4008; H, H, Cl, H, Ph, t-Bu], [RC4009; H, H, Cl, H, Ph, c -PrCH ₂ ], [RC4010; H, H, Cl, H, Ph, Ph], [RC4011; H, H, Cl, H, Ph, Bn], [RC4012; H, H, Cl, H, Ph, CF ₃ ], [RC4013; H, H, Cl, H, Ph, CF ₃ CH ₂ ], [RC4014; H, H, Cl, H, Ph, CF ₃ CF ₂ ], [RC4015; H, H, Cl , H, Ph, CF ₂ H], [RC4016; H, H, Cl, H, Ph, CF ₂ HCF ₂ ], [RC4017; H, H, Cl, Cl, Ph, Me], [RC4018; H, H, Cl, Cl, Ph, Et], [RC4019; H, H, Cl, Cl, Ph, Pr], [RC4020; H, H, Cl, Cl, Ph, i-Pr], [RC4021; H, H, Cl, Cl, Ph, c-Pr], [RC4022; H, H, Cl, Cl, Ph, Bu], [RC4023; H, H, Cl, Cl, Ph, i-Bu], [RC4024; H, H, Cl, Cl, Ph, t-Bu], [RC4025; H, H, Cl, Cl, Ph, c-PrCH ₂ ], [RC4026; H, H, Cl, Cl, Ph, Ph], [RC4027; H, H, Cl, Cl, Ph, Bn], [RC4028; H, H, Cl, Cl, Ph, CF ₃ ], [RC4029; H, H, Cl, Cl, Ph, CF ₃ CH ₂ ], [RC4030; H, H, Cl, Cl, Ph, CF ₃ CF ₂ ], [RC4031; H, H, Cl, Cl, Ph, CF ₂ H], [RC4032; H, H, Cl, Cl, Ph, CF ₂ HCF ₂ ], [RC4033; F, H, H, H, H, Me], [RC4034; F, H, H, H, H, Et], [RC4035; F, H, H, H , H, Pr], [RC4036; F, H, H, H, H, i-Pr], [RC4037; F, H, H, H, H, c-Pr], [RC4038; F, H, H, H, H, Bu], [RC4039; F, H, H, H, H, i-Bu], [RC4040; F, H, H, H, H, t-Bu], [ RC4041; F, H, H, H, H, c-PrCH ₂ ], [RC4042; F, H, H, H, H, Ph], [RC4043; F, H, H, H, H, Bn], [RC4044; F, H, H, H, H, CF ₃ ], [RC4045; F, H, H, H, H, CF ₃ CH ₂ ], [RC4046; F, H, H, H, H, CF ₃ CF ₂ ], [RC4047; F, H, H, H, H, CF ₂ H], [RC4048; F, H, H, H, H, CF ₂ HCF ₂ ], [RC4049; F, H, H , Me, H, Me], [RC4050; F, H, H, Me, H, Et], [RC4051; F, H, H, Me, H, Pr], [RC4052; F, H, H, Me , H, i-Pr], [RC4053; F, H, H, Me, H, c-Pr], [RC4054; F, H, H, Me, H, Bu], [RC4055; F, H, H , Me, H, i-Bu], [RC4056; F, H, H, Me, H, t-Bu], [RC4057; F, H, H, Me, H, c-PrCH ₂ ], [RC4058; F, H, H, Me, H, Ph], [RC4059; F, H, H, Me, H, Bn], [RC4060; F, H, H, Me, H, CF ₃ ], [RC4061; F , H, H, Me, H, CF ₃ CH ₂ ], [RC4062; F, H, H, Me, H, CF ₃ CF ₂ ], [RC4063; F, H, H, Me, H, CF ₂ H ], [RC4064; F, H, H, Me, H, CF ₂ HCF ₂ ], [RC4065; F, H, Me, Me, H, Me], [RC4066; F, H, Me, Me, H, Et], [RC4067; F, H, Me, Me, H, Pr], [RC4068; F, H, Me, Me, H, i-Pr], [RC4069; F, H, Me, Me, H, c-Pr], [RC4070; F, H, Me, Me, H, Bu], [RC4071; F, H, Me, Me, H, i-Bu], [RC4072; F, H, Me, Me, H, t-Bu], [RC4073; F, H, Me, Me, H, c-PrCH ₂ ], [RC4074; F, H, Me, Me, H, Ph], [RC4075; F, H, Me , Me, H, Bn], [RC4076; F, H, Me, Me, H, CF ₃ ], [R C4077; F, H, Me, Me, H, CF ₃ CH ₂ ], [RC4078; F, H, Me, Me, H, CF ₃ CF ₂ ], [RC4079; F, H, Me, Me, H, CF ₂ H], [RC4080; F, H, Me, Me, H, CF ₂ HCF ₂ ], [RC4081; F, H, Me, Et, H, Me], [RC4082; F, H, Me, Et , H, Et], [RC4083; F, H, Me, Et, H, Pr], [RC4084; F, H, Me, Et, H, i-Pr], [RC4085; F, H, Me, Et , H, c-Pr], [RC4086; F, H, Me, Et, H, Bu], [RC4087; F, H, Me, Et, H, i-Bu], [RC4088; F, H, Me , Et, H, t-Bu], [RC4089; F, H, Me, Et, H, c-PrCH ₂ ], [RC4090; F, H, Me, Et, H, Ph], [RC4091; F, H, Me, Et, H, Bn], [RC4092; F, H, Me, Et, H, CF ₃ ], [RC4093; F, H, Me, Et, H, CF ₃ CH ₂ ], [RC4094; F, H, Me, Et, H, CF ₃ CF ₂ ], [RC4095; F, H, Me, Et, H, CF ₂ H], [RC4096; F, H, Me, Et, H, CF ₂ HCF ₂ ], [RC4097; F, H, Me, F, H, Me], [RC4098; F, H, Me, F, H, Et], [RC4099; F, H, Me, F, H, Pr] , [RC4100; F, H, Me, F, H, i-Pr], [RC4101; F, H, Me, F, H, c-Pr], [RC4102; F, H, Me, F, H, Bu], [RC4103; F, H, Me, F, H, i-Bu], [RC4104; F, H, Me, F, H, t-Bu], [RC4105; F, H, Me, F, H, c-PrCH ₂ ], [RC4106; F, H, Me, F, H, Ph], [RC4107; F, H, Me, F, H, Bn], [RC4108; F, H, Me, F , H, CF ₃ ], [RC4109; F, H, Me, F, H, CF ₃ CH ₂ ], [RC4110; F, H, Me, F, H, CF ₃ CF ₂ ], [RC4111; F, H, Me, F, H, CF ₂ H], [RC4112; F, H, Me, F, H, CF ₂ HCF ₂ ], [RC4113; F, H, Me, Cl, H, Me], [RC4114 ; F, H, Me, Cl, H, Et], [RC4115; F, H, Me, Cl, H, Pr], [RC4116; F, H, Me, Cl, H, i-Pr], [RC4117 ; F, H, Me, Cl, H, c-Pr], [RC4118; F, H, Me, Cl, H, Bu], [RC4119; F, H, Me, Cl, H, i-Bu], [RC4120; F, H, Me, Cl, H, t-Bu], [RC4121; F, H, Me, Cl, H, c-PrCH ₂ ], [RC4122; F, H, Me, Cl, H, Ph], [RC4123; F, H, Me, Cl, H, Bn], [RC4124; F, H, Me, Cl, H, CF ₃ ], [RC4125; F, H, Me, Cl, H, CF ₃ CH ₂ ], [RC4126; F, H, Me, Cl, H, CF ₃ CF ₂ ], [RC4127; F, H, Me, Cl, H, CF ₂ H], [RC4128; F, H, Me , Cl, H, CF ₂ HCF ₂ ], [RC4129; F, H, Et, H, H, Me], [RC4130; F, H, Et, H, H, Et], [RC4131; F, H, Et, H, H, Pr], [RC4132; F, H, Et, H, H, i-Pr], [RC4133; F, H, Et, H, H, c-Pr], [RC4134; F, H, Et, H, H, Bu], [RC4135; F, H, Et, H, H, i-Bu], [RC4136; F, H, Et, H, H, t-Bu], [RC4137; F, H, Et, H, H, c-PrCH ₂ ], [RC4138; F, H, Et, H, H, Ph], [RC4139; F, H, Et, H, H, Bn], [RC4140 ; F, H, Et, H, H, CF ₃ ], [RC4141; F, H, Et, H, H, CF ₃ CH ₂ ], [RC4142; F, H, Et, H, H, CF ₃ CF ₂ ], [RC4143; F, H, Et, H, H, CF ₂ H], [RC4144; F, H, Et, H, H, CF ₂ HCF ₂ ], [RC4145; F, H, Et, F , H, Me], [RC4146; F, H, Et, F, H, Et], [RC4147; F, H, Et, F, H, Pr], [RC4148; F, H, Et, F, H , i-Pr], [RC4149; F, H, Et, F, H, c-Pr], [RC4150; F, H, Et, F, H, Bu], [RC4151; F, H, Et, F , H, i-Bu], [RC4152; F, H, Et, F, H , t-Bu], [RC4153; F, H, Et, F, H, c-PrCH ₂ ], [RC4154; F, H, Et, F, H, Ph], [RC4155; F, H, Et, F, H, Bn], [RC4156; F, H, Et, F, H, CF ₃ ], [RC4157; F, H, Et, F, H, CF ₃ CH ₂ ], [RC4158; F, H, Et, F, H, CF ₃ CF ₂ ], [RC4159; F, H, Et, F, H, CF ₂ H], [RC4160; F, H, Et, F, H, CF ₂ HCF ₂ ], [ RC4161; F, H, Et, Cl, H, Me], [RC4162; F, H, Et, Cl, H, Et], [RC4163; F, H, Et, Cl, H, Pr], [RC4164; F, H, Et, Cl, H, i-Pr], [RC4165; F, H, Et, Cl, H, c-Pr], [RC4166; F, H, Et, Cl, H, Bu], [ RC4167; F, H, Et, Cl, H, i-Bu], [RC4168; F, H, Et, Cl, H, t-Bu], [RC4169; F, H, Et, Cl, H, c- PrCH ₂ ], [RC4170; F, H, Et, Cl, H, Ph], [RC4171; F, H, Et, Cl, H, Bn], [RC4172; F, H, Et, Cl, H, CF ₃ ], [RC4173; F, H, Et, Cl, H, CF ₃ CH ₂ ], [RC4174; F, H, Et, Cl, H, CF ₃ CF ₂ ], [RC4175; F, H, Et, Cl, H, CF ₂ H], [RC4176; F, H, Et, Cl, H, CF ₂ HCF ₂ ], [RC4177; F, H, F, H, H, Me], [RC4178; F, H , F, H, H, Et], [RC4179; F, H, F, H, H, Pr], [RC4180; F, H, F, H, H, i-Pr], [RC4181; F, H , F, H, H, c-Pr], [RC4182; F, H, F, H, H, Bu], [RC4183; F, H, F, H, H, i-Bu], [RC4184; F , H, F, H, H, t-Bu], [RC4185; F, H, F, H, H, c-PrCH ₂ ], [RC4186; F, H, F, H, H, Ph], [ RC4187; F, H, F, H, H, Bn], [RC4188; F, H, F, H, H, CF ₃ ], [RC4189; F, H, F, H, H, CF ₃ CH ₂ ] , [RC4190; F, H, F, H, H, CF ₃ CF ₂ ], [RC4191; F, H, F, H, H, CF ₂ H], [RC4192; F, H, F, H, H, CF ₂ HCF ₂ ], [RC4193; F, H, F, F, H, Me], [RC4194; F, H, F, F, H, Et], [RC4195; F, H, F, F, H, Pr], [RC4196; F, H, F, F, H, i-Pr], [RC4197; F, H, F, F, H, c-Pr], [RC4198; F, H, F, F, H, Bu], [RC4199; F, H, F, F, H, i-Bu], [RC4200; F, H, F, F, H, t-Bu],

[RC4201; F, H, F, F, H, c-PrCH ₂ ], [RC4202; F, H, F, F, H, Ph], [RC4203; F, H, F, F, H, Bn] , [RC4204; F, H, F, F, H, CF ₃ ], [RC4205; F, H, F, F, H, CF ₃ CH ₂ ], [RC4206; F, H, F, F, H, CF ₃ CF ₂ ], [RC4207; F, H, F, F, H, CF ₂ H], [RC4208; F, H, F, F, H, CF ₂ HCF ₂ ], [RC4209; F, H, F, Cl, H, Me], [RC4210; F, H, F, Cl, H, Et], [RC4211; F, H, F, Cl, H, Pr], [RC4212; F, H, F, Cl, H, i-Pr], [RC4213; F, H, F, Cl, H, c-Pr], [RC4214; F, H, F, Cl, H, Bu], [RC4215; F, H, F, Cl, H, i-Bu], [RC4216; F, H, F, Cl, H, t-Bu], [RC4217; F, H, F, Cl, H, c-PrCH ₂ ], [RC4218 ; F, H, F, Cl, H, Ph], [RC4219; F, H, F, Cl, H, Bn], [RC4220; F, H, F, Cl, H, CF ₃ ], [RC4221; F, H, F, Cl, H, CF ₃ CH ₂ ], [RC4222; F, H, F, Cl, H, CF ₃ CF ₂ ], [RC4223; F, H, F, Cl, H, CF ₂ H], [RC4224; F, H, F, Cl, H, CF ₂ HCF ₂ ], [RC4225; F, H, Cl, H, H, Me], [RC4226; F, H, Cl, H, H , Et], [RC4227; F, H, Cl, H, H, Pr], [RC4228; F, H, Cl, H, H, i-Pr], [RC4229; F, H, Cl, H, H , c-Pr], [RC4230; F, H, Cl, H, H, Bu], [RC4231; F, H, Cl, H, H, i-Bu], [RC4232; F, H, Cl, H , H, t-Bu], [RC4233; F, H, Cl, H, H, c-PrCH ₂ ], [RC4234; F, H, Cl, H, H, Ph], [RC4235; F, H, Cl, H, H, Bn], [RC4236; F, H, Cl, H, H, CF ₃ ], [RC4237; F, H, Cl, H, H, CF ₃ CH ₂ ], [RC4238; F, H, Cl, H, H, CF ₃ CF ₂ ], [RC4239; F, H, Cl , H, H, CF ₂ H], [RC4240; F, H, Cl, H, H, CF ₂ HCF ₂ ], [RC4241; F, H, Cl, Cl, H, Me], [RC4242; F, H, Cl, Cl, H, Et], [RC4243; F, H, Cl, Cl, H, Pr], [RC4244; F, H, Cl, Cl, H, i-Pr], [RC4245; F, H, Cl, Cl, H, c-Pr], [RC4246; F, H, Cl, Cl, H, Bu], [RC4247; F, H, Cl, Cl, H, i-Bu], [RC4248; F, H, Cl, Cl, H, t-Bu], [RC4249; F, H, Cl, Cl, H, c-PrCH ₂ ], [RC4250; F, H, Cl, Cl, H, Ph], [RC4251; F, H, Cl, Cl, H, Bn], [RC4252; F, H, Cl, Cl, H, CF ₃ ], [RC4253; F, H, Cl, Cl, H, CF ₃ CH ₂ ], [RC4254; F, H, Cl, Cl, H, CF ₃ CF ₂ ], [RC4255; F, H, Cl, Cl, H, CF ₂ H], [RC4256; F, H, Cl, Cl, H, CF ₂ HCF ₂ ], [RC4257; F, H, H, H, Me, Me], [RC4258; F, H, H, H, Me, Et], [RC4259; F, H, H, H , Me, Pr], [RC4260; F, H, H, H, Me, i-Pr], [RC4261; F, H, H, H, Me, c-Pr], [RC4262; F, H, H , H, Me, Bu], [RC4263; F, H, H, H, Me, i-Bu], [RC4264; F, H, H, H, Me, t-Bu], [RC4265; F, H , H, H, Me, c-PrCH ₂ ], [RC4266; F, H, H, H, Me, Ph], [RC4267; F, H, H, H, Me, Bn], [RC4268; F, H, H, H, Me, CF ₃ ], [RC4269; F, H, H, H, Me, CF ₃ CH ₂ ], [RC4270; F, H, H, H, Me, CF ₃ CF ₂ ], [RC4271; F, H, H, H, Me, CF ₂ H], [RC4272; F, H, H, H, Me, CF ₂ HCF ₂ ], [RC4273; F, H, H, Me, Me, Me], [RC4274; F, H, H, Me, Me, Et], [RC4275; F, H, H, Me, Me, Pr], [RC4276; F, H, H, Me, Me, i- Pr], [RC4277; F, H , H, Me, Me, c-Pr], [RC4278; F, H, H, Me, Me, Bu], [RC4279; F, H, H, Me, Me, i-Bu], [RC4280; F , H, H, Me, Me, t-Bu], [RC4281; F, H, H, Me, Me, c-PrCH ₂ ], [RC4282; F, H, H, Me, Me, Ph], [ RC4283; F, H, H, Me, Me, Bn], [RC4284; F, H, H, Me, Me, CF ₃ ], [RC4285; F, H, H, Me, Me, CF ₃ CH ₂ ] , [RC4286; F, H, H, Me, Me, CF ₃ CF ₂ ], [RC4287; F, H, H, Me, Me, CF ₂ H], [RC4288; F, H, H, Me, Me , CF ₂ HCF ₂ ], [RC4289; F, H, Me, Me, Me, Me], [RC4290; F, H, Me, Me, Me, Et], [RC4291; F, H, Me, Me, Me, Pr], [RC4292; F, H, Me, Me, Me, i-Pr], [RC4293; F, H, Me, Me, Me, c-Pr], [RC4294; F, H, Me, Me, Me, Bu], [RC4295; F, H, Me, Me, Me, i-Bu], [RC4296; F, H, Me, Me, Me, t-Bu], [RC4297; F, H, Me, Me, Me, c-PrCH ₂ ], [RC4298; F, H, Me, Me, Me, Ph], [RC4299; F, H, Me, Me, Me, Bn], [RC4300; F, H , Me, Me, Me, CF ₃ ], [RC4301; F, H, Me, Me, Me, CF ₃ CH ₂ ], [RC4302; F, H, Me, Me, Me, CF ₃ CF ₂ ], [ RC4303; F, H, Me, Me, Me, CF ₂ H], [RC4304; F, H, Me, Me, Me, CF ₂ HCF ₂ ], [RC4305; F, H, Me, Et, Me, Me ], [RC4306; F, H, Me, Et, Me, Et], [RC4307; F, H, Me, Et, Me, Pr], [RC4308; F, H, Me, Et, Me, i-Pr ], [RC4309; F, H, Me, Et, Me, c-Pr], [RC4310; F, H, Me, Et, Me, Bu], [RC4311; F, H, Me, Et, Me, i -Bu], [RC4312; F, H, Me, Et, Me, t-Bu], [RC4313; F, H, Me, Et, Me, c- PrCH ₂ ], [RC4314; F, H, Me, Et, Me, Ph], [RC4315; F, H, Me, Et, Me, Bn], [RC4316; F, H, Me, Et, Me, CF ₃ ], [RC4317; F, H, Me, Et, Me, CF ₃ CH ₂ ], [RC4318; F, H, Me, Et, Me, CF ₃ CF ₂ ], [RC4319; F, H, Me, Et, Me, CF ₂ H], [RC4320; F, H, Me, Et, Me, CF ₂ HCF ₂ ], [RC4321; F, H, Me, F, Me, Me], [RC4322; F, H , Me, F, Me, Et], [RC4323; F, H, Me, F, Me, Pr], [RC4324; F, H, Me, F, Me, i-Pr], [RC4325; F, H , Me, F, Me, c-Pr], [RC4326; F, H, Me, F, Me, Bu], [RC4327; F, H, Me, F, Me, i-Bu], [RC4328; F , H, Me, F, Me, t-Bu], [RC4329; F, H, Me, F, Me, c-PrCH ₂ ], [RC4330; F, H, Me, F, Me, Ph], [ RC4331; F, H, Me, F, Me, Bn], [RC4332; F, H, Me, F, Me, CF ₃ ], [RC4333; F, H, Me, F, Me, CF ₃ CH ₂ ] , [RC4334; F, H, Me, F, Me, CF ₃ CF ₂ ], [RC4335; F, H, Me, F, Me, CF ₂ H], [RC4336; F, H, Me, F, Me , CF ₂ HCF ₂ ], [RC4337; F, H, Me, Cl, Me, Me], [RC4338; F, H, Me, Cl, Me, Et], [RC4339; F, H, Me, Cl, Me, Pr], [RC4340; F, H, Me, Cl, Me, i-Pr], [RC4341; F, H, Me, Cl, Me, c-Pr], [RC4342; F, H, Me, Cl, Me, Bu], [RC4343; F, H, Me, Cl, Me, i-Bu], [RC4344; F, H, Me, Cl, Me, t-Bu], [RC4345; F, H, Me, Cl, Me, c-PrCH ₂ ], [RC4346; F, H, Me, Cl, Me, Ph], [RC4347; F, H, Me, Cl, Me, Bn], [RC4348; F, H , Me, Cl, Me, CF ₃ ], [RC4349; F, H, Me, Cl, Me, CF ₃ CH ₂ ], [R C4350; F, H, Me, Cl, Me, CF ₃ CF ₂ ], [RC4351; F, H, Me, Cl, Me, CF ₂ H], [RC4352; F, H, Me, Cl, Me, CF ₂ HCF ₂ ], [RC4353; F, H, Et, H, Me, Me], [RC4354; F, H, Et, H, Me, Et], [RC4355; F, H, Et, H, Me, Pr], [RC4356; F, H, Et, H, Me, i-Pr], [RC4357; F, H, Et, H, Me, c-Pr], [RC4358; F, H, Et, H, Me, Bu], [RC4359; F, H, Et, H, Me, i-Bu], [RC4360; F, H, Et, H, Me, t-Bu], [RC4361; F, H, Et, H, Me, c-PrCH ₂ ], [RC4362; F, H, Et, H, Me, Ph], [RC4363; F, H, Et, H, Me, Bn], [RC4364; F, H, Et , H, Me, CF ₃ ], [RC4365; F, H, Et, H, Me, CF ₃ CH ₂ ], [RC4366; F, H, Et, H, Me, CF ₃ CF ₂ ], [RC4367; F, H, Et, H, Me, CF ₂ H], [RC4368; F, H, Et, H, Me, CF ₂ HCF ₂ ], [RC4369; F, H, Et, F, Me, Me], [RC4370; F, H, Et, F, Me, Et], [RC4371; F, H, Et, F, Me, Pr], [RC4372; F, H, Et, F, Me, i-Pr], [RC4373; F, H, Et, F, Me, c-Pr], [RC4374; F, H, Et, F, Me, Bu], [RC4375; F, H, Et, F, Me, i-Bu ], [RC4376; F, H, Et, F, Me, t-Bu], [RC4377; F, H, Et, F, Me, c-PrCH ₂ ], [RC4378; F, H, Et, F, Me, Ph], [RC4379; F, H, Et, F, Me, Bn], [RC4380; F, H, Et, F, Me, CF ₃ ], [RC4381; F, H, Et, F, Me , CF ₃ CH ₂ ], [RC4382; F, H, Et, F, Me, CF ₃ CF ₂ ], [RC4383; F, H, Et, F, Me, CF ₂ H], [RC4384; F, H , Et, F, Me, CF ₂ HCF ₂ ], [RC4385; F, H, Et, Cl, Me, Me], [RC4386; F, H, Et, Cl, M e, Et], [RC4387; F, H, Et, Cl, Me, Pr], [RC4388; F, H, Et, Cl, Me, i-Pr], [RC4389; F, H, Et, Cl, Me, c-Pr], [RC4390; F, H, Et, Cl, Me, Bu], [RC4391; F, H, Et, Cl, Me, i-Bu], [RC4392; F, H, Et, Cl, Me, t-Bu], [RC4393; F, H, Et, Cl, Me, c-PrCH ₂ ], [RC4394; F, H, Et, Cl, Me, Ph], [RC4395; F, H , Et, Cl, Me, Bn], [RC4396; F, H, Et, Cl, Me, CF ₃ ], [RC4397; F, H, Et, Cl, Me, CF ₃ CH ₂ ], [RC4398; F , H, Et, Cl, Me, CF ₃ CF ₂ ], [RC4399; F, H, Et, Cl, Me, CF ₂ H], [RC4400; F, H, Et, Cl, Me, CF ₂ HCF ₂ ],

[RC4401; F, H, F, H, Me, Me], [RC4402; F, H, F, H, Me, Et], [RC4403; F, H, F, H, Me, Pr], [RC4404 ; F, H, F, H, Me, i-Pr], [RC4405; F, H, F, H, Me, c-Pr], [RC4406; F, H, F, H, Me, Bu], [RC4407; F, H, F, H, Me, i-Bu], [RC4408; F, H, F, H, Me, t-Bu], [RC4409; F, H, F, H, Me, c -PrCH ₂ ], [RC4410; F, H, F, H, Me, Ph], [RC4411; F, H, F, H, Me, Bn], [RC4412; F, H, F, H, Me, CF ₃ ], [RC4413; F, H, F, H, Me, CF ₃ CH ₂ ], [RC4414; F, H, F, H, Me, CF ₃ CF ₂ ], [RC4415; F, H, F , H, Me, CF ₂ H], [RC4416; F, H, F, H, Me, CF ₂ HCF ₂ ], [RC4417; F, H, F, F, Me, Me], [RC4418; F, H, F, F, Me, Et], [RC4419; F, H, F, F, Me, Pr], [RC4420; F, H, F, F, Me, i-Pr], [RC4421; F, H, F, F, Me, c-Pr], [RC4422; F, H, F, F, Me, Bu], [RC4423; F, H, F, F, Me, i-Bu], [RC4424; F, H, F, F, Me, t-Bu], [RC4425; F, H, F, F, Me, c-PrCH ₂ ], [RC4426; F, H, F, F, Me, Ph], [RC4427; F, H, F, F, Me, Bn], [RC4428; F, H, F, F, Me, CF ₃ ], [RC4429; F, H, F, F, Me, CF ₃ CH ₂ ], [RC4430; F, H, F, F, Me, CF ₃ CF ₂ ], [RC4431; F, H, F, F, Me, CF ₂ H], [RC4432; F, H, F, F, Me, CF ₂ HCF ₂ ], [RC4433; F, H, F, Cl, Me, Me], [RC4434; F, H, F, Cl, Me, Et], [RC4435; F, H, F, Cl , Me, Pr], [RC4436; F, H, F, Cl, Me, i-Pr], [RC4437; F, H, F, Cl, Me, c-Pr], [RC4438; F, H, F , Cl, Me, Bu], [RC4439; F, H, F, Cl, Me, i- Bu], [RC4440; F, H, F, Cl, Me, t-Bu], [RC4441; F, H, F, Cl, Me, c-PrCH ₂ ], [RC4442; F, H, F, Cl , Me, Ph], [RC4443; F, H, F, Cl, Me, Bn], [RC4444; F, H, F, Cl, Me, CF ₃ ], [RC4445; F, H, F, Cl, Me, CF ₃ CH ₂ ], [RC4446; F, H, F, Cl, Me, CF ₃ CF ₂ ], [RC4447; F, H, F, Cl, Me, CF ₂ H], [RC4448; F, H, F, Cl, Me, CF ₂ HCF ₂ ], [RC4449; F, H, Cl, H, Me, Me], [RC4450; F, H, Cl, H, Me, Et], [RC4451; F , H, Cl, H, Me, Pr], [RC4452; F, H, Cl, H, Me, i-Pr], [RC4453; F, H, Cl, H, Me, c-Pr], [RC4454 ; F, H, Cl, H, Me, Bu], [RC4455; F, H, Cl, H, Me, i-Bu], [RC4456; F, H, Cl, H, Me, t-Bu], [RC4457; F, H, Cl, H, Me, c-PrCH ₂ ], [RC4458; F, H, Cl, H, Me, Ph], [RC4459; F, H, Cl, H, Me, Bn] , [RC4460; F, H, Cl, H, Me, CF ₃ ], [RC4461; F, H, Cl, H, Me, CF ₃ CH ₂ ], [RC4462; F, H, Cl, H, Me, CF ₃ CF ₂ ], [RC4463; F, H, Cl, H, Me, CF ₂ H], [RC4464; F, H, Cl, H, Me, CF ₂ HCF ₂ ], [RC4465; F, H, Cl, Cl, Me, Me], [RC4466; F, H, Cl, Cl, Me, Et], [RC4467; F, H, Cl, Cl, Me, Pr], [RC4468; F, H, Cl, Cl, Me, i-Pr], [RC4469; F, H, Cl, Cl, Me, c-Pr], [RC4470; F, H, Cl, Cl, Me, Bu], [RC4471; F, H, Cl, Cl, Me, i-Bu], [RC4472; F, H, Cl, Cl, Me, t-Bu], [RC4473; F, H, Cl, Cl, Me, c-PrCH ₂ ], [RC4474 ; F, H, Cl, Cl, Me, Ph], [RC4475; F, H, Cl, Cl, Me, Bn], [RC4476; F, H, Cl, Cl, Me, CF ₃ ], [RC4477; F, H, Cl, Cl, Me, CF ₃ CH ₂ ], [RC4478; F, H, Cl, Cl, Me, CF ₃ CF ₂ ], [RC4479; F, H , Cl, Cl, Me, CF ₂ H], [RC4480; F, H, Cl, Cl, Me, CF ₂ HCF ₂ ], [RC4481; F, H, H, H, Et, Me], [RC4482; F, H, H, H, Et, Et], [RC4483; F, H, H, H, Et, Pr], [RC4484; F, H, H, H, Et, i-Pr], [RC4485; F, H, H, H, Et, c-Pr], [RC4486; F, H, H, H, Et, Bu], [RC4487; F, H, H, H, Et, i-Bu], [ RC4488; F, H, H, H, Et, t-Bu], [RC4489; F, H, H, H, Et, c-PrCH ₂ ], [RC4490; F, H, H, H, Et, Ph ], [RC4491; F, H, H, H, Et, Bn], [RC4492; F, H, H, H, Et, CF ₃ ], [RC4493; F, H, H, H, Et, CF ₃ CH ₂ ], [RC4494; F, H, H, H, Et, CF ₃ CF ₂ ], [RC4495; F, H, H, H, Et, CF ₂ H], [RC4496; F, H, H, H, Et, CF ₂ HCF ₂ ], [RC4497; F, H, H, Me, Et, Me], [RC4498; F, H, H, Me, Et, Et], [RC4499; F, H, H , Me, Et, Pr], [RC4500; F, H, H, Me, Et, i-Pr], [RC4501; F, H, H, Me, Et, c-Pr], [RC4502; F, H , H, Me, Et, Bu], [RC4503; F, H, H, Me, Et, i-Bu], [RC4504; F, H, H, Me, Et, t-Bu], [RC4505; F , H, H, Me, Et, c-PrCH ₂ ], [RC4506; F, H, H, Me, Et, Ph], [RC4507; F, H, H, Me, Et, Bn], [RC4508; F, H, H, Me, Et, CF ₃ ], [RC4509; F, H, H, Me, Et, CF ₃ CH ₂ ], [RC4510; F, H, H, Me, Et, CF ₃ CF ₂ ], [RC4511; F, H, H, Me, Et, CF ₂ H], [RC4512; F, H, H, Me, Et, CF ₂ HCF ₂ ], [RC4513; F, H, Me, Me, Et, Me], [RC4514; F, H, Me, Me, Et, Et], [RC4515; F, H, Me, Me, Et, Pr], [RC4516; F, H, Me, Me, Et, i-Pr], [RC4517; F, H, Me, Me, Et, c-Pr], [RC4518; F, H, Me, Me, Et, Bu], [RC4519; F, H, Me, Me, Et, i-Bu], [RC4520; F, H, Me, Me, Et, t-Bu], [RC4521; F, H, Me, Me, Et, c-PrCH ₂ ], [RC4522; F , H, Me, Me, Et, Ph], [RC4523; F, H, Me, Me, Et, Bn], [RC4524; F, H, Me, Me, Et, CF ₃ ], [RC4525; F, H, Me, Me, Et, CF ₃ CH ₂ ], [RC4526; F, H, Me, Me, Et, CF ₃ CF ₂ ], [RC4527; F, H, Me, Me, Et, CF ₂ H] , [RC4528; F, H, Me, Me, Et, CF ₂ HCF ₂ ], [RC4529; F, H, Me, Et, Et, Me], [RC4530; F, H, Me, Et, Et, Et ], [RC4531; F, H, Me, Et, Et, Pr], [RC4532; F, H, Me, Et, Et, i-Pr], [RC4533; F, H, Me, Et, Et, c -Pr], [RC4534; F, H, Me, Et, Et, Bu], [RC4535; F, H, Me, Et, Et, i-Bu], [RC4536; F, H, Me, Et, Et , t-Bu], [RC4537; F, H, Me, Et, Et, c-PrCH ₂ ], [RC4538; F, H, Me, Et, Et, Ph], [RC4539; F, H, Me, Et, Et, Bn], [RC4540; F, H, Me, Et, Et, CF ₃ ], [RC4541; F, H, Me, Et, Et, CF ₃ CH ₂ ], [RC4542; F, H, Me, Et, Et, CF ₃ CF ₂ ], [RC4543; F, H, Me, Et, Et, CF ₂ H], [RC4544; F, H, Me, Et, Et, CF ₂ HCF ₂ ], [ RC4545; F, H, Me, F, Et, Me], [RC4546; F, H, Me, F, Et, Et], [RC4547; F, H, Me, F, Et, Pr], [RC4548; F, H, Me, F, Et, i-Pr], [RC4549; F, H, Me, F, Et, cP r], [RC4550; F, H, Me, F, Et, Bu], [RC4551; F, H, Me, F, Et, i-Bu], [RC4552; F, H, Me, F, Et, t-Bu], [RC4553; F, H, Me, F, Et, c-PrCH ₂ ], [RC4554; F, H, Me, F, Et, Ph], [RC4555; F, H, Me, F , Et, Bn], [RC4556; F, H, Me, F, Et, CF ₃ ], [RC4557; F, H, Me, F, Et, CF ₃ CH ₂ ], [RC4558; F, H, Me , F, Et, CF ₃ CF ₂ ], [RC4559; F, H, Me, F, Et, CF ₂ H], [RC4560; F, H, Me, F, Et, CF ₂ HCF ₂ ], [RC4561 ; F, H, Me, Cl, Et, Me], [RC4562; F, H, Me, Cl, Et, Et], [RC4563; F, H, Me, Cl, Et, Pr], [RC4564; F , H, Me, Cl, Et, i-Pr], [RC4565; F, H, Me, Cl, Et, c-Pr], [RC4566; F, H, Me, Cl, Et, Bu], [RC4567 ; F, H, Me, Cl, Et, i-Bu], [RC4568; F, H, Me, Cl, Et, t-Bu], [RC4569; F, H, Me, Cl, Et, c-PrCH ₂ ], [RC4570; F, H, Me, Cl, Et, Ph], [RC4571; F, H, Me, Cl, Et, Bn], [RC4572; F, H, Me, Cl, Et, CF ₃ ], [RC4573; F, H, Me, Cl, Et, CF ₃ CH ₂ ], [RC4574; F, H, Me, Cl, Et, CF ₃ CF ₂ ], [RC4575; F, H, Me, Cl _{, Et, CF 2 H],} [RC4576; F, H, Me, Cl, Et, CF 2 HCF 2], [RC4577; F, H, Et, H, Et, Me], [RC4578; F, H, Et, H, Et, Et], [RC4579; F, H, Et, H, Et, Pr], [RC4580; F, H, Et, H, Et, i-Pr], [RC4581; F, H, Et, H, Et, c-Pr], [RC4582; F, H, Et, H, Et, Bu], [RC4583; F, H, Et, H, Et, i-Bu], [RC4584; F, H, Et, H, Et, t-Bu], [RC4585; F, H, Et, H, Et, c-PrCH ₂ ], [RC4586; F, H, Et, H, Et, Ph], [RC4587; F, H, Et, H, Et, Bn], [RC4588; F, H, Et, H, Et, CF ₃ ], [RC4589; F, H, Et , H, Et, CF ₃ CH ₂ ], [RC4590; F, H, Et, H, Et, CF ₃ CF ₂ ], [RC4591; F, H, Et, H, Et, CF ₂ H], [RC4592 ; F, H, Et, H, Et, CF ₂ HCF ₂ ], [RC4593; F, H, Et, F, Et, Me], [RC4594; F, H, Et, F, Et, Et], [ RC4595; F, H, Et, F, Et, Pr], [RC4596; F, H, Et, F, Et, i-Pr], [RC4597; F, H, Et, F, Et, c-Pr] , [RC4598; F, H, Et, F, Et, Bu], [RC4599; F, H, Et, F, Et, i-Bu], [RC4600; F, H, Et, F, Et, t- Bu],

[RC4601; F, H, Et, F, Et, c-PrCH ₂ ], [RC4602; F, H, Et, F, Et, Ph], [RC4603; F, H, Et, F, Et, Bn] , [RC4604; F, H, Et, F, Et, CF ₃ ], [RC4605; F, H, Et, F, Et, CF ₃ CH ₂ ], [RC4606; F, H, Et, F, Et, CF ₃ CF ₂ ], [RC4607; F, H, Et, F, Et, CF ₂ H], [RC4608; F, H, Et, F, Et, CF ₂ HCF ₂ ], [RC4609; F, H, Et, Cl, Et, Me], [RC4610; F, H, Et, Cl, Et, Et], [RC4611; F, H, Et, Cl, Et, Pr], [RC4612; F, H, Et, Cl, Et, i-Pr], [RC4613; F, H, Et, Cl, Et, c-Pr], [RC4614; F, H, Et, Cl, Et, Bu], [RC4615; F, H, Et, Cl, Et, i-Bu], [RC4616; F, H, Et, Cl, Et, t-Bu], [RC4617; F, H, Et, Cl, Et, c-PrCH ₂ ], [RC4618 ; F, H, Et, Cl, Et, Ph], [RC4619; F, H, Et, Cl, Et, Bn], [RC4620; F, H, Et, Cl, Et, CF ₃ ], [RC4621; F, H, Et, Cl, Et, CF ₃ CH ₂ ], [RC4622; F, H, Et, Cl, Et, CF ₃ CF ₂ ], [RC4623; F, H, Et, Cl, Et, CF ₂ H], [RC4624; F, H, Et, Cl, Et, CF ₂ HCF ₂ ], [RC4625; F, H, F, H, Et, Me], [RC4626; F, H, F, H, Et , Et], [RC4627; F, H, F, H, Et, Pr], [RC4628; F, H, F, H, Et, i-Pr], [RC4629; F, H, F, H, Et , c-Pr], [RC4630; F, H, F, H, Et, Bu], [RC4631; F, H, F, H, Et, i-Bu], [RC4632; F, H, F, H , Et, t-Bu], [RC4633; F, H, F, H, Et, c-PrCH ₂ ], [RC4634; F, H, F, H, Et, Ph], [RC4635; F, H, F, H, Et, Bn], [RC4636; F, H, F, H, Et, CF ₃ ], [RC4637; F, H, F, H, Et, CF ₃ CH ₂ ], [RC4638; F, H, F, H, Et, CF ₃ CF ₂ ], [RC4639; F, H, F, H, Et, CF ₂ H], [RC4640; F, H, F, H, Et, CF ₂ HCF ₂ ], [RC4641; F, H, F, F, Et, Me], [RC4642; F, H, F, F, Et, Et], [RC4643; F, H, F, F , Et, Pr], [RC4644; F, H, F, F, Et, i-Pr], [RC4645; F, H, F, F, Et, c-Pr], [RC4646; F, H, F , F, Et, Bu], [RC4647; F, H, F, F, Et, i-Bu], [RC4648; F, H, F, F, Et, t-Bu], [RC4649; F, H , F, F, Et, c-PrCH ₂ ], [RC4650; F, H, F, F, Et, Ph], [RC4651; F, H, F, F, Et, Bn], [RC4652; F, H, F, F, Et, CF ₃ ], [RC4653; F, H, F, F, Et, CF ₃ CH ₂ ], [RC4654; F, H, F, F, Et, CF ₃ CF ₂ ], [RC4655; F, H, F, F, Et, CF ₂ H], [RC4656; F, H, F, F, Et, CF ₂ HCF ₂ ], [RC4657; F, H, F, Cl, Et, Me], [RC4658; F, H, F, Cl, Et, Et], [RC4659; F, H, F, Cl, Et, Pr], [RC4660; F, H, F, Cl, Et, i- Pr], [RC4661; F, H, F, Cl, Et, c-Pr], [RC4662; F, H, F, Cl, Et, Bu], [RC4663; F, H, F, Cl, Et, i-Bu], [RC4664; F, H, F, Cl, Et, t-Bu], [RC4665; F, H, F, Cl, Et, c-PrCH ₂ ], [RC4666; F, H, F , Cl, Et, Ph], [RC4667; F, H, F, Cl, Et, Bn], [RC4668; F, H, F, Cl, Et, CF ₃ ], [RC4669; F, H, F, Cl, Et, CF ₃ CH ₂ ], [RC4670; F, H, F, Cl, Et, CF ₃ CF ₂ ], [RC4671; F, H, F, Cl, Et, CF ₂ H], [RC4672; F, H, F, Cl, Et, CF ₂ HCF ₂ ], [RC4673; F, H, Cl, H, Et, Me], [RC4674; F, H, Cl, H, Et, Et], [RC4675 ; F, H, C l, H, Et, Pr], [RC4676; F, H, Cl, H, Et, i-Pr], [RC4677; F, H, Cl, H, Et, c-Pr], [RC4678; F, H, Cl, H, Et, Bu], [RC4679; F, H, Cl, H, Et, i-Bu], [RC4680; F, H, Cl, H, Et, t-Bu], [RC4681; F, H, Cl, H, Et, c-PrCH ₂ ], [RC4682; F, H, Cl, H, Et, Ph], [RC4683; F, H, Cl, H, Et, Bn], [RC4684 ; F, H, Cl, H, Et, CF ₃ ], [RC4685; F, H, Cl, H, Et, CF ₃ CH ₂ ], [RC4686; F, H, Cl, H, Et, CF ₃ CF ₂ ], [RC4687; F, H, Cl, H, Et, CF ₂ H], [RC4688; F, H, Cl, H, Et, CF ₂ HCF ₂ ], [RC4689; F, H, Cl, Cl , Et, Me], [RC4690; F, H, Cl, Cl, Et, Et], [RC4691; F, H, Cl, Cl, Et, Pr], [RC4692; F, H, Cl, Cl, Et , i-Pr], [RC4693; F, H, Cl, Cl, Et, c-Pr], [RC4694; F, H, Cl, Cl, Et, Bu], [RC4695; F, H, Cl, Cl , Et, i-Bu], [RC4696; F, H, Cl, Cl, Et, t-Bu], [RC4697; F, H, Cl, Cl, Et, c-PrCH ₂ ], [RC4698; F, H, Cl, Cl, Et, Ph], [RC4699; F, H, Cl, Cl, Et, Bn], [RC4700; F, H, Cl, Cl, Et, CF ₃ ], [RC4701; F, H , Cl, Cl, Et, CF ₃ CH ₂ ], [RC4702; F, H, Cl, Cl, Et, CF ₃ CF ₂ ], [RC4703; F, H, Cl, Cl, Et, CF ₂ H], [RC4704; F, H, Cl, Cl, Et, CF ₂ HCF ₂ ], [RC4705; F, H, H, H, Pr, Me], [RC4706; F, H, H, H, Pr, Et] , [RC4707; F, H, H, H, Pr, Pr], [RC4708; F, H, H, H, Pr, i-Pr], [RC4709; F, H, H, H, Pr, c- Pr], [RC4710; F, H, H, H, Pr, Bu], [RC4711; F, H, H, H, Pr, i-Bu], [RC4712; F, H, H, H, Pr, t-Bu], [RC4713; F, H, H, H, Pr, c-PrCH ₂ ], [RC4714; F, H, H, H, Pr, Ph], [RC4715; F, H, H , H, Pr, Bn], [RC4716; F, H, H, H, Pr, CF ₃ ], [RC4717; F, H, H, H, Pr, CF ₃ CH ₂ ], [RC4718; F, H , H, H, Pr, CF ₃ CF ₂ ], [RC4719; F, H, H, H, Pr, CF ₂ H], [RC4720; F, H, H, H, Pr, CF ₂ HCF ₂ ], [RC4721; F, H, H, Me, Pr, Me], [RC4722; F, H, H, Me, Pr, Et], [RC4723; F, H, H, Me, Pr, Pr], [RC4724 ; F, H, H, Me, Pr, i-Pr], [RC4725; F, H, H, Me, Pr, c-Pr], [RC4726; F, H, H, Me, Pr, Bu], [RC4727; F, H, H, Me, Pr, i-Bu], [RC4728; F, H, H, Me, Pr, t-Bu], [RC4729; F, H, H, Me, Pr, c -PrCH ₂ ], [RC4730; F, H, H, Me, Pr, Ph], [RC4731; F, H, H, Me, Pr, Bn], [RC4732; F, H, H, Me, Pr, CF ₃ ], [RC4733; F, H, H, Me, Pr, CF ₃ CH ₂ ], [RC4734; F, H, H, Me, Pr, CF ₃ CF ₂ ], [RC4735; F, H, H , Me, Pr, CF ₂ H], [RC4736; F, H, H, Me, Pr, CF ₂ HCF ₂ ], [RC4737; F, H, Me, Me, Pr, Me], [RC4738; F, H, Me, Me, Pr, Et], [RC4739; F, H, Me, Me, Pr, Pr], [RC4740; F, H, Me, Me, Pr, i-Pr], [RC4741; F, H, Me, Me, Pr, c-Pr], [RC4742; F, H, Me, Me, Pr, Bu], [RC4743; F, H, Me, Me, Pr, i-Bu], [RC4744; F, H, Me, Me, Pr, t-Bu], [RC4745; F, H, Me, Me, Pr, c-PrCH ₂ ], [RC4746; F, H, Me, Me, Pr, Ph], [RC4747; F, H, Me, Me, Pr, Bn], [RC4748; F, H, Me, Me, Pr, CF ₃ ], [RC4749; F, H, Me, Me, P r, CF ₃ CH ₂ ], [RC4750; F, H, Me, Me, Pr, CF ₃ CF ₂ ], [RC4751; F, H, Me, Me, Pr, CF ₂ H], [RC4752; F, H, Me, Me, Pr, CF ₂ HCF ₂ ], [RC4753; F, H, Me, Et, Pr, Me], [RC4754; F, H, Me, Et, Pr, Et], [RC4755; F , H, Me, Et, Pr, Pr], [RC4756; F, H, Me, Et, Pr, i-Pr], [RC4757; F, H, Me, Et, Pr, c-Pr], [RC4758 ; F, H, Me, Et, Pr, Bu], [RC4759; F, H, Me, Et, Pr, i-Bu], [RC4760; F, H, Me, Et, Pr, t-Bu], [RC4761; F, H, Me, Et, Pr, c-PrCH ₂ ], [RC4762; F, H, Me, Et, Pr, Ph], [RC4763; F, H, Me, Et, Pr, Bn] , [RC4764; F, H, Me, Et, Pr, CF ₃ ], [RC4765; F, H, Me, Et, Pr, CF ₃ CH ₂ ], [RC4766; F, H, Me, Et, Pr, CF ₃ CF ₂ ], [RC4767; F, H, Me, Et, Pr, CF ₂ H], [RC4768; F, H, Me, Et, Pr, CF ₂ HCF ₂ ], [RC4769; F, H, Me, F, Pr, Me], [RC4770; F, H, Me, F, Pr, Et], [RC4771; F, H, Me, F, Pr, Pr], [RC4772; F, H, Me, F, Pr, i-Pr], [RC4773; F, H, Me, F, Pr, c-Pr], [RC4774; F, H, Me, F, Pr, Bu], [RC4775; F, H, Me, F, Pr, i-Bu], [RC4776; F, H, Me, F, Pr, t-Bu], [RC4777; F, H, Me, F, Pr, c-PrCH ₂ ], [RC4778 ; F, H, Me, F, Pr, Ph], [RC4779; F, H, Me, F, Pr, Bn], [RC4780; F, H, Me, F, Pr, CF ₃ ], [RC4781; F, H, Me, F, Pr, CF ₃ CH ₂ ], [RC4782; F, H, Me, F, Pr, CF ₃ CF ₂ ], [RC4783; F, H, Me, F, Pr, CF ₂ H], [RC4784; F, H, Me, F, Pr, CF ₂ HCF ₂ ], [RC4785; F, H, Me, Cl, Pr, Me], [RC4786; F, H, Me, Cl, Pr, Et], [RC4787; F, H, Me, Cl, Pr, Pr], [RC4788; F, H, Me, Cl, Pr, i-Pr], [RC4789; F, H, Me, Cl, Pr, c-Pr], [RC4790; F, H, Me, Cl, Pr, Bu], [RC4791; F, H, Me, Cl, Pr, i-Bu], [RC4792; F, H, Me, Cl, Pr, t-Bu], [RC4793; F, H, Me, Cl, Pr, c-PrCH ₂ ], [RC4794 ; F, H, Me, Cl, Pr, Ph], [RC4795; F, H, Me, Cl, Pr, Bn], [RC4796; F, H, Me, Cl, Pr, CF ₃ ], [RC4797; F, H, Me, Cl, Pr, CF ₃ CH ₂ ], [RC4798; F, H, Me, Cl, Pr, CF ₃ CF ₂ ], [RC4799; F, H, Me, Cl, Pr, CF ₂ H], [RC4800; F, H, Me, Cl, Pr, CF ₂ HCF ₂ ],

[RC4801; F, H, Et, H, Pr, Me], [RC4802; F, H, Et, H, Pr, Et], [RC4803; F, H, Et, H, Pr, Pr], [RC4804 ; F, H, Et, H, Pr, i-Pr], [RC4805; F, H, Et, H, Pr, c-Pr], [RC4806; F, H, Et, H, Pr, Bu], [RC4807; F, H, Et, H, Pr, i-Bu], [RC4808; F, H, Et, H, Pr, t-Bu], [RC4809; F, H, Et, H, Pr, c -PrCH ₂ ], [RC4810; F, H, Et, H, Pr, Ph], [RC4811; F, H, Et, H, Pr, Bn], [RC4812; F, H, Et, H, Pr, CF ₃ ], [RC4813; F, H, Et, H, Pr, CF ₃ CH ₂ ], [RC4814; F, H, Et, H, Pr, CF ₃ CF ₂ ], [RC4815; F, H, Et , H, Pr, CF ₂ H], [RC4816; F, H, Et, H, Pr, CF ₂ HCF ₂ ], [RC4817; F, H, Et, F, Pr, Me], [RC4818; F, H, Et, F, Pr, Et], [RC4819; F, H, Et, F, Pr, Pr], [RC4820; F, H, Et, F, Pr, i-Pr], [RC4821; F, H, Et, F, Pr, c-Pr], [RC4822; F, H, Et, F, Pr, Bu], [RC4823; F, H, Et, F, Pr, i-Bu], [RC4824; F, H, Et, F, Pr, t-Bu], [RC4825; F, H, Et, F, Pr, c-PrCH ₂ ], [RC4826; F, H, Et, F, Pr, Ph], [RC4827; F, H, Et, F, Pr, Bn], [RC4828; F, H, Et, F, Pr, CF ₃ ], [RC4829; F, H, Et, F, Pr, CF ₃ CH ₂ ], [RC4830; F, H, Et, F, Pr, CF ₃ CF ₂ ], [RC4831; F, H, Et, F, Pr, CF ₂ H], [RC4832; F, H, Et, F, Pr, CF ₂ HCF ₂ ], [RC4833; F, H, Et, Cl, Pr, Me], [RC4834; F, H, Et, Cl, Pr, Et], [RC4835; F, H, Et, Cl , Pr, Pr], [RC4836; F, H, Et, Cl, Pr, i-Pr], [RC4837; F, H, Et, Cl, Pr, c-Pr], [RC4838; F , H, Et, Cl, Pr, Bu], [RC4839; F, H, Et, Cl, Pr, i-Bu], [RC4840; F, H, Et, Cl, Pr, t-Bu], [RC4841 ; F, H, Et, Cl, Pr, c-PrCH ₂ ], [RC4842; F, H, Et, Cl, Pr, Ph], [RC4843; F, H, Et, Cl, Pr, Bn], [ RC4844; F, H, Et, Cl, Pr, CF ₃ ], [RC4845; F, H, Et, Cl, Pr, CF ₃ CH ₂ ], [RC4846; F, H, Et, Cl, Pr, CF ₃ CF ₂ ], [RC4847; F, H, Et, Cl, Pr, CF ₂ H], [RC4848; F, H, Et, Cl, Pr, CF ₂ HCF ₂ ], [RC4849; F, H, F, H, Pr, Me], [RC4850; F, H, F, H, Pr, Et], [RC4851; F, H, F, H, Pr, Pr], [RC4852; F, H, F, H, Pr, i-Pr], [RC4853; F, H, F, H, Pr, c-Pr], [RC4854; F, H, F, H, Pr, Bu], [RC4855; F, H, F, H, Pr, i-Bu], [RC4856; F, H, F, H, Pr, t-Bu], [RC4857; F, H, F, H, Pr, c-PrCH ₂ ], [RC4858; F , H, F, H, Pr, Ph], [RC4859; F, H, F, H, Pr, Bn], [RC4860; F, H, F, H, Pr, CF ₃ ], [RC4861; F, H, F, H, Pr, CF ₃ CH ₂ ], [RC4862; F, H, F, H, Pr, CF ₃ CF ₂ ], [RC4863; F, H, F, H, Pr, CF ₂ H] , [RC4864; F, H, F, H, Pr, CF ₂ HCF ₂ ], [RC4865; F, H, F, F, Pr, Me], [RC4866; F, H, F, F, Pr, Et ], [RC4867; F, H, F, F, Pr, Pr], [RC4868; F, H, F, F, Pr, i-Pr], [RC4869; F, H, F, F, Pr, c -Pr], [RC4870; F, H, F, F, Pr, Bu], [RC4871; F, H, F, F, Pr, i-Bu], [RC4872; F, H, F, F, Pr , t-Bu], [RC4873; F, H, F, F, Pr, c-PrCH ₂ ], [RC4874; F, H, F, F, Pr, Ph], [RC4875; F, H, F, F, Pr, Bn], [RC4876; F, H, F, F, Pr, CF ₃ ], [RC4877; F, H, F, F, Pr, CF ₃ CH ₂ ], [RC4878; F, H, F, F, Pr, CF ₃ CF ₂ ], [RC4879; F, H, F, F, Pr, CF ₂ H], [RC4880; F, H, F, F, Pr, CF ₂ HCF ₂ ], [RC4881; F, H, F, Cl, Pr, Me], [RC4882; F, H, F, Cl, Pr, Et], [RC4883; F, H, F, Cl, Pr, Pr], [RC4884; F, H, F, Cl, Pr, i-Pr], [RC4885; F, H, F, Cl, Pr, c-Pr], [RC4886; F, H, F, Cl, Pr, Bu], [RC4887; F, H, F, Cl, Pr, i-Bu], [RC4888; F, H, F, Cl, Pr, t-Bu], [RC4889; F, H, F, Cl, Pr, c-PrCH ₂ ], [RC4890; F, H , F, Cl, Pr, Ph], [RC4891; F, H, F, Cl, Pr, Bn], [RC4892; F, H, F, Cl, Pr, CF ₃ ], [RC4893; F, H, F, Cl, Pr, CF ₃ CH ₂ ], [RC4894; F, H, F, Cl, Pr, CF ₃ CF ₂ ], [RC4895; F, H, F, Cl, Pr, CF ₂ H], [ RC4896; F, H, F, Cl, Pr, CF ₂ HCF ₂ ], [RC4897; F, H, Cl, H, Pr, Me], [RC4898; F, H, Cl, H, Pr, Et], [RC4899; F, H, Cl, H, Pr, Pr], [RC4900; F, H, Cl, H, Pr, i-Pr], [RC4901; F, H, Cl, H, Pr, c-Pr ], [RC4902; F, H, Cl, H, Pr, Bu], [RC4903; F, H, Cl, H, Pr, i-Bu], [RC4904; F, H, Cl, H, Pr, t -Bu], [RC4905; F, H, Cl, H, Pr, c-PrCH ₂ ], [RC4906; F, H, Cl, H, Pr, Ph], [RC4907; F, H, Cl, H, Pr, Bn], [RC4908; F, H, Cl, H, Pr, CF ₃ ], [RC4909; F, H, Cl, H, Pr, CF ₃ CH ₂ ], [RC4910; F, H, Cl, H, Pr, CF ₃ CF ₂ ], [RC4911; F, H, Cl, H, Pr, CF ₂ H], [RC4912; F, H, Cl, H, Pr, CF ₂ HCF ₂ ] , [RC4913; F, H, Cl, Cl, Pr, Me], [RC4914; F, H, Cl, Cl, Pr, Et], [RC4915; F, H, Cl, Cl, Pr, Pr], [ RC4916; F, H, Cl, Cl, Pr, i-Pr], [RC4917; F, H, Cl, Cl, Pr, c-Pr], [RC4918; F, H, Cl, Cl, Pr, Bu] , [RC4919; F, H, Cl, Cl, Pr, i-Bu], [RC4920; F, H, Cl, Cl, Pr, t-Bu], [RC4921; F, H, Cl, Cl, Pr, c-PrCH ₂ ], [RC4922; F, H, Cl, Cl, Pr, Ph], [RC4923; F, H, Cl, Cl, Pr, Bn], [RC4924; F, H, Cl, Cl, Pr , CF ₃ ], [RC4925; F, H, Cl, Cl, Pr, CF ₃ CH ₂ ], [RC4926; F, H, Cl, Cl, Pr, CF ₃ CF ₂ ], [RC4927; F, H, Cl, Cl, Pr, CF ₂ H], [RC4928; F, H, Cl, Cl, Pr, CF ₂ HCF ₂ ], [RC4929; F, H, H, H, Bu, Me], [RC4930; F , H, H, H, Bu, Et], [RC4931; F, H, H, H, Bu, Pr], [RC4932; F, H, H, H, Bu, i-Pr], [RC4933; F , H, H, H, Bu, c-Pr], [RC4934; F, H, H, H, Bu, Bu], [RC4935; F, H, H, H, Bu, i-Bu], [RC4936 ; F, H, H, H, Bu, t-Bu], [RC4937; F, H, H, H, Bu, c-PrCH ₂ ], [RC4938; F, H, H, H, Bu, Ph] , [RC4939; F, H, H, H, Bu, Bn], [RC4940; F, H, H, H, Bu, CF ₃ ], [RC4941; F, H, H, H, Bu, CF ₃ CH ₂ ], [RC4942; F, H, H, H, Bu, CF ₃ CF ₂ ], [RC4943; F, H, H, H, Bu, CF ₂ H], [RC4944; F, H, H, H , Bu, CF ₂ HCF ₂ ], [RC4945; F, H, H, Me, Bu, Me], [RC4946; F, H, H, Me, Bu, Et], [RC4947; F, H, H, Me, Bu, Pr], [RC4948; F, H, H, Me, Bu, i-Pr], [RC4949; F, H, H, Me, Bu, c-Pr], [RC4950; F, H, H , Me, Bu, Bu], [RC4951; F, H, H, Me, Bu, i-Bu], [RC4952; F, H, H, Me, Bu, t-Bu], [RC4953; F, H , H, Me, Bu, c-PrCH ₂ ], [RC4954; F, H, H, Me, Bu, Ph], [RC4955; F, H, H, Me, Bu, Bn], [RC4956; F, H, H, Me, Bu, CF ₃ ], [RC4957; F, H, H, Me, Bu, CF ₃ CH ₂ ], [RC4958; F, H, H, Me, Bu, CF ₃ CF ₂ ], [RC4959; F, H, H, Me, Bu, CF ₂ H], [RC4960; F, H, H, Me, Bu, CF ₂ HCF ₂ ], [RC4961; F, H, Me, Me, Bu, Me], [RC4962; F, H, Me, Me, Bu, Et], [RC4963; F, H, Me, Me, Bu, Pr], [RC4964; F, H, Me, Me, Bu, i- Pr], [RC4965; F, H, Me, Me, Bu, c-Pr], [RC4966; F, H, Me, Me, Bu, Bu], [RC4967; F, H, Me, Me, Bu, i-Bu], [RC4968; F, H, Me, Me, Bu, t-Bu], [RC4969; F, H, Me, Me, Bu, c-PrCH ₂ ], [RC4970; F, H, Me , Me, Bu, Ph], [RC4971; F, H, Me, Me, Bu, Bn], [RC4972; F, H, Me, Me, Bu, CF ₃ ], [RC4973; F, H, Me, Me, Bu, CF ₃ CH ₂ ], [RC4974; F, H, Me, Me, Bu, CF ₃ CF ₂ ], [RC4975; F, H, Me, Me, Bu, CF ₂ H], [RC4976; F, H, Me, Me, Bu, CF ₂ HCF ₂ ], [RC4977; F, H, Me, Et, Bu, Me], [RC4978; F, H, Me, Et, Bu, Et], [RC4979 ; F, H, Me, Et, Bu, Pr], [RC4980; F, H, Me, Et, Bu, i-Pr], [RC4981; F, H, Me, Et, Bu, c-Pr], [RC4982; F, H, Me, Et, Bu, Bu], [RC4983; F, H, Me, Et, Bu, i-Bu], [RC4984; F, H, Me, Et, Bu, t-Bu ], [RC4985; F, H, Me, Et, Bu, c-PrCH ₂ ], [RC4986; F, H, Me, Et, B u, Ph], [RC4987; F, H, Me, Et, Bu, Bn], [RC4988; F, H, Me, Et, Bu, CF ₃ ], [RC4989; F, H, Me, Et, Bu , CF ₃ CH ₂ ], [RC4990; F, H, Me, Et, Bu, CF ₃ CF ₂ ], [RC4991; F, H, Me, Et, Bu, CF ₂ H], [RC4992; F, H , Me, Et, Bu, CF ₂ HCF ₂ ], [RC4993; F, H, Me, F, Bu, Me], [RC4994; F, H, Me, F, Bu, Et], [RC4995; F, H, Me, F, Bu, Pr], [RC4996; F, H, Me, F, Bu, i-Pr], [RC4997; F, H, Me, F, Bu, c-Pr], [RC4998; F, H, Me, F, Bu, Bu], [RC4999; F, H, Me, F, Bu, i-Bu], [RC5000; F, H, Me, F, Bu, t-Bu],

[RC5001; F, H, Me, F, Bu, c-PrCH ₂ ], [RC5002; F, H, Me, F, Bu, Ph], [RC5003; F, H, Me, F, Bu, Bn] , [RC5004; F, H, Me, F, Bu, CF ₃ ], [RC5005; F, H, Me, F, Bu, CF ₃ CH ₂ ], [RC5006; F, H, Me, F, Bu, CF ₃ CF ₂ ], [RC5007; F, H, Me, F, Bu, CF ₂ H], [RC5008; F, H, Me, F, Bu, CF ₂ HCF ₂ ], [RC5009; F, H, Me, Cl, Bu, Me], [RC5010; F, H, Me, Cl, Bu, Et], [RC5011; F, H, Me, Cl, Bu, Pr], [RC5012; F, H, Me, Cl, Bu, i-Pr], [RC5013; F, H, Me, Cl, Bu, c-Pr], [RC5014; F, H, Me, Cl, Bu, Bu], [RC5015; F, H, Me, Cl, Bu, i-Bu], [RC5016; F, H, Me, Cl, Bu, t-Bu], [RC5017; F, H, Me, Cl, Bu, c-PrCH ₂ ], [RC5018 ; F, H, Me, Cl, Bu, Ph], [RC5019; F, H, Me, Cl, Bu, Bn], [RC5020; F, H, Me, Cl, Bu, CF ₃ ], [RC5021; F, H, Me, Cl, Bu, CF ₃ CH ₂ ], [RC5022; F, H, Me, Cl, Bu, CF ₃ CF ₂ ], [RC5023; F, H, Me, Cl, Bu, CF ₂ H], [RC5024; F, H, Me, Cl, Bu, CF ₂ HCF ₂ ], [RC5025; F, H, Et, H, Bu, Me], [RC5026; F, H, Et, H, Bu , Et], [RC5027; F, H, Et, H, Bu, Pr], [RC5028; F, H, Et, H, Bu, i-Pr], [RC5029; F, H, Et, H, Bu , c-Pr], [RC5030; F, H, Et, H, Bu, Bu], [RC5031; F, H, Et, H, Bu, i-Bu], [RC5032; F, H, Et, H , Bu, t-Bu], [RC5033; F, H, Et, H, Bu, c-PrCH ₂ ], [RC5034; F, H, Et, H, Bu, Ph], [RC5035; F, H, Et, H, Bu, Bn], [RC5036; F, H, Et, H, Bu, CF ₃ ], [RC5037; F, H, Et, H , Bu, CF ₃ CH ₂ ], [RC5038; F, H, Et, H, Bu, CF ₃ CF ₂ ], [RC5039; F, H, Et, H, Bu, CF ₂ H], [RC5040; F , H, Et, H, Bu, CF ₂ HCF ₂ ], [RC5041; F, H, Et, F, Bu, Me], [RC5042; F, H, Et, F, Bu, Et], [RC5043; F, H, Et, F, Bu, Pr], [RC5044; F, H, Et, F, Bu, i-Pr], [RC5045; F, H, Et, F, Bu, c-Pr], [ RC5046; F, H, Et, F, Bu, Bu], [RC5047; F, H, Et, F, Bu, i-Bu], [RC5048; F, H, Et, F, Bu, t-Bu] , [RC5049; F, H, Et, F, Bu, c-PrCH ₂ ], [RC5050; F, H, Et, F, Bu, Ph], [RC5051; F, H, Et, F, Bu, Bn ], [RC5052; F, H, Et, F, Bu, CF ₃ ], [RC5053; F, H, Et, F, Bu, CF ₃ CH ₂ ], [RC5054; F, H, Et, F, Bu , CF ₃ CF ₂ ], [RC5055; F, H, Et, F, Bu, CF ₂ H], [RC5056; F, H, Et, F, Bu, CF ₂ HCF ₂ ], [RC5057; F, H , Et, Cl, Bu, Me], [RC5058; F, H, Et, Cl, Bu, Et], [RC5059; F, H, Et, Cl, Bu, Pr], [RC5060; F, H, Et , Cl, Bu, i-Pr], [RC5061; F, H, Et, Cl, Bu, c-Pr], [RC5062; F, H, Et, Cl, Bu, Bu], [RC5063; F, H , Et, Cl, Bu, i-Bu], [RC5064; F, H, Et, Cl, Bu, t-Bu], [RC5065; F, H, Et, Cl, Bu, c-PrCH ₂ ], [ RC5066; F, H, Et, Cl, Bu, Ph], [RC5067; F, H, Et, Cl, Bu, Bn], [RC5068; F, H, Et, Cl, Bu, CF ₃ ], [RC5069 ; F, H, Et, Cl, Bu, CF ₃ CH ₂ ], [RC5070; F, H, Et, Cl, Bu, CF ₃ CF ₂ ], [RC5071; F, H, Et, Cl, Bu, CF ₂ H], [RC5072; F, H, Et, Cl, Bu, CF ₂ HCF ₂ ], [RC5073; F, H, F , H, Bu, Me], [RC5074; F, H, F, H, Bu, Et], [RC5075; F, H, F, H, Bu, Pr], [RC5076; F, H, F, H , Bu, i-Pr], [RC5077; F, H, F, H, Bu, c-Pr], [RC5078; F, H, F, H, Bu, Bu], [RC5079; F, H, F , H, Bu, i-Bu], [RC5080; F, H, F, H, Bu, t-Bu], [RC5081; F, H, F, H, Bu, c-PrCH ₂ ], [RC5082; F, H, F, H, Bu, Ph], [RC5083; F, H, F, H, Bu, Bn], [RC5084; F, H, F, H, Bu, CF ₃ ], [RC5085; F , H, F, H, Bu, CF ₃ CH ₂ ], [RC5086; F, H, F, H, Bu, CF ₃ CF ₂ ], [RC5087; F, H, F, H, Bu, CF ₂ H ], [RC5088; F, H, F, H, Bu, CF ₂ HCF ₂ ], [RC5089; F, H, F, F, Bu, Me], [RC5090; F, H, F, F, Bu, Et], [RC5091; F, H, F, F, Bu, Pr], [RC5092; F, H, F, F, Bu, i-Pr], [RC5093; F, H, F, F, Bu, c-Pr], [RC5094; F, H, F, F, Bu, Bu], [RC5095; F, H, F, F, Bu, i-Bu], [RC5096; F, H, F, F, Bu, t-Bu], [RC5097; F, H, F, F, Bu, c-PrCH ₂ ], [RC5098; F, H, F, F, Bu, Ph], [RC5099; F, H, F , F, Bu, Bn], [RC5100; F, H, F, F, Bu, CF ₃ ], [RC5101; F, H, F, F, Bu, CF ₃ CH ₂ ], [RC5102; F, H , F, F, Bu, CF ₃ CF ₂ ], [RC5103; F, H, F, F, Bu, CF ₂ H], [RC5104; F, H, F, F, Bu, CF ₂ HCF ₂ ], [RC5105; F, H, F, Cl, Bu, Me], [RC5106; F, H, F, Cl, Bu, Et], [RC5107; F, H, F, Cl, Bu, Pr], [RC5108 ; F, H, F, Cl, Bu, i-Pr], [RC5109; F, H, F, Cl, Bu, c-Pr], [RC5110; F, H, F, Cl, Bu, Bu], [RC5111; F, H, F, Cl, Bu, i-Bu], [RC5112; F , H, F, Cl, Bu, t-Bu], [RC5113; F, H, F, Cl, Bu, c-PrCH ₂ ], [RC5114; F, H, F, Cl, Bu, Ph], [ RC5115; F, H, F, Cl, Bu, Bn], [RC5116; F, H, F, Cl, Bu, CF ₃ ], [RC5117; F, H, F, Cl, Bu, CF ₃ CH ₂ ] , [RC5118; F, H, F, Cl, Bu, CF ₃ CF ₂ ], [RC5119; F, H, F, Cl, Bu, CF ₂ H], [RC5120; F, H, F, Cl, Bu , CF ₂ HCF ₂ ], [RC5121; F, H, Cl, H, Bu, Me], [RC5122; F, H, Cl, H, Bu, Et], [RC5123; F, H, Cl, H, Bu, Pr], [RC5124; F, H, Cl, H, Bu, i-Pr], [RC5125; F, H, Cl, H, Bu, c-Pr], [RC5126; F, H, Cl, H, Bu, Bu], [RC5127; F, H, Cl, H, Bu, i-Bu], [RC5128; F, H, Cl, H, Bu, t-Bu], [RC5129; F, H, Cl, H, Bu, c-PrCH ₂ ], [RC5130; F, H, Cl, H, Bu, Ph], [RC5131; F, H, Cl, H, Bu, Bn], [RC5132; F, H , Cl, H, Bu, CF ₃ ], [RC5133; F, H, Cl, H, Bu, CF ₃ CH ₂ ], [RC5134; F, H, Cl, H, Bu, CF ₃ CF ₂ ], [ RC5135; F, H, Cl, H, Bu, CF ₂ H], [RC5136; F, H, Cl, H, Bu, CF ₂ HCF ₂ ], [RC5137; F, H, Cl, Cl, Bu, Me ], [RC5138; F, H, Cl, Cl, Bu, Et], [RC5139; F, H, Cl, Cl, Bu, Pr], [RC5140; F, H, Cl, Cl, Bu, i-Pr ], [RC5141; F, H, Cl, Cl, Bu, c-Pr], [RC5142; F, H, Cl, Cl, Bu, Bu], [RC5143; F, H, Cl, Cl, Bu, i -Bu], [RC5144; F, H, Cl, Cl, Bu, t-Bu], [RC5145; F, H, Cl, Cl, Bu, c-PrCH ₂ ], [RC5146; F, H, Cl, Cl, Bu, Ph], [RC5147; F, H, Cl, Cl, Bu, Bn], [RC5148; F, H, Cl, Cl, Bu, CF ₃ ], [RC 5149; F, H, Cl, Cl, Bu, CF ₃ CH ₂ ], [RC5150; F, H, Cl, Cl, Bu, CF ₃ CF ₂ ], [RC5151; F, H, Cl, Cl, Bu, CF ₂ H], [RC5152; F, H, Cl, Cl, Bu, CF ₂ HCF ₂ ], [RC5153; F, H, H, H, i-Pr, Me], [RC5154; F, H, H , H, i-Pr, Et], [RC5155; F, H, H, H, i-Pr, Pr], [RC5156; F, H, H, H, i-Pr, i-Pr], [RC5157 ; F, H, H, H, i-Pr, c-Pr], [RC5158; F, H, H, H, i-Pr, Bu], [RC5159; F, H, H, H, i-Pr , i-Bu], [RC5160; F, H, H, H, i-Pr, t-Bu], [RC5161; F, H, H, H, i-Pr, c-PrCH ₂ ], [RC5162; F, H, H, H, i-Pr, Ph], [RC5163; F, H, H, H, i-Pr, Bn], [RC5164; F, H, H, H, i-Pr, CF ₃ ], [RC5165; F, H, H, H, i-Pr, CF ₃ CH ₂ ], [RC5166; F, H, H, H, i-Pr, CF ₃ CF ₂ ], [RC5167; F, H , H, H, i-Pr, CF ₂ H], [RC5168; F, H, H, H, i-Pr, CF ₂ HCF ₂ ], [RC5169; F, H, H, Me, i-Pr, Me], [RC5170; F, H, H, Me, i-Pr, Et], [RC5171; F, H, H, Me, i-Pr, Pr], [RC5172; F, H, H, Me, i-Pr, i-Pr], [RC5173; F, H, H, Me, i-Pr, c-Pr], [RC5174; F, H, H, Me, i-Pr, Bu], [RC5175; F, H, H, Me, i-Pr, i-Bu], [RC5176; F, H, H, Me, i-Pr, t-Bu], [RC5177; F, H, H, Me, i- Pr, c-PrCH ₂ ], [RC5178; F, H, H, Me, i-Pr, Ph], [RC5179; F, H, H, Me, i-Pr, Bn], [RC5180; F, H , H, Me, i-Pr, CF ₃ ], [RC5181; F, H, H, Me, i-Pr, CF ₃ CH ₂ ], [RC5182; F, H, H, Me, i-Pr, CF ₃ CF ₂ ], [RC5183; F, H, H, Me, i-Pr, CF ₂ H] , [RC5184; F, H, H, Me, i-Pr, CF ₂ HCF ₂ ], [RC5185; F, H, Me, Me, i-Pr, Me], [RC5186; F, H, Me, Me , i-Pr, Et], [RC5187; F, H, Me, Me, i-Pr, Pr], [RC5188; F, H, Me, Me, i-Pr, i-Pr], [RC5189; F , H, Me, Me, i-Pr, c-Pr], [RC5190; F, H, Me, Me, i-Pr, Bu], [RC5191; F, H, Me, Me, i-Pr, i -Bu], [RC5192; F, H, Me, Me, i-Pr, t-Bu], [RC5193; F, H, Me, Me, i-Pr, c-PrCH ₂ ], [RC5194; F, H, Me, Me, i-Pr, Ph], [RC5195; F, H, Me, Me, i-Pr, Bn], [RC5196; F, H, Me, Me, i-Pr, CF ₃ ], [RC5197; F, H, Me, Me, i-Pr, CF ₃ CH ₂ ], [RC5198; F, H, Me, Me, i-Pr, CF ₃ CF ₂ ], [RC5199; F, H, Me , Me, i-Pr, CF ₂ H], [RC5200; F, H, Me, Me, i-Pr, CF ₂ HCF ₂ ],

[RC5201; F, H, Me, Et, i-Pr, Me], [RC5202; F, H, Me, Et, i-Pr, Et], [RC5203; F, H, Me, Et, i-Pr , Pr], [RC5204; F, H, Me, Et, i-Pr, i-Pr], [RC5205; F, H, Me, Et, i-Pr, c-Pr], [RC5206; F, H , Me, Et, i-Pr, Bu], [RC5207; F, H, Me, Et, i-Pr, i-Bu], [RC5208; F, H, Me, Et, i-Pr, t-Bu ], [RC5209; F, H, Me, Et, i-Pr, c-PrCH ₂ ], [RC5210; F, H, Me, Et, i-Pr, Ph], [RC5211; F, H, Me, Et, i-Pr, Bn], [RC5212; F, H, Me, Et, i-Pr, CF ₃ ], [RC5213; F, H, Me, Et, i-Pr, CF ₃ CH ₂ ], [ RC5214; F, H, Me, Et, i-Pr, CF ₃ CF ₂ ], [RC5215; F, H, Me, Et, i-Pr, CF ₂ H], [RC5216; F, H, Me, Et , i-Pr, CF ₂ HCF ₂ ], [RC5217; F, H, Me, F, i-Pr, Me], [RC5218; F, H, Me, F, i-Pr, Et], [RC5219; F, H, Me, F, i-Pr, Pr], [RC5220; F, H, Me, F, i-Pr, i-Pr], [RC5221; F, H, Me, F, i-Pr, c-Pr], [RC5222; F, H, Me, F, i-Pr, Bu], [RC5223; F, H, Me, F, i-Pr, i-Bu], [RC5224; F, H, Me, F, i-Pr, t-Bu], [RC5225; F, H, Me, F, i-Pr, c-PrCH ₂ ], [RC5226; F, H, Me, F, i-Pr, Ph ], [RC5227; F, H, Me, F, i-Pr, Bn], [RC5228; F, H, Me, F, i-Pr, CF ₃ ], [RC5229; F, H, Me, F, i-Pr, CF ₃ CH ₂ ], [RC5230; F, H, Me, F, i-Pr, CF ₃ CF ₂ ], [RC5231; F, H, Me, F, i-Pr, CF ₂ H] , [RC5232; F, H, Me, F, i-Pr, CF ₂ HCF ₂ ], [RC5233; F, H, Me, Cl, i-Pr, Me], [RC5234; F, H, Me, Cl , i-Pr, Et], [RC5 235; F, H, Me, Cl, i-Pr, Pr], [RC5236; F, H, Me, Cl, i-Pr, i-Pr], [RC5237; F, H, Me, Cl, i- Pr, c-Pr], [RC5238; F, H, Me, Cl, i-Pr, Bu], [RC5239; F, H, Me, Cl, i-Pr, i-Bu], [RC5240; F, H, Me, Cl, i-Pr, t-Bu], [RC5241; F, H, Me, Cl, i-Pr, c-PrCH ₂ ], [RC5242; F, H, Me, Cl, i-Pr , Ph], [RC5243; F, H, Me, Cl, i-Pr, Bn], [RC5244; F, H, Me, Cl, i-Pr, CF ₃ ], [RC5245; F, H, Me, Cl, i-Pr, CF ₃ CH ₂ ], [RC5246; F, H, Me, Cl, i-Pr, CF ₃ CF ₂ ], [RC5247; F, H, Me, Cl, i-Pr, CF ₂ H], [RC5248; F, H, Me, Cl, i-Pr, CF ₂ HCF ₂ ], [RC5249; F, H, Et, H, i-Pr, Me], [RC5250; F, H, Et , H, i-Pr, Et], [RC5251; F, H, Et, H, i-Pr, Pr], [RC5252; F, H, Et, H, i-Pr, i-Pr], [RC5253 ; F, H, Et, H, i-Pr, c-Pr], [RC5254; F, H, Et, H, i-Pr, Bu], [RC5255; F, H, Et, H, i-Pr , i-Bu], [RC5256; F, H, Et, H, i-Pr, t-Bu], [RC5257; F, H, Et, H, i-Pr, c-PrCH ₂ ], [RC5258; F, H, Et, H, i-Pr, Ph], [RC5259; F, H, Et, H, i-Pr, Bn], [RC5260; F, H, Et, H, i-Pr, CF ₃ ], [RC5261; F, H, Et, H, i-Pr, CF ₃ CH ₂ ], [RC5262; F, H, Et, H, i-Pr, CF ₃ CF ₂ ], [RC5263; F, H , Et, H, i-Pr, CF ₂ H], [RC5264; F, H, Et, H, i-Pr, CF ₂ HCF ₂ ], [RC5265; F, H, Et, F, i-Pr, Me], [RC5266; F, H, Et, F, i-Pr, Et], [RC5267; F, H, Et, F, i-Pr, Pr], [RC5268; F, H, Et, F, i-Pr, i-Pr], [RC5269; F, H, Et, F, i-Pr, c-Pr], [RC5270; F, H, Et, F, i-Pr, Bu], [RC5271; F, H, Et, F, i-Pr, i- Bu], [RC5272; F, H, Et, F, i-Pr, t-Bu], [RC5273; F, H, Et, F, i-Pr, c-PrCH ₂ ], [RC5274; F, H , Et, F, i-Pr, Ph], [RC5275; F, H, Et, F, i-Pr, Bn], [RC5276; F, H, Et, F, i-Pr, CF ₃ ], [ RC5277; F, H, Et, F, i-Pr, CF ₃ CH ₂ ], [RC5278; F, H, Et, F, i-Pr, CF ₃ CF ₂ ], [RC5279; F, H, Et, F, i-Pr, CF ₂ H], [RC5280; F, H, Et, F, i-Pr, CF ₂ HCF ₂ ], [RC5281; F, H, Et, Cl, i-Pr, Me], [RC5282; F, H, Et, Cl, i-Pr, Et], [RC5283; F, H, Et, Cl, i-Pr, Pr], [RC5284; F, H, Et, Cl, i-Pr , i-Pr], [RC5285; F, H, Et, Cl, i-Pr, c-Pr], [RC5286; F, H, Et, Cl, i-Pr, Bu], [RC5287; F, H , Et, Cl, i-Pr, i-Bu], [RC5288; F, H, Et, Cl, i-Pr, t-Bu], [RC5289; F, H, Et, Cl, i-Pr, c -PrCH ₂ ], [RC5290; F, H, Et, Cl, i-Pr, Ph], [RC5291; F, H, Et, Cl, i-Pr, Bn], [RC5292; F, H, Et, Cl, i-Pr, CF ₃ ], [RC5293; F, H, Et, Cl, i-Pr, CF ₃ CH ₂ ], [RC5294; F, H, Et, Cl, i-Pr, CF ₃ CF ₂ ], [RC5295; F, H, Et, Cl, i-Pr, CF ₂ H], [RC5296; F, H, Et, Cl, i-Pr, CF ₂ HCF ₂ ], [RC5297; F, H, F, H, i-Pr, Me], [RC5298; F, H, F, H, i-Pr, Et], [RC5299; F, H, F, H, i-Pr, Pr], [RC5300; F, H, F, H, i-Pr, i-Pr], [RC5301; F, H, F, H, i-Pr, c-Pr], [RC5302; F, H, F, H, i- Pr, Bu], [RC5303; F, H, F, H, i-Pr , i-Bu], [RC5304; F, H, F, H, i-Pr, t-Bu], [RC5305; F, H, F, H, i-Pr, c-PrCH ₂ ], [RC5306; F, H, F, H, i-Pr, Ph], [RC5307; F, H, F, H, i-Pr, Bn], [RC5308; F, H, F, H, i-Pr, CF ₃ ], [RC5309; F, H, F, H, i-Pr, CF ₃ CH ₂ ], [RC5310; F, H, F, H, i-Pr, CF ₃ CF ₂ ], [RC5311; F, H , F, H, i-Pr, CF ₂ H], [RC5312; F, H, F, H, i-Pr, CF ₂ HCF ₂ ], [RC5313; F, H, F, F, i-Pr, Me], [RC5314; F, H, F, F, i-Pr, Et], [RC5315; F, H, F, F, i-Pr, Pr], [RC5316; F, H, F, F, i-Pr, i-Pr], [RC5317; F, H, F, F, i-Pr, c-Pr], [RC5318; F, H, F, F, i-Pr, Bu], [RC5319; F, H, F, F, i-Pr, i-Bu], [RC5320; F, H, F, F, i-Pr, t-Bu], [RC5321; F, H, F, F, i- Pr, c-PrCH ₂ ], [RC5322; F, H, F, F, i-Pr, Ph], [RC5323; F, H, F, F, i-Pr, Bn], [RC5324; F, H , F, F, i-Pr, CF ₃ ], [RC5325; F, H, F, F, i-Pr, CF ₃ CH ₂ ], [RC5326; F, H, F, F, i-Pr, CF ₃ CF ₂ ], [RC5327; F, H, F, F, i-Pr, CF ₂ H], [RC5328; F, H, F, F, i-Pr, CF ₂ HCF ₂ ], [RC5329; F , H, F, Cl, i-Pr, Me], [RC5330; F, H, F, Cl, i-Pr, Et], [RC5331; F, H, F, Cl, i-Pr, Pr], [RC5332; F, H, F, Cl, i-Pr, i-Pr], [RC5333; F, H, F, Cl, i-Pr, c-Pr], [RC5334; F, H, F, Cl , i-Pr, Bu], [RC5335; F, H, F, Cl, i-Pr, i-Bu], [RC5336; F, H, F, Cl, i-Pr, t-Bu], [RC5337 ; F, H, F, Cl, i-Pr, c-PrCH ₂ ], [RC5338; F, H, F, Cl, i-Pr, Ph], [RC53 39; F, H, F, Cl, i-Pr, Bn], [RC5340; F, H, F, Cl, i-Pr, CF ₃ ], [RC5341; F, H, F, Cl, i-Pr , CF ₃ CH ₂ ], [RC5342; F, H, F, Cl, i-Pr, CF ₃ CF ₂ ], [RC5343; F, H, F, Cl, i-Pr, CF ₂ H], [RC5344 ; F, H, F, Cl, i-Pr, CF ₂ HCF ₂ ], [RC5345; F, H, Cl, H, i-Pr, Me], [RC5346; F, H, Cl, H, i- Pr, Et], [RC5347; F, H, Cl, H, i-Pr, Pr], [RC5348; F, H, Cl, H, i-Pr, i-Pr], [RC5349; F, H, Cl, H, i-Pr, c-Pr], [RC5350; F, H, Cl, H, i-Pr, Bu], [RC5351; F, H, Cl, H, i-Pr, i-Bu] , [RC5352; F, H, Cl, H, i-Pr, t-Bu], [RC5353; F, H, Cl, H, i-Pr, c-PrCH ₂ ], [RC5354; F, H, Cl , H, i-Pr, Ph], [RC5355; F, H, Cl, H, i-Pr, Bn], [RC5356; F, H, Cl, H, i-Pr, CF ₃ ], [RC5357; F, H, Cl, H, i-Pr, CF ₃ CH ₂ ], [RC5358; F, H, Cl, H, i-Pr, CF ₃ CF ₂ ], [RC5359; F, H, Cl, H, i-Pr, CF ₂ H], [RC5360; F, H, Cl, H, i-Pr, CF ₂ HCF ₂ ], [RC5361; F, H, Cl, Cl, i-Pr, Me], [RC5362 ; F, H, Cl, Cl, i-Pr, Et], [RC5363; F, H, Cl, Cl, i-Pr, Pr], [RC5364; F, H, Cl, Cl, i-Pr, i -Pr], [RC5365; F, H, Cl, Cl, i-Pr, c-Pr], [RC5366; F, H, Cl, Cl, i-Pr, Bu], [RC5367; F, H, Cl , Cl, i-Pr, i-Bu], [RC5368; F, H, Cl, Cl, i-Pr, t-Bu], [RC5369; F, H, Cl, Cl, i-Pr, c-PrCH ₂ ], [RC5370; F, H, Cl, Cl, i-Pr, Ph], [RC5371; F, H, Cl, Cl, i-Pr, Bn], [RC5372; F, H, Cl, Cl, i-Pr, CF ₃ ], [RC5373; F, H, Cl, Cl, i-Pr, CF ₃ CH ₂ ], [RC5374; F, H, Cl, Cl, i-Pr, CF ₃ CF ₂ ], [RC5375; F, H, Cl, Cl, i-Pr, CF ₂ H], [RC5376; F, H, Cl, Cl, i-Pr, CF ₂ HCF ₂ ], [RC5377; F, H, H, H, c-Pr, Me], [RC5378; F, H , H, H, c-Pr, Et], [RC5379; F, H, H, H, c-Pr, Pr], [RC5380; F, H, H, H, c-Pr, i-Pr], [RC5381; F, H, H, H, c-Pr, c-Pr], [RC5382; F, H, H, H, c-Pr, Bu], [RC5383; F, H, H, H, c -Pr, i-Bu], [RC5384; F, H, H, H, c-Pr, t-Bu], [RC5385; F, H, H, H, c-Pr, c-PrCH ₂ ], [ RC5386; F, H, H, H, c-Pr, Ph], [RC5387; F, H, H, H, c-Pr, Bn], [RC5388; F, H, H, H, c-Pr, CF ₃ ], [RC5389; F, H, H, H, c-Pr, CF ₃ CH ₂ ], [RC5390; F, H, H, H, c-Pr, CF ₃ CF ₂ ], [RC5391; F , H, H, H, c-Pr, CF ₂ H], [RC5392; F, H, H, H, c-Pr, CF ₂ HCF ₂ ], [RC5393; F, H, H, Me, c- Pr, Me], [RC5394; F, H, H, Me, c-Pr, Et], [RC5395; F, H, H, Me, c-Pr, Pr], [RC5396; F, H, H, Me, c-Pr, i-Pr], [RC5397; F, H, H, Me, c-Pr, c-Pr], [RC5398; F, H, H, Me, c-Pr, Bu], [ RC5399; F, H, H, Me, c-Pr, i-Bu], [RC5400; F, H, H, Me, c-Pr, t-Bu],

[RC5401; F, H, H, Me, c-Pr, c-PrCH ₂ ], [RC5402; F, H, H, Me, c-Pr, Ph], [RC5403; F, H, H, Me, c-Pr, Bn], [RC5404; F, H, H, Me, c-Pr, CF ₃ ], [RC5405; F, H, H, Me, c-Pr, CF ₃ CH ₂ ], [RC5406; F, H, H, Me, c-Pr, CF ₃ CF ₂ ], [RC5407; F, H, H, Me, c-Pr, CF ₂ H], [RC5408; F, H, H, Me, c -Pr, CF ₂ HCF ₂ ], [RC5409; F, H, Me, Me, c-Pr, Me], [RC5410; F, H, Me, Me, c-Pr, Et], [RC5411; F, H, Me, Me, c-Pr, Pr], [RC5412; F, H, Me, Me, c-Pr, i-Pr], [RC5413; F, H, Me, Me, c-Pr, c- Pr], [RC5414; F, H, Me, Me, c-Pr, Bu], [RC5415; F, H, Me, Me, c-Pr, i-Bu], [RC5416; F, H, Me, Me, c-Pr, t-Bu], [RC5417; F, H, Me, Me, c-Pr, c-PrCH ₂ ], [RC5418; F, H, Me, Me, c-Pr, Ph], [RC5419; F, H, Me, Me, c-Pr, Bn], [RC5420; F, H, Me, Me, c-Pr, CF ₃ ], [RC5421; F, H, Me, Me, c- Pr, CF ₃ CH ₂ ], [RC5422; F, H, Me, Me, c-Pr, CF ₃ CF ₂ ], [RC5423; F, H, Me, Me, c-Pr, CF ₂ H], [ RC5424; F, H, Me, Me, c-Pr, CF ₂ HCF ₂ ], [RC5425; F, H, Me, Et, c-Pr, Me], [RC5426; F, H, Me, Et, c -Pr, Et], [RC5427; F, H, Me, Et, c-Pr, Pr], [RC5428; F, H, Me, Et, c-Pr, i-Pr], [RC5429; F, H , Me, Et, c-Pr, c-Pr], [RC5430; F, H, Me, Et, c-Pr, Bu], [RC5431; F, H, Me, Et, c-Pr, i-Bu ], [RC5432; F, H, Me, Et, c-Pr, t-Bu], [RC5433; F, H, Me, Et, c-Pr, c-PrCH ₂ ], [RC5434; F, H, Me, E t, c-Pr, Ph], [RC5435; F, H, Me, Et, c-Pr, Bn], [RC5436; F, H, Me, Et, c-Pr, CF ₃ ], [RC5437; F , H, Me, Et, c-Pr, CF ₃ CH ₂ ], [RC5438; F, H, Me, Et, c-Pr, CF ₃ CF ₂ ], [RC5439; F, H, Me, Et, c -Pr, CF ₂ H], [RC5440; F, H, Me, Et, c-Pr, CF ₂ HCF ₂ ], [RC5441; F, H, Me, F, c-Pr, Me], [RC5442; F, H, Me, F, c-Pr, Et], [RC5443; F, H, Me, F, c-Pr, Pr], [RC5444; F, H, Me, F, c-Pr, i- Pr], [RC5445; F, H, Me, F, c-Pr, c-Pr], [RC5446; F, H, Me, F, c-Pr, Bu], [RC5447; F, H, Me, F, c-Pr, i-Bu], [RC5448; F, H, Me, F, c-Pr, t-Bu], [RC5449; F, H, Me, F, c-Pr, c-PrCH ₂ ], [RC5450; F, H, Me, F, c-Pr, Ph], [RC5451; F, H, Me, F, c-Pr, Bn], [RC5452; F, H, Me, F, c -Pr, CF ₃ ], [RC5453; F, H, Me, F, c-Pr, CF ₃ CH ₂ ], [RC5454; F, H, Me, F, c-Pr, CF ₃ CF ₂ ], [ RC5455; F, H, Me, F, c-Pr, CF ₂ H], [RC5456; F, H, Me, F, c-Pr, CF ₂ HCF ₂ ], [RC5457; F, H, Me, Cl , c-Pr, Me], [RC5458; F, H, Me, Cl, c-Pr, Et], [RC5459; F, H, Me, Cl, c-Pr, Pr], [RC5460; F, H , Me, Cl, c-Pr, i-Pr], [RC5461; F, H, Me, Cl, c-Pr, c-Pr], [RC5462; F, H, Me, Cl, c-Pr, Bu ], [RC5463; F, H, Me, Cl, c-Pr, i-Bu], [RC5464; F, H, Me, Cl, c-Pr, t-Bu], [RC5465; F, H, Me , Cl, c-Pr, c-PrCH ₂ ], [RC5466; F, H, Me, Cl, c-Pr, Ph], [RC5467; F, H, Me, Cl, c-Pr, Bn], [ RC5468; F, H, Me, Cl, c- Pr, CF ₃ ], [RC5469; F, H, Me, Cl, c-Pr, CF ₃ CH ₂ ], [RC5470; F, H, Me, Cl, c-Pr, CF ₃ CF ₂ ], [RC5471 ; F, H, Me, Cl, c-Pr, CF ₂ H], [RC5472; F, H, Me, Cl, c-Pr, CF ₂ HCF ₂ ], [RC5473; F, H, Et, H, c-Pr, Me], [RC5474; F, H, Et, H, c-Pr, Et], [RC5475; F, H, Et, H, c-Pr, Pr], [RC5476; F, H, Et, H, c-Pr, i-Pr], [RC5477; F, H, Et, H, c-Pr, c-Pr], [RC5478; F, H, Et, H, c-Pr, Bu] , [RC5479; F, H, Et, H, c-Pr, i-Bu], [RC5480; F, H, Et, H, c-Pr, t-Bu], [RC5481; F, H, Et, H, c-Pr, c-PrCH ₂ ], [RC5482; F, H, Et, H, c-Pr, Ph], [RC5483; F, H, Et, H, c-Pr, Bn], [RC5484 ; F, H, Et, H, c-Pr, CF ₃ ], [RC5485; F, H, Et, H, c-Pr, CF ₃ CH ₂ ], [RC5486; F, H, Et, H, c -Pr, CF ₃ CF ₂ ], [RC5487; F, H, Et, H, c-Pr, CF ₂ H], [RC5488; F, H, Et, H, c-Pr, CF ₂ HCF ₂ ], [RC5489; F, H, Et, F, c-Pr, Me], [RC5490; F, H, Et, F, c-Pr, Et], [RC5491; F, H, Et, F, c-Pr , Pr], [RC5492; F, H, Et, F, c-Pr, i-Pr], [RC5493; F, H, Et, F, c-Pr, c-Pr], [RC5494; F, H , Et, F, c-Pr, Bu], [RC5495; F, H, Et, F, c-Pr, i-Bu], [RC5496; F, H, Et, F, c-Pr, t-Bu ], [RC5497; F, H, Et, F, c-Pr, c-PrCH ₂ ], [RC5498; F, H, Et, F, c-Pr, Ph], [RC5499; F, H, Et, F, c-Pr, Bn], [RC5500; F, H, Et, F, c-Pr, CF ₃ ], [RC5501; F, H, Et, F, c-Pr, CF ₃ CH ₂ ], [ RC5502; F, H, Et, F, c-Pr, CF ₃ CF ₂ ], [RC5503; F, H, Et, F, c-Pr, CF ₂ H], [RC5504; F, H, Et, F, c-Pr, CF ₂ HCF ₂ ], [RC5505; F, H, Et, Cl, c-Pr, Me], [RC5506; F, H, Et, Cl, c-Pr, Et], [RC5507; F, H, Et, Cl, c-Pr, Pr], [ RC5508; F, H, Et, Cl, c-Pr, i-Pr], [RC5509; F, H, Et, Cl, c-Pr, c-Pr], [RC5510; F, H, Et, Cl, c-Pr, Bu], [RC5511; F, H, Et, Cl, c-Pr, i-Bu], [RC5512; F, H, Et, Cl, c-Pr, t-Bu], [RC5513; F, H, Et, Cl, c-Pr, c-PrCH ₂ ], [RC5514; F, H, Et, Cl, c-Pr, Ph], [RC5515; F, H, Et, Cl, c-Pr , Bn], [RC5516; F, H, Et, Cl, c-Pr, CF ₃ ], [RC5517; F, H, Et, Cl, c-Pr, CF ₃ CH ₂ ], [RC5518; F, H , Et, Cl, c-Pr, CF ₃ CF ₂ ], [RC5519; F, H, Et, Cl, c-Pr, CF ₂ H], [RC5520; F, H, Et, Cl, c-Pr, CF ₂ HCF ₂ ], [RC5521; F, H, F, H, c-Pr, Me], [RC5522; F, H, F, H, c-Pr, Et], [RC5523; F, H, F , H, c-Pr, Pr], [RC5524; F, H, F, H, c-Pr, i-Pr], [RC5525; F, H, F, H, c-Pr, c-Pr], [RC5526; F, H, F, H, c-Pr, Bu], [RC5527; F, H, F, H, c-Pr, i-Bu], [RC5528; F, H, F, H, c -Pr, t-Bu], [RC5529; F, H, F, H, c-Pr, c-PrCH ₂ ], [RC5530; F, H, F, H, c-Pr, Ph], [RC5531; F, H, F, H, c-Pr, Bn], [RC5532; F, H, F, H, c-Pr, CF ₃ ], [RC5533; F, H, F, H, c-Pr, CF ₃ CH ₂ ], [RC5534; F, H, F, H, c-Pr, CF ₃ CF ₂ ], [RC5535; F, H, F, H, c-Pr, CF ₂ H], [RC5536; F , H, F, H, c-Pr, CF ₂ HCF ₂ ], [ RC5537; F, H, F, F, c-Pr, Me], [RC5538; F, H, F, F, c-Pr, Et], [RC5539; F, H, F, F, c-Pr, Pr], [RC5540; F, H, F, F, c-Pr, i-Pr], [RC5541; F, H, F, F, c-Pr, c-Pr], [RC5542; F, H, F, F, c-Pr, Bu], [RC5543; F, H, F, F, c-Pr, i-Bu], [RC5544; F, H, F, F, c-Pr, t-Bu] , [RC5545; F, H, F, F, c-Pr, c-PrCH ₂ ], [RC5546; F, H, F, F, c-Pr, Ph], [RC5547; F, H, F, F , c-Pr, Bn], [RC5548; F, H, F, F, c-Pr, CF ₃ ], [RC5549; F, H, F, F, c-Pr, CF ₃ CH ₂ ], [RC5550 ; F, H, F, F, c-Pr, CF ₃ CF ₂ ], [RC5551; F, H, F, F, c-Pr, CF ₂ H], [RC5552; F, H, F, F, c-Pr, CF ₂ HCF ₂ ], [RC5553; F, H, F, Cl, c-Pr, Me], [RC5554; F, H, F, Cl, c-Pr, Et], [RC5555; F , H, F, Cl, c-Pr, Pr], [RC5556; F, H, F, Cl, c-Pr, i-Pr], [RC5557; F, H, F, Cl, c-Pr, c -Pr], [RC5558; F, H, F, Cl, c-Pr, Bu], [RC5559; F, H, F, Cl, c-Pr, i-Bu], [RC5560; F, H, F , Cl, c-Pr, t-Bu], [RC5561; F, H, F, Cl, c-Pr, c-PrCH ₂ ], [RC5562; F, H, F, Cl, c-Pr, Ph] , [RC5563; F, H, F, Cl, c-Pr, Bn], [RC5564; F, H, F, Cl, c-Pr, CF ₃ ], [RC5565; F, H, F, Cl, c -Pr, CF ₃ CH ₂ ], [RC5566; F, H, F, Cl, c-Pr, CF ₃ CF ₂ ], [RC5567; F, H, F, Cl, c-Pr, CF ₂ H], [RC5568; F, H, F, Cl, c-Pr, CF ₂ HCF ₂ ], [RC5569; F, H, Cl, H, c-Pr, Me], [RC5570; F, H, Cl, H, c-Pr, Et], [RC5571; F, H, Cl, H, c-Pr, Pr], [RC5572; F, H, C l, H, c-Pr, i-Pr], [RC5573; F, H, Cl, H, c-Pr, c-Pr], [RC5574; F, H, Cl, H, c-Pr, Bu] , [RC5575; F, H, Cl, H, c-Pr, i-Bu], [RC5576; F, H, Cl, H, c-Pr, t-Bu], [RC5577; F, H, Cl, H, c-Pr, c-PrCH ₂ ], [RC5578; F, H, Cl, H, c-Pr, Ph], [RC5579; F, H, Cl, H, c-Pr, Bn], [RC5580 ; F, H, Cl, H, c-Pr, CF ₃ ], [RC5581; F, H, Cl, H, c-Pr, CF ₃ CH ₂ ], [RC5582; F, H, Cl, H, c -Pr, CF ₃ CF ₂ ], [RC5583; F, H, Cl, H, c-Pr, CF ₂ H], [RC5584; F, H, Cl, H, c-Pr, CF ₂ HCF ₂ ], [RC5585; F, H, Cl, Cl, c-Pr, Me], [RC5586; F, H, Cl, Cl, c-Pr, Et], [RC5587; F, H, Cl, Cl, c-Pr , Pr], [RC5588; F, H, Cl, Cl, c-Pr, i-Pr], [RC5589; F, H, Cl, Cl, c-Pr, c-Pr], [RC5590; F, H , Cl, Cl, c-Pr, Bu], [RC5591; F, H, Cl, Cl, c-Pr, i-Bu], [RC5592; F, H, Cl, Cl, c-Pr, t-Bu ], [RC5593; F, H, Cl, Cl, c-Pr, c-PrCH ₂ ], [RC5594; F, H, Cl, Cl, c-Pr, Ph], [RC5595; F, H, Cl, Cl, c-Pr, Bn], [RC5596; F, H, Cl, Cl, c-Pr, CF ₃ ], [RC5597; F, H, Cl, Cl, c-Pr, CF ₃ CH ₂ ], [ RC5598; F, H, Cl, Cl, c-Pr, CF ₃ CF ₂ ], [RC5599; F, H, Cl, Cl, c-Pr, CF ₂ H], [RC5600; F, H, Cl, Cl , c-Pr, CF ₂ HCF ₂ ],

[RC5601; F, H, H, H, i-Bu, Me], [RC5602; F, H, H, H, i-Bu, Et], [RC5603; F, H, H, H, i-Bu , Pr], [RC5604; F, H, H, H, i-Bu, i-Pr], [RC5605; F, H, H, H, i-Bu, c-Pr], [RC5606; F, H , H, H, i-Bu, Bu], [RC5607; F, H, H, H, i-Bu, i-Bu], [RC5608; F, H, H, H, i-Bu, t-Bu ], [RC5609; F, H, H, H, i-Bu, c-PrCH ₂ ], [RC5610; F, H, H, H, i-Bu, Ph], [RC5611; F, H, H, H, i-Bu, Bn], [RC5612; F, H, H, H, i-Bu, CF ₃ ], [RC5613; F, H, H, H, i-Bu, CF ₃ CH ₂ ], [ RC5614; F, H, H, H, i-Bu, CF ₃ CF ₂ ], [RC5615; F, H, H, H, i-Bu, CF ₂ H], [RC5616; F, H, H, H , i-Bu, CF ₂ HCF ₂ ], [RC5617; F, H, H, Me, i-Bu, Me], [RC5618; F, H, H, Me, i-Bu, Et], [RC5619; F, H, H, Me, i-Bu, Pr], [RC5620; F, H, H, Me, i-Bu, i-Pr], [RC5621; F, H, H, Me, i-Bu, c-Pr], [RC5622; F, H, H, Me, i-Bu, Bu], [RC5623; F, H, H, Me, i-Bu, i-Bu], [RC5624; F, H, H, Me, i-Bu, t-Bu], [RC5625; F, H, H, Me, i-Bu, c-PrCH ₂ ], [RC5626; F, H, H, Me, i-Bu, Ph ], [RC5627; F, H, H, Me, i-Bu, Bn], [RC5628; F, H, H, Me, i-Bu, CF ₃ ], [RC5629; F, H, H, Me, i-Bu, CF ₃ CH ₂ ], [RC5630; F, H, H, Me, i-Bu, CF ₃ CF ₂ ], [RC5631; F, H, H, Me, i-Bu, CF ₂ H] , [RC5632; F, H, H, Me, i-Bu, CF ₂ HCF ₂ ], [RC5633; F, H, Me, Me, i-Bu, Me], [RC5634; F, H, Me, Me , i-Bu, Et], [RC5635; F, H, Me, Me, i-Bu, Pr], [RC5636; F , H, Me, Me, i-Bu, i-Pr], [RC5637; F, H, Me, Me, i-Bu, c-Pr], [RC5638; F, H, Me, Me, i-Bu , Bu], [RC5639; F, H, Me, Me, i-Bu, i-Bu], [RC5640; F, H, Me, Me, i-Bu, t-Bu], [RC5641; F, H , Me, Me, i-Bu, c-PrCH ₂ ], [RC5642; F, H, Me, Me, i-Bu, Ph], [RC5643; F, H, Me, Me, i-Bu, Bn] , [RC5644; F, H, Me, Me, i-Bu, CF ₃ ], [RC5645; F, H, Me, Me, i-Bu, CF ₃ CH ₂ ], [RC5646; F, H, Me, Me, i-Bu, CF ₃ CF ₂ ], [RC5647; F, H, Me, Me, i-Bu, CF ₂ H], [RC5648; F, H, Me, Me, i-Bu, CF ₂ HCF ₂ ], [RC5649; F, H, Me, Et, i-Bu, Me], [RC5650; F, H, Me, Et, i-Bu, Et], [RC5651; F, H, Me, Et, i-Bu, Pr], [RC5652; F, H, Me, Et, i-Bu, i-Pr], [RC5653; F, H, Me, Et, i-Bu, c-Pr], [RC5654; F, H, Me, Et, i-Bu, Bu], [RC5655; F, H, Me, Et, i-Bu, i-Bu], [RC5656; F, H, Me, Et, i-Bu, t-Bu], [RC5657; F, H, Me, Et, i-Bu, c-PrCH ₂ ], [RC5658; F, H, Me, Et, i-Bu, Ph], [RC5659; F, H , Me, Et, i-Bu, Bn], [RC5660; F, H, Me, Et, i-Bu, CF ₃ ], [RC5661; F, H, Me, Et, i-Bu, CF ₃ CH ₂ ], [RC5662; F, H, Me, Et, i-Bu, CF ₃ CF ₂ ], [RC5663; F, H, Me, Et, i-Bu, CF ₂ H], [RC5664; F, H, Me, Et, i-Bu, CF ₂ HCF ₂ ], [RC5665; F, H, Me, F, i-Bu, Me], [RC5666; F, H, Me, F, i-Bu, Et], [RC5667; F, H, Me, F, i-Bu, Pr], [RC5668; F, H, Me, F, i-Bu, i-Pr], [RC5669; F, H, Me, F, i -Bu, c-Pr ], [RC5670; F, H, Me, F, i-Bu, Bu], [RC5671; F, H, Me, F, i-Bu, i-Bu], [RC5672; F, H, Me, F , i-Bu, t-Bu], [RC5673; F, H, Me, F, i-Bu, c-PrCH ₂ ], [RC5674; F, H, Me, F, i-Bu, Ph], [ RC5675; F, H, Me, F, i-Bu, Bn], [RC5676; F, H, Me, F, i-Bu, CF ₃ ], [RC5677; F, H, Me, F, i-Bu , CF ₃ CH ₂ ], [RC5678; F, H, Me, F, i-Bu, CF ₃ CF ₂ ], [RC5679; F, H, Me, F, i-Bu, CF ₂ H], [RC5680 ; F, H, Me, F, i-Bu, CF ₂ HCF ₂ ], [RC5681; F, H, Me, Cl, i-Bu, Me], [RC5682; F, H, Me, Cl, i- Bu, Et], [RC5683; F, H, Me, Cl, i-Bu, Pr], [RC5684; F, H, Me, Cl, i-Bu, i-Pr], [RC5685; F, H, Me, Cl, i-Bu, c-Pr], [RC5686; F, H, Me, Cl, i-Bu, Bu], [RC5687; F, H, Me, Cl, i-Bu, i-Bu] , [RC5688; F, H, Me, Cl, i-Bu, t-Bu], [RC5689; F, H, Me, Cl, i-Bu, c-PrCH ₂ ], [RC5690; F, H, Me , Cl, i-Bu, Ph], [RC5691; F, H, Me, Cl, i-Bu, Bn], [RC5692; F, H, Me, Cl, i-Bu, CF ₃ ], [RC5693; F, H, Me, Cl, i-Bu, CF ₃ CH ₂ ], [RC5694; F, H, Me, Cl, i-Bu, CF ₃ CF ₂ ], [RC5695; F, H, Me, Cl, i-Bu, CF ₂ H], [RC5696; F, H, Me, Cl, i-Bu, CF ₂ HCF ₂ ], [RC5697; F, H, Et, H, i-Bu, Me], [RC5698 ; F, H, Et, H, i-Bu, Et], [RC5699; F, H, Et, H, i-Bu, Pr], [RC5700; F, H, Et, H, i-Bu, i -Pr], [RC5701; F, H, Et, H, i-Bu, c-Pr], [RC5702; F, H, Et, H, i-Bu, Bu], [RC5703; F, H, Et , H, i-Bu, i-Bu], [R C5704; F, H, Et, H, i-Bu, t-Bu], [RC5705; F, H, Et, H, i-Bu, c-PrCH ₂ ], [RC5706; F, H, Et, H , i-Bu, Ph], [RC5707; F, H, Et, H, i-Bu, Bn], [RC5708; F, H, Et, H, i-Bu, CF ₃ ], [RC5709; F, H, Et, H, i-Bu, CF ₃ CH ₂ ], [RC5710; F, H, Et, H, i-Bu, CF ₃ CF ₂ ], [RC5711; F, H, Et, H, i- Bu, CF ₂ H], [RC5712; F, H, Et, H, i-Bu, CF ₂ HCF ₂ ], [RC5713; F, H, Et, F, i-Bu, Me], [RC5714; F , H, Et, F, i-Bu, Et], [RC5715; F, H, Et, F, i-Bu, Pr], [RC5716; F, H, Et, F, i-Bu, i-Pr ], [RC5717; F, H, Et, F, i-Bu, c-Pr], [RC5718; F, H, Et, F, i-Bu, Bu], [RC5719; F, H, Et, F , i-Bu, i-Bu], [RC5720; F, H, Et, F, i-Bu, t-Bu], [RC5721; F, H, Et, F, i-Bu, c-PrCH ₂ ] , [RC5722; F, H, Et, F, i-Bu, Ph], [RC5723; F, H, Et, F, i-Bu, Bn], [RC5724; F, H, Et, F, i- Bu, CF ₃ ], [RC5725; F, H, Et, F, i-Bu, CF ₃ CH ₂ ], [RC5726; F, H, Et, F, i-Bu, CF ₃ CF ₂ ], [RC5727 ; F, H, Et, F, i-Bu, CF ₂ H], [RC5728; F, H, Et, F, i-Bu, CF ₂ HCF ₂ ], [RC5729; F, H, Et, Cl, i-Bu, Me], [RC5730; F, H, Et, Cl, i-Bu, Et], [RC5731; F, H, Et, Cl, i-Bu, Pr], [RC5732; F, H, Et, Cl, i-Bu, i-Pr], [RC5733; F, H, Et, Cl, i-Bu, c-Pr], [RC5734; F, H, Et, Cl, i-Bu, Bu] , [RC5735; F, H, Et, Cl, i-Bu, i-Bu], [RC5736; F, H, Et, Cl, i-Bu, t-Bu], [RC5737; F, H, Et, Cl, i-Bu, c-PrCH ₂ ], [RC573 8; F, H, Et, Cl, i-Bu, Ph], [RC5739; F, H, Et, Cl, i-Bu, Bn], [RC5740; F, H, Et, Cl, i-Bu, CF ₃ ], [RC5741; F, H, Et, Cl, i-Bu, CF ₃ CH ₂ ], [RC5742; F, H, Et, Cl, i-Bu, CF ₃ CF ₂ ], [RC5743; F , H, Et, Cl, i-Bu, CF ₂ H], [RC5744; F, H, Et, Cl, i-Bu, CF ₂ HCF ₂ ], [RC5745; F, H, F, H, i- Bu, Me], [RC5746; F, H, F, H, i-Bu, Et], [RC5747; F, H, F, H, i-Bu, Pr], [RC5748; F, H, F, H, i-Bu, i-Pr], [RC5749; F, H, F, H, i-Bu, c-Pr], [RC5750; F, H, F, H, i-Bu, Bu], [ RC5751; F, H, F, H, i-Bu, i-Bu], [RC5752; F, H, F, H, i-Bu, t-Bu], [RC5753; F, H, F, H, i-Bu, c-PrCH ₂ ], [RC5754; F, H, F, H, i-Bu, Ph], [RC5755; F, H, F, H, i-Bu, Bn], [RC5756; F , H, F, H, i-Bu, CF ₃ ], [RC5757; F, H, F, H, i-Bu, CF ₃ CH ₂ ], [RC5758; F, H, F, H, i-Bu , CF ₃ CF ₂ ], [RC5759; F, H, F, H, i-Bu, CF ₂ H], [RC5760; F, H, F, H, i-Bu, CF ₂ HCF ₂ ], [RC5761 ; F, H, F, F, i-Bu, Me], [RC5762; F, H, F, F, i-Bu, Et], [RC5763; F, H, F, F, i-Bu, Pr ], [RC5764; F, H, F, F, i-Bu, i-Pr], [RC5765; F, H, F, F, i-Bu, c-Pr], [RC5766; F, H, F , F, i-Bu, Bu], [RC5767; F, H, F, F, i-Bu, i-Bu], [RC5768; F, H, F, F, i-Bu, t-Bu], [RC5769; F, H, F, F, i-Bu, c-PrCH ₂ ], [RC5770; F, H, F, F, i-Bu, Ph], [RC5771; F, H, F, F, i-Bu, Bn], [RC5772; F, H, F, F, i-Bu, CF ₃ ], [RC5773; F, H, F, F, i-Bu , CF ₃ CH ₂ ], [RC5774; F, H, F, F, i-Bu, CF ₃ CF ₂ ], [RC5775; F, H, F, F, i-Bu, CF ₂ H], [RC5776 ; F, H, F, F, i-Bu, CF ₂ HCF ₂ ], [RC5777; F, H, F, Cl, i-Bu, Me], [RC5778; F, H, F, Cl, i- Bu, Et], [RC5779; F, H, F, Cl, i-Bu, Pr], [RC5780; F, H, F, Cl, i-Bu, i-Pr], [RC5781; F, H, F, Cl, i-Bu, c-Pr], [RC5782; F, H, F, Cl, i-Bu, Bu], [RC5783; F, H, F, Cl, i-Bu, i-Bu] , [RC5784; F, H, F, Cl, i-Bu, t-Bu], [RC5785; F, H, F, Cl, i-Bu, c-PrCH ₂ ], [RC5786; F, H, F , Cl, i-Bu, Ph], [RC5787; F, H, F, Cl, i-Bu, Bn], [RC5788; F, H, F, Cl, i-Bu, CF ₃ ], [RC5789; F, H, F, Cl, i-Bu, CF ₃ CH ₂ ], [RC5790; F, H, F, Cl, i-Bu, CF ₃ CF ₂ ], [RC5791; F, H, F, Cl, i-Bu, CF ₂ H], [RC5792; F, H, F, Cl, i-Bu, CF ₂ HCF ₂ ], [RC5793; F, H, Cl, H, i-Bu, Me], [RC5794 ; F, H, Cl, H, i-Bu, Et], [RC5795; F, H, Cl, H, i-Bu, Pr], [RC5796; F, H, Cl, H, i-Bu, i -Pr], [RC5797; F, H, Cl, H, i-Bu, c-Pr], [RC5798; F, H, Cl, H, i-Bu, Bu], [RC5799; F, H, Cl , H, i-Bu, i-Bu], [RC5800; F, H, Cl, H, i-Bu, t-Bu],

[RC5801; F, H, Cl, H, i-Bu, c-PrCH ₂ ], [RC5802; F, H, Cl, H, i-Bu, Ph], [RC5803; F, H, Cl, H, i-Bu, Bn], [RC5804; F, H, Cl, H, i-Bu, CF ₃ ], [RC5805; F, H, Cl, H, i-Bu, CF ₃ CH ₂ ], [RC5806; F, H, Cl, H, i-Bu, CF ₃ CF ₂ ], [RC5807; F, H, Cl, H, i-Bu, CF ₂ H], [RC5808; F, H, Cl, H, i -Bu, CF ₂ HCF ₂ ], [RC5809; F, H, Cl, Cl, i-Bu, Me], [RC5810; F, H, Cl, Cl, i-Bu, Et], [RC5811; F, H, Cl, Cl, i-Bu, Pr], [RC5812; F, H, Cl, Cl, i-Bu, i-Pr], [RC5813; F, H, Cl, Cl, i-Bu, c- Pr], [RC5814; F, H, Cl, Cl, i-Bu, Bu], [RC5815; F, H, Cl, Cl, i-Bu, i-Bu], [RC5816; F, H, Cl, Cl, i-Bu, t-Bu], [RC5817; F, H, Cl, Cl, i-Bu, c-PrCH ₂ ], [RC5818; F, H, Cl, Cl, i-Bu, Ph], [RC5819; F, H, Cl, Cl, i-Bu, Bn], [RC5820; F, H, Cl, Cl, i-Bu, CF ₃ ], [RC5821; F, H, Cl, Cl, i- Bu, CF ₃ CH ₂ ], [RC5822; F, H, Cl, Cl, i-Bu, CF ₃ CF ₂ ], [RC5823; F, H, Cl, Cl, i-Bu, CF ₂ H], [ RC5824; F, H, Cl, Cl, i-Bu, CF ₂ HCF ₂ ], [RC5825; F, H, H, H, t-Bu, Me], [RC5826; F, H, H, H, t -Bu, Et], [RC5827; F, H, H, H, t-Bu, Pr], [RC5828; F, H, H, H, t-Bu, i-Pr], [RC5829; F, H , H, H, t-Bu, c-Pr], [RC5830; F, H, H, H, t-Bu, Bu], [RC5831; F, H, H, H, t-Bu, i-Bu ], [RC5832; F, H, H, H, t-Bu, t-Bu], [RC5833; F, H, H, H, t-Bu, c-PrCH ₂ ], [RC5834; F, H, H, H, t-Bu, Ph], [RC5835; F , H, H, H, t-Bu, Bn], [RC5836; F, H, H, H, t-Bu, CF ₃ ], [RC5837; F, H, H, H, t-Bu, CF ₃ CH ₂ ], [RC5838; F, H, H, H, t-Bu, CF ₃ CF ₂ ], [RC5839; F, H, H, H, t-Bu, CF ₂ H], [RC5840; F, H, H, H, t-Bu, CF ₂ HCF ₂ ], [RC5841; F, H, H, Me, t-Bu, Me], [RC5842; F, H, H, Me, t-Bu, Et ], [RC5843; F, H, H, Me, t-Bu, Pr], [RC5844; F, H, H, Me, t-Bu, i-Pr], [RC5845; F, H, H, Me , t-Bu, c-Pr], [RC5846; F, H, H, Me, t-Bu, Bu], [RC5847; F, H, H, Me, t-Bu, i-Bu], [RC5848 ; F, H, H, Me, t-Bu, t-Bu], [RC5849; F, H, H, Me, t-Bu, c-PrCH ₂ ], [RC5850; F, H, H, Me, t-Bu, Ph], [RC5851; F, H, H, Me, t-Bu, Bn], [RC5852; F, H, H, Me, t-Bu, CF ₃ ], [RC5853; F, H , H, Me, t-Bu, CF ₃ CH ₂ ], [RC5854; F, H, H, Me, t-Bu, CF ₃ CF ₂ ], [RC5855; F, H, H, Me, t-Bu , CF ₂ H], [RC5856; F, H, H, Me, t-Bu, CF ₂ HCF ₂ ], [RC5857; F, H, Me, Me, t-Bu, Me], [RC5858; F, H, Me, Me, t-Bu, Et], [RC5859; F, H, Me, Me, t-Bu, Pr], [RC5860; F, H, Me, Me, t-Bu, i-Pr] , [RC5861; F, H, Me, Me, t-Bu, c-Pr], [RC5862; F, H, Me, Me, t-Bu, Bu], [RC5863; F, H, Me, Me, t-Bu, i-Bu], [RC5864; F, H, Me, Me, t-Bu, t-Bu], [RC5865; F, H, Me, Me, t-Bu, c-PrCH ₂ ], [RC5866; F, H, Me, Me, t-Bu, Ph], [RC5867; F, H, Me, Me, t-Bu, Bn], [RC5868; F, H, Me, Me, t-Bu , CF ₃ ], [RC5869; F, H, Me, Me, t-Bu , CF ₃ CH ₂ ], [RC5870; F, H, Me, Me, t-Bu, CF ₃ CF ₂ ], [RC5871; F, H, Me, Me, t-Bu, CF ₂ H], [RC5872 ; F, H, Me, Me, t-Bu, CF ₂ HCF ₂ ], [RC5873; F, H, Me, Et, t-Bu, Me], [RC5874; F, H, Me, Et, t- Bu, Et], [RC5875; F, H, Me, Et, t-Bu, Pr], [RC5876; F, H, Me, Et, t-Bu, i-Pr], [RC5877; F, H, Me, Et, t-Bu, c-Pr], [RC5878; F, H, Me, Et, t-Bu, Bu], [RC5879; F, H, Me, Et, t-Bu, i-Bu] , [RC5880; F, H, Me, Et, t-Bu, t-Bu], [RC5881; F, H, Me, Et, t-Bu, c-PrCH ₂ ], [RC5882; F, H, Me , Et, t-Bu, Ph], [RC5883; F, H, Me, Et, t-Bu, Bn], [RC5884; F, H, Me, Et, t-Bu, CF ₃ ], [RC5885; F, H, Me, Et, t-Bu, CF ₃ CH ₂ ], [RC5886; F, H, Me, Et, t-Bu, CF ₃ CF ₂ ], [RC5887; F, H, Me, Et, t-Bu, CF ₂ H], [RC5888; F, H, Me, Et, t-Bu, CF ₂ HCF ₂ ], [RC5889; F, H, Me, F, t-Bu, Me], [RC5890 ; F, H, Me, F, t-Bu, Et], [RC5891; F, H, Me, F, t-Bu, Pr], [RC5892; F, H, Me, F, t-Bu, i -Pr], [RC5893; F, H, Me, F, t-Bu, c-Pr], [RC5894; F, H, Me, F, t-Bu, Bu], [RC5895; F, H, Me , F, t-Bu, i-Bu], [RC5896; F, H, Me, F, t-Bu, t-Bu], [RC5897; F, H, Me, F, t-Bu, c-PrCH ₂ ], [RC5898; F, H, Me, F, t-Bu, Ph], [RC5899; F, H, Me, F, t-Bu, Bn], [RC5900; F, H, Me, F, t-Bu, CF ₃ ], [RC5901; F, H, Me, F, t-Bu, CF ₃ CH ₂ ], [RC5902; F, H, Me, F, t-Bu, CF ₃ CF ₂ ], [RC5903; F, H, Me, F, t-Bu, CF ₂ H], [RC5904; F, H, Me, F, t-Bu, CF ₂ HCF ₂ ], [RC5905; F, H, Me, Cl, t -Bu, Me], [RC5906; F, H, Me, Cl, t-Bu, Et], [RC5907; F, H, Me, Cl, t-Bu, Pr], [RC5908; F, H, Me , Cl, t-Bu, i-Pr], [RC5909; F, H, Me, Cl, t-Bu, c-Pr], [RC5910; F, H, Me, Cl, t-Bu, Bu], [RC5911; F, H, Me, Cl, t-Bu, i-Bu], [RC5912; F, H, Me, Cl, t-Bu, t-Bu], [RC5913; F, H, Me, Cl , t-Bu, c-PrCH ₂ ], [RC5914; F, H, Me, Cl, t-Bu, Ph], [RC5915; F, H, Me, Cl, t-Bu, Bn], [RC5916; F, H, Me, Cl, t-Bu, CF ₃ ], [RC5917; F, H, Me, Cl, t-Bu, CF ₃ CH ₂ ], [RC5918; F, H, Me, Cl, t- Bu, CF ₃ CF ₂ ], [RC5919; F, H, Me, Cl, t-Bu, CF ₂ H], [RC5920; F, H, Me, Cl, t-Bu, CF ₂ HCF ₂ ], [ RC5921; F, H, Et, H, t-Bu, Me], [RC5922; F, H, Et, H, t-Bu, Et], [RC5923; F, H, Et, H, t-Bu, Pr], [RC5924; F, H, Et, H, t-Bu, i-Pr], [RC5925; F, H, Et, H, t-Bu, c-Pr], [RC5926; F, H, Et, H, t-Bu, Bu], [RC5927; F, H, Et, H, t-Bu, i-Bu], [RC5928; F, H, Et, H, t-Bu, t-Bu] , [RC5929; F, H, Et, H, t-Bu, c-PrCH ₂ ], [RC5930; F, H, Et, H, t-Bu, Ph], [RC5931; F, H, Et, H , t-Bu, Bn], [RC5932; F, H, Et, H, t-Bu, CF ₃ ], [RC5933; F, H, Et, H, t-Bu, CF ₃ CH ₂ ], [RC5934 ; F, H, Et, H, t-Bu, CF ₃ CF ₂ ], [RC5935; F, H, Et, H, t-Bu, CF ₂ H], [RC5936; F, H, Et, H, t-Bu, CF ₂ HCF ₂ ], [ RC5937; F, H, Et, F, t-Bu, Me], [RC5938; F, H, Et, F, t-Bu, Et], [RC5939; F, H, Et, F, t-Bu, Pr], [RC5940; F, H, Et, F, t-Bu, i-Pr], [RC5941; F, H, Et, F, t-Bu, c-Pr], [RC5942; F, H, Et, F, t-Bu, Bu], [RC5943; F, H, Et, F, t-Bu, i-Bu], [RC5944; F, H, Et, F, t-Bu, t-Bu] , [RC5945; F, H, Et, F, t-Bu, c-PrCH ₂ ], [RC5946; F, H, Et, F, t-Bu, Ph], [RC5947; F, H, Et, F , t-Bu, Bn], [RC5948; F, H, Et, F, t-Bu, CF ₃ ], [RC5949; F, H, Et, F, t-Bu, CF ₃ CH ₂ ], [RC5950 ; F, H, Et, F, t-Bu, CF ₃ CF ₂ ], [RC5951; F, H, Et, F, t-Bu, CF ₂ H], [RC5952; F, H, Et, F, t-Bu, CF ₂ HCF ₂ ], [RC5953; F, H, Et, Cl, t-Bu, Me], [RC5954; F, H, Et, Cl, t-Bu, Et], [RC5955; F , H, Et, Cl, t-Bu, Pr], [RC5956; F, H, Et, Cl, t-Bu, i-Pr], [RC5957; F, H, Et, Cl, t-Bu, c -Pr], [RC5958; F, H, Et, Cl, t-Bu, Bu], [RC5959; F, H, Et, Cl, t-Bu, i-Bu], [RC5960; F, H, Et , Cl, t-Bu, t-Bu], [RC5961; F, H, Et, Cl, t-Bu, c-PrCH ₂ ], [RC5962; F, H, Et, Cl, t-Bu, Ph] , [RC5963; F, H, Et, Cl, t-Bu, Bn], [RC5964; F, H, Et, Cl, t-Bu, CF ₃ ], [RC5965; F, H, Et, Cl, t -Bu, CF ₃ CH ₂ ], [RC5966; F, H, Et, Cl, t-Bu, CF ₃ CF ₂ ], [RC5967; F, H, Et, Cl, t-Bu, CF ₂ H], [RC5968; F, H, Et, Cl, t-Bu, CF ₂ HCF ₂ ], [RC5969; F, H, F, H, t-Bu, Me], [RC5970; F, H, F, H, t-Bu, Et], [RC5971; F , H, F, H, t-Bu, Pr], [RC5972; F, H, F, H, t-Bu, i-Pr], [RC5973; F, H, F, H, t-Bu, c -Pr], [RC5974; F, H, F, H, t-Bu, Bu], [RC5975; F, H, F, H, t-Bu, i-Bu], [RC5976; F, H, F , H, t-Bu, t-Bu], [RC5977; F, H, F, H, t-Bu, c-PrCH ₂ ], [RC5978; F, H, F, H, t-Bu, Ph] , [RC5979; F, H, F, H, t-Bu, Bn], [RC5980; F, H, F, H, t-Bu, CF ₃ ], [RC5981; F, H, F, H, t -Bu, CF ₃ CH ₂ ], [RC5982; F, H, F, H, t-Bu, CF ₃ CF ₂ ], [RC5983; F, H, F, H, t-Bu, CF ₂ H], [RC5984; F, H, F, H, t-Bu, CF ₂ HCF ₂ ], [RC5985; F, H, F, F, t-Bu, Me], [RC5986; F, H, F, F, t-Bu, Et], [RC5987; F, H, F, F, t-Bu, Pr], [RC5988; F, H, F, F, t-Bu, i-Pr], [RC5989; F, H, F, F, t-Bu, c-Pr], [RC5990; F, H, F, F, t-Bu, Bu], [RC5991; F, H, F, F, t-Bu, i- Bu], [RC5992; F, H, F, F, t-Bu, t-Bu], [RC5993; F, H, F, F, t-Bu, c-PrCH ₂ ], [RC5994; F, H , F, F, t-Bu, Ph], [RC5995; F, H, F, F, t-Bu, Bn], [RC5996; F, H, F, F, t-Bu, CF ₃ ], [ RC5997; F, H, F, F, t-Bu, CF ₃ CH ₂ ], [RC5998; F, H, F, F, t-Bu, CF ₃ CF ₂ ], [RC5999; F, H, F, F, t-Bu, CF ₂ H], [RC6000; F, H, F, F, t-Bu, CF ₂ HCF ₂ ],

[RC6001; F, H, F, Cl, t-Bu, Me], [RC6002; F, H, F, Cl, t-Bu, Et], [RC6003; F, H, F, Cl, t-Bu , Pr], [RC6004; F, H, F, Cl, t-Bu, i-Pr], [RC6005; F, H, F, Cl, t-Bu, c-Pr], [RC6006; F, H , F, Cl, t-Bu, Bu], [RC6007; F, H, F, Cl, t-Bu, i-Bu], [RC6008; F, H, F, Cl, t-Bu, t-Bu ], [RC6009; F, H, F, Cl, t-Bu, c-PrCH ₂ ], [RC6010; F, H, F, Cl, t-Bu, Ph], [RC6011; F, H, F, Cl, t-Bu, Bn], [RC6012; F, H, F, Cl, t-Bu, CF ₃ ], [RC6013; F, H, F, Cl, t-Bu, CF ₃ CH ₂ ], [ RC6014; F, H, F, Cl, t-Bu, CF ₃ CF ₂ ], [RC6015; F, H, F, Cl, t-Bu, CF ₂ H], [RC6016; F, H, F, Cl , t-Bu, CF ₂ HCF ₂ ], [RC6017; F, H, Cl, H, t-Bu, Me], [RC6018; F, H, Cl, H, t-Bu, Et], [RC6019; F, H, Cl, H, t-Bu, Pr], [RC6020; F, H, Cl, H, t-Bu, i-Pr], [RC6021; F, H, Cl, H, t-Bu, c-Pr], [RC6022; F, H, Cl, H, t-Bu, Bu], [RC6023; F, H, Cl, H, t-Bu, i-Bu], [RC6024; F, H, Cl, H, t-Bu, t-Bu], [RC6025; F, H, Cl, H, t-Bu, c-PrCH ₂ ], [RC6026; F, H, Cl, H, t-Bu, Ph ], [RC6027; F, H, Cl, H, t-Bu, Bn], [RC6028; F, H, Cl, H, t-Bu, CF ₃ ], [RC6029; F, H, Cl, H, t-Bu, CF ₃ CH ₂ ], [RC6030; F, H, Cl, H, t-Bu, CF ₃ CF ₂ ], [RC6031; F, H, Cl, H, t-Bu, CF ₂ H] , [RC6032; F, H, Cl, H, t-Bu, CF ₂ HCF ₂ ], [RC6033; F, H, Cl, Cl, t-Bu, Me], [RC6034; F, H, Cl, Cl , t-Bu, Et], [RC6035; F, H, Cl, Cl, t- Bu, Pr], [RC6036; F, H, Cl, Cl, t-Bu, i-Pr], [RC6037; F, H, Cl, Cl, t-Bu, c-Pr], [RC6038; F, H, Cl, Cl, t-Bu, Bu], [RC6039; F, H, Cl, Cl, t-Bu, i-Bu], [RC6040; F, H, Cl, Cl, t-Bu, t- Bu], [RC6041; F, H, Cl, Cl, t-Bu, c-PrCH ₂ ], [RC6042; F, H, Cl, Cl, t-Bu, Ph], [RC6043; F, H, Cl , Cl, t-Bu, Bn], [RC6044; F, H, Cl, Cl, t-Bu, CF ₃ ], [RC6045; F, H, Cl, Cl, t-Bu, CF ₃ CH ₂ ], [RC6046; F, H, Cl, Cl, t-Bu, CF ₃ CF ₂ ], [RC6047; F, H, Cl, Cl, t-Bu, CF ₂ H], [RC6048; F, H, Cl, Cl, t-Bu, CF ₂ HCF ₂ ], [RC6049; F, H, H, H, CF ₂ H, Me], [RC6050; F, H, H, H, CF ₂ H, Et], [RC6051 ; F, H, H, H, CF ₂ H, Pr], [RC6052; F, H, H, H, CF ₂ H, i-Pr], [RC6053; F, H, H, H, CF ₂ H , c-Pr], [RC6054; F, H, H, H, CF ₂ H, Bu], [RC6055; F, H, H, H, CF ₂ H, i-Bu], [RC6056; F, H , H, H, CF ₂ H, t-Bu], [RC6057; F, H, H, H, CF ₂ H, c-PrCH ₂ ], [RC6058; F, H, H, H, CF ₂ H, Ph], [RC6059; F, H, H, H, CF ₂ H, Bn], [RC6060; F, H, H, H, CF ₂ H, CF ₃ ], [RC6061; F, H, H, H , CF ₂ H, CF ₃ CH ₂ ], [RC6062; F, H, H, H, CF ₂ H, CF ₃ CF ₂ ], [RC6063; F, H, H, H, CF ₂ H, CF ₂ H ], [RC6064; F, H, H, H, CF ₂ H, CF ₂ HCF ₂ ], [RC6065; F, H, H, Me, CF ₂ H, Me], [RC6066; F, H, H, Me, CF ₂ H, Et], [RC6067; F, H, H, Me, CF ₂ H, Pr], [RC6068; F, H, H, Me, CF ₂ H, i-Pr], [R C6069; F, H, H, Me, CF ₂ H, c-Pr], [RC6070; F, H, H, Me, CF ₂ H, Bu], [RC6071; F, H, H, Me, CF ₂ H, i-Bu], [RC6072; F, H, H, Me, CF ₂ H, t-Bu], [RC6073; F, H, H, Me, CF ₂ H, c-PrCH ₂ ], [RC6074 ; F, H, H, Me, CF ₂ H, Ph], [RC6075; F, H, H, Me, CF ₂ H, Bn], [RC6076; F, H, H, Me, CF ₂ H, CF ₃ ], [RC6077; F, H, H, Me, CF ₂ H, CF ₃ CH ₂ ], [RC6078; F, H, H, Me, CF ₂ H, CF ₃ CF ₂ ], [RC6079; F, H, H, Me, CF ₂ H, CF ₂ H], [RC6080; F, H, H, Me, CF ₂ H, CF ₂ HCF ₂ ], [RC6081; F, H, Me, Me, CF ₂ H , Me], [RC6082; F, H, Me, Me, CF ₂ H, Et], [RC6083; F, H, Me, Me, CF ₂ H, Pr], [RC6084; F, H, Me, Me , CF ₂ H, i-Pr], [RC6085; F, H, Me, Me, CF ₂ H, c-Pr], [RC6086; F, H, Me, Me, CF ₂ H, Bu], [RC6087 ; F, H, Me, Me, CF ₂ H, i-Bu], [RC6088; F, H, Me, Me, CF ₂ H, t-Bu], [RC6089; F, H, Me, Me, CF ₂ H, c-PrCH ₂ ], [RC6090; F, H, Me, Me, CF ₂ H, Ph], [RC6091; F, H, Me, Me, CF ₂ H, Bn], [RC6092; F, H, Me, Me, CF ₂ H, CF ₃ ], [RC6093; F, H, Me, Me, CF ₂ H, CF ₃ CH ₂ ], [RC6094; F, H, Me, Me, CF ₂ H, CF ₃ CF ₂ ], [RC6095; F, H, Me, Me, CF ₂ H, CF ₂ H], [RC6096; F, H, Me, Me, CF ₂ H, CF ₂ HCF ₂ ], [RC6097; F, H, Me, Et, CF ₂ H, Me], [RC6098; F, H, Me, Et, CF ₂ H, Et], [RC6099; F, H, Me, Et, CF ₂ H, Pr] , [RC6100; F, H, Me, Et, CF ₂ H, i-Pr], [RC6101; F, H, Me, Et, CF ₂ H, c-Pr], [RC6102; F, H, Me, Et, CF ₂ H, Bu], [RC6103; F, H, Me, Et, CF ₂ H, i-Bu], [RC6104; F, H, Me, Et, CF ₂ H, t-Bu], [RC6105; F, H, Me, Et, CF ₂ H, c-PrCH ₂ ], [RC6106; F, H, Me, Et, CF ₂ H, Ph], [RC6107; F, H, Me, Et, CF ₂ H, Bn], [RC6108; F, H, Me , Et, CF ₂ H, CF ₃ ], [RC6109; F, H, Me, Et, CF ₂ H, CF ₃ CH ₂ ], [RC6110; F, H, Me, Et, CF ₂ H, CF ₃ CF ₂ ], [RC6111; F, H, Me, Et, CF ₂ H, CF ₂ H], [RC6112; F, H, Me, Et, CF ₂ H, CF ₂ HCF ₂ ], [RC6113; F, H , Me, F, CF ₂ H, Me], [RC6114; F, H, Me, F, CF ₂ H, Et], [RC6115; F, H, Me, F, CF ₂ H, Pr], [RC6116 ; F, H, Me, F, CF ₂ H, i-Pr], [RC6117; F, H, Me, F, CF ₂ H, c-Pr], [RC6118; F, H, Me, F, CF ₂ H, Bu], [RC6119; F, H, Me, F, CF ₂ H, i-Bu], [RC6120; F, H, Me, F, CF ₂ H, t-Bu], [RC6121; F , H, Me, F, CF ₂ H, c-PrCH ₂ ], [RC6122; F, H, Me, F, CF ₂ H, Ph], [RC6123; F, H, Me, F, CF ₂ H, Bn], [RC6124; F, H, Me, F, CF ₂ H, CF ₃ ], [RC6125; F, H, Me, F, CF ₂ H, CF ₃ CH ₂ ], [RC6126; F, H, Me, F, CF ₂ H, CF ₃ CF ₂ ], [RC6127; F, H, Me, F, CF ₂ H, CF ₂ H], [RC6128; F, H, Me, F, CF ₂ H, CF ₂ HCF ₂ ], [RC6129; F, H, Me, Cl, CF ₂ H, Me], [RC6130; F, H, Me, Cl, CF ₂ H, Et], [RC6131; F, H, Me, Cl, CF ₂ H, Pr], [RC6132; F, H, Me, Cl , CF ₂ H, i-Pr], [RC6133; F, H, Me, Cl, CF ₂ H, c-Pr], [RC6134; F, H, Me, Cl, CF ₂ H, Bu], [RC6135 ; F, H, Me, Cl, CF ₂ H, i-Bu], [RC6136; F, H, Me, Cl, CF ₂ H, t-Bu], [RC6137; F, H, Me, Cl, CF ₂ H, c-PrCH ₂ ], [RC6138; F, H, Me, Cl, CF ₂ H, Ph], [RC6139; F, H, Me, Cl, CF ₂ H, Bn], [RC6140; F, H, Me, Cl, CF ₂ H, CF ₃ ], [RC6141; F, H, Me, Cl, CF ₂ H, CF ₃ CH ₂ ], [RC6142; F, H, Me, Cl, CF ₂ H, CF ₃ CF ₂ ], [RC6143; F, H, Me, Cl, CF ₂ H, CF ₂ H], [RC6144; F, H, Me, Cl, CF ₂ H, CF ₂ HCF ₂ ], [RC6145; F, H, Et, H, CF ₂ H, Me], [RC6146; F, H, Et, H, CF ₂ H, Et], [RC6147; F, H, Et, H, CF ₂ H, Pr] , [RC6148; F, H, Et, H, CF ₂ H, i-Pr], [RC6149; F, H, Et, H, CF ₂ H, c-Pr], [RC6150; F, H, Et, H, CF ₂ H, Bu], [RC6151; F, H, Et, H, CF ₂ H, i-Bu], [RC6152; F, H, Et, H, CF ₂ H, t-Bu], [ RC6153; F, H, Et, H, CF ₂ H, c-PrCH ₂ ], [RC6154; F, H, Et, H, CF ₂ H, Ph], [RC6155; F, H, Et, H, CF ₂ H, Bn], [RC6156; F, H, Et, H, CF ₂ H, CF ₃ ], [RC6157; F, H, Et, H, CF ₂ H, CF ₃ CH ₂ ], [RC6158; F , H, Et, H, CF ₂ H, CF ₃ CF ₂ ], [RC6159; F, H, Et, H, CF ₂ H, CF ₂ H], [RC6160; F, H, Et, H, CF ₂ H, CF ₂ HCF ₂ ], [RC6161; F, H, Et, F, CF ₂ H, Me], [RC6162; F, H, Et, F, CF ₂ H, Et], [RC6163; F, H , Et, F, CF ₂ H, Pr], [RC6164; F, H, Et , F, CF ₂ H, i-Pr], [RC6165; F, H, Et, F, CF ₂ H, c-Pr], [RC6166; F, H, Et, F, CF ₂ H, Bu], [RC6167; F, H, Et, F, CF ₂ H, i-Bu], [RC6168; F, H, Et, F, CF ₂ H, t-Bu], [RC6169; F, H, Et, F , CF ₂ H, c-PrCH ₂ ], [RC6170; F, H, Et, F, CF ₂ H, Ph], [RC6171; F, H, Et, F, CF ₂ H, Bn], [RC6172; F, H, Et, F, CF ₂ H, CF ₃ ], [RC6173; F, H, Et, F, CF ₂ H, CF ₃ CH ₂ ], [RC6174; F, H, Et, F, CF ₂ H, CF ₃ CF ₂ ], [RC6175; F, H, Et, F, CF ₂ H, CF ₂ H], [RC6176; F, H, Et, F, CF ₂ H, CF ₂ HCF ₂ ], [ RC6177; F, H, Et, Cl, CF ₂ H, Me], [RC6178; F, H, Et, Cl, CF ₂ H, Et], [RC6179; F, H, Et, Cl, CF ₂ H, Pr], [RC6180; F, H, Et, Cl, CF ₂ H, i-Pr], [RC6181; F, H, Et, Cl, CF ₂ H, c-Pr], [RC6182; F, H, Et, Cl, CF ₂ H, Bu], [RC6183; F, H, Et, Cl, CF ₂ H, i-Bu], [RC6184; F, H, Et, Cl, CF ₂ H, t-Bu] , [RC6185; F, H, Et, Cl, CF ₂ H, c-PrCH ₂ ], [RC6186; F, H, Et, Cl, CF ₂ H, Ph], [RC6187; F, H, Et, Cl , CF ₂ H, Bn], [RC6188; F, H, Et, Cl, CF ₂ H, CF ₃ ], [RC6189; F, H, Et, Cl, CF ₂ H, CF ₃ CH ₂ ], [RC6190 ; F, H, Et, Cl, CF ₂ H, CF ₃ CF ₂ ], [RC6191; F, H, Et, Cl, CF ₂ H, CF ₂ H], [RC6192; F, H, Et, Cl, CF ₂ H, CF ₂ HCF ₂ ], [RC6193; F, H, F, H, CF ₂ H, Me], [RC6194; F, H, F, H, CF ₂ H, Et], [RC6195; F , H, F, H, CF ₂ H, Pr], [RC6196; F, H , F, H, CF ₂ H, i-Pr], [RC6197; F, H, F, H, CF ₂ H, c-Pr], [RC6198; F, H, F, H, CF ₂ H, Bu ], [RC6199; F, H, F, H, CF ₂ H, i-Bu], [RC6200; F, H, F, H, CF ₂ H, t-Bu],

[RC6201; F, H, F, H, CF ₂ H, c-PrCH ₂ ], [RC6202; F, H, F, H, CF ₂ H, Ph], [RC6203; F, H, F, H, CF ₂ H, Bn], [RC6204; F, H, F, H, CF ₂ H, CF ₃ ], [RC6205; F, H, F, H, CF ₂ H, CF ₃ CH ₂ ], [RC6206; F, H, F, H, CF ₂ H, CF ₃ CF ₂ ], [RC6207; F, H, F, H, CF ₂ H, CF ₂ H], [RC6208; F, H, F, H, CF ₂ H, CF ₂ HCF ₂ ], [RC6209; F, H, F, F, CF ₂ H, Me], [RC6210; F, H, F, F, CF ₂ H, Et], [RC6211; F, H, F, F, CF ₂ H, Pr], [RC6212; F, H, F, F, CF ₂ H, i-Pr], [RC6213; F, H, F, F, CF ₂ H, c- Pr], [RC6214; F, H, F, F, CF ₂ H, Bu], [RC6215; F, H, F, F, CF ₂ H, i-Bu], [RC6216; F, H, F, F, CF ₂ H, t-Bu], [RC6217; F, H, F, F, CF ₂ H, c-PrCH ₂ ], [RC6218; F, H, F, F, CF ₂ H, Ph], [RC6219; F, H, F, F, CF ₂ H, Bn], [RC6220; F, H, F, F, CF ₂ H, CF ₃ ], [RC6221; F, H, F, F, CF ₂ H, CF ₃ CH ₂ ], [RC6222; F, H, F, F, CF ₂ H, CF ₃ CF ₂ ], [RC6223; F, H, F, F, CF ₂ H, CF ₂ H], [ RC6224; F, H, F, F, CF ₂ H, CF ₂ HCF ₂ ], [RC6225; F, H, F, Cl, CF ₂ H, Me], [RC6226; F, H, F, Cl, CF ₂ H, Et], [RC6227; F, H, F, Cl, CF ₂ H, Pr], [RC6228; F, H, F, Cl, CF ₂ H, i-Pr], [RC6229; F, H , F, Cl, CF ₂ H, c-Pr], [RC6230; F, H, F, Cl, CF ₂ H, Bu], [RC6231; F, H, F, Cl, CF ₂ H, i-Bu ], [RC6232; F, H, F, Cl, CF ₂ H, t-Bu], [RC6233; F, H, F, Cl, CF ₂ H, c-PrCH ₂ ] , [RC6234; F, H, F, Cl, CF ₂ H, Ph], [RC6235; F, H, F, Cl, CF ₂ H, Bn], [RC6236; F, H, F, Cl, CF ₂ H, CF ₃ ], [RC6237; F, H, F, Cl, CF ₂ H, CF ₃ CH ₂ ], [RC6238; F, H, F, Cl, CF ₂ H, CF ₃ CF ₂ ], [RC6239 ; F, H, F, Cl, CF ₂ H, CF ₂ H], [RC6240; F, H, F, Cl, CF ₂ H, CF ₂ HCF ₂ ], [RC6241; F, H, Cl, H, CF ₂ H, Me], [RC6242; F, H, Cl, H, CF ₂ H, Et], [RC6243; F, H, Cl, H, CF ₂ H, Pr], [RC6244; F, H, Cl, H, CF ₂ H, i-Pr], [RC6245; F, H, Cl, H, CF ₂ H, c-Pr], [RC6246; F, H, Cl, H, CF ₂ H, Bu] , [RC6247; F, H, Cl, H, CF ₂ H, i-Bu], [RC6248; F, H, Cl, H, CF ₂ H, t-Bu], [RC6249; F, H, Cl, H, CF ₂ H, c-PrCH ₂ ], [RC6250; F, H, Cl, H, CF ₂ H, Ph], [RC6251; F, H, Cl, H, CF ₂ H, Bn], [RC6252 ; F, H, Cl, H, CF ₂ H, CF ₃ ], [RC6253; F, H, Cl, H, CF ₂ H, CF ₃ CH ₂ ], [RC6254; F, H, Cl, H, CF ₂ H, CF ₃ CF ₂ ], [RC6255; F, H, Cl, H, CF ₂ H, CF ₂ H], [RC6256; F, H, Cl, H, CF ₂ H, CF ₂ HCF ₂ ], [RC6257; F, H, Cl, Cl, CF ₂ H, Me], [RC6258; F, H, Cl, Cl, CF ₂ H, Et], [RC6259; F, H, Cl, Cl, CF ₂ H , Pr], [RC6260; F, H, Cl, Cl, CF ₂ H, i-Pr], [RC6261; F, H, Cl, Cl, CF ₂ H, c-Pr], [RC6262; F, H , Cl, Cl, CF ₂ H, Bu], [RC6263; F, H, Cl, Cl, CF ₂ H, i-Bu], [RC6264; F, H, Cl, Cl, CF ₂ H, t-Bu ], [RC6265; F, H, Cl, Cl, CF ₂ H, c-PrCH ₂ ], [RC6266; F, H, Cl, Cl, CF ₂ H, Ph], [RC6267; F, H, Cl, Cl, CF ₂ H, Bn], [RC6268; F, H, Cl, Cl, CF ₂ H , CF ₃ ], [RC6269; F, H, Cl, Cl, CF ₂ H, CF ₃ CH ₂ ], [RC6270; F, H, Cl, Cl, CF ₂ H, CF ₃ CF ₂ ], [RC6271; F, H, Cl, Cl, CF ₂ H, CF ₂ H], [RC6272; F, H, Cl, Cl, CF ₂ H, CF ₂ HCF ₂ ], [RC6273; F, H, H, H, CF ₃ , Me], [RC6274; F, H, H, H, CF ₃ , Et], [RC6275; F, H, H, H, CF ₃ , Pr], [RC6276; F, H, H, H, CF ₃ , i-Pr], [RC6277; F, H, H, H, CF ₃ , c-Pr], [RC6278; F, H, H, H, CF ₃ , Bu], [RC6279; F, H , H, H, CF ₃ , i-Bu], [RC6280; F, H, H, H, CF ₃ , t-Bu], [RC6281; F, H, H, H, CF ₃ , c-PrCH ₂ ], [RC6282; F, H, H, H, CF ₃ , Ph], [RC6283; F, H, H, H, CF ₃ , Bn], [RC6284; F, H, H, H, CF ₃ , CF ₃ ], [RC6285; F, H, H, H, CF ₃ , CF ₃ CH ₂ ], [RC6286; F, H, H, H, CF ₃ , CF ₃ CF ₂ ], [RC6287; F, H , H, H, CF ₃ , CF ₂ H], [RC6288; F, H, H, H, CF ₃ , CF ₂ HCF ₂ ], [RC6289; F, H, H, Me, CF ₃ , Me], [RC6290; F, H, H, Me, CF ₃ , Et], [RC6291; F, H, H, Me, CF ₃ , Pr], [RC6292; F, H, H, Me, CF ₃ , i- Pr], [RC6293; F, H, H, Me, CF ₃ , c-Pr], [RC6294; F, H, H, Me, CF ₃ , Bu], [RC6295; F, H, H, Me, CF ₃ , i-Bu], [RC6296; F, H, H, Me, CF ₃ , t-Bu], [RC6297; F, H, H, Me, CF ₃ , c-PrCH ₂ ], [RC6298; F, H, H, Me, CF ₃ , Ph], [RC6299; F, H, H, Me, CF ₃ , Bn], [RC6300; F, H, H, Me, CF ₃ , CF ₃ ], [RC6301; F, H, H, Me, CF ₃ , CF ₃ CH ₂ ], [RC6302; F, H , H, Me, CF ₃ , CF ₃ CF ₂ ], [RC6303; F, H, H, Me, CF ₃ , CF ₂ H], [RC6304; F, H, H, Me, CF ₃ , CF ₂ HCF ₂ ], [RC6305; F, H, Me, Me, CF ₃ , Me], [RC6306; F, H, Me, Me, CF ₃ , Et], [RC6307; F, H, Me, Me, CF ₃ , Pr], [RC6308; F, H, Me, Me, CF ₃ , i-Pr], [RC6309; F, H, Me, Me, CF ₃ , c-Pr], [RC6310; F, H, Me , Me, CF ₃ , Bu], [RC6311; F, H, Me, Me, CF ₃ , i-Bu], [RC6312; F, H, Me, Me, CF ₃ , t-Bu], [RC6313; F, H, Me, Me, CF ₃ , c-PrCH ₂ ], [RC6314; F, H, Me, Me, CF ₃ , Ph], [RC6315; F, H, Me, Me, CF ₃ , Bn] , [RC6316; F, H, Me, Me, CF ₃ , CF ₃ ], [RC6317; F, H, Me, Me, CF ₃ , CF ₃ CH ₂ ], [RC6318; F, H, Me, Me, CF ₃ , CF ₃ CF ₂ ], [RC6319; F, H, Me, Me, CF ₃ , CF ₂ H], [RC6320; F, H, Me, Me, CF ₃ , CF ₂ HCF ₂ ], [RC6321 ; F, H, Me, Et, CF ₃ , Me], [RC6322; F, H, Me, Et, CF ₃ , Et], [RC6323; F, H, Me, Et, CF ₃ , Pr], [ RC6324; F, H, Me, Et, CF ₃ , i-Pr], [RC6325; F, H, Me, Et, CF ₃ , c-Pr], [RC6326; F, H, Me, Et, CF ₃ , Bu], [RC6327; F, H, Me, Et, CF ₃ , i-Bu], [RC6328; F, H, Me, Et, CF ₃ , t-Bu], [RC6329; F, H, Me , Et, CF ₃ , c-PrCH ₂ ], [RC6330; F, H, Me, Et, CF ₃ , Ph], [RC6331; F, H, Me, Et, CF ₃ , Bn], [RC63 32; F, H, Me, Et, CF ₃ , CF ₃ ], [RC6333; F, H, Me, Et, CF ₃ , CF ₃ CH ₂ ], [RC6334; F, H, Me, Et, CF ₃ , CF ₃ CF ₂ ], [RC6335; F, H, Me, Et, CF ₃ , CF ₂ H], [RC6336; F, H, Me, Et, CF ₃ , CF ₂ HCF ₂ ], [RC6337; F , H, Me, F, CF ₃ , Me], [RC6338; F, H, Me, F, CF ₃ , Et], [RC6339; F, H, Me, F, CF ₃ , Pr], [RC6340; F, H, Me, F, CF ₃ , i-Pr], [RC6341; F, H, Me, F, CF ₃ , c-Pr], [RC6342; F, H, Me, F, CF ₃ , Bu ], [RC6343; F, H, Me, F, CF ₃ , i-Bu], [RC6344; F, H, Me, F, CF ₃ , t-Bu], [RC6345; F, H, Me, F , CF ₃ , c-PrCH ₂ ], [RC6346; F, H, Me, F, CF ₃ , Ph], [RC6347; F, H, Me, F, CF ₃ , Bn], [RC6348; F, H , Me, F, CF ₃ , CF ₃ ], [RC6349; F, H, Me, F, CF ₃ , CF ₃ CH ₂ ], [RC6350; F, H, Me, F, CF ₃ , CF ₃ CF ₂ ], [RC6351; F, H, Me, F, CF ₃ , CF ₂ H], [RC6352; F, H, Me, F, CF ₃ , CF ₂ HCF ₂ ], [RC6353; F, H, Me, Cl, CF ₃ , Me], [RC6354; F, H, Me, Cl, CF ₃ , Et], [RC6355; F, H, Me, Cl, CF ₃ , Pr], [RC6356; F, H, Me , Cl, CF ₃ , i-Pr], [RC6357; F, H, Me, Cl, CF ₃ , c-Pr], [RC6358; F, H, Me, Cl, CF ₃ , Bu], [RC6359; F, H, Me, Cl, CF ₃ , i-Bu], [RC6360; F, H, Me, Cl, CF ₃ , t-Bu], [RC6361; F, H, Me, Cl, CF ₃ , c -PrCH ₂ ], [RC6362; F, H, Me, Cl, CF ₃ , Ph], [RC6363; F, H, Me, Cl, CF ₃ , Bn], [RC6364; F, H, Me, Cl, CF ₃ , CF ₃ ], [RC6365; F, H, Me, Cl, CF ₃ , CF ₃ CH ₂ ], [RC6366; F, H, Me, Cl, CF ₃ , CF ₃ CF ₂ ], [RC6367; F, H, Me, Cl , CF ₃ , CF ₂ H], [RC6368; F, H, Me, Cl, CF ₃ , CF ₂ HCF ₂ ], [RC6369; F, H, Et, H, CF ₃ , Me], [RC6370; F , H, Et, H, CF ₃ , Et], [RC6371; F, H, Et, H, CF ₃ , Pr], [RC6372; F, H, Et, H, CF ₃ , i-Pr], [ RC6373; F, H, Et, H, CF ₃ , c-Pr], [RC6374; F, H, Et, H, CF ₃ , Bu], [RC6375; F, H, Et, H, CF ₃ , i -Bu], [RC6376; F, H, Et, H, CF ₃ , t-Bu], [RC6377; F, H, Et, H, CF ₃ , c-PrCH ₂ ], [RC6378; F, H, Et, H, CF ₃ , Ph], [RC6379; F, H, Et, H, CF ₃ , Bn], [RC6380; F, H, Et, H, CF ₃ , CF ₃ ], [RC6381; F, H, Et, H, CF ₃ , CF ₃ CH ₂ ], [RC6382; F, H, Et, H, CF ₃ , CF ₃ CF ₂ ], [RC6383; F, H, Et, H, CF ₃ , CF ₂ H], [RC6384; F, H, Et, H, CF ₃ , CF ₂ HCF ₂ ], [RC6385; F, H, Et, F, CF ₃ , Me], [RC6386; F, H, Et, F, CF ₃ , Et], [RC6387; F, H, Et, F, CF ₃ , Pr], [RC6388; F, H, Et, F, CF ₃ , i-Pr], [RC6389; F, H , Et, F, CF ₃ , c-Pr], [RC6390; F, H, Et, F, CF ₃ , Bu], [RC6391; F, H, Et, F, CF ₃ , i-Bu], [ RC6392; F, H, Et, F, CF ₃ , t-Bu], [RC6393; F, H, Et, F, CF ₃ , c-PrCH ₂ ], [RC6394; F, H, Et, F, CF ₃ , Ph], [RC6395; F, H, Et, F, CF ₃ , Bn], [RC6396; F, H, Et, F, CF ₃ , CF ₃ ], [RC6397; F, H, Et, F , CF ₃ , CF ₃ CH ₂ ], [RC 6398; F, H, Et, F, CF ₃ , CF ₃ CF ₂ ], [RC6399; F, H, Et, F, CF ₃ , CF ₂ H], [RC6400; F, H, Et, F, CF ₃ , CF ₂ HCF ₂ ],

[RC6401; F, H, Et, Cl, CF ₃ , Me], [RC6402; F, H, Et, Cl, CF ₃ , Et], [RC6403; F, H, Et, Cl, CF ₃ , Pr] , [RC6404; F, H, Et, Cl, CF ₃ , i-Pr], [RC6405; F, H, Et, Cl, CF ₃ , c-Pr], [RC6406; F, H, Et, Cl, CF ₃ , Bu], [RC6407; F, H, Et, Cl, CF ₃ , i-Bu], [RC6408; F, H, Et, Cl, CF ₃ , t-Bu], [RC6409; F, H , Et, Cl, CF ₃ , c-PrCH ₂ ], [RC6410; F, H, Et, Cl, CF ₃ , Ph], [RC6411; F, H, Et, Cl, CF ₃ , Bn], [RC6412 ; F, H, Et, Cl, CF ₃ , CF ₃ ], [RC6413; F, H, Et, Cl, CF ₃ , CF ₃ CH ₂ ], [RC6414; F, H, Et, Cl, CF ₃ , CF ₃ CF ₂ ], [RC6415; F, H, Et, Cl, CF ₃ , CF ₂ H], [RC6416; F, H, Et, Cl, CF ₃ , CF ₂ HCF ₂ ], [RC6417; F, H, F, H, CF ₃ , Me], [RC6418; F, H, F, H, CF ₃ , Et], [RC6419; F, H, F, H, CF ₃ , Pr], [RC6420; F , H, F, H, CF ₃ , i-Pr], [RC6421; F, H, F, H, CF ₃ , c-Pr], [RC6422; F, H, F, H, CF ₃ , Bu] , [RC6423; F, H, F, H, CF ₃ , i-Bu], [RC6424; F, H, F, H, CF ₃ , t-Bu], [RC6425; F, H, F, H, CF ₃ , c-PrCH ₂ ], [RC6426; F, H, F, H, CF ₃ , Ph], [RC6427; F, H, F, H, CF ₃ , Bn], [RC6428; F, H, F, H, CF ₃ , CF ₃ ], [RC6429; F, H, F, H, CF ₃ , CF ₃ CH ₂ ], [RC6430; F, H, F, H, CF ₃ , CF ₃ CF ₂ ] , [RC6431; F, H, F, H, CF ₃ , CF ₂ H], [RC6432; F, H, F, H, CF ₃ , CF ₂ HCF ₂ ], [RC6433; F, H, F, F , CF ₃ , Me], [RC6434; F, H, F, F, CF ₃ , Et], [RC6435; F, H, F, F, CF ₃ , Pr], [RC6436; F, H, F, F, CF ₃ , i-Pr], [RC6437; F, H, F , F, CF ₃ , c-Pr], [RC6438; F, H, F, F, CF ₃ , Bu], [RC6439; F, H, F, F, CF ₃ , i-Bu], [RC6440; F, H, F, F, CF ₃ , t-Bu], [RC6441; F, H, F, F, CF ₃ , c-PrCH ₂ ], [RC6442; F, H, F, F, CF ₃ , Ph], [RC6443; F, H, F, F, CF ₃ , Bn], [RC6444; F, H, F, F, CF ₃ , CF ₃ ], [RC6445; F, H, F, F, CF ₃ , CF ₃ CH ₂ ], [RC6446; F, H, F, F, CF ₃ , CF ₃ CF ₂ ], [RC6447; F, H, F, F, CF ₃ , CF ₂ H], [RC6448; F, H, F, F, CF ₃ , CF ₂ HCF ₂ ], [RC6449; F, H, F, Cl, CF ₃ , Me], [RC6450; F, H, F, Cl, CF ₃ , Et] , [RC6451; F, H, F, Cl, CF ₃ , Pr], [RC6452; F, H, F, Cl, CF ₃ , i-Pr], [RC6453; F, H, F, Cl, CF ₃ , c-Pr], [RC6454; F, H, F, Cl, CF ₃ , Bu], [RC6455; F, H, F, Cl, CF ₃ , i-Bu], [RC6456; F, H, F , Cl, CF ₃ , t-Bu], [RC6457; F, H, F, Cl, CF ₃ , c-PrCH ₂ ], [RC6458; F, H, F, Cl, CF ₃ , Ph], [RC6459 ; F, H, F, Cl, CF ₃ , Bn], [RC6460; F, H, F, Cl, CF ₃ , CF ₃ ], [RC6461; F, H, F, Cl, CF ₃ , CF ₃ CH ₂ ], [RC6462; F, H, F, Cl, CF ₃ , CF ₃ CF ₂ ], [RC6463; F, H, F, Cl, CF ₃ , CF ₂ H], [RC6464; F, H, F , Cl, CF ₃ , CF ₂ HCF ₂ ], [RC6465; F, H, Cl, H, CF ₃ , Me], [RC6466; F, H, Cl, H, CF ₃ , Et], [RC6467; F , H, Cl, H, CF ₃ , Pr], [RC6468; F, H, Cl, H, CF ₃ , i-Pr], [RC6469; F, H, Cl, H, CF ₃ , c-Pr], [RC6470; F, H, Cl, H, CF ₃ , Bu], [RC6471; F, H, Cl, H, CF ₃ , i-Bu], [RC6472; F, H, Cl, H, CF ₃ , t-Bu], [RC6473; F, H, Cl, H, CF ₃ , c-PrCH ₂ ] , [RC6474; F, H, Cl, H, CF ₃ , Ph], [RC6475; F, H, Cl, H, CF ₃ , Bn], [RC6476; F, H, Cl, H, CF ₃ , CF ₃ ], [RC6477; F, H, Cl, H, CF ₃ , CF ₃ CH ₂ ], [RC6478; F, H, Cl, H, CF ₃ , CF ₃ CF ₂ ], [RC6479; F, H, Cl, H, CF ₃ , CF ₂ H], [RC6480; F, H, Cl, H, CF ₃ , CF ₂ HCF ₂ ], [RC6481; F, H, Cl, Cl, CF ₃ , Me], [ RC6482; F, H, Cl, Cl, CF ₃ , Et], [RC6483; F, H, Cl, Cl, CF ₃ , Pr], [RC6484; F, H, Cl, Cl, CF ₃ , i-Pr ], [RC6485; F, H, Cl, Cl, CF ₃ , c-Pr], [RC6486; F, H, Cl, Cl, CF ₃ , Bu], [RC6487; F, H, Cl, Cl, CF ₃ , i-Bu], [RC6488; F, H, Cl, Cl, CF ₃ , t-Bu], [RC6489; F, H, Cl, Cl, CF ₃ , c-PrCH ₂ ], [RC6490; F , H, Cl, Cl, CF ₃ , Ph], [RC6491; F, H, Cl, Cl, CF ₃ , Bn], [RC6492; F, H, Cl, Cl, CF ₃ , CF ₃ ], [RC6493 ; F, H, Cl, Cl, CF ₃ , CF ₃ CH ₂ ], [RC6494; F, H, Cl, Cl, CF ₃ , CF ₃ CF ₂ ], [RC6495; F, H, Cl, Cl, CF ₃ , CF ₂ H], [RC6496; F, H, Cl, Cl, CF ₃ , CF ₂ HCF ₂ ], [RC6497; F, H, H, H, CF ₂ HCH ₂ , Me], [RC6498; F , H, H, H, CF ₂ HCH ₂ , Et], [RC6499; F, H, H, H, CF ₂ HCH ₂ , Pr], [RC6500; F, H, H, H, CF ₂ HCH ₂ , i- Pr], [RC6501; F, H, H, H, CF ₂ HCH ₂ , c-Pr], [RC6502; F, H, H, H, CF ₂ HCH ₂ , Bu], [RC6503; F, H, H, H, CF ₂ HCH ₂ , i-Bu], [RC6504; F, H, H, H, CF ₂ HCH ₂ , t-Bu], [RC6505; F, H, H, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC6506; F, H, H, H, CF ₂ HCH ₂ , Ph], [RC6507; F, H, H, H, CF ₂ HCH ₂ , Bn], [RC6508; F, H, H, H, CF ₂ HCH ₂ , CF ₃ ], [RC6509; F, H, H, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC6510; F, H, H, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC6511; F, H, H, H, CF ₂ HCH ₂ , CF ₂ H], [RC6512; F, H, H, H, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC6513; F, H, H, Me, CF ₂ HCH ₂ , Me], [RC6514; F, H, H, Me, CF ₂ HCH ₂ , Et], [RC6515; F, H, H, Me , CF ₂ HCH ₂ , Pr], [RC6516; F, H, H, Me, CF ₂ HCH ₂ , i-Pr], [RC6517; F, H, H, Me, CF ₂ HCH ₂ , c-Pr] , [RC6518; F, H, H, Me, CF ₂ HCH ₂ , Bu], [RC6519; F, H, H, Me, CF ₂ HCH ₂ , i-Bu], [RC6520; F, H, H, Me, CF ₂ HCH ₂ , t-Bu], [RC6521; F, H, H, Me, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC6522; F, H, H, Me, CF ₂ HCH ₂ , Ph], [RC6523; F, H, H, Me, CF ₂ HCH ₂ , Bn], [RC6524; F, H, H, Me, CF ₂ HCH ₂ , CF ₃ ], [RC6525; F, H, H , Me, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC6526; F, H, H, Me, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC6527; F, H, H, Me, CF ₂ HCH ₂ , CF ₂ H], [RC6528; F, H, H, Me, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC6529; F, H, Me, Me, CF ₂ HCH ₂ , Me], [RC6530; F, H, Me, Me, CF ₂ HCH ₂ , Et], [RC6531; F, H, Me , Me, CF ₂ HCH ₂ , Pr], [RC6532; F, H, Me, Me, CF ₂ HCH ₂ , i-Pr], [RC6533; F, H, Me, Me, CF ₂ HCH ₂ , c- Pr], [RC6534; F, H, Me, Me, CF ₂ HCH ₂ , Bu], [RC6535; F, H, Me, Me, CF ₂ HCH ₂ , i-Bu], [RC6536; F, H, Me, Me, CF ₂ HCH ₂ , t-Bu], [RC6537; F, H, Me, Me, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC6538; F, H, Me, Me, CF ₂ HCH _{2, Ph], [RC6539;} F, H, Me, Me, CF 2 HCH 2, Bn], [RC6540; F, H, Me, Me, CF 2 HCH 2, CF 3], [RC6541; F, H , Me, Me, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC6542; F, H, Me, Me, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC6543; F, H, Me, Me, CF ₂ HCH ₂ , CF ₂ H], [RC6544; F, H, Me, Me, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC6545; F, H, Me, Et, CF ₂ HCH ₂ , Me], [RC6546; F, H, Me, Et, CF ₂ HCH ₂ , Et], [RC6547; F, H, Me, Et, CF ₂ HCH ₂ , Pr], [RC6548; F, H, Me, Et, CF ₂ HCH ₂ , i-Pr], [RC6549; F, H, Me, Et, CF ₂ HCH ₂ , c-Pr], [RC6550; F, H, Me, Et, CF ₂ HCH ₂ , Bu], [ RC6551; F, H, Me, Et, CF ₂ HCH ₂ , i-Bu], [RC6552; F, H, Me, Et, CF ₂ HCH ₂ , t-Bu], [RC6553; F, H, Me, Et, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC6554; F, H, Me, Et, CF ₂ HCH ₂ , Ph], [RC6555; F, H, Me, Et, CF ₂ HCH ₂ , Bn] , [RC6556; F, H, Me, Et, CF ₂ HCH ₂ , CF ₃ ], [RC6557; F, H, Me, Et, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC6558; F, H, Me, Et, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC6559; F, H, Me, Et, CF ₂ HCH ₂ , CF ₂ H], [RC6560; F, H, Me, Et, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC6561; F, H, Me, F, CF ₂ HCH ₂ , Me], [RC6562; F, H, Me, F, CF ₂ HCH ₂ , Et], [RC6563; F, H, Me, F, CF ₂ HCH ₂ , Pr], [RC6564; F, H, Me, F, CF ₂ HCH ₂ , i-Pr], [RC6565; F, H, Me, F, CF ₂ HCH ₂ , c-Pr], [ RC6566; F, H, Me, F, CF ₂ HCH ₂ , Bu], [RC6567; F, H, Me, F, CF ₂ HCH ₂ , i-Bu], [RC6568; F, H, Me, F, CF ₂ HCH ₂ , t-Bu], [RC6569; F, H, Me, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC6570; F, H, Me, F, CF ₂ HCH ₂ , Ph] , [RC6571; F, H, Me, F, CF ₂ HCH ₂ , Bn], [RC6572; F, H, Me, F, CF ₂ HCH ₂ , CF ₃ ], [RC6573; F, H, Me, F , CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC6574; F, H, Me, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC6575; F, H, Me, F, CF ₂ HCH ₂ , CF ₂ H], [RC6576; F, H, Me, F, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC6577; F, H, Me, Cl, CF ₂ HCH ₂ , Me], [RC6578; F , H, Me, Cl, CF ₂ HCH ₂ , Et], [RC6579; F, H, Me, Cl, CF ₂ HCH ₂ , Pr], [RC6580; F, H, Me, Cl, CF ₂ HCH ₂ , i-Pr], [RC6581; F, H, Me, Cl, CF ₂ HCH ₂ , c-Pr], [RC6582; F, H, Me, Cl, CF ₂ HCH ₂ , Bu], [RC6583; F, H, Me, Cl, CF ₂ HCH ₂ , i-Bu], [RC6584; F, H, Me, Cl, CF ₂ HCH ₂ , t-Bu], [RC6585; F, H, Me, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC6586; F, H, Me, Cl, CF ₂ HCH ₂ , Ph], [RC6587; F, H, Me, Cl, CF ₂ HCH ₂ , Bn], [RC6588; F, H, Me, Cl, CF ₂ HCH ₂ , CF ₃ ], [RC6589; F, H, Me, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC6590; F, H, Me, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC6591; F, H, Me, Cl, CF ₂ HCH ₂ , CF ₂ H], [RC6592; F, H, Me, Cl, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC6593; F, H, Et, H, CF ₂ HCH ₂ , Me], [RC6594; F, H, Et, H, CF ₂ HCH ₂ , Et], [RC6595; F, H, Et, H, CF ₂ HCH ₂ , Pr ], [RC6596; F, H, Et, H, CF ₂ HCH ₂ , i-Pr], [RC6597; F, H, Et, H, CF ₂ HCH ₂ , c-Pr], [RC6598; F, H , Et, H, CF ₂ HCH ₂ , Bu], [RC6599; F, H
, Et, H, CF ₂ HCH ₂ , i-Bu], [RC6600; F, H, Et, H, CF ₂ HCH ₂ , t-Bu],

[RC6601; F, H, Et, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC6602; F, H, Et, H, CF ₂ HCH ₂ , Ph], [RC6603; F, H, Et, H, CF ₂ HCH ₂ , Bn], [RC6604; F, H, Et, H, CF ₂ HCH ₂ , CF ₃ ], [RC6605; F, H, Et, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC6606; F, H, Et, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC6607; F, H, Et, H, CF ₂ HCH ₂ , CF ₂ H], [RC6608; F, H, Et, H, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC6609; F, H, Et, F, CF ₂ HCH ₂ , Me], [RC6610; F, H, Et, F, CF ₂ HCH ₂ , Et], [RC6611; F, H, Et, F, CF ₂ HCH ₂ , Pr], [RC6612; F, H, Et, F, CF ₂ HCH ₂ , i-Pr], [RC6613; F, H, Et, F, CF ₂ HCH ₂ , c-Pr], [RC6614; F, H, Et, F, CF ₂ HCH ₂ , Bu], [RC6615; F, H, Et, F, CF ₂ HCH ₂ , i-Bu], [RC6616; F, H, Et, F, CF ₂ HCH ₂ , t-Bu], [RC6617; F, H, Et, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [ RC6618; F, H, Et, F, CF ₂ HCH ₂ , Ph], [RC6619; F, H, Et, F, CF ₂ HCH ₂ , Bn], [RC6620; F, H, Et, F, CF ₂ HCH ₂ , CF ₃ ], [RC6621; F, H, Et, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC6622; F, H, Et, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ] , [RC6623; F, H, Et, F, CF ₂ HCH ₂ , CF ₂ H], [RC6624; F, H, Et, F, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC6625; F, H , Et, Cl, CF ₂ HCH ₂ , Me], [RC6626; F, H, Et, Cl, CF ₂ HCH ₂ , Et], [RC6627; F, H, Et, Cl, CF ₂ HCH ₂ , Pr] , [RC6628; F, H, Et, Cl, CF ₂ HCH ₂ , i-Pr], [RC6629; F, H, Et, Cl, CF ₂ HCH ₂ , c-Pr], [RC6630; F, H, Et, Cl, CF ₂ HCH ₂ , Bu], [ RC6631; F, H, Et, Cl, CF ₂ HCH ₂ , i-Bu], [RC6632; F, H, Et, Cl, CF ₂ HCH ₂ , t-Bu], [RC6633; F, H, Et, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC6634; F, H, Et, Cl, CF ₂ HCH ₂ , Ph], [RC6635; F, H, Et, Cl, CF ₂ HCH ₂ , Bn] , [RC6636; F, H, Et, Cl, CF ₂ HCH ₂ , CF ₃ ], [RC6637; F, H, Et, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC6638; F, H, Et, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC6639; F, H, Et, Cl, CF ₂ HCH ₂ , CF ₂ H], [RC6640; F, H, Et, Cl, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC6641; F, H, F, H, CF ₂ HCH ₂ , Me], [RC6642; F, H, F, H, CF ₂ HCH ₂ , Et], [RC6643; F , H, F, H, CF ₂ HCH ₂ , Pr], [RC6644; F, H, F, H, CF ₂ HCH ₂ , i-Pr], [RC6645; F, H, F, H, CF ₂ HCH _{2, c-Pr], [} RC6646; F, H, F, H, CF 2 HCH 2, Bu], [RC6647; F, H, F, H, CF 2 HCH 2, i-Bu], [RC6648; F, H, F, H, CF ₂ HCH ₂ , t-Bu], [RC6649; F, H, F, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC6650; F, H, F, H , CF ₂ HCH ₂ , Ph], [RC6651; F, H, F, H, CF ₂ HCH ₂ , Bn], [RC6652; F, H, F, H, CF ₂ HCH ₂ , CF ₃ ], [RC6653 ; F, H, F, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC6654; F, H, F, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC6655; F, H, F , H, CF ₂ HCH ₂ , CF ₂ H], [RC6656; F, H, F , H, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC6657; F, H, F, F, CF ₂ HCH ₂ , Me], [RC6658; F, H, F, F, CF ₂ HCH ₂ , Et ], [RC6659; F, H, F, F, CF ₂ HCH ₂ , Pr], [RC6660; F, H, F, F, CF ₂ HCH ₂ , i-Pr], [RC6661; F, H, F , F, CF ₂ HCH ₂ , c-Pr], [RC6662; F, H, F, F, CF ₂ HCH ₂ , Bu], [RC6663; F, H, F, F, CF ₂ HCH ₂ , i- Bu], [RC6664; F, H, F, F, CF ₂ HCH ₂ , t-Bu], [RC6665; F, H, F, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC6666; F , H, F, F, CF ₂ HCH ₂ , Ph], [RC6667; F, H, F, F, CF ₂ HCH ₂ , Bn], [RC6668; F, H, F, F, CF ₂ HCH ₂ , CF ₃ ], [RC6669; F, H, F, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC6670; F, H, F, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC6671 ; F, H, F, F, CF ₂ HCH ₂ , CF ₂ H], [RC6672; F, H, F, F, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC6673; F, H, F, Cl, CF ₂ HCH ₂ , Me], [RC6674; F, H, F, Cl, CF ₂ HCH ₂ , Et], [RC6675; F, H, F, Cl, CF ₂ HCH ₂ , Pr], [RC6676 ; F, H, F, Cl, CF ₂ HCH ₂ , i-Pr], [RC6677; F, H, F, Cl, CF ₂ HCH ₂ , c-Pr], [RC6678; F, H, F, Cl , CF ₂ HCH ₂ , Bu], [RC6679; F, H, F, Cl, CF ₂ HCH ₂ , i-Bu], [RC6680; F, H, F, Cl, CF ₂ HCH ₂ , t-Bu] , [RC6681; F, H, F, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC6682; F, H, F, Cl, CF ₂ HCH ₂ , Ph], [RC6683; F, H, F , Cl, CF ₂ HCH ₂ , Bn], [RC6684; F, H, F, Cl, CF ₂ HCH ₂ , CF ₃ ] , [RC6685; F, H, F, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC6686; F, H, F, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC6687; F, H, F, Cl, CF ₂ HCH ₂ , CF ₂ H], [RC6688; F, H, F, Cl, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC6689; F, H, Cl, H, CF ₂ HCH ₂ , Me], [RC6690; F, H, Cl, H, CF ₂ HCH ₂ , Et], [RC6691; F, H, Cl, H, CF ₂ HCH ₂ , Pr], [RC6692; F, H, Cl, H, CF ₂ HCH ₂ , i-Pr], [RC6693; F, H, Cl, H, CF ₂ HCH ₂ , c-Pr], [RC6694; F, H, Cl, H, CF ₂ HCH ₂ , Bu], [RC6695; F, H, Cl, H, CF ₂ HCH ₂ , i-Bu], [RC6696; F, H, Cl, H, CF ₂ HCH ₂ , t-Bu], [RC6697 ; F, H, Cl, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC6698; F, H, Cl, H, CF ₂ HCH ₂ , Ph], [RC6699; F, H, Cl, H, CF ₂ HCH ₂ , Bn], [RC6700; F, H, Cl, H, CF ₂ HCH ₂ , CF ₃ ], [RC6701; F, H, Cl, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC6702; F, H, Cl, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC6703; F, H, Cl, H, CF ₂ HCH ₂ , CF ₂ H], [RC6704; F, H, Cl, H, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC6705; F, H, Cl, Cl, CF ₂ HCH ₂ , Me], [RC6706; F, H, Cl, Cl, CF ₂ HCH ₂ , Et], [RC6707; F, H, Cl, Cl, CF ₂ HCH ₂ , Pr], [RC6708; F, H, Cl, Cl, CF ₂ HCH ₂ , i-Pr], [RC6709; F, H, Cl, Cl, CF ₂ HCH ₂ , c-Pr], [RC6710; F, H, Cl, Cl, CF ₂ HCH ₂ , Bu], [RC6711; F, H, Cl, Cl, CF ₂ HCH ₂ , i -Bu], [RC6712; F, H, Cl, Cl, C F ₂ HCH ₂ , t-Bu], [RC6713; F, H, Cl, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC6714; F, H, Cl, Cl, CF ₂ HCH ₂ , Ph] , [RC6715; F, H, Cl, Cl, CF ₂ HCH ₂ , Bn], [RC6716; F, H, Cl, Cl, CF ₂ HCH ₂ , CF ₃ ], [RC6717; F, H, Cl, Cl , CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC6718; F, H, Cl, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC6719; F, H, Cl, Cl, CF ₂ HCH ₂ , CF ₂ H], [RC6720; F, H, Cl, Cl, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC6721; F, H, H, H, CF ₃ CH ₂ , Me], [RC6722; F , H, H, H, CF ₃ CH ₂ , Et], [RC6723; F, H, H, H, CF ₃ CH ₂ , Pr], [RC6724; F, H, H, H, CF ₃ CH ₂ , i-Pr], [RC6725; F, H, H, H, CF ₃ CH ₂ , c-Pr], [RC6726; F, H, H, H, CF ₃ CH ₂ , Bu], [RC6727; F, H, H, H, CF ₃ CH ₂ , i-Bu], [RC6728; F, H, H, H, CF ₃ CH ₂ , t-Bu], [RC6729; F, H, H, H, CF _{3 CH 2, c-PrCH 2]} , [RC6730; F, H, H, H, CF 3 CH 2, Ph], [RC6731; F, H, H, H, CF 3 CH 2, Bn], [RC6732; F, H, H, H, CF ₃ CH ₂ , CF ₃ ], [RC6733; F, H, H, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC6734; F, H, H, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC6735; F, H, H, H, CF ₃ CH ₂ , CF ₂ H], [RC6736; F, H, H, H, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC6737; F, H, H, Me, CF ₃ CH ₂ , Me], [RC6738; F, H, H, Me, CF ₃ CH ₂ , Et], [RC6739; F, H, H , Me, CF ₃ CH ₂ , Pr], [RC6740; F, H, H, Me, CF ₃ CH ₂ , i-Pr] , [RC6741; F, H, H, Me, CF ₃ CH ₂ , c-Pr], [RC6742; F, H, H, Me, CF ₃ CH ₂ , Bu], [RC6743; F, H, H, Me, CF ₃ CH ₂ , i-Bu], [RC6744; F, H, H, Me, CF ₃ CH ₂ , t-Bu], [RC6745; F, H, H, Me, CF ₃ CH ₂ , c -PrCH ₂ ], [RC6746; F, H, H, Me, CF ₃ CH ₂ , Ph], [RC6747; F, H, H, Me, CF ₃ CH ₂ , Bn], [RC6748; F, H, H, Me, CF ₃ CH ₂ , CF ₃ ], [RC6749; F, H, H, Me, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC6750; F, H, H, Me, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC6751; F, H, H, Me, CF ₃ CH ₂ , CF ₂ H], [RC6752; F, H, H, Me, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC6753; F, H, Me, Me, CF ₃ CH ₂ , Me], [RC6754; F, H, Me, Me, CF ₃ CH ₂ , Et], [RC6755; F, H, Me, Me, CF ₃ CH ₂ , Pr], [RC6756; F, H, Me, Me, CF ₃ CH ₂ , i-Pr], [RC6757; F, H, Me, Me, CF ₃ CH ₂ , c-Pr], [ RC6758; F, H, Me, Me, CF ₃ CH ₂ , Bu], [RC6759; F, H, Me, Me, CF ₃ CH ₂ , i-Bu], [RC6760; F, H, Me, Me, CF ₃ CH ₂ , t-Bu], [RC6761; F, H, Me, Me, CF ₃ CH ₂ , c-PrCH ₂ ], [RC6762; F, H, Me, Me, CF ₃ CH ₂ , Ph] , [RC6763; F, H, Me, Me, CF ₃ CH ₂ , Bn], [RC6764; F, H, Me, Me, CF ₃ CH ₂ , CF ₃ ], [RC6765; F, H, Me, Me , CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC6766; F, H, Me, Me, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC6767; F, H, Me, Me, CF ₃ CH ₂ , CF ₂ H], [RC6768; F, H, Me, Me, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC6769; F, H, Me, Et, CF ₃ CH ₂ , Me], [RC6770; F, H, Me, Et, CF ₃ CH ₂ , Et], [RC6771; F, H, Me, Et, CF ₃ CH ₂ , Pr], [RC6772; F, H, Me, Et, CF ₃ CH ₂ , i-Pr], [RC6773; F, H, Me, Et, CF ₃ CH ₂ , c-Pr ], [RC6774; F, H, Me, Et, CF ₃ CH ₂ , Bu], [RC6775; F, H
, Me, Et, CF ₃ CH ₂ , i-Bu], [RC6776; F, H, Me, Et, CF ₃ CH ₂ , t-Bu], [RC6777; F, H, Me, Et, CF ₃ CH ₂ , c-PrCH ₂ ], [RC6778; F, H, Me, Et, CF ₃ CH ₂ , Ph], [RC6779; F, H, Me, Et, CF ₃ CH ₂ , Bn], [RC6780; F , H, Me, Et, CF ₃ CH ₂ , CF ₃ ], [RC6781; F, H, Me, Et, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC6782; F, H, Me, Et, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC6783; F, H, Me, Et, CF ₃ CH ₂ , CF ₂ H], [RC6784; F, H, Me, Et, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC6785; F, H, Me, F, CF ₃ CH ₂ , Me], [RC6786; F, H, Me, F, CF ₃ CH ₂ , Et], [RC6787; F, H, Me, F, CF ₃ CH ₂ , Pr], [RC6788; F, H, Me, F, CF ₃ CH ₂ , i-Pr], [RC6789; F, H, Me, F, CF ₃ CH ₂ , c-Pr ], [RC6790; F, H, Me, F, CF ₃ CH ₂ , Bu], [RC6791; F, H, Me, F, CF ₃ CH ₂ , i-Bu], [RC6792; F, H, Me , F, CF ₃ CH ₂ , t-Bu], [RC6793; F, H, Me, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RC6794; F, H, Me, F, CF ₃ CH ₂ , Ph], [RC6795; F, H, Me, F, CF ₃ CH ₂ , Bn], [RC6796; F, H, Me, F, CF ₃ CH ₂ , CF ₃ ], [RC6797; F, H, Me, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC6798; F, H, Me, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC6799; F, H, Me, F, CF ₃ CH ₂ , CF ₂ H], [RC6800; F, H, Me, F, CF ₃ CH ₂ , CF ₂ HCF ₂ ],

[RC6801; F, H, Me, Cl, CF ₃ CH ₂ , Me], [RC6802; F, H, Me, Cl, CF ₃ CH ₂ , Et], [RC6803; F, H, Me, Cl, CF ₃ CH ₂ , Pr], [RC6804; F, H, Me, Cl, CF ₃ CH ₂ , i-Pr], [RC6805; F, H, Me, Cl, CF ₃ CH ₂ , c-Pr], [ RC6806; F, H, Me, Cl, CF ₃ CH ₂ , Bu], [RC6807; F, H, Me, Cl, CF ₃ CH ₂ , i-Bu], [RC6808; F, H, Me, Cl, CF ₃ CH ₂ , t-Bu], [RC6809; F, H, Me, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RC6810; F, H, Me, Cl, CF ₃ CH ₂ , Ph] , [RC6811; F, H, Me, Cl, CF ₃ CH ₂ , Bn], [RC6812; F, H, Me, Cl, CF ₃ CH ₂ , CF ₃ ], [RC6813; F, H, Me, Cl , CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC6814; F, H, Me, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC6815; F, H, Me, Cl, CF ₃ CH ₂ , CF ₂ H], [RC6816; F, H, Me, Cl, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC6817; F, H, Et, H, CF ₃ CH ₂ , Me], [RC6818; F , H, Et, H, CF ₃ CH ₂ , Et], [RC6819; F, H, Et, H, CF ₃ CH ₂ , Pr], [RC6820; F, H, Et, H, CF ₃ CH ₂ , i-Pr], [RC6821; F, H, Et, H, CF ₃ CH ₂ , c-Pr], [RC6822; F, H, Et, H, CF ₃ CH ₂ , Bu], [RC6823; F, H, Et, H, CF ₃ CH ₂ , i-Bu], [RC6824; F, H, Et, H, CF ₃ CH ₂ , t-Bu], [RC6825; F, H, Et, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RC6826; F, H, Et, H, CF ₃ CH ₂ , Ph], [RC6827; F, H, Et, H, CF ₃ CH ₂ , Bn], [RC6828; F, H, Et, H, CF ₃ CH ₂ , CF ₃ ], [RC6829; F, H, Et, H, CF ₃ C H ₂ , CF ₃ CH ₂ ], [RC6830; F, H, Et, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC6831; F, H, Et, H, CF ₃ CH ₂ , CF ₂ H ], [RC6832; F, H, Et, H, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC6833; F, H, Et, F, CF ₃ CH ₂ , Me], [RC6834; F, H, Et, F, CF ₃ CH ₂ , Et], [RC6835; F, H, Et, F, CF ₃ CH ₂ , Pr], [RC6836; F, H, Et, F, CF ₃ CH ₂ , i-Pr ], [RC6837; F, H, Et, F, CF ₃ CH ₂ , c-Pr], [RC6838; F, H, Et, F, CF ₃ CH ₂ , Bu], [RC6839; F, H, Et , F, CF ₃ CH ₂ , i-Bu], [RC6840; F, H, Et, F, CF ₃ CH ₂ , t-Bu], [RC6841; F, H, Et, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RC6842; F, H, Et, F, CF ₃ CH ₂ , Ph], [RC6843; F, H, Et, F, CF ₃ CH ₂ , Bn], [RC6844; F, H , Et, F, CF ₃ CH ₂ , CF ₃ ], [RC6845; F, H, Et, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC6846; F, H, Et, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC6847; F, H, Et, F, CF ₃ CH ₂ , CF ₂ H], [RC6848; F, H, Et, F, CF ₃ CH ₂ , CF ₂ HCF ₂ ] , [RC6849; F, H, Et, Cl, CF ₃ CH ₂ , Me], [RC6850; F, H, Et, Cl, CF ₃ CH ₂ , Et], [RC6851; F, H, Et, Cl, CF ₃ CH ₂ , Pr], [RC6852; F, H, Et, Cl, CF ₃ CH ₂ , i-Pr], [RC6853; F, H, Et, Cl, CF ₃ CH ₂ , c-Pr], [RC6854; F, H, Et, Cl, CF ₃ CH ₂ , Bu], [RC6855; F, H, Et, Cl, CF ₃ CH ₂ , i-Bu], [RC6856; F, H, Et, Cl , CF ₃ CH ₂ , t-Bu], [RC6857; F, H, Et, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RC6858; F, H, Et, Cl, CF ₃ CH ₂ , Ph], [RC6859; F, H, Et, Cl, CF ₃ CH ₂ , Bn], [RC6860; F, H, Et, Cl, CF ₃ CH ₂ , CF ₃ ], [RC6861; F, H, Et, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC6862; F, H, Et, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC6863; F, H, Et, Cl, CF ₃ CH ₂ , CF ₂ H], [RC6864; F, H, Et, Cl, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC6865 ; F, H, F, H, CF ₃ CH ₂ , Me], [RC6866; F, H, F, H, CF ₃ CH ₂ , Et], [RC6867; F, H, F, H, CF ₃ CH ₂ , Pr], [RC6868; F, H, F, H, CF ₃ CH ₂ , i-Pr], [RC6869; F, H, F, H, CF ₃ CH ₂ , c-Pr], [RC6870; F, H, F, H, CF ₃ CH ₂ , Bu], [RC6871; F, H, F, H, CF ₃ CH ₂ , i-Bu], [RC6872; F, H, F, H, CF ₃ CH ₂ , t-Bu], [RC6873; F, H, F, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RC6874; F, H, F, H, CF ₃ CH ₂ , Ph], [ RC6875; F, H, F, H, CF ₃ CH ₂ , Bn], [RC6876; F, H, F, H, CF ₃ CH ₂ , CF ₃ ], [RC6877; F, H, F, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC6878; F, H, F, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC6879; F, H, F, H, CF ₃ CH ₂ , CF ₂ H], [RC6880; F, H, F, H, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC6881; F, H, F, F, CF ₃ CH ₂ , Me], [RC6882; F, H , F, F, CF ₃ CH ₂ , Et], [RC6883; F, H, F, F, CF ₃ CH ₂ , Pr], [RC6884; F, H, F, F, CF ₃ CH ₂ , i- Pr], [RC6885; F, H, F, F, CF ₃ CH ₂ , c-Pr], [RC6886; F, H, F, F, CF ₃ CH ₂ , Bu] , [RC6887; F, H, F, F, CF ₃ CH ₂ , i-Bu], [RC6888; F, H, F, F, CF ₃ CH ₂ , t-Bu], [RC6889; F, H, F, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RC6890; F, H, F, F, CF ₃ CH ₂ , Ph], [RC6891; F, H, F, F, CF ₃ CH ₂ , Bn], [RC6892; F, H, F, F, CF ₃ CH ₂ , CF ₃ ], [RC6893; F, H, F, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC6894; F, H, F, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC6895; F, H, F, F, CF ₃ CH ₂ , CF ₂ H], [RC6896; F, H, F, F, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC6897; F, H, F, Cl, CF ₃ CH ₂ , Me], [RC6898; F, H, F, Cl, CF ₃ CH ₂ , Et], [RC6899 ; F, H, F, Cl, CF ₃ CH ₂ , Pr], [RC6900; F, H, F, Cl, CF ₃ CH ₂ , i-Pr], [RC6901; F, H, F, Cl, CF ₃ CH ₂ , c-Pr], [RC6902; F, H, F, Cl, CF ₃ CH ₂ , Bu], [RC6903; F, H, F, Cl, CF ₃ CH ₂ , i-Bu], [ RC6904; F, H, F, Cl, CF ₃ CH ₂ , t-Bu], [RC6905; F, H, F, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RC6906; F, H, F , Cl, CF ₃ CH ₂ , Ph], [RC6907; F, H, F, Cl, CF ₃ CH ₂ , Bn], [RC6908; F, H, F, Cl, CF ₃ CH ₂ , CF ₃ ], [RC6909; F, H, F, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC6910; F, H, F, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC6911; F, H , F, Cl, CF ₃ CH ₂ , CF ₂ H], [RC6912; F, H, F, Cl, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC6913; F, H, Cl, H, CF ₃ CH ₂ , Me], [RC6914; F, H, Cl, H, CF ₃ CH ₂ , Et], [RC6915; F, H, Cl, H, CF ₃ C H ₂ , Pr], [RC6916; F, H, Cl, H, CF ₃ CH ₂ , i-Pr], [RC6917; F, H, Cl, H, CF ₃ CH ₂ , c-Pr], [RC6918 ; F, H, Cl, H, CF ₃ CH ₂ , Bu], [RC6919; F, H, Cl, H, CF ₃ CH ₂ , i-Bu], [RC6920; F, H, Cl, H, CF ₃ CH ₂ , t-Bu], [RC6921; F, H, Cl, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RC6922; F, H, Cl, H, CF ₃ CH ₂ , Ph], [RC6923; F, H, Cl, H, CF ₃ CH ₂ , Bn], [RC6924; F, H, Cl, H, CF ₃ CH ₂ , CF ₃ ], [RC6925; F, H, Cl, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC6926; F, H, Cl, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC6927; F, H, Cl, H, CF ₃ CH ₂ , CF ₂ H], [RC6928; F, H, Cl, H, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC6929; F, H, Cl, Cl, CF ₃ CH ₂ , Me], [RC6930; F, H, Cl, Cl, CF ₃ CH ₂ , Et], [RC6931; F, H, Cl, Cl, CF ₃ CH ₂ , Pr], [RC6932; F, H, Cl, Cl, CF ₃ CH ₂ , i -Pr], [RC6933; F, H, Cl, Cl, CF ₃ CH ₂ , c-Pr], [RC6934; F, H, Cl, Cl, CF ₃ CH ₂ , Bu], [RC6935; F, H , Cl, Cl, CF ₃ CH ₂ , i-Bu], [RC6936; F, H, Cl, Cl, CF ₃ CH ₂ , t-Bu], [RC6937; F, H, Cl, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RC6938; F, H, Cl, Cl, CF ₃ CH ₂ , Ph], [RC6939; F, H, Cl, Cl, CF ₃ CH ₂ , Bn], [RC6940; F , H, Cl, Cl, CF ₃ CH ₂ , CF ₃ ], [RC6941; F, H, Cl, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC6942; F, H, Cl, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC6943; F, H, Cl, Cl, CF ₃ CH ₂ , CF ₂ H], [RC6944; F, H, Cl, Cl, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC6945; F, H, H, H, HCCCH ₂ , Me], [RC6946; F, H, H, H, HCCCH ₂ , Et], [RC6947; F, H, H, H, HCCCH ₂ , Pr], [RC6948; F, H, H, H, HCCCH ₂ , i-Pr], [RC6949; F , H, H, H, HCCCH ₂ , c-Pr], [RC6950; F, H, H, H, HCCCH ₂ , Bu], [RC6951; F, H, H, H, HCCCH ₂ , i-Bu] , [RC6952; F, H, H, H, HCCCH ₂ , t-Bu], [RC6953; F, H, H, H, HCCCH ₂ , c-PrCH ₂ ], [RC6954; F, H, H, H , HCCCH ₂ , Ph], [RC6955; F, H, H, H, HCCCH ₂ , Bn], [RC6956; F, H, H, H, HCCCH ₂ , CF ₃ ], [RC6957; F, H, H , H, HCCCH ₂ , CF ₃ CH ₂ ], [RC6958; F, H, H, H, HCCCH ₂ , CF ₃ CF ₂ ], [RC6959; F, H, H, H, HCCCH ₂ , CF ₂ H] , [RC6960; F, H, H, H, HCCCH ₂ , CF ₂ HCF ₂ ], [RC6961; F, H, H, Me, HCCCH ₂ , Me], [RC6962; F, H, H, Me, HCCCH ₂ , Et], [RC6963; F, H, H, Me, HCCCH ₂ , Pr], [RC6964; F, H, H, Me, HCCCH ₂ , i-Pr], [RC6965; F, H, H, Me, HCCCH ₂ , c-Pr], [RC6966; F, H, H, Me, HCCCH ₂ , Bu], [RC6967; F, H, H, Me, HCCCH ₂ , i-Bu], [RC6968; F , H, H, Me, HCCCH ₂ , t-Bu], [RC6969; F, H, H, Me, HCCCH ₂ , c-PrCH ₂ ], [RC6970; F, H, H, Me, HCCCH ₂ , Ph ], [RC6971; F, H, H, Me, HCCCH ₂ , Bn], [RC6972; F, H, H, Me, HCCCH ₂ , CF ₃ ], [RC6973; F, H, H, Me, HCCCH ₂ , CF ₃ CH ₂ ], [RC6974; F, H, H, Me, HCCCH ₂ , CF ₃ CF ₂ ], [RC6975; F, H, H, Me, HCCCH ₂ , CF ₂ H], [RC6976; F, H, H, Me, HCCCH ₂ , CF ₂ HCF ₂ ], [RC6977; F, H, Me, Me, HCCCH ₂ , Me], [RC6978; F, H, Me, Me, HCCCH ₂ , Et], [RC6979; F, H, Me, Me, HCCCH ₂ , Pr], [RC6980; F , H, Me, Me, HCCCH ₂ , i-Pr], [RC6981; F, H, Me, Me, HCCCH ₂ , c-Pr], [RC6982; F, H, Me, Me, HCCCH ₂ , Bu] , [RC6983; F, H, Me, Me, HCCCH ₂ , i-Bu], [RC6984; F, H, Me, Me, HCCCH ₂ , t-Bu], [RC6985; F, H, Me, Me, HCCCH ₂ , c-PrCH ₂ ], [
RC6986; F, H, Me, Me, HCCCH ₂ , Ph], [RC6987; F, H, Me, Me, HCCCH ₂ , Bn], [RC6988; F, H, Me, Me, HCCCH ₂ , CF ₃ ] , [RC6989; F, H, Me, Me, HCCCH ₂ , CF ₃ CH ₂ ], [RC6990; F, H, Me, Me, HCCCH ₂ , CF ₃ CF ₂ ], [RC6991; F, H, Me, Me, HCCCH ₂ , CF ₂ H], [RC6992; F, H, Me, Me, HCCCH ₂ , CF ₂ HCF ₂ ], [RC6993; F, H, Me, Et, HCCCH ₂ , Me], [RC6994; F, H, Me, Et, HCCCH ₂ , Et], [RC6995; F, H, Me, Et, HCCCH ₂ , Pr], [RC6996; F, H, Me, Et, HCCCH ₂ , i-Pr], [RC6997; F, H, Me, Et, HCCCH ₂ , c-Pr], [RC6998; F, H, Me, Et, HCCCH ₂ , Bu], [RC6999; F, H, Me, Et, HCCCH ₂ , i-Bu], [RC7000; F, H, Me, Et, HCCCH ₂ , t-Bu],

[RC7001; F, H, Me, Et, HCCCH ₂ , c-PrCH ₂ ], [RC7002; F, H, Me, Et, HCCCH ₂ , Ph], [RC7003; F, H, Me, Et, HCCCH ₂ , Bn], [RC7004; F, H, Me, Et, HCCCH ₂ , CF ₃ ], [RC7005; F, H, Me, Et, HCCCH ₂ , CF ₃ CH ₂ ], [RC7006; F, H, Me , Et, HCCCH ₂ , CF ₃ CF ₂ ], [RC7007; F, H, Me, Et, HCCCH ₂ , CF ₂ H], [RC7008; F, H, Me, Et, HCCCH ₂ , CF ₂ HCF ₂ ] , [RC7009; F, H, Me, F, HCCCH ₂ , Me], [RC7010; F, H, Me, F, HCCCH ₂ , Et], [RC7011; F, H, Me, F, HCCCH ₂ , Pr ], [RC7012; F, H, Me, F, HCCCH ₂ , i-Pr], [RC7013; F, H, Me, F, HCCCH ₂ , c-Pr], [RC7014; F, H, Me, F , HCCCH ₂ , Bu], [RC7015; F, H, Me, F, HCCCH ₂ , i-Bu], [RC7016; F, H, Me, F, HCCCH ₂ , t-Bu], [RC7017; F, H, Me, F, HCCCH ₂ , c-PrCH ₂ ], [RC7018; F, H, Me, F, HCCCH ₂ , Ph], [RC7019; F, H, Me, F, HCCCH ₂ , Bn], [ RC7020; F, H, Me, F, HCCCH ₂ , CF ₃ ], [RC7021; F, H, Me, F, HCCCH ₂ , CF ₃ CH ₂ ], [RC7022; F, H, Me, F, HCCCH ₂ , CF ₃ CF ₂ ], [RC7023; F, H, Me, F, HCCCH ₂ , CF ₂ H], [RC7024; F, H, Me, F, HCCCH ₂ , CF ₂ HCF ₂ ], [RC7025; F , H, Me, Cl, HCCCH ₂ , Me], [RC7026; F, H, Me, Cl, HCCCH ₂ , Et], [RC7027; F, H, Me, Cl, HCCCH ₂ , Pr], [RC7028; F, H, Me, Cl, HCCCH 2, i-Pr], [RC7029; F, H, Me, Cl, HCCCH 2, c-Pr], [RC7030; F, H, Me, Cl, HCCCH 2, Bu], [RC7031; F, H, Me, Cl, HCCCH ₂ , i-Bu], [RC7032; F, H, Me, Cl, HCCCH ₂ , t-Bu], [RC7033; F, H, Me, Cl, HCCCH ₂ , c-PrCH ₂ ], [RC7034; F, H, Me, Cl, HCCCH ₂ , Ph], [RC7035; F, H, Me, Cl, HCCCH ₂ , Bn], [RC7036; F, H, Me, Cl, HCCCH ₂ , CF ₃ ], [RC7037; F, H, Me, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RC7038; F, H, Me, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RC7039; F, H, Me, Cl, HCCCH ₂ , CF ₂ H], [RC7040; F, H, Me, Cl, HCCCH ₂ , CF ₂ HCF ₂ ], [RC7041; F, H, Et , H, HCCCH ₂ , Me], [RC7042; F, H, Et, H, HCCCH ₂ , Et], [RC7043; F, H, Et, H, HCCCH ₂ , Pr], [RC7044; F, H, Et, H, HCCCH ₂ , i-Pr], [RC7045; F, H, Et, H, HCCCH ₂ , c-Pr], [RC7046; F, H, Et, H, HCCCH ₂ , Bu], [RC7047 ; F, H, Et, H, HCCCH ₂ , i-Bu], [RC7048; F, H, Et, H, HCCCH ₂ , t-Bu], [RC7049; F, H, Et, H, HCCCH ₂ , c-PrCH ₂ ], [RC7050; F, H, Et, H, HCCCH ₂ , Ph], [RC7051; F, H, Et, H, HCCCH ₂ , Bn], [RC7052; F, H, Et, H , HCCCH ₂ , CF ₃ ], [RC7053; F, H, Et, H, HCCCH ₂ , CF ₃ CH ₂ ], [RC7054; F, H, Et, H, HCCCH ₂ , CF ₃ CF ₂ ], [RC7055 ; F, H, Et, H, HCCCH ₂ , CF ₂ H], [RC7056; F, H, Et, H, HCCCH ₂ , CF ₂ HCF ₂ ], [RC7057; F, H, Et, F, HCCCH ₂ , Me], [RC7058; F, H, Et, F, HCCCH ₂ , Et], [RC7059; F, H, Et, F, HCCCH ₂ , Pr], [RC7060; F, H, Et, F, HCCCH ₂ , i-Pr], [RC7061; F, H, Et, F, HCCCH ₂ , c-Pr], [RC7062; F, H, Et, F, HCCCH ₂ , Bu], [RC7063; F, H, Et, F, HCCCH ₂ , i-Bu], [RC7064; F, H, Et, F, HCCCH ₂ , t-Bu], [RC7065; F, H, Et, F, HCCCH ₂ , c-PrCH ₂ ], [ RC7066; F, H, Et, F, HCCCH ₂ , Ph], [RC7067; F, H, Et, F, HCCCH ₂ , Bn], [RC7068; F, H, Et, F, HCCCH ₂ , CF ₃ ] , [RC7069; F, H, Et, F, HCCCH ₂ , CF ₃ CH ₂ ], [RC7070; F, H, Et, F, HCCCH ₂ , CF ₃ CF ₂ ], [RC7071; F, H, Et, F, HCCCH ₂ , CF ₂ H], [RC7072; F, H, Et, F, HCCCH ₂ , CF ₂ HCF ₂ ], [RC7073; F, H, Et, Cl, HCCCH ₂ , Me], [RC7074; F, H, Et, Cl, HCCCH ₂ , Et], [RC7075; F, H, Et, Cl, HCCCH ₂ , Pr], [RC7076; F, H, Et, Cl, HCCCH ₂ , i-Pr], [RC7077; F, H, Et, Cl, HCCCH ₂ , c-Pr], [RC7078; F, H, Et, Cl, HCCCH ₂ , Bu], [RC7079; F, H, Et, Cl, HCCCH ₂ , i-Bu], [RC7080; F, H, Et, Cl, HCCCH ₂ , t-Bu], [RC7081; F, H, Et, Cl, HCCCH ₂ , c-PrCH ₂ ], [RC7082; F, H , Et, Cl, HCCCH ₂ , Ph], [RC7083; F, H, Et, Cl, HCCCH ₂ , Bn], [RC7084; F, H, Et, Cl, HCCCH ₂ , CF ₃ ], [RC7085; F , H, Et, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RC7086; F, H, Et, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RC7087; F, H, Et, Cl, HCCCH ₂ , CF ₂ H], [RC7088; F, H, Et, Cl, HCCCH ₂ , CF ₂ HCF ₂ ], [RC7089; F, H, F, H, HCCCH ₂ , Me], [RC7090; F, H, F , H, H CCCH ₂ , Et], [RC7091; F, H, F, H, HCCCH ₂ , Pr], [RC7092; F, H, F, H, HCCCH ₂ , i-Pr], [RC7093; F, H, F , H, HCCCH ₂ , c-Pr], [RC7094; F, H, F, H, HCCCH ₂ , Bu], [RC7095; F, H, F, H, HCCCH ₂ , i-Bu], [RC7096; F, H, F, H, HCCCH ₂ , t-Bu], [RC7097; F, H, F, H, HCCCH ₂ , c-PrCH ₂ ], [RC7098; F, H, F, H, HCCCH ₂ , Ph], [RC7099; F, H, F, H, HCCCH ₂ , Bn], [RC7100; F, H, F, H, HCCCH ₂ , CF ₃ ], [RC7101; F, H, F, H, HCCCH ₂ , CF ₃ CH ₂ ], [RC7102; F, H, F, H, HCCCH ₂ , CF ₃ CF ₂ ], [RC7103; F, H, F, H, HCCCH ₂ , CF ₂ H], [RC7104; F, H, F, H, HCCCH ₂ , CF ₂ HCF ₂ ], [RC7105; F, H, F, F, HCCCH ₂ , Me], [RC7106; F, H, F, F, HCCCH ₂ , Et] , [RC7107; F, H, F, F, HCCCH ₂ , Pr], [RC7108; F, H, F, F, HCCCH ₂ , i-Pr], [RC7109; F, H, F, F, HCCCH ₂ , c-Pr], [RC7110; F, H, F, F, HCCCH ₂ , Bu], [RC7111; F, H, F, F, HCCCH ₂ , i-Bu], [RC7112; F, H, F , F, HCCCH ₂ , t-Bu], [RC7113; F, H, F, F, HCCCH ₂ , c-PrCH ₂ ], [RC7114; F, H, F, F, HCCCH ₂ , Ph], [RC7115 ; F, H, F, F, HCCCH ₂ , Bn], [RC7116; F, H, F, F, HCCCH ₂ , CF ₃ ], [RC7117; F, H, F, F, HCCCH ₂ , CF ₃ CH ₂ ], [RC7118; F, H, F, F, HCCCH ₂ , CF ₃ CF ₂ ], [RC7119; F, H, F, F, HCCCH ₂ , CF ₂ H], [RC7120; F, H, F , F, HCCCH ₂ , CF ₂ HCF ₂ ], [RC7121; F, H, F, Cl, HCCCH ₂ , Me], [RC7122; F, H, F, Cl, HCCCH ₂ , Et], [RC7123; F, H, F, Cl, HCCCH ₂ , Pr], [RC7124; F, H, F, Cl, HCCCH _{2, i-Pr], [} RC7125; F, H, F, Cl, HCCCH 2, c-Pr], [RC7126; F, H, F, Cl, HCCCH 2, Bu], [RC7127; F, H, F, Cl, HCCCH ₂ , i-Bu], [RC7128; F, H, F, Cl, HCCCH ₂ , t-Bu], [RC7129; F, H, F, Cl, HCCCH ₂ , c-PrCH ₂ ] , [RC7130; F, H, F, Cl, HCCCH ₂ , Ph], [RC7131; F, H, F, Cl, HCCCH ₂ , Bn], [RC7132; F, H, F, Cl, HCCCH ₂ , CF ₃ ], [RC7133; F, H, F, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RC7134; F, H, F, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RC7135; F, H, F, Cl, HCCCH ₂ , CF ₂ H], [RC7136; F, H, F, Cl, HCCCH ₂ , CF ₂ HCF ₂ ], [RC7137; F, H, Cl, H, HCCCH ₂ , Me], [ RC7138; F, H, Cl, H, HCCCH ₂ , Et], [RC7139; F, H, Cl, H, HCCCH ₂ , Pr], [RC7140; F, H, Cl, H, HCCCH ₂ , i-Pr ], [RC7141; F, H, Cl, H, HCCCH ₂ , c-Pr], [RC7142; F, H, Cl, H, HCCCH ₂ , Bu], [RC7143; F, H, Cl, H, HCCCH ₂ , i-Bu], [RC7144; F, H, Cl, H, HCCCH ₂ , t-Bu], [RC7145; F, H, Cl, H, HCCCH ₂ , c-PrCH ₂ ], [RC7146; F , H, Cl, H, HCCCH ₂ , Ph], [RC7147; F, H, Cl, H, HCCCH ₂ , Bn], [RC7148; F, H, Cl, H, HCCCH ₂ , CF ₃ ], [RC7149 ; F, H, Cl, H, HCCCH ₂ , CF ₃ CH ₂ ], [RC7150; F, H, Cl, H, HCCCH ₂ , CF ₃ CF ₂ ], [RC7151; F, H, Cl, H, HCCCH ₂ , CF ₂ H], [RC7152; F , H, Cl, H, HCCCH ₂ , CF ₂ HCF ₂ ], [RC7153; F, H, Cl, Cl, HCCCH ₂ , Me], [RC7154; F, H, Cl, Cl, HCCCH ₂ , Et], [RC7155; F, H, Cl, Cl, HCCCH ₂ , Pr], [RC7156; F, H, Cl, Cl, HCCCH ₂ , i-Pr], [RC7157; F, H, Cl, Cl, HCCCH ₂ , c-Pr], [RC7158; F, H, Cl, Cl, HCCCH ₂ , Bu], [RC7159; F, H, Cl, Cl, HCCCH ₂ , i-Bu], [RC7160; F, H, Cl, Cl, HCCCH ₂ , t-Bu], [RC7161; F, H, Cl, Cl, HCCCH ₂ , c-PrCH ₂ ], [RC7162; F, H, Cl, Cl, HCCCH ₂ , Ph], [RC7163; F, H, Cl, Cl, HCCCH ₂ , Bn], [RC7164; F, H, Cl, Cl, HCCCH ₂ , CF ₃ ], [RC7165; F, H, Cl, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RC7166; F, H, Cl, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RC7167; F, H, Cl, Cl, HCCCH ₂ , CF ₂ H], [RC7168; F, H, Cl, Cl, HCCCH ₂ , CF ₂ HCF ₂ ], [RC7169; F, H, H, H, CH ₃ CCCH ₂ , Me], [RC7170; F, H, H, H, CH ₃ CCCH ₂ , Et], [ RC7171; F, H, H, H, CH ₃ CCCH ₂ , Pr], [RC7172; F, H, H, H, CH ₃ CCCH ₂ , i-Pr], [RC7173; F, H, H, H, CH ₃ CCCH ₂ , c-Pr], [RC7174; F, H, H, H, CH ₃ CCCH ₂ , Bu], [RC7175; F, H, H, H, CH ₃ CCCH ₂ , i-Bu], [RC7176; F, H, H, H, CH ₃ CCCH ₂ , t-Bu], [RC7177; F, H, H, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC7178; F, H, H, H, CH ₃ CCCH ₂ , Ph], [RC7179; F, H, H, H, CH ₃ CCCH ₂ , Bn], [RC7180; F, H, H, H, CH ₃ CCCH ₂ , CF ₃ ] , [RC7181; F, H, H , H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC7182; F, H, H, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC7183; F, H, H, H, CH ₃ CCCH ₂ , CF ₂ H], [RC7184; F, H, H, H, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC7185; F, H, H, Me, CH ₃ CCCH ₂ , Me], [RC7186 ; F, H, H, Me, CH ₃ CCCH ₂ , Et], [RC7187; F, H, H, Me, CH ₃ CCCH ₂ , Pr], [RC7188; F, H, H, Me, CH ₃ CCCH ₂ , i-Pr], [RC7189; F, H, H, Me, CH ₃ CCCH ₂ , c-Pr], [RC7190; F, H, H, Me, CH ₃ CCCH ₂ , Bu], [RC7191; F, H, H, Me, CH ₃ CCCH ₂ , i-Bu], [RC7192; F, H, H, Me, CH ₃ CCCH ₂ , t-Bu], [RC7193; F, H, H, Me, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC7194; F, H, H, Me, CH ₃ CCCH ₂ , Ph], [RC7195; F, H, H, Me, CH ₃ CCCH ₂ , Bn], [ RC7196; F, H, H, Me, CH ₃ CCCH ₂ , CF ₃ ], [RC7197; F, H, H, Me, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC7198; F, H, H, Me, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC7199; F, H, H, Me, CH ₃ CCCH ₂ , CF ₂ H], [RC7200; F, H, H, Me, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ],

[RC7201; F, H, Me, Me, CH ₃ CCCH ₂ , Me], [RC7202; F, H, Me, Me, CH ₃ CCCH ₂ , Et], [RC7203; F, H, Me, Me, CH ₃ CCCH ₂ , Pr], [RC7204; F, H, Me, Me, CH ₃ CCCH ₂ , i-Pr], [RC7205; F, H, Me, Me, CH ₃ CCCH ₂ , c-Pr], [ RC7206; F, H, Me, Me, CH ₃ CCCH ₂ , Bu], [RC7207; F, H, Me, Me, CH ₃ CCCH ₂ , i-Bu], [RC7208; F, H, Me, Me, CH ₃ CCCH ₂ , t-Bu], [RC7209; F, H, Me, Me, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC7210; F, H, Me, Me, CH ₃ CCCH ₂ , Ph] , [RC7211; F, H, Me, Me, CH ₃ CCCH ₂ , Bn], [RC7212; F, H, Me, Me, CH ₃ CCCH ₂ , CF ₃ ], [RC7213; F, H, Me, Me , CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC7214; F, H, Me, Me, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC7215; F, H, Me, Me, CH ₃ CCCH ₂ , CF ₂ H], [RC7216; F, H, Me, Me, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC7217; F, H, Me, Et, CH ₃ CCCH ₂ , Me], [RC7218; F , H, Me, Et, CH ₃ CCCH ₂ , Et], [RC7219; F, H, Me, Et, CH ₃ CCCH ₂ , Pr], [RC7220; F, H, Me, Et, CH ₃ CCCH ₂ , i-Pr], [RC7221; F, H, Me, Et, CH ₃ CCCH ₂ , c-Pr], [RC7222; F, H, Me, Et, CH ₃ CCCH ₂ , Bu], [RC7223; F, H, Me, Et, CH ₃ CCCH ₂ , i-Bu], [RC7224; F, H, Me, Et, CH ₃ CCCH ₂ , t-Bu], [RC7225; F, H, Me, Et, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC7226; F, H, Me, Et, CH ₃ CCCH ₂ , Ph], [RC7227; F, H, Me, Et, CH ₃ CCCH ₂ , Bn], [RC7228; F, H, Me, Et, CH ₃ CCCH ₂ , CF ₃ ], [RC7229; F, H, Me, Et, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC7230; F, H, Me, Et, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC7231; F, H, Me, Et, CH ₃ CCCH ₂ , CF ₂ H], [RC7232; F, H, Me, Et , CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC7233; F, H, Me, F, CH ₃ CCCH ₂ , Me], [RC7234; F, H, Me, F, CH ₃ CCCH ₂ , Et], [RC7235; F, H, Me, F, CH ₃ CCCH ₂ , Pr], [RC7236; F, H, Me, F, CH ₃ CCCH ₂ , i-Pr], [RC7237; F, H, Me, F , CH ₃ CCCH ₂ , c-Pr], [RC7238; F, H, Me, F, CH ₃ CCCH ₂ , Bu], [RC7239; F, H, Me, F, CH ₃ CCCH ₂ , i-Bu] , [RC7240; F, H, Me, F, CH ₃ CCCH ₂ , t-Bu], [RC7241; F, H, Me, F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC7242; F, H , Me, F, CH ₃ CCCH ₂ , Ph], [RC7243; F, H, Me, F, CH ₃ CCCH ₂ , Bn], [RC7244; F, H, Me, F, CH ₃ CCCH ₂ , CF ₃ ], [RC7245; F, H, Me, F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC7246; F, H, Me, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC7247; F , H, Me, F, CH ₃ CCCH ₂ , CF ₂ H], [RC7248; F, H, Me, F, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC7249; F, H, Me, Cl, CH ₃ CCCH ₂ , Me], [RC7250; F, H, Me, Cl, CH ₃ CCCH ₂ , Et], [RC7251; F, H, Me, Cl, CH ₃ CCCH ₂ , Pr], [RC7252; F , H, Me, Cl, CH ₃ CCCH ₂ , i-Pr], [RC7253; F, H, Me, Cl, CH ₃ CCCH ₂ , c-Pr], [RC7254; F, H, Me, C l, CH ₃ CCCH ₂ , Bu], [RC7255; F, H, Me, Cl, CH ₃ CCCH ₂ , i-Bu], [RC7256; F, H, Me, Cl, CH ₃ CCCH ₂ , t-Bu ], [RC7257; F, H, Me, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC7258; F, H, Me, Cl, CH ₃ CCCH ₂ , Ph], [RC7259; F, H, Me, Cl, CH ₃ CCCH ₂ , Bn], [RC7260; F, H, Me, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RC7261; F, H, Me, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC7262; F, H, Me, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC7263; F, H, Me, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RC7264; F, H, Me, Cl, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC7265; F, H, Et, H, CH ₃ CCCH ₂ , Me], [RC7266; F, H, Et, H, CH ₃ CCCH ₂ , Et], [RC7267; F, H, Et, H, CH ₃ CCCH ₂ , Pr], [RC7268; F, H, Et, H, CH ₃ CCCH ₂ , i-Pr], [RC7269; F, H, Et, H, CH ₃ CCCH ₂ , c-Pr], [RC7270; F, H, Et, H, CH ₃ CCCH ₂ , Bu], [RC7271; F, H, Et, H, CH ₃ CCCH ₂ , i-Bu], [RC7272; F, H, Et, H, CH ₃ CCCH ₂ , t-Bu], [RC7273; F, H, Et, H, CH ₃ CCCH ₂ , c-PrCH ₂ ] , [RC7274; F, H, Et, H, CH ₃ CCCH ₂ , Ph], [RC7275; F, H, Et, H, CH ₃ CCCH ₂ , Bn], [RC7276; F, H, Et, H, CH ₃ CCCH ₂ , CF ₃ ], [RC7277; F, H, Et, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC7278; F, H, Et, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC7279; F, H, Et, H, CH ₃ CCCH ₂ , CF ₂ H], [RC7280; F, H, Et, H, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC7281; F, H, Et, F, CH ₃ CCCH ₂ , Me], [RC7282; F, H, Et, F, CH ₃ CCCH ₂ , Et], [RC7283; F, H, Et, F , CH ₃ CCCH ₂ , Pr], [RC7284; F, H, Et, F, CH ₃ CCCH ₂ , i-Pr], [RC7285; F, H, Et, F, CH ₃ CCCH ₂ , c-Pr] , [RC7286; F, H, Et, F, CH ₃ CCCH ₂ , Bu], [RC7287; F, H, Et, F, CH ₃ CCCH ₂ , i-Bu], [RC7288; F, H, Et, F, CH ₃ CCCH ₂ , t-Bu], [RC7289; F, H, Et, F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC7290; F, H, Et, F, CH ₃ CCCH ₂ , Ph], [RC7291; F, H, Et, F, CH ₃ CCCH ₂ , Bn], [RC7292; F, H, Et, F, CH ₃ CCCH ₂ , CF ₃ ], [RC7293; F, H, Et , F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC7294; F, H, Et, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC7295; F, H, Et, F, CH ₃ CCCH ₂ , CF ₂ H], [RC7296; F, H, Et, F, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC7297; F, H, Et, Cl, CH ₃ CCCH ₂ , Me], [RC7298 ; F, H, Et, Cl, CH ₃ CCCH ₂ , Et], [RC7299; F, H, Et, Cl, CH ₃ CCCH ₂ , Pr], [RC7300; F, H, Et, Cl, CH ₃ CCCH ₂ , i-Pr], [RC7301; F, H, Et, Cl, CH ₃ CCCH ₂ , c-Pr], [RC7302; F, H, Et, Cl, CH ₃ CCCH ₂ , Bu], [RC7303; F, H, Et, Cl, CH ₃ CCCH ₂ , i-Bu], [RC7304; F, H, Et, Cl, CH ₃ CCCH ₂ , t-Bu], [RC7305; F, H, Et, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC7306; F, H, Et, Cl, CH ₃ CCCH ₂ , Ph], [RC7307; F, H, Et, Cl, CH ₃ CCCH ₂ , Bn], [ RC730 8; F, H, Et, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RC7309; F, H, Et, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC7310; F, H, Et, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC7311; F, H, Et, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RC7312; F, H, Et, Cl, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC7313; F, H, F, H, CH ₃ CCCH ₂ , Me], [RC7314; F, H, F, H, CH ₃ CCCH ₂ , Et], [RC7315; F, H , F, H, CH ₃ CCCH ₂ , Pr], [RC7316; F, H, F, H, CH ₃ CCCH ₂ , i-Pr], [RC7317; F, H, F, H, CH ₃ CCCH ₂ , c-Pr], [RC7318; F, H, F, H, CH ₃ CCCH ₂ , Bu], [RC7319; F, H, F, H, CH ₃ CCCH ₂ , i-Bu], [RC7320; F, H, F, H, CH ₃ CCCH ₂ , t-Bu], [RC7321; F, H, F, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC7322; F, H, F, H, CH ₃ CCCH ₂ , Ph], [RC7323; F, H, F, H, CH ₃ CCCH ₂ , Bn], [RC7324; F, H, F, H, CH ₃ CCCH ₂ , CF ₃ ], [RC7325; F , H, F, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC7326; F, H, F, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC7327; F, H, F, H , CH ₃ CCCH ₂ , CF ₂ H], [RC7328; F, H, F, H, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC7329; F, H, F, F, CH ₃ CCCH ₂ , Me ], [RC7330; F, H, F, F, CH ₃ CCCH ₂ , Et], [RC7331; F, H, F, F, CH ₃ CCCH ₂ , Pr], [RC7332; F, H, F, F , CH ₃ CCCH ₂ , i-Pr], [RC7333; F, H, F, F, CH ₃ CCCH ₂ , c-Pr], [RC7334; F, H, F, F, CH ₃ CCCH ₂ , Bu] , [RC7335; F, H, F, F, CH ₃ C CCH ₂ , i-Bu], [RC7336; F, H, F, F, CH ₃ CCCH ₂ , t-Bu], [RC7337; F, H, F, F, CH ₃ CCCH ₂ , c-PrCH ₂ ] , [RC7338; F, H, F, F, CH ₃ CCCH ₂ , Ph], [RC7339; F, H, F, F, CH ₃ CCCH ₂ , Bn], [RC7340; F, H, F, F, CH ₃ CCCH ₂ , CF ₃ ], [RC7341; F, H, F, F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC7342; F, H, F, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC7343; F, H, F, F, CH ₃ CCCH ₂ , CF ₂ H], [RC7344; F, H, F, F, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC7345; F , H, F, Cl, CH ₃ CCCH ₂ , Me], [RC7346; F, H, F, Cl, CH ₃ CCCH ₂ , Et], [RC7347; F, H, F, Cl, CH ₃ CCCH ₂ , Pr], [RC7348; F, H, F, Cl, CH ₃ CCCH ₂ , i-Pr], [RC7349; F, H, F, Cl, CH ₃ CCCH ₂ , c-Pr], [RC7350; F, H, F, Cl, CH ₃ CCCH ₂ , Bu], [RC7351; F, H, F, Cl, CH ₃ CCCH ₂ , i-Bu], [RC7352; F, H, F, Cl, CH ₃ CCCH ₂ , t-Bu], [RC7353; F, H, F, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC7354; F, H, F, Cl, CH ₃ CCCH ₂ , Ph], [RC7355; F, H, F, Cl, CH ₃ CCCH ₂ , Bn], [RC7356; F, H, F, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RC7357; F, H, F, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC7358; F, H, F, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC7359; F, H, F, Cl, CH ₃ CCCH ₂ , CF ₂ H] , [RC7360; F, H, F, Cl, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC7361; F, H, Cl, H, CH ₃ CCCH ₂ , Me], [RC7362; F, H, Cl , H, CH ₃ CC _{CH 2, Et], [RC7363} ; F, H, Cl, H, CH 3 CCCH 2, Pr], [RC7364; F, H, Cl, H, CH 3 CCCH 2, i-Pr], [RC7365; F , H, Cl, H, CH ₃ CCCH ₂ , c-Pr], [RC7366; F, H, Cl, H, CH ₃ CCCH ₂ , Bu], [RC7367; F, H, Cl, H, CH ₃ CCCH ₂ , i-Bu], [RC7368; F, H, Cl, H, CH ₃ CCCH ₂ , t-Bu], [RC7369; F, H, Cl, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC7370; F, H, Cl, H, CH ₃ CCCH ₂ , Ph], [RC7371; F, H, Cl, H, CH ₃ CCCH ₂ , Bn], [RC7372; F, H, C
l, H, CH ₃ CCCH ₂ , CF ₃ ], [RC7373; F, H, Cl, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC7374; F, H, Cl, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC7375; F, H, Cl, H, CH ₃ CCCH ₂ , CF ₂ H], [RC7376; F, H, Cl, H, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC7377; F, H, Cl, Cl, CH ₃ CCCH ₂ , Me], [RC7378; F, H, Cl, Cl, CH ₃ CCCH ₂ , Et], [RC7379; F, H, Cl, Cl, CH ₃ CCCH ₂ , Pr], [RC7380; F, H, Cl, Cl, CH ₃ CCCH ₂ , i-Pr], [RC7381; F, H, Cl, Cl, CH ₃ CCCH ₂ , c-Pr], [ RC7382; F, H, Cl, Cl, CH ₃ CCCH ₂ , Bu], [RC7383; F, H, Cl, Cl, CH ₃ CCCH ₂ , i-Bu], [RC7384; F, H, Cl, Cl, CH ₃ CCCH ₂ , t-Bu], [RC7385; F, H, Cl, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC7386; F, H, Cl, Cl, CH ₃ CCCH ₂ , Ph] , [RC7387; F, H, Cl, Cl, CH ₃ CCCH ₂ , Bn], [RC7388; F, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RC7389; F, H, Cl, Cl , CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC7390; F, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC7391; F, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RC7392; F, H, Cl, Cl, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC7393; F, H, H, H, c-Pr, Me], [RC7394; F, H, H, H, c-Pr, Et], [RC7395; F, H, H, H, c-Pr, Pr], [RC7396; F, H, H, H, c-Pr, i-Pr] , [RC7397; F, H, H, H, c-Pr, c-Pr], [RC7398; F, H, H, H, c-Pr, Bu], [RC7399; F, H, H, H, c-Pr, i-Bu], [RC7400; F, H, H, H, c-Pr, t- Bu],

[RC7401; F, H, H, H, c-Pr, c-PrCH ₂ ], [RC7402; F, H, H, H, c-Pr, Ph], [RC7403; F, H, H, H, c-Pr, Bn], [RC7404; F, H, H, H, c-Pr, CF ₃ ], [RC7405; F, H, H, H, c-Pr, CF ₃ CH ₂ ], [RC7406; F, H, H, H, c-Pr, CF ₃ CF ₂ ], [RC7407; F, H, H, H, c-Pr, CF ₂ H], [RC7408; F, H, H, H, c -Pr, CF ₂ HCF ₂ ], [RC7409; F, H, H, Me, c-Pr, Me], [RC7410; F, H, H, Me, c-Pr, Et], [RC7411; F, H, H, Me, c-Pr, Pr], [RC7412; F, H, H, Me, c-Pr, i-Pr], [RC7413; F, H, H, Me, c-Pr, c- Pr], [RC7414; F, H, H, Me, c-Pr, Bu], [RC7415; F, H, H, Me, c-Pr, i-Bu], [RC7416; F, H, H, Me, c-Pr, t-Bu], [RC7417; F, H, H, Me, c-Pr, c-PrCH ₂ ], [RC7418; F, H, H, Me, c-Pr, Ph], [RC7419; F, H, H, Me, c-Pr, Bn], [RC7420; F, H, H, Me, c-Pr, CF ₃ ], [RC7421; F, H, H, Me, c- Pr, CF ₃ CH ₂ ], [RC7422; F, H, H, Me, c-Pr, CF ₃ CF ₂ ], [RC7423; F, H, H, Me, c-Pr, CF ₂ H], [ RC7424; F, H, H, Me, c-Pr, CF ₂ HCF ₂ ], [RC7425; F, H, Me, Me, c-Pr, Me], [RC7426; F, H, Me, Me, c -Pr, Et], [RC7427; F, H, Me, Me, c-Pr, Pr], [RC7428; F, H, Me, Me, c-Pr, i-Pr], [RC7429; F, H , Me, Me, c-Pr, c-Pr], [RC7430; F, H, Me, Me, c-Pr, Bu], [RC7431; F, H, Me, Me, c-Pr, i-Bu ], [RC7432; F, H, Me, Me, c-Pr, t-Bu], [RC7433; F, H, Me, Me, c-Pr, c-PrCH ₂ ], [RC7434; F, H, Me, Me, c-Pr, Ph], [RC7435; F, H, M e, Me, c-Pr, Bn], [RC7436; F, H, Me, Me, c-Pr, CF ₃ ], [RC7437; F, H, Me, Me, c-Pr, CF ₃ CH ₂ ] , [RC7438; F, H, Me, Me, c-Pr, CF ₃ CF ₂ ], [RC7439; F, H, Me, Me, c-Pr, CF ₂ H], [RC7440; F, H, Me , Me, c-Pr, CF ₂ HCF ₂ ], [RC7441; F, H, Me, Et, c-Pr, Me], [RC7442; F, H, Me, Et, c-Pr, Et], [ RC7443; F, H, Me, Et, c-Pr, Pr], [RC7444; F, H, Me, Et, c-Pr, i-Pr], [RC7445; F, H, Me, Et, c- Pr, c-Pr], [RC7446; F, H, Me, Et, c-Pr, Bu], [RC7447; F, H, Me, Et, c-Pr, i-Bu], [RC7448; F, H, Me, Et, c-Pr, t-Bu], [RC7449; F, H, Me, Et, c-Pr, c-PrCH ₂ ], [RC7450; F, H, Me, Et, c-Pr , Ph], [RC7451; F, H, Me, Et, c-Pr, Bn], [RC7452; F, H, Me, Et, c-Pr, CF ₃ ], [RC7453; F, H, Me, Et, c-Pr, CF ₃ CH ₂ ], [RC7454; F, H, Me, Et, c-Pr, CF ₃ CF ₂ ], [RC7455; F, H, Me, Et, c-Pr, CF ₂ H], [RC7456; F, H, Me, Et, c-Pr, CF ₂ HCF ₂ ], [RC7457; F, H, Me, F, c-Pr, Me], [RC7458; F, H, Me , F, c-Pr, Et], [RC7459; F, H, Me, F, c-Pr, Pr], [RC7460; F, H, Me, F, c-Pr, i-Pr], [RC7461 ; F, H, Me, F, c-Pr, c-Pr], [RC7462; F, H, Me, F, c-Pr, Bu], [RC7463; F, H, Me, F, c-Pr , i-Bu], [RC7464; F, H, Me, F, c-Pr, t-Bu], [RC7465; F, H, Me, F, c-Pr, c-PrCH ₂ ], [RC7466; F, H, Me, F, c-Pr, Ph], [RC7467; F, H, Me, F, c-Pr, Bn], [RC7468; F, H, Me, F, c-Pr, CF ₃ ], [RC7469; F, H, Me, F, c-Pr, CF ₃ CH ₂ ], [RC7470; F, H, Me, F, c-Pr, CF ₃ CF ₂ ], [RC7471; F, H, Me, F, c- Pr, CF ₂ H], [RC7472; F, H, Me, F, c-Pr, CF ₂ HCF ₂ ], [RC7473; F, H, Me, Cl, c-Pr, Me], [RC7474; F , H, Me, Cl, c-Pr, Et], [RC7475; F, H, Me, Cl, c-Pr, Pr], [RC7476; F, H, Me, Cl, c-Pr, i-Pr ], [RC7477; F, H, Me, Cl, c-Pr, c-Pr], [RC7478; F, H, Me, Cl, c-Pr, Bu], [RC7479; F, H, Me, Cl , c-Pr, i-Bu], [RC7480; F, H, Me, Cl, c-Pr, t-Bu], [RC7481; F, H, Me, Cl, c-Pr, c-PrCH ₂ ] , [RC7482; F, H, Me, Cl, c-Pr, Ph], [RC7483; F, H, Me, Cl, c-Pr, Bn], [RC7484; F, H, Me, Cl, c- Pr, CF ₃ ], [RC7485; F, H, Me, Cl, c-Pr, CF ₃ CH ₂ ], [RC7486; F, H, Me, Cl, c-Pr, CF ₃ CF ₂ ], [RC7487 ; F, H, Me, Cl, c-Pr, CF ₂ H], [RC7488; F, H, Me, Cl, c-Pr, CF ₂ HCF ₂ ], [RC7489; F, H, Et, H, c-Pr, Me], [RC7490; F, H, Et, H, c-Pr, Et], [RC7491; F, H, Et, H, c-Pr, Pr], [RC7492; F, H, Et, H, c-Pr, i-Pr], [RC7493; F, H, Et, H, c-Pr, c-Pr], [RC7494; F, H, Et, H, c-Pr, Bu] , [RC7495; F, H, Et, H, c-Pr, i-Bu], [RC7496; F, H, Et, H, c-Pr, t-Bu], [RC7497; F, H, Et, H, c-Pr, c-PrCH ₂ ], [RC7498; F, H, Et, H, c-Pr, Ph], [RC7499; F, H, Et, H, c-Pr, Bn], [RC7500 ; F, H, Et, H, c-Pr, CF ₃ ], [RC7501; F, H, Et, H, c-Pr, CF ₃ CH ₂ ], [RC7502; F, H, Et, H, c -Pr, CF ₃ CF ₂ ], [RC7503; F, H, Et, H, c-Pr, CF ₂ H], [RC7504; F, H, Et, H, c-Pr, CF ₂ HCF ₂ ], [RC7505; F, H, Et, F, c-Pr, Me], [RC7506; F, H, Et, F, c-Pr, Et], [RC7507; F, H, Et, F, c-Pr, Pr], [RC7508; F, H, Et, F, c-Pr, i-Pr], [RC7509; F, H, Et, F, c-Pr, c-Pr], [RC7510; F, H, Et, F, c-Pr, Bu], [RC7511; F, H, Et, F, c-Pr, i-Bu], [RC7512; F, H, Et, F, c-Pr, t-Bu], [RC7513; F, H, Et, F, c-Pr, c-PrCH ₂ ], [RC7514; F, H, Et, F, c-Pr, Ph], [RC7515; F, H, Et, F, c-Pr, Bn], [RC7516; F, H, Et, F, c-Pr, CF ₃ ], [RC7517; F, H, Et, F, c-Pr, CF ₃ CH ₂ ], [RC7518; F, H, Et, F , c-Pr, CF ₃ CF ₂ ], [RC7519; F, H, Et, F, c-Pr, CF ₂ H], [RC7520; F, H, Et, F, c-Pr, CF ₂ HCF ₂ ], [RC7521; F, H, Et, Cl, c-Pr, Me], [RC7522; F, H, Et, Cl, c-Pr, Et], [RC7523; F, H, Et, Cl, c -Pr, Pr], [RC7524; F, H, Et, Cl, c-Pr, i-Pr], [RC7525; F, H, Et, Cl, c-Pr, c-Pr], [RC7526; F , H, Et, Cl, c-Pr, Bu], [RC7527; F, H, Et, Cl, c-Pr, i-Bu], [RC7528; F, H, Et, Cl, c-Pr, t -Bu], [RC7529; F, H, Et, Cl, c-Pr, c-PrCH ₂ ], [RC7530; F, H, Et, Cl, c-Pr, Ph], [RC7531; F, H, Et, Cl, c-Pr, Bn], [RC7532; F, H, Et, Cl, c-Pr, CF ₃ ], [RC7533; F, H, Et, Cl, c-Pr, CF ₃ CH ₂ ] , [RC7534; F, H, Et, Cl, c-Pr, CF ₃ CF ₂ ], [RC7535; F, H, Et, Cl, c-Pr, CF ₂ H], [RC7536; F, H, Et , Cl, c-Pr, CF ₂ H CF ₂ ], [RC7537; F, H, F, H, c-Pr, Me], [RC7538; F, H, F, H, c-Pr, Et], [RC7539; F, H, F, H , c-Pr, Pr], [RC7540; F, H, F, H, c-Pr, i-Pr], [RC7541; F, H, F, H, c-Pr, c-Pr], [RC7542 ; F, H, F, H, c-Pr, Bu], [RC7543; F, H, F, H, c-Pr, i-Bu], [RC7544; F, H, F, H, c-Pr , t-Bu], [RC7545; F, H, F, H, c-Pr, c-PrCH ₂ ], [RC7546; F, H, F, H, c-Pr, Ph], [RC7547; F, H, F, H, c-Pr, Bn], [RC7548; F, H, F, H, c-Pr, CF ₃ ], [RC7549; F, H, F, H, c-Pr, CF ₃ CH ₂ ], [RC7550; F, H, F, H, c-Pr, CF ₃ CF ₂ ], [RC7551; F, H, F, H, c-Pr, CF ₂ H], [RC7552; F, H , F, H, c-Pr, CF ₂ HCF ₂ ], [RC7553; F, H, F, F, c-Pr, Me], [RC7554; F, H, F, F, c-Pr, Et] , [RC7555; F, H, F, F, c-Pr, Pr], [RC7556; F, H, F, F, c-Pr, i-Pr], [RC7557; F, H, F, F, c-Pr, c-Pr], [RC7558; F, H, F, F, c-Pr, Bu], [RC7559; F, H, F, F, c-Pr, i-Bu], [RC7560; F, H, F, F, c-Pr, t-Bu], [RC7561; F, H, F, F, c-Pr, c-PrCH ₂ ], [RC7562; F, H, F, F, c -Pr, Ph], [RC7563; F, H, F, F, c-Pr, Bn], [RC7564; F, H, F, F, c-Pr, CF ₃ ], [RC7565; F, H, F, F, c-Pr, CF ₃ CH ₂ ], [RC7566; F, H, F, F, c-Pr, CF ₃ CF ₂ ], [RC7567; F, H, F, F, c-Pr, CF ₂ H], [RC7568; F, H, F, F, c-Pr, CF ₂ HCF ₂ ], [RC7569; F, H, F, Cl, c-Pr, Me], [RC7570; F, H , F, Cl, c-Pr, Et], [RC7571; F, H, F, Cl, c-Pr, Pr], [RC7572; F, H, F, Cl, c-Pr , i-Pr], [RC7573; F, H, F, Cl, c-Pr, c-Pr], [RC7574; F, H, F, Cl, c-Pr, Bu], [RC7575; F, H , F, Cl, c-Pr, i-Bu], [RC7576; F, H, F, Cl, c-Pr, t-Bu], [RC7577; F, H, F, Cl, c-Pr, c -PrCH ₂ ], [RC7578; F, H, F, Cl, c-Pr, Ph], [RC7579; F, H, F, Cl, c-Pr, Bn], [RC7580; F, H, F, Cl, c-Pr, CF ₃ ], [RC7581; F, H, F, Cl, c-Pr, CF ₃ CH ₂ ], [RC7582; F, H, F, Cl, c-Pr, CF ₃ CF ₂ ], [RC7583; F, H, F, Cl, c-Pr, CF ₂ H], [RC7584; F, H, F, Cl, c-Pr, CF ₂ HCF ₂ ], [RC7585; F, H, Cl, H, c-Pr, Me], [RC7586; F, H, Cl, H, c-Pr, Et], [RC7587; F, H, Cl, H, c-Pr, Pr], [RC7588; F, H, Cl, H, c-Pr, i-Pr], [RC7589; F, H, Cl, H, c-Pr, c-Pr], [RC7590; F, H, Cl, H, c- Pr, Bu], [RC7591; F, H, Cl, H, c-Pr, i-Bu], [RC7592; F, H, Cl, H, c-Pr, t-Bu], [RC7593; F, H, Cl, H, c-Pr, c-PrCH ₂ ], [RC7594; F, H, Cl, H, c-Pr, Ph], [RC7595; F, H, Cl, H, c-Pr, Bn ], [RC7596; F, H, Cl, H, c-Pr, CF ₃ ], [RC7597; F, H, Cl, H, c-Pr, CF ₃ CH ₂ ], [RC7598; F, H, Cl , H, c-Pr, CF ₃ CF ₂ ], [RC7599; F, H, Cl, H, c-Pr, CF ₂ H], [RC7600; F, H, Cl, H, c-Pr, CF ₂ HCF ₂ ],

[RC7601; F, H, Cl, Cl, c-Pr, Me], [RC7602; F, H, Cl, Cl, c-Pr, Et], [RC7603; F, H, Cl, Cl, c-Pr , Pr], [RC7604; F, H, Cl, Cl, c-Pr, i-Pr], [RC7605; F, H, Cl, Cl, c-Pr, c-Pr], [RC7606; F, H , Cl, Cl, c-Pr, Bu], [RC7607; F, H, Cl, Cl, c-Pr, i-Bu], [RC7608; F, H, Cl, Cl, c-Pr, t-Bu ], [RC7609; F, H, Cl, Cl, c-Pr, c-PrCH ₂ ], [RC7610; F, H, Cl, Cl, c-Pr, Ph], [RC7611; F, H, Cl, Cl, c-Pr, Bn], [RC7612; F, H, Cl, Cl, c-Pr, CF ₃ ], [RC7613; F, H, Cl, Cl, c-Pr, CF ₃ CH ₂ ], [ RC7614; F, H, Cl, Cl, c-Pr, CF ₃ CF ₂ ], [RC7615; F, H, Cl, Cl, c-Pr, CF ₂ H], [RC7616; F, H, Cl, Cl , c-Pr, CF ₂ HCF ₂ ], [RC7617; F, H, H, H, Bn, Me], [RC7618; F, H, H, H, Bn, Et], [RC7619; F, H, H, H, Bn, Pr], [RC7620; F, H, H, H, Bn, i-Pr], [RC7621; F, H, H, H, Bn, c-Pr], [RC7622; F, H, H, H, Bn, Bu], [RC7623; F, H, H, H, Bn, i-Bu], [RC7624; F, H, H, H, Bn, t-Bu], [RC7625; F, H, H, H, Bn, c-PrCH ₂ ], [RC7626; F, H, H, H, Bn, Ph], [RC7627; F, H, H, H, Bn, Bn], [RC7628 ; F, H, H, H, Bn, CF ₃ ], [RC7629; F, H, H, H, Bn, CF ₃ CH ₂ ], [RC7630; F, H, H, H, Bn, CF ₃ CF ₂ ], [RC7631; F, H, H, H, Bn, CF ₂ H], [RC7632; F, H, H, H, Bn, CF ₂ HCF ₂ ], [RC7633; F, H, H, Me , Bn, Me], [RC7634; F, H, H, Me, Bn, Et], [RC7635; F, H, H, Me, Bn, Pr], [RC7636; F, H, H, Me, Bn , i-Pr], [RC7637; F, H, H, Me, Bn, c-Pr], [RC7638; F, H, H, Me, Bn, Bu], [RC7639; F, H, H, Me, Bn, i-Bu], [ RC7640; F, H, H, Me, Bn, t-Bu], [RC7641; F, H, H, Me, Bn, c-PrCH ₂ ], [RC7642; F, H, H, Me, Bn, Ph ], [RC7643; F, H, H, Me, Bn, Bn], [RC7644; F, H, H, Me, Bn, CF ₃ ], [RC7645; F, H, H, Me, Bn, CF ₃ CH ₂ ], [RC7646; F, H, H, Me, Bn, CF ₃ CF ₂ ], [RC7647; F, H, H, Me, Bn, CF ₂ H], [RC7648; F, H, H, Me, Bn, CF ₂ HCF ₂ ], [RC7649; F, H, Me, Me, Bn, Me], [RC7650; F, H, Me, Me, Bn, Et], [RC7651; F, H, Me , Me, Bn, Pr], [RC7652; F, H, Me, Me, Bn, i-Pr], [RC7653; F, H, Me, Me, Bn, c-Pr], [RC7654; F, H , Me, Me, Bn, Bu], [RC7655; F, H, Me, Me, Bn, i-Bu], [RC7656; F, H, Me, Me, Bn, t-Bu], [RC7657; F , H, Me, Me, Bn, c-PrCH ₂ ], [RC7658; F, H, Me, Me, Bn, Ph], [RC7659; F, H, Me, Me, Bn, Bn], [RC7660; F, H, Me, Me, Bn, CF ₃ ], [RC7661; F, H, Me, Me, Bn, CF ₃ CH ₂ ], [RC7662; F, H, Me, Me, Bn, CF ₃ CF ₂ ], [RC7663; F, H, Me, Me, Bn, CF ₂ H], [RC7664; F, H, Me, Me, Bn, CF ₂ HCF ₂ ], [RC7665; F, H, Me, Et, Bn, Me], [RC7666; F, H, Me, Et, Bn, Et], [RC7667; F, H, Me, Et, Bn, Pr], [RC7668; F, H, Me, Et, Bn, i-Pr], [RC7669; F, H, Me, Et, Bn, c-Pr], [RC7670; F, H, Me, Et, Bn, Bu], [RC7671; F, H, Me, Et, Bn, i-Bu], [RC7672; F, H, Me, Et, Bn, t-Bu], [RC7673; F, H, Me, Et, Bn , c-PrCH ₂ ], [RC7674; F, H, Me, Et, Bn, Ph], [RC7675; F, H, Me, Et, Bn, Bn], [RC7676; F, H, Me, Et, Bn, CF ₃ ], [RC7677; F, H, Me, Et, Bn, CF ₃ CH ₂ ], [RC7678; F, H, Me, Et, Bn, CF ₃ CF ₂ ], [RC7679; F, H , Me, Et, Bn, CF ₂ H], [RC7680; F, H, Me, Et, Bn, CF ₂ HCF ₂ ], [RC7681; F, H, Me, F, Bn, Me], [RC7682; F, H, Me, F, Bn, Et], [RC7683; F, H, Me, F, Bn, Pr], [RC7684; F, H, Me, F, Bn, i-Pr], [RC7685; F, H, Me, F, Bn, c-Pr], [RC7686; F, H, Me, F, Bn, Bu], [RC7687; F, H, Me, F, Bn, i-Bu], [ RC7688; F, H, Me, F, Bn, t-Bu], [RC7689; F, H, Me, F, Bn, c-PrCH ₂ ], [RC7690; F, H, Me, F, Bn, Ph ], [RC7691; F, H, Me, F, Bn, Bn], [RC7692; F, H, Me, F, Bn, CF ₃ ], [RC7693; F, H, Me, F, Bn, CF ₃ CH ₂ ], [RC7694; F, H, Me, F, Bn, CF ₃ CF ₂ ], [RC7695; F, H, Me, F, Bn, CF ₂ H], [RC7696; F, H, Me, F, Bn, CF ₂ HCF ₂ ], [RC7697; F, H, Me, Cl, Bn, Me], [RC7698; F, H, Me, Cl, Bn, Et], [RC7699; F, H, Me , Cl, Bn, Pr], [RC7700; F, H, Me, Cl, Bn, i-Pr], [RC7701; F, H, Me, Cl, Bn, c-Pr], [RC7702; F, H , Me, Cl, Bn, Bu], [RC7703; F, H, Me, Cl, Bn, i-Bu], [RC7704; F, H, Me, Cl, Bn, t-Bu], [RC7705; F , H, Me, Cl, Bn, c-PrCH ₂ ], [RC7706; F, H, Me, Cl, Bn, Ph], [RC7707; F, H, Me, Cl, Bn, Bn], [RC7708; F, H, Me, Cl, Bn, CF ₃ ], [RC7709; F, H, Me, Cl, Bn, CF ₃ CH ₂ ] , [RC7710; F, H, Me, Cl, Bn, CF ₃ CF ₂ ], [RC7711; F, H, Me, Cl, Bn, CF ₂ H], [RC7712; F, H, Me, Cl, Bn , CF ₂ HCF ₂ ], [RC7713; F, H, Et, H, Bn, Me], [RC7714; F, H, Et, H, Bn, Et], [RC7715; F, H, Et, H, Bn, Pr], [RC7716; F, H, Et, H, Bn, i-Pr], [RC7717; F, H, Et, H, Bn, c-Pr], [RC7718; F, H, Et, H, Bn, Bu], [RC7719; F, H, Et, H, Bn, i-Bu], [RC7720; F, H, Et, H, Bn, t-Bu], [RC7721; F, H, Et, H, Bn, c-PrCH ₂ ], [RC7722; F, H, Et, H, Bn, Ph], [RC7723; F, H, Et, H, Bn, Bn], [RC7724; F, H , Et, H, Bn, CF ₃ ], [RC7725; F, H, Et, H, Bn, CF ₃ CH ₂ ], [RC7726; F, H, Et, H, Bn, CF ₃ CF ₂ ], [ RC7727; F, H, Et, H, Bn, CF ₂ H], [RC7728; F, H, Et, H, Bn, CF ₂ HCF ₂ ], [RC7729; F, H, Et, F, Bn, Me ], [RC7730; F, H, Et, F, Bn, Et], [RC7731; F, H, Et, F, Bn, Pr], [RC7732; F, H, Et, F, Bn, i-Pr ], [RC7733; F, H, Et, F, Bn, c-Pr], [RC7734; F, H, Et, F, Bn, Bu], [RC7735; F, H, Et, F, Bn, i -Bu], [RC7736; F, H, Et, F, Bn, t-Bu], [RC7737; F, H, Et, F, Bn, c-PrCH ₂ ], [RC7738; F, H, Et, F, Bn, Ph], [RC7739; F, H, Et, F, Bn, Bn], [RC7740; F, H, Et, F, Bn, CF ₃ ], [RC7741; F, H, Et, F , Bn, CF ₃ CH ₂ ], [RC7742; F, H, Et, F, Bn, CF ₃ CF ₂ ], [RC7743; F, H, Et, F, Bn, CF ₂ H], [RC7744; F , H, Et, F, Bn, CF ₂ HCF ₂ ], [RC7745; F, H, Et, Cl, Bn, Me], [RC7746; F, H, Et, C l, Bn, Et], [RC7747; F, H, Et, Cl, Bn, Pr], [RC7748; F, H, Et, Cl, Bn, i-Pr], [RC7749; F, H, Et, Cl, Bn, c-Pr], [RC7750; F, H, Et, Cl, Bn, Bu], [RC7751; F, H, Et, Cl, Bn, i-Bu], [RC7752; F, H, Et, Cl, Bn, t-Bu], [RC7753; F, H, Et, Cl, Bn, c-PrCH ₂ ], [RC7754; F, H, Et, Cl, Bn, Ph], [RC7755; F , H, Et, Cl, Bn, Bn], [RC7756; F, H, Et, Cl, Bn, CF ₃ ], [RC7757; F, H, Et, Cl, Bn, CF ₃ CH ₂ ], [RC7758 ; F, H, Et, Cl, Bn, CF ₃ CF ₂ ], [RC7759; F, H, Et, Cl, Bn, CF ₂ H], [RC7760; F, H, Et, Cl, Bn, CF ₂ HCF ₂ ], [RC7761; F, H, F, H, Bn, Me], [RC7762; F, H, F, H, Bn, Et], [RC7763; F, H, F, H, Bn, Pr ], [RC7764; F, H, F, H, Bn, i-Pr], [RC7765; F, H, F, H, Bn, c-Pr], [RC7766; F, H, F, H, Bn , Bu], [RC7767; F, H, F, H, Bn, i-Bu], [RC7768; F, H, F, H, Bn, t-Bu], [RC7769; F, H, F, H , Bn, c-PrCH ₂ ], [RC7770; F, H, F, H, Bn, Ph], [RC7771; F, H, F, H, Bn, Bn], [RC7772; F, H, F, H, Bn, CF ₃ ], [RC7773; F, H, F, H, Bn, CF ₃ CH ₂ ], [RC7774; F, H, F, H, Bn, CF ₃ CF ₂ ], [RC7775; F , H, F, H, Bn, CF ₂ H], [RC7776; F, H, F, H, Bn, CF ₂ HCF ₂ ], [RC7777; F, H, F, F, Bn, Me], [ RC7778; F, H, F, F, Bn, Et], [RC7779; F, H, F, F, Bn, Pr], [RC7780; F, H, F, F, Bn, i-Pr], [ RC7781; F, H, F, F, Bn, c-Pr], [RC7782; F, H, F, F, Bn, Bu], [RC7783; F, H, F, F, Bn, i-Bu] , [RC7784; F, H, F, F, Bn, t-Bu], [RC7785; F, H, F, F, Bn, c-PrCH ₂ ], [RC7786; F, H, F, F, Bn, Ph], [RC7787; F , H, F, F, Bn, Bn], [RC7788; F, H, F, F, Bn, CF ₃ ], [RC7789; F, H, F, F, Bn, CF ₃ CH ₂ ], [RC7790 ; F, H, F, F, Bn, CF ₃ CF ₂ ], [RC7791; F, H, F, F, Bn, CF ₂ H], [RC7792; F, H, F, F, Bn, CF ₂ HCF ₂ ], [RC7793; F, H, F, Cl, Bn, Me], [RC7794; F, H, F, Cl, Bn, Et], [RC7795; F, H, F, Cl, Bn, Pr ], [RC7796; F, H, F, Cl, Bn, i-Pr], [RC7797; F, H, F, Cl, Bn, c-Pr], [RC7798; F, H, F, Cl, Bn , Bu], [RC7799; F, H, F, Cl, Bn, i-Bu], [RC7800; F, H, F, Cl, Bn, t-Bu],

[RC7801; F, H, F, Cl, Bn, c-PrCH ₂ ], [RC7802; F, H, F, Cl, Bn, Ph], [RC7803; F, H, F, Cl, Bn, Bn] , [RC7804; F, H, F, Cl, Bn, CF ₃ ], [RC7805; F, H, F, Cl, Bn, CF ₃ CH ₂ ], [RC7806; F, H, F, Cl, Bn, CF ₃ CF ₂ ], [RC7807; F, H, F, Cl, Bn, CF ₂ H], [RC7808; F, H, F, Cl, Bn, CF ₂ HCF ₂ ], [RC7809; F, H, Cl, H, Bn, Me], [RC7810; F, H, Cl, H, Bn, Et], [RC7811; F, H, Cl, H, Bn, Pr], [RC7812; F, H, Cl, H, Bn, i-Pr], [RC7813; F, H, Cl, H, Bn, c-Pr], [RC7814; F, H, Cl, H, Bn, Bu], [RC7815; F, H, Cl, H, Bn, i-Bu], [RC7816; F, H, Cl, H, Bn, t-Bu], [RC7817; F, H, Cl, H, Bn, c-PrCH ₂ ], [RC7818 ; F, H, Cl, H, Bn, Ph], [RC7819; F, H, Cl, H, Bn, Bn], [RC7820; F, H, Cl, H, Bn, CF ₃ ], [RC7821; F, H, Cl, H, Bn, CF ₃ CH ₂ ], [RC7822; F, H, Cl, H, Bn, CF ₃ CF ₂ ], [RC7823; F, H, Cl, H, Bn, CF ₂ H], [RC7824; F, H, Cl, H, Bn, CF ₂ HCF ₂ ], [RC7825; F, H, Cl, Cl, Bn, Me], [RC7826; F, H, Cl, Cl, Bn , Et], [RC7827; F, H, Cl, Cl, Bn, Pr], [RC7828; F, H, Cl, Cl, Bn, i-Pr], [RC7829; F, H, Cl, Cl, Bn , c-Pr], [RC7830; F, H, Cl, Cl, Bn, Bu], [RC7831; F, H, Cl, Cl, Bn, i-Bu], [RC7832; F, H, Cl, Cl , Bn, t-Bu], [RC7833; F, H, Cl, Cl, Bn, c-PrCH ₂ ], [RC7834; F, H, Cl, Cl, Bn, Ph], [RC7835; F, H, Cl, Cl, Bn, Bn], [RC7836; F, H, Cl, Cl, Bn, CF ₃ ], [RC7837; F, H, Cl, Cl, Bn , CF ₃ CH ₂ ], [RC7838; F, H, Cl, Cl, Bn, CF ₃ CF ₂ ], [RC7839; F, H, Cl, Cl, Bn, CF ₂ H], [RC7840; F, H , Cl, Cl, Bn, CF ₂ HCF ₂ ], [RC7841; F, H, H, H, Ph, Me], [RC7842; F, H, H, H, Ph, Et], [RC7843; F, H, H, H, Ph, Pr], [RC7844; F, H, H, H, Ph, i-Pr], [RC7845; F, H, H, H, Ph, c-Pr], [RC7846; F, H, H, H, Ph, Bu], [RC7847; F, H, H, H, Ph, i-Bu], [RC7848; F, H, H, H, Ph, t-Bu], [ RC7849; F, H, H, H, Ph, c-PrCH ₂ ], [RC7850; F, H, H, H, Ph, Ph], [RC7851; F, H, H, H, Ph, Bn], [RC7852; F, H, H, H, Ph, CF ₃ ], [RC7853; F, H, H, H, Ph, CF ₃ CH ₂ ], [RC7854; F, H, H, H, Ph, CF ₃ CF ₂ ], [RC7855; F, H, H, H, Ph, CF ₂ H], [RC7856; F, H, H, H, Ph, CF ₂ HCF ₂ ], [RC7857; F, H, H , Me, Ph, Me], [RC7858; F, H, H, Me, Ph, Et], [RC7859; F, H, H, Me, Ph, Pr], [RC7860; F, H, H, Me , Ph, i-Pr], [RC7861; F, H, H, Me, Ph, c-Pr], [RC7862; F, H, H, Me, Ph, Bu], [RC7863; F, H, H , Me, Ph, i-Bu], [RC7864; F, H, H, Me, Ph, t-Bu], [RC7865; F, H, H, Me, Ph, c-PrCH ₂ ], [RC7866; F, H, H, Me, Ph, Ph], [RC7867; F, H, H, Me, Ph, Bn], [RC7868; F, H, H, Me, Ph, CF ₃ ], [RC7869; F , H, H, Me, Ph, CF ₃ CH ₂ ], [RC7870; F, H, H, Me, Ph, CF ₃ CF ₂ ], [RC7871; F, H, H, Me, Ph, CF ₂ H ], [RC7872; F, H, H, Me, Ph, CF ₂ HCF ₂ ], [RC7873; F, H, Me, Me, Ph, Me], [RC7874; F, H, Me, Me, Ph , Et], [RC7875; F, H, Me, Me, Ph, Pr], [RC7876; F, H, Me, Me, Ph, i-Pr], [RC7877; F, H, Me, Me, Ph , c-Pr], [RC7878; F, H, Me, Me, Ph, Bu], [RC7879; F, H, Me, Me, Ph, i-Bu], [RC7880; F, H, Me, Me , Ph, t-Bu], [RC7881; F, H, Me, Me, Ph, c-PrCH ₂ ], [RC7882; F, H, Me, Me, Ph, Ph], [RC7883; F, H, Me, Me, Ph, Bn], [RC7884; F, H, Me, Me, Ph, CF ₃ ], [RC7885; F, H, Me, Me, Ph, CF ₃ CH ₂ ], [RC7886; F, H, Me, Me, Ph, CF ₃ CF ₂ ], [RC7887; F, H, Me, Me, Ph, CF ₂ H], [RC7888; F, H, Me, Me, Ph, CF ₂ HCF ₂ ] , [RC7889; F, H, Me, Et, Ph, Me], [RC7890; F, H, Me, Et, Ph, Et], [RC7891; F, H, Me, Et, Ph, Pr], [ RC7892; F, H, Me, Et, Ph, i-Pr], [RC7893; F, H, Me, Et, Ph, c-Pr], [RC7894; F, H, Me, Et, Ph, Bu] , [RC7895; F, H, Me, Et, Ph, i-Bu], [RC7896; F, H, Me, Et, Ph, t-Bu], [RC7897; F, H, Me, Et, Ph, c-PrCH ₂ ], [RC7898; F, H, Me, Et, Ph, Ph], [RC7899; F, H, Me, Et, Ph, Bn], [RC7900; F, H, Me, Et, Ph , CF ₃ ], [RC7901; F, H, Me, Et, Ph, CF ₃ CH ₂ ], [RC7902; F, H, Me, Et, Ph, CF ₃ CF ₂ ], [RC7903; F, H, Me, Et, Ph, CF ₂ H], [RC7904; F, H, Me, Et, Ph, CF ₂ HCF ₂ ], [RC7905; F, H, Me, F, Ph, Me], [RC7906; F , H, Me, F, Ph, Et], [RC7907; F, H, Me, F, Ph, Pr], [RC7908; F, H, Me, F, Ph, i-Pr], [RC7909; F , H, Me, F, Ph, c-Pr], [RC7910; F, H, Me, F, Ph, Bu], [RC 7911; F, H, Me, F, Ph, i-Bu], [RC7912; F, H, Me, F, Ph, t-Bu], [RC7913; F, H, Me, F, Ph, c- PrCH ₂ ], [RC7914; F, H, Me, F, Ph, Ph], [RC7915; F, H, Me, F, Ph, Bn], [RC7916; F, H, Me, F, Ph, CF ₃ ], [RC7917; F, H, Me, F, Ph, CF ₃ CH ₂ ], [RC7918; F, H, Me, F, Ph, CF ₃ CF ₂ ], [RC7919; F, H, Me, F, Ph, CF ₂ H], [RC7920; F, H, Me, F, Ph, CF ₂ HCF ₂ ], [RC7921; F, H, Me, Cl, Ph, Me], [RC7922; F, H , Me, Cl, Ph, Et], [RC7923; F, H, Me, Cl, Ph, Pr], [RC7924; F, H, Me, Cl, Ph, i-Pr], [RC7925; F, H , Me, Cl, Ph, c-Pr], [RC7926; F, H, Me, Cl, Ph, Bu], [RC7927; F, H, Me, Cl, Ph, i-Bu], [RC7928; F , H, Me, Cl, Ph, t-Bu], [RC7929; F, H, Me, Cl, Ph, c-PrCH ₂ ], [RC7930; F, H, Me, Cl, Ph, Ph], [ RC7931; F, H, Me, Cl, Ph, Bn], [RC7932; F, H, Me, Cl, Ph, CF ₃ ], [RC7933; F, H, Me, Cl, Ph, CF ₃ CH ₂ ] , [RC7934; F, H, Me, Cl, Ph, CF ₃ CF ₂ ], [RC7935; F, H, Me, Cl, Ph, CF ₂ H], [RC7936; F, H, Me, Cl, Ph , CF ₂ HCF ₂ ], [RC7937; F, H, Et, H, Ph, Me], [RC7938; F, H, Et, H, Ph, Et], [RC7939; F, H, Et, H, Ph, Pr], [RC7940; F, H, Et, H, Ph, i-Pr], [RC7941; F, H, Et, H, Ph, c-Pr], [RC7942; F, H, Et, H, Ph, Bu], [RC7943; F, H, Et, H, Ph, i-Bu], [RC7944; F, H, Et, H, Ph, t-Bu], [RC7945; F, H, Et, H, Ph, c-PrCH ₂ ], [RC7946; F, H, Et, H, Ph, Ph], [RC7947; F, H, Et, H, P h, Bn], [RC7948; F, H, Et, H, Ph, CF ₃ ], [RC7949; F, H, Et, H, Ph, CF ₃ CH ₂ ], [RC7950; F, H, Et, H, Ph, CF ₃ CF ₂ ], [RC7951; F, H, Et, H, Ph, CF ₂ H], [RC7952; F, H, Et, H, Ph, CF ₂ HCF ₂ ], [RC7953; F, H, Et, F, Ph, Me], [RC7954; F, H, Et, F, Ph, Et], [RC7955; F, H, Et, F, Ph, Pr], [RC7956; F, H, Et, F, Ph, i-Pr], [RC7957; F, H, Et, F, Ph, c-Pr], [RC7958; F, H, Et, F, Ph, Bu], [RC7959; F, H, Et, F, Ph, i-Bu], [RC7960; F, H, Et, F, Ph, t-Bu], [RC7961; F, H, Et, F, Ph, c-PrCH ₂ ], [RC7962; F, H, Et, F, Ph, Ph], [RC7963; F, H, Et, F, Ph, Bn], [RC7964; F, H, Et, F, Ph, CF ₃ ] , [RC7965; F, H, Et, F, Ph, CF ₃ CH ₂ ], [RC7966; F, H, Et, F, Ph, CF ₃ CF ₂ ], [RC7967; F, H, Et, F, Ph, CF ₂ H], [RC7968; F, H, Et, F, Ph, CF ₂ HCF ₂ ], [RC7969; F, H, Et, Cl, Ph, Me], [RC7970; F, H, Et , Cl, Ph, Et], [RC7971; F, H, Et, Cl, Ph, Pr], [RC7972; F, H, Et, Cl, Ph, i-Pr], [RC7973; F, H, Et , Cl, Ph, c-Pr], [RC7974; F, H, Et, Cl, Ph, Bu], [RC7975; F, H, Et, Cl, Ph, i-Bu], [RC7976; F, H , Et, Cl, Ph, t-Bu], [RC7977; F, H, Et, Cl, Ph, c-PrCH ₂ ], [RC7978; F, H, Et, Cl, Ph, Ph], [RC7979; F, H, Et, Cl, Ph, Bn], [RC7980; F, H, Et, Cl, Ph, CF ₃ ], [RC7981; F, H, Et, Cl, Ph, CF ₃ CH ₂ ], [ RC7982; F, H, Et, Cl, Ph, CF ₃ CF ₂ ], [RC7983; F, H, Et, Cl, Ph, CF ₂ H ], [RC7984; F, H, Et, Cl, Ph, CF ₂ HCF ₂ ], [RC7985; F, H, F, H, Ph, Me], [RC7986; F, H, F, H, Ph, Et], [RC7987; F, H, F, H, Ph, Pr], [RC7988; F, H, F, H, Ph, i-Pr], [RC7989; F, H, F, H, Ph, c-Pr], [RC7990; F, H, F, H, Ph, Bu], [RC7991; F, H, F, H, Ph, i-Bu], [RC7992; F, H, F, H, Ph, t-Bu], [RC7993; F, H, F, H, Ph, c-PrCH ₂ ], [RC7994; F, H, F, H, Ph, Ph], [RC7995; F, H, F , H, Ph, Bn], [RC7996; F, H, F, H, Ph, CF ₃ ], [RC7997; F, H, F, H, Ph, CF ₃ CH ₂ ], [RC7998; F, H , F, H, Ph, CF ₃ CF ₂ ], [RC7999; F, H, F, H, Ph, CF ₂ H], [RC8000; F, H, F, H, Ph, CF ₂ HCF ₂ ],

[RC8001; F, H, F, F, Ph, Me], [RC8002; F, H, F, F, Ph, Et], [RC8003; F, H, F, F, Ph, Pr], [RC8004 ; F, H, F, F, Ph, i-Pr], [RC8005; F, H, F, F, Ph, c-Pr], [RC8006; F, H, F, F, Ph, Bu], [RC8007; F, H, F, F, Ph, i-Bu], [RC8008; F, H, F, F, Ph, t-Bu], [RC8009; F, H, F, F, Ph, c -PrCH ₂ ], [RC8010; F, H, F, F, Ph, Ph], [RC8011; F, H, F, F, Ph, Bn], [RC8012; F, H, F, F, Ph, CF ₃ ], [RC8013; F, H, F, F, Ph, CF ₃ CH ₂ ], [RC8014; F, H, F, F, Ph, CF ₃ CF ₂ ], [RC8015; F, H, F , F, Ph, CF ₂ H], [RC8016; F, H, F, F, Ph, CF ₂ HCF ₂ ], [RC8017; F, H, F, Cl, Ph, Me], [RC8018; F, H, F, Cl, Ph, Et], [RC8019; F, H, F, Cl, Ph, Pr], [RC8020; F, H, F, Cl, Ph, i-Pr], [RC8021; F, H, F, Cl, Ph, c-Pr], [RC8022; F, H, F, Cl, Ph, Bu], [RC8023; F, H, F, Cl, Ph, i-Bu], [RC8024; F, H, F, Cl, Ph, t-Bu], [RC8025; F, H, F, Cl, Ph, c-PrCH ₂ ], [RC8026; F, H, F, Cl, Ph, Ph], [RC8027; F, H, F, Cl, Ph, Bn], [RC8028; F, H, F, Cl, Ph, CF ₃ ], [RC8029; F, H, F, Cl, Ph, CF ₃ CH ₂ ], [RC8030; F, H, F, Cl, Ph, CF ₃ CF ₂ ], [RC8031; F, H, F, Cl, Ph, CF ₂ H], [RC8032; F, H, F, Cl, Ph, CF ₂ HCF ₂ ], [RC8033; F, H, Cl, H, Ph, Me], [RC8034; F, H, Cl, H, Ph, Et], [RC8035; F, H, Cl, H , Ph, Pr], [RC8036; F, H, Cl, H, Ph, i-Pr], [RC8037; F, H, Cl, H, Ph, c-Pr], [RC8038; F, H, Cl , H, Ph, Bu], [RC803 9; F, H, Cl, H, Ph, i-Bu], [RC8040; F, H, Cl, H, Ph, t-Bu], [RC8041; F, H, Cl, H, Ph, c- PrCH ₂ ], [RC8042; F, H, Cl, H, Ph, Ph], [RC8043; F, H, Cl, H, Ph, Bn], [RC8044; F, H, Cl, H, Ph, CF ₃ ], [RC8045; F, H, Cl, H, Ph, CF ₃ CH ₂ ], [RC8046; F, H, Cl, H, Ph, CF ₃ CF ₂ ], [RC8047; F, H, Cl, H, Ph, CF ₂ H], [RC8048; F, H, Cl, H, Ph, CF ₂ HCF ₂ ], [RC8049; F, H, Cl, Cl, Ph, Me], [RC8050; F, H , Cl, Cl, Ph, Et], [RC8051; F, H, Cl, Cl, Ph, Pr], [RC8052; F, H, Cl, Cl, Ph, i-Pr], [RC8053; F, H , Cl, Cl, Ph, c-Pr], [RC8054; F, H, Cl, Cl, Ph, Bu], [RC8055; F, H, Cl, Cl, Ph, i-Bu], [RC8056; F , H, Cl, Cl, Ph, t-Bu], [RC8057; F, H, Cl, Cl, Ph, c-PrCH ₂ ], [RC8058; F, H, Cl, Cl, Ph, Ph], [ RC8059; F, H, Cl, Cl, Ph, Bn], [RC8060; F, H, Cl, Cl, Ph, CF ₃ ], [RC8061; F, H, Cl, Cl, Ph, CF ₃ CH ₂ ] , [RC8062; F, H, Cl, Cl, Ph, CF ₃ CF ₂ ], [RC8063; F, H, Cl, Cl, Ph, CF ₂ H], [RC8064; F, H, Cl, Cl, Ph , CF ₂ HCF ₂ ], [RC8065; H, F, H, H, H, Me], [RC8066; H, F, H, H, H, Et], [RC8067; H, F, H, H, H, Pr], [RC8068; H, F, H, H, H, i-Pr], [RC8069; H, F, H, H, H, c-Pr], [RC8070; H, F, H, H, H, Bu], [RC8071; H, F, H, H, H, i-Bu], [RC8072; H, F, H, H, H, t-Bu], [RC8073; H, F, H, H, H, c-PrCH ₂ ], [RC8074; H, F, H, H, H, Ph], [RC8075; H, F, H, H, H, Bn], [RC8076; H, F , H, H, H, C F ₃ ], [RC8077; H, F, H, H, H, CF ₃ CH ₂ ], [RC8078; H, F, H, H, H, CF ₃ CF ₂ ], [RC8079; H, F, H , H, H, CF ₂ H], [RC8080; H, F, H, H, H, CF ₂ HCF ₂ ], [RC8081; H, F, H, Me, H, Me], [RC8082; H, F, H, Me, H, Et], [RC8083; H, F, H, Me, H, Pr], [RC8084; H, F, H, Me, H, i-Pr], [RC8085; H, F, H, Me, H, c-Pr], [RC8086; H, F, H, Me, H, Bu], [RC8087; H, F, H, Me, H, i-Bu], [RC8088; H, F, H, Me, H, t-Bu], [RC8089; H, F, H, Me, H, c-PrCH ₂ ], [RC8090; H, F, H, Me, H, Ph], [RC8091; H, F, H, Me, H, Bn], [RC8092; H, F, H, Me, H, CF ₃ ], [RC8093; H, F, H, Me, H, CF ₃ CH ₂ ], [RC8094; H, F, H, Me, H, CF ₃ CF ₂ ], [RC8095; H, F, H, Me, H, CF ₂ H], [RC8096; H, F, H, Me, H, CF ₂ HCF ₂ ], [RC8097; H, F, Me, Me, H, Me], [RC8098; H, F, Me, Me, H, Et], [RC8099; H, F, Me, Me , H, Pr], [RC8100; H, F, Me, Me, H, i-Pr], [RC8101; H, F, Me, Me, H, c-Pr], [RC8102; H, F, Me , Me, H, Bu], [RC8103; H, F, Me, Me, H, i-Bu], [RC8104; H, F, Me, Me, H, t-Bu], [RC8105; H, F , Me, Me, H, c-PrCH ₂ ], [RC8106; H, F, Me, Me, H, Ph], [RC8107; H, F, Me, Me, H, Bn], [RC8108; H, F, Me, Me, H, CF ₃ ], [RC8109; H, F, Me, Me, H, CF ₃ CH ₂ ], [RC8110; H, F, Me, Me, H, CF ₃ CF ₂ ], [RC8111; H, F, Me, Me, H, CF ₂ H], [RC8112; H, F, Me, Me, H, CF ₂ HCF ₂ ], [RC8113; H, F, Me, Et, H, Me], [RC8114 ; H, F, Me, Et, H, Et], [RC8115; H, F, Me, Et, H, Pr], [RC8116; H, F, Me, Et, H, i-Pr], [RC8117 ; H, F, Me, Et, H, c-Pr], [RC8118; H, F, Me, Et, H, Bu], [RC8119; H, F, Me, Et, H, i-Bu], [RC8120; H, F, Me, Et, H, t-Bu], [RC8121; H, F, Me, Et, H, c-PrCH ₂ ], [RC8122; H, F, Me, Et, H, Ph], [RC8123; H, F, Me, Et, H, Bn], [RC8124; H, F, Me, Et, H, CF ₃ ], [RC8125; H, F, Me, Et, H, CF ₃ CH ₂ ], [RC8126; H, F, Me, Et, H, CF ₃ CF ₂ ], [RC8127; H, F, Me, Et, H, CF ₂ H], [RC8128; H, F, Me , Et, H, CF ₂ HCF ₂ ], [RC8129; H, F, Me, F, H, Me], [RC8130; H, F, Me, F, H, Et], [RC8131; H, F, Me, F, H, Pr], [RC8132; H, F, Me, F, H, i-Pr], [RC8133; H, F, Me, F, H, c-Pr], [RC8134; H, F, Me, F, H, Bu], [RC8135; H, F, Me, F, H, i-Bu], [RC8136; H, F, Me, F, H, t-Bu], [RC8137; H, F, Me, F, H, c-PrCH ₂ ], [RC8138; H, F, Me, F, H, Ph], [RC8139; H, F, Me, F, H, Bn], [RC8140 ; H, F, Me, F, H, CF ₃ ], [RC8141; H, F, Me, F, H, CF ₃ CH ₂ ], [RC8142; H, F, Me, F, H, CF ₃ CF ₂ ], [RC8143; H, F, Me, F, H, CF ₂ H], [RC8144; H, F, Me, F, H, CF ₂ HCF ₂ ], [RC8145; H, F, Me, Cl , H, Me], [RC8146; H, F, Me, Cl, H, Et], [RC8147; H, F, Me, Cl, H, Pr], [RC8148; H, F, Me, Cl, H , i-Pr], [RC8149; H, F, Me, Cl, H, c-Pr], [RC8150; H, F, Me, Cl, H, Bu], [RC8151; H, F, Me, Cl , H, i-Bu], [RC8152; H, F , Me, Cl, H, t-Bu], [RC8153; H, F, Me, Cl, H, c-PrCH ₂ ], [RC8154; H, F, Me, Cl, H, Ph], [RC8155; H, F, Me, Cl, H, Bn], [RC8156; H, F, Me, Cl, H, CF ₃ ], [RC8157; H, F, Me, Cl, H, CF ₃ CH ₂ ], [ RC8158; H, F, Me, Cl, H, CF ₃ CF ₂ ], [RC8159; H, F, Me, Cl, H, CF ₂ H], [RC8160; H, F, Me, Cl, H, CF ₂ HCF ₂ ], [RC8161; H, F, Et, H, H, Me], [RC8162; H, F, Et, H, H, Et], [RC8163; H, F, Et, H, H, Pr], [RC8164; H, F, Et, H, H, i-Pr], [RC8165; H, F, Et, H, H, c-Pr], [RC8166; H, F, Et, H, H, Bu], [RC8167; H, F, Et, H, H, i-Bu], [RC8168; H, F, Et, H, H, t-Bu], [RC8169; H, F, Et, H, H, c-PrCH ₂ ], [RC8170; H, F, Et, H, H, Ph], [RC8171; H, F, Et, H, H, Bn], [RC8172; H, F, Et , H, H, CF ₃ ], [RC8173; H, F, Et, H, H, CF ₃ CH ₂ ], [RC8174; H, F, Et, H, H, CF ₃ CF ₂ ], [RC8175; H, F, Et, H, H, CF ₂ H], [RC8176; H, F, Et, H, H, CF ₂ HCF ₂ ], [RC8177; H, F, Et, F, H, Me], [RC8178; H, F, Et, F, H, Et], [RC8179; H, F, Et, F, H, Pr], [RC8180; H, F, Et, F, H, i-Pr], [RC8181; H, F, Et, F, H, c-Pr], [RC8182; H, F, Et, F, H, Bu], [RC8183; H, F, Et, F, H, i-Bu ], [RC8184; H, F, Et, F, H, t-Bu], [RC8185; H, F, Et, F, H, c-PrCH ₂ ], [RC8186; H, F, Et, F, H, Ph], [RC8187; H, F, Et, F, H, Bn], [RC8188; H, F, Et, F, H, CF ₃ ], [RC8189; H, F, Et, F, H , CF ₃ CH ₂ ], [RC8190; H, F, Et , F, H, CF ₃ CF ₂ ], [RC8191; H, F, Et, F, H, CF ₂ H], [RC8192; H, F, Et, F, H, CF ₂ HCF ₂ ], [RC8193 ; H, F, Et, Cl, H, Me], [RC8194; H, F, Et, Cl, H, Et], [RC8195; H, F, Et, Cl, H, Pr], [RC8196; H , F, Et, Cl, H, i-Pr], [RC8197; H, F, Et, Cl, H, c-Pr], [RC8198; H, F, Et, Cl, H, Bu], [RC8199 ; H, F, Et, Cl, H, i-Bu], [RC8200; H, F, Et, Cl, H, t-Bu],

[RC8201; H, F, Et, Cl, H, c-PrCH ₂ ], [RC8202; H, F, Et, Cl, H, Ph], [RC8203; H, F, Et, Cl, H, Bn] , [RC8204; H, F, Et, Cl, H, CF ₃ ], [RC8205; H, F, Et, Cl, H, CF ₃ CH ₂ ], [RC8206; H, F, Et, Cl, H, CF ₃ CF ₂ ], [RC8207; H, F, Et, Cl, H, CF ₂ H], [RC8208; H, F, Et, Cl, H, CF ₂ HCF ₂ ], [RC8209; H, F, F, H, H, Me], [RC8210; H, F, F, H, H, Et], [RC8211; H, F, F, H, H, Pr], [RC8212; H, F, F, H, H, i-Pr], [RC8213; H, F, F, H, H, c-Pr], [RC8214; H, F, F, H, H, Bu], [RC8215; H, F, F, H, H, i-Bu], [RC8216; H, F, F, H, H, t-Bu], [RC8217; H, F, F, H, H, c-PrCH ₂ ], [RC8218 ; H, F, F, H, H, Ph], [RC8219; H, F, F, H, H, Bn], [RC8220; H, F, F, H, H, CF ₃ ], [RC8221; H, F, F, H, H, CF ₃ CH ₂ ], [RC8222; H, F, F, H, H, CF ₃ CF ₂ ], [RC8223; H, F, F, H, H, CF ₂ H], [RC8224; H, F, F, H, H, CF ₂ HCF ₂ ], [RC8225; H, F, F, F, H, Me], [RC8226; H, F, F, F, H , Et], [RC8227; H, F, F, F, H, Pr], [RC8228; H, F, F, F, H, i-Pr], [RC8229; H, F, F, F, H , c-Pr], [RC8230; H, F, F, F, H, Bu], [RC8231; H, F, F, F, H, i-Bu], [RC8232; H, F, F, F , H, t-Bu], [RC8233; H, F, F, F, H, c-PrCH ₂ ], [RC8234; H, F, F, F, H, Ph], [RC8235; H, F, F, F, H, Bn], [RC8236; H, F, F, F, H, CF ₃ ], [RC8237; H, F, F, F, H, CF ₃ CH ₂ ], [RC8238; H, F, F, F, H, CF ₃ CF ₂ ], [RC8239; H, F, F, F, H, CF ₂ H], [R C8240; H, F, F, F, H, CF ₂ HCF ₂ ], [RC8241; H, F, F, Cl, H, Me], [RC8242; H, F, F, Cl, H, Et], [RC8243; H, F, F, Cl, H, Pr], [RC8244; H, F, F, Cl, H, i-Pr], [RC8245; H, F, F, Cl, H, c-Pr ], [RC8246; H, F, F, Cl, H, Bu], [RC8247; H, F, F, Cl, H, i-Bu], [RC8248; H, F, F, Cl, H, t -Bu], [RC8249; H, F, F, Cl, H, c-PrCH ₂ ], [RC8250; H, F, F, Cl, H, Ph], [RC8251; H, F, F, Cl, H, Bn], [RC8252; H, F, F, Cl, H, CF ₃ ], [RC8253; H, F, F, Cl, H, CF ₃ CH ₂ ], [RC8254; H, F, F, Cl, H, CF ₃ CF ₂ ], [RC8255; H, F, F, Cl, H, CF ₂ H], [RC8256; H, F, F, Cl, H, CF ₂ HCF ₂ ], [RC8257; H, F, Cl, H, H, Me], [RC8258; H, F, Cl, H, H, Et], [RC8259; H, F, Cl, H, H, Pr], [RC8260; H, F, Cl, H, H, i-Pr], [RC8261; H, F, Cl, H, H, c-Pr], [RC8262; H, F, Cl, H, H, Bu], [RC8263; H, F, Cl, H, H, i-Bu], [RC8264; H, F, Cl, H, H, t-Bu], [RC8265; H, F, Cl, H, H, c-PrCH ₂ ], [RC8266; H, F, Cl, H, H, Ph], [RC8267; H, F, Cl, H, H, Bn], [RC8268; H, F, Cl, H, H, CF ₃ ] , [RC8269; H, F, Cl, H, H, CF ₃ CH ₂ ], [RC8270; H, F, Cl, H, H, CF ₃ CF ₂ ], [RC8271; H, F, Cl, H, H, CF ₂ H], [RC8272; H, F, Cl, H, H, CF ₂ HCF ₂ ], [RC8273; H, F, Cl, Cl, H, Me], [RC8274; H, F, Cl , Cl, H, Et], [RC8275; H, F, Cl, Cl, H, Pr], [RC8276; H, F, Cl, Cl, H, i-Pr], [RC8277; H, F, Cl , Cl, H, c-Pr], [RC8278; H, F, Cl, Cl , H, Bu], [RC8279; H, F, Cl, Cl, H, i-Bu], [RC8280; H, F, Cl, Cl, H, t-Bu], [RC8281; H, F, Cl , Cl, H, c-PrCH ₂ ], [RC8282; H, F, Cl, Cl, H, Ph], [RC8283; H, F, Cl, Cl, H, Bn], [RC8284; H, F, Cl, Cl, H, CF ₃ ], [RC8285; H, F, Cl, Cl, H, CF ₃ CH ₂ ], [RC8286; H, F, Cl, Cl, H, CF ₃ CF ₂ ], [RC8287 ; H, F, Cl, Cl, H, CF ₂ H], [RC8288; H, F, Cl, Cl, H, CF ₂ HCF ₂ ], [RC8289; H, F, H, H, Me, Me] , [RC8290; H, F, H, H, Me, Et], [RC8291; H, F, H, H, Me, Pr], [RC8292; H, F, H, H, Me, i-Pr] , [RC8293; H, F, H, H, Me, c-Pr], [RC8294; H, F, H, H, Me, Bu], [RC8295; H, F, H, H, Me, i- Bu], [RC8296; H, F, H, H, Me, t-Bu], [RC8297; H, F, H, H, Me, c-PrCH ₂ ], [RC8298; H, F, H, H , Me, Ph], [RC8299; H, F, H, H, Me, Bn], [RC8300; H, F, H, H, Me, CF ₃ ], [RC8301; H, F, H, H, Me, CF ₃ CH ₂ ], [RC8302; H, F, H, H, Me, CF ₃ CF ₂ ], [RC8303; H, F, H, H, Me, CF ₂ H], [RC8304; H, F, H, H, Me, CF ₂ HCF ₂ ], [RC8305; H, F, H, Me, Me, Me], [RC8306; H, F, H, Me, Me, Et], [RC8307; H , F, H, Me, Me, Pr], [RC8308; H, F, H, Me, Me, i-Pr], [RC8309; H, F, H, Me, Me, c-Pr], [RC8310 ; H, F, H, Me, Me, Bu], [RC8311; H, F, H, Me, Me, i-Bu], [RC8312; H, F, H, Me, Me, t-Bu], [RC8313; H, F, H, Me, Me, c-PrCH ₂ ], [RC8314; H, F, H, Me, Me, Ph], [RC8315; H, F, H, Me, Me, Bn] , [RC8316; H, F, H, Me , Me, CF ₃ ], [RC8317; H, F, H, Me, Me, CF ₃ CH ₂ ], [RC8318; H, F, H, Me, Me, CF ₃ CF ₂ ], [RC8319; H, F, H, Me, Me, CF ₂ H], [RC8320; H, F, H, Me, Me, CF ₂ HCF ₂ ], [RC8321; H, F, Me, Me, Me, Me], [RC8322 ; H, F, Me, Me, Me, Et], [RC8323; H, F, Me, Me, Me, Pr], [RC8324; H, F, Me, Me, Me, i-Pr], [RC8325 ; H, F, Me, Me, Me, c-Pr], [RC8326; H, F, Me, Me, Me, Bu], [RC8327; H, F, Me, Me, Me, i-Bu], [RC8328; H, F, Me, Me, Me, t-Bu], [RC8329; H, F, Me, Me, Me, c-PrCH ₂ ], [RC8330; H, F, Me, Me, Me, Ph], [RC8331; H, F, Me, Me, Me, Bn], [RC8332; H, F, Me, Me, Me, CF ₃ ], [RC8333; H, F, Me, Me, Me, CF ₃ CH ₂ ], [RC8334; H, F, Me, Me, Me, CF ₃ CF ₂ ], [RC8335; H, F, Me, Me, Me, CF ₂ H], [RC8336; H, F, Me , Me, Me, CF ₂ HCF ₂ ], [RC8337; H, F, Me, Et, Me, Me], [RC8338; H, F, Me, Et, Me, Et], [RC8339; H, F, Me, Et, Me, Pr], [RC8340; H, F, Me, Et, Me, i-Pr], [RC8341; H, F, Me, Et, Me, c-Pr], [RC8342; H, F, Me, Et, Me, Bu], [RC8343; H, F, Me, Et, Me, i-Bu], [RC8344; H, F, Me, Et, Me, t-Bu], [RC8345; H, F, Me, Et, Me, c-PrCH ₂ ], [RC8346; H, F, Me, Et, Me, Ph], [RC8347; H, F, Me, Et, Me, Bn], [RC8348 ; H, F, Me, Et, Me, CF ₃ ], [RC8349; H, F, Me, Et, Me, CF ₃ CH ₂ ], [RC8350; H, F, Me, Et, Me, CF ₃ CF ₂ ], [RC8351; H, F, Me, Et, Me, CF ₂ H], [RC8 352; H, F, Me, Et, Me, CF ₂ HCF ₂ ], [RC8353; H, F, Me, F, Me, Me], [RC8354; H, F, Me, F, Me, Et], [RC8355; H, F, Me, F, Me, Pr], [RC8356; H, F, Me, F, Me, i-Pr], [RC8357; H, F, Me, F, Me, c-Pr ], [RC8358; H, F, Me, F, Me, Bu], [RC8359; H, F, Me, F, Me, i-Bu], [RC8360; H, F, Me, F, Me, t -Bu], [RC8361; H, F, Me, F, Me, c-PrCH ₂ ], [RC8362; H, F, Me, F, Me, Ph], [RC8363; H, F, Me, F, Me, Bn], [RC8364; H, F, Me, F, Me, CF ₃ ], [RC8365; H, F, Me, F, Me, CF ₃ CH ₂ ], [RC8366; H, F, Me, F, Me, CF ₃ CF ₂ ], [RC8367; H, F, Me, F, Me, CF ₂ H], [RC8368; H, F, Me, F, Me, CF ₂ HCF ₂ ], [RC8369; H, F, Me, Cl, Me, Me], [RC8370; H, F, Me, Cl, Me, Et], [RC8371; H, F, Me, Cl, Me, Pr], [RC8372; H, F, Me, Cl, Me, i-Pr], [RC8373; H, F, Me, Cl, Me, c-Pr], [RC8374; H, F, Me, Cl, Me, Bu], [RC8375; H, F, Me, Cl, Me, i-Bu], [RC8376; H, F, Me, Cl, Me, t-Bu], [RC8377; H, F, Me, Cl, Me, c-PrCH ₂ ], [RC8378; H, F, Me, Cl, Me, Ph], [RC8379; H, F, Me, Cl, Me, Bn], [RC8380; H, F, Me, Cl, Me, CF ₃ ] , [RC8381; H, F, Me, Cl, Me, CF ₃ CH ₂ ], [RC8382; H, F, Me, Cl, Me, CF ₃ CF ₂ ], [RC8383; H, F, Me, Cl, Me, CF ₂ H], [RC8384; H, F, Me, Cl, Me, CF ₂ HCF ₂ ], [RC8385; H, F, Et, H, Me, Me], [RC8386; H, F, Et , H, Me, Et], [RC8387; H, F, Et, H, Me, Pr], [RC8388; H, F, Et, H, Me, i-Pr], [RC8389; H, F, Et, H, Me, c-Pr], [RC8390; H, F, Et, H, Me, Bu], [RC8391; H, F, Et, H, Me, i-Bu], [RC8392; H, F, Et, H, Me, t-Bu], [RC8393; H, F, Et, H, Me, c-PrCH ₂ ], [RC8394; H, F , Et, H, Me, Ph], [RC8395; H, F, Et, H, Me, Bn], [RC8396; H, F, Et, H, Me, CF ₃ ], [RC8397; H, F, Et, H, Me, CF ₃ CH ₂ ], [RC8398; H, F, Et, H, Me, CF ₃ CF ₂ ], [RC8399; H, F, Et, H, Me, CF ₂ H], [ RC8400; H, F, Et, H, Me, CF ₂ HCF ₂ ],

[RC8401; H, F, Et, F, Me, Me], [RC8402; H, F, Et, F, Me, Et], [RC8403; H, F, Et, F, Me, Pr], [RC8404 ; H, F, Et, F, Me, i-Pr], [RC8405; H, F, Et, F, Me, c-Pr], [RC8406; H, F, Et, F, Me, Bu], [RC8407; H, F, Et, F, Me, i-Bu], [RC8408; H, F, Et, F, Me, t-Bu], [RC8409; H, F, Et, F, Me, c -PrCH ₂ ], [RC8410; H, F, Et, F, Me, Ph], [RC8411; H, F, Et, F, Me, Bn], [RC8412; H, F, Et, F, Me, CF ₃ ], [RC8413; H, F, Et, F, Me, CF ₃ CH ₂ ], [RC8414; H, F, Et, F, Me, CF ₃ CF ₂ ], [RC8415; H, F, Et , F, Me, CF ₂ H], [RC8416; H, F, Et, F, Me, CF ₂ HCF ₂ ], [RC8417; H, F, Et, Cl, Me, Me], [RC8418; H, F, Et, Cl, Me, Et], [RC8419; H, F, Et, Cl, Me, Pr], [RC8420; H, F, Et, Cl, Me, i-Pr], [RC8421; H, F, Et, Cl, Me, c-Pr], [RC8422; H, F, Et, Cl, Me, Bu], [RC8423; H, F, Et, Cl, Me, i-Bu], [RC8424; H, F, Et, Cl, Me, t-Bu], [RC8425; H, F, Et, Cl, Me, c-PrCH ₂ ], [RC8426; H, F, Et, Cl, Me, Ph], [RC8427; H, F, Et, Cl, Me, Bn], [RC8428; H, F, Et, Cl, Me, CF ₃ ], [RC8429; H, F, Et, Cl, Me, CF ₃ CH ₂ ], [RC8430; H, F, Et, Cl, Me, CF ₃ CF ₂ ], [RC8431; H, F, Et, Cl, Me, CF ₂ H], [RC8432; H, F, Et, Cl, Me, CF ₂ HCF ₂ ], [RC8433; H, F, F, H, Me, Me], [RC8434; H, F, F, H, Me, Et], [RC8435; H, F, F, H , Me, Pr], [RC8436; H, F, F, H, Me, i-Pr], [RC8437; H, F, F, H, Me, c-Pr], [RC 8438; H, F, F, H, Me, Bu], [RC8439; H, F, F, H, Me, i-Bu], [RC8440; H, F, F, H, Me, t-Bu] , [RC8441; H, F, F, H, Me, c-PrCH ₂ ], [RC8442; H, F, F, H, Me, Ph], [RC8443; H, F, F, H, Me, Bn ], [RC8444; H, F, F, H, Me, CF ₃ ], [RC8445; H, F, F, H, Me, CF ₃ CH ₂ ], [RC8446; H, F, F, H, Me , CF ₃ CF ₂ ], [RC8447; H, F, F, H, Me, CF ₂ H], [RC8448; H, F, F, H, Me, CF ₂ HCF ₂ ], [RC8449; H, F , F, F, Me, Me], [RC8450; H, F, F, F, Me, Et], [RC8451; H, F, F, F, Me, Pr], [RC8452; H, F, F , F, Me, i-Pr], [RC8453; H, F, F, F, Me, c-Pr], [RC8454; H, F, F, F, Me, Bu], [RC8455; H, F , F, F, Me, i-Bu], [RC8456; H, F, F, F, Me, t-Bu], [RC8457; H, F, F, F, Me, c-PrCH ₂ ], [ RC8458; H, F, F, F, Me, Ph], [RC8459; H, F, F, F, Me, Bn], [RC8460; H, F, F, F, Me, CF ₃ ], [RC8461 ; H, F, F, F, Me, CF ₃ CH ₂ ], [RC8462; H, F, F, F, Me, CF ₃ CF ₂ ], [RC8463; H, F, F, F, Me, CF ₂ H], [RC8464; H, F, F, F, Me, CF ₂ HCF ₂ ], [RC8465; H, F, F, Cl, Me, Me], [RC8466; H, F, F, Cl, Me, Et], [RC8467; H, F, F, Cl, Me, Pr], [RC8468; H, F, F, Cl, Me, i-Pr], [RC8469; H, F, F, Cl, Me, c-Pr], [RC8470; H, F, F, Cl, Me, Bu], [RC8471; H, F, F, Cl, Me, i-Bu], [RC8472; H, F, F, Cl, Me, t-Bu], [RC8473; H, F, F, Cl, Me, c-PrCH ₂ ], [RC8474; H, F, F, Cl, Me, Ph], [RC8475; H, F , F, Cl, Me, Bn], [RC8476; H, F, F , Cl, Me, CF ₃ ], [RC8477; H, F, F, Cl, Me, CF ₃ CH ₂ ], [RC8478; H, F, F, Cl, Me, CF ₃ CF ₂ ], [RC8479; H, F, F, Cl, Me, CF ₂ H], [RC8480; H, F, F, Cl, Me, CF ₂ HCF ₂ ], [RC8481; H, F, Cl, H, Me, Me], [RC8482; H, F, Cl, H, Me, Et], [RC8483; H, F, Cl, H, Me, Pr], [RC8484; H, F, Cl, H, Me, i-Pr], [RC8485; H, F, Cl, H, Me, c-Pr], [RC8486; H, F, Cl, H, Me, Bu], [RC8487; H, F, Cl, H, Me, i-Bu ], [RC8488; H, F, Cl, H, Me, t-Bu], [RC8489; H, F, Cl, H, Me, c-PrCH ₂ ], [RC8490; H, F, Cl, H, Me, Ph], [RC8491; H, F, Cl, H, Me, Bn], [RC8492; H, F, Cl, H, Me, CF ₃ ], [RC8493; H, F, Cl, H, Me , CF ₃ CH ₂ ], [RC8494; H, F, Cl, H, Me, CF ₃ CF ₂ ], [RC8495; H, F, Cl, H, Me, CF ₂ H], [RC8496; H, F , Cl, H, Me, CF ₂ HCF ₂ ], [RC8497; H, F, Cl, Cl, Me, Me], [RC8498; H, F, Cl, Cl, Me, Et], [RC8499; H, F, Cl, Cl, Me, Pr], [RC8500; H, F, Cl, Cl, Me, i-Pr], [RC8501; H, F, Cl, Cl, Me, c-Pr], [RC8502; H, F, Cl, Cl, Me, Bu], [RC8503; H, F, Cl, Cl, Me, i-Bu], [RC8504; H, F, Cl, Cl, Me, t-Bu], [ RC8505; H, F, Cl, Cl, Me, c-PrCH ₂ ], [RC8506; H, F, Cl, Cl, Me, Ph], [RC8507; H, F, Cl, Cl, Me, Bn], [RC8508; H, F, Cl, Cl, Me, CF ₃ ], [RC8509; H, F, Cl, Cl, Me, CF ₃ CH ₂ ], [RC8510; H, F, Cl, Cl, Me, CF ₃ CF ₂ ], [RC8511; H, F, Cl, Cl, Me, CF ₂ H], [RC8512; H, F, Cl, Cl , Me, CF ₂ HCF ₂ ], [RC8513; H, F, H, H, Et, Me], [RC8514; H, F, H, H, Et, Et], [RC8515; H, F, H, H, Et, Pr], [RC8516; H, F, H, H, Et, i-Pr], [RC8517; H, F, H, H, Et, c-Pr], [RC8518; H, F, H, H, Et, Bu], [RC8519; H, F, H, H, Et, i-Bu], [RC8520; H, F, H, H, Et, t-Bu], [RC8521; H, F, H, H, Et, c-PrCH ₂ ], [RC8522; H, F, H, H, Et, Ph], [RC8523; H, F, H, H, Et, Bn], [RC8524; H , F, H, H, Et, CF ₃ ], [RC8525; H, F, H, H, Et, CF ₃ CH ₂ ], [RC8526; H, F, H, H, Et, CF ₃ CF ₂ ] , [RC8527; H, F, H, H, Et, CF ₂ H], [RC8528; H, F, H, H, Et, CF ₂ HCF ₂ ], [RC8529; H, F, H, Me, Et , Me], [RC8530; H, F, H, Me, Et, Et], [RC8531; H, F, H, Me, Et, Pr], [RC8532; H, F, H, Me, Et, i -Pr], [RC8533; H, F, H, Me, Et, c-Pr], [RC8534; H, F, H, Me, Et, Bu], [RC8535; H, F, H, Me, Et , i-Bu], [RC8536; H, F, H, Me, Et, t-Bu], [RC8537; H, F, H, Me, Et, c-PrCH ₂ ], [RC8538; H, F, H, Me, Et, Ph], [RC8539; H, F, H, Me, Et, Bn], [RC8540; H, F, H, Me, Et, CF ₃ ], [RC8541; H, F, H , Me, Et, CF ₃ CH ₂ ], [RC8542; H, F, H, Me, Et, CF ₃ CF ₂ ], [RC8543; H, F, H, Me, Et, CF ₂ H], [RC8544 ; H, F, H, Me, Et, CF ₂ HCF ₂ ], [RC8545; H, F, Me, Me, Et, Me], [RC8546; H, F, Me, Me, Et, Et], [ RC8547; H, F, Me, Me, Et, Pr], [RC8548; H, F, Me, Me, Et, i-Pr], [RC8549; H, F, Me, Me, Et, c-Pr] , [RC8550; H, F, Me, Me, Et, Bu], [RC8551; H, F, Me, Me, Et, i-Bu], [RC8552; H, F, Me, Me, Et, t-Bu], [ RC8553; H, F, Me, Me, Et, c-PrCH ₂ ], [RC8554; H, F, Me, Me, Et, Ph], [RC8555; H, F, Me, Me, Et, Bn], [RC8556; H, F, Me, Me, Et, CF ₃ ], [RC8557; H, F, Me, Me, Et, CF ₃ CH ₂ ], [RC8558; H, F, Me, Me, Et, CF ₃ CF ₂ ], [RC8559; H, F, Me, Me, Et, CF ₂ H], [RC8560; H, F, Me, Me, Et, CF ₂ HCF ₂ ], [RC8561; H, F, Me , Et, Et, Me], [RC8562; H, F, Me, Et, Et, Et], [RC8563; H, F, Me, Et, Et, Pr], [RC8564; H, F, Me, Et , Et, i-Pr], [RC8565; H, F, Me, Et, Et, c-Pr], [RC8566; H, F, Me, Et, Et, Bu], [RC8567; H, F, Me , Et, Et, i-Bu], [RC8568; H, F, Me, Et, Et, t-Bu], [RC8569; H, F, Me, Et, Et, c-PrCH ₂ ], [RC8570; H, F, Me, Et, Et, Ph], [RC8571; H, F, Me, Et, Et, Bn], [RC8572; H, F, Me, Et, Et, CF ₃ ], [RC8573; H , F, Me, Et, Et, CF ₃ CH ₂ ], [RC8574; H, F, Me, Et, Et, CF ₃ CF ₂ ], [RC8575; H, F, Me, Et, Et, CF ₂ H ], [RC8576; H, F, Me, Et, Et, CF ₂ HCF ₂ ], [RC8577; H, F, Me, F, Et, Me], [RC8578; H, F, Me, F, Et, Et], [RC8579; H, F, Me, F, Et, Pr], [RC8580; H, F, Me, F, Et, i-Pr], [RC8581; H, F, Me, F, Et, c-Pr], [RC8582; H, F, Me, F, Et, Bu], [RC8583; H, F, Me, F, Et, i-Bu], [RC8584; H, F, Me, F, Et, t-Bu], [RC8585; H, F, Me, F, Et, c-PrCH ₂ ], [RC8586; H, F, Me, F, Et, Ph], [RC8587; H, F, Me, F, Et, Bn], [RC8588; H, F, Me, F, Et, CF ₃ ], [RC8589; H, F, Me , F, Et, CF ₃ CH ₂ ], [RC8590; H, F, Me, F, Et, CF ₃ CF ₂ ], [RC8591; H, F, Me, F, Et, CF ₂ H], [RC8592 ; H, F, Me, F, Et, CF ₂ HCF ₂ ], [RC8593; H, F, Me, Cl, Et, Me], [RC8594; H, F, Me, Cl, Et, Et], [ RC8595; H, F, Me, Cl, Et, Pr], [RC8596; H, F, Me, Cl, Et, i-Pr], [RC8597; H, F, Me, Cl, Et, c-Pr] , [RC8598; H, F, Me, Cl, Et, Bu], [RC8599; H, F, Me, Cl, Et, i-Bu], [RC8600; H, F, Me, Cl, Et, t- Bu],

[RC8601; H, F, Me, Cl, Et, c-PrCH ₂ ], [RC8602; H, F, Me, Cl, Et, Ph], [RC8603; H, F, Me, Cl, Et, Bn] , [RC8604; H, F, Me, Cl, Et, CF ₃ ], [RC8605; H, F, Me, Cl, Et, CF ₃ CH ₂ ], [RC8606; H, F, Me, Cl, Et, CF ₃ CF ₂ ], [RC8607; H, F, Me, Cl, Et, CF ₂ H], [RC8608; H, F, Me, Cl, Et, CF ₂ HCF ₂ ], [RC8609; H, F, Et, H, Et, Me], [RC8610; H, F, Et, H, Et, Et], [RC8611; H, F, Et, H, Et, Pr], [RC8612; H, F, Et, H, Et, i-Pr], [RC8613; H, F, Et, H, Et, c-Pr], [RC8614; H, F, Et, H, Et, Bu], [RC8615; H, F, Et, H, Et, i-Bu], [RC8616; H, F, Et, H, Et, t-Bu], [RC8617; H, F, Et, H, Et, c-PrCH ₂ ], [RC8618 ; H, F, Et, H, Et, Ph], [RC8619; H, F, Et, H, Et, Bn], [RC8620; H, F, Et, H, Et, CF ₃ ], [RC8621; H, F, Et, H, Et, CF ₃ CH ₂ ], [RC8622; H, F, Et, H, Et, CF ₃ CF ₂ ], [RC8623; H, F, Et, H, Et, CF ₂ H], [RC8624; H, F, Et, H, Et, CF ₂ HCF ₂ ], [RC8625; H, F, Et, F, Et, Me], [RC8626; H, F, Et, F, Et , Et], [RC8627; H, F, Et, F, Et, Pr], [RC8628; H, F, Et, F, Et, i-Pr], [RC8629; H, F, Et, F, Et , c-Pr], [RC8630; H, F, Et, F, Et, Bu], [RC8631; H, F, Et, F, Et, i-Bu], [RC8632; H, F, Et, F , Et, t-Bu], [RC8633; H, F, Et, F, Et, c-PrCH ₂ ], [RC8634; H, F, Et, F, Et, Ph], [RC8635; H, F, Et, F, Et, Bn], [RC8636; H, F, Et, F, Et, CF ₃ ], [RC8637; H, F, Et, F, Et, CF ₃ CH ₂ ], [RC8638; H, F, Et, F, Et, CF ₃ CF ₂ ], [RC8639; H, F, Et, F, Et, CF ₂ H], [RC8640; H, F, Et, F, Et, CF ₂ HCF ₂ ], [RC8641; H, F, Et, Cl, Et, Me], [RC8642; H, F, Et, Cl, Et, Et], [RC8643; H, F, Et , Cl, Et, Pr], [RC8644; H, F, Et, Cl, Et, i-Pr], [RC8645; H, F, Et, Cl, Et, c-Pr], [RC8646; H, F , Et, Cl, Et, Bu], [RC8647; H, F, Et, Cl, Et, i-Bu], [RC8648; H, F, Et, Cl, Et, t-Bu], [RC8649; H , F, Et, Cl, Et, c-PrCH ₂ ], [RC8650; H, F, Et, Cl, Et, Ph], [RC8651; H, F, Et, Cl, Et, Bn], [RC8652; H, F, Et, Cl, Et, CF ₃ ], [RC8653; H, F, Et, Cl, Et, CF ₃ CH ₂ ], [RC8654; H, F, Et, Cl, Et, CF ₃ CF ₂ ], [RC8655; H, F, Et, Cl, Et, CF ₂ H], [RC8656; H, F, Et, Cl, Et, CF ₂ HCF ₂ ], [RC8657; H, F, F, H, Et, Me], [RC8658; H, F, F, H, Et, Et], [RC8659; H, F, F, H, Et, Pr], [RC8660; H, F, F, H, Et, i-Pr], [RC8661; H, F, F, H, Et, c-Pr], [RC8662; H, F, F, H, Et, Bu], [RC8663; H, F, F, H, Et, i-Bu], [RC8664; H, F, F, H, Et, t-Bu], [RC8665; H, F, F, H, Et, c-PrCH ₂ ], [RC8666; H, F , F, H, Et, Ph], [RC8667; H, F, F, H, Et, Bn], [RC8668; H, F, F, H, Et, CF ₃ ], [RC8669; H, F, F, H, Et, CF ₃ CH ₂ ], [RC8670; H, F, F, H, Et, CF ₃ CF ₂ ], [RC8671; H, F, F, H, Et, CF ₂ H], [ RC8672; H, F, F, H, Et, CF ₂ HCF ₂ ], [RC8673; H, F, F, F, Et, Me], [RC8674; H, F, F, F, Et, Et], [RC8675; H, F, F, F, Et, Pr], [RC8676; H, F, F, F, Et, i-Pr], [RC8677; H, F, F, F, Et, c-Pr], [RC8678; H, F, F, F, Et, Bu], [RC8679; H, F, F, F, Et, i-Bu], [RC8680; H, F, F, F, Et, t-Bu], [RC8681; H, F, F, F, Et, c-PrCH ₂ ], [RC8682; H, F, F, F, Et, Ph], [RC8683; H , F, F, F, Et, Bn], [RC8684; H, F, F, F, Et, CF ₃ ], [RC8685; H, F, F, F, Et, CF ₃ CH ₂ ], [RC8686 ; H, F, F, F, Et, CF ₃ CF ₂ ], [RC8687; H, F, F, F, Et, CF ₂ H], [RC8688; H, F, F, F, Et, CF ₂ HCF ₂ ], [RC8689; H, F, F, Cl, Et, Me], [RC8690; H, F, F, Cl, Et, Et], [RC8691; H, F, F, Cl, Et, Pr ], [RC8692; H, F, F, Cl, Et, i-Pr], [RC8693; H, F, F, Cl, Et, c-Pr], [RC8694; H, F, F, Cl, Et , Bu], [RC8695; H, F, F, Cl, Et, i-Bu], [RC8696; H, F, F, Cl, Et, t-Bu], [RC8697; H, F, F, Cl , Et, c-PrCH ₂ ], [RC8698; H, F, F, Cl, Et, Ph], [RC8699; H, F, F, Cl, Et, Bn], [RC8700; H, F, F, Cl, Et, CF ₃ ], [RC8701; H, F, F, Cl, Et, CF ₃ CH ₂ ], [RC8702; H, F, F, Cl, Et, CF ₃ CF ₂ ], [RC8703; H , F, F, Cl, Et, CF ₂ H], [RC8704; H, F, F, Cl, Et, CF ₂ HCF ₂ ], [RC8705; H, F, Cl, H, Et, Me], [ RC8706; H, F, Cl, H, Et, Et], [RC8707; H, F, Cl, H, Et, Pr], [RC8708; H, F, Cl, H, Et, i-Pr], [ RC8709; H, F, Cl, H, Et, c-Pr], [RC8710; H, F, Cl, H, Et, Bu], [RC8711; H, F, Cl, H, Et, i-Bu] , [RC8712; H, F, Cl, H, Et, t-Bu], [RC8713; H, F, Cl, H, Et, c-PrCH ₂ ], [RC8714; H, F, Cl, H, Et, Ph], [RC8715; H, F, Cl , H, Et, Bn], [RC8716; H, F, Cl, H, Et, CF ₃ ], [RC8717; H, F, Cl, H, Et, CF ₃ CH ₂ ], [RC8718; H, F , Cl, H, Et, CF ₃ CF ₂ ], [RC8719; H, F, Cl, H, Et, CF ₂ H], [RC8720; H, F, Cl, H, Et, CF ₂ HCF ₂ ], [RC8721; H, F, Cl, Cl, Et, Me], [RC8722; H, F, Cl, Cl, Et, Et], [RC8723; H, F, Cl, Cl, Et, Pr], [RC8724 ; H, F, Cl, Cl, Et, i-Pr], [RC8725; H, F, Cl, Cl, Et, c-Pr], [RC8726; H, F, Cl, Cl, Et, Bu], [RC8727; H, F, Cl, Cl, Et, i-Bu], [RC8728; H, F, Cl, Cl, Et, t-Bu], [RC8729; H, F, Cl, Cl, Et, c -PrCH ₂ ], [RC8730; H, F, Cl, Cl, Et, Ph], [RC8731; H, F, Cl, Cl, Et, Bn], [RC8732; H, F, Cl, Cl, Et, CF ₃ ], [RC8733; H, F, Cl, Cl, Et, CF ₃ CH ₂ ], [RC8734; H, F, Cl, Cl, Et, CF ₃ CF ₂ ], [RC8735; H, F, Cl , Cl, Et, CF ₂ H], [RC8736; H, F, Cl, Cl, Et, CF ₂ HCF ₂ ], [RC8737; H, F, H, H, Pr, Me], [RC8738; H, F, H, H, Pr, Et], [RC8739; H, F, H, H, Pr, Pr], [RC8740; H, F, H, H, Pr, i-Pr], [RC8741; H, F, H, H, Pr, c-Pr], [RC8742; H, F, H, H, Pr, Bu], [RC8743; H, F, H, H, Pr, i-Bu], [RC8744; H, F, H, H, Pr, t-Bu], [RC8745; H, F, H, H, Pr, c-PrCH ₂ ], [RC8746; H, F, H, H, Pr, Ph], [RC8747; H, F, H, H, Pr, Bn], [RC8748; H, F, H, H, Pr, CF ₃ ], [RC8749; H, F, H, H, Pr, CF ₃ CH ₂ ], [RC8750; H, F, H, H, Pr, CF ₃ CF ₂ ], [RC8751; H, F, H, H, Pr, CF ₂ H], [RC8752; H, F, H, H, Pr, CF ₂ HCF ₂ ], [RC8753; H, F, H, Me, Pr, Me], [RC8754; H, F, H, Me, Pr, Et], [RC8755; H, F , H, Me, Pr, Pr], [RC8756; H, F, H, Me, Pr, i-Pr], [RC8757; H, F, H, Me, Pr, c-Pr], [RC8758; H , F, H, Me, Pr, Bu], [RC8759; H, F, H, Me, Pr, i-Bu], [RC8760; H, F, H, Me, Pr, t-Bu], [RC8761 ; H, F, H, Me, Pr, c-PrCH ₂ ], [RC8762; H, F, H, Me, Pr, Ph], [RC8763; H, F, H, Me, Pr, Bn], [ RC8764; H, F, H, Me, Pr, CF ₃ ], [RC8765; H, F, H, Me, Pr, CF ₃ CH ₂ ], [RC8766; H, F, H, Me, Pr, CF ₃ CF ₂ ], [RC8767; H, F, H, Me, Pr, CF ₂ H], [RC8768; H, F, H, Me, Pr, CF ₂ HCF ₂ ], [RC8769; H, F, Me, Me, Pr, Me], [RC8770; H, F, Me, Me, Pr, Et], [RC8771; H, F, Me, Me, Pr, Pr], [RC8772; H, F, Me, Me, Pr, i-Pr], [RC8773; H, F, Me, Me, Pr, c-Pr], [RC8774; H, F, Me, Me, Pr, Bu], [RC8775; H, F, Me, Me, Pr, i-Bu], [RC8776; H, F, Me, Me, Pr, t-Bu], [RC8777; H, F, Me, Me, Pr, c-PrCH ₂ ], [RC8778; H , F, Me, Me, Pr, Ph], [RC8779; H, F, Me, Me, Pr, Bn], [RC8780; H, F, Me, Me, Pr, CF ₃ ], [RC8781; H, F, Me, Me, Pr, CF ₃ CH ₂ ], [RC8782; H, F, Me, Me, Pr, CF ₃ CF ₂ ], [RC8783; H, F, Me, Me, Pr, CF ₂ H] , [RC8784; H, F, Me, Me, Pr, CF ₂ HCF ₂ ], [RC8785; H, F, Me, Et, Pr , Me], [RC8786; H, F, Me, Et, Pr, Et], [RC8787; H, F, Me, Et, Pr, Pr], [RC8788; H, F, Me, Et, Pr, i -Pr], [RC8789; H, F, Me, Et, Pr, c-Pr], [RC8790; H, F, Me, Et, Pr, Bu], [RC8791; H, F, Me, Et, Pr , i-Bu], [RC8792; H, F, Me, Et, Pr, t-Bu], [RC8793; H, F, Me, Et, Pr, c-PrCH ₂ ], [RC8794; H, F, Me, Et, Pr, Ph], [RC8795; H, F, Me, Et, Pr, Bn], [RC8796; H, F, Me, Et, Pr, CF ₃ ], [RC8797; H, F, Me , Et, Pr, CF ₃ CH ₂ ], [RC8798; H, F, Me, Et, Pr, CF ₃ CF ₂ ], [RC8799; H, F, Me, Et, Pr, CF ₂ H], [RC8800 ; H, F, Me, Et, Pr, CF ₂ HCF ₂ ],

[RC8801; H, F, Me, F, Pr, Me], [RC8802; H, F, Me, F, Pr, Et], [RC8803; H, F, Me, F, Pr, Pr], [RC8804 ; H, F, Me, F, Pr, i-Pr], [RC8805; H, F, Me, F, Pr, c-Pr], [RC8806; H, F, Me, F, Pr, Bu], [RC8807; H, F, Me, F, Pr, i-Bu], [RC8808; H, F, Me, F, Pr, t-Bu], [RC8809; H, F, Me, F, Pr, c -PrCH ₂ ], [RC8810; H, F, Me, F, Pr, Ph], [RC8811; H, F, Me, F, Pr, Bn], [RC8812; H, F, Me, F, Pr, CF ₃ ], [RC8813; H, F, Me, F, Pr, CF ₃ CH ₂ ], [RC8814; H, F, Me, F, Pr, CF ₃ CF ₂ ], [RC8815; H, F, Me , F, Pr, CF ₂ H], [RC8816; H, F, Me, F, Pr, CF ₂ HCF ₂ ], [RC8817; H, F, Me, Cl, Pr, Me], [RC8818; H, F, Me, Cl, Pr, Et], [RC8819; H, F, Me, Cl, Pr, Pr], [RC8820; H, F, Me, Cl, Pr, i-Pr], [RC8821; H, F, Me, Cl, Pr, c-Pr], [RC8822; H, F, Me, Cl, Pr, Bu], [RC8823; H, F, Me, Cl, Pr, i-Bu], [RC8824; H, F, Me, Cl, Pr, t-Bu], [RC8825; H, F, Me, Cl, Pr, c-PrCH ₂ ], [RC8826; H, F, Me, Cl, Pr, Ph], [RC8827; H, F, Me, Cl, Pr, Bn], [RC8828; H, F, Me, Cl, Pr, CF ₃ ], [RC8829; H, F, Me, Cl, Pr, CF ₃ CH ₂ ], [RC8830; H, F, Me, Cl, Pr, CF ₃ CF ₂ ], [RC8831; H, F, Me, Cl, Pr, CF ₂ H], [RC8832; H, F, Me, Cl, Pr, CF ₂ HCF ₂ ], [RC8833; H, F, Et, H, Pr, Me], [RC8834; H, F, Et, H, Pr, Et], [RC8835; H, F, Et, H , Pr, Pr], [RC8836; H, F, Et, H, Pr, i-Pr], [RC8837; H, F, Et, H, Pr, c-Pr ], [RC8838; H, F, Et, H, Pr, Bu], [RC8839; H, F, Et, H, Pr, i-Bu], [RC8840; H, F, Et, H, Pr, t -Bu], [RC8841; H, F, Et, H, Pr, c-PrCH ₂ ], [RC8842; H, F, Et, H, Pr, Ph], [RC8843; H, F, Et, H, Pr, Bn], [RC8844; H, F, Et, H, Pr, CF ₃ ], [RC8845; H, F, Et, H, Pr, CF ₃ CH ₂ ], [RC8846; H, F, Et, H, Pr, CF ₃ CF ₂ ], [RC8847; H, F, Et, H, Pr, CF ₂ H], [RC8848; H, F, Et, H, Pr, CF ₂ HCF ₂ ], [RC8849; H, F, Et, F, Pr, Me], [RC8850; H, F, Et, F, Pr, Et], [RC8851; H, F, Et, F, Pr, Pr], [RC8852; H, F, Et, F, Pr, i-Pr], [RC8853; H, F, Et, F, Pr, c-Pr], [RC8854; H, F, Et, F, Pr, Bu], [RC8855; H, F, Et, F, Pr, i-Bu], [RC8856; H, F, Et, F, Pr, t-Bu], [RC8857; H, F, Et, F, Pr, c-PrCH ₂ ], [RC8858; H, F, Et, F, Pr, Ph], [RC8859; H, F, Et, F, Pr, Bn], [RC8860; H, F, Et, F, Pr, CF ₃ ] , [RC8861; H, F, Et, F, Pr, CF ₃ CH ₂ ], [RC8862; H, F, Et, F, Pr, CF ₃ CF ₂ ], [RC8863; H, F, Et, F, Pr, CF ₂ H], [RC8864; H, F, Et, F, Pr, CF ₂ HCF ₂ ], [RC8865; H, F, Et, Cl, Pr, Me], [RC8866; H, F, Et , Cl, Pr, Et], [RC8867; H, F, Et, Cl, Pr, Pr], [RC8868; H, F, Et, Cl, Pr, i-Pr], [RC8869; H, F, Et , Cl, Pr, c-Pr], [RC8870; H, F, Et, Cl, Pr, Bu], [RC8871; H, F, Et, Cl, Pr, i-Bu], [RC8872; H, F , Et, Cl, Pr, t-Bu], [RC8873; H, F, Et, Cl, Pr, c-PrCH ₂ ], [RC8874; H, F, Et, Cl, Pr , Ph], [RC8875; H, F, Et, Cl, Pr, Bn], [RC8876; H, F, Et, Cl, Pr, CF ₃ ], [RC8877; H, F, Et, Cl, Pr, CF ₃ CH ₂ ], [RC8878; H, F, Et, Cl, Pr, CF ₃ CF ₂ ], [RC8879; H, F, Et, Cl, Pr, CF ₂ H], [RC8880; H, F, Et, Cl, Pr, CF ₂ HCF ₂ ], [RC8881; H, F, F, H, Pr, Me], [RC8882; H, F, F, H, Pr, Et], [RC8883; H, F , F, H, Pr, Pr], [RC8884; H, F, F, H, Pr, i-Pr], [RC8885; H, F, F, H, Pr, c-Pr], [RC8886; H , F, F, H, Pr, Bu], [RC8887; H, F, F, H, Pr, i-Bu], [RC8888; H, F, F, H, Pr, t-Bu], [RC8889 ; H, F, F, H, Pr, c-PrCH ₂ ], [RC8890; H, F, F, H, Pr, Ph], [RC8891; H, F, F, H, Pr, Bn], [ RC8892; H, F, F, H, Pr, CF ₃ ], [RC8893; H, F, F, H, Pr, CF ₃ CH ₂ ], [RC8894; H, F, F, H, Pr, CF ₃ CF ₂ ], [RC8895; H, F, F, H, Pr, CF ₂ H], [RC8896; H, F, F, H, Pr, CF ₂ HCF ₂ ], [RC8897; H, F, F, F, Pr, Me], [RC8898; H, F, F, F, Pr, Et], [RC8899; H, F, F, F, Pr, Pr], [RC8900; H, F, F, F, Pr, i-Pr], [RC8901; H, F, F, F, Pr, c-Pr], [RC8902; H, F, F, F, Pr, Bu], [RC8903; H, F, F, F, Pr, i-Bu], [RC8904; H, F, F, F, Pr, t-Bu], [RC8905; H, F, F, F, Pr, c-PrCH ₂ ], [RC8906; H , F, F, F, Pr, Ph], [RC8907; H, F, F, F, Pr, Bn], [RC8908; H, F, F, F, Pr, CF ₃ ], [RC8909; H, F, F, F, Pr, CF ₃ CH ₂ ], [RC8910; H, F, F, F, Pr, CF ₃ CF ₂ ], [RC8911; H, F, F, F, Pr, CF ₂ H] , [RC8912; H, F, F, F , Pr, CF ₂ HCF ₂ ], [RC8913; H, F, F, Cl, Pr, Me], [RC8914; H, F, F, Cl, Pr, Et], [RC8915; H, F, F, Cl, Pr, Pr], [RC8916; H, F, F, Cl, Pr, i-Pr], [RC8917; H, F, F, Cl, Pr, c-Pr], [RC8918; H, F, F, Cl, Pr, Bu], [RC8919; H, F, F, Cl, Pr, i-Bu], [RC8920; H, F, F, Cl, Pr, t-Bu], [RC8921; H, F, F, Cl, Pr, c-PrCH ₂ ], [RC8922; H, F, F, Cl, Pr, Ph], [RC8923; H, F, F, Cl, Pr, Bn], [RC8924; H , F, F, Cl, Pr, CF ₃ ], [RC8925; H, F, F, Cl, Pr, CF ₃ CH ₂ ], [RC8926; H, F, F, Cl, Pr, CF ₃ CF ₂ ] , [RC8927; H, F, F, Cl, Pr, CF ₂ H], [RC8928; H, F, F, Cl, Pr, CF ₂ HCF ₂ ], [RC8929; H, F, Cl, H, Pr , Me], [RC8930; H, F, Cl, H, Pr, Et], [RC8931; H, F, Cl, H, Pr, Pr], [RC8932; H, F, Cl, H, Pr, i -Pr], [RC8933; H, F, Cl, H, Pr, c-Pr], [RC8934; H, F, Cl, H, Pr, Bu], [RC8935; H, F, Cl, H, Pr , i-Bu], [RC8936; H, F, Cl, H, Pr, t-Bu], [RC8937; H, F, Cl, H, Pr, c-PrCH ₂ ], [RC8938; H, F, Cl, H, Pr, Ph], [RC8939; H, F, Cl, H, Pr, Bn], [RC8940; H, F, Cl, H, Pr, CF ₃ ], [RC8941; H, F, Cl , H, Pr, CF ₃ CH ₂ ], [RC8942; H, F, Cl, H, Pr, CF ₃ CF ₂ ], [RC8943; H, F, Cl, H, Pr, CF ₂ H], [RC8944 ; H, F, Cl, H, Pr, CF ₂ HCF ₂ ], [RC8945; H, F, Cl, Cl, Pr, Me], [RC8946; H, F, Cl, Cl, Pr, Et], [ RC8947; H, F, Cl, Cl, Pr, Pr], [RC8948; H, F, Cl, Cl, Pr, i-Pr], [RC8949; H, F, Cl, Cl, P r, c-Pr], [RC8950; H, F, Cl, Cl, Pr, Bu], [RC8951; H, F, Cl, Cl, Pr, i-Bu], [RC8952; H, F, Cl, Cl, Pr, t-Bu], [RC8953; H, F, Cl, Cl, Pr, c-PrCH ₂ ], [RC8954; H, F, Cl, Cl, Pr, Ph], [RC8955; H, F , Cl, Cl, Pr, Bn], [RC8956; H, F, Cl, Cl, Pr, CF ₃ ], [RC8957; H, F, Cl, Cl, Pr, CF ₃ CH ₂ ], [RC8958; H , F, Cl, Cl, Pr, CF ₃ CF ₂ ], [RC8959; H, F, Cl, Cl, Pr, CF ₂ H], [RC8960; H, F, Cl, Cl, Pr, CF ₂ HCF ₂ ], [RC8961; H, F, H, H, Bu, Me], [RC8962; H, F, H, H, Bu, Et], [RC8963; H, F, H, H, Bu, Pr], [RC8964; H, F, H, H, Bu, i-Pr], [RC8965; H, F, H, H, Bu, c-Pr], [RC8966; H, F, H, H, Bu, Bu ], [RC8967; H, F, H, H, Bu, i-Bu], [RC8968; H, F, H, H, Bu, t-Bu], [RC8969; H, F, H, H, Bu , c-PrCH ₂ ], [RC8970; H, F, H, H, Bu, Ph], [RC8971; H, F, H, H, Bu, Bn], [RC8972; H, F, H, H, Bu, CF ₃ ], [RC8973; H, F, H, H, Bu, CF ₃ CH ₂ ], [RC8974; H, F, H, H, Bu, CF ₃ CF ₂ ], [RC8975; H, F , H, H, Bu, CF ₂ H], [RC8976; H, F, H, H, Bu, CF ₂ HCF ₂ ], [RC8977; H, F, H, Me, Bu, Me], [RC8978; H, F, H, Me, Bu, Et], [RC8979; H, F, H, Me, Bu, Pr], [RC8980; H, F, H, Me, Bu, i-Pr], [RC8981; H, F, H, Me, Bu, c-Pr], [RC8982; H, F, H, Me, Bu, Bu], [RC8983; H, F, H, Me, Bu, i-Bu], [ RC8984; H, F, H, Me, Bu, t-Bu], [RC8985; H, F, H, Me, Bu, c-PrCH ₂ ], [RC8986; H, F, H, Me, Bu, Ph ], [RC8 987; H, F, H, Me, Bu, Bn], [RC8988; H, F, H, Me, Bu, CF ₃ ], [RC8989; H, F, H, Me, Bu, CF ₃ CH ₂ ] , [RC8990; H, F, H, Me, Bu, CF ₃ CF ₂ ], [RC8991; H, F, H, Me, Bu, CF ₂ H], [RC8992; H, F, H, Me, Bu , CF ₂ HCF ₂ ], [RC8993; H, F, Me, Me, Bu, Me], [RC8994; H, F, Me, Me, Bu, Et], [RC8995; H, F, Me, Me, Bu, Pr], [RC8996; H, F, Me, Me, Bu, i-Pr], [RC8997; H, F, Me, Me, Bu, c-Pr], [RC8998; H, F, Me, Me, Bu, Bu], [RC8999; H, F, Me, Me, Bu, i-Bu], [RC9000; H, F, Me, Me, Bu, t-Bu],

[RC9001; H, F, Me, Me, Bu, c-PrCH ₂ ], [RC9002; H, F, Me, Me, Bu, Ph], [RC9003; H, F, Me, Me, Bu, Bn] , [RC9004; H, F, Me, Me, Bu, CF ₃ ], [RC9005; H, F, Me, Me, Bu, CF ₃ CH ₂ ], [RC9006; H, F, Me, Me, Bu, CF ₃ CF ₂ ], [RC9007; H, F, Me, Me, Bu, CF ₂ H], [RC9008; H, F, Me, Me, Bu, CF ₂ HCF ₂ ], [RC9009; H, F, Me, Et, Bu, Me], [RC9010; H, F, Me, Et, Bu, Et], [RC9011; H, F, Me, Et, Bu, Pr], [RC9012; H, F, Me, Et, Bu, i-Pr], [RC9013; H, F, Me, Et, Bu, c-Pr], [RC9014; H, F, Me, Et, Bu, Bu], [RC9015; H, F, Me, Et, Bu, i-Bu], [RC9016; H, F, Me, Et, Bu, t-Bu], [RC9017; H, F, Me, Et, Bu, c-PrCH ₂ ], [RC9018 ; H, F, Me, Et, Bu, Ph], [RC9019; H, F, Me, Et, Bu, Bn], [RC9020; H, F, Me, Et, Bu, CF ₃ ], [RC9021; H, F, Me, Et, Bu, CF ₃ CH ₂ ], [RC9022; H, F, Me, Et, Bu, CF ₃ CF ₂ ], [RC9023; H, F, Me, Et, Bu, CF ₂ H], [RC9024; H, F, Me, Et, Bu, CF ₂ HCF ₂ ], [RC9025; H, F, Me, F, Bu, Me], [RC9026; H, F, Me, F, Bu , Et], [RC9027; H, F, Me, F, Bu, Pr], [RC9028; H, F, Me, F, Bu, i-Pr], [RC9029; H, F, Me, F, Bu , c-Pr], [RC9030; H, F, Me, F, Bu, Bu], [RC9031; H, F, Me, F, Bu, i-Bu], [RC9032; H, F, Me, F , Bu, t-Bu], [RC9033; H, F, Me, F, Bu, c-PrCH ₂ ], [RC9034; H, F, Me, F, Bu, Ph], [RC9035; H, F, Me, F, Bu, Bn], [RC9036; H, F, Me, F, Bu, CF ₃ ], [RC9037; H, F, Me, F, Bu, CF ₃ CH ₂ ], [RC9038; H, F, Me, F, Bu, CF ₃ CF ₂ ], [RC9039; H, F, Me, F, Bu, CF ₂ H], [RC9040; H, F, Me, F, Bu, CF ₂ HCF ₂ ], [RC9041; H, F, Me, Cl, Bu, Me], [RC9042; H, F, Me, Cl, Bu , Et], [RC9043; H, F, Me, Cl, Bu, Pr], [RC9044; H, F, Me, Cl, Bu, i-Pr], [RC9045; H, F, Me, Cl, Bu , c-Pr], [RC9046; H, F, Me, Cl, Bu, Bu], [RC9047; H, F, Me, Cl, Bu, i-Bu], [RC9048; H, F, Me, Cl , Bu, t-Bu], [RC9049; H, F, Me, Cl, Bu, c-PrCH ₂ ], [RC9050; H, F, Me, Cl, Bu, Ph], [RC9051; H, F, Me, Cl, Bu, Bn], [RC9052; H, F, Me, Cl, Bu, CF ₃ ], [RC9053; H, F, Me, Cl, Bu, CF ₃ CH ₂ ], [RC9054; H, F, Me, Cl, Bu, CF ₃ CF ₂ ], [RC9055; H, F, Me, Cl, Bu, CF ₂ H], [RC9056; H, F, Me, Cl, Bu, CF ₂ HCF ₂ ] , [RC9057; H, F, Et, H, Bu, Me], [RC9058; H, F, Et, H, Bu, Et], [RC9059; H, F, Et, H, Bu, Pr], [ RC9060; H, F, Et, H, Bu, i-Pr], [RC9061; H, F, Et, H, Bu, c-Pr], [RC9062; H, F, Et, H, Bu, Bu] , [RC9063; H, F, Et, H, Bu, i-Bu], [RC9064; H, F, Et, H, Bu, t-Bu], [RC9065; H, F, Et, H, Bu, c-PrCH ₂ ], [RC9066; H, F, Et, H, Bu, Ph], [RC9067; H, F, Et, H, Bu, Bn], [RC9068; H, F, Et, H, Bu , CF ₃ ], [RC9069; H, F, Et, H, Bu, CF ₃ CH ₂ ], [RC9070; H, F, Et, H, Bu, CF ₃ CF ₂ ], [RC9071; H, F, Et, H, Bu, CF ₂ H], [RC9072; H, F, Et, H, Bu, CF ₂ HCF ₂ ], [RC90 73; H, F, Et, F, Bu, Me], [RC9074; H, F, Et, F, Bu, Et], [RC9075; H, F, Et, F, Bu, Pr], [RC9076; H, F, Et, F, Bu, i-Pr], [RC9077; H, F, Et, F, Bu, c-Pr], [RC9078; H, F, Et, F, Bu, Bu], [ RC9079; H, F, Et, F, Bu, i-Bu], [RC9080; H, F, Et, F, Bu, t-Bu], [RC9081; H, F, Et, F, Bu, c- PrCH ₂ ], [RC9082; H, F, Et, F, Bu, Ph], [RC9083; H, F, Et, F, Bu, Bn], [RC9084; H, F, Et, F, Bu, CF ₃ ], [RC9085; H, F, Et, F, Bu, CF ₃ CH ₂ ], [RC9086; H, F, Et, F, Bu, CF ₃ CF ₂ ], [RC9087; H, F, Et, F, Bu, CF ₂ H], [RC9088; H, F, Et, F, Bu, CF ₂ HCF ₂ ], [RC9089; H, F, Et, Cl, Bu, Me], [RC9090; H, F , Et, Cl, Bu, Et], [RC9091; H, F, Et, Cl, Bu, Pr], [RC9092; H, F, Et, Cl, Bu, i-Pr], [RC9093; H, F , Et, Cl, Bu, c-Pr], [RC9094; H, F, Et, Cl, Bu, Bu], [RC9095; H, F, Et, Cl, Bu, i-Bu], [RC9096; H , F, Et, Cl, Bu, t-Bu], [RC9097; H, F, Et, Cl, Bu, c-PrCH ₂ ], [RC9098; H, F, Et, Cl, Bu, Ph], [ RC9099; H, F, Et, Cl, Bu, Bn], [RC9100; H, F, Et, Cl, Bu, CF ₃ ], [RC9101; H, F, Et, Cl, Bu, CF ₃ CH ₂ ] , [RC9102; H, F, Et, Cl, Bu, CF ₃ CF ₂ ], [RC9103; H, F, Et, Cl, Bu, CF ₂ H], [RC9104; H, F, Et, Cl, Bu , CF ₂ HCF ₂ ], [RC9105; H, F, F, H, Bu, Me], [RC9106; H, F, F, H, Bu, Et], [RC9107; H, F, F, H, Bu, Pr], [RC9108; H, F, F, H, Bu, i-Pr], [RC9109; H, F, F, H, Bu, c-Pr], [RC9110; H, F, F, H, Bu, Bu], [RC9111; H, F, F, H, Bu, i-Bu], [RC9112; H, F, F, H, Bu, t-Bu], [ RC9113; H, F, F, H, Bu, c-PrCH ₂ ], [RC9114; H, F, F, H, Bu, Ph], [RC9115; H, F, F, H, Bu, Bn], [RC9116; H, F, F, H, Bu, CF ₃ ], [RC9117; H, F, F, H, Bu, CF ₃ CH ₂ ], [RC9118; H, F, F, H, Bu, CF ₃ CF ₂ ], [RC9119; H, F, F, H, Bu, CF ₂ H], [RC9120; H, F, F, H, Bu, CF ₂ HCF ₂ ], [RC9121; H, F, F , F, Bu, Me], [RC9122; H, F, F, F, Bu, Et], [RC9123; H, F, F, F, Bu, Pr], [RC9124; H, F, F, F , Bu, i-Pr], [RC9125; H, F, F, F, Bu, c-Pr], [RC9126; H, F, F, F, Bu, Bu], [RC9127; H, F, F , F, Bu, i-Bu], [RC9128; H, F, F, F, Bu, t-Bu], [RC9129; H, F, F, F, Bu, c-PrCH ₂ ], [RC9130; H, F, F, F, Bu, Ph], [RC9131; H, F, F, F, Bu, Bn], [RC9132; H, F, F, F, Bu, CF ₃ ], [RC9133; H , F, F, F, Bu, CF ₃ CH ₂ ], [RC9134; H, F, F, F, Bu, CF ₃ CF ₂ ], [RC9135; H, F, F, F, Bu, CF ₂ H ], [RC9136; H, F, F, F, Bu, CF ₂ HCF ₂ ], [RC9137; H, F, F, Cl, Bu, Me], [RC9138; H, F, F, Cl, Bu, Et], [RC9139; H, F, F, Cl, Bu, Pr], [RC9140; H, F, F, Cl, Bu, i-Pr], [RC9141; H, F, F, Cl, Bu, c-Pr], [RC9142; H, F, F, Cl, Bu, Bu], [RC9143; H, F, F, Cl, Bu, i-Bu], [RC9144; H, F, F, Cl, Bu, t-Bu], [RC9145; H, F, F, Cl, Bu, c-PrCH ₂ ], [RC9146; H, F, F, Cl, Bu, Ph], [RC9147; H, F, F , Cl, Bu, Bn], [RC9148; H, F, F, Cl, B u, CF ₃ ], [RC9149; H, F, F, Cl, Bu, CF ₃ CH ₂ ], [RC9150; H, F, F, Cl, Bu, CF ₃ CF ₂ ], [RC9151; H, F , F, Cl, Bu, CF ₂ H], [RC9152; H, F, F, Cl, Bu, CF ₂ HCF ₂ ], [RC9153; H, F, Cl, H, Bu, Me], [RC9154; H, F, Cl, H, Bu, Et], [RC9155; H, F, Cl, H, Bu, Pr], [RC9156; H, F, Cl, H, Bu, i-Pr], [RC9157; H, F, Cl, H, Bu, c-Pr], [RC9158; H, F, Cl, H, Bu, Bu], [RC9159; H, F, Cl, H, Bu, i-Bu], [ RC9160; H, F, Cl, H, Bu, t-Bu], [RC9161; H, F, Cl, H, Bu, c-PrCH ₂ ], [RC9162; H, F, Cl, H, Bu, Ph ], [RC9163; H, F, Cl, H, Bu, Bn], [RC9164; H, F, Cl, H, Bu, CF ₃ ], [RC9165; H, F, Cl, H, Bu, CF ₃ CH ₂ ], [RC9166; H, F, Cl, H, Bu, CF ₃ CF ₂ ], [RC9167; H, F, Cl, H, Bu, CF ₂ H], [RC9168; H, F, Cl, H, Bu, CF ₂ HCF ₂ ], [RC9169; H, F, Cl, Cl, Bu, Me], [RC9170; H, F, Cl, Cl, Bu, Et], [RC9171; H, F, Cl , Cl, Bu, Pr], [RC9172; H, F, Cl, Cl, Bu, i-Pr], [RC9173; H, F, Cl, Cl, Bu, c-Pr], [RC9174; H, F , Cl, Cl, Bu, Bu], [RC9175; H, F, Cl, Cl, Bu, i-Bu], [RC9176; H, F, Cl, Cl, Bu, t-Bu], [RC9177; H , F, Cl, Cl, Bu, c-PrCH ₂ ], [RC9178; H, F, Cl, Cl, Bu, Ph], [RC9179; H, F, Cl, Cl, Bu, Bn], [RC9180; H, F, Cl, Cl, Bu, CF ₃ ], [RC9181; H, F, Cl, Cl, Bu, CF ₃ CH ₂ ], [RC9182; H, F, Cl, Cl, Bu, CF ₃ CF ₂ ], [RC9183; H, F, Cl, Cl, Bu, CF ₂ H], [RC9184; H, F, Cl, Cl, Bu, C F ₂ HCF ₂ ], [RC9185; H, F, H, H, i-Pr, Me], [RC9186; H, F, H, H, i-Pr, Et], [RC9187; H, F, H , H, i-Pr, Pr], [RC9188; H, F, H, H, i-Pr, i-Pr], [RC9189; H, F, H, H, i-Pr, c-Pr], [RC9190; H, F, H, H, i-Pr, Bu], [RC9191; H, F, H, H, i-Pr, i-Bu], [RC9192; H, F, H, H, i -Pr, t-Bu], [RC9193; H, F, H, H, i-Pr, c-PrCH ₂ ], [RC9194; H, F, H, H, i-Pr, Ph], [RC9195; H, F, H, H, i-Pr, Bn], [RC9196; H, F, H, H, i-Pr, CF ₃ ], [RC9197; H, F, H, H, i-Pr, CF ₃ CH ₂ ], [RC9198; H, F, H, H, i-Pr, CF ₃ CF ₂ ], [RC9199; H, F, H, H, i-Pr, CF ₂ H], [RC9200; H , F, H, H, i-Pr, CF ₂ HCF ₂ ],

[RC9201; H, F, H, Me, i-Pr, Me], [RC9202; H, F, H, Me, i-Pr, Et], [RC9203; H, F, H, Me, i-Pr , Pr], [RC9204; H, F, H, Me, i-Pr, i-Pr], [RC9205; H, F, H, Me, i-Pr, c-Pr], [RC9206; H, F , H, Me, i-Pr, Bu], [RC9207; H, F, H, Me, i-Pr, i-Bu], [RC9208; H, F, H, Me, i-Pr, t-Bu ], [RC9209; H, F, H, Me, i-Pr, c-PrCH ₂ ], [RC9210; H, F, H, Me, i-Pr, Ph], [RC9211; H, F, H, Me, i-Pr, Bn], [RC9212; H, F, H, Me, i-Pr, CF ₃ ], [RC9213; H, F, H, Me, i-Pr, CF ₃ CH ₂ ], [ RC9214; H, F, H, Me, i-Pr, CF ₃ CF ₂ ], [RC9215; H, F, H, Me, i-Pr, CF ₂ H], [RC9216; H, F, H, Me , i-Pr, CF ₂ HCF ₂ ], [RC9217; H, F, Me, Me, i-Pr, Me], [RC9218; H, F, Me, Me, i-Pr, Et], [RC9219; H, F, Me, Me, i-Pr, Pr], [RC9220; H, F, Me, Me, i-Pr, i-Pr], [RC9221; H, F, Me, Me, i-Pr, c-Pr], [RC9222; H, F, Me, Me, i-Pr, Bu], [RC9223; H, F, Me, Me, i-Pr, i-Bu], [RC9224; H, F, Me, Me, i-Pr, t-Bu], [RC9225; H, F, Me, Me, i-Pr, c-PrCH ₂ ], [RC9226; H, F, Me, Me, i-Pr, Ph ], [RC9227; H, F, Me, Me, i-Pr, Bn], [RC9228; H, F, Me, Me, i-Pr, CF ₃ ], [RC9229; H, F, Me, Me, i-Pr, CF ₃ CH ₂ ], [RC9230; H, F, Me, Me, i-Pr, CF ₃ CF ₂ ], [RC9231; H, F, Me, Me, i-Pr, CF ₂ H] , [RC9232; H, F, Me, Me, i-Pr, CF ₂ HCF ₂ ], [RC9233; H, F, Me, Et, i-Pr, Me], [RC9234; H, F, Me, Et , i-Pr, Et], [RC9 235; H, F, Me, Et, i-Pr, Pr], [RC9236; H, F, Me, Et, i-Pr, i-Pr], [RC9237; H, F, Me, Et, i- Pr, c-Pr], [RC9238; H, F, Me, Et, i-Pr, Bu], [RC9239; H, F, Me, Et, i-Pr, i-Bu], [RC9240; H, F, Me, Et, i-Pr, t-Bu], [RC9241; H, F, Me, Et, i-Pr, c-PrCH ₂ ], [RC9242; H, F, Me, Et, i-Pr , Ph], [RC9243; H, F, Me, Et, i-Pr, Bn], [RC9244; H, F, Me, Et, i-Pr, CF ₃ ], [RC9245; H, F, Me, Et, i-Pr, CF ₃ CH ₂ ], [RC9246; H, F, Me, Et, i-Pr, CF ₃ CF ₂ ], [RC9247; H, F, Me, Et, i-Pr, CF ₂ H], [RC9248; H, F, Me, Et, i-Pr, CF ₂ HCF ₂ ], [RC9249; H, F, Me, F, i-Pr, Me], [RC9250; H, F, Me , F, i-Pr, Et], [RC9251; H, F, Me, F, i-Pr, Pr], [RC9252; H, F, Me, F, i-Pr, i-Pr], [RC9253 ; H, F, Me, F, i-Pr, c-Pr], [RC9254; H, F, Me, F, i-Pr, Bu], [RC9255; H, F, Me, F, i-Pr , i-Bu], [RC9256; H, F, Me, F, i-Pr, t-Bu], [RC9257; H, F, Me, F, i-Pr, c-PrCH ₂ ], [RC9258; H, F, Me, F, i-Pr, Ph], [RC9259; H, F, Me, F, i-Pr, Bn], [RC9260; H, F, Me, F, i-Pr, CF ₃ ], [RC9261; H, F, Me, F, i-Pr, CF ₃ CH ₂ ], [RC9262; H, F, Me, F, i-Pr, CF ₃ CF ₂ ], [RC9263; H, F , Me, F, i-Pr, CF ₂ H], [RC9264; H, F, Me, F, i-Pr, CF ₂ HCF ₂ ], [RC9265; H, F, Me, Cl, i-Pr, Me], [RC9266; H, F, Me, Cl, i-Pr, Et], [RC9267; H, F, Me, Cl, i-Pr, Pr], [RC9268; H, F, Me, Cl, i-Pr, i-Pr], [RC926 9; H, F, Me, Cl, i-Pr, c-Pr], [RC9270; H, F, Me, Cl, i-Pr, Bu], [RC9271; H, F, Me, Cl, i- Pr, i-Bu], [RC9272; H, F, Me, Cl, i-Pr, t-Bu], [RC9273; H, F, Me, Cl, i-Pr, c-PrCH ₂ ], [RC9274 ; H, F, Me, Cl, i-Pr, Ph], [RC9275; H, F, Me, Cl, i-Pr, Bn], [RC9276; H, F, Me, Cl, i-Pr, CF ₃ ], [RC9277; H, F, Me, Cl, i-Pr, CF ₃ CH ₂ ], [RC9278; H, F, Me, Cl, i-Pr, CF ₃ CF ₂ ], [RC9279; H, F, Me, Cl, i-Pr, CF ₂ H], [RC9280; H, F, Me, Cl, i-Pr, CF ₂ HCF ₂ ], [RC9281; H, F, Et, H, i-Pr , Me], [RC9282; H, F, Et, H, i-Pr, Et], [RC9283; H, F, Et, H, i-Pr, Pr], [RC9284; H, F, Et, H , i-Pr, i-Pr], [RC9285; H, F, Et, H, i-Pr, c-Pr], [RC9286; H, F, Et, H, i-Pr, Bu], [RC9287 ; H, F, Et, H, i-Pr, i-Bu], [RC9288; H, F, Et, H, i-Pr, t-Bu], [RC9289; H, F, Et, H, i -Pr, c-PrCH ₂ ], [RC9290; H, F, Et, H, i-Pr, Ph], [RC9291; H, F, Et, H, i-Pr, Bn], [RC9292; H, F, Et, H, i-Pr, CF ₃ ], [RC9293; H, F, Et, H, i-Pr, CF ₃ CH ₂ ], [RC9294; H, F, Et, H, i-Pr, CF ₃ CF ₂ ], [RC9295; H, F, Et, H, i-Pr, CF ₂ H], [RC9296; H, F, Et, H, i-Pr, CF ₂ HCF ₂ ], [RC9297; H, F, Et, F, i-Pr, Me], [RC9298; H, F, Et, F, i-Pr, Et], [RC9299; H, F, Et, F, i-Pr, Pr] , [RC9300; H, F, Et, F, i-Pr, i-Pr], [RC9301; H, F, Et, F, i-Pr, c-Pr], [RC9302; H, F, Et, F, i-Pr, Bu], [RC9303; H, F, Et , F, i-Pr, i-Bu], [RC9304; H, F, Et, F, i-Pr, t-Bu], [RC9305; H, F, Et, F, i-Pr, c-PrCH ₂ ], [RC9306; H, F, Et, F, i-Pr, Ph], [RC9307; H, F, Et, F, i-Pr, Bn], [RC9308; H, F, Et, F, i-Pr, CF ₃ ], [RC9309; H, F, Et, F, i-Pr, CF ₃ CH ₂ ], [RC9310; H, F, Et, F, i-Pr, CF ₃ CF ₂ ], [RC9311; H, F, Et, F, i-Pr, CF ₂ H], [RC9312; H, F, Et, F, i-Pr, CF ₂ HCF ₂ ], [RC9313; H, F, Et, Cl, i-Pr, Me], [RC9314; H, F, Et, Cl, i-Pr, Et], [RC9315; H, F, Et, Cl, i-Pr, Pr], [RC9316; H, F, Et, Cl, i-Pr, i-Pr], [RC9317; H, F, Et, Cl, i-Pr, c-Pr], [RC9318; H, F, Et, Cl, i-Pr, Bu], [RC9319; H, F, Et, Cl, i-Pr, i-Bu], [RC9320; H, F, Et, Cl, i-Pr, t-Bu], [RC9321; H, F, Et, Cl, i-Pr, c-PrCH ₂ ], [RC9322; H, F, Et, Cl, i-Pr, Ph], [RC9323; H, F, Et, Cl, i-Pr, Bn], [RC9324; H, F, Et, Cl, i-Pr, CF ₃ ], [RC9325; H, F, Et, Cl, i-Pr, CF ₃ CH ₂ ], [RC9326; H, F, Et, Cl , i-Pr, CF ₃ CF ₂ ], [RC9327; H, F, Et, Cl, i-Pr, CF ₂ H], [RC9328; H, F, Et, Cl, i-Pr, CF ₂ HCF ₂ ], [RC9329; H, F, F, H, i-Pr, Me], [RC9330; H, F, F, H, i-Pr, Et], [RC9331; H, F, F, H, i -Pr, Pr], [RC9332; H, F, F, H, i-Pr, i-Pr], [RC9333; H, F, F, H, i-Pr, c-Pr], [RC9334; H , F, F, H, i-Pr, Bu], [RC9335; H, F, F, H, i-Pr, i-Bu], [RC9336; H, F, F, H, i-Pr, t -Bu], [RC9337; H, F, F, H, i-Pr, cP rCH ₂ ], [RC9338; H, F, F, H, i-Pr, Ph], [RC9339; H, F, F, H, i-Pr, Bn], [RC9340; H, F, F, H , i-Pr, CF ₃ ], [RC9341; H, F, F, H, i-Pr, CF ₃ CH ₂ ], [RC9342; H, F, F, H, i-Pr, CF ₃ CF ₂ ] , [RC9343; H, F, F, H, i-Pr, CF ₂ H], [RC9344; H, F, F, H, i-Pr, CF ₂ HCF ₂ ], [RC9345; H, F, F , F, i-Pr, Me], [RC9346; H, F, F, F, i-Pr, Et], [RC9347; H, F, F, F, i-Pr, Pr], [RC9348; H , F, F, F, i-Pr, i-Pr], [RC9349; H, F, F, F, i-Pr, c-Pr], [RC9350; H, F, F, F, i-Pr , Bu], [RC9351; H, F, F, F, i-Pr, i-Bu], [RC9352; H, F, F, F, i-Pr, t-Bu], [RC9353; H, F , F, F, i-Pr, c-PrCH ₂ ], [RC9354; H, F, F, F, i-Pr, Ph], [RC9355; H, F, F, F, i-Pr, Bn] , [RC9356; H, F, F, F, i-Pr, CF ₃ ], [RC9357; H, F, F, F, i-Pr, CF ₃ CH ₂ ], [RC9358; H, F, F, F, i-Pr, CF ₃ CF ₂ ], [RC9359; H, F, F, F, i-Pr, CF ₂ H], [RC9360; H, F, F, F, i-Pr, CF ₂ HCF ₂ ], [RC9361; H, F, F, Cl, i-Pr, Me], [RC9362; H, F, F, Cl, i-Pr, Et], [RC9363; H, F, F, Cl, i-Pr, Pr], [RC9364; H, F, F, Cl, i-Pr, i-Pr], [RC9365; H, F, F, Cl, i-Pr, c-Pr], [RC9366; H, F, F, Cl, i-Pr, Bu], [RC9367; H, F, F, Cl, i-Pr, i-Bu], [RC9368; H, F, F, Cl, i-Pr, t-Bu], [RC9369; H, F, F, Cl, i-Pr, c-PrCH ₂ ], [RC9370; H, F, F, Cl, i-Pr, Ph], [RC9371; H, F , F, Cl, i-Pr, Bn], [RC9372; H, F, F, Cl, i-Pr, CF ₃ ], [RC9373; H, F, F, Cl, i-Pr, CF ₃ CH ₂ ], [RC9374; H, F, F, Cl, i-Pr, CF ₃ CF ₂ ], [RC9375; H, F, F, Cl, i-Pr, CF ₂ H], [RC9376; H, F, F, Cl, i-Pr, CF ₂ HCF ₂ ], [RC9377; H, F, Cl, H, i-Pr, Me], [RC9378 ; H, F, Cl, H, i-Pr, Et], [RC9379; H, F, Cl, H, i-Pr, Pr], [RC9380; H, F, Cl, H, i-Pr, i -Pr], [RC9381; H, F, Cl, H, i-Pr, c-Pr], [RC9382; H, F, Cl, H, i-Pr, Bu], [RC9383; H, F, Cl , H, i-Pr, i-Bu], [RC9384; H, F, Cl, H, i-Pr, t-Bu], [RC9385; H, F, Cl, H, i-Pr, c-PrCH ₂ ], [RC9386; H, F, Cl, H, i-Pr, Ph], [RC9387; H, F, Cl, H, i-Pr, Bn], [RC9388; H, F, Cl, H, i-Pr, CF ₃ ], [RC9389; H, F, Cl, H, i-Pr, CF ₃ CH ₂ ], [RC9390; H, F, Cl, H, i-Pr, CF ₃ CF ₂ ], [RC9391; H, F, Cl, H, i-Pr, CF ₂ H], [RC9392; H, F, Cl, H, i-Pr, CF ₂ HCF ₂ ], [RC9393; H, F, Cl, Cl, i-Pr, Me], [RC9394; H, F, Cl, Cl, i-Pr, Et], [RC9395; H, F, Cl, Cl, i-Pr, Pr], [RC9396; H, F, Cl, Cl, i-Pr, i-Pr], [RC9397; H, F, Cl, Cl, i-Pr, c-Pr], [RC9398; H, F, Cl, Cl, i-Pr, Bu], [RC9399; H, F, Cl, Cl, i-Pr, i-Bu], [RC9400; H, F, Cl, Cl, i-Pr, t-Bu],

[RC9401; H, F, Cl, Cl, i-Pr, c-PrCH ₂ ], [RC9402; H, F, Cl, Cl, i-Pr, Ph], [RC9403; H, F, Cl, Cl, i-Pr, Bn], [RC9404; H, F, Cl, Cl, i-Pr, CF ₃ ], [RC9405; H, F, Cl, Cl, i-Pr, CF ₃ CH ₂ ], [RC9406; H, F, Cl, Cl, i-Pr, CF ₃ CF ₂ ], [RC9407; H, F, Cl, Cl, i-Pr, CF ₂ H], [RC9408; H, F, Cl, Cl, i -Pr, CF ₂ HCF ₂ ], [RC9409; H, F, H, H, c-Pr, Me], [RC9410; H, F, H, H, c-Pr, Et], [RC9411; H, F, H, H, c-Pr, Pr], [RC9412; H, F, H, H, c-Pr, i-Pr], [RC9413; H, F, H, H, c-Pr, c- Pr], [RC9414; H, F, H, H, c-Pr, Bu], [RC9415; H, F, H, H, c-Pr, i-Bu], [RC9416; H, F, H, H, c-Pr, t-Bu], [RC9417; H, F, H, H, c-Pr, c-PrCH ₂ ], [RC9418; H, F, H, H, c-Pr, Ph], [RC9419; H, F, H, H, c-Pr, Bn], [RC9420; H, F, H, H, c-Pr, CF ₃ ], [RC9421; H, F, H, H, c- Pr, CF ₃ CH ₂ ], [RC9422; H, F, H, H, c-Pr, CF ₃ CF ₂ ], [RC9423; H, F, H, H, c-Pr, CF ₂ H], [ RC9424; H, F, H, H, c-Pr, CF ₂ HCF ₂ ], [RC9425; H, F, H, Me, c-Pr, Me], [RC9426; H, F, H, Me, c -Pr, Et], [RC9427; H, F, H, Me, c-Pr, Pr], [RC9428; H, F, H, Me, c-Pr, i-Pr], [RC9429; H, F , H, Me, c-Pr, c-Pr], [RC9430; H, F, H, Me, c-Pr, Bu], [RC9431; H, F, H, Me, c-Pr, i-Bu ], [RC9432; H, F, H, Me, c-Pr, t-Bu], [RC9433; H, F, H, Me, c-Pr, c-PrCH ₂ ], [RC9434; H, F, H, Me, c-Pr, Ph], [RC9435; H, F, H, Me, c-Pr, B n], [RC9436; H, F, H, Me, c-Pr, CF ₃ ], [RC9437; H, F, H, Me, c-Pr, CF ₃ CH ₂ ], [RC9438; H, F, H, Me, c-Pr, CF ₃ CF ₂ ], [RC9439; H, F, H, Me, c-Pr, CF ₂ H], [RC9440; H, F, H, Me, c-Pr, CF ₂ HCF ₂ ], [RC9441; H, F, Me, Me, c-Pr, Me], [RC9442; H, F, Me, Me, c-Pr, Et], [RC9443; H, F, Me, Me, c-Pr, Pr], [RC9444; H, F, Me, Me, c-Pr, i-Pr], [RC9445; H, F, Me, Me, c-Pr, c-Pr], [ RC9446; H, F, Me, Me, c-Pr, Bu], [RC9447; H, F, Me, Me, c-Pr, i-Bu], [RC9448; H, F, Me, Me, c- Pr, t-Bu], [RC9449; H, F, Me, Me, c-Pr, c-PrCH ₂ ], [RC9450; H, F, Me, Me, c-Pr, Ph], [RC9451; H , F, Me, Me, c-Pr, Bn], [RC9452; H, F, Me, Me, c-Pr, CF ₃ ], [RC9453; H, F, Me, Me, c-Pr, CF ₃ CH ₂ ], [RC9454; H, F, Me, Me, c-Pr, CF ₃ CF ₂ ], [RC9455; H, F, Me, Me, c-Pr, CF ₂ H], [RC9456; H, F, Me, Me, c-Pr, CF ₂ HCF ₂ ], [RC9457; H, F, Me, Et, c-Pr, Me], [RC9458; H, F, Me, Et, c-Pr, Et ], [RC9459; H, F, Me, Et, c-Pr, Pr], [RC9460; H, F, Me, Et, c-Pr, i-Pr], [RC9461; H, F, Me, Et , c-Pr, c-Pr], [RC9462; H, F, Me, Et, c-Pr, Bu], [RC9463; H, F, Me, Et, c-Pr, i-Bu], [RC9464 ; H, F, Me, Et, c-Pr, t-Bu], [RC9465; H, F, Me, Et, c-Pr, c-PrCH ₂ ], [RC9466; H, F, Me, Et, c-Pr, Ph], [RC9467; H, F, Me, Et, c-Pr, Bn], [RC9468; H, F, Me, Et, c-Pr, CF ₃ ], [RC9469; H, F , Me , Et, c-Pr, CF ₃ CH ₂ ], [RC9470; H, F, Me, Et, c-Pr, CF ₃ CF ₂ ], [RC9471; H, F, Me, Et, c-Pr, CF ₂ H], [RC9472; H, F, Me, Et, c-Pr, CF ₂ HCF ₂ ], [RC9473; H, F, Me, F, c-Pr, Me], [RC9474; H, F, Me, F, c-Pr, Et], [RC9475; H, F, Me, F, c-Pr, Pr], [RC9476; H, F, Me, F, c-Pr, i-Pr], [ RC9477; H, F, Me, F, c-Pr, c-Pr], [RC9478; H, F, Me, F, c-Pr, Bu], [RC9479; H, F, Me, F, c- Pr, i-Bu], [RC9480; H, F, Me, F, c-Pr, t-Bu], [RC9481; H, F, Me, F, c-Pr, c-PrCH ₂ ], [RC9482 ; H, F, Me, F, c-Pr, Ph], [RC9483; H, F, Me, F, c-Pr, Bn], [RC9484; H, F, Me, F, c-Pr, CF ₃ ], [RC9485; H, F, Me, F, c-Pr, CF ₃ CH ₂ ], [RC9486; H, F, Me, F, c-Pr, CF ₃ CF ₂ ], [RC9487; H, F, Me, F, c-Pr, CF ₂ H], [RC9488; H, F, Me, F, c-Pr, CF ₂ HCF ₂ ], [RC9489; H, F, Me, Cl, c-Pr , Me], [RC9490; H, F, Me, Cl, c-Pr, Et], [RC9491; H, F, Me, Cl, c-Pr, Pr], [RC9492; H, F, Me, Cl , c-Pr, i-Pr], [RC9493; H, F, Me, Cl, c-Pr, c-Pr], [RC9494; H, F, Me, Cl, c-Pr, Bu], [RC9495 ; H, F, Me, Cl, c-Pr, i-Bu], [RC9496; H, F, Me, Cl, c-Pr, t-Bu], [RC9497; H, F, Me, Cl, c -Pr, c-PrCH ₂ ], [RC9498; H, F, Me, Cl, c-Pr, Ph], [RC9499; H, F, Me, Cl, c-Pr, Bn], [RC9500; H, F, Me, Cl, c-Pr, CF ₃ ], [RC9501; H, F, Me, Cl, c-Pr, CF ₃ CH ₂ ], [RC9502; H, F, Me, Cl, c-Pr, CF ₃ CF ₂ ], [R C9503; H, F, Me, Cl, c-Pr, CF ₂ H], [RC9504; H, F, Me, Cl, c-Pr, CF ₂ HCF ₂ ], [RC9505; H, F, Et, H , c-Pr, Me], [RC9506; H, F, Et, H, c-Pr, Et], [RC9507; H, F, Et, H, c-Pr, Pr], [RC9508; H, F , Et, H, c-Pr, i-Pr], [RC9509; H, F, Et, H, c-Pr, c-Pr], [RC9510; H, F, Et, H, c-Pr, Bu ], [RC9511; H, F, Et, H, c-Pr, i-Bu], [RC9512; H, F, Et, H, c-Pr, t-Bu], [RC9513; H, F, Et , H, c-Pr, c-PrCH ₂ ], [RC9514; H, F, Et, H, c-Pr, Ph], [RC9515; H, F, Et, H, c-Pr, Bn], [ RC9516; H, F, Et, H, c-Pr, CF ₃ ], [RC9517; H, F, Et, H, c-Pr, CF ₃ CH ₂ ], [RC9518; H, F, Et, H, c-Pr, CF ₃ CF ₂ ], [RC9519; H, F, Et, H, c-Pr, CF ₂ H], [RC9520; H, F, Et, H, c-Pr, CF ₂ HCF ₂ ] , [RC9521; H, F, Et, F, c-Pr, Me], [RC9522; H, F, Et, F, c-Pr, Et], [RC9523; H, F, Et, F, c- Pr, Pr], [RC9524; H, F, Et, F, c-Pr, i-Pr], [RC9525; H, F, Et, F, c-Pr, c-Pr], [RC9526; H, F, Et, F, c-Pr, Bu], [RC9527; H, F, Et, F, c-Pr, i-Bu], [RC9528; H, F, Et, F, c-Pr, t- Bu], [RC9529; H, F, Et, F, c-Pr, c-PrCH ₂ ], [RC9530; H, F, Et, F, c-Pr, Ph], [RC9531; H, F, Et , F, c-Pr, Bn], [RC9532; H, F, Et, F, c-Pr, CF ₃ ], [RC9533; H, F, Et, F, c-Pr, CF ₃ CH ₂ ], [RC9534; H, F, Et, F, c-Pr, CF ₃ CF ₂ ], [RC9535; H, F, Et, F, c-Pr, CF ₂ H], [RC9536; H, F, Et, F, c-Pr, CF ₂ HCF ₂ ], [RC9537; H , F, Et, Cl, c-Pr, Me], [RC9538; H, F, Et, Cl, c-Pr, Et], [RC9539; H, F, Et, Cl, c-Pr, Pr], [RC9540; H, F, Et, Cl, c-Pr, i-Pr], [RC9541; H, F, Et, Cl, c-Pr, c-Pr], [RC9542; H, F, Et, Cl , c-Pr, Bu], [RC9543; H, F, Et, Cl, c-Pr, i-Bu], [RC9544; H, F, Et, Cl, c-Pr, t-Bu], [RC9545 ; H, F, Et, Cl, c-Pr, c-PrCH ₂ ], [RC9546; H, F, Et, Cl, c-Pr, Ph], [RC9547; H, F, Et, Cl, c- Pr, Bn], [RC9548; H, F, Et, Cl, c-Pr, CF ₃ ], [RC9549; H, F, Et, Cl, c-Pr, CF ₃ CH ₂ ], [RC9550; H, F, Et, Cl, c-Pr, CF ₃ CF ₂ ], [RC9551; H, F, Et, Cl, c-Pr, CF ₂ H], [RC9552; H, F, Et, Cl, c-Pr , CF ₂ HCF ₂ ], [RC9553; H, F, F, H, c-Pr, Me], [RC9554; H, F, F, H, c-Pr, Et], [RC9555; H, F, F, H, c-Pr, Pr], [RC9556; H, F, F, H, c-Pr, i-Pr], [RC9557; H, F, F, H, c-Pr, c-Pr] , [RC9558; H, F, F, H, c-Pr, Bu], [RC9559; H, F, F, H, c-Pr, i-Bu], [RC9560; H, F, F, H, c-Pr, t-Bu], [RC9561; H, F, F, H, c-Pr, c-PrCH ₂ ], [RC9562; H, F, F, H, c-Pr, Ph], [RC9563 ; H, F, F, H, c-Pr, Bn], [RC9564; H, F, F, H, c-Pr, CF ₃ ], [RC9565; H, F, F, H, c-Pr, CF ₃ CH ₂ ], [RC9566; H, F, F, H, c-Pr, CF ₃ CF ₂ ], [RC9567; H, F, F, H, c-Pr, CF ₂ H], [RC9568; H, F, F, H, c-Pr, CF ₂ HCF ₂ ], [RC9569; H, F, F, F, c-Pr, Me], [RC9570; H, F, F, F, c-Pr , Et], [RC9571; H, F, F, F, c-Pr, Pr], [RC9572; H, F, F, F, c-Pr, i-Pr], [RC9573; H, F, F, F, c-Pr, c-Pr], [RC9574; H, F, F, F, c- Pr, Bu], [RC9575; H, F, F, F, c-Pr, i-Bu], [RC9576; H, F, F, F, c-Pr, t-Bu], [RC9577; H, F, F, F, c-Pr, c-PrCH ₂ ], [RC9578; H, F, F, F, c-Pr, Ph], [RC9579; H, F, F, F, c-Pr, Bn ], [RC9580; H, F, F, F, c-Pr, CF ₃ ], [RC9581; H, F, F, F, c-Pr, CF ₃ CH ₂ ], [RC9582; H, F, F , F, c-Pr, CF ₃ CF ₂ ], [RC9583; H, F, F, F, c-Pr, CF ₂ H], [RC9584; H, F, F, F, c-Pr, CF ₂ HCF ₂ ], [RC9585; H, F, F, Cl, c-Pr, Me], [RC9586; H, F, F, Cl, c-Pr, Et], [RC9587; H, F, F, Cl , c-Pr, Pr], [RC9588; H, F, F, Cl, c-Pr, i-Pr], [RC9589; H, F, F, Cl, c-Pr, c-Pr], [RC9590 ; H, F, F, Cl, c-Pr, Bu], [RC9591; H, F, F, Cl, c-Pr, i-Bu], [RC9592; H, F, F, Cl, c-Pr , t-Bu], [RC9593; H, F, F, Cl, c-Pr, c-PrCH ₂ ], [RC9594; H, F, F, Cl, c-Pr, Ph], [RC9595; H, F, F, Cl, c-Pr, Bn], [RC9596; H, F, F, Cl, c-Pr, CF ₃ ], [RC9597; H, F, F, Cl, c-Pr, CF ₃ CH ₂ ], [RC9598; H, F, F, Cl, c-Pr, CF ₃ CF ₂ ], [RC9599; H, F, F, Cl, c-Pr, CF ₂ H], [RC9600; H, F , F, Cl, c-Pr, CF ₂ HCF ₂ ],

[RC9601; H, F, Cl, H, c-Pr, Me], [RC9602; H, F, Cl, H, c-Pr, Et], [RC9603; H, F, Cl, H, c-Pr , Pr], [RC9604; H, F, Cl, H, c-Pr, i-Pr], [RC9605; H, F, Cl, H, c-Pr, c-Pr], [RC9606; H, F , Cl, H, c-Pr, Bu], [RC9607; H, F, Cl, H, c-Pr, i-Bu], [RC9608; H, F, Cl, H, c-Pr, t-Bu ], [RC9609; H, F, Cl, H, c-Pr, c-PrCH ₂ ], [RC9610; H, F, Cl, H, c-Pr, Ph], [RC9611; H, F, Cl, H, c-Pr, Bn], [RC9612; H, F, Cl, H, c-Pr, CF ₃ ], [RC9613; H, F, Cl, H, c-Pr, CF ₃ CH ₂ ], [ RC9614; H, F, Cl, H, c-Pr, CF ₃ CF ₂ ], [RC9615; H, F, Cl, H, c-Pr, CF ₂ H], [RC9616; H, F, Cl, H , c-Pr, CF ₂ HCF ₂ ], [RC9617; H, F, Cl, Cl, c-Pr, Me], [RC9618; H, F, Cl, Cl, c-Pr, Et], [RC9619; H, F, Cl, Cl, c-Pr, Pr], [RC9620; H, F, Cl, Cl, c-Pr, i-Pr], [RC9621; H, F, Cl, Cl, c-Pr, c-Pr], [RC9622; H, F, Cl, Cl, c-Pr, Bu], [RC9623; H, F, Cl, Cl, c-Pr, i-Bu], [RC9624; H, F, Cl, Cl, c-Pr, t-Bu], [RC9625; H, F, Cl, Cl, c-Pr, c-PrCH ₂ ], [RC9626; H, F, Cl, Cl, c-Pr, Ph ], [RC9627; H, F, Cl, Cl, c-Pr, Bn], [RC9628; H, F, Cl, Cl, c-Pr, CF ₃ ], [RC9629; H, F, Cl, Cl, c-Pr, CF ₃ CH ₂ ], [RC9630; H, F, Cl, Cl, c-Pr, CF ₃ CF ₂ ], [RC9631; H, F, Cl, Cl, c-Pr, CF ₂ H] , [RC9632; H, F, Cl, Cl, c-Pr, CF ₂ HCF ₂ ], [RC9633; H, F, H, H, i-Bu, Me], [RC9634; H, F, H, H , i-Bu, Et], [RC9635; H, F, H, H, i-Bu, Pr], [RC9636; H, F, H, H, i-Bu, i-Pr], [RC9637; H, F, H, H, i-Bu, c-Pr], [RC9638; H, F, H, H, i-Bu, Bu], [RC9639; H, F, H, H, i-Bu, i-Bu], [RC9640; H, F, H, H, i-Bu, t-Bu], [RC9641; H, F, H, H, i-Bu, c-PrCH ₂ ], [RC9642; H, F, H, H, i-Bu, Ph ], [RC9643; H, F, H, H, i-Bu, Bn], [RC9644; H, F, H, H, i-Bu, CF ₃ ], [RC9645; H, F, H, H, i-Bu, CF ₃ CH ₂ ], [RC9646; H, F, H, H, i-Bu, CF ₃ CF ₂ ], [RC9647; H, F, H, H, i-Bu, CF ₂ H] , [RC9648; H, F, H, H, i-Bu, CF ₂ HCF ₂ ], [RC9649; H, F, H, Me, i-Bu, Me], [RC9650; H, F, H, Me , i-Bu, Et], [RC9651; H, F, H, Me, i-Bu, Pr], [RC9652; H, F, H, Me, i-Bu, i-Pr], [RC9653; H , F, H, Me, i-Bu, c-Pr], [RC9654; H, F, H, Me, i-Bu, Bu], [RC9655; H, F, H, Me, i-Bu, i -Bu], [RC9656; H, F, H, Me, i-Bu, t-Bu], [RC9657; H, F, H, Me, i-Bu, c-PrCH ₂ ], [RC9658; H, F, H, Me, i-Bu, Ph], [RC9659; H, F, H, Me, i-Bu, Bn], [RC9660; H, F, H, Me, i-Bu, CF ₃ ], [RC9661; H, F, H, Me, i-Bu, CF ₃ CH ₂ ], [RC9662; H, F, H, Me, i-Bu, CF ₃ CF ₂ ], [RC9663; H, F, H , Me, i-Bu, CF ₂ H], [RC9664; H, F, H, Me, i-Bu, CF ₂ HCF ₂ ], [RC9665; H, F, Me, Me, i-Bu, Me] , [RC9666; H, F, Me, Me, i-Bu, Et], [RC9667; H, F, Me, Me, i-Bu, Pr], [RC9668; H, F, Me, Me, i- Bu, i-Pr], [RC9669; H, F, Me, Me, i-Bu, c-Pr], [RC9670; H , F, Me, Me, i-Bu, Bu], [RC9671; H, F, Me, Me, i-Bu, i-Bu], [RC9672; H, F, Me, Me, i-Bu, t -Bu], [RC9673; H, F, Me, Me, i-Bu, c-PrCH ₂ ], [RC9674; H, F, Me, Me, i-Bu, Ph], [RC9675; H, F, Me, Me, i-Bu, Bn], [RC9676; H, F, Me, Me, i-Bu, CF ₃ ], [RC9677; H, F, Me, Me, i-Bu, CF ₃ CH ₂ ] , [RC9678; H, F, Me, Me, i-Bu, CF ₃ CF ₂ ], [RC9679; H, F, Me, Me, i-Bu, CF ₂ H], [RC9680; H, F, Me , Me, i-Bu, CF ₂ HCF ₂ ], [RC9681; H, F, Me, Et, i-Bu, Me], [RC9682; H, F, Me, Et, i-Bu, Et], [ RC9683; H, F, Me, Et, i-Bu, Pr], [RC9684; H, F, Me, Et, i-Bu, i-Pr], [RC9685; H, F, Me, Et, i- Bu, c-Pr], [RC9686; H, F, Me, Et, i-Bu, Bu], [RC9687; H, F, Me, Et, i-Bu, i-Bu], [RC9688; H, F, Me, Et, i-Bu, t-Bu], [RC9689; H, F, Me, Et, i-Bu, c-PrCH ₂ ], [RC9690; H, F, Me, Et, i-Bu , Ph], [RC9691; H, F, Me, Et, i-Bu, Bn], [RC9692; H, F, Me, Et, i-Bu, CF ₃ ], [RC9693; H, F, Me, Et, i-Bu, CF ₃ CH ₂ ], [RC9694; H, F, Me, Et, i-Bu, CF ₃ CF ₂ ], [RC9695; H, F, Me, Et, i-Bu, CF ₂ H], [RC9696; H, F, Me, Et, i-Bu, CF ₂ HCF ₂ ], [RC9697; H, F, Me, F, i-Bu, Me], [RC9698; H, F, Me , F, i-Bu, Et], [RC9699; H, F, Me, F, i-Bu, Pr], [RC9700; H, F, Me, F, i-Bu, i-Pr], [RC9701 ; H, F, Me, F, i-Bu, c-Pr], [RC9702; H, F, Me, F, i-Bu, Bu], [RC9703; H, F, Me, F, i-Bu , i-Bu], [R C9704; H, F, Me, F, i-Bu, t-Bu], [RC9705; H, F, Me, F, i-Bu, c-PrCH ₂ ], [RC9706; H, F, Me, F , i-Bu, Ph], [RC9707; H, F, Me, F, i-Bu, Bn], [RC9708; H, F, Me, F, i-Bu, CF ₃ ], [RC9709; H, F, Me, F, i-Bu, CF ₃ CH ₂ ], [RC9710; H, F, Me, F, i-Bu, CF ₃ CF ₂ ], [RC9711; H, F, Me, F, i- Bu, CF ₂ H], [RC9712; H, F, Me, F, i-Bu, CF ₂ HCF ₂ ], [RC9713; H, F, Me, Cl, i-Bu, Me], [RC9714; H , F, Me, Cl, i-Bu, Et], [RC9715; H, F, Me, Cl, i-Bu, Pr], [RC9716; H, F, Me, Cl, i-Bu, i-Pr ], [RC9717; H, F, Me, Cl, i-Bu, c-Pr], [RC9718; H, F, Me, Cl, i-Bu, Bu], [RC9719; H, F, Me, Cl , i-Bu, i-Bu], [RC9720; H, F, Me, Cl, i-Bu, t-Bu], [RC9721; H, F, Me, Cl, i-Bu, c-PrCH ₂ ] , [RC9722; H, F, Me, Cl, i-Bu, Ph], [RC9723; H, F, Me, Cl, i-Bu, Bn], [RC9724; H, F, Me, Cl, i- Bu, CF ₃ ], [RC9725; H, F, Me, Cl, i-Bu, CF ₃ CH ₂ ], [RC9726; H, F, Me, Cl, i-Bu, CF ₃ CF ₂ ], [RC9727 ; H, F, Me, Cl, i-Bu, CF ₂ H], [RC9728; H, F, Me, Cl, i-Bu, CF ₂ HCF ₂ ], [RC9729; H, F, Et, H, i-Bu, Me], [RC9730; H, F, Et, H, i-Bu, Et], [RC9731; H, F, Et, H, i-Bu, Pr], [RC9732; H, F, Et, H, i-Bu, i-Pr], [RC9733; H, F, Et, H, i-Bu, c-Pr], [RC9734; H, F, Et, H, i-Bu, Bu] , [RC9735; H, F, Et, H, i-Bu, i-Bu], [RC9736; H, F, Et, H, i-Bu, t-Bu], [RC9737; H, F, Et, H, i-Bu, c-PrCH ₂ ] , [RC9738; H, F, Et, H, i-Bu, Ph], [RC9739; H, F, Et, H, i-Bu, Bn], [RC9740; H, F, Et, H, i- Bu, CF ₃ ], [RC9741; H, F, Et, H, i-Bu, CF ₃ CH ₂ ], [RC9742; H, F, Et, H, i-Bu, CF ₃ CF ₂ ], [RC9743 ; H, F, Et, H, i-Bu, CF ₂ H], [RC9744; H, F, Et, H, i-Bu, CF ₂ HCF ₂ ], [RC9745; H, F, Et, F, i-Bu, Me], [RC9746; H, F, Et, F, i-Bu, Et], [RC9747; H, F, Et, F, i-Bu, Pr], [RC9748; H, F, Et, F, i-Bu, i-Pr], [RC9749; H, F, Et, F, i-Bu, c-Pr], [RC9750; H, F, Et, F, i-Bu, Bu] , [RC9751; H, F, Et, F, i-Bu, i-Bu], [RC9752; H, F, Et, F, i-Bu, t-Bu], [RC9753; H, F, Et, F, i-Bu, c-PrCH ₂ ], [RC9754; H, F, Et, F, i-Bu, Ph], [RC9755; H, F, Et, F, i-Bu, Bn], [RC9756 ; H, F, Et, F, i-Bu, CF ₃ ], [RC9757; H, F, Et, F, i-Bu, CF ₃ CH ₂ ], [RC9758; H, F, Et, F, i -Bu, CF ₃ CF ₂ ], [RC9759; H, F, Et, F, i-Bu, CF ₂ H], [RC9760; H, F, Et, F, i-Bu, CF ₂ HCF ₂ ], [RC9761; H, F, Et, Cl, i-Bu, Me], [RC9762; H, F, Et, Cl, i-Bu, Et], [RC9763; H, F, Et, Cl, i-Bu , Pr], [RC9764; H, F, Et, Cl, i-Bu, i-Pr], [RC9765; H, F, Et, Cl, i-Bu, c-Pr], [RC9766; H, F , Et, Cl, i-Bu, Bu], [RC9767; H, F, Et, Cl, i-Bu, i-Bu], [RC9768; H, F, Et, Cl, i-Bu, t-Bu ], [RC9769; H, F, Et, Cl, i-Bu, c-PrCH ₂ ], [RC9770; H, F, Et, Cl, i-Bu, Ph], [RC9771; H, F, Et, Cl, i-Bu, Bn], [RC9772; H, F, Et, Cl, i-Bu, CF ₃ ], [RC9773; H, F, Et, Cl, i-Bu, CF ₃ CH ₂ ], [RC9774; H, F, Et, Cl, i-Bu, CF ₃ CF ₂ ], [RC9775; H, F, Et, Cl, i-Bu, CF ₂ H], [RC9776; H, F, Et, Cl, i-Bu, CF ₂ HCF ₂ ], [RC9777; H, F, F, H, i-Bu, Me], [RC9778; H, F, F, H, i-Bu, Et], [RC9779; H, F, F, H, i-Bu, Pr] , [RC9780; H, F, F, H, i-Bu, i-Pr], [RC9781; H, F, F, H, i-Bu, c-Pr], [RC9782; H, F, F, H, i-Bu, Bu], [RC9783; H, F, F, H, i-Bu, i-Bu], [RC9784; H, F, F, H, i-Bu, t-Bu], [ RC9785; H, F, F, H, i-Bu, c-PrCH ₂ ], [RC9786; H, F, F, H, i-Bu, Ph], [RC9787; H, F, F, H, i -Bu, Bn], [RC9788; H, F, F, H, i-Bu, CF ₃ ], [RC9789; H, F, F, H, i-Bu, CF ₃ CH ₂ ], [RC9790; H , F, F, H, i-Bu, CF ₃ CF ₂ ], [RC9791; H, F, F, H, i-Bu, CF ₂ H], [RC9792; H, F, F, H, i- Bu, CF ₂ HCF ₂ ], [RC9793; H, F, F, F, i-Bu, Me], [RC9794; H, F, F, F, i-Bu, Et], [RC9795; H, F , F, F, i-Bu, Pr], [RC9796; H, F, F, F, i-Bu, i-Pr], [RC9797; H, F, F, F, i-Bu, c-Pr ], [RC9798; H, F, F, F, i-Bu, Bu], [RC9799; H, F, F, F, i-Bu, i-Bu], [RC9800; H, F, F, F , i-Bu, t-Bu],

[RC9801; H, F, F, F, i-Bu, c-PrCH ₂ ], [RC9802; H, F, F, F, i-Bu, Ph], [RC9803; H, F, F, F, i-Bu, Bn], [RC9804; H, F, F, F, i-Bu, CF ₃ ], [RC9805; H, F, F, F, i-Bu, CF ₃ CH ₂ ], [RC9806; H, F, F, F, i-Bu, CF ₃ CF ₂ ], [RC9807; H, F, F, F, i-Bu, CF ₂ H], [RC9808; H, F, F, F, i -Bu, CF ₂ HCF ₂ ], [RC9809; H, F, F, Cl, i-Bu, Me], [RC9810; H, F, F, Cl, i-Bu, Et], [RC9811; H, F, F, Cl, i-Bu, Pr], [RC9812; H, F, F, Cl, i-Bu, i-Pr], [RC9813; H, F, F, Cl, i-Bu, c- Pr], [RC9814; H, F, F, Cl, i-Bu, Bu], [RC9815; H, F, F, Cl, i-Bu, i-Bu], [RC9816; H, F, F, Cl, i-Bu, t-Bu], [RC9817; H, F, F, Cl, i-Bu, c-PrCH ₂ ], [RC9818; H, F, F, Cl, i-Bu, Ph], [RC9819; H, F, F, Cl, i-Bu, Bn], [RC9820; H, F, F, Cl, i-Bu, CF ₃ ], [RC9821; H, F, F, Cl, i- Bu, CF ₃ CH ₂ ], [RC9822; H, F, F, Cl, i-Bu, CF ₃ CF ₂ ], [RC9823; H, F, F, Cl, i-Bu, CF ₂ H], [ RC9824; H, F, F, Cl, i-Bu, CF ₂ HCF ₂ ], [RC9825; H, F, Cl, H, i-Bu, Me], [RC9826; H, F, Cl, H, i -Bu, Et], [RC9827; H, F, Cl, H, i-Bu, Pr], [RC9828; H, F, Cl, H, i-Bu, i-Pr], [RC9829; H, F , Cl, H, i-Bu, c-Pr], [RC9830; H, F, Cl, H, i-Bu, Bu], [RC9831; H, F, Cl, H, i-Bu, i-Bu ], [RC9832; H, F, Cl, H, i-Bu, t-Bu], [RC9833; H, F, Cl, H, i-Bu, c-PrCH ₂ ], [RC9834; H, F, Cl, H, i-Bu, Ph], [RC9835; H, F, Cl, H, i-Bu, B n], [RC9836; H, F, Cl, H, i-Bu, CF ₃ ], [RC9837; H, F, Cl, H, i-Bu, CF ₃ CH ₂ ], [RC9838; H, F, Cl, H, i-Bu, CF ₃ CF ₂ ], [RC9839; H, F, Cl, H, i-Bu, CF ₂ H], [RC9840; H, F, Cl, H, i-Bu, CF ₂ HCF ₂ ], [RC9841; H, F, Cl, Cl, i-Bu, Me], [RC9842; H, F, Cl, Cl, i-Bu, Et], [RC9843; H, F, Cl, Cl, i-Bu, Pr], [RC9844; H, F, Cl, Cl, i-Bu, i-Pr], [RC9845; H, F, Cl, Cl, i-Bu, c-Pr], [ RC9846; H, F, Cl, Cl, i-Bu, Bu], [RC9847; H, F, Cl, Cl, i-Bu, i-Bu], [RC9848; H, F, Cl, Cl, i- Bu, t-Bu], [RC9849; H, F, Cl, Cl, i-Bu, c-PrCH ₂ ], [RC9850; H, F, Cl, Cl, i-Bu, Ph], [RC9851; H , F, Cl, Cl, i-Bu, Bn], [RC9852; H, F, Cl, Cl, i-Bu, CF ₃ ], [RC9853; H, F, Cl, Cl, i-Bu, CF ₃ CH ₂ ], [RC9854; H, F, Cl, Cl, i-Bu, CF ₃ CF ₂ ], [RC9855; H, F, Cl, Cl, i-Bu, CF ₂ H], [RC9856; H, F, Cl, Cl, i-Bu, CF ₂ HCF ₂ ], [RC9857; H, F, H, H, t-Bu, Me], [RC9858; H, F, H, H, t-Bu, Et ], [RC9859; H, F, H, H, t-Bu, Pr], [RC9860; H, F, H, H, t-Bu, i-Pr], [RC9861; H, F, H, H , t-Bu, c-Pr], [RC9862; H, F, H, H, t-Bu, Bu], [RC9863; H, F, H, H, t-Bu, i-Bu], [RC9864 ; H, F, H, H, t-Bu, t-Bu], [RC9865; H, F, H, H, t-Bu, c-PrCH ₂ ], [RC9866; H, F, H, H, t-Bu, Ph], [RC9867; H, F, H, H, t-Bu, Bn], [RC9868; H, F, H, H, t-Bu, CF ₃ ], [RC9869; H, F , H, H, t-Bu, CF ₃ CH ₂ ], [RC98 70; H, F, H, H, t-Bu, CF ₃ CF ₂ ], [RC9871; H, F, H, H, t-Bu, CF ₂ H], [RC9872; H, F, H, H , t-Bu, CF ₂ HCF ₂ ], [RC9873; H, F, H, Me, t-Bu, Me], [RC9874; H, F, H, Me, t-Bu, Et], [RC9875; H, F, H, Me, t-Bu, Pr], [RC9876; H, F, H, Me, t-Bu, i-Pr], [RC9877; H, F, H, Me, t-Bu, c-Pr], [RC9878; H, F, H, Me, t-Bu, Bu], [RC9879; H, F, H, Me, t-Bu, i-Bu], [RC9880; H, F, H, Me, t-Bu, t-Bu], [RC9881; H, F, H, Me, t-Bu, c-PrCH ₂ ], [RC9882; H, F, H, Me, t-Bu, Ph ], [RC9883; H, F, H, Me, t-Bu, Bn], [RC9884; H, F, H, Me, t-Bu, CF ₃ ], [RC9885; H, F, H, Me, t-Bu, CF ₃ CH ₂ ], [RC9886; H, F, H, Me, t-Bu, CF ₃ CF ₂ ], [RC9887; H, F, H, Me, t-Bu, CF ₂ H] , [RC9888; H, F, H, Me, t-Bu, CF ₂ HCF ₂ ], [RC9889; H, F, Me, Me, t-Bu, Me], [RC9890; H, F, Me, Me , t-Bu, Et], [RC9891; H, F, Me, Me, t-Bu, Pr], [RC9892; H, F, Me, Me, t-Bu, i-Pr], [RC9893; H , F, Me, Me, t-Bu, c-Pr], [RC9894; H, F, Me, Me, t-Bu, Bu], [RC9895; H, F, Me, Me, t-Bu, i -Bu], [RC9896; H, F, Me, Me, t-Bu, t-Bu], [RC9897; H, F, Me, Me, t-Bu, c-PrCH ₂ ], [RC9898; H, F, Me, Me, t-Bu, Ph], [RC9899; H, F, Me, Me, t-Bu, Bn], [RC9900; H, F, Me, Me, t-Bu, CF ₃ ], [RC9901; H, F, Me, Me, t-Bu, CF ₃ CH ₂ ], [RC9902; H, F, Me, Me, t-Bu, CF ₃ CF ₂ ], [RC9903; H, F, Me , Me, t-Bu, CF ₂ H], [RC 9904; H, F, Me, Me, t-Bu, CF ₂ HCF ₂ ], [RC9905; H, F, Me, Et, t-Bu, Me], [RC9906; H, F, Me, Et, t -Bu, Et], [RC9907; H, F, Me, Et, t-Bu, Pr], [RC9908; H, F, Me, Et, t-Bu, i-Pr], [RC9909; H, F , Me, Et, t-Bu, c-Pr], [RC9910; H, F, Me, Et, t-Bu, Bu], [RC9911; H, F, Me, Et, t-Bu, i-Bu ], [RC9912; H, F, Me, Et, t-Bu, t-Bu], [RC9913; H, F, Me, Et, t-Bu, c-PrCH ₂ ], [RC9914; H, F, Me, Et, t-Bu, Ph], [RC9915; H, F, Me, Et, t-Bu, Bn], [RC9916; H, F, Me, Et, t-Bu, CF ₃ ], [RC9917 ; H, F, Me, Et, t-Bu, CF ₃ CH ₂ ], [RC9918; H, F, Me, Et, t-Bu, CF ₃ CF ₂ ], [RC9919; H, F, Me, Et , t-Bu, CF ₂ H], [RC9920; H, F, Me, Et, t-Bu, CF ₂ HCF ₂ ], [RC9921; H, F, Me, F, t-Bu, Me], [ RC9922; H, F, Me, F, t-Bu, Et], [RC9923; H, F, Me, F, t-Bu, Pr], [RC9924; H, F, Me, F, t-Bu, i-Pr], [RC9925; H, F, Me, F, t-Bu, c-Pr], [RC9926; H, F, Me, F, t-Bu, Bu], [RC9927; H, F, Me, F, t-Bu, i-Bu], [RC9928; H, F, Me, F, t-Bu, t-Bu], [RC9929; H, F, Me, F, t-Bu, c- PrCH ₂ ], [RC9930; H, F, Me, F, t-Bu, Ph], [RC9931; H, F, Me, F, t-Bu, Bn], [RC9932; H, F, Me, F , t-Bu, CF ₃ ], [RC9933; H, F, Me, F, t-Bu, CF ₃ CH ₂ ], [RC9934; H, F, Me, F, t-Bu, CF ₃ CF ₂ ] , [RC9935; H, F, Me, F, t-Bu, CF ₂ H], [RC9936; H, F, Me, F, t-Bu, CF ₂ HCF ₂ ], [RC9937; H, F, Me , Cl, t-Bu, Me ], [RC9938; H, F, Me, Cl, t-Bu, Et], [RC9939; H, F, Me, Cl, t-Bu, Pr], [RC9940; H, F, Me, Cl, t -Bu, i-Pr], [RC9941; H, F, Me, Cl, t-Bu, c-Pr], [RC9942; H, F, Me, Cl, t-Bu, Bu], [RC9943; H , F, Me, Cl, t-Bu, i-Bu], [RC9944; H, F, Me, Cl, t-Bu, t-Bu], [RC9945; H, F, Me, Cl, t-Bu , c-PrCH ₂ ], [RC9946; H, F, Me, Cl, t-Bu, Ph], [RC9947; H, F, Me, Cl, t-Bu, Bn], [RC9948; H, F, Me, Cl, t-Bu, CF ₃ ], [RC9949; H, F, Me, Cl, t-Bu, CF ₃ CH ₂ ], [RC9950; H, F, Me, Cl, t-Bu, CF ₃ CF ₂ ], [RC9951; H, F, Me, Cl, t-Bu, CF ₂ H], [RC9952; H, F, Me, Cl, t-Bu, CF ₂ HCF ₂ ], [RC9953; H, F, Et, H, t-Bu, Me], [RC9954; H, F, Et, H, t-Bu, Et], [RC9955; H, F, Et, H, t-Bu, Pr], [ RC9956; H, F, Et, H, t-Bu, i-Pr], [RC9957; H, F, Et, H, t-Bu, c-Pr], [RC9958; H, F, Et, H, t-Bu, Bu], [RC9959; H, F, Et, H, t-Bu, i-Bu], [RC9960; H, F, Et, H, t-Bu, t-Bu], [RC9961; H, F, Et, H, t-Bu, c-PrCH ₂ ], [RC9962; H, F, Et, H, t-Bu, Ph], [RC9963; H, F, Et, H, t-Bu , Bn], [RC9964; H, F, Et, H, t-Bu, CF ₃ ], [RC9965; H, F, Et, H, t-Bu, CF ₃ CH ₂ ], [RC9966; H, F , Et, H, t-Bu, CF ₃ CF ₂ ], [RC9967; H, F, Et, H, t-Bu, CF ₂ H], [RC9968; H, F, Et, H, t-Bu, CF ₂ HCF ₂ ], [RC9969; H, F, Et, F, t-Bu, Me], [RC9970; H, F, Et, F, t-Bu, Et], [RC9971; H, F, Et , F, t-Bu, Pr], [RC99 72; H, F, Et, F, t-Bu, i-Pr], [RC9973; H, F, Et, F, t-Bu, c-Pr], [RC9974; H, F, Et, F, t-Bu, Bu], [RC9975; H, F, Et, F, t-Bu, i-Bu], [RC9976; H, F, Et, F, t-Bu, t-Bu], [RC9977; H, F, Et, F, t-Bu, c-PrCH ₂ ], [RC9978; H, F, Et, F, t-Bu, Ph], [RC9979; H, F, Et, F, t-Bu , Bn], [RC9980; H, F, Et, F, t-Bu, CF ₃ ], [RC9981; H, F, Et, F, t-Bu, CF ₃ CH ₂ ], [RC9982; H, F , Et, F, t-Bu, CF ₃ CF ₂ ], [RC9983; H, F, Et, F, t-Bu, CF ₂ H], [RC9984; H, F, Et, F, t-Bu, CF ₂ HCF ₂ ], [RC9985; H, F, Et, Cl, t-Bu, Me], [RC9986; H, F, Et, Cl, t-Bu, Et], [RC9987; H, F, Et , Cl, t-Bu, Pr], [RC9988; H, F, Et, Cl, t-Bu, i-Pr], [RC9989; H, F, Et, Cl, t-Bu, c-Pr], [RC9990; H, F, Et, Cl, t-Bu, Bu], [RC9991; H, F, Et, Cl, t-Bu, i-Bu], [RC9992; H, F, Et, Cl, t -Bu, t-Bu], [RC9993; H, F, Et, Cl, t-Bu, c-PrCH ₂ ], [RC9994; H, F, Et, Cl, t-Bu, Ph], [RC9995; H, F, Et, Cl, t-Bu, Bn], [RC9996; H, F, Et, Cl, t-Bu, CF ₃ ], [RC9997; H, F, Et, Cl, t-Bu, CF ₃ CH ₂ ], [RC9998; H, F, Et, Cl, t-Bu, CF ₃ CF ₂ ], [RC9999; H, F, Et, Cl, t-Bu, CF ₂ H], [RC10000; H , F, Et, Cl, t-Bu, CF ₂ HCF ₂ ],

[RC10001; H, F, F, H, t-Bu, Me], [RC10002; H, F, F, H, t-Bu, Et], [RC10003; H, F, F, H, t-Bu , Pr], [RC10004; H, F, F, H, t-Bu, i-Pr], [RC10005; H, F, F, H, t-Bu, c-Pr], [RC10006; H, F , F, H, t-Bu, Bu], [RC10007; H, F, F, H, t-Bu, i-Bu], [RC10008; H, F, F, H, t-Bu, t-Bu ], [RC10009; H, F, F, H, t-Bu, c-PrCH ₂ ], [RC10010; H, F, F, H, t-Bu, Ph], [RC10011; H, F, F, H, t-Bu, Bn], [RC10012; H, F, F, H, t-Bu, CF ₃ ], [RC10013; H, F, F, H, t-Bu, CF ₃ CH ₂ ], [ RC10014; H, F, F, H, t-Bu, CF ₃ CF ₂ ], [RC10015; H, F, F, H, t-Bu, CF ₂ H], [RC10016; H, F, F, H , t-Bu, CF ₂ HCF ₂ ], [RC10017; H, F, F, F, t-Bu, Me], [RC10018; H, F, F, F, t-Bu, Et], [RC10019; H, F, F, F, t-Bu, Pr], [RC10020; H, F, F, F, t-Bu, i-Pr], [RC10021; H, F, F, F, t-Bu, c-Pr], [RC10022; H, F, F, F, t-Bu, Bu], [RC10023; H, F, F, F, t-Bu, i-Bu], [RC10024; H, F, F, F, t-Bu, t-Bu], [RC10025; H, F, F, F, t-Bu, c-PrCH ₂ ], [RC10026; H, F, F, F, t-Bu, Ph ], [RC10027; H, F, F, F, t-Bu, Bn], [RC10028; H, F, F, F, t-Bu, CF ₃ ], [RC10029; H, F, F, F, t-Bu, CF ₃ CH ₂ ], [RC10030; H, F, F, F, t-Bu, CF ₃ CF ₂ ], [RC10031; H, F, F, F, t-Bu, CF ₂ H] , [RC10032; H, F, F, F, t-Bu, CF ₂ HCF ₂ ], [RC10033; H, F, F, Cl, t-Bu, Me], [RC10034; H, F, F, Cl , t-Bu, Et], [RC10035; H, F, F, Cl, t- Bu, Pr], [RC10036; H, F, F, Cl, t-Bu, i-Pr], [RC10037; H, F, F, Cl, t-Bu, c-Pr], [RC10038; H, F, F, Cl, t-Bu, Bu], [RC10039; H, F, F, Cl, t-Bu, i-Bu], [RC10040; H, F, F, Cl, t-Bu, t- Bu], [RC10041; H, F, F, Cl, t-Bu, c-PrCH ₂ ], [RC10042; H, F, F, Cl, t-Bu, Ph], [RC10043; H, F, F , Cl, t-Bu, Bn], [RC10044; H, F, F, Cl, t-Bu, CF ₃ ], [RC10045; H, F, F, Cl, t-Bu, CF ₃ CH ₂ ], [RC10046; H, F, F, Cl, t-Bu, CF ₃ CF ₂ ], [RC10047; H, F, F, Cl, t-Bu, CF ₂ H], [RC10048; H, F, F, Cl, t-Bu, CF ₂ HCF ₂ ], [RC10049; H, F, Cl, H, t-Bu, Me], [RC10050; H, F, Cl, H, t-Bu, Et], [RC10051 ; H, F, Cl, H, t-Bu, Pr], [RC10052; H, F, Cl, H, t-Bu, i-Pr], [RC10053; H, F, Cl, H, t-Bu , c-Pr], [RC10054; H, F, Cl, H, t-Bu, Bu], [RC10055; H, F, Cl, H, t-Bu, i-Bu], [RC10056; H, F , Cl, H, t-Bu, t-Bu], [RC10057; H, F, Cl, H, t-Bu, c-PrCH ₂ ], [RC10058; H, F, Cl, H, t-Bu, Ph], [RC10059; H, F, Cl, H, t-Bu, Bn], [RC10060; H, F, Cl, H, t-Bu, CF ₃ ], [RC10061; H, F, Cl, H , t-Bu, CF ₃ CH ₂ ], [RC10062; H, F, Cl, H, t-Bu, CF ₃ CF ₂ ], [RC10063; H, F, Cl, H, t-Bu, CF ₂ H ], [RC10064; H, F, Cl, H, t-Bu, CF ₂ HCF ₂ ], [RC10065; H, F, Cl, Cl, t-Bu, Me], [RC10066; H, F, Cl, Cl, t-Bu, Et], [RC10067; H, F, Cl, Cl, t-Bu, Pr], [RC10068; H, F, Cl, Cl, t-Bu, i-Pr], [R C10069; H, F, Cl, Cl, t-Bu, c-Pr], [RC10070; H, F, Cl, Cl, t-Bu, Bu], [RC10071; H, F, Cl, Cl, t- Bu, i-Bu], [RC10072; H, F, Cl, Cl, t-Bu, t-Bu], [RC10073; H, F, Cl, Cl, t-Bu, c-PrCH ₂ ], [RC10074 ; H, F, Cl, Cl, t-Bu, Ph], [RC10075; H, F, Cl, Cl, t-Bu, Bn], [RC10076; H, F, Cl, Cl, t-Bu, CF ₃ ], [RC10077; H, F, Cl, Cl, t-Bu, CF ₃ CH ₂ ], [RC10078; H, F, Cl, Cl, t-Bu, CF ₃ CF ₂ ], [RC10079; H, F, Cl, Cl, t-Bu, CF ₂ H], [RC10080; H, F, Cl, Cl, t-Bu, CF ₂ HCF ₂ ], [RC10081; H, F, H, H, CF ₂ H , Me], [RC10082; H, F, H, H, CF ₂ H, Et], [RC10083; H, F, H, H, CF ₂ H, Pr], [RC10084; H, F, H, H , CF ₂ H, i-Pr], [RC10085; H, F, H, H, CF ₂ H, c-Pr], [RC10086; H, F, H, H, CF ₂ H, Bu], [RC10087 ; H, F, H, H, CF ₂ H, i-Bu], [RC10088; H, F, H, H, CF ₂ H, t-Bu], [RC10089; H, F, H, H, CF ₂ H, c-PrCH ₂ ], [RC10090; H, F, H, H, CF ₂ H, Ph], [RC10091; H, F, H, H, CF ₂ H, Bn], [RC10092; H, F, H, H, CF ₂ H, CF ₃ ], [RC10093; H, F, H, H, CF ₂ H, CF ₃ CH ₂ ], [RC10094; H, F, H, H, CF ₂ H, CF ₃ CF ₂ ], [RC10095; H, F, H, H, CF ₂ H, CF ₂ H], [RC10096; H, F, H, H, CF ₂ H, CF ₂ HCF ₂ ], [RC10097; H, F, H, Me, CF ₂ H, Me], [RC10098; H, F, H, Me, CF ₂ H, Et], [RC10099; H, F, H, Me, CF ₂ H, Pr] , [RC10100; H, F, H, Me, CF ₂ H, i-Pr], [RC10101 ; H, F, H, Me, CF ₂ H, c-Pr], [RC10102; H, F, H, Me, CF ₂ H, Bu], [RC10103; H, F, H, Me, CF ₂ H , i-Bu], [RC10104; H, F, H, Me, CF ₂ H, t-Bu], [RC10105; H, F, H, Me, CF ₂ H, c-PrCH ₂ ], [RC10106; H, F, H, Me, CF ₂ H, Ph], [RC10107; H, F, H, Me, CF ₂ H, Bn], [RC10108; H, F, H, Me, CF ₂ H, CF ₃ ], [RC10109; H, F, H, Me, CF ₂ H, CF ₃ CH ₂ ], [RC10110; H, F, H, Me, CF ₂ H, CF ₃ CF ₂ ], [RC10111; H, F , H, Me, CF ₂ H, CF ₂ H], [RC10112; H, F, H, Me, CF ₂ H, CF ₂ HCF ₂ ], [RC10113; H, F, Me, Me, CF ₂ H, Me], [RC10114; H, F, Me, Me, CF ₂ H, Et], [RC10115; H, F, Me, Me, CF ₂ H, Pr], [RC10116; H, F, Me, Me, CF ₂ H, i-Pr], [RC10117; H, F, Me, Me, CF ₂ H, c-Pr], [RC10118; H, F, Me, Me, CF ₂ H, Bu], [RC10119; H, F, Me, Me, CF ₂ H, i-Bu], [RC10120; H, F, Me, Me, CF ₂ H, t-Bu], [RC10121; H, F, Me, Me, CF ₂ H, c-PrCH ₂ ], [RC10122; H, F, Me, Me, CF ₂ H, Ph], [RC10123; H, F, Me, Me, CF ₂ H, Bn], [RC10124; H, F , Me, Me, CF ₂ H, CF ₃ ], [RC10125; H, F, Me, Me, CF ₂ H, CF ₃ CH ₂ ], [RC10126; H, F, Me, Me, CF ₂ H, CF ₃ CF ₂ ], [RC10127; H, F, Me, Me, CF ₂ H, CF ₂ H], [RC10128; H, F, Me, Me, CF ₂ H, CF ₂ HCF ₂ ], [RC10129; H , F, Me, Et, CF ₂ H, Me], [RC10130; H, F, Me, Et, CF ₂ H, Et], [RC10131; H, F, Me, Et, CF ₂ H, Pr ], [RC10132; H, F, Me, Et, CF ₂ H, i-Pr], [RC10133; H, F, Me, Et, CF ₂ H, c-Pr], [RC10134; H, F, Me , Et, CF ₂ H, Bu], [RC10135; H, F, Me, Et, CF ₂ H, i-Bu], [RC10136; H, F, Me, Et, CF ₂ H, t-Bu], [RC10137; H, F, Me, Et, CF ₂ H, c-PrCH ₂ ], [RC10138; H, F, Me, Et, CF ₂ H, Ph], [RC10139; H, F, Me, Et, CF ₂ H, Bn], [RC10140; H, F, Me, Et, CF ₂ H, CF ₃ ], [RC10141; H, F, Me, Et, CF ₂ H, CF ₃ CH ₂ ], [RC10142; H, F, Me, Et, CF ₂ H, CF ₃ CF ₂ ], [RC10143; H, F, Me, Et, CF ₂ H, CF ₂ H], [RC10144; H, F, Me, Et, CF ₂ H, CF ₂ HCF ₂ ], [RC10145; H, F, Me, F, CF ₂ H, Me], [RC10146; H, F, Me, F, CF ₂ H, Et], [RC10147; H, F, Me, F, CF ₂ H, Pr], [RC10148; H, F, Me, F, CF ₂ H, i-Pr], [RC10149; H, F, Me, F, CF ₂ H, c- Pr], [RC10150; H, F, Me, F, CF ₂ H, Bu], [RC10151; H, F, Me, F, CF ₂ H, i-Bu], [RC10152; H, F, Me, F, CF ₂ H, t-Bu], [RC10153; H, F, Me, F, CF ₂ H, c-PrCH ₂ ], [RC10154; H, F, Me, F, CF ₂ H, Ph], [RC10155; H, F, Me, F, CF ₂ H, Bn], [RC10156; H, F, Me, F, CF ₂ H, CF ₃ ], [RC10157; H, F, Me, F, CF ₂ H, CF ₃ CH ₂ ], [RC10158; H, F, Me, F, CF ₂ H, CF ₃ CF ₂ ], [RC10159; H, F, Me, F, CF ₂ H, CF ₂ H], [ RC10160; H, F, Me, F, CF ₂ H, CF ₂ HCF ₂ ], [RC10161; H, F, Me, Cl, CF ₂ H, Me], [RC10162; H, F, Me, Cl, C F ₂ H, Et], [RC10163; H, F, Me, Cl, CF ₂ H, Pr], [RC10164; H, F, Me, Cl, CF ₂ H, i-Pr], [RC10165; H, F, Me, Cl, CF ₂ H, c-Pr], [RC10166; H, F, Me, Cl, CF ₂ H, Bu], [RC10167; H, F, Me, Cl, CF ₂ H, i- Bu], [RC10168; H, F, Me, Cl, CF ₂ H, t-Bu], [RC10169; H, F, Me, Cl, CF ₂ H, c-PrCH ₂ ], [RC10170; H, F , Me, Cl, CF ₂ H, Ph], [RC10171; H, F, Me, Cl, CF ₂ H, Bn], [RC10172; H, F, Me, Cl, CF ₂ H, CF ₃ ], [ RC10173; H, F, Me, Cl, CF ₂ H, CF ₃ CH ₂ ], [RC10174; H, F, Me, Cl, CF ₂ H, CF ₃ CF ₂ ], [RC10175; H, F, Me, Cl, CF ₂ H, CF ₂ H], [RC10176; H, F, Me, Cl, CF ₂ H, CF ₂ HCF ₂ ], [RC10177; H, F, Et, H, CF ₂ H, Me], [RC10178; H, F, Et, H, CF ₂ H, Et], [RC10179; H, F, Et, H, CF ₂ H, Pr], [RC10180; H, F, Et, H, CF ₂ H , i-Pr], [RC10181; H, F, Et, H, CF ₂ H, c-Pr], [RC10182; H, F, Et, H, CF ₂ H, Bu], [RC10183; H, F , Et, H, CF ₂ H, i-Bu], [RC10184; H, F, Et, H, CF ₂ H, t-Bu], [RC10185; H, F, Et, H, CF ₂ H, c -PrCH ₂ ], [RC10186; H, F, Et, H, CF ₂ H, Ph], [RC10187; H, F, Et, H, CF ₂ H, Bn], [RC10188; H, F, Et, H, CF ₂ H, CF ₃ ], [RC10189; H, F, Et, H, CF ₂ H, CF ₃ CH ₂ ], [RC10190; H, F, Et, H, CF ₂ H, CF ₃ CF ₂ ], [RC10191; H, F, Et, H, CF ₂ H, CF ₂ H], [RC10192; H, F, Et, H, CF ₂ H, CF ₂ HCF ₂ ], [RC10193; H, F , Et, F, CF ₂ H, Me], [RC10194; H, F, Et, F, CF ₂ H, Et], [RC10195; H, F, Et, F, CF ₂ H, Pr], [RC10196 ; H, F, Et, F, CF ₂ H, i-Pr], [RC10197; H, F, Et, F, CF ₂ H, c-Pr], [RC10198; H, F, Et, F, CF ₂ H, Bu], [RC10199; H, F, Et, F, CF ₂ H, i-Bu], [RC10200; H, F, Et, F, CF ₂ H, t-Bu],

[RC10201; H, F, Et, F, CF ₂ H, c-PrCH ₂ ], [RC10202; H, F, Et, F, CF ₂ H, Ph], [RC10203; H, F, Et, F, CF ₂ H, Bn], [RC10204; H, F, Et, F, CF ₂ H, CF ₃ ], [RC10205; H, F, Et, F, CF ₂ H, CF ₃ CH ₂ ], [RC10206; H, F, Et, F, CF ₂ H, CF ₃ CF ₂ ], [RC10207; H, F, Et, F, CF ₂ H, CF ₂ H], [RC10208; H, F, Et, F, CF ₂ H, CF ₂ HCF ₂ ], [RC10209; H, F, Et, Cl, CF ₂ H, Me], [RC10210; H, F, Et, Cl, CF ₂ H, Et], [RC10211; H, F, Et, Cl, CF ₂ H, Pr], [RC10212; H, F, Et, Cl, CF ₂ H, i-Pr], [RC10213; H, F, Et, Cl, CF ₂ H, c- Pr], [RC10214; H, F, Et, Cl, CF ₂ H, Bu], [RC10215; H, F, Et, Cl, CF ₂ H, i-Bu], [RC10216; H, F, Et, Cl, CF ₂ H, t-Bu], [RC10217; H, F, Et, Cl, CF ₂ H, c-PrCH ₂ ], [RC10218; H, F, Et, Cl, CF ₂ H, Ph], [RC10219; H, F, Et, Cl, CF ₂ H, Bn], [RC10220; H, F, Et, Cl, CF ₂ H, CF ₃ ], [RC10221; H, F, Et, Cl, CF ₂ H, CF ₃ CH ₂ ], [RC10222; H, F, Et, Cl, CF ₂ H, CF ₃ CF ₂ ], [RC10223; H, F, Et, Cl, CF ₂ H, CF ₂ H], [ RC10224; H, F, Et, Cl, CF ₂ H, CF ₂ HCF ₂ ], [RC10225; H, F, F, H, CF ₂ H, Me], [RC10226; H, F, F, H, CF ₂ H, Et], [RC10227; H, F, F, H, CF ₂ H, Pr], [RC10228; H, F, F, H, CF ₂ H, i-Pr], [RC10229; H, F , F, H, CF ₂ H, c-Pr], [RC10230; H, F, F, H, CF ₂ H, Bu], [RC10231; H, F, F, H, CF ₂ H, i-Bu ], [RC10232; H, F, F, H, CF ₂ H, t-Bu], [RC10233; H, F, F, H, CF ₂ H, c-PrCH ₂ ], [RC10234; H, F, F, H, CF ₂ H, Ph], [RC10235; H, F, F, H, CF ₂ H, Bn], [RC10236; H, F, F, H, CF ₂ H, CF ₃ ], [RC10237; H , F, F, H, CF ₂ H, CF ₃ CH ₂ ], [RC10238; H, F, F, H, CF ₂ H, CF ₃ CF ₂ ], [RC10239; H, F, F, H, CF ₂ H, CF ₂ H], [RC10240; H, F, F, H, CF ₂ H, CF ₂ HCF ₂ ], [RC10241; H, F, F, F, CF ₂ H, Me], [RC10242; H, F, F, F, CF ₂ H, Et], [RC10243; H, F, F, F, CF ₂ H, Pr], [RC10244; H, F, F, F, CF ₂ H, i- Pr], [RC10245; H, F, F, F, CF ₂ H, c-Pr], [RC10246; H, F, F, F, CF ₂ H, Bu], [RC10247; H, F, F, F, CF ₂ H, i-Bu], [RC10248; H, F, F, F, CF ₂ H, t-Bu], [RC10249; H, F, F, F, CF ₂ H, c-PrCH ₂ ], [RC10250; H, F, F, F, CF ₂ H, Ph], [RC10251; H, F, F, F, CF ₂ H, Bn], [RC10252; H, F, F, F, CF ₂ H, CF ₃ ], [RC10253; H, F, F, F, CF ₂ H, CF ₃ CH ₂ ], [RC10254; H, F, F, F, CF ₂ H, CF ₃ CF ₂ ], [ RC10255; H, F, F, F, CF ₂ H, CF ₂ H], [RC10256; H, F, F, F, CF ₂ H, CF ₂ HCF ₂ ], [RC10257; H, F, F, Cl , CF ₂ H, Me], [RC10258; H, F, F, Cl, CF ₂ H, Et], [RC10259; H, F, F, Cl, CF ₂ H, Pr], [RC10260; H, F , F, Cl, CF ₂ H, i-Pr], [RC10261; H, F, F, Cl, CF ₂ H, c-Pr], [RC10262; H, F, F, Cl, CF ₂ H, Bu ], [RC10263; H, F, F, Cl, CF ₂ H, i-Bu], [RC 10264; H, F, F, Cl, CF ₂ H, t-Bu], [RC10265; H, F, F, Cl, CF ₂ H, c-PrCH ₂ ], [RC10266; H, F, F, Cl , CF ₂ H, Ph], [RC10267; H, F, F, Cl, CF ₂ H, Bn], [RC10268; H, F, F, Cl, CF ₂ H, CF ₃ ], [RC10269; H, F, F, Cl, CF ₂ H, CF ₃ CH ₂ ], [RC10270; H, F, F, Cl, CF ₂ H, CF ₃ CF ₂ ], [RC10271; H, F, F, Cl, CF ₂ H, CF ₂ H], [RC10272; H, F, F, Cl, CF ₂ H, CF ₂ HCF ₂ ], [RC10273; H, F, Cl, H, CF ₂ H, Me], [RC10274; H , F, Cl, H, CF ₂ H, Et], [RC10275; H, F, Cl, H, CF ₂ H, Pr], [RC10276; H, F, Cl, H, CF ₂ H, i-Pr ], [RC10277; H, F, Cl, H, CF ₂ H, c-Pr], [RC10278; H, F, Cl, H, CF ₂ H, Bu], [RC10279; H, F, Cl, H , CF ₂ H, i-Bu], [RC10280; H, F, Cl, H, CF ₂ H, t-Bu], [RC10281; H, F, Cl, H, CF ₂ H, c-PrCH ₂ ] , [RC10282; H, F, Cl, H, CF ₂ H, Ph], [RC10283; H, F, Cl, H, CF ₂ H, Bn], [RC10284; H, F, Cl, H, CF ₂ H, CF ₃ ], [RC10285; H, F, Cl, H, CF ₂ H, CF ₃ CH ₂ ], [RC10286; H, F, Cl, H, CF ₂ H, CF ₃ CF ₂ ], [RC10287 ; H, F, Cl, H, CF ₂ H, CF ₂ H], [RC10288; H, F, Cl, H, CF ₂ H, CF ₂ HCF ₂ ], [RC10289; H, F, Cl, Cl, CF ₂ H, Me], [RC10290; H, F, Cl, Cl, CF ₂ H, Et], [RC10291; H, F, Cl, Cl, CF ₂ H, Pr], [RC10292; H, F, Cl, Cl, CF ₂ H, i-Pr], [RC10293; H, F, Cl, Cl, CF ₂ H, c-Pr], [RC10294; H, F, Cl, Cl, CF ₂ H, Bu] , [RC102 95; H, F, Cl, Cl, CF ₂ H, i-Bu], [RC10296; H, F, Cl, Cl, CF ₂ H, t-Bu], [RC10297; H, F, Cl, Cl, CF ₂ H, c-PrCH ₂ ], [RC10298; H, F, Cl, Cl, CF ₂ H, Ph], [RC10299; H, F, Cl, Cl, CF ₂ H, Bn], [RC10300; H , F, Cl, Cl, CF ₂ H, CF ₃ ], [RC10301; H, F, Cl, Cl, CF ₂ H, CF ₃ CH ₂ ], [RC10302; H, F, Cl, Cl, CF ₂ H , CF ₃ CF ₂ ], [RC10303; H, F, Cl, Cl, CF ₂ H, CF ₂ H], [RC10304; H, F, Cl, Cl, CF ₂ H, CF ₂ HCF ₂ ], [RC10305 ; H, F, H, H, CF ₃ , Me], [RC10306; H, F, H, H, CF ₃ , Et], [RC10307; H, F, H, H, CF ₃ , Pr], [ RC10308; H, F, H, H, CF ₃ , i-Pr], [RC10309; H, F, H, H, CF ₃ , c-Pr], [RC10310; H, F, H, H, CF ₃ , Bu], [RC10311; H, F, H, H, CF ₃ , i-Bu], [RC10312; H, F, H, H, CF ₃ , t-Bu], [RC10313; H, F, H , H, CF ₃ , c-PrCH ₂ ], [RC10314; H, F, H, H, CF ₃ , Ph], [RC10315; H, F, H, H, CF ₃ , Bn], [RC10316; H , F, H, H, CF ₃ , CF ₃ ], [RC10317; H, F, H, H, CF ₃ , CF ₃ CH ₂ ], [RC10318; H, F, H, H, CF ₃ , CF ₃ CF ₂ ], [RC10319; H, F, H, H, CF ₃ , CF ₂ H], [RC10320; H, F, H, H, CF ₃ , CF ₂ HCF ₂ ], [RC10321; H, F, H, Me, CF ₃ , Me], [RC10322; H, F, H, Me, CF ₃ , Et], [RC10323; H, F, H, Me, CF ₃ , Pr], [RC10324; H, F , H, Me, CF ₃ , i-Pr], [RC10325; H, F, H, Me, CF ₃ , c-Pr], [RC10326; H, F, H, Me, CF ₃ , Bu], [ RC10327; H, F , H, Me, CF ₃ , i-Bu], [RC10328; H, F, H, Me, CF ₃ , t-Bu], [RC10329; H, F, H, Me, CF ₃ , c-PrCH ₂ ], [RC10330; H, F, H, Me, CF ₃ , Ph], [RC10331; H, F, H, Me, CF ₃ , Bn], [RC10332; H, F, H, Me, CF ₃ , CF ₃ ], [RC10333; H, F, H, Me, CF ₃ , CF ₃ CH ₂ ], [RC10334; H, F, H, Me, CF ₃ , CF ₃ CF ₂ ], [RC10335; H, F , H, Me, CF ₃ , CF ₂ H], [RC10336; H, F, H, Me, CF ₃ , CF ₂ HCF ₂ ], [RC10337; H, F, Me, Me, CF ₃ , Me], [RC10338; H, F, Me, Me, CF ₃ , Et], [RC10339; H, F, Me, Me, CF ₃ , Pr], [RC10340; H, F, Me, Me, CF ₃ , i- Pr], [RC10341; H, F, Me, Me, CF ₃ , c-Pr], [RC10342; H, F, Me, Me, CF ₃ , Bu], [RC10343; H, F, Me, Me, CF ₃ , i-Bu], [RC10344; H, F, Me, Me, CF ₃ , t-Bu], [RC10345; H, F, Me, Me, CF ₃ , c-PrCH ₂ ], [RC10346; H, F, Me, Me, CF ₃ , Ph], [RC10347; H, F, Me, Me, CF ₃ , Bn], [RC10348; H, F, Me, Me, CF ₃ , CF ₃ ], [ RC10349; H, F, Me, Me, CF ₃ , CF ₃ CH ₂ ], [RC10350; H, F, Me, Me, CF ₃ , CF ₃ CF ₂ ], [RC10351; H, F, Me, Me, CF ₃ , CF ₂ H], [RC10352; H, F, Me, Me, CF ₃ , CF ₂ HCF ₂ ], [RC10353; H, F, Me, Et, CF ₃ , Me], [RC10354; H, F, Me, Et, CF ₃ , Et], [RC10355; H, F, Me, Et, CF ₃ , Pr], [RC10356; H, F, Me, Et, CF ₃ , i-Pr], [RC10357 ; H, F, Me, Et, CF ₃ , c-Pr], [RC10358; H, F, Me, Et, CF ₃ , Bu], [RC10359; H, F, Me, Et, CF ₃ , i-Bu], [RC10360; H, F, Me, Et, CF ₃ , t-Bu], [RC10361; H, F, Me, Et, CF ₃ , c-PrCH ₂ ], [RC10362; H, F, Me, Et, CF ₃ , Ph], [RC10363; H, F, Me, Et, CF ₃ , Bn], [RC10364; H, F, Me , Et, CF ₃ , CF ₃ ], [RC10365; H, F, Me, Et, CF ₃ , CF ₃ CH ₂ ], [RC10366; H, F, Me, Et, CF ₃ , CF ₃ CF ₂ ], [RC10367; H, F, Me, Et, CF ₃ , CF ₂ H], [RC10368; H, F, Me, Et, CF ₃ , CF ₂ HCF ₂ ], [RC10369; H, F, Me, F, CF ₃ , Me], [RC10370; H, F, Me, F, CF ₃ , Et], [RC10371; H, F, Me, F, CF ₃ , Pr], [RC10372; H, F, Me, F , CF ₃ , i-Pr], [RC10373; H, F, Me, F, CF ₃ , c-Pr], [RC10374; H, F, Me, F, CF ₃ , Bu], [RC10375; H, F, Me, F, CF ₃ , i-Bu], [RC10376; H, F, Me, F, CF ₃ , t-Bu], [RC10377; H, F, Me, F, CF ₃ , c-PrCH ₂ ], [RC10378; H, F, Me, F, CF ₃ , Ph], [RC10379; H, F, Me, F, CF ₃ , Bn], [RC10380; H, F, Me, F, CF ₃ , CF ₃ ], [RC10381; H, F, Me, F, CF ₃ , CF ₃ CH ₂ ], [RC10382; H, F, Me, F, CF ₃ , CF ₃ CF ₂ ], [RC10383; H, F, Me, F, CF ₃ , CF ₂ H], [RC10384; H, F, Me, F, CF ₃ , CF ₂ HCF ₂ ], [RC10385; H, F, Me, Cl, CF ₃ , Me] , [RC10386; H, F, Me, Cl, CF ₃ , Et], [RC10387; H, F, Me, Cl, CF ₃ , Pr], [RC10388; H, F, Me, Cl, CF ₃ , i -Pr], [RC10389; H, F, Me, Cl, CF ₃ , c-Pr], [RC10390; H, F, Me, Cl, CF ₃ , Bu], [RC10391; H, F, Me, Cl, CF ₃ , i-Bu], [RC10392; H, F, Me, Cl, CF ₃ , t-Bu], [RC10393; H, F, Me , Cl, CF ₃ , c-PrCH ₂ ], [RC10394; H, F, Me, Cl, CF ₃ , Ph], [RC10395; H, F, Me, Cl, CF ₃ , Bn], [RC10396; H , F, Me, Cl, CF ₃ , CF ₃ ], [RC10397; H, F, Me, Cl, CF ₃ , CF ₃ CH ₂ ], [RC10398; H, F, Me, Cl, CF ₃ , CF ₃ CF ₂ ], [RC10399; H, F, Me, Cl, CF ₃ , CF ₂ H], [RC10400; H, F, Me, Cl, CF ₃ , CF ₂ HCF ₂ ],

[RC10401; H, F, Et, H, CF ₃ , Me], [RC10402; H, F, Et, H, CF ₃ , Et], [RC10403; H, F, Et, H, CF ₃ , Pr] , [RC10404; H, F, Et, H, CF ₃ , i-Pr], [RC10405; H, F, Et, H, CF ₃ , c-Pr], [RC10406; H, F, Et, H, CF ₃ , Bu], [RC10407; H, F, Et, H, CF ₃ , i-Bu], [RC10408; H, F, Et, H, CF ₃ , t-Bu], [RC10409; H, F , Et, H, CF ₃ , c-PrCH ₂ ], [RC10410; H, F, Et, H, CF ₃ , Ph], [RC10411; H, F, Et, H, CF ₃ , Bn], [RC10412 ; H, F, Et, H, CF ₃ , CF ₃ ], [RC10413; H, F, Et, H, CF ₃ , CF ₃ CH ₂ ], [RC10414; H, F, Et, H, CF ₃ , CF ₃ CF ₂ ], [RC10415; H, F, Et, H, CF ₃ , CF ₂ H], [RC10416; H, F, Et, H, CF ₃ , CF ₂ HCF ₂ ], [RC10417; H, F, Et, F, CF ₃ , Me], [RC10418; H, F, Et, F, CF ₃ , Et], [RC10419; H, F, Et, F, CF ₃ , Pr], [RC10420; H , F, Et, F, CF ₃ , i-Pr], [RC10421; H, F, Et, F, CF ₃ , c-Pr], [RC10422; H, F, Et, F, CF ₃ , Bu] , [RC10423; H, F, Et, F, CF ₃ , i-Bu], [RC10424; H, F, Et, F, CF ₃ , t-Bu], [RC10425; H, F, Et, F, CF ₃ , c-PrCH ₂ ], [RC10426; H, F, Et, F, CF ₃ , Ph], [RC10427; H, F, Et, F, CF ₃ , Bn], [RC10428; H, F, Et, F, CF ₃ , CF ₃ ], [RC10429; H, F, Et, F, CF ₃ , CF ₃ CH ₂ ], [RC10430; H, F, Et, F, CF ₃ , CF ₃ CF ₂ ] , [RC10431; H, F, Et, F, CF ₃ , CF ₂ H], [RC10432; H, F, Et, F, CF ₃ , CF ₂ HCF ₂ ], [RC10433; H , F, Et, Cl, CF ₃ , Me], [RC10434; H, F, Et, Cl, CF ₃ , Et], [RC10435; H, F, Et, Cl, CF ₃ , Pr], [RC10436; H, F, Et, Cl, CF ₃ , i-Pr], [RC10437; H, F, Et, Cl, CF ₃ , c-Pr], [RC10438; H, F, Et, Cl, CF ₃ , Bu ], [RC10439; H, F, Et, Cl, CF ₃ , i-Bu], [RC10440; H, F, Et, Cl, CF ₃ , t-Bu], [RC10441; H, F, Et, Cl , CF ₃ , c-PrCH ₂ ], [RC10442; H, F, Et, Cl, CF ₃ , Ph], [RC10443; H, F, Et, Cl, CF ₃ , Bn], [RC10444; H, F , Et, Cl, CF ₃ , CF ₃ ], [RC10445; H, F, Et, Cl, CF ₃ , CF ₃ CH ₂ ], [RC10446; H, F, Et, Cl, CF ₃ , CF ₃ CF ₂ ], [RC10447; H, F, Et, Cl, CF ₃ , CF ₂ H], [RC10448; H, F, Et, Cl, CF ₃ , CF ₂ HCF ₂ ], [RC10449; H, F, F, H, CF ₃ , Me], [RC10450; H, F, F, H, CF ₃ , Et], [RC10451; H, F, F, H, CF ₃ , Pr], [RC10452; H, F, F , H, CF ₃ , i-Pr], [RC10453; H, F, F, H, CF ₃ , c-Pr], [RC10454; H, F, F, H, CF ₃ , Bu], [RC10455; H, F, F, H, CF ₃ , i-Bu], [RC10456; H, F, F, H, CF ₃ , t-Bu], [RC10457; H, F, F, H, CF ₃ , c -PrCH ₂ ], [RC10458; H, F, F, H, CF ₃ , Ph], [RC10459; H, F, F, H, CF ₃ , Bn], [RC10460; H, F, F, H, CF ₃ , CF ₃ ], [RC10461; H, F, F, H, CF ₃ , CF ₃ CH ₂ ], [RC10462; H, F, F, H, CF ₃ , CF ₃ CF ₂ ], [RC10463; H, F, F, H, CF ₃ , CF ₂ H], [RC10464; H, F, F, H, CF ₃ , CF ₂ HCF ₂ ], [RC10465; H, F, F, F, CF ₃ , Me], [RC10466; H, F, F, F, CF ₃ , Et], [RC10467; H, F, F, F, CF ₃ , Pr], [RC10468; H, F, F, F, CF ₃ , i-Pr], [RC10469; H, F, F, F, CF ₃ , c-Pr], [RC10470; H, F, F, F, CF ₃ , Bu], [RC10471; H, F , F, F, CF ₃ , i-Bu], [RC10472; H, F, F, F, CF ₃ , t-Bu], [RC10473; H, F, F, F, CF ₃ , c-PrCH ₂ ], [RC10474; H, F, F, F, CF ₃ , Ph], [RC10475; H, F, F, F, CF ₃ , Bn], [RC10476; H, F, F, F, CF ₃ , CF ₃ ], [RC10477; H, F, F, F, CF ₃ , CF ₃ CH ₂ ], [RC10478; H, F, F, F, CF ₃ , CF ₃ CF ₂ ], [RC10479; H, F , F, F, CF ₃ , CF ₂ H], [RC10480; H, F, F, F, CF ₃ , CF ₂ HCF ₂ ], [RC10481; H, F, F, Cl, CF ₃ , Me], [RC10482; H, F, F, Cl, CF ₃ , Et], [RC10483; H, F, F, Cl, CF ₃ , Pr], [RC10484; H, F, F, Cl, CF ₃ , i- Pr], [RC10485; H, F, F, Cl, CF ₃ , c-Pr], [RC10486; H, F, F, Cl, CF ₃ , Bu], [RC10487; H, F, F, Cl, CF ₃ , i-Bu], [RC10488; H, F, F, Cl, CF ₃ , t-Bu], [RC10489; H, F, F, Cl, CF ₃ , c-PrCH ₂ ], [RC10490; H, F, F, Cl, CF ₃ , Ph], [RC10491; H, F, F, Cl, CF ₃ , Bn], [RC10492; H, F, F, Cl, CF ₃ , CF ₃ ], [ RC10493; H, F, F, Cl, CF ₃ , CF ₃ CH ₂ ], [RC10494; H, F, F, Cl, CF ₃ , CF ₃ CF ₂ ], [RC10495; H, F, F, Cl, CF ₃ , CF ₂ H], [RC10496; H, F, F, Cl, CF ₃ , CF ₂ HCF ₂ ], [RC10497; H, F, Cl, H, CF ₃ , Me], [RC10498; H, F, Cl, H, CF ₃ , Et], [RC10499; H, F, Cl, H, CF ₃ , Pr], [RC10500; H, F, Cl, H, CF ₃ , i-Pr], [RC10501; H, F, Cl , H, CF ₃ , c-Pr], [RC10502; H, F, Cl, H, CF ₃ , Bu], [RC10503; H, F, Cl, H, CF ₃ , i-Bu], [RC10504; H, F, Cl, H, CF ₃ , t-Bu], [RC10505; H, F, Cl, H, CF ₃ , c-PrCH ₂ ], [RC10506; H, F, Cl, H, CF ₃ , Ph], [RC10507; H, F, Cl, H, CF ₃ , Bn], [RC10508; H, F, Cl, H, CF ₃ , CF ₃ ], [RC10509; H, F, Cl, H, CF ₃ , CF ₃ CH ₂ ], [RC10510; H, F, Cl, H, CF ₃ , CF ₃ CF ₂ ], [RC10511; H, F, Cl, H, CF ₃ , CF ₂ H], [RC10512; H, F, Cl, H, CF ₃ , CF ₂ HCF ₂ ], [RC10513; H, F, Cl, Cl, CF ₃ , Me], [RC10514; H, F, Cl, Cl, CF ₃ , Et] , [RC10515; H, F, Cl, Cl, CF ₃ , Pr], [RC10516; H, F, Cl, Cl, CF ₃ , i-Pr], [RC10517; H, F, Cl, Cl, CF ₃ , c-Pr], [RC10518; H, F, Cl, Cl, CF ₃ , Bu], [RC10519; H, F, Cl, Cl, CF ₃ , i-Bu], [RC10520; H, F, Cl , Cl, CF ₃ , t-Bu], [RC10521; H, F, Cl, Cl, CF ₃ , c-PrCH ₂ ], [RC10522; H, F, Cl, Cl, CF ₃ , Ph], [RC10523 ; H, F, Cl, Cl, CF ₃ , Bn], [RC10524; H, F, Cl, Cl, CF ₃ , CF ₃ ], [RC10525; H, F, Cl, Cl, CF ₃ , CF ₃ CH ₂ ], [RC10526; H, F, Cl, Cl, CF ₃ , CF ₃ CF ₂ ], [RC10527; H, F, Cl, Cl, CF ₃ , CF ₂ H], [RC10528; H, F, Cl , Cl, CF ₃ , CF ₂ HCF ₂ ], [RC10529; H, F, H, H, CF ₂ HCH ₂ , Me], [RC1053 0; H, F, H, H, CF ₂ HCH ₂ , Et], [RC10531; H, F, H, H, CF ₂ HCH ₂ , Pr], [RC10532; H, F, H, H, CF ₂ HCH ₂ , i-Pr], [RC10533; H, F, H, H, CF ₂ HCH ₂ , c-Pr], [RC10534; H, F, H, H, CF ₂ HCH ₂ , Bu], [RC10535 ; H, F, H, H, CF ₂ HCH ₂ , i-Bu], [RC10536; H, F, H, H, CF ₂ HCH ₂ , t-Bu], [RC10537; H, F, H, H , CF ₂ HCH ₂ , c-PrCH ₂ ], [RC10538; H, F, H, H, CF ₂ HCH ₂ , Ph], [RC10539; H, F, H, H, CF ₂ HCH ₂ , Bn], [RC10540; H, F, H, H, CF ₂ HCH ₂ , CF ₃ ], [RC10541; H, F, H, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC10542; H, F, H , H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC10543; H, F, H, H, CF ₂ HCH ₂ , CF ₂ H], [RC10544; H, F, H, H, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC10545; H, F, H, Me, CF ₂ HCH ₂ , Me], [RC10546; H, F, H, Me, CF ₂ HCH ₂ , Et], [RC10547; H, F, H, Me, CF ₂ HCH ₂ , Pr], [RC10548; H, F, H, Me, CF ₂ HCH ₂ , i-Pr], [RC10549; H, F, H, Me, CF ₂ HCH ₂ , c-Pr], [RC10550; H, F, H, Me, CF ₂ HCH ₂ , Bu], [RC10551; H, F, H, Me, CF ₂ HCH ₂ , i-Bu], [RC10552; H , F, H, Me, CF ₂ HCH ₂ , t-Bu], [RC10553; H, F, H, Me, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC10554; H, F, H, Me, CF ₂ HCH ₂ , Ph], [RC10555; H, F, H, Me, CF ₂ HCH ₂ , Bn], [RC10556; H, F, H, Me, CF ₂ HCH ₂ , CF ₃ ], [RC10557; H, F, H, Me, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC10558; H, F, H, Me, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC10559; H, F, H, Me, CF ₂ HCH ₂ , CF ₂ H], [RC10560; H, F, H, Me, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC10561; H, F, Me, Me, CF ₂ HCH ₂ , Me], [RC10562; H, F, Me, Me, CF ₂ HCH ₂ , Et], [RC10563; H, F, Me, Me, CF ₂ HCH ₂ , Pr], [RC10564; H, F, Me, Me, CF ₂ HCH ₂ , i-Pr], [RC10565; H, F, Me, Me, CF ₂ HCH ₂ , c-Pr], [RC10566; H, F, Me, Me, CF ₂ HCH ₂ , Bu], [RC10567; H, F, Me, Me, CF ₂ HCH ₂ , i-Bu], [RC10568; H, F, Me, Me, CF ₂ HCH ₂ , t-Bu], [RC10569; H, F, Me, Me, CF ₂ HCH ₂ , c-PrCH ₂ ], [ RC10570; H, F, Me, Me, CF ₂ HCH ₂ , Ph], [RC10571; H, F, Me, Me, CF ₂ HCH ₂ , Bn], [RC10572; H, F, Me, Me, CF ₂ HCH ₂ , CF ₃ ], [RC10573; H, F, Me, Me, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC10574; H, F, Me, Me, CF ₂ HCH ₂ , CF ₃ CF ₂ ] , [RC10575; H, F, Me, Me, CF ₂ HCH ₂ , CF ₂ H], [RC10576; H, F, Me, Me, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC10577; H, F , Me, Et, CF ₂ HCH ₂ , Me], [RC10578; H, F, Me, Et, CF ₂ HCH ₂ , Et], [RC10579; H, F, Me, Et, CF ₂ HCH ₂ , Pr] , [RC10580; H, F, Me, Et, CF ₂ HCH ₂ , i-Pr], [RC10581; H, F, Me, Et, CF ₂ HCH ₂ , c-Pr], [RC10582; H, F, Me, Et, CF ₂ HCH ₂ , Bu], [RC10583; H, F, Me, Et, CF ₂ HCH ₂ , i-Bu], [RC10584; H, F, Me, Et, CF ₂ HCH ₂ , t-Bu], [RC10585; H, F, Me, Et, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC10586; H, F, Me, Et, CF ₂ HCH ₂ , Ph], [RC10587; H, F, Me, Et, CF ₂ HCH ₂ , Bn], [RC10588; H, F, Me, Et, CF ₂ HCH ₂ , CF ₃ ], [RC10589; H, F, Me , Et, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC10590; H, F, Me, Et, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC10591; H, F, Me, Et, CF ₂ HCH ₂ , CF ₂ H], [RC10592; H, F, Me, Et, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC10593; H, F, Me, F, CF ₂ HCH ₂ , Me], [RC10594 ; H, F, Me, F, CF ₂ HCH ₂ , Et], [RC10595; H, F, Me, F, CF ₂ HCH ₂ , Pr], [RC10596; H, F, Me, F, CF ₂ HCH ₂ , i-Pr], [RC10597; H, F, Me, F, CF ₂ HCH ₂ , c-Pr], [RC10598; H, F, Me, F, CF ₂ HCH ₂ , Bu], [RC10599; H, F, Me, F, CF ₂ HCH ₂ , i-Bu], [RC10600; H, F, Me, F, CF ₂ HCH ₂ , t-Bu],

