WO2011045760A3 - Micronized olmesartan medoxomil compositions - Google Patents

Micronized olmesartan medoxomil compositions Download PDF

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Publication number
WO2011045760A3
WO2011045760A3 PCT/IB2010/054641 IB2010054641W WO2011045760A3 WO 2011045760 A3 WO2011045760 A3 WO 2011045760A3 IB 2010054641 W IB2010054641 W IB 2010054641W WO 2011045760 A3 WO2011045760 A3 WO 2011045760A3
Authority
WO
WIPO (PCT)
Prior art keywords
micronized
compositions
olmesartan medoxomil
medoxomil
olmesartan
Prior art date
Application number
PCT/IB2010/054641
Other languages
French (fr)
Other versions
WO2011045760A2 (en
Inventor
Arun Gupta
Madhusudan Vattikonda
Anupam Trehan
Vinod Kumar Arora
Original Assignee
Ranbaxy Laboratories Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ranbaxy Laboratories Limited filed Critical Ranbaxy Laboratories Limited
Publication of WO2011045760A2 publication Critical patent/WO2011045760A2/en
Publication of WO2011045760A3 publication Critical patent/WO2011045760A3/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/549—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame having two or more nitrogen atoms in the same ring, e.g. hydrochlorothiazide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The present invention relates to pharmaceutical compositions comprising micronized particles of olmesartan medoxomil and processes thereof.
PCT/IB2010/054641 2009-10-13 2010-10-13 Micronized olmesartan medoxomil compositions WO2011045760A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN2119DE2009 2009-10-13
IN2119/DEL/2009 2009-10-13

Publications (2)

Publication Number Publication Date
WO2011045760A2 WO2011045760A2 (en) 2011-04-21
WO2011045760A3 true WO2011045760A3 (en) 2012-01-05

Family

ID=43413907

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/IB2010/054641 WO2011045760A2 (en) 2009-10-13 2010-10-13 Micronized olmesartan medoxomil compositions

Country Status (1)

Country Link
WO (1) WO2011045760A2 (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2554159A1 (en) * 2011-08-04 2013-02-06 ratiopharm GmbH Dosage forms comprising apixaban and content uniformity enhancer
WO2014002011A1 (en) * 2012-06-26 2014-01-03 Micro Labs Limited Micronized particles of olmesartan medoxomil and pharmaceutical composition thereof
WO2014030082A1 (en) 2012-08-22 2014-02-27 Lupin Limited Novel method to obtain olmesartan medoxomil with reduced particle size
CN103263395A (en) * 2013-06-10 2013-08-28 南京正宽医药科技有限公司 Telmisartan tablet preparation and preparation method thereof
JP6653116B2 (en) * 2014-08-27 2020-02-26 日本ケミファ株式会社 Olmesartan prodrug formulations
JP2017008018A (en) * 2015-06-19 2017-01-12 日本ジェネリック株式会社 Olmesartan medoxomil tablet in which elution properties are improved

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20060281800A1 (en) * 2005-04-12 2006-12-14 Glenmark Pharmaceuticals Limited Polymorphic form of olmesartan and process for its preparation
WO2007128478A2 (en) * 2006-05-04 2007-11-15 Lek Pharmaceuticals D.D. Pharmaceutical composition
CA2681591A1 (en) * 2007-03-23 2008-10-02 Daiichi Sankyo Company, Limited Pulverized crystals of olmesartan medoxomil
WO2009113420A1 (en) * 2008-03-13 2009-09-17 第一三共株式会社 Improvement of dissolvability of preparation containing olmesartan medoxomil

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5616599A (en) 1991-02-21 1997-04-01 Sankyo Company, Limited Angiotensin II antagosist 1-biphenylmethylimidazole compounds and their therapeutic use
WO2007047838A2 (en) 2005-10-20 2007-04-26 Dr. Reddy's Laboratories Ltd. Process for preparing olmesartan medoxomil

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20060281800A1 (en) * 2005-04-12 2006-12-14 Glenmark Pharmaceuticals Limited Polymorphic form of olmesartan and process for its preparation
WO2007128478A2 (en) * 2006-05-04 2007-11-15 Lek Pharmaceuticals D.D. Pharmaceutical composition
CA2681591A1 (en) * 2007-03-23 2008-10-02 Daiichi Sankyo Company, Limited Pulverized crystals of olmesartan medoxomil
WO2009113420A1 (en) * 2008-03-13 2009-09-17 第一三共株式会社 Improvement of dissolvability of preparation containing olmesartan medoxomil
EP2253318A1 (en) * 2008-03-13 2010-11-24 Daiichi Sankyo Company, Limited Improvement of dissolvability of preparation containing olmesartan medoxomil

Also Published As

Publication number Publication date
WO2011045760A2 (en) 2011-04-21

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