WO2009047534A3 - Composés, procédé et utilisation - Google Patents
Composés, procédé et utilisation Download PDFInfo
- Publication number
- WO2009047534A3 WO2009047534A3 PCT/GB2008/003456 GB2008003456W WO2009047534A3 WO 2009047534 A3 WO2009047534 A3 WO 2009047534A3 GB 2008003456 W GB2008003456 W GB 2008003456W WO 2009047534 A3 WO2009047534 A3 WO 2009047534A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- optionally substituted
- compounds
- formula
- photoantimicrobials
- fused
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 5
- 238000002360 preparation method Methods 0.000 title 1
- 125000000547 substituted alkyl group Chemical group 0.000 abstract 3
- 230000000845 anti-microbial effect Effects 0.000 abstract 2
- 229910052736 halogen Chemical class 0.000 abstract 2
- 150000002367 halogens Chemical class 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 229920006395 saturated elastomer Polymers 0.000 abstract 2
- 125000005415 substituted alkoxy group Chemical group 0.000 abstract 2
- BUGBHKTXTAQXES-UHFFFAOYSA-N Selenium Chemical compound [Se] BUGBHKTXTAQXES-UHFFFAOYSA-N 0.000 abstract 1
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
- 239000005864 Sulphur Substances 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- 150000001450 anions Chemical class 0.000 abstract 1
- 125000004429 atom Chemical group 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 229910052711 selenium Inorganic materials 0.000 abstract 1
- 239000011669 selenium Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
- C07D513/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C09—DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
- C09B—ORGANIC DYES OR CLOSELY-RELATED COMPOUNDS FOR PRODUCING DYES, e.g. PIGMENTS; MORDANTS; LAKES
- C09B21/00—Thiazine dyes
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Agronomy & Crop Science (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- Dentistry (AREA)
- Plant Pathology (AREA)
- Pest Control & Pesticides (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La présente invention porte sur des composés de Formule 4 et sur des composés antimicrobiens et des compositions antimicrobiennes à base des composés de Formule 4 : dans laquelle : X comprend du soufre ou du sélénium; Y comprend un anion pharmaceutiquement acceptable; R1 et R9 représentent chacun indépendamment hydrogène, alkyle facultativement substitué, alcoxyle facultativement substitué, amine facultativement substituée ou halogène; et R3a, R3b, R7a et R7b sont chacun indépendamment H ou alkyle facultativement substitué, à la condition qu'au moins l'un de R3a ou R3b et/ou R7a ou R7b conjointement avec les atomes d'azote auxquels ils sont attachés forment un noyau à 6 ou 7 chaînons facultativement saturé, facultativement substitué avec R2 ou R4 et/ou R6 ou R8; et R2, R4, R6 et R8 respectivement représentent chacun indépendamment hydrogène, alkyle facultativement substitué, alcoxyle facultativement substitué ou halogène, pour autant qu'au moins l'un parmi R2, R4, R6 ou R8 conjointement avec les atomes auxquels ils sont attachés forment un noyau à 6 ou 7 chaînons facultativement saturé, facultativement substitué avec R3a ou R3b et/ou R7b ou R7a respectivement; et à la condition que les composés ne soient pas de Formule 3a ou 3b.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0719834.4 | 2007-10-11 | ||
| GB0719834A GB2453564A (en) | 2007-10-11 | 2007-10-11 | Ring-fused derivatives of 3,7-diamino- phenothiazinium & phenoselenazinium salts for use as antimicrobial agents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| WO2009047534A2 WO2009047534A2 (fr) | 2009-04-16 |
| WO2009047534A3 true WO2009047534A3 (fr) | 2009-05-28 |
Family
ID=38787960
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PCT/GB2008/003456 WO2009047534A2 (fr) | 2007-10-11 | 2008-10-13 | Composés, procédé et utilisation |
Country Status (2)
| Country | Link |
|---|---|
| GB (1) | GB2453564A (fr) |
| WO (1) | WO2009047534A2 (fr) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB201004450D0 (en) * | 2010-03-17 | 2010-05-05 | Pharmalucia Ltd | Compounds and methods relating thereto |
| CN114391446A (zh) * | 2022-01-24 | 2022-04-26 | 邯郸市农业科学院 | 一种脱毒生姜原原种的生产方法 |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2373787A (en) * | 2001-03-08 | 2002-10-02 | Univ Central Lancashire | Phenothiazinium derivatives and their use to reduce pathogenic contaminants |
| WO2005054217A1 (fr) * | 2003-11-28 | 2005-06-16 | Photopharmica Limited | Derives ameliores (2) de bleu de methylene biologiquement actifs |
-
2007
- 2007-10-11 GB GB0719834A patent/GB2453564A/en not_active Withdrawn
-
2008
- 2008-10-13 WO PCT/GB2008/003456 patent/WO2009047534A2/fr active Application Filing
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2373787A (en) * | 2001-03-08 | 2002-10-02 | Univ Central Lancashire | Phenothiazinium derivatives and their use to reduce pathogenic contaminants |
| WO2005054217A1 (fr) * | 2003-11-28 | 2005-06-16 | Photopharmica Limited | Derives ameliores (2) de bleu de methylene biologiquement actifs |
Non-Patent Citations (1)
| Title |
|---|
| WAINWRIGHT, MARK ET AL: "phenothiazinium-based photobactericidal meterials", JOURNAL OF PHOTOCHEMISTRY AND PHOTOBIOLOGY B:BIOLOGY, vol. 84, 2006, pages 227 - 230, XP025227644 * |
Also Published As
| Publication number | Publication date |
|---|---|
| GB2453564A (en) | 2009-04-15 |
| GB0719834D0 (en) | 2007-11-21 |
| WO2009047534A2 (fr) | 2009-04-16 |
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