WO2007139948A3 - Composés d'imidazo-azépinone - Google Patents
Composés d'imidazo-azépinone Download PDFInfo
- Publication number
- WO2007139948A3 WO2007139948A3 PCT/US2007/012516 US2007012516W WO2007139948A3 WO 2007139948 A3 WO2007139948 A3 WO 2007139948A3 US 2007012516 W US2007012516 W US 2007012516W WO 2007139948 A3 WO2007139948 A3 WO 2007139948A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- imidazoazepinone
- