WO2010060513A3 - Method for the photo stabilisation of ascorbic acid derivatives - Google Patents

Method for the photo stabilisation of ascorbic acid derivatives Download PDF

Info

Publication number
WO2010060513A3
WO2010060513A3 PCT/EP2009/007685 EP2009007685W WO2010060513A3 WO 2010060513 A3 WO2010060513 A3 WO 2010060513A3 EP 2009007685 W EP2009007685 W EP 2009007685W WO 2010060513 A3 WO2010060513 A3 WO 2010060513A3
Authority
WO
WIPO (PCT)
Prior art keywords
ascorbic acid
stabilisation
photo
acid derivatives
filters
Prior art date
Application number
PCT/EP2009/007685
Other languages
German (de)
French (fr)
Other versions
WO2010060513A2 (en
Inventor
Thomas Rudolph
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of WO2010060513A2 publication Critical patent/WO2010060513A2/en
Publication of WO2010060513A3 publication Critical patent/WO2010060513A3/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q17/00—Barrier preparations; Preparations brought into direct contact with the skin for affording protection against external influences, e.g. sunlight, X-rays or other harmful rays, corrosive materials, bacteria or insect stings
    • A61Q17/04—Topical preparations for affording protection against sunlight or other radiation; Topical sun tanning preparations
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/35—Ketones, e.g. benzophenone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/37—Esters of carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/40—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing nitrogen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/67—Vitamins
    • A61K8/676—Ascorbic acid, i.e. vitamin C
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/40—Chemical, physico-chemical or functional or structural properties of particular ingredients
    • A61K2800/52—Stabilizers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q5/00—Preparations for care of the hair
    • A61Q5/06—Preparations for styling the hair, e.g. by temporary shaping or colouring
    • A61Q5/065—Preparations for temporary colouring the hair, e.g. direct dyes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q5/00—Preparations for care of the hair
    • A61Q5/10—Preparations for permanently dyeing the hair

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Birds (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cosmetics (AREA)

Abstract

The invention relates to the use of a compound selected from the group containing diphenyl acrylate UV filters, phenolic antioxidants or mixtures of the same, for improving the UV stability of a preparation containing at least one ascorbic acid derivative as a UV filter.
PCT/EP2009/007685 2008-11-26 2009-10-28 Method for the photo stabilisation of ascorbic acid derivatives WO2010060513A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08020511.5 2008-11-26
EP08020511 2008-11-26

Publications (2)

Publication Number Publication Date
WO2010060513A2 WO2010060513A2 (en) 2010-06-03
WO2010060513A3 true WO2010060513A3 (en) 2010-09-23

Family

ID=41722724

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2009/007685 WO2010060513A2 (en) 2008-11-26 2009-10-28 Method for the photo stabilisation of ascorbic acid derivatives

Country Status (1)

Country Link
WO (1) WO2010060513A2 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2427443B1 (en) 2009-05-08 2014-10-15 Merck Patent GmbH Cinnamic acid ascorbates
CN117043202A (en) 2021-03-05 2023-11-10 H.B.富乐公司 Cyanoacrylate compositions containing hazard-free stabilizers

Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0664290A1 (en) * 1994-01-20 1995-07-26 L'oreal Mono- and di-esters of cinnamic acid or of one of his derivatives and of vitamine C, their process of preparation and their use as antioxydants in cosmetic, pharmaceutical or alimentary compositions
DE10013156A1 (en) * 2000-03-17 2001-09-20 Volkhard Jenning Water-containing vehicle for cosmetic or dermatological compositions, in which active agents or auxiliaries are stabilized by combination of ascorbic acid or derivative, polyphenol and buffer
US20050154054A1 (en) * 2004-01-13 2005-07-14 Skinceuticals, Inc. Stabilized ascorbic acid compositions and methods therefor
EP1591099A2 (en) * 2004-04-28 2005-11-02 MERCK PATENT GmbH Methods for stabilizing ingredients within cosmetics, personal care and household products
WO2007048645A2 (en) * 2005-10-24 2007-05-03 Ciba Holding Inc. Protection of oxidizable agents
WO2008017346A2 (en) * 2006-08-11 2008-02-14 Merck Patent Gmbh Use of ascorbic acid derivatives for the functionalization of matrices

Patent Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0664290A1 (en) * 1994-01-20 1995-07-26 L'oreal Mono- and di-esters of cinnamic acid or of one of his derivatives and of vitamine C, their process of preparation and their use as antioxydants in cosmetic, pharmaceutical or alimentary compositions
DE10013156A1 (en) * 2000-03-17 2001-09-20 Volkhard Jenning Water-containing vehicle for cosmetic or dermatological compositions, in which active agents or auxiliaries are stabilized by combination of ascorbic acid or derivative, polyphenol and buffer
US20050154054A1 (en) * 2004-01-13 2005-07-14 Skinceuticals, Inc. Stabilized ascorbic acid compositions and methods therefor
EP1591099A2 (en) * 2004-04-28 2005-11-02 MERCK PATENT GmbH Methods for stabilizing ingredients within cosmetics, personal care and household products
WO2007048645A2 (en) * 2005-10-24 2007-05-03 Ciba Holding Inc. Protection of oxidizable agents
WO2008017346A2 (en) * 2006-08-11 2008-02-14 Merck Patent Gmbh Use of ascorbic acid derivatives for the functionalization of matrices

Non-Patent Citations (3)

* Cited by examiner, † Cited by third party
Title
GASPAR ET AL: "Photostability and efficacy studies of topical formulations containing UV-filters combination and vitamins A, C and E", INTERNATIONAL JOURNAL OF PHARMACEUTICS, ELSEVIER BV, NL, vol. 343, no. 1-2, 30 August 2007 (2007-08-30), pages 181 - 189, XP022223265, ISSN: 0378-5173 *
LIN F-H ET AL: "Ferulic acid stabilizes a solution of vitamin C and E and doubles its photoprotection of skin", JOURNAL OF INVESTIGATIVE DERMATOLOGY, NATURE PUBLISHING GROUP, GB, vol. 125, no. 4, 1 October 2005 (2005-10-01), pages 826 - 832, XP008101490, ISSN: 0022-202X *
MURRAY J C ET AL: "A topical antioxidant solution containing vitamins C and E stabilized by ferulic acid provides protection for human skin against damage caused by ultraviolet irradiation", JOURNAL OF THE AMERICAN ACADEMY OF DERMATOLOGY, C.V. MOSBY, ST. LOUIS, MO, US, vol. 59, no. 3, 1 September 2008 (2008-09-01), pages 418 - 425, XP024518729, ISSN: 0190-9622, [retrieved on 20080707] *

Also Published As

Publication number Publication date
WO2010060513A2 (en) 2010-06-03

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