WO2015092810A2 - Forme amorphe d'idélalisib - Google Patents
Forme amorphe d'idélalisib Download PDFInfo
- Publication number
- WO2015092810A2 WO2015092810A2 PCT/IN2014/000724 IN2014000724W WO2015092810A2 WO 2015092810 A2 WO2015092810 A2 WO 2015092810A2 IN 2014000724 W IN2014000724 W IN 2014000724W WO 2015092810 A2 WO2015092810 A2 WO 2015092810A2
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- idelalisib
- less
- pharmaceutically acceptable
- amorphous
- solid dispersion
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
- C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Anesthesiology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicinal Preparation (AREA)
Abstract
La présente invention concerne une forme amorphe d'idélalisib et des procédés pour la préparation de ladite forme amorphe. L'invention concerne également des compositions pharmaceutiques qui contiennent ladite forme amorphe d'idélalisib.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN3641/MUM/2013 | 2013-11-20 | ||
IN3641MU2013 IN2013MU03641A (fr) | 2013-11-20 | 2014-11-19 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2015092810A2 true WO2015092810A2 (fr) | 2015-06-25 |
WO2015092810A3 WO2015092810A3 (fr) | 2015-08-13 |
Family
ID=52785145
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/IN2014/000724 WO2015092810A2 (fr) | 2013-11-20 | 2014-11-19 | Forme amorphe d'idélalisib |
Country Status (2)
Country | Link |
---|---|
IN (1) | IN2013MU03641A (fr) |
WO (1) | WO2015092810A2 (fr) |
Cited By (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2016097314A1 (fr) * | 2014-12-19 | 2016-06-23 | Sandoz Ag | Formes amorphes et cristallines d'idélalisib et procédé pour les produire |
WO2016147206A1 (fr) | 2015-03-13 | 2016-09-22 | Mylan Laboratories Limited | Procédé pour la préparation d'idélalisib amorphe et son mélange préliminaire |
WO2016157136A1 (fr) | 2015-04-02 | 2016-10-06 | Mylan Laboratories Ltd | Formes cristallines de l'idélalisib |
WO2016165618A1 (fr) * | 2015-04-15 | 2016-10-20 | 上海方楠生物科技有限公司 | Substance amorphe d'idélalisibe et procédé de préparation associé |
WO2017137097A1 (fr) * | 2016-02-12 | 2017-08-17 | Synthon B.V. | Composition pharmaceutique comprenant de l'idelalisib sous forme amorphe |
WO2017175184A1 (fr) * | 2016-04-07 | 2017-10-12 | Laurus Labs Limited | Procédé de préparation de la forme amorphe d'idélalisib |
EP3272348A1 (fr) | 2016-07-21 | 2018-01-24 | LEK Pharmaceuticals d.d. | Composition pharmaceutique comportant de l'idelalisib |
WO2019178596A1 (fr) | 2018-03-16 | 2019-09-19 | Johnson Matthey Public Limited Company | Formes à l'état solide solvatées de pyridine ou de n,n-diméthylacétamide d'idélalisib solvaté, leur utilisation et leur préparation |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2005113556A1 (fr) | 2004-05-13 | 2005-12-01 | Icos Corporation | Quinazolinones utilisees en tant qu'inhibiteurs de la phosphatidylinositol 3-kinase delta humaine |
WO2013134288A1 (fr) | 2012-03-05 | 2013-09-12 | Gilead Calistoga Llc | Formes polymorphes de l'acide -2-(1-(9h-purine-6-ylamino)propyl)-5-fluoro-3-phénylquinazolin-4(3h)-one |
-
2014
- 2014-11-19 IN IN3641MU2013 patent/IN2013MU03641A/en unknown
- 2014-11-19 WO PCT/IN2014/000724 patent/WO2015092810A2/fr active Application Filing
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2005113556A1 (fr) | 2004-05-13 | 2005-12-01 | Icos Corporation | Quinazolinones utilisees en tant qu'inhibiteurs de la phosphatidylinositol 3-kinase delta humaine |
WO2013134288A1 (fr) | 2012-03-05 | 2013-09-12 | Gilead Calistoga Llc | Formes polymorphes de l'acide -2-(1-(9h-purine-6-ylamino)propyl)-5-fluoro-3-phénylquinazolin-4(3h)-one |
Cited By (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2016097314A1 (fr) * | 2014-12-19 | 2016-06-23 | Sandoz Ag | Formes amorphes et cristallines d'idélalisib et procédé pour les produire |
WO2016147206A1 (fr) | 2015-03-13 | 2016-09-22 | Mylan Laboratories Limited | Procédé pour la préparation d'idélalisib amorphe et son mélange préliminaire |
US20180064714A1 (en) * | 2015-03-13 | 2018-03-08 | Mylan Laboratories Ltd | Process for the Preparation of Amorphous Idelalisib and its Premix |
WO2016157136A1 (fr) | 2015-04-02 | 2016-10-06 | Mylan Laboratories Ltd | Formes cristallines de l'idélalisib |
WO2016165618A1 (fr) * | 2015-04-15 | 2016-10-20 | 上海方楠生物科技有限公司 | Substance amorphe d'idélalisibe et procédé de préparation associé |
US10370376B2 (en) | 2015-04-15 | 2019-08-06 | Alnova Pharmaceuticals, Ltd. | Amorphous substance of Idelalisib and preparation method therefor |
WO2017137097A1 (fr) * | 2016-02-12 | 2017-08-17 | Synthon B.V. | Composition pharmaceutique comprenant de l'idelalisib sous forme amorphe |
WO2017175184A1 (fr) * | 2016-04-07 | 2017-10-12 | Laurus Labs Limited | Procédé de préparation de la forme amorphe d'idélalisib |
EP3272348A1 (fr) | 2016-07-21 | 2018-01-24 | LEK Pharmaceuticals d.d. | Composition pharmaceutique comportant de l'idelalisib |
WO2019178596A1 (fr) | 2018-03-16 | 2019-09-19 | Johnson Matthey Public Limited Company | Formes à l'état solide solvatées de pyridine ou de n,n-diméthylacétamide d'idélalisib solvaté, leur utilisation et leur préparation |
US11358966B2 (en) | 2018-03-16 | 2022-06-14 | Johnson Matthey Public Limited Company | Pyridine or N,N-dimethyl acetamide solvated solid state forms of solvated idelalisib, their use and preparation |
Also Published As
Publication number | Publication date |
---|---|
IN2013MU03641A (fr) | 2015-07-31 |
WO2015092810A3 (fr) | 2015-08-13 |
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