WO2009011367A1 - 水系組成物 - Google Patents

水系組成物 Download PDF

Info

Publication number
WO2009011367A1
WO2009011367A1 PCT/JP2008/062853 JP2008062853W WO2009011367A1 WO 2009011367 A1 WO2009011367 A1 WO 2009011367A1 JP 2008062853 W JP2008062853 W JP 2008062853W WO 2009011367 A1 WO2009011367 A1 WO 2009011367A1
Authority
WO
WIPO (PCT)
Prior art keywords
aqueous composition
solid content
aqueous
mass
additive
Prior art date
Application number
PCT/JP2008/062853
Other languages
English (en)
French (fr)
Inventor
Yoshihito Yaginuma
Naoya Yoshida
Original Assignee
Asahi Kasei Chemicals Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Asahi Kasei Chemicals Corporation filed Critical Asahi Kasei Chemicals Corporation
Priority to US12/663,961 priority Critical patent/US8765187B2/en
Priority to JP2009523662A priority patent/JP5283623B2/ja
Publication of WO2009011367A1 publication Critical patent/WO2009011367A1/ja

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • A61K9/5047—Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A61K9/2081—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets with microcapsules or coated microparticles according to A61K9/50
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core

Abstract

　アクリル酸エチル・メタクリル酸メチルコポリマー又は可塑化酢酸ビニルポリマー（ａ）、エチルセルロース（ｂ）、水溶性医薬用添加剤（ｃ）、酸化チタン（ｄ）、及び水（ｅ）を含んでなる水系組成物であって、該（ａ）、（ｂ）、（ｃ）、及び（ｄ）の固形分質量比ａ：ｂ：ｃ：ｄが、１００：（５～５０）：（１～５０）：（０．５～１０）であり、該水系組成物に対する固形分濃度が０．５％～４０質量％である上記水系組成物。
PCT/JP2008/062853 2007-07-17 2008-07-16 水系組成物 WO2009011367A1 (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
US12/663,961 US8765187B2 (en) 2007-07-17 2008-07-16 Aqueous composition
JP2009523662A JP5283623B2 (ja) 2007-07-17 2008-07-16 水系組成物

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2007185357 2007-07-17
JP2007-185357 2007-07-17

Publications (1)

Publication Number Publication Date
WO2009011367A1 true WO2009011367A1 (ja) 2009-01-22

Family

ID=40259699

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/JP2008/062853 WO2009011367A1 (ja) 2007-07-17 2008-07-16 水系組成物

Country Status (3)

Country Link
US (1) US8765187B2 (ja)
JP (1) JP5283623B2 (ja)
WO (1) WO2009011367A1 (ja)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011043370A1 (ja) 2009-10-09 2011-04-14 旭化成ケミカルズ株式会社 コーティングフィルム、及びそれを用いた顆粒、錠剤

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8268356B2 (en) * 2007-11-16 2012-09-18 Asahi Kasei Chemicals Corporation Aqueous film coating solution, film coated granule and tablet using the same

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4728513A (en) * 1985-07-31 1988-03-01 Zyma Sa Granular delayed-release form of pharmaceutically active substances
WO1988007369A1 (en) * 1987-03-27 1988-10-06 The Wellcome Foundation Limited Pharmaceutical formulations
JPH04169522A (ja) * 1990-11-01 1992-06-17 Shin Etsu Chem Co Ltd 徐放性錠剤およびその製造方法
EP1238662A2 (en) * 2001-03-07 2002-09-11 Sumitomo Pharmaceuticals Company, Limited Method for manufacturing drug granules, the drug granules and pharmaceutical preparation containing the drug granules
WO2003000169A1 (en) * 2001-06-20 2003-01-03 Takeda Chemical Industries, Ltd. Method of manufacturing tablet

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6468561B1 (en) * 1986-06-19 2002-10-22 Bpsi Holdings, Inc. Aqueous film coating with improved properties
WO2002026845A1 (de) 2000-09-29 2002-04-04 Basf Aktiengesellschaft Wässrige polymerdispersion
JP4438268B2 (ja) 2001-03-07 2010-03-24 大日本住友製薬株式会社 薬物顆粒の製造方法、および薬物顆粒、ならびにそれを用いた医薬製剤