[RC10601; H, F, Me, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC10602; H, F, Me, F, CF ₂ HCH ₂ , Ph], [RC10603; H, F, Me, F, CF ₂ HCH ₂ , Bn], [RC10604; H, F, Me, F, CF ₂ HCH ₂ , CF ₃ ], [RC10605; H, F, Me, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC10606; H, F, Me, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC10607; H, F, Me, F, CF ₂ HCH ₂ , CF ₂ H], [RC10608; H, F, Me, F, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC10609; H, F, Me, Cl, CF ₂ HCH ₂ , Me], [RC10610; H, F, Me, Cl, CF ₂ HCH ₂ , Et], [RC10611; H, F, Me, Cl, CF ₂ HCH ₂ , Pr], [RC10612; H, F, Me, Cl, CF ₂ HCH ₂ , i-Pr], [RC10613; H, F, Me, Cl, CF ₂ HCH ₂ , c-Pr], [RC10614; H, F, Me, Cl, CF ₂ HCH ₂ , Bu], [RC10615; H, F, Me, Cl, CF ₂ HCH ₂ , i-Bu], [RC10616; H, F, Me, Cl, CF ₂ HCH ₂ , t-Bu], [RC10617; H, F, Me, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [ RC10618; H, F, Me, Cl, CF ₂ HCH ₂ , Ph], [RC10619; H, F, Me, Cl, CF ₂ HCH ₂ , Bn], [RC10620; H, F, Me, Cl, CF ₂ HCH ₂ , CF ₃ ], [RC10621; H, F, Me, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC10622; H, F, Me, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ] , [RC10623; H, F, Me, Cl, CF ₂ HCH ₂ , CF ₂ H], [RC10624; H, F, Me, Cl, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC10625; H, F , Et, H, CF ₂ HCH ₂ , Me], [RC10626; H, F, Et, H, CF ₂ HCH ₂ , Et], [RC10627; H, F, E t, H, CF ₂ HCH ₂ , Pr], [RC10628; H, F, Et, H, CF ₂ HCH ₂ , i-Pr], [RC10629; H, F, Et, H, CF ₂ HCH ₂ , c -Pr], [RC10630; H, F, Et, H, CF ₂ HCH ₂ , Bu], [RC10631; H, F, Et, H, CF ₂ HCH ₂ , i-Bu], [RC10632; H, F , Et, H, CF ₂ HCH ₂ , t-Bu], [RC10633; H, F, Et, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC10634; H, F, Et, H, CF _{2 HCH 2, Ph], [RC10635} ; H, F, Et, H, CF 2 HCH 2, Bn], [RC10636; H, F, Et, H, CF 2 HCH 2, CF 3], [RC10637; H, F, Et, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC10638; H, F, Et, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC10639; H, F, Et, H, CF ₂ HCH ₂ , CF ₂ H], [RC10640; H, F, Et, H, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC10641; H, F, Et, F, CF ₂ HCH ₂ , Me] , [RC10642; H, F, Et, F, CF ₂ HCH ₂ , Et], [RC10643; H, F, Et, F, CF ₂ HCH ₂ , Pr], [RC10644; H, F, Et, F, CF ₂ HCH ₂ , i-Pr], [RC10645; H, F, Et, F, CF ₂ HCH ₂ , c-Pr], [RC10646; H, F, Et, F, CF ₂ HCH ₂ , Bu], [RC10647; H, F, Et, F, CF ₂ HCH ₂ , i-Bu], [RC10648; H, F, Et, F, CF ₂ HCH ₂ , t-Bu], [RC10649; H, F, Et , F, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC10650; H, F, Et, F, CF ₂ HCH ₂ , Ph], [RC10651; H, F, Et, F, CF ₂ HCH ₂ , Bn ], [RC10652; H, F, Et, F, CF ₂ HCH ₂ , CF ₃ ], [RC10653; H, F, Et, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC10654; H, F , Et, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC10655; H, F, Et, F, CF ₂ HCH ₂ , CF ₂ H], [RC10656; H, F, Et, F, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC10657; H, F, Et, Cl, CF ₂ HCH ₂ , Me], [RC10658; H, F, Et, Cl, CF ₂ HCH ₂ , Et], [RC10659; H, F, Et, Cl , CF ₂ HCH ₂ , Pr], [RC10660; H, F, Et, Cl, CF ₂ HCH ₂ , i-Pr], [RC10661; H, F, Et, Cl, CF ₂ HCH ₂ , c-Pr] , [RC10662; H, F, Et, Cl, CF ₂ HCH ₂ , Bu], [RC10663; H, F, Et, Cl, CF ₂ HCH ₂ , i-Bu], [RC10664; H, F, Et, Cl, CF ₂ HCH ₂ , t-Bu], [RC10665; H, F, Et, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC10666; H, F, Et, Cl, CF ₂ HCH ₂ , Ph], [RC10667; H, F, Et, Cl, CF ₂ HCH ₂ , Bn], [RC10668; H, F, Et, Cl, CF ₂ HCH ₂ , CF ₃ ], [RC10669; H, F, Et , Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC10670; H, F, Et, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC10671; H, F, Et, Cl, CF ₂ HCH ₂ , CF ₂ H], [RC10672; H, F, Et, Cl, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC10673; H, F, F, H, CF ₂ HCH ₂ , Me], [RC10674 ; H, F, F, H, CF ₂ HCH ₂ , Et], [RC10675; H, F, F, H, CF ₂ HCH ₂ , Pr], [RC10676; H, F, F, H, CF ₂ HCH ₂ , i-Pr], [RC10677; H, F, F, H, CF ₂ HCH ₂ , c-Pr], [RC10678; H, F, F, H, CF ₂ HCH ₂ , Bu], [RC10679; H, F, F, H, CF ₂ HCH ₂ , i-Bu], [RC10680; H, F, F, H, CF ₂ HCH ₂ , t-Bu], [RC10681; H, F, F, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC10682; H, F, F, H, CF ₂ HCH ₂ , Ph], [RC10683; H, F, F, H, CF ₂ HCH ₂ , Bn], [RC10684; H, F, F, H, CF ₂ HCH ₂ , CF ₃ ], [RC10685; H, F, F, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC10686; H, F, F, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC10687; H, F, F, H, CF ₂ HCH ₂ , CF ₂ H], [RC10688; H, F, F, H, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC10689; H, F, F, F, CF ₂ HCH ₂ , Me], [RC10690; H, F, F, F, CF ₂ HCH ₂ , Et], [RC10691; H, F, F , F, CF ₂ HCH ₂ , Pr], [RC10692; H, F, F, F, CF ₂ HCH ₂ , i-Pr], [RC10693; H, F, F, F, CF ₂ HCH ₂ , c- Pr], [RC10694; H, F, F, F, CF ₂ HCH ₂ , Bu], [RC10695; H, F, F, F, CF ₂ HCH ₂ , i-Bu], [RC10696; H, F, F, F, CF ₂ HCH ₂ , t-Bu], [RC10697; H, F, F, F, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC10698; H, F, F, F, CF ₂ HCH ₂ , Ph], [RC10699; H, F, F, F, CF ₂ HCH ₂ , Bn], [RC10700; H, F, F, F, CF ₂ HCH ₂ , CF ₃ ], [RC10701; H, F , F, F, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC10702; H, F, F, F, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC10703; H, F, F, F, CF ₂ HCH ₂ , CF ₂ H], [RC10704; H, F, F, F, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC10705; H, F, F, Cl, CF ₂ HCH ₂ , Me], [RC10706; H, F, F, Cl, CF ₂ HCH ₂ , Et], [RC10707; H, F, F, Cl, CF ₂ HCH ₂ , Pr], [RC10708; H, F, F, Cl, CF ₂ HCH ₂ , i-Pr], [RC10 709; H, F, F, Cl, CF ₂ HCH ₂ , c-Pr], [RC10710; H, F, F, Cl, CF ₂ HCH ₂ , Bu], [RC10711; H, F, F, Cl, CF ₂ HCH ₂ , i-Bu], [RC10712; H, F, F, Cl, CF ₂ HCH ₂ , t-Bu], [RC10713; H, F, F, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC10714; H, F, F, Cl, CF ₂ HCH ₂ , Ph], [RC10715; H, F, F, Cl, CF ₂ HCH ₂ , Bn], [RC10716; H, F, F, Cl, CF ₂ HCH ₂ , CF ₃ ], [RC10717; H, F, F, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC10718; H, F, F, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC10719; H, F, F, Cl, CF ₂ HCH ₂ , CF ₂ H], [RC10720; H, F, F, Cl, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC10721 ; H, F, Cl, H, CF ₂ HCH ₂ , Me], [RC10722; H, F, Cl, H, CF ₂ HCH ₂ , Et], [RC10723; H, F, Cl, H, CF ₂ HCH ₂ , Pr], [RC10724; H, F, Cl, H, CF ₂ HCH ₂ , i-Pr], [RC10725; H, F, Cl, H, CF ₂ HCH ₂ , c-Pr], [RC10726; H, F, Cl, H, CF ₂ HCH ₂ , Bu], [RC10727; H, F, Cl, H, CF ₂ HCH ₂ , i-Bu], [RC10728; H, F, Cl, H, CF ₂ HCH ₂ , t-Bu], [RC10729; H, F, Cl, H, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC10730; H, F, Cl, H, CF ₂ HCH ₂ , Ph], [ RC10731; H, F, Cl, H, CF ₂ HCH ₂ , Bn], [RC10732; H, F, Cl, H, CF ₂ HCH ₂ , CF ₃ ], [RC10733; H, F, Cl, H, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC10734; H, F, Cl, H, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC10735; H, F, Cl, H, CF ₂ HCH ₂ , CF ₂ H], [RC1 0736; H, F, Cl, H, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC10737; H, F, Cl, Cl, CF ₂ HCH ₂ , Me], [RC10738; H, F, Cl, Cl , CF ₂ HCH ₂ , Et], [RC10739; H, F, Cl, Cl, CF ₂ HCH ₂ , Pr], [RC10740; H, F, Cl, Cl, CF ₂ HCH ₂ , i-Pr], [ RC10741; H, F, Cl, Cl, CF ₂ HCH ₂ , c-Pr], [RC10742; H, F, Cl, Cl, CF ₂ HCH ₂ , Bu], [RC10743; H, F, Cl, Cl, CF ₂ HCH ₂ , i-Bu], [RC10744; H, F, Cl, Cl, CF ₂ HCH ₂ , t-Bu], [RC10745; H, F, Cl, Cl, CF ₂ HCH ₂ , c-PrCH ₂ ], [RC10746; H, F, Cl, Cl, CF ₂ HCH ₂ , Ph], [RC10747; H, F, Cl, Cl, CF ₂ HCH ₂ , Bn], [RC10748; H, F, Cl, Cl, CF ₂ HCH ₂ , CF ₃ ], [RC10749; H, F, Cl, Cl, CF ₂ HCH ₂ , CF ₃ CH ₂ ], [RC10750; H, F, Cl, Cl, CF ₂ HCH ₂ , CF ₃ CF ₂ ], [RC10751; H, F, Cl, Cl, CF ₂ HCH ₂ , CF ₂ H], [RC10752; H, F, Cl, Cl, CF ₂ HCH ₂ , CF ₂ HCF ₂ ], [RC10753 ; H, F, H, H, CF ₃ CH ₂ , Me], [RC10754; H, F, H, H, CF ₃ CH ₂ , Et], [RC10755; H, F, H, H, CF ₃ CH ₂ , Pr], [RC10756; H, F, H, H, CF ₃ CH ₂ , i-Pr], [RC10757; H, F, H, H, CF ₃ CH ₂ , c-Pr], [RC10758; H, F, H, H, CF ₃ CH ₂ , Bu], [RC10759; H, F, H, H, CF ₃ CH ₂ , i-Bu], [RC10760; H, F, H, H, CF ₃ CH ₂ , t-Bu], [RC10761; H, F, H, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RC10762; H, F, H, H, CF ₃ CH ₂ , Ph], [ RC10763; H, F, H, H, CF ₃ CH ₂ , Bn], [RC10764; H, F, H, H, CF ₃ CH ₂ , CF ₃ ], [RC10765; H, F, H, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [ RC10766; H, F, H, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC10767; H, F, H, H, CF ₃ CH ₂ , CF ₂ H], [RC10768; H, F, H , H, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC10769; H, F, H, Me, CF ₃ CH ₂ , Me], [RC10770; H, F, H, Me, CF ₃ CH ₂ , Et ], [RC10771; H, F, H, Me, C
F ₃ CH ₂ , Pr], [RC10772; H, F, H, Me, CF ₃ CH ₂ , i-Pr], [RC10773; H, F, H, Me, CF ₃ CH ₂ , c-Pr], [RC10774; H, F, H, Me, CF ₃ CH ₂ , Bu], [RC10775; H, F, H, Me, CF ₃ CH ₂ , i-Bu], [RC10776; H, F, H, Me , CF ₃ CH ₂ , t-Bu], [RC10777; H, F, H, Me, CF ₃ CH ₂ , c-PrCH ₂ ], [RC10778; H, F, H, Me, CF ₃ CH ₂ , Ph ], [RC10779; H, F, H, Me, CF ₃ CH ₂ , Bn], [RC10780; H, F, H, Me, CF ₃ CH ₂ , CF ₃ ], [RC10781; H, F, H, Me, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC10782; H, F, H, Me, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC10783; H, F, H, Me, CF ₃ CH ₂ , CF ₂ H], [RC10784; H, F, H, Me, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC10785; H, F, Me, Me, CF ₃ CH ₂ , Me], [RC10786; H, F, Me, Me, CF ₃ CH ₂ , Et], [RC10787; H, F, Me, Me, CF ₃ CH ₂ , Pr], [RC10788; H, F, Me, Me, CF ₃ CH ₂ , i-Pr], [RC10789; H, F, Me, Me, CF ₃ CH ₂ , c-Pr], [RC10790; H, F, Me, Me, CF ₃ CH ₂ , Bu], [RC10791; H , F, Me, Me, CF ₃ CH ₂ , i-Bu], [RC10792; H, F, Me, Me, CF ₃ CH ₂ , t-Bu], [RC10793; H, F, Me, Me, CF ₃ CH ₂ , c-PrCH ₂ ], [RC10794; H, F, Me, Me, CF ₃ CH ₂ , Ph], [RC10795; H, F, Me, Me, CF ₃ CH ₂ , Bn], [RC10796 ; H, F, Me, Me, CF ₃ CH ₂ , CF ₃ ], [RC10797; H, F, Me, Me, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC10798; H, F, Me, Me , CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC10799; H, F, Me, Me, CF ₃ CH ₂ , CF ₂ H], [RC10800; H, F, Me, Me, CF ₃ CH ₂ , CF ₂ HCF ₂ ],

[RC10801; H, F, Me, Et, CF ₃ CH ₂ , Me], [RC10802; H, F, Me, Et, CF ₃ CH ₂ , Et], [RC10803; H, F, Me, Et, CF ₃ CH ₂ , Pr], [RC10804; H, F, Me, Et, CF ₃ CH ₂ , i-Pr], [RC10805; H, F, Me, Et, CF ₃ CH ₂ , c-Pr], [ RC10806; H, F, Me, Et, CF ₃ CH ₂ , Bu], [RC10807; H, F, Me, Et, CF ₃ CH ₂ , i-Bu], [RC10808; H, F, Me, Et, CF ₃ CH ₂ , t-Bu], [RC10809; H, F, Me, Et, CF ₃ CH ₂ , c-PrCH ₂ ], [RC10810; H, F, Me, Et, CF ₃ CH ₂ , Ph] , [RC10811; H, F, Me, Et, CF ₃ CH ₂ , Bn], [RC10812; H, F, Me, Et, CF ₃ CH ₂ , CF ₃ ], [RC10813; H, F, Me, Et , CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC10814; H, F, Me, Et, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC10815; H, F, Me, Et, CF ₃ CH ₂ , CF ₂ H], [RC10816; H, F, Me, Et, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC10817; H, F, Me, F, CF ₃ CH ₂ , Me], [RC10818; H , F, Me, F, CF ₃ CH ₂ , Et], [RC10819; H, F, Me, F, CF ₃ CH ₂ , Pr], [RC10820; H, F, Me, F, CF ₃ CH ₂ , i-Pr], [RC10821; H, F, Me, F, CF ₃ CH ₂ , c-Pr], [RC10822; H, F, Me, F, CF ₃ CH ₂ , Bu], [RC10823; H, F, Me, F, CF ₃ CH ₂ , i-Bu], [RC10824; H, F, Me, F, CF ₃ CH ₂ , t-Bu], [RC10825; H, F, Me, F, CF _{3 CH 2, c-PrCH 2]} , [RC10826; H, F, Me, F, CF 3 CH 2, Ph], [RC10827; H, F, Me, F, CF 3 CH 2, Bn], [RC10828; H, F, Me, F, CF ₃ CH ₂ , CF ₃ ], [RC10829; H, F, Me, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC10830; H, F, Me, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC10831; H, F, Me, F, CF ₃ CH ₂ , CF ₂ H], [RC10832; H, F, Me, F, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC10833; H, F, Me, Cl , CF ₃ CH ₂ , Me], [RC10834; H, F, Me, Cl, CF ₃ CH ₂ , Et], [RC10835; H, F, Me, Cl, CF ₃ CH ₂ , Pr], [RC10836; H, F, Me, Cl, CF ₃ CH ₂ , i-Pr], [RC10837; H, F, Me, Cl, CF ₃ CH ₂ , c-Pr], [RC10838; H, F, Me, Cl, CF ₃ CH ₂ , Bu], [RC10839; H, F, Me, Cl, CF ₃ CH ₂ , i-Bu], [RC10840; H, F, Me, Cl, CF ₃ CH ₂ , t-Bu], [RC10841; H, F, Me, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RC10842; H, F, Me, Cl, CF ₃ CH ₂ , Ph], [RC10843; H, F, Me, Cl, CF ₃ CH ₂ , Bn], [RC10844; H, F, Me, Cl, CF ₃ CH ₂ , CF ₃ ], [RC10845; H, F, Me, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC10846; H, F, Me, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC10847; H, F, Me, Cl, CF ₃ CH ₂ , CF ₂ H], [RC10848; H, F, Me, Cl, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC10849; H, F, Et, H, CF ₃ CH ₂ , Me], [RC10850; H, F, Et, H, CF ₃ CH ₂ , Et], [RC10851; H, F, Et, H, CF ₃ CH ₂ , Pr], [RC10852; H, F, Et, H, CF ₃ CH ₂ , i-Pr], [RC10853; H, F, Et, H, CF ₃ CH ₂ , c-Pr], [RC10854; H, F, Et, H, CF ₃ CH ₂ , Bu], [RC10855; H, F, Et, H, CF ₃ CH ₂ , i-Bu], [RC108 56; H, F, Et, H, CF ₃ CH ₂ , t-Bu], [RC10857; H, F, Et, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RC10858; H, F, Et , H, CF ₃ CH ₂ , Ph], [RC10859; H, F, Et, H, CF ₃ CH ₂ , Bn], [RC10860; H, F, Et, H, CF ₃ CH ₂ , CF ₃ ], [RC10861; H, F, Et, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC10862; H, F, Et, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC10863; H, F , Et, H, CF ₃ CH ₂ , CF ₂ H], [RC10864; H, F, Et, H, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC10865; H, F, Et, F, CF _{3 CH 2, Me], [RC10866} ; H, F, Et, F, CF 3 CH 2, Et], [RC10867; H, F, Et, F, CF 3 CH 2, Pr], [RC10868; H, F , Et, F, CF ₃ CH ₂ , i-Pr], [RC10869; H, F, Et, F, CF ₃ CH ₂ , c-Pr], [RC10870; H, F, Et, F, CF ₃ CH ₂ , Bu], [RC10871; H, F, Et, F, CF ₃ CH ₂ , i-Bu], [RC10872; H, F, Et, F, CF ₃ CH ₂ , t-Bu], [RC10873; H, F, Et, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RC10874; H, F, Et, F, CF ₃ CH ₂ , Ph], [RC10875; H, F, Et, F, CF ₃ CH ₂ , Bn], [RC10876; H, F, Et, F, CF ₃ CH ₂ , CF ₃ ], [RC10877; H, F, Et, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [ RC10878; H, F, Et, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC10879; H, F, Et, F, CF ₃ CH ₂ , CF ₂ H], [RC10880; H, F, Et , F, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC10881; H, F, Et, Cl, CF ₃ CH ₂ , Me], [RC10882; H, F, Et, Cl, CF ₃ CH ₂ , Et ], [RC10883; H, F, Et, Cl, CF ₃ C H ₂ , Pr], [RC10884; H, F, Et, Cl, CF ₃ CH ₂ , i-Pr], [RC10885; H, F, Et, Cl, CF ₃ CH ₂ , c-Pr], [RC10886 ; H, F, Et, Cl, CF ₃ CH ₂ , Bu], [RC10887; H, F, Et, Cl, CF ₃ CH ₂ , i-Bu], [RC10888; H, F, Et, Cl, CF ₃ CH ₂ , t-Bu], [RC10889; H, F, Et, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RC10890; H, F, Et, Cl, CF ₃ CH ₂ , Ph], [RC10891; H, F, Et, Cl, CF ₃ CH ₂ , Bn], [RC10892; H, F, Et, Cl, CF ₃ CH ₂ , CF ₃ ], [RC10893; H, F, Et, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC10894; H, F, Et, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC10895; H, F, Et, Cl, CF ₃ CH ₂ , CF ₂ H], [RC10896; H, F, Et, Cl, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC10897; H, F, F, H, CF ₃ CH ₂ , Me], [RC10898; H, F, F, H, CF ₃ CH ₂ , Et], [RC10899; H, F, F, H, CF ₃ CH ₂ , Pr], [RC10900; H, F, F, H, CF ₃ CH ₂ , i -Pr], [RC10901; H, F, F, H, CF ₃ CH ₂ , c-Pr], [RC10902; H, F, F, H, CF ₃ CH ₂ , Bu], [RC10903; H, F , F, H, CF ₃ CH ₂ , i-Bu], [RC10904; H, F, F, H, CF ₃ CH ₂ , t-Bu], [RC10905; H, F, F, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RC10906; H, F, F, H, CF ₃ CH ₂ , Ph], [RC10907; H, F, F, H, CF ₃ CH ₂ , Bn], [RC10908; H , F, F, H, CF ₃ CH ₂ , CF ₃ ], [RC10909; H, F, F, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC10910; H, F, F, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC10911; H, F, F, H, CF ₃ CH ₂ , CF ₂ H], [RC10912; H, F, F, H, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC10913; H, F, F, F, CF ₃ CH ₂ , Me], [RC10914; H, F, F, F, CF ₃ CH ₂ , Et], [RC10915; H, F, F, F, CF ₃ CH ₂ , Pr], [RC10916; H, F, F, F, CF ₃ CH ₂ , i-Pr], [RC10917; H, F, F, F, CF ₃ CH ₂ , c-Pr], [RC10918; H, F, F, F, CF ₃ CH ₂ , Bu], [ RC10919; H, F, F, F, CF ₃ CH ₂ , i-Bu], [RC10920; H, F, F, F, CF ₃ CH ₂ , t-Bu], [RC10921; H, F, F, F, CF ₃ CH ₂ , c-PrCH ₂ ], [RC10922; H, F, F, F, CF ₃ CH ₂ , Ph], [RC10923; H, F, F, F, CF ₃ CH ₂ , Bn] , [RC10924; H, F, F, F, CF ₃ CH ₂ , CF ₃ ], [RC10925; H, F, F, F, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC10926; H, F, F, F, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC10927; H, F, F, F, CF ₃ CH ₂ , CF ₂ H], [RC10928; H, F, F, F, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC10929; H, F, F, Cl, CF ₃ CH ₂ , Me], [RC10930; H, F, F, Cl, CF ₃ CH ₂ , Et], [RC10931; H , F, F, Cl, CF ₃ CH ₂ , Pr], [RC10932; H, F, F, Cl, CF ₃ CH ₂ , i-Pr], [RC10933; H, F, F, Cl, CF ₃ CH _{2, c-Pr], [} RC10934; H, F, F, Cl, CF 3 CH 2, Bu], [RC10935; H, F, F, Cl, CF 3 CH 2, i-Bu], [RC10936; H, F, F, Cl, CF ₃ CH ₂ , t-Bu], [RC10937; H, F, F, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RC10938; H, F, F, Cl , CF ₃ CH ₂ , Ph], [RC10939; H, F, F, Cl, CF ₃ CH ₂ , Bn], [RC109 40; H, F, F, Cl, CF ₃ CH ₂ , CF ₃ ], [RC10941; H, F, F, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC10942; H, F, F, Cl, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC10943; H, F, F, Cl, CF ₃ CH ₂ , CF ₂ H], [RC10944; H, F, F, Cl, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC10945; H, F, Cl, H, CF ₃ CH ₂ , Me], [RC10946; H, F, Cl, H, CF ₃ CH ₂ , Et], [RC10947; H, F , Cl, H, CF ₃ CH ₂ , Pr], [RC10948; H, F, Cl, H, CF ₃ CH ₂ , i-Pr], [RC10949; H, F, Cl, H, CF ₃ CH ₂ , c-Pr], [RC10950; H, F, Cl, H, CF ₃ CH ₂ , Bu], [RC10951; H, F, Cl, H, CF ₃ CH ₂ , i-Bu], [RC10952; H, F, Cl, H, CF ₃ CH ₂ , t-Bu], [RC10953; H, F, Cl, H, CF ₃ CH ₂ , c-PrCH ₂ ], [RC10954; H, F, Cl, H, CF ₃ CH ₂ , Ph], [RC10955; H, F, Cl, H, CF ₃ CH ₂ , Bn], [RC10956; H, F, Cl, H, CF ₃ CH ₂ , CF ₃ ], [RC10957; H , F, Cl, H, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC10958; H, F, Cl, H, CF ₃ CH ₂ , CF ₃ CF ₂ ], [RC10959; H, F, Cl, H , CF ₃ CH ₂ , CF ₂ H], [RC10960; H, F, Cl, H, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC10961; H, F, Cl, Cl, CF ₃ CH ₂ , Me ], [RC10962; H, F, Cl, Cl, CF ₃ CH ₂ , Et], [RC10963; H, F, Cl, Cl, CF ₃ CH ₂ , Pr], [RC10964; H, F, Cl, Cl , CF ₃ CH ₂ , i-Pr], [RC10965; H, F, Cl, Cl, CF ₃ CH ₂ , c-Pr], [RC10966; H, F, Cl, Cl, CF ₃ CH ₂ , Bu] , [RC10967; H, F, Cl, Cl, CF ₃ CH ₂ , i-Bu], [RC10968; H, F, Cl, Cl, CF ₃ CH ₂ , t-Bu], [RC10969; H, F, Cl, Cl, CF ₃ CH ₂ , c-PrCH ₂ ], [RC10970; H, F, Cl, Cl, CF ₃ CH ₂ , Ph], [RC10971; H, F, Cl, Cl, CF ₃ CH ₂ , Bn], [RC10972; H, F, Cl, Cl, CF ₃ CH ₂ , CF ₃ ], [RC10973; H, F, Cl, Cl, CF ₃ CH ₂ , CF ₃ CH ₂ ], [RC10974; H, F, Cl, Cl, CF ₃ CH ₂
, CF ₃ CF ₂ ], [RC10975; H, F, Cl, Cl, CF ₃ CH ₂ , CF ₂ H], [RC10976; H, F, Cl, Cl, CF ₃ CH ₂ , CF ₂ HCF ₂ ], [RC10977; H, F, H, H, HCCCH ₂ , Me], [RC10978; H, F, H, H, HCCCH ₂ , Et], [RC10979; H, F, H, H, HCCCH ₂ , Pr] , [RC10980; H, F, H, H, HCCCH ₂ , i-Pr], [RC10981; H, F, H, H, HCCCH ₂ , c-Pr], [RC10982; H, F, H, H, HCCCH ₂ , Bu], [RC10983; H, F, H, H, HCCCH ₂ , i-Bu], [RC10984; H, F, H, H, HCCCH ₂ , t-Bu], [RC10985; H, F , H, H, HCCCH ₂ , c-PrCH ₂ ], [RC10986; H, F, H, H, HCCCH ₂ , Ph], [RC10987; H, F, H, H, HCCCH ₂ , Bn], [RC10988 ; H, F, H, H, HCCCH ₂ , CF ₃ ], [RC10989; H, F, H, H, HCCCH ₂ , CF ₃ CH ₂ ], [RC10990; H, F, H, H, HCCCH ₂ , CF ₃ CF ₂ ], [RC10991; H, F, H, H, HCCCH ₂ , CF ₂ H], [RC10992; H, F, H, H, HCCCH ₂ , CF ₂ HCF ₂ ], [RC10993; H, F, H, Me, HCCCH ₂ , Me], [RC10994; H, F, H, Me, HCCCH ₂ , Et], [RC10995; H, F, H, Me, HCCCH ₂ , Pr], [RC10996; H , F, H, Me, HCCCH ₂ , i-Pr], [RC10997; H, F, H, Me, HCCCH ₂ , c-Pr], [RC10998; H, F, H, Me, HCCCH ₂ , Bu] , [RC10999; H, F, H, Me, HCCCH ₂ , i-Bu], [RC11000; H, F, H, Me, HCCCH ₂ , t-Bu],

[RC11001; H, F, H, Me, HCCCH ₂ , c-PrCH ₂ ], [RC11002; H, F, H, Me, HCCCH ₂ , Ph], [RC11003; H, F, H, Me, HCCCH ₂ , Bn], [RC11004; H, F, H, Me, HCCCH ₂ , CF ₃ ], [RC11005; H, F, H, Me, HCCCH ₂ , CF ₃ CH ₂ ], [RC11006; H, F, H , Me, HCCCH ₂ , CF ₃ CF ₂ ], [RC11007; H, F, H, Me, HCCCH ₂ , CF ₂ H], [RC11008; H, F, H, Me, HCCCH ₂ , CF ₂ HCF ₂ ] , [RC11009; H, F, Me, Me, HCCCH ₂ , Me], [RC11010; H, F, Me, Me, HCCCH ₂ , Et], [RC11011; H, F, Me, Me, HCCCH ₂ , Pr ], [RC11012; H, F, Me, Me, HCCCH ₂ , i-Pr], [RC11013; H, F, Me, Me, HCCCH ₂ , c-Pr], [RC11014; H, F, Me, Me , HCCCH ₂ , Bu], [RC11015; H, F, Me, Me, HCCCH ₂ , i-Bu], [RC11016; H, F, Me, Me, HCCCH ₂ , t-Bu], [RC11017; H, F, Me, Me, HCCCH ₂ , c-PrCH ₂ ], [RC11018; H, F, Me, Me, HCCCH ₂ , Ph], [RC11019; H, F, Me, Me, HCCCH ₂ , Bn], [ RC11020; H, F, Me, Me, HCCCH ₂ , CF ₃ ], [RC11021; H, F, Me, Me, HCCCH ₂ , CF ₃ CH ₂ ], [RC11022; H, F, Me, Me, HCCCH ₂ , CF ₃ CF ₂ ], [RC11023; H, F, Me, Me, HCCCH ₂ , CF ₂ H], [RC11024; H, F, Me, Me, HCCCH ₂ , CF ₂ HCF ₂ ], [RC11025; H , F, Me, Et, HCCCH ₂ , Me], [RC11026; H, F, Me, Et, HCCCH ₂ , Et], [RC11027; H, F, Me, Et, HCCCH ₂ , Pr], [RC11028; H, F, Me, Et, HCCCH ₂ , i-Pr], [RC11029; H, F, Me, Et, HCCCH ₂ , c-Pr], [RC11030; H, F, Me, Et, HCCCH ₂ , Bu], [RC11031; H, F, Me, Et, HCCCH ₂ , i-Bu], [RC11032; H, F, Me, Et, HCCCH ₂ , t-Bu], [RC11033; H, F, Me, Et, HCCCH ₂ , c-PrCH ₂ ], [RC11034; H, F, Me, Et, HCCCH ₂ , Ph], [ RC11035; H, F, Me, Et, HCCCH ₂ , Bn], [RC11036; H, F, Me, Et, HCCCH ₂ , CF ₃ ], [RC11037; H, F, Me, Et, HCCCH ₂ , CF ₃ CH ₂ ], [RC11038; H, F, Me, Et, HCCCH ₂ , CF ₃ CF ₂ ], [RC11039; H, F, Me, Et, HCCCH ₂ , CF ₂ H], [RC11040; H, F, Me, Et, HCCCH ₂ , CF ₂ HCF ₂ ], [RC11041; H, F, Me, F, HCCCH ₂ , Me], [RC11042; H, F, Me, F, HCCCH ₂ , Et], [RC11043; H, F, Me, F, HCCCH ₂ , Pr], [RC11044; H, F, Me, F, HCCCH ₂ , i-Pr], [RC11045; H, F, Me, F, HCCCH ₂ , c-Pr ], [RC11046; H, F, Me, F, HCCCH ₂ , Bu], [RC11047; H, F, Me, F, HCCCH ₂ , i-Bu], [RC11048; H, F, Me, F, HCCCH ₂ , t-Bu], [RC11049; H, F, Me, F, HCCCH ₂ , c-PrCH ₂ ], [RC11050; H, F, Me, F, HCCCH ₂ , Ph], [RC11051; H, F _{, Me, F, HCCCH 2,} Bn], [RC11052; H, F, Me, F, HCCCH 2, CF 3], [RC11053; H, F, Me, F, HCCCH 2, CF 3 CH 2], [ RC11054; H, F, Me, F, HCCCH ₂ , CF ₃ CF ₂ ], [RC11055; H, F, Me, F, HCCCH ₂ , CF ₂ H], [RC11056; H, F, Me, F, HCCCH ₂ , CF ₂ HCF ₂ ], [RC11057; H, F, Me, Cl, HCCCH ₂ , Me], [RC11058; H, F, Me, Cl, H CCCH ₂ , Et], [RC11059; H, F, Me, Cl, HCCCH ₂ , Pr], [RC11060; H, F, Me, Cl, HCCCH ₂ , i-Pr], [RC11061; H, F, Me , Cl, HCCCH ₂ , c-Pr], [RC11062; H, F, Me, Cl, HCCCH ₂ , Bu], [RC11063; H, F, Me, Cl, HCCCH ₂ , i-Bu], [RC11064; H, F, Me, Cl, HCCCH ₂ , t-Bu], [RC11065; H, F, Me, Cl, HCCCH ₂ , c-PrCH ₂ ], [RC11066; H, F, Me, Cl, HCCCH ₂ , Ph], [RC11067; H, F, Me, Cl, HCCCH ₂ , Bn], [RC11068; H, F, Me, Cl, HCCCH ₂ , CF ₃ ], [RC11069; H, F, Me, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RC11070; H, F, Me, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RC11071; H, F, Me, Cl, HCCCH ₂ , CF ₂ H], [RC11072; H, F, Me, Cl, HCCCH ₂ , CF ₂ HCF ₂ ], [RC11073; H, F, Et, H, HCCCH ₂ , Me], [RC11074; H, F, Et, H, HCCCH ₂ , Et] , [RC11075; H, F, Et, H, HCCCH ₂ , Pr], [RC11076; H, F, Et, H, HCCCH ₂ , i-Pr], [RC11077; H, F, Et, H, HCCCH ₂ , c-Pr], [RC11078; H, F, Et, H, HCCCH ₂ , Bu], [RC11079; H, F, Et, H, HCCCH ₂ , i-Bu], [RC11080; H, F, Et , H, HCCCH ₂ , t-Bu], [RC11081; H, F, Et, H, HCCCH ₂ , c-PrCH ₂ ], [RC11082; H, F, Et, H, HCCCH ₂ , Ph], [RC11083 ; H, F, Et, H, HCCCH ₂ , Bn], [RC11084; H, F, Et, H, HCCCH ₂ , CF ₃ ], [RC11085; H, F, Et, H, HCCCH ₂ , CF ₃ CH ₂ ], [RC11086; H, F, Et, H, HCCCH ₂ , CF ₃ CF ₂ ], [RC11087; H, F, Et, H, HCCCH ₂ , CF ₂ H], [RC11088; H, F, Et, H, HCCCH ₂ , CF ₂ HCF ₂ ], [RC11089; H, F, Et, F, HCCCH ₂ , Me], [RC11090; H, F, Et, F, HCCCH ₂ , Et], [RC11091; H, F, Et, F, HCCCH ₂ , Pr], [RC11092; H, F, Et, F, HCCCH ₂ , i-Pr], [RC11093; H , F, Et, F, HCCCH ₂ , c-Pr], [RC11094; H, F, Et, F, HCCCH ₂ , Bu], [RC11095; H, F, Et, F, HCCCH ₂ , i-Bu] , [RC11096; H, F, Et, F, HCCCH ₂ , t-Bu], [RC11097; H, F, Et, F, HCCCH ₂ , c-PrCH ₂ ], [RC11098; H, F, Et, F , HCCCH ₂ , Ph], [RC11099; H, F, Et, F, HCCCH ₂ , Bn], [RC11100; H, F, Et, F, HCCCH ₂ , CF ₃ ], [RC11101; H, F, Et , F, HCCCH ₂ , CF ₃ CH ₂ ], [RC11102; H, F, Et, F, HCCCH ₂ , CF ₃ CF ₂ ], [RC11103; H, F, Et, F, HCCCH ₂ , CF ₂ H] , [RC11104; H, F, Et, F, HCCCH ₂ , CF ₂ HCF ₂ ], [RC11105; H, F, Et, Cl, HCCCH ₂ , Me], [RC11106; H, F, Et, Cl, HCCCH _{2, Et], [RC11107;} H, F, Et, Cl, HCCCH 2, Pr], [RC11108; H, F, Et, Cl, HCCCH 2, i-Pr], [RC11109; H, F, Et, Cl, HCCCH ₂ , c-Pr], [RC11110; H, F, Et, Cl, HCCCH ₂ , Bu], [RC11111; H, F, Et, Cl, HCCCH ₂ , i-Bu], [RC11112; H , F, Et, Cl, HCCCH ₂ , t-Bu], [RC11113; H, F, Et, Cl, HCCCH ₂ , c-PrCH ₂ ], [RC11114; H, F, Et, Cl, HCCCH ₂ , Ph ], [RC11115; H, F, Et, Cl, HCCCH ₂ , Bn], [RC11116; H, F, Et, Cl, HCCCH ₂ , CF ₃ ], [RC11 117; H, F, Et, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RC11118; H, F, Et, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RC11119; H, F, Et, Cl, HCCCH ₂ , CF ₂ H], [RC11120; H, F, Et, Cl, HCCCH ₂ , CF ₂ HCF ₂ ], [RC11121; H, F, F, H, HCCCH ₂ , Me], [RC11122; H, F, F, H, HCCCH ₂ , Et], [RC11123; H, F, F, H, HCCCH ₂ , Pr], [RC11124; H, F, F, H, HCCCH ₂ , i-Pr], [RC11125 ; H, F, F, H, HCCCH ₂ , c-Pr], [RC11126; H, F, F, H, HCCCH ₂ , Bu], [RC11127; H, F, F, H, HCCCH ₂ , i- Bu], [RC11128; H, F, F, H, HCCCH ₂ , t-Bu], [RC11129; H, F, F, H, HCCCH ₂ , c-PrCH ₂ ], [RC11130; H, F, F , H, HCCCH ₂ , Ph], [RC11131; H, F, F, H, HCCCH ₂ , Bn], [RC11132; H, F, F, H, HCCCH ₂ , CF ₃ ], [RC11133; H, F , F, H, HCCCH ₂ , CF ₃ CH ₂ ], [RC11134; H, F, F, H, HCCCH ₂ , CF ₃ CF ₂ ], [RC11135; H, F, F, H, HCCCH ₂ , CF ₂ H], [RC11136; H, F, F, H, HCCCH ₂ , CF ₂ HCF ₂ ], [RC11137; H, F, F, F, HCCCH ₂ , Me], [RC11138; H, F, F, F , HCCCH ₂ , Et], [RC11139; H, F, F, F, HCCCH ₂ , Pr], [RC11140; H, F, F, F, HCCCH ₂ , i-Pr], [RC11141; H, F, F, F, HCCCH ₂ , c-Pr], [RC11142; H, F, F, F, HCCCH ₂ , Bu], [RC11143; H, F, F, F, HCCCH ₂ , i-Bu], [RC11144 ; H, F, F, F, HCCCH ₂ , t-Bu], [RC11145; H, F, F, F, HCCCH ₂ , c-PrCH ₂ ], [RC11146; H, F, F, F, HCCCH ₂ , Ph], [RC111 47; H, F, F, F, HCCCH ₂ , Bn], [RC11148; H, F, F, F, HCCCH ₂ , CF ₃ ], [RC11149; H, F, F, F, HCCCH ₂ , CF ₃ CH ₂ ], [RC11150; H, F, F, F, HCCCH ₂ , CF ₃ CF ₂ ], [RC11151; H, F, F, F, HCCCH ₂ , CF ₂ H], [RC11152; H, F, F, F, HCCCH ₂ , CF ₂ HCF ₂ ], [RC11153; H, F, F, Cl, HCCCH ₂ , Me], [RC11154; H, F, F, Cl, HCCCH ₂ , Et], [RC11155; H, F, F, Cl, HCCCH ₂ , Pr], [RC11156; H, F, F, Cl, HCCCH ₂ , i-Pr], [RC11157; H, F, F, Cl, HCCCH ₂ , c-Pr ], [RC11158; H, F, F, Cl, HCCCH ₂ , Bu], [RC11159; H, F, F, Cl, HCCCH ₂ , i-Bu], [RC11160; H, F, F, Cl, HCCCH ₂ , t-Bu], [RC11161; H, F, F, Cl, HCCCH ₂ , c-PrCH ₂ ], [RC11162; H, F, F, Cl, HCCCH ₂ , Ph], [RC11163; H, F , F, Cl, HCCCH ₂ , Bn], [RC11164; H, F, F, Cl, HCCCH ₂ , CF ₃ ], [RC11165; H, F, F, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [ RC11166; H, F, F, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RC11167; H, F, F, Cl, HCCCH ₂ , CF ₂ H], [RC11168; H, F, F, Cl, HCCCH ₂ , CF ₂ HCF ₂ ], [RC11169; H, F, Cl, H, HCCCH ₂ , Me], [RC11170; H, F, Cl, H, HCCCH ₂ , Et], [RC11171; H, F, Cl , H, HCCCH ₂ , Pr], [RC11172; H, F, Cl, H, HCCCH ₂ , i-Pr], [RC11173; H, F, Cl, H, HCCCH ₂ , c-Pr], [RC11174; H, F, Cl, H, HCCCH ₂ , Bu], [RC11175; H, F, Cl, H, HCCCH ₂ , i-Bu], [RC11176; H, F, Cl, H, HCCCH ₂ , t -Bu], [RC11177; H, F, Cl, H, HCCCH ₂ , c-PrCH ₂ ], [RC11178; H, F, Cl, H, HCCCH ₂ , Ph], [RC11179; H, F, Cl, H, HCCCH ₂ , Bn], [RC11180; H, F, Cl, H, HCCCH ₂ , CF ₃ ], [RC11181; H, F, Cl, H, HCCCH ₂ , CF ₃ CH ₂ ], [RC11182; H , F, Cl, H, HCCCH ₂ , CF ₃ CF ₂ ], [RC11183; H, F, Cl, H, HCCCH ₂ , CF ₂ H], [RC11184; H, F, Cl, H, HCCCH ₂ , CF ₂ HCF ₂ ], [RC11185; H, F, Cl, Cl, HCCCH ₂ , Me], [RC11186; H, F, Cl, Cl, HCCCH ₂ , Et], [RC11187; H, F, Cl, Cl, HCCCH ₂ , Pr], [RC11188; H, F, Cl, Cl, HCCCH ₂ , i-Pr], [RC11189; H, F, Cl, Cl, HCCCH ₂ , c-Pr], [RC11190; H, F , Cl, Cl, HCCCH ₂ , Bu], [RC11191; H, F, Cl, Cl, HCCCH ₂ , i-Bu], [RC11192; H, F, Cl, Cl, HCCCH ₂ , t-Bu], [ RC11193; H, F, Cl, Cl, HCCCH ₂ , c-PrCH ₂ ], [RC11194; H, F, Cl, Cl, HCCCH ₂ , Ph], [RC11195; H, F, Cl, Cl, HCCCH ₂ , Bn], [RC11196; H, F, Cl, Cl, HCCCH ₂ , CF ₃ ], [RC11197; H, F, Cl, Cl, HCCCH ₂ , CF ₃ CH ₂ ], [RC11198; H, F, Cl, Cl, HCCCH ₂ , CF ₃ CF ₂ ], [RC11199; H, F, Cl, Cl, HCCCH ₂ , CF ₂ H], [RC11200; H, F, Cl, Cl, HCCCH ₂ , CF ₂ HCF ₂ ],

[RC11201; H, F, H, H, CH ₃ CCCH ₂ , Me], [RC11202; H, F, H, H, CH ₃ CCCH ₂ , Et], [RC11203; H, F, H, H, CH ₃ CCCH ₂ , Pr], [RC11204; H, F, H, H, CH ₃ CCCH ₂ , i-Pr], [RC11205; H, F, H, H, CH ₃ CCCH ₂ , c-Pr], [ RC11206; H, F, H, H, CH ₃ CCCH ₂ , Bu], [RC11207; H, F, H, H, CH ₃ CCCH ₂ , i-Bu], [RC11208; H, F, H, H, CH ₃ CCCH ₂ , t-Bu], [RC11209; H, F, H, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC11210; H, F, H, H, CH ₃ CCCH ₂ , Ph] , [RC11211; H, F, H, H, CH ₃ CCCH ₂ , Bn], [RC11212; H, F, H, H, CH ₃ CCCH ₂ , CF ₃ ], [RC11213; H, F, H, H , CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC11214; H, F, H, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC11215; H, F, H, H, CH ₃ CCCH ₂ , CF ₂ H], [RC11216; H, F, H, H, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC11217; H, F, H, Me, CH ₃ CCCH ₂ , Me], [RC11218; H , F, H, Me, CH ₃ CCCH ₂ , Et], [RC11219; H, F, H, Me, CH ₃ CCCH ₂ , Pr], [RC11220; H, F, H, Me, CH ₃ CCCH ₂ , i-Pr], [RC11221; H, F, H, Me, CH ₃ CCCH ₂ , c-Pr], [RC11222; H, F, H, Me, CH ₃ CCCH ₂ , Bu], [RC11223; H, F, H, Me, CH ₃ CCCH ₂ , i-Bu], [RC11224; H, F, H, Me, CH ₃ CCCH ₂ , t-Bu], [RC11225; H, F, H, Me, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC11226; H, F, H, Me, CH ₃ CCCH ₂ , Ph], [RC11227; H, F, H, Me, CH ₃ CCCH ₂ , Bn], [RC11228; H, F, H, Me, CH ₃ CCCH ₂ , CF ₃ ], [RC11229; H, F, H, Me, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC11230; H, F, H, Me, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC11231; H, F, H, Me, CH ₃ CCCH ₂ , CF ₂ H], [RC11232; H, F, H, Me, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC11233; H, F, Me, Me, CH ₃ CCCH ₂ , Me], [RC11234; H, F, Me, Me, CH ₃ CCCH ₂ , Et], [RC11235; H, F, Me , Me, CH ₃ CCCH ₂ , Pr], [RC11236; H, F, Me, Me, CH ₃ CCCH ₂ , i-Pr], [RC11237; H, F, Me, Me, CH ₃ CCCH ₂ , c- Pr], [RC11238; H, F, Me, Me, CH ₃ CCCH ₂ , Bu], [RC11239; H, F, Me, Me, CH ₃ CCCH ₂ , i-Bu], [RC11240; H, F, Me, Me, CH ₃ CCCH ₂ , t-Bu], [RC11241; H, F, Me, Me, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC11242; H, F, Me, Me, CH ₃ CCCH ₂ , Ph], [RC11243; H, F, Me, Me, CH ₃ CCCH ₂ , Bn], [RC11244; H, F, Me, Me, CH ₃ CCCH ₂ , CF ₃ ], [RC11245; H, F , Me, Me, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC11246; H, F, Me, Me, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC11247; H, F, Me, Me, CH ₃ CCCH ₂ , CF ₂ H], [RC11248; H, F, Me, Me, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC11249; H, F, Me, Et, CH ₃ CCCH ₂ , Me], [RC11250; H, F, Me, Et, CH ₃ CCCH ₂ , Et], [RC11251; H, F, Me, Et, CH ₃ CCCH ₂ , Pr], [RC11252; H, F, Me, Et, CH ₃ CCCH ₂ , i-Pr], [RC11253; H, F, Me, Et, CH ₃ CCCH ₂ , c -Pr], [RC11254; H, F, Me, Et, CH ₃ CCCH ₂ , Bu], [RC11255; H, F, Me, Et, CH ₃ CCCH ₂ , i-Bu], [RC11256; H, F , Me, Et, CH ₃ CCCH ₂ , t-Bu], [RC11257; H, F, Me, Et, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC11258; H, F, Me, Et, CH ₃ CCCH ₂ , Ph], [RC11259; H, F, Me, Et, CH ₃ CCCH ₂ , Bn], [RC11260; H, F, Me, Et, CH ₃ CCCH ₂ , CF ₃ ], [RC11261; H, F, Me, Et, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC11262; H, F, Me, Et, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC11263; H, F, Me, Et, CH ₃ CCCH ₂ , CF ₂ H], [RC11264; H, F, Me, Et, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC11265; H, F, Me, F, CH ₃ CCCH ₂ , Me] , [RC11266; H, F, Me, F, CH ₃ CCCH ₂ , Et], [RC11267; H, F, Me, F, CH ₃ CCCH ₂ , Pr], [RC11268; H, F, Me, F, CH ₃ CCCH ₂ , i-Pr], [RC11269; H, F, Me, F, CH ₃ CCCH ₂ , c-Pr], [RC11270; H, F, Me, F, CH ₃ CCCH ₂ , Bu], [RC11271; H, F, Me, F, CH ₃ CCCH ₂ , i-Bu], [RC11272; H, F, Me, F, CH ₃ CCCH ₂ , t-Bu], [RC11273; H, F, Me , F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC11274; H, F, Me, F, CH ₃ CCCH ₂ , Ph], [RC11275; H, F, Me, F, CH ₃ CCCH ₂ , Bn ], [RC11276; H, F, Me, F, CH ₃ CCCH ₂ , CF ₃ ], [RC11277; H, F, Me, F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC11278; H, F , Me, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC11279; H, F, Me, F, CH ₃ CCCH ₂ , C F ₂ H], [RC11280; H, F, Me, F, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC11281; H, F, Me, Cl, CH ₃ CCCH ₂ , Me], [RC11282; H , F, Me, Cl, CH ₃ CCCH ₂ , Et], [RC11283; H, F, Me, Cl, CH ₃ CCCH ₂ , Pr], [RC11284; H, F, Me, Cl, CH ₃ CCCH ₂ , i-Pr], [RC11285; H, F, Me, Cl, CH ₃ CCCH ₂ , c-Pr], [RC11286; H, F, Me, Cl, CH ₃ CCCH ₂ , Bu], [RC11287; H, F, Me, Cl, CH ₃ CCCH ₂ , i-Bu], [RC11288; H, F, Me, Cl, CH ₃ CCCH ₂ , t-Bu], [RC11289; H, F, Me, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC11290; H, F, Me, Cl, CH ₃ CCCH ₂ , Ph], [RC11291; H, F, Me, Cl, CH ₃ CCCH ₂ , Bn], [RC11292; H, F, Me, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RC11293; H, F, Me, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC11294; H, F, Me, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC11295; H, F, Me, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RC11296; H, F, Me, Cl, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC11297; H, F, Et, H, CH ₃ CCCH ₂ , Me], [RC11298; H, F, Et, H, CH ₃ CCCH ₂ , Et], [RC11299; H, F, Et , H, CH ₃ CCCH ₂ , Pr], [RC11300; H, F, Et, H, CH ₃ CCCH ₂ , i-Pr], [RC11301; H, F, Et, H, CH ₃ CCCH ₂ , c- Pr], [RC11302; H, F, Et, H, CH ₃ CCCH ₂ , Bu], [RC11303; H, F, Et, H, CH ₃ CCCH ₂ , i-Bu], [RC11304; H, F, Et, H, CH ₃ CCCH ₂ , t-Bu], [RC11305; H, F, Et, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC11306; H, F, Et, H, CH ₃ CCCH ₂ , Ph], [RC11307; H, F, Et, H, CH ₃ CCCH ₂ , Bn], [RC11308; H, F, Et, H, CH ₃ CCCH ₂ , CF ₃ ], [RC11309; H, F, Et, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC11310; H, F, Et, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC11311; H, F, Et, H, CH ₃ CCCH ₂ , CF ₂ H], [RC11312; H, F, Et, H, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC11313 ; H, F, Et, F, CH ₃ CCCH ₂ , Me], [RC11314; H, F, Et, F, CH ₃ CCCH ₂ , Et], [RC11315; H, F, Et, F, CH ₃ CCCH ₂ , Pr], [RC11316; H, F, Et, F, CH ₃ CCCH ₂ , i-Pr], [RC11317; H, F, Et, F, CH ₃ CCCH ₂ , c-Pr], [RC11318; H, F, Et, F, CH ₃ CCCH ₂ , Bu], [RC11319; H, F, Et, F, CH ₃ CCCH ₂ , i-Bu], [RC11320; H, F, Et, F, CH ₃ CCCH ₂ , t-Bu], [RC11321; H, F, Et, F, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC11322; H, F, Et, F, CH ₃ CCCH ₂ , Ph], [ RC11323; H, F, Et, F, CH ₃ CCCH ₂ , Bn], [RC11324; H, F, Et, F, CH ₃ CCCH ₂ , CF ₃ ], [RC11325; H, F, Et, F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC11326; H, F, Et, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC11327; H, F, Et, F, CH ₃ CCCH ₂ , CF ₂ H], [RC11328; H, F, Et, F, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC11329; H, F, Et, Cl, CH ₃ CCCH ₂ , Me], [RC11330; H, F , Et, Cl, CH ₃ CCCH ₂ , Et], [RC11331; H, F, Et, Cl, CH ₃ CCCH ₂ , Pr], [RC1 1332; H, F, Et, Cl, CH ₃ CCCH ₂ , i-Pr], [RC11333; H, F, Et, Cl, CH ₃ CCCH ₂ , c-Pr], [RC11334; H, F, Et, Cl, CH ₃ CCCH ₂ , Bu], [RC11335; H, F, Et, Cl, CH ₃ CCCH ₂ , i-Bu], [RC11336; H, F, Et, Cl, CH ₃ CCCH ₂ , t-Bu ], [RC11337; H, F, Et, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC11338; H, F, Et, Cl, CH ₃ CCCH ₂ , Ph], [RC11339; H, F, Et, Cl, CH ₃ CCCH ₂ , Bn], [RC11340; H, F, Et, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RC11341; H, F, Et, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC11342; H, F, Et, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC11343; H, F, Et, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RC11344; H, F, Et, Cl, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC11345; H, F, F, H, CH ₃ CCCH ₂ , Me], [RC11346; H, F, F, H, CH ₃ CCCH ₂ , Et], [RC11347; H, F, F, H, CH ₃ CCCH ₂ , Pr], [RC11348; H, F, F, H, CH ₃ CCCH ₂ , i-Pr], [RC11349; H, F, F, H, CH ₃ CCCH ₂ , c-Pr], [RC11350; H, F, F, H, CH ₃ CCCH ₂ , Bu], [RC11351; H, F, F, H, CH ₃ CCCH ₂ , i-Bu], [RC11352; H, F, F, H, CH ₃ CCCH ₂ , t-Bu], [RC11353; H, F, F, H, CH ₃ CCCH ₂ , c-PrCH ₂ ] , [RC11354; H, F, F, H, CH ₃ CCCH ₂ , Ph], [RC11355; H, F, F, H, CH ₃ CCCH ₂ , Bn], [RC11356; H, F, F, H, CH ₃ CCCH ₂ , CF ₃ ], [RC11357; H, F, F, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC11358; H, F, F, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC11359; H, F, F, H, CH ₃ CCCH ₂ , CF ₂ H], [RC11360; H, F, F, H, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC11361; H, F, F, F, CH ₃ CCCH ₂ , Me], [RC11362; H, F, F, F, CH ₃ CCCH ₂ , Et], [RC11363; H, F, F, F , CH ₃ CCCH ₂ , Pr], [RC11364; H, F, F, F, CH ₃ CCCH ₂ , i-Pr], [RC11365; H, F, F, F, CH ₃ CCCH ₂ , c-Pr] , [RC11366; H, F, F, F, CH ₃ CCCH ₂ , Bu], [RC11367; H, F, F, F, CH ₃ CCCH ₂ , i-Bu], [RC11368; H, F, F, F, CH ₃ CCCH ₂ , t-Bu], [RC11369; H, F, F, F, CH ₃
CCCH ₂ , c-PrCH ₂ ], [RC11370; H, F, F, F, CH ₃ CCCH ₂ , Ph], [RC11371; H, F, F, F, CH ₃ CCCH ₂ , Bn], [RC11372; H, F, F, F, CH ₃ CCCH ₂ , CF ₃ ], [RC11373; H, F, F, F, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC11374; H, F, F, F, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC11375; H, F, F, F, CH ₃ CCCH ₂ , CF ₂ H], [RC11376; H, F, F, F, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC11377; H, F, F, Cl, CH ₃ CCCH ₂ , Me], [RC11378; H, F, F, Cl, CH ₃ CCCH ₂ , Et], [RC11379; H, F, F , Cl, CH ₃ CCCH ₂ , Pr], [RC11380; H, F, F, Cl, CH ₃ CCCH ₂ , i-Pr], [RC11381; H, F, F, Cl, CH ₃ CCCH ₂ , c- Pr], [RC11382; H, F, F, Cl, CH ₃ CCCH ₂ , Bu], [RC11383; H, F, F, Cl, CH ₃ CCCH ₂ , i-Bu], [RC11384; H, F, F, Cl, CH ₃ CCCH ₂ , t-Bu], [RC11385; H, F, F, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC11386; H, F, F, Cl, CH ₃ CCCH ₂ , Ph], [RC11387; H, F, F, Cl, CH ₃ CCCH ₂ , Bn], [RC11388; H, F, F, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RC11389; H, F , F, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC11390; H, F, F, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC11391; H, F, F, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RC11392; H, F, F, Cl, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC11393; H, F, Cl, H, CH ₃ CCCH ₂ , Me], [RC11394; H, F, Cl, H, CH ₃ CCCH ₂ , Et], [RC11395; H, F, Cl, H, CH ₃ CCCH ₂ , Pr] , [RC11396; H, F, Cl, H, CH ₃ CCCH ₂ , i-Pr], [RC11397; H, F, Cl, H, CH ₃ CCCH ₂ , c-Pr], [RC11398; H, F, Cl, H, CH ₃ CCCH ₂ , Bu], [RC11399; H, F, Cl, H, CH ₃ CCCH ₂ , i-Bu], [RC11400; H, F, Cl, H, CH ₃ CCCH ₂ , t -Bu],

[RC11401; H, F, Cl, H, CH ₃ CCCH ₂ , c-PrCH ₂ ], [RC11402; H, F, Cl, H, CH ₃ CCCH ₂ , Ph], [RC11403; H, F, Cl, H, CH ₃ CCCH ₂ , Bn], [RC11404; H, F, Cl, H, CH ₃ CCCH ₂ , CF ₃ ], [RC11405; H, F, Cl, H, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC11406; H, F, Cl, H, CH ₃ CCCH ₂ , CF ₃ CF ₂ ], [RC11407; H, F, Cl, H, CH ₃ CCCH ₂ , CF ₂ H], [RC11408; H, F, Cl, H, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC11409; H, F, Cl, Cl, CH ₃ CCCH ₂ , Me], [RC11410; H, F, Cl, Cl, CH ₃ CCCH ₂ , Et], [RC11411; H, F, Cl, Cl, CH ₃ CCCH ₂ , Pr], [RC11412; H, F, Cl, Cl, CH ₃ CCCH ₂ , i-Pr], [RC11413; H, F, Cl, Cl, CH ₃ CCCH ₂ , c-Pr], [RC11414; H, F, Cl, Cl, CH ₃ CCCH ₂ , Bu], [RC11415; H, F, Cl, Cl, CH ₃ CCCH ₂ , i-Bu], [RC11416; H, F, Cl, Cl, CH ₃ CCCH ₂ , t-Bu], [RC11417; H, F, Cl, Cl, CH ₃ CCCH ₂ , c-PrCH ₂ ], [ RC11418; H, F, Cl, Cl, CH ₃ CCCH ₂ , Ph], [RC11419; H, F, Cl, Cl, CH ₃ CCCH ₂ , Bn], [RC11420; H, F, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ ], [RC11421; H, F, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ CH ₂ ], [RC11422; H, F, Cl, Cl, CH ₃ CCCH ₂ , CF ₃ CF ₂ ] , [RC11423; H, F, Cl, Cl, CH ₃ CCCH ₂ , CF ₂ H], [RC11424; H, F, Cl, Cl, CH ₃ CCCH ₂ , CF ₂ HCF ₂ ], [RC11425; H, F , H, H, c-Pr, Me], [RC11426; H, F, H, H, c-Pr, Et], [RC114 27; H, F, H, H, c-Pr, Pr], [RC11428; H, F, H, H, c-Pr, i-Pr], [RC11429; H, F, H, H, c- Pr, c-Pr], [RC11430; H, F, H, H, c-Pr, Bu], [RC11431; H, F, H, H, c-Pr, i-Bu], [RC11432; H, F, H, H, c-Pr, t-Bu], [RC11433; H, F, H, H, c-Pr, c-PrCH ₂ ], [RC11434; H, F, H, H, c-Pr , Ph], [RC11435; H, F, H, H, c-Pr, Bn], [RC11436; H, F, H, H, c-Pr, CF ₃ ], [RC11437; H, F, H, H, c-Pr, CF ₃ CH ₂ ], [RC11438; H, F, H, H, c-Pr, CF ₃ CF ₂ ], [RC11439; H, F, H, H, c-Pr, CF ₂ H], [RC11440; H, F, H, H, c-Pr, CF ₂ HCF ₂ ], [RC11441; H, F, H, Me, c-Pr, Me], [RC11442; H, F, H , Me, c-Pr, Et], [RC11443; H, F, H, Me, c-Pr, Pr], [RC11444; H, F, H, Me, c-Pr, i-Pr], [RC11445 ; H, F, H, Me, c-Pr, c-Pr], [RC11446; H, F, H, Me, c-Pr, Bu], [RC11447; H, F, H, Me, c-Pr , i-Bu], [RC11448; H, F, H, Me, c-Pr, t-Bu], [RC11449; H, F, H, Me, c-Pr, c-PrCH ₂ ], [RC11450; H, F, H, Me, c-Pr, Ph], [RC11451; H, F, H, Me, c-Pr, Bn], [RC11452; H, F, H, Me, c-Pr, CF ₃ ], [RC11453; H, F, H, Me, c-Pr, CF ₃ CH ₂ ], [RC11454; H, F, H, Me, c-Pr, CF ₃ CF ₂ ], [RC11455; H, F , H, Me, c-Pr, CF ₂ H], [RC11456; H, F, H, Me, c-Pr, CF ₂ HCF ₂ ], [RC11457; H, F, Me, Me, c-Pr, Me], [RC11458; H, F, Me, Me, c-Pr, Et], [RC11459; H, F, Me, Me, c-Pr, Pr], [RC11460; H, F, Me, Me, c-Pr, i-Pr], [R C11461; H, F, Me, Me, c-Pr, c-Pr], [RC11462; H, F, Me, Me, c-Pr, Bu], [RC11463; H, F, Me, Me, c- Pr, i-Bu], [RC11464; H, F, Me, Me, c-Pr, t-Bu], [RC11465; H, F, Me, Me, c-Pr, c-PrCH ₂ ], [RC11466 ; H, F, Me, Me, c-Pr, Ph], [RC11467; H, F, Me, Me, c-Pr, Bn], [RC11468; H, F, Me, Me, c-Pr, CF ₃ ], [RC11469; H, F, Me, Me, c-Pr, CF ₃ CH ₂ ], [RC11470; H, F, Me, Me, c-Pr, CF ₃ CF ₂ ], [RC11471; H, F, Me, Me, c-Pr, CF ₂ H], [RC11472; H, F, Me, Me, c-Pr, CF ₂ HCF ₂ ], [RC11473; H, F, Me, Et, c-Pr , Me], [RC11474; H, F, Me, Et, c-Pr, Et], [RC11475; H, F, Me, Et, c-Pr, Pr], [RC11476; H, F, Me, Et , c-Pr, i-Pr], [RC11477; H, F, Me, Et, c-Pr, c-Pr], [RC11478; H, F, Me, Et, c-Pr, Bu], [RC11479 ; H, F, Me, Et, c-Pr, i-Bu], [RC11480; H, F, Me, Et, c-Pr, t-Bu], [RC11481; H, F, Me, Et, c -Pr, c-PrCH ₂ ], [RC11482; H, F, Me, Et, c-Pr, Ph], [RC11483; H, F, Me, Et, c-Pr, Bn], [RC11484; H, F, Me, Et, c-Pr, CF ₃ ], [RC11485; H, F, Me, Et, c-Pr, CF ₃ CH ₂ ], [RC11486; H, F, Me, Et, c-Pr, CF ₃ CF ₂ ], [RC11487; H, F, Me, Et, c-Pr, CF ₂ H], [RC11488; H, F, Me, Et, c-Pr, CF ₂ HCF ₂ ], [RC11489; H, F, Me, F, c-Pr, Me], [RC11490; H, F, Me, F, c-Pr, Et], [RC11491; H, F, Me, F, c-Pr, Pr] , [RC11492; H, F, Me, F, c-Pr, i-Pr], [RC11493; H, F, Me, F, c-Pr, c-Pr], [RC11494; H, F, Me, F, c-Pr, Bu], [RC11495; H, F, Me, F, c-Pr, i-Bu], [ RC11496; H, F, Me, F, c-Pr, t-Bu], [RC11497; H, F, Me, F, c-Pr, c-PrCH ₂ ], [RC11498; H, F, Me, F , c-Pr, Ph], [RC11499; H, F, Me, F, c-Pr, Bn], [RC11500; H, F, Me, F, c-Pr, CF ₃ ], [RC11501; H, F, Me, F, c-Pr, CF ₃ CH ₂ ], [RC11502; H, F, Me, F, c-Pr, CF ₃ CF ₂ ], [RC11503; H, F, Me, F, c- Pr, CF ₂ H], [RC11504; H, F, Me, F, c-Pr, CF ₂ HCF ₂ ], [RC11505; H, F, Me, Cl, c-Pr, Me], [RC11506; H , F, Me, Cl, c-Pr, Et], [RC11507; H, F, Me, Cl, c-Pr, Pr], [RC11508; H, F, Me, Cl, c-Pr, i-Pr ], [RC11509; H, F, Me, Cl, c-Pr, c-Pr], [RC11510; H, F, Me, Cl, c-Pr, Bu], [RC11511; H, F, Me, Cl , c-Pr, i-Bu], [RC11512; H, F, Me, Cl, c-Pr, t-Bu], [RC11513; H, F, Me, Cl, c-Pr, c-PrCH ₂ ] , [RC11514; H, F, Me, Cl, c-Pr, Ph], [RC11515; H, F, Me, Cl, c-Pr, Bn], [RC11516; H, F, Me, Cl, c- Pr, CF ₃ ], [RC11517; H, F, Me, Cl, c-Pr, CF ₃ CH ₂ ], [RC11518; H, F, Me, Cl, c-Pr, CF ₃ CF ₂ ], [RC11519 ; H, F, Me, Cl, c-Pr, CF ₂ H], [RC11520; H, F, Me, Cl, c-Pr, CF ₂ HCF ₂ ], [RC11521; H, F, Et, H, c-Pr, Me], [RC11522; H, F, Et, H, c-Pr, Et], [RC11523; H, F, Et, H, c-Pr, Pr], [RC11524; H, F, Et, H, c-Pr, i-Pr], [RC11525; H, F, Et, H, c-Pr, c-Pr], [RC11526; H, F, Et, H, c-Pr, Bu], [RC11527; H, F, Et, H, c-Pr, i-Bu], [RC11528; H, F, Et, H, c-Pr, t-Bu] , [RC11529; H, F, Et, H, c-Pr, c-PrCH ₂ ], [RC11530; H, F, Et, H, c-Pr, Ph], [RC11531; H, F, Et, H , c-Pr, Bn], [RC11532; H, F, Et, H, c-Pr, CF ₃ ], [RC11533; H, F, Et, H, c-Pr, CF ₃ CH ₂ ], [RC11534 ; H, F, Et, H, c-Pr, CF ₃ CF ₂ ], [RC11535; H, F, Et, H, c-Pr, CF ₂ H], [RC11536; H, F, Et, H, c-Pr, CF ₂ HCF ₂ ], [RC11537; H, F, Et, F, c-Pr, Me], [RC11538; H, F, Et, F, c-Pr, Et], [RC11539; H , F, Et, F, c-Pr, Pr], [RC11540; H, F, Et, F, c-Pr, i-Pr], [RC11541; H, F, Et, F, c-Pr, c -Pr], [RC11542; H, F, Et, F, c-Pr, Bu], [RC11543; H, F, Et, F, c-Pr, i-Bu], [RC11544; H, F, Et , F, c-Pr, t-Bu], [RC11545; H, F, Et, F, c-Pr, c-PrCH ₂ ], [RC11546; H, F, Et, F, c-Pr, Ph] , [RC11547; H, F, Et, F, c-Pr, Bn], [RC11548; H, F, Et, F, c-Pr, CF ₃ ], [RC11549; H, F, Et, F, c -Pr, CF ₃ CH ₂ ], [RC11550; H, F, Et, F, c-Pr, CF ₃ CF ₂ ], [RC11551; H, F, Et, F, c-Pr, CF ₂ H], [RC11552; H, F, Et, F, c-Pr, CF ₂ HCF ₂ ], [RC11553; H, F, Et, Cl, c-Pr, Me], [RC11554; H, F, Et, Cl, c-Pr, Et], [RC11555; H, F, Et, Cl, c-Pr, Pr], [RC11556; H, F, Et, Cl, c-Pr, i-Pr], [RC11557; H, F, Et, Cl, c-Pr, c-Pr], [RC11558; H, F, Et, Cl, c-Pr, Bu], [RC11559; H, F, Et, Cl, cP r, i-Bu], [RC11560; H, F, Et, Cl, c-Pr, t-Bu], [RC11561; H, F, Et, Cl, c-Pr, c-PrCH ₂ ], [RC11562 ; H, F, Et, Cl, c-Pr, Ph], [RC11563; H, F, Et, Cl, c-Pr, Bn], [RC11564; H, F, Et, Cl, c-Pr, CF ₃ ], [RC11565; H, F, Et, Cl, c-Pr, CF ₃ CH ₂ ], [RC11566; H, F, Et, Cl, c-Pr, CF ₃ CF ₂ ], [RC11567; H, F, Et, Cl, c-Pr, CF ₂ H], [RC11568; H, F, Et, Cl, c-Pr, CF ₂ HCF ₂ ], [RC11569; H, F, F, H, c-Pr , Me], [RC11570; H, F, F, H, c-Pr, Et], [RC11571; H, F, F, H, c-Pr, Pr], [RC11572; H, F, F, H , c-Pr, i-Pr], [RC11573; H, F, F, H, c-Pr, c-Pr], [RC11574; H, F, F, H, c-Pr, Bu], [RC11575 ; H, F, F, H, c-Pr, i-Bu], [RC11576; H, F, F, H, c-Pr, t-Bu], [RC11577; H, F, F, H, c -Pr, c-PrCH ₂ ], [RC11578; H, F, F, H, c-Pr, Ph], [RC11579; H, F, F, H, c-Pr, Bn], [RC11580; H, F, F, H, c-Pr, CF ₃ ], [RC11581; H, F, F, H, c-Pr, CF ₃ CH ₂ ], [RC11582; H, F, F, H, c-Pr, CF ₃ CF ₂ ], [RC11583; H, F, F, H, c-Pr, CF ₂ H], [RC11584; H, F, F, H, c-Pr, CF ₂ HCF ₂ ], [RC11585; H, F, F, F, c-Pr, Me], [RC11586; H, F, F, F, c-Pr, Et], [RC11587; H, F, F, F, c-Pr, Pr] , [RC11588; H, F, F, F, c-Pr, i-Pr], [RC11589; H, F, F, F, c-Pr, c-Pr], [RC11590; H, F, F, F, c-Pr, Bu], [RC11591; H, F, F, F, c-Pr, i-Bu], [RC11592; H, F, F, F, c-Pr, t-Bu], [ RC11593; H, F, F, F, cP r, c-PrCH ₂ ], [RC11594; H, F, F, F, c-Pr, Ph], [RC11595; H, F, F, F, c-Pr, Bn], [RC11596; H, F , F, F, c-Pr, CF ₃ ], [RC11597; H, F, F, F, c-Pr, CF ₃ CH ₂ ], [RC11598; H, F, F, F, c-Pr, CF ₃ CF ₂ ], [RC11599; H, F, F, F, c-Pr, CF ₂ H], [RC11600; H, F, F, F, c-Pr, CF ₂ HCF ₂ ],

[RC11601; H, F, F, Cl, c-Pr, Me], [RC11602; H, F, F, Cl, c-Pr, Et], [RC11603; H, F, F, Cl, c-Pr , Pr], [RC11604; H, F, F, Cl, c-Pr, i-Pr], [RC11605; H, F, F, Cl, c-Pr, c-Pr], [RC11606; H, F , F, Cl, c-Pr, Bu], [RC11607; H, F, F, Cl, c-Pr, i-Bu], [RC11608; H, F, F, Cl, c-Pr, t-Bu ], [RC11609; H, F, F, Cl, c-Pr, c-PrCH ₂ ], [RC11610; H, F, F, Cl, c-Pr, Ph], [RC11611; H, F, F, Cl, c-Pr, Bn], [RC11612; H, F, F, Cl, c-Pr, CF ₃ ], [RC11613; H, F, F, Cl, c-Pr, CF ₃ CH ₂ ], [ RC11614; H, F, F, Cl, c-Pr, CF ₃ CF ₂ ], [RC11615; H, F, F, Cl, c-Pr, CF ₂ H], [RC11616; H, F, F, Cl , c-Pr, CF ₂ HCF ₂ ], [RC11617; H, F, Cl, H, c-Pr, Me], [RC11618; H, F, Cl, H, c-Pr, Et], [RC11619; H, F, Cl, H, c-Pr, Pr], [RC11620; H, F, Cl, H, c-Pr, i-Pr], [RC11621; H, F, Cl, H, c-Pr, c-Pr], [RC11622; H, F, Cl, H, c-Pr, Bu], [RC11623; H, F, Cl, H, c-Pr, i-Bu], [RC11624; H, F, Cl, H, c-Pr, t-Bu], [RC11625; H, F, Cl, H, c-Pr, c-PrCH ₂ ], [RC11626; H, F, Cl, H, c-Pr, Ph ], [RC11627; H, F, Cl, H, c-Pr, Bn], [RC11628; H, F, Cl, H, c-Pr, CF ₃ ], [RC11629; H, F, Cl, H, c-Pr, CF ₃ CH ₂ ], [RC11630; H, F, Cl, H, c-Pr, CF ₃ CF ₂ ], [RC11631; H, F, Cl, H, c-Pr, CF ₂ H] , [RC11632; H, F, Cl, H, c-Pr, CF ₂ HCF ₂ ], [RC11633; H, F, Cl, Cl, c-Pr, Me], [RC11634; H, F, C l, Cl, c-Pr, Et], [RC11635; H, F, Cl, Cl, c-Pr, Pr], [RC11636; H, F, Cl, Cl, c-Pr, i-Pr], [ RC11637; H, F, Cl, Cl, c-Pr, c-Pr], [RC11638; H, F, Cl, Cl, c-Pr, Bu], [RC11639; H, F, Cl, Cl, c- Pr, i-Bu], [RC11640; H, F, Cl, Cl, c-Pr, t-Bu], [RC11641; H, F, Cl, Cl, c-Pr, c-PrCH ₂ ], [RC11642 ; H, F, Cl, Cl, c-Pr, Ph], [RC11643; H, F, Cl, Cl, c-Pr, Bn], [RC11644; H, F, Cl, Cl, c-Pr, CF ₃ ], [RC11645; H, F, Cl, Cl, c-Pr, CF ₃ CH ₂ ], [RC11646; H, F, Cl, Cl, c-Pr, CF ₃ CF ₂ ], [RC11647; H, F, Cl, Cl, c-Pr, CF ₂ H], [RC11648; H, F, Cl, Cl, c-Pr, CF ₂ HCF ₂ ], [RC11649; H, F, H, H, Bn, Me ], [RC11650; H, F, H, H, Bn, Et], [RC11651; H, F, H, H, Bn, Pr], [RC11652; H, F, H, H, Bn, i-Pr ], [RC11653; H, F, H, H, Bn, c-Pr], [RC11654; H, F, H, H, Bn, Bu], [RC11655; H, F, H, H, Bn, i -Bu], [RC11656; H, F, H, H, Bn, t-Bu], [RC11657; H, F, H, H, Bn, c-PrCH ₂ ], [RC11658; H, F, H, H, Bn, Ph], [RC11659; H, F, H, H, Bn, Bn], [RC11660; H, F, H, H, Bn, CF ₃ ], [RC11661; H, F, H, H , Bn, CF ₃ CH ₂ ], [RC11662; H, F, H, H, Bn, CF ₃ CF ₂ ], [RC11663; H, F, H, H, Bn, CF ₂ H], [RC11664; H , F, H, H, Bn, CF ₂ HCF ₂ ], [RC11665; H, F, H, Me, Bn, Me], [RC11666; H, F, H, Me, Bn, Et], [RC11667; H, F, H, Me, Bn, Pr], [RC11668; H, F, H, Me, Bn, i-Pr], [RC11669; H, F, H , Me, Bn, c-Pr], [RC11670; H, F, H, Me, Bn, Bu], [RC11671; H, F, H, Me, Bn, i-Bu], [RC11672; H, F , H, Me, Bn, t-Bu], [RC11673; H, F, H, Me, Bn, c-PrCH ₂ ], [RC11674; H, F, H, Me, Bn, Ph], [RC11675; H, F, H, Me, Bn, Bn], [RC11676; H, F, H, Me, Bn, CF ₃ ], [RC11677; H, F, H, Me, Bn, CF ₃ CH ₂ ], [ RC11678; H, F, H, Me, Bn, CF ₃ CF ₂ ], [RC11679; H, F, H, Me, Bn, CF ₂ H], [RC11680; H, F, H, Me, Bn, CF ₂ HCF ₂ ], [RC11681; H, F, Me, Me, Bn, Me], [RC11682; H, F, Me, Me, Bn, Et], [RC11683; H, F, Me, Me, Bn, Pr], [RC11684; H, F, Me, Me, Bn, i-Pr], [RC11685; H, F, Me, Me, Bn, c-Pr], [RC11686; H, F, Me, Me, Bn, Bu], [RC11687; H, F, Me, Me, Bn, i-Bu], [RC11688; H, F, Me, Me, Bn, t-Bu], [RC11689; H, F, Me, Me, Bn, c-PrCH ₂ ], [RC11690; H, F, Me, Me, Bn, Ph], [RC11691; H, F, Me, Me, Bn, Bn], [RC11692; H, F, Me , Me, Bn, CF ₃ ], [RC11693; H, F, Me, Me, Bn, CF ₃ CH ₂ ], [RC11694; H, F, Me, Me, Bn, CF ₃ CF ₂ ], [RC11695; H, F, Me, Me, Bn, CF ₂ H], [RC11696; H, F, Me, Me, Bn, CF ₂ HCF ₂ ], [RC11697; H, F, Me, Et, Bn, Me], [RC11698; H, F, Me, Et, Bn, Et], [RC11699; H, F, Me, Et, Bn, Pr], [RC11700; H, F, Me, Et, Bn, i-Pr], [RC11701; H, F, Me, Et, Bn, c-Pr], [RC11702; H, F, Me, Et, Bn, Bu], [RC11703; H, F, Me, Et, Bn, i-Bu ], [RC11704; H, F, Me, Et , Bn, t-Bu], [RC11705; H, F, Me, Et, Bn, c-PrCH ₂ ], [RC11706; H, F, Me, Et, Bn, Ph], [RC11707; H, F, Me, Et, Bn, Bn], [RC11708; H, F, Me, Et, Bn, CF ₃ ], [RC11709; H, F, Me, Et, Bn, CF ₃ CH ₂ ], [RC11710; H, F, Me, Et, Bn, CF ₃ CF ₂ ], [RC11711; H, F, Me, Et, Bn, CF ₂ H], [RC11712; H, F, Me, Et, Bn, CF ₂ HCF ₂ ] , [RC11713; H, F, Me, F, Bn, Me], [RC11714; H, F, Me, F, Bn, Et], [RC11715; H, F, Me, F, Bn, Pr], [ RC11716; H, F, Me, F, Bn, i-Pr], [RC11717; H, F, Me, F, Bn, c-Pr], [RC11718; H, F, Me, F, Bn, Bu] , [RC11719; H, F, Me, F, Bn, i-Bu], [RC11720; H, F, Me, F, Bn, t-Bu], [RC11721; H, F, Me, F, Bn, c-PrCH ₂ ], [RC11722; H, F, Me, F, Bn, Ph], [RC11723; H, F, Me, F, Bn, Bn], [RC11724; H, F, Me, F, Bn , CF ₃ ], [RC11725; H, F, Me, F, Bn, CF ₃ CH ₂ ], [RC11726; H, F, Me, F, Bn, CF ₃ CF ₂ ], [RC11727; H, F, Me, F, Bn, CF ₂ H], [RC11728; H, F, Me, F, Bn, CF ₂ HCF ₂ ], [RC11729; H, F, Me, Cl, Bn, Me], [RC11730; H , F, Me, Cl, Bn, Et], [RC11731; H, F, Me, Cl, Bn, Pr], [RC11732; H, F, Me, Cl, Bn, i-Pr], [RC11733; H , F, Me, Cl, Bn, c-Pr], [RC11734; H, F, Me, Cl, Bn, Bu], [RC11735; H, F, Me, Cl, Bn, i-Bu], [RC11736 ; H, F, Me, Cl, Bn, t-Bu], [RC11737; H, F, Me, Cl, Bn, c-PrCH ₂ ], [RC11738; H, F, Me, Cl, Bn, Ph] , [RC11739; H, F, Me, Cl, Bn , Bn], [RC11740; H, F, Me, Cl, Bn, CF ₃ ], [RC11741; H, F, Me, Cl, Bn, CF ₃ CH ₂ ], [RC11742; H, F, Me, Cl , Bn, CF ₃ CF ₂ ], [RC11743; H, F, Me, Cl, Bn, CF ₂ H], [RC11744; H, F, Me, Cl, Bn, CF ₂ HCF ₂ ], [RC11745; H , F, Et, H, Bn, Me], [RC11746; H, F, Et, H, Bn, Et], [RC11747; H, F, Et, H, Bn, Pr], [RC11748; H, F , Et, H, Bn, i-Pr], [RC11749; H, F, Et, H, Bn, c-Pr], [RC11750; H, F, Et, H, Bn, Bu], [RC11751; H , F, Et, H, Bn, i-Bu], [RC11752; H, F, Et, H, Bn, t-Bu], [RC11753; H, F, Et, H, Bn, c-PrCH ₂ ] , [RC11754; H, F, Et, H, Bn, Ph], [RC11755; H, F, Et, H, Bn, Bn], [RC11756; H, F, Et, H, Bn, CF ₃ ], [RC11757; H, F, Et, H, Bn, CF ₃ CH ₂ ], [RC11758; H, F, Et, H, Bn, CF ₃ CF ₂ ], [RC11759; H, F, Et, H, Bn , CF ₂ H], [RC11760; H, F, Et, H, Bn, CF ₂ HCF ₂ ], [RC11761; H, F, Et, F, Bn, Me], [RC11762; H, F, Et, F, Bn, Et], [RC11763; H, F, Et, F, Bn, Pr], [RC11764; H, F, Et, F, Bn, i-Pr], [RC11765; H, F, Et, F, Bn, c-Pr], [RC11766; H, F, Et, F, Bn, Bu], [RC11767; H, F, Et, F, Bn, i-Bu], [RC11768; H, F, Et, F, Bn, t-Bu], [RC11769; H, F, Et, F, Bn, c-PrCH ₂ ], [RC11770; H, F, Et, F, Bn, Ph], [RC11771; H , F, Et, F, Bn, Bn], [RC11772; H, F, Et, F, Bn, CF ₃ ], [RC11773; H, F, Et, F, Bn, CF ₃ CH ₂ ], [RC11774 ; H, F, Et, F, Bn, CF ₃ CF ₂ ], [R C11775; H, F, Et, F, Bn, CF ₂ H], [RC11776; H, F, Et, F, Bn, CF ₂ HCF ₂ ], [RC11777; H, F, Et, Cl, Bn, Me ], [RC11778; H, F, Et, Cl, Bn, Et], [RC11779; H, F, Et, Cl, Bn, Pr], [RC11780; H, F, Et, Cl, Bn, i-Pr ], [RC11781; H, F, Et, Cl, Bn, c-Pr], [RC11782; H, F, Et, Cl, Bn, Bu], [RC11783; H, F, Et, Cl, Bn, i -Bu], [RC11784; H, F, Et, Cl, Bn, t-Bu], [RC11785; H, F, Et, Cl, Bn, c-PrCH ₂ ], [RC11786; H, F, Et, Cl, Bn, Ph], [RC11787; H, F, Et, Cl, Bn, Bn], [RC11788; H, F, Et, Cl, Bn, CF ₃ ], [RC11789; H, F, Et, Cl , Bn, CF ₃ CH ₂ ], [RC11790; H, F, Et, Cl, Bn, CF ₃ CF ₂ ], [RC11791; H, F, Et, Cl, Bn, CF ₂ H], [RC11792; H , F, Et, Cl, Bn, CF ₂ HCF ₂ ], [RC11793; H, F, F, H, Bn, Me], [RC11794; H, F, F, H, Bn, Et], [RC11795; H, F, F, H, Bn, Pr], [RC11796; H, F, F, H, Bn, i-Pr], [RC11797; H, F, F, H, Bn, c-Pr], [ RC11798; H, F, F, H, Bn, Bu], [RC11799; H, F, F, H, Bn, i-Bu], [RC11800; H, F, F, H, Bn, t-Bu] ,

[RC11801; H, F, F, H, Bn, c-PrCH ₂ ], [RC11802; H, F, F, H, Bn, Ph], [RC11803; H, F, F, H, Bn, Bn] , [RC11804; H, F, F, H, Bn, CF ₃ ], [RC11805; H, F, F, H, Bn, CF ₃ CH ₂ ], [RC11806; H, F, F, H, Bn, CF ₃ CF ₂ ], [RC11807; H, F, F, H, Bn, CF ₂ H], [RC11808; H, F, F, H, Bn, CF ₂ HCF ₂ ], [RC11809; H, F, F, F, Bn, Me], [RC11810; H, F, F, F, Bn, Et], [RC11811; H, F, F, F, Bn, Pr], [RC11812; H, F, F, F, Bn, i-Pr], [RC11813; H, F, F, F, Bn, c-Pr], [RC11814; H, F, F, F, Bn, Bu], [RC11815; H, F, F, F, Bn, i-Bu], [RC11816; H, F, F, F, Bn, t-Bu], [RC11817; H, F, F, F, Bn, c-PrCH ₂ ], [RC11818 ; H, F, F, F, Bn, Ph], [RC11819; H, F, F, F, Bn, Bn], [RC11820; H, F, F, F, Bn, CF ₃ ], [RC11821; H, F, F, F, Bn, CF ₃ CH ₂ ], [RC11822; H, F, F, F, Bn, CF ₃ CF ₂ ], [RC11823; H, F, F, F, Bn, CF ₂ H], [RC11824; H, F, F, F, Bn, CF ₂ HCF ₂ ], [RC11825; H, F, F, Cl, Bn, Me], [RC11826; H, F, F, Cl, Bn , Et], [RC11827; H, F, F, Cl, Bn, Pr], [RC11828; H, F, F, Cl, Bn, i-Pr], [RC11829; H, F, F, Cl, Bn , c-Pr], [RC11830; H, F, F, Cl, Bn, Bu], [RC11831; H, F, F, Cl, Bn, i-Bu], [RC11832; H, F, F, Cl , Bn, t-Bu], [RC11833; H, F, F, Cl, Bn, c-PrCH ₂ ], [RC11834; H, F, F, Cl, Bn, Ph], [RC11835; H, F, F, Cl, Bn, Bn], [RC11836; H, F, F, Cl, Bn, CF ₃ ], [RC11837; H, F, F, Cl, Bn , CF ₃ CH ₂ ], [RC11838; H, F, F, Cl, Bn, CF ₃ CF ₂ ], [RC11839; H, F, F, Cl, Bn, CF ₂ H], [RC11840; H, F , F, Cl, Bn, CF ₂ HCF ₂ ], [RC11841; H, F, Cl, H, Bn, Me], [RC11842; H, F, Cl, H, Bn, Et], [RC11843; H, F, Cl, H, Bn, Pr], [RC11844; H, F, Cl, H, Bn, i-Pr], [RC11845; H, F, Cl, H, Bn, c-Pr], [RC11846; H, F, Cl, H, Bn, Bu], [RC11847; H, F, Cl, H, Bn, i-Bu], [RC11848; H, F, Cl, H, Bn, t-Bu], [ RC11849; H, F, Cl, H, Bn, c-PrCH ₂ ], [RC11850; H, F, Cl, H, Bn, Ph], [RC11851; H, F, Cl, H, Bn, Bn], [RC11852; H, F, Cl, H, Bn, CF ₃ ], [RC11853; H, F, Cl, H, Bn, CF ₃ CH ₂ ], [RC11854; H, F, Cl, H, Bn, CF ₃ CF ₂ ], [RC11855; H, F, Cl, H, Bn, CF ₂ H], [RC11856; H, F, Cl, H, Bn, CF ₂ HCF ₂ ], [RC11857; H, F, Cl , Cl, Bn, Me], [RC11858; H, F, Cl, Cl, Bn, Et], [RC11859; H, F, Cl, Cl, Bn, Pr], [RC11860; H, F, Cl, Cl , Bn, i-Pr], [RC11861; H, F, Cl, Cl, Bn, c-Pr], [RC11862; H, F, Cl, Cl, Bn, Bu], [RC11863; H, F, Cl , Cl, Bn, i-Bu], [RC11864; H, F, Cl, Cl, Bn, t-Bu], [RC11865; H, F, Cl, Cl, Bn, c-PrCH ₂ ], [RC11866; H, F, Cl, Cl, Bn, Ph], [RC11867; H, F, Cl, Cl, Bn, Bn], [RC11868; H, F, Cl, Cl, Bn, CF ₃ ], [RC11869; H , F, Cl, Cl, Bn, CF ₃ CH ₂ ], [RC11870; H, F, Cl, Cl, Bn, CF ₃ CF ₂ ], [RC11871; H, F, Cl, Cl, Bn, CF ₂ H ], [RC11872; H, F, Cl, Cl, Bn, CF ₂ HCF ₂ ], [RC11873; H, F, H, H, Ph, Me], [RC11874; H, F, H, H, Ph, Et], [RC11875; H, F, H , H, Ph, Pr], [RC11876; H, F, H, H, Ph, i-Pr], [RC11877; H, F, H, H, Ph, c-Pr], [RC11878; H, F , H, H, Ph, Bu], [RC11879; H, F, H, H, Ph, i-Bu], [RC11880; H, F, H, H, Ph, t-Bu], [RC11881; H , F, H, H, Ph, c-PrCH ₂ ], [RC11882; H, F, H, H, Ph, Ph], [RC11883; H, F, H, H, Ph, Bn], [RC11884; H, F, H, H, Ph, CF ₃ ], [RC11885; H, F, H, H, Ph, CF ₃ CH ₂ ], [RC11886; H, F, H, H, Ph, CF ₃ CF ₂ ], [RC11887; H, F, H, H, Ph, CF ₂ H], [RC11888; H, F, H, H, Ph, CF ₂ HCF ₂ ], [RC11889; H, F, H, Me, Ph, Me], [RC11890; H, F, H, Me, Ph, Et], [RC11891; H, F, H, Me, Ph, Pr], [RC11892; H, F, H, Me, Ph, i-Pr], [RC11893; H, F, H, Me, Ph, c-Pr], [RC11894; H, F, H, Me, Ph, Bu], [RC11895; H, F, H, Me, Ph, i-Bu], [RC11896; H, F, H, Me, Ph, t-Bu], [RC11897; H, F, H, Me, Ph, c-PrCH ₂ ], [RC11898; H, F , H, Me, Ph, Ph], [RC11899; H, F, H, Me, Ph, Bn], [RC11900; H, F, H, Me, Ph, CF ₃ ], [RC11901; H, F, H, Me, Ph, CF ₃ CH ₂ ], [RC11902; H, F, H, Me, Ph, CF ₃ CF ₂ ], [RC11903; H, F, H, Me, Ph, CF ₂ H], [ RC11904; H, F, H, Me, Ph, CF ₂ HCF ₂ ], [RC11905; H, F, Me, Me, Ph, Me], [RC11906; H, F, Me, Me, Ph, Et], [RC11907; H, F, Me, Me, Ph, Pr], [RC11908; H, F, Me, Me, Ph, iP r], [RC11909; H, F, Me, Me, Ph, c-Pr], [RC11910; H, F, Me, Me, Ph, Bu], [RC11911; H, F, Me, Me, Ph, i-Bu], [RC11912; H, F, Me, Me, Ph, t-Bu], [RC11913; H, F, Me, Me, Ph, c-PrCH ₂ ], [RC11914; H, F, Me , Me, Ph, Ph], [RC11915; H, F, Me, Me, Ph, Bn], [RC11916; H, F, Me, Me, Ph, CF ₃ ], [RC11917; H, F, Me, Me, Ph, CF ₃ CH ₂ ], [RC11918; H, F, Me, Me, Ph, CF ₃ CF ₂ ], [RC11919; H, F, Me, Me, Ph, CF ₂ H], [RC11920; H, F, Me, Me, Ph, CF ₂ HCF ₂ ], [RC11921; H, F, Me, Et, Ph, Me], [RC11922; H, F, Me, Et, Ph, Et], [RC11923 ; H, F, Me, Et, Ph, Pr], [RC11924; H, F, Me, Et, Ph, i-Pr], [RC11925; H, F, Me, Et, Ph, c-Pr], [RC11926; H, F, Me, Et, Ph, Bu], [RC11927; H, F, Me, Et, Ph, i-Bu], [RC11928; H, F, Me, Et, Ph, t-Bu ], [RC11929; H, F, Me, Et, Ph, c-PrCH ₂ ], [RC11930; H, F, Me, Et, Ph, Ph], [RC11931; H, F, Me, Et, Ph, Bn], [RC11932; H, F, Me, Et, Ph, CF ₃ ], [RC11933; H, F, Me, Et, Ph, CF ₃ CH ₂ ], [RC11934; H, F, Me, Et, Ph, CF ₃ CF ₂ ], [RC11935; H, F, Me, Et, Ph, CF ₂ H], [RC11936; H, F, Me, Et, Ph, CF ₂ HCF ₂ ], [RC11937; H, F, Me, F, Ph, Me], [RC11938; H, F, Me, F, Ph, Et], [RC11939; H, F, Me, F, Ph, Pr], [RC11940; H, F, Me, F, Ph, i-Pr], [RC11941; H, F, Me, F, Ph, c-Pr], [RC11942; H, F, Me, F, Ph, Bu], [RC11943; H, F, Me, F, Ph, i- Bu], [RC11944; H, F, Me, F, Ph, t-Bu], [RC11945; H, F, Me, F, Ph, c-PrCH ₂ ], [RC11946; H, F, Me, F , Ph, Ph], [RC11947; H, F, Me, F, Ph, Bn], [RC11948; H, F, Me, F, Ph, CF ₃ ], [RC11949; H, F, Me, F, Ph, CF ₃ CH ₂ ], [RC11950; H, F, Me, F, Ph, CF ₃ CF ₂ ], [RC11951; H, F, Me, F, Ph, CF ₂ H], [RC11952; H, F, Me, F, Ph, CF ₂ HCF ₂ ], [RC11953; H, F, Me, Cl, Ph, Me], [RC11954; H, F, Me, Cl, Ph, Et], [RC11955; H , F, Me, Cl, Ph, Pr], [RC11956; H, F, Me, Cl, Ph, i-Pr], [RC11957; H, F, Me, Cl, Ph, c-Pr], [RC11958 ; H, F, Me, Cl, Ph, Bu], [RC11959; H, F, Me, Cl, Ph, i-Bu], [RC11960; H, F, Me, Cl, Ph, t-Bu], [RC11961; H, F, Me, Cl, Ph, c-PrCH ₂ ], [RC11962; H, F, Me, Cl, Ph, Ph], [RC11963; H, F, Me, Cl, Ph, Bn] , [RC11964; H, F, Me, Cl, Ph, CF ₃ ], [RC11965; H, F, Me, Cl, Ph, CF ₃ CH ₂ ], [RC11966; H, F, Me, Cl, Ph, CF ₃ CF ₂ ], [RC11967; H, F, Me, Cl, Ph, CF ₂ H], [RC11968; H, F, Me, Cl, Ph, CF ₂ HCF ₂ ], [RC11969; H, F, Et, H, Ph, Me], [RC11970; H, F, Et, H, Ph, Et], [RC11971; H, F, Et, H, Ph, Pr], [RC11972; H, F, Et, H, Ph, i-Pr], [RC11973; H, F, Et, H, Ph, c-Pr], [RC11974; H, F, Et, H, Ph, Bu], [RC11975; H, F, Et, H, Ph, i-Bu], [RC11976; H, F, Et, H, Ph, t-Bu], [RC11977; H, F, Et, H, Ph, c-PrCH ₂ ], [RC11978 ; H, F, Et, H, Ph, Ph], [R C11979; H, F, Et, H, Ph, Bn], [RC11980; H, F, Et, H, Ph, CF ₃ ], [RC11981; H, F, Et, H, Ph, CF ₃ CH ₂ ] , [RC11982; H, F, Et, H, Ph, CF ₃ CF ₂ ], [RC11983; H, F, Et, H, Ph, CF ₂ H], [RC11984; H, F, Et, H, Ph , CF ₂ HCF ₂ ], [RC11985; H, F, Et, F, Ph, Me], [RC11986; H, F, Et, F, Ph, Et], [RC11987; H, F, Et, F, Ph, Pr], [RC11988; H, F, Et, F, Ph, i-Pr], [RC11989; H, F, Et, F, Ph, c-Pr], [RC11990; H, F, Et, F, Ph, Bu], [RC11991; H, F, Et, F, Ph, i-Bu], [RC11992; H, F, Et, F, Ph, t-Bu], [RC11993; H, F, Et, F, Ph, c-PrCH ₂ ], [RC11994; H, F, Et, F, Ph, Ph], [RC11995; H, F, Et, F, Ph, Bn], [RC11996; H, F , Et, F, Ph, CF ₃ ], [RC11997; H, F, Et, F, Ph, CF ₃ CH ₂ ], [RC11998; H, F, Et, F, Ph, CF ₃ CF ₂ ], [ RC11999; H, F, Et, F, Ph, CF ₂ H], [RC12000; H, F, Et, F, Ph, CF ₂ HCF ₂ ],

[RC12001; H, F, Et, Cl, Ph, Me], [RC12002; H, F, Et, Cl, Ph, Et], [RC12003; H, F, Et, Cl, Ph, Pr], [RC12004 ; H, F, Et, Cl, Ph, i-Pr], [RC12005; H, F, Et, Cl, Ph, c-Pr], [RC12006; H, F, Et, Cl, Ph, Bu], [RC12007; H, F, Et, Cl, Ph, i-Bu], [RC12008; H, F, Et, Cl, Ph, t-Bu], [RC12009; H, F, Et, Cl, Ph, c -PrCH ₂ ], [RC12010; H, F, Et, Cl, Ph, Ph], [RC12011; H, F, Et, Cl, Ph, Bn], [RC12012; H, F, Et, Cl, Ph, CF ₃ ], [RC12013; H, F, Et, Cl, Ph, CF ₃ CH ₂ ], [RC12014; H, F, Et, Cl, Ph, CF ₃ CF ₂ ], [RC12015; H, F, Et , Cl, Ph, CF ₂ H], [RC12016; H, F, Et, Cl, Ph, CF ₂ HCF ₂ ], [RC12017; H, F, F, H, Ph, Me], [RC12018; H, F, F, H, Ph, Et], [RC12019; H, F, F, H, Ph, Pr], [RC12020; H, F, F, H, Ph, i-Pr], [RC12021; H, F, F, H, Ph, c-Pr], [RC12022; H, F, F, H, Ph, Bu], [RC12023; H, F, F, H, Ph, i-Bu], [RC12024; H, F, F, H, Ph, t-Bu], [RC12025; H, F, F, H, Ph, c-PrCH ₂ ], [RC12026; H, F, F, H, Ph, Ph], [RC12027; H, F, F, H, Ph, Bn], [RC12028; H, F, F, H, Ph, CF ₃ ], [RC12029; H, F, F, H, Ph, CF ₃ CH ₂ ], [RC12030; H, F, F, H, Ph, CF ₃ CF ₂ ], [RC12031; H, F, F, H, Ph, CF ₂ H], [RC12032; H, F, F, H, Ph, CF ₂ HCF ₂ ], [RC12033; H, F, F, F, Ph, Me], [RC12034; H, F, F, F, Ph, Et], [RC12035; H, F, F, F , Ph, Pr], [RC12036; H, F, F, F, Ph, i-Pr], [RC12037 ; H, F, F, F, Ph, c-Pr], [RC12038; H, F, F, F, Ph, Bu], [RC12039; H, F, F, F, Ph, i-Bu], [RC12040; H, F, F, F, Ph, t-Bu], [RC12041; H, F, F, F, Ph, c-PrCH ₂ ], [RC12042; H, F, F, F, Ph, Ph], [RC12043; H, F, F, F, Ph, Bn], [RC12044; H, F, F, F, Ph, CF ₃ ], [RC12045; H, F, F, F, Ph, CF ₃ CH ₂ ], [RC12046; H, F, F, F, Ph, CF ₃ CF ₂ ], [RC12047; H, F, F, F, Ph, CF ₂ H], [RC12048; H, F, F , F, Ph, CF ₂ HCF ₂ ], [RC12049; H, F, F, Cl, Ph, Me], [RC12050; H, F, F, Cl, Ph, Et], [RC12051; H, F, F, Cl, Ph, Pr], [RC12052; H, F, F, Cl, Ph, i-Pr], [RC12053; H, F, F, Cl, Ph, c-Pr], [RC12054; H, F, F, Cl, Ph, Bu], [RC12055; H, F, F, Cl, Ph, i-Bu], [RC12056; H, F, F, Cl, Ph, t-Bu], [RC12057; H, F, F, Cl, Ph, c-PrCH ₂ ], [RC12058; H, F, F, Cl, Ph, Ph], [RC12059; H, F, F, Cl, Ph, Bn], [RC12060 ; H, F, F, Cl, Ph, CF ₃ ], [RC12061; H, F, F, Cl, Ph, CF ₃ CH ₂ ], [RC12062; H, F, F, Cl, Ph, CF ₃ CF ₂ ], [RC12063; H, F, F, Cl, Ph, CF ₂ H], [RC12064; H, F, F, Cl, Ph, CF ₂ HCF ₂ ], [RC12065; H, F, Cl, H , Ph, Me], [RC12066; H, F, Cl, H, Ph, Et], [RC12067; H, F, Cl, H, Ph, Pr], [RC12068; H, F, Cl, H, Ph , i-Pr], [RC12069; H, F, Cl, H, Ph, c-Pr], [RC12070; H, F, Cl, H, Ph, Bu], [RC12071; H, F, Cl, H , Ph, i-Bu], [RC12072; H, F, Cl, H, Ph, t-Bu], [RC12073; H, F, Cl, H, Ph , c-PrCH ₂ ], [RC12074; H, F, Cl, H, Ph, Ph], [RC12075; H, F, Cl, H, Ph, Bn], [RC12076; H, F, Cl, H, Ph, CF ₃ ], [RC12077; H, F, Cl, H, Ph, CF ₃ CH ₂ ], [RC12078; H, F, Cl, H, Ph, CF ₃ CF ₂ ], [RC12079; H, F , Cl, H, Ph, CF ₂ H], [RC12080; H, F, Cl, H, Ph, CF ₂ HCF ₂ ], [RC12081; H, F, Cl, Cl, Ph, Me], [RC12082; H, F, Cl, Cl, Ph, Et], [RC12083; H, F, Cl, Cl, Ph, Pr], [RC12084; H, F, Cl, Cl, Ph, i-Pr], [RC12085; H, F, Cl, Cl, Ph, c-Pr], [RC12086; H, F, Cl, Cl, Ph, Bu], [RC12087; H, F, Cl, Cl, Ph, i-Bu], [ RC12088; H, F, Cl, Cl, Ph, t-Bu], [RC12089; H, F, Cl, Cl, Ph, c-PrCH ₂ ], [RC12090; H, F, Cl, Cl, Ph, Ph ], [RC12091; H, F, Cl, Cl, Ph, Bn], [RC12092; H, F, Cl, Cl, Ph, CF ₃ ], [RC12093; H, F, Cl, Cl, Ph, CF ₃ CH ₂ ], [RC12094; H, F, Cl, Cl, Ph, CF ₃ CF ₂ ], [RC12095; H, F, Cl, Cl, Ph, CF ₂ H], [RC12096; H, F, Cl, Cl, Ph, CF ₂ HCF ₂ ].

The present compound RA, the present compound RB, the present compound RC and the present compound RD are referred to as the present compound A.

The present compound or the present compound can be used in combination or in combination with a bactericidal active ingredient, an insecticidal active ingredient, an acaricidal active ingredient, a nematocidal active ingredient or a plant growth regulating ingredient (hereinafter collectively referred to as this ingredient). .
Treating a plant or soil with one or more selected from the group consisting of bactericidal active ingredients, insecticidal active ingredients, acaricidal active ingredients, nematicidal active ingredients and plant growth regulating ingredients, and a composition containing the compound of the present invention It is possible to control pests such as harmful arthropods, harmful linear animals, and plant pathogens. Moreover, this invention compound and this component can be applied separately and a pest can be controlled.
A bactericidal active ingredient is an ingredient used to protect plants from diseases caused by phytopathogenic fungi (filamentous fungi and bacteria). For example, it is prescribed by FRAC (Fungicide Resistance Action Committee) etc. Can be mentioned.
Examples of the insecticidal active ingredient, acaricidal active ingredient and nematocidal active ingredient include those prescribed by, for example, IRAC (Insecticide Resistance Action Committee).
The plant growth regulating component means a component that regulates plant growth, such as fruiting promotion and rooting promotion, and examples thereof include indole butyric acid.

Below, the example of the combination of this compound or this invention compound and this component is described. For example, tebuconazole + SX means a combination of tebuconazole and SX. The abbreviation SX means any one compound selected from Compound A. The numbers in parentheses represent CAS registration numbers.
Tebuconazole + SX, prothioconazole + SX, metconazole + SX, ipconazole + SX, triticonazole + SX, difenoconazole + SX, imazalil + SX triadimenol) + SX, tetraconazole + SX, flutriafol + SX, bromuconazole + SX, propiconazole + SX, mefentrifluconazole + SX, ipfentrifluconazole (SX) ipfentrifluconazole) + SX, epoxiconazole + SX, cyproconazole + SX, mandestrobin + SX, azoxystrobin + SX, pyraclostrobin + SX, trifloxystrobin ( trifloxystrobin) + SX, fluoxast Robin (fluoxastrobin) + SX, picoxystrobin (SX), fenamidone (fenamidone) + SX, dimoxystrobin (SX) + metominostrobin (SX), pyribencarb (SX), sedaxane (SX) Penflufen + SX, fluxapyroxad + SX, fluopyram + SX, benzovindiflupyr + SX, boscalid + SX, carboxin + SX, penthiopyrad + SX, flutolanil (flutolanil) + SX, bixafen + SX, pydiflumetofen + SX, 3-difluoromethyl-N- (7-fluoro-1,1,3-trimethylindan-4-yl) -1-methylpyrazole -4-carboxamide (1383809-87-7) + SX, N-cyclopropyl-3- (difluoromethyl) -5 Fluoro-N- (5-chloro-2-isopropylbenzyl) -1-methyl-1H-pyrazole-4-carboxamide (1255734-28-1) + SX, 3-difluoromethyl-1-methyl-N- (1,1 , 3-Trimethylindan-4-yl) pyrazole-4-carboxamide (141573-94-6) + SX, 3-difluoromethyl-1-methyl-N-[(3R) -1,1,3-trimethylindan-4 -Yl] pyrazole-4-carboxamide (1352994-67-2) + SX, metalaxyl + SX, metalaxyl-M + SX, metrafenone + SX, cyflufenamid + SX, proquinazid + SX, 3-chloro-5-phenyl-6-methyl-4- (2,6-difluorophenyl) pyridazine (1358061-55-8) + SX, 1- (2-{[1- (4-chlorophenyl) -1H-pi Zol-3-yl] oxymethyl} -3-methylphenyl) -4-methyl-1,4-dihydrotetrazol-5-one (1472649-01-6) + SX, 4- (2-bromo-4-fluorophenyl) ) -N- (2-chloro-6-fluorophenyl) -1,3-dimethyl-1H-pyrazol-5-amine (1362477-26-6) + SX, fenpicoxamid + SX, N '-( 2,5-dimethyl-4-phenoxyphenyl) -N-ethyl-N-methylmethanimidamide (1052688-31-9) + SX, isotianil + SX, oxolinic acid + SX, ferimzone + SX , Phthalide + SX, kasugamycin + SX, tebufloquin + SX, quinofumelin + SX, fenpyrazamine + SX, procymidone + SX, fludioxonil nil) + SX, tolclofos-methyl + SX, thiabendazole + SX, ethaboxam + SX, picarbutrazox + SX, oxathiapiprolin + SX, iminoctadine triacetate + SX, iminoctadine albesilate + SX, fenpropimorph + SX, fenpropidin + SX, spiroxamine + SX, chlorothalonil + SX, folpet + SX, captan ( captan + SX, thiram + SX, silthiofam + SX, mancozeb + SX, cartap + SX, clothianidin + SX, thiamethoxam + SX, imidacloprid + SX, thiacloprid + SX, thiacloprid + SX + SX, flupyradifurone + SX, Sulfoxaflor + SX, triflumezopyrim + SX, dicloromezotiaz + SX, beta-cyfluthrin + SX, tefluthrin + SX, fipronil + SX, chlorantraniliprolol (chlorantraniliprole) + SX, cyantraniliprole + SX, tetraniliprole + SX, thiodicarb + SX, carbofuran + SX, fluxametamide + SX, afoxolaner + SX, uralflner + SX, broflanilide + SX, abamectin + SX, fluensulfone + SX, fluazaindolizine + SX, tioxazafen + SX, (E) -N- {1-[(6-chloro Pyridin-3-yl) methyl] pyridine-2 (1H) Iridene} -2,2,2-trifluoroacetamide (1689566-03-7) + SX, Mycorrhizal Fungi + SX, Bacillus firmus + SX, Bacillus amyloliquefaciens (Bacillus) amyloliquefaciens) + SX, Pasteuria nishizawae + SX, Pasteuria penetrans + SX.

The ratio of the present compound or the present compound and the present component is not particularly limited, but is 1000: 1 to 1: 1000, 500: 500 by weight ratio (the present compound: the present component or the present compound: the present component). 1 to 1: 500, 100: 1 to 1: 100, 50: 1 to 1:50, 20: 1 to 1:20, 10: 1 to 1:10, 3: 1 to 1: 3, 1: 1 to 1: 500, 1: 1 to 1: 100, 1: 1 to 1:50, 1: 1 to 1:20, 1: 1 to 1:10, and the like.

By treating the present compound or the present compound with a plant, improvement of seedling establishment rate, increase in the number of healthy leaves, increase in plant height, increase in plant weight, increase in leaf area, increase in the number or weight of seeds or fruits, number of flowers or The effect of promoting the growth of plants, such as an increase in the number of fruits and an increase in root growth, can be obtained. Moreover, by treating the present compound or the present compound with a plant, resistance to temperature stress such as high temperature stress or low temperature stress, moisture stress such as drought stress or excessive humidity stress, or abiotic stress such as salt stress is improved. Is done.

Next, formulation examples are shown. In the preparation examples, “part” means “part by weight”.

Formulation Example 1 A formulation is obtained by thoroughly pulverizing and mixing 50 parts of any one of the present compounds A, 3 parts of calcium lignin sulfonate, 2 parts of magnesium lauryl sulfate and 45 parts of wet silica.

Formulation Example 2 After mixing 20 parts of any one of the present compounds A and 1.5 parts of sorbitan trioleate with 28.5 parts of an aqueous solution containing 2 parts of polyvinyl alcohol, To this, 40 parts of an aqueous solution containing 0.05 part of xanthan gum and 0.1 part of aluminum magnesium silicate is added, and further 10 parts of propylene glycol is added and stirred to obtain a preparation.

Formulation Example 3 A formulation is obtained by thoroughly crushing and mixing 2 parts of any one of the present compounds A, 88 parts of kaolin clay and 10 parts of talc.

Formulation Example 4 A formulation is obtained by thoroughly mixing 5 parts of any one of the present compounds A, 14 parts of polyoxyethylene styryl phenyl ether, 6 parts of calcium dodecylbenzenesulfonate and 75 parts of xylene.

Formulation Example 5 After thoroughly mixing 2 parts of any one of the present compounds A, 1 part of wet silica, 2 parts of calcium lignin sulfonate, 30 parts of bentonite and 65 parts of kaolin clay, add water and knead well. The preparation is obtained by grain drying.

Formulation Example 6 A mixture of 35 parts of a mixture of polyoxyethylene alkyl ether sulfate ammonium salt and wet silica (weight ratio 1: 1), 20 parts of any one of the present compounds A, and 45 parts of water is sufficiently mixed. Get.

Next, test examples are shown. The untreated section in Test Example 1 or Test Example 2 is a test conducted under the same conditions as described in each test example except that dimethyl sulfoxide was dispensed instead of the dimethyl sulfoxide diluting solution containing this compound. Represents a ward. The term “no treatment” in Test Example 3 to Test Example 15 means that the foliage spraying of the water-diluted solution of the preparation containing the present compound was not performed.

Test Example 1 Control test against tomato leaf mold fungus (Cladosporium fulvum) Compound 2, 6, 8, 9, 11, 14, 19, 21, 26, 28, 33-37, 39, 46, 49, 51, 56 of the present invention , 63 or 64 is diluted with dimethyl sulfoxide so as to contain 1500 ppm, and 1 μL is dispensed into a titer plate (96-well), and then the tomato leaf blight fungus (cytochrome b encoding gene 129th of cytochrome b) 150 μL of a potato broth liquid medium (PDB medium) inoculated with spores of a QoI resistant strain whose nucleotide sequence was mutated so that the amino acid residue was substituted from phenylalanine to leucine was dispensed. This plate was cultured at 18 ° C. for 5 days to proliferate the tomato leaf mold, and then the absorbance at 550 nm of each well of the titer plate was measured, and the value was taken as the growth degree of the tomato leaf mold. As a result, the degree of growth in the section treated with the compound 2, 6, 8, 9, 11, 14, 19, 21, 26, 28, 33-37, 39, 46, 49, 51, 56, 63 or 64 of the present invention. All were 40% or less of the degree of growth in the untreated section.

Test Example 2 Control Test Against Wheat Leaf Blight Fungus (Septoria tritici) Compound 2, 4, 9, 12, 15-18, 22-27, 30, 33-40, 42, 46, 50, 56, 61, 63 of the present invention Alternatively, after diluting with dimethyl sulfoxide to contain 1500 ppm of 64 and dispensing 1 μL into a titer plate (96 well), 150 μL of potato broth liquid medium (PDB medium) inoculated with wheat leaf blight fungus spores in advance is dispensed. did. This plate was cultured at 18 ° C. for 5 days to grow wheat leaf blight fungi. Then, the absorbance at 550 nm of each well of the titer plate was measured, and the value was taken as the growth degree of wheat leaf blight fungi. As a result, the growth degree in the section treated with the compound 2, 4, 9, 12, 15-18, 22-27, 30, 33-40, 42, 46, 50, 56, 61, 63 or 64 of the present invention is increased. Was 40% or less of the degree of growth in the untreated area.

Test Example 3 Control Test for Soybean Rust (Phakopsora pachyrhizi) A plastic pot was filled with soil, and then soybean (cultivar; Kurosengoku) was sown there, grown in a greenhouse for 10 days, and an aqueous suspension of soybean rust fungus spores. Was spray-inoculated. After inoculation, the present compound 1 was formulated according to the method described in Formulation Example 6 after placing soybeans in a humid room at 23 ° C. in the daytime and 20 ° C. for 1 day in a humid room and then cultivating in the greenhouse for 2 days. -7, 9-26, 28-46, 49-51, 53, 56-59, 61, 63, 64 or the present compound 1 is mixed with water to a concentration of 200 ppm, The foliage was sprayed so as to adhere well to the leaf surface. After spraying, the soybeans were air-dried and cultivated in a greenhouse for 8 days, and then the lesion area was examined. As a result, there was no lesion area in soybeans treated with the present compounds 1-7, 9-26, 28-46, 49-51, 53, 56-59, 61, 63, 64 or the present compound 1. It was 30% or less of the lesion area in the treated soybean.

Test Example 4 Control test against soybean rust (Phakopsora pachyrhizi) A plastic pot was filled with soil, and soybean (cultivar; Kurosengoku) was sown therein and allowed to grow in a greenhouse for 13 days. The present compounds 1-26, 28-44, 46-59, 61-64 or the present compound 1 formulated according to the method described in Formulation Example 6 is mixed with water to a concentration of 200 ppm, The mixture was sprayed on the foliage so that it sufficiently adhered to the leaf surface of the soybean. After spraying, the soybeans were air-dried, and after 4 days, sprayed with a water suspension of soybean rust spores. After inoculation, soybeans were placed in a humid room at 23 ° C. in the daytime and at 20 ° C. for one day under high humidity, then cultivated in the greenhouse for 14 days, and then the lesion area was examined. As a result, the lesion area in the soybean treated with the present compounds 1-26, 28-44, 46-59, 61-64 or the present compound 1 was 30% or less of the lesion area in the untreated soybean. there were.

Test Example 5 Control test against rice blast (Magnaporthe grisea) A plastic pot was filled with soil, rice (cultivar: Hinohikari) was sown there, and cultivated in a greenhouse for 20 days. The compound 1, 4, 5, 6, 37, 43 or 44 of the present invention formulated according to the method described in Formulation Example 6 is mixed with water to a concentration of 500 ppm, and the mixture is mixed with the above rice The foliage was sprayed so as to adhere well to the leaf surface. After spraying, the rice is air-dried and left for 6 days in contact with a rice seedling (variety: Hinohikari) that has been treated with the rice blast fungus under a high humidity of 24 ° C in the daytime and 20 ° C in the nighttime. The lesion area was investigated. As a result, the lesion area in the rice treated with the present compound 1, 4, 5, 6, 37, 43 or 44 was 30% or less of the lesion area in the untreated rice.

Test Example 6 Control test against rice blast (Magnaporthe grisea) A plastic pot was filled with soil, rice (cultivar: Hinohikari) was sown there, and cultivated in a greenhouse for 20 days. Thereafter, the present compound 2, 5, 14, 15, 19, 31, 34, 43, 44 or 46 formulated according to the method described in Formulation Example 6 is mixed with water so that the concentration becomes 200 ppm. The mixture was sprayed on the foliage so that it sufficiently adhered to the leaf surface of the rice. After spraying, the rice is air-dried and left for 6 days in contact with a rice seedling (variety: Hinohikari) that has been treated with the rice blast fungus under a high humidity of 24 ° C in the daytime and 20 ° C in the nighttime. The lesion area was investigated. As a result, the lesion area in the rice treated with the present compound 2, 5, 14, 15, 19, 31, 34, 43, 44 or 46 is 30% or less of the lesion area in the untreated rice. there were.

Test Example 7 Control test against wheat leaf blight (Septoria tritici) A plastic pot was filled with soil, and wheat (cultivar; Apoge) was sown therein and cultivated in a greenhouse for 10 days. The present compound 1-7, 9-18, 22-24, 38, 43 or the present compound 1 formulated according to the method described in Formulation Example 6 is mixed with water so that the concentration becomes 500 ppm, The mixture was sprayed on the foliage so as to adhere well to the leaf surface of the wheat. After spraying, the wheat was air-dried, and after 4 days, a water suspension containing spores of wheat leaf blight was spray-inoculated. After inoculation, the wheat was placed under high humidity at 18 ° C. for 3 days, then cultivated under illumination for 14 to 18 days, and then the lesion area was examined. As a result, the lesion area in the wheat treated with the present compounds 1-7, 9-18, 22-24, 38, 43 or the present compound 1 was 30% or less of the lesion area in the untreated wheat. there were.

Test Example 8 Control test against wheat leaf blight (Septoria tritici) A plastic pot was filled with soil, and wheat (cultivar; Apoge) was sown therein and cultivated in a greenhouse for 10 days. Compound 1, 2, 6, 9-20, 22-24, 26, 28-34, 38, 44, 46, 48, 50, 51, 53 of the present invention formulated according to the method described in Formulation Example 6 ~ 59, 63, or 64 was mixed with water to a concentration of 200 ppm, and the mixture was sprayed on the foliage so as to adhere well to the leaf surface of the wheat. After spraying, the wheat was air-dried, and after 4 days, a water suspension containing spores of wheat leaf blight was spray-inoculated. After inoculation, the wheat was placed under high humidity at 18 ° C. for 3 days, then cultivated under illumination for 14 to 18 days, and then the lesion area was examined. As a result, in wheat treated with the compounds 1, 2, 6, 9-20, 22-24, 26, 28-34, 38, 44, 46, 48, 50, 51, 53-59, 63 or 64 of the present invention. The lesion area was 30% or less of the lesion area in untreated wheat.

Test Example 9 Control test against wheat leaf blight (Septoria tritici) A plastic pot was filled with soil, seeded with wheat (variety; apoge), cultivated in a greenhouse for 10 days, and water suspension of wheat leaf blight fungus spores The solution was spray inoculated. After inoculation, the wheat was placed under high humidity at 18 ° C. for 3 days, and then the compound 9 of the present invention formulated according to the method described in Formulation Example 6 was mixed with water to a concentration of 200 ppm. The foliage was sprayed so as to adhere well to the leaf surface of the wheat. After spraying, the wheat was air-dried and placed under illumination for 14 to 18 days, and then the lesion area was examined. As a result, the lesion area in the wheat treated with Compound 9 of the present invention was 30% or less of the lesion area in the untreated wheat.

Test Example 10 Control test against wheat rust (Puccinia recondita) A plastic pot was stuffed with soil, seeded with wheat (cultivar: Shirogane), and cultivated in a greenhouse for 9 days. The present compound 1-7, 9-18, 22-25, 27-29, 37, 38, 40, 42-44 or the present compound 1 formulated according to the method described in Formulation Example 6 at a concentration of 500 ppm Then, the mixture was sprayed with foliage so as to adhere well to the leaf surface of the wheat. After spraying, the wheat was air-dried and cultivated under light at 20 ° C. for 5 days, and then sprinkled with spores of wheat rust fungus. After inoculation, the wheat was placed in a dark and humid environment at 23 ° C. for 1 day, and then cultivated at 20 ° C. for 8 days under illumination. As a result, the lesion areas in the wheat treated with the present compounds 1-7, 9-18, 22-25, 27-29, 37, 38, 40, 42-44 or the present compound 1 were all untreated. It was 30% or less of the lesion area in wheat.

Test Example 11 Control test against wheat rust (Puccinia recondita) A plastic pot was stuffed with soil, seeded with wheat (cultivar: Shirogane), and cultivated in a greenhouse for 9 days. Compounds of the present invention 1, 4, 6, 9 to 26, 28 to 31, 37, 38, 42 to 44, 46 to 48, 51 to 54, 56 to 59 formulated according to the method described in Formulation Example 6 61-64 or the present compound 1 was mixed with water to a concentration of 200 ppm, and the mixture was sprayed on the foliage so as to adhere well to the leaf surface of the wheat. After spraying, the wheat was air-dried and cultivated under light at 20 ° C. for 5 days, and then sprinkled with spores of wheat rust fungus. After inoculation, the wheat was placed in a dark and humid environment at 23 ° C. for 1 day, and then cultivated at 20 ° C. for 8 days under illumination. As a result, the present compound 1, 4, 6, 9 to 26, 28 to 31, 37, 38, 42 to 44, 46 to 48, 51 to 54, 56 to 59, 61 to 64 or the present compound 1 was treated. The lesion area in wheat was 30% or less of the lesion area in untreated wheat.

Test Example 12 Control test against soybean powdery mildew (Microsphaera diffusa) A plastic pot was filled with soil, and then soybean (cultivar; Kurosengoku) was sown, cultivated in a greenhouse for 10 days, and soybean affected with soybean powdery mildew The seedlings (variety: Kurosengoku) were sprinkled and inoculated. Soybeans are cultivated in a greenhouse at 24 ° C. during the daytime and 20 ° C. during the night for 2 days, and then formulated according to the method described in Formulation Example 6, Compounds 1, 4-6, 10-20, 22-29, 31 of the present invention. , 33, 34, 37, 38, 42, 46, 50, 58, 61, 63 or this compound 1 is mixed with water to a concentration of 200 ppm, and the mixture adheres sufficiently to the leaf surface of the soybean. So that the foliage was sprayed. After spraying, the soybean was air-dried and cultivated in a greenhouse for 9 days, and then the lesion area was examined. As a result, the present compound 1, 4-6, 10-20, 22-29, 31, 33, 34, 37, 38, 42, 46, 50, 58, 61, 63 or soybean treated with the present compound 1 The lesion area was 30% or less of the lesion area in untreated soybean.

Test Example 13 Control test against soybean powdery mildew (Microsphaera diffusa) A plastic pot was filled with soil, and then soybean (cultivar; Kurosengoku) was sown therein and cultivated in a greenhouse for 13 days. The present compound 1, 5, 6, 10 to 18, 22, 23, 28, 37 or 38 formulated according to the method described in Formulation Example 6 is mixed with water so that the concentration becomes 200 ppm, The mixture was sprayed on the foliage so that it sufficiently adhered to the leaf surface of the soybean. After spraying, the soybeans were air-dried, and one day later, they were sprinkled with spores of soybean seedlings (variety: Kurosengoku) afflicted with soybean powdery mildew. After inoculation, soybeans were cultivated in a greenhouse at 24 ° C. during the day and 20 ° C. during the night for 11 days, and then the lesion area was examined. As a result, the lesion area in the soybean treated with the compound 1, 5, 6, 10 to 18, 22, 23, 28, 37 or 38 of the present invention was 30% or less of the lesion area in the untreated soybean. there were.

Test Example 14 Pyrephorophora teres control test A plastic pot was filled with soil, and barley (cultivar: Nishinohoshi) was sown therein and cultivated in a greenhouse for 7 days. The compound 6, 9, 11, 14, 18 or 24 of the present invention formulated according to the method described in Formulation Example 6 is mixed with water to a concentration of 500 ppm, and the mixture is mixed with the above-mentioned barley leaves. The foliage was sprayed so as to adhere well to the surface. After spraying, the barley was air-dried, and two days later, a water suspension of barley reticular fungus spores was spray-inoculated. After inoculation, the barley was placed under high humidity in a greenhouse at 23 ° C. during the daytime and 20 ° C. during the night for 3 days and then cultivated in the greenhouse for 7 days. As a result, the lesion area in the barley treated with the present compound 6, 9, 11, 14, 18 or 24 was 30% or less of the lesion area in the untreated barley.

Test Example 15
The compound 1, 40, 41 or 45 of the present invention formulated according to the method described in Formulation Example 6 was mixed with water so that the concentration was 500 ppm. The mixture was sprayed on the foliage so that it sufficiently adhered to the leaf surface of the cabbage seedling (second to third leaf development stage) planted in the container. After spraying, the cabbage was air-dried, and the stems and leaves of this seedling were cut out and placed in a container with filter paper. To this, five 5th instar larvae were released. After 5 days, the number of live insects was counted, and the death rate was calculated from the following formula.
Death rate% = (1−Number of surviving insects / 5) × 100
As a result, the death rate when the present compound 1, 40, 41 or 45 was treated was 80% or more.

This compound has a controlling effect against plant diseases and can be used for controlling plant diseases.

Claims (8)

1. Formula (I)
   

   

   [Where,
   G is a thiophene ring, furan ring, pyrrole ring, imidazole ring, oxazole ring, isoxazole ring, thiazole ring, isothiazole ring, oxadiazole ring, thiadiazole ring, pyrazole ring, pyridine ring, pyrazine ring, pyridazine ring, pyrimidine Ring or benzene ring {the thiophene ring, the furan ring, the pyrrole ring, the imidazole ring, the oxazole ring, the isoxazole ring, the thiazole ring, the isothiazole ring, the pyrazole ring, the pyridine ring, the pyrazine ring , The pyridazine ring, the pyrimidine ring and the benzene ring each may have one or more substituents selected from group D}
   n represents 1, 2, 3 or 4;
   when n is 2, 3 or 4, the plurality of R ¹ and the plurality of R ² are the same or different,
   The combination of L, X and R ² is
   L is C (O), X is a single bond, NR ³ or an oxygen atom, and R ² is a C1-C6 alkyl group optionally having one or more substituents selected from group A, group A C1-C6 alkoxy group optionally having one or more substituents selected from B, a phenyl group optionally having one or more substituents selected from Group D, one or more selected from Group D An optionally substituted 5-6 membered aromatic heterocyclic group, one or more substituents selected from group D, a C3-C6 cycloalkyl group, a hydrogen atom, a halogen atom or cyano A combination that is a group, or
   L is S (O) ₂ , X is NR ³ or an oxygen atom, R ² is a C1-C6 alkyl group optionally having one or more substituents selected from group A, from group B A C1-C6 alkoxy group optionally having one or more substituents selected, a phenyl group optionally having one or more substituents selected from Group D, one or more substituents selected from Group D A combination of a 5- to 6-membered aromatic heterocyclic group optionally having one or more, a C3-C6 cycloalkyl group optionally having one or more substituents selected from Group D, a halogen atom or a cyano group Represent,
   R ¹ is a C1-C6 alkyl group optionally having one or more substituents selected from group A, a C1-C6 alkoxy group optionally having one or more substituents selected from group B, A phenyl group optionally having one or more substituents selected from group D, a 5-6-membered aromatic heterocyclic group optionally having one or more substituents selected from group D, from group D Represents a C3-C6 cycloalkyl group optionally having one or more selected substituents, a hydrogen atom, a halogen atom or a cyano group,
   R ¹ and R ^2, together with the carbon atoms to which they are attached, 3-7 membered cycloalkylene group, or 3-7-membered saturated heterocyclic ring (wherein 3-7 membered cycloalkylene group, and 3-7-membered saturated heterocyclic The ring may have one or more substituents selected from group D),
   R ³ is a C1-C6 alkyl group optionally having one or more substituents selected from group A, a C3-C6 alkenyl group optionally having one or more substituents selected from group A, A C3-C6 alkynyl group optionally having one or more substituents selected from group A, a C1-C6 alkoxy group optionally having one or more halogen atoms, one or more substituents selected from group D A C3-C6 cycloalkyl group optionally having a group, a phenyl group optionally having one or more substituents selected from group D, and one or more substituents selected from group D May represent a 5-6 membered aromatic heterocyclic group or a hydrogen atom,
   Z is a C3-C6 cycloalkyl group, a phenyl group, a 5-6 membered aromatic heterocyclic group, a 3-6 membered non-aromatic heterocyclic group (the C3-C6 cycloalkyl group, the phenyl group, the 5-6 And the 3-6-membered non-aromatic heterocyclic group may have one or more substituents selected from group D), CR ⁴ R ⁵ R ⁶ , NR ⁷ R Represents ⁸ or OR ⁹ or
   X and Z together with L to which they are attached form a 4-7 membered heterocycle (the 4-7 membered heterocycle may have one or more substituents selected from group D) You may,
   R ⁴ , R ⁵ and R ⁶ are the same or different and are a C1-C6 alkyl group optionally having one or more substituents selected from the group consisting of Group A and Group E, 1 selected from Group A A C3-C6 alkenyl group optionally having one or more substituents, a C3-C6 alkynyl group optionally having one or more substituents selected from group A, and one or more substituents selected from group B A C1-C6 alkoxy group which may have, a C3-C6 cycloalkyl group which may have one or more substituents selected from group D, and one or more substituents selected from group D An optionally substituted phenyl group, a 5-6 membered aromatic heterocyclic group optionally having one or more substituents selected from group D, a hydrogen atom, a halogen atom or a cyano group;
   R ⁷ and R ⁸ are the same or different and are each a C1-C6 alkyl group optionally having one or more substituents selected from the group consisting of group A and group E; one or more substituents selected from group A A C3-C6 alkenyl group which may have a group, a C3-C6 alkynyl group which may have one or more substituents selected from group A, and a C1 which may have one or more halogen atoms -C6 alkoxy group, C3-C6 cycloalkyl group optionally having one or more substituents selected from group D, phenyl group optionally having one or more substituents selected from group D, group Represents a 5- or 6-membered aromatic heterocyclic group which may have one or more substituents selected from D or a hydrogen atom, or R ⁷ and R ⁸ together with the nitrogen atom to which they are bonded 3-8 membered heterocycle (the 3-8 membered heterocycle is group D It may form may also be) have one or more substituents selected,
   R ⁹ may have one or more substituents selected from the group consisting of group A and group E, and may have one or more substituents selected from group A. C3-C6 alkenyl group, C3-C6 alkynyl group optionally having one or more substituents selected from group A, C3-C6 cyclo optionally having one or more substituents selected from group D An alkyl group, a phenyl group optionally having one or more substituents selected from group D, a 5-6-membered aromatic heterocyclic group optionally having one or more substituents selected from group D, or Represents a hydrogen atom.
   Group A: a C1-C6 alkoxy group optionally having one or more halogen atoms, a C1-C6 alkylthio group optionally having one or more halogen atoms, one or more substituents selected from group C A C3-C6 cycloalkyl group which may have, a phenyl group which may have one or more substituents selected from group F, and one or more substituents selected from group F. A group consisting of a 5-6 membered aromatic heterocyclic group, a halogen atom, a nitro group and a cyano group.
   Group B: C1-C6 alkylthio group optionally having one or more halogen atoms, phenyl group optionally having one or more substituents selected from Group F, one or more substituents selected from Group F A group consisting of a 5-6-membered aromatic heterocyclic group, a halogen atom, a nitro group and a cyano group, which may have a group;
   Group C: Group consisting of halogen atom, nitro group and cyano group.
   Group D: a C1-C6 alkyl group optionally having one or more substituents selected from group C, a C3-C6 cycloalkyl group optionally having one or more substituents selected from group C, C1-C6 alkoxy group which may have one or more halogen atoms, C3-C6 alkenyloxy group which may have one or more halogen atoms, C3 which may have one or more halogen atoms -C6 alkynyloxy group, C1-C6 alkylthio group optionally having one or more halogen atoms, C1-C6 alkylsulfonyloxy group optionally having one or more halogen atoms, halogen atom, cyano group, A group consisting of a nitro group, a hydroxy group and an amino group.
   Group E: (C1-C6 alkyl) carbonylamino group optionally having one or more substituents selected from group C, or one or more substituents selected from group C (C1-C6) C6 alkyl) aminocarbonyl group, di (C1-C6 alkyl) aminocarbonyl group optionally having one or more substituents selected from group C, having one or more substituents selected from group C A C1-C6 alkylsulfonylamino group, a C1-C6 alkylaminosulfonyl group optionally having one or more substituents selected from group C, and one or more substituents selected from group C. A group consisting of a di (C1-C6 alkyl) aminosulfonyl group, a hydroxy group and an amino group.
   Group F: a group consisting of a C1-C6 alkyl group optionally having one or more halogen atoms, a C1-C6 alkoxy group optionally having one or more halogen atoms, a halogen atom and a cyano group. ]
   The plant disease control method by processing the compound shown by a plant or soil.
2. Formula (II)
   

   

   [Where,
   G ^X represents thiophene ring, furan ring, pyrrole ring, imidazole ring, oxazole ring, isoxazole ring, thiazole ring, isothiazole ring, oxadiazole ring, thiadiazole ring, pyrazole ring, pyridine ring, pyrazine ring, pyridazine ring, Pyrimidine ring or benzene ring {the thiophene ring, the furan ring, the pyrrole ring, the imidazole ring, the oxazole ring, the isoxazole ring, the thiazole ring, the isothiazole ring, the pyrazole ring, the pyridine ring, the pyrazine The ring, the pyridazine ring, the pyrimidine ring, and the benzene ring may have one or more substituents selected from the group D ^X },
   m represents 1, 2, 3 or 4;
   when m is 2, 3 or 4, a plurality of R ^1X and a plurality of R ^2X are the same or different, respectively,
   The combination of L ^X, X ^X and R ^2X is
   L ^X is C (O), X ^X is NR ^3X or an oxygen atom, R ^2X is a C1-C6 alkyl group optionally having one or more substituents selected from group A ^X , 1 or more substituents optionally may C1-C6 alkoxy group which may have a phenyl group which may have one or more substituents selected from the group D ^X selected from B ^X, is selected from the group D ^X A 5-6 membered aromatic heterocyclic group optionally having one or more substituents, a C3-C6 cycloalkyl group optionally having one or more substituents selected from the group D ^X , a hydrogen atom, A combination that is a halogen atom or a cyano group, or
   L ^X is S (O) ₂ , X ^X is NR ^3X or an oxygen atom, and R ^2X may have one or more substituents selected from group A ^X , 1 or more substituents optionally may C1-C6 alkoxy group which may have a phenyl group which may have one or more substituents selected from the group D ^X selected from the group B ^X, selected from the group D ^X A 5- or 6-membered aromatic heterocyclic group optionally having one or more substituents, a C3-C6 cycloalkyl group optionally having one or more substituents selected from group D ^X , a halogen atom Or represents a combination that is a cyano group,
   R ^1X is one or more substituents optionally may be C1-C6 alkyl group optionally having a one or more substituents may C1-C6 alkoxy which may have a selected from the group B ^X selected from the group A ^X group, one or more substituents phenyl group which may have a one or more substituents may be a 5-6 membered aromatic heterocyclic group selected from the group D ^X is selected from the group D ^X represents one or more substituents optionally may be C3-C6 cycloalkyl group having a hydrogen atom, a halogen atom or a cyano group selected from the group D ^X,
   R ^1X and R ^2X , together with the carbon atom to which they are attached, represent a 3-7 membered cycloalkylene group or a 3-7 membered saturated heterocycle (the 3-7 membered cycloalkylene group and 3-7 membered saturated heterocycle). The ring may have one or more substituents selected from group D ^X ),
   R ^3X is one or more substituents optionally may C1-C6 alkyl group which may have one or more substituents may C3-C6 alkenyl which may have a selected from the group A ^X selected from the group A ^X A group, a C3-C6 alkynyl group optionally having one or more substituents selected from group A ^X , a C1-C6 alkoxy group optionally having one or more halogen atoms, selected from group D ^X 1 or may C3-C6 have a substituent of the cycloalkyl group, one or more substituents phenyl group which may have a selected from the group D ^X, one or more substituents selected from the group D ^X A 6-membered aromatic heterocyclic group which may have a group or a hydrogen atom,
   Z ^X represents C3-C6 cycloalkyl group, phenyl group, 6-membered aromatic heterocyclic group, 3-6-membered non-aromatic heterocyclic group, pyrazol-4-yl group, thienyl group, furyl group, imidazolyl group, oxazolyl Group, isoxazolyl group, thiazolyl group, isothiazolyl group, oxadiazolyl group, thiadiazolyl group (the C3-C6 cycloalkyl group, the phenyl group, the 6-membered aromatic heterocyclic group, the 3-6-membered non-aromatic heterocyclic group, The pyrazol-4-yl group, the thienyl group, the furyl group, the imidazolyl group, the oxazolyl group, the isoxazolyl group, the thiazolyl group, the isothiazolyl group, the oxadiazolyl group, and the thiadiazolyl group are selected from the group D ^X Or may represent one or more substituents), CR ^4X R ^5X R ^6X , NR ^7X R ^8X or OR ^9X , or
   X ^X and Z ^X together with L ^{X to} which they are bonded have a 4-7 membered heterocycle (the 4-7 membered heterocycle may have one or more substituents selected from group D ^X Good)
   R ^4X, R ^5X and R ^6X are identical or different phases, one or more substituents optionally may C1-C6 alkyl group which may have a selected from the group consisting of the group A ^X and the group E ^X, from the group A ^X C3-C6 alkenyl group optionally having one or more substituents selected, C3-C6 alkynyl group optionally having one or more substituents selected from group A ^X , selected from group B ^X 1 or more substituents optionally may C1-C6 alkoxy group which may have one or more substituents may be a C3-C6 cycloalkyl group selected from the group D ^X, 1 is selected from the group D ^X A phenyl group optionally having the above substituents, a 5-6 membered aromatic heterocyclic group optionally having one or more substituents selected from the group D ^X , a hydrogen atom, a halogen atom or a cyano group Represents
   R ^7X and R ^8X are the same or different and are a C1-C6 alkyl group optionally having one or more substituents selected from the group consisting of group A ^X and group E ^X , 1 selected from group A ^X or more substituents may have a C3-C6 alkenyl group, one or more substituents optionally may C3-C6 alkynyl group which may have a selected from the group a ^X, have one or more halogen atoms it may also be C1-C6 alkoxy group, one or more substituents the have optionally may C3-C6 cycloalkyl group selected from the group D ^X, have one or more substituents selected from the group D ^X Or a phenyl group, a 5- or 6-membered aromatic heterocyclic group which may have one or more substituents selected from the group D ^X or a hydrogen atom, or R ^7X and R ^8X are Combined with the nitrogen atom to be bonded, a 3-8 membered heterocycle (the 3-8 membered Ring may form a good) have one or more substituents selected from the group D ^X,
   R ^9X is one or more substituents optionally may C1-C3 alkyl group which may have a selected from the group consisting of the group E ^X and the group G ^X, have one or more substituents selected from the group A ^X An optionally substituted C3-C6 alkenyl group, a C3-C6 alkynyl group optionally having one or more substituents selected from group A ^X , and one or more substituents selected from group D ^X good C3-C6 cycloalkyl group optionally substituted with one or more substituents phenyl group which may have a one or more substituents selected from the group D ^X is selected from the group D ^X 5-6 Represents a membered aromatic heterocyclic group or a hydrogen atom.
   Group A ^X : C1-C6 alkoxy group optionally having one or more halogen atoms, C1-C6 alkylthio group optionally having one or more halogen atoms, one or more substitutions selected from Group C ^X optionally may be C3-C6 cycloalkyl group having a group, one or more substituents phenyl group which may have a selected from the group F ^X, have one or more substituents selected from the group F ^X A group consisting of a 5-6 membered aromatic heterocyclic group, a halogen atom, a nitro group and a cyano group, which may be
   Group B ^X: 1 or more halogen atoms optionally may C1-C6 alkylthio group which may have one or more substituents phenyl group which may have a selected from the group F ^X, 1 is selected from the group F ^X A group consisting of a 5-6 membered aromatic heterocyclic group, a halogen atom, a nitro group and a cyano group, which may have the above substituents.
   Group C ^X: a halogen atom, the group consisting of a nitro group and a cyano group.
   Group D ^X: 1 or more substituents optionally may C1-C6 alkyl group which may have one or more substituents may C3-C6 cycloalkyl which may have a selected from the group C ^X selected from the group C ^X An alkyl group, a C1-C6 alkoxy group optionally having one or more halogen atoms, a C3-C6 alkenyloxy group optionally having one or more halogen atoms, and having one or more halogen atoms. A C3-C6 alkynyloxy group, a C1-C6 alkylthio group optionally having one or more halogen atoms, a C1-C6 alkylsulfonyloxy group optionally having one or more halogen atoms, a halogen atom, A group consisting of a cyano group, a nitro group, a hydroxy group and an amino group.
   Group E ^X : may have one or more substituents selected from group C ^X (C1-C6 alkyl) carbonylamino group, may have one or more substituents selected from group C ^X (C1-C6 alkyl) aminocarbonyl group, one or more may have a substituent di (C1-C6 alkyl) aminocarbonyl group, one or more substituents selected from the group C ^X selected from the group C ^X the a and may C1-C6 alkylsulfonylamino group, one or more may C1-C6 be substituted alkylaminosulfonyl group selected from the group C ^X, one or more selected from the group C ^X A group consisting of a di (C1-C6 alkyl) aminosulfonyl group, a hydroxy group and an amino group, which may have a substituent.
   Group F ^X : A group consisting of a C1-C6 alkyl group optionally having one or more halogen atoms, a C1-C6 alkoxy group optionally having one or more halogen atoms, a halogen atom and a cyano group.
   Group G ^X : C1-C6 alkoxy group optionally having one or more halogen atoms, C1-C6 alkylthio group optionally having one or more halogen atoms, one or more substitutions selected from Group C ^X optionally may be C3-C6 cycloalkyl group having a group, one or more substituents phenyl group which may have a selected from the group F ^X, have one or more substituents selected from the group F ^X A group consisting of a 5-membered aromatic heterocyclic group, a halogen atom, a nitro group, and a cyano group, which may be ]
   A compound represented by
3. G ^X is a benzene ring optionally having one or more substituents selected from the group consisting of a halogen atom and a C1-C6 alkyl group;
   The combination of L ^X, X ^X and R ^2X is,
   L ^X is C a (O), X ^X is a NR ^3X or an oxygen atom, R ^2X is C1-C6 alkyl group, or a combination of a hydrogen atom or halogen atom, or L ^X is S (O) ₂ , X ^X is NR ^3X , R ^2X is a combination of a C1-C6 alkyl group or a halogen atom,
   R ^1X is a C1-C6 alkyl group, a hydrogen atom or a halogen atom,
   R ^3X may have one or more substituents selected from group A ^X, and may have one or more substituents selected from group A ^X, C3-C6 alkynyl group, one or more halogen atoms optionally may C1-C6 alkoxy group which may have one or more substituents have may be C3-C6 cycloalkyl group selected from the group D ^X, selected from the group D ^X is one or more substituents phenyl group which may have a one or more 6-membered aromatic or substituted heterocyclic group or a hydrogen atom selected from the group D ^X to be,
   Z ^X is 1 or more may C3-C6 have a substituent of the cycloalkyl group, one or more substituents phenyl group which may have a selected from the group D ^X selected from the group D ^X, A 6-membered aromatic heterocyclic group ^optionally having one or more substituents selected from the group D ^X , CR ^4X R ^5X R ^6X , NR ^7X R ^8X or OR ^9X , or
   X ^X and Z ^X together with L ^{X to} which they are attached may have a 5-6 membered heterocycle (the 5-6 membered heterocycle may have one or more substituents selected from group D ^X Good) and
   Z ^X -L ^X -X ^X- (CR ^1X R ^2X ) _m on G ^X is bonded to the meta or para position with respect to the oxadiazole ring,
   R ^4X, R ^5X and R ^6X are the same or different phases, one or more substituents optionally may C1-C6 alkyl group which may have a selected from the group consisting of the group A ^X and the group E ^X, from the group A ^X C3-C6 alkynyl group optionally having one or more substituents selected, C1-C6 alkoxy group optionally having one or more substituents selected from group B ^X , selected from group D ^X 1 or may C3-C6 have a substituent of the cycloalkyl group, one or more substituents phenyl group which may have a selected from the group D ^X, one or more substituents selected from the group D ^X A 5-6 membered aromatic heterocyclic group optionally having a group, a hydrogen atom, a halogen atom or a cyano group,
   R ^7X and R ^8X are the same or different and are a C1-C6 alkyl group optionally having one or more substituents selected from the group consisting of group A ^X and group E ^X , 1 selected from group A ^X A C3-C6 alkynyl group optionally having one or more substituents, a C1-C6 alkoxy group optionally having one or more halogen atoms, and one or more substituents selected from the group D ^X. An optionally substituted C3-C6 cycloalkyl group, a phenyl group optionally having one or more substituents selected from group D ^X , and an optionally substituted one or more substituents selected from group D ^X 5 A 6-membered aromatic heterocyclic group or a hydrogen atom, or R ^7X and R ^8X together with the nitrogen atom to which they are bonded (the 3-6-membered heterocyclic ring is have one or more substituents selected from the group D ^X forms also may), A compound according to Motomeko 2.
4. G ^X is a benzene ring optionally having one or more halogen atoms,
   m is 1,
   The combination of L ^X, X ^X and R ^2X is,
   L ^X is C (O), X ^X is an oxygen atom, R ^2X is a combination of hydrogen atoms, or L ^X is S (O) ₂ , X ^X is NR ^3X , R ^2X Is a C1-C3 alkyl group,
   R ^1X is a hydrogen atom,
   R ^3X is a hydrogen atom,
   Z ^X is CR ^4X R ^5X R ^6X or NR ^7X R ^8X ;
   G ^X on the ^{Z X -L X -X X - (} CR 1X R 2X) m is attached at the para position relative to the oxadiazole ring,
   R ^4X , R ^5X and R ^6X are the same or different and are a C1-C6 alkyl group or a hydrogen atom,
   R ^7X and R ^8X are the same or different and have a C1-C6 alkyl group (the C1-C6 alkyl group has one or more substituents selected from the group consisting of a cyano group and a C1-C3 alkoxy group). Or a C3-C6 cycloalkyl group.
5. A pest control agent comprising the compound according to claim 2, 3 or 4.
6. A method for controlling pests by treating a plant or soil with an effective amount of the compound according to claim 2, 3 or 4.
7. Use of the compound according to claim 2, 3 or 4 for controlling pests.
8. A composition containing one or more selected from the group consisting of a bactericidal active ingredient, an insecticidal active ingredient, an acaricidal active ingredient, a nematicidal active ingredient and a plant growth regulating ingredient, and the compound according to claim 2, 3 or 4.