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4728513A (en) * 1985-07-31 1988-03-01 Zyma Sa Granular delayed-release form of pharmaceutically active substances
WO1988007369A1 (en) * 1987-03-27 1988-10-06 The Wellcome Foundation Limited Pharmaceutical formulations
JPH04169522A (ja) * 1990-11-01 1992-06-17 Shin Etsu Chem Co Ltd 徐放性錠剤およびその製造方法
EP1238662A2 (en) * 2001-03-07 2002-09-11 Sumitomo Pharmaceuticals Company, Limited Method for manufacturing drug granules, the drug granules and pharmaceutical preparation containing the drug granules
WO2003000169A1 (en) * 2001-06-20 2003-01-03 Takeda Chemical Industries, Ltd. Method of manufacturing tablet

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011043370A1 (ja) 2009-10-09 2011-04-14 旭化成ケミカルズ株式会社 コーティングフィルム、及びそれを用いた顆粒、錠剤
US8992988B2 (en) 2009-10-09 2015-03-31 Asahi Kasei Chemicals Corporation Coating film, and granules and tablets each utilizing same
JP5787762B2 (ja) * 2009-10-09 2015-09-30 旭化成ケミカルズ株式会社 コーティングフィルム、及びそれを用いた顆粒、錠剤
US9439865B2 (en) 2009-10-09 2016-09-13 Asahi Kasei Chemicals Corporation Coating film, and granules and tablets each utilizing same

Also Published As

Publication number Publication date
JP5283623B2 (ja) 2013-09-04
US20100172978A1 (en) 2010-07-08
JPWO2009011367A1 (ja) 2010-09-24
US8765187B2 (en) 2014-07-01

Similar Documents

Publication Publication Date Title
WO2007089451A3 (en) Blends of biopolymers with acrylic copolymers
WO2007017196A3 (de) Öl-in-wasser emulsionen
WO2008037716A3 (en) Pharmaceutical compositions comprising nilotinib or its salt
JP2009516717A5 (ja)
WO2006127637A3 (en) Compressed pharmaceutical composition comprising coated pellets and a direct compression mixture, and method of preparation thereof
EP2113532A8 (en) Resin composition, and molded article produced from the same
DE502006005477D1 (de) Herstellung eines wasserabsorbierenden harzes unter einmischen eines teilchenförmigen additivs
WO2008036334A3 (en) Toughened poly(hydroxyalkanoic acid) compositions
WO2008018044A3 (en) Absorbent articles including an improved odour control system
TWI370155B (en) Conductive copolymer, conductive copolymer composition, film and opto-electronic device using the same
WO2009038112A1 (ja) Ｎｐｙｙ５受容体拮抗剤を含有する固形製剤
EP2060605A4 (en) COMPOSITION CONTAINING COPOLYMER OF POLYHYDROXYALCANOATE AND POLYLACTIC ACID, AS FOAM
WO2007041156A3 (en) Antibiotic formulations, unit doses, kits, and methods
IL179069A0 (en) Lactone copolymer and radiation-sensitive resin composition
WO2009077693A3 (fr) Compositions comprenant au moins un derive de l'acide naphtoique, du peroxyde de benzoyle et au moins un agent filmogene
EP1704853A3 (en) Water-in-silicone emulsion compositions
WO2008039472A3 (en) Stabilizing compositions for antibiotics and methods of use
WO2010035122A3 (fr) Complexe constitue d'un polysaccharide et d'une hpb
WO2008123582A1 (ja) テトラヒドロイソキノリン化合物
BRPI0810335A2 (pt) "pó depolímero redispersável, dispersão aquosa, composição de polímero e uso da composição de polímero"
WO2009063916A1 (ja) 水系フィルムコーティング液、および、フィルムコーティング顆粒、ならびに、これを用いた錠剤
WO2007100524A3 (en) Repeat sequence protein polymer nanoparticles optionally containing active agents and their preparation
MX340436B (es) Formulacion farmaceutica estable con descoloramiento limitado.
WO2007080172A3 (en) Plasticizer of natural origin for nail polish
WO2009011367A1 (ja) 水系組成物

Legal Events

Date Code Title Description
121 Ep: the epo has been informed by wipo that ep was designated in this application

Ref document number: 08778204

Country of ref document: EP

Kind code of ref document: A1

ENP Entry into the national phase

Ref document number: 2009523662

Country of ref document: JP

Kind code of ref document: A

WWE Wipo information: entry into national phase

Ref document number: 12663961

Country of ref document: US

NENP Non-entry into the national phase

Ref country code: DE

122 Ep: pct application non-entry in european phase

Ref document number: 08778204

Country of ref document: EP

Kind code of ref document: A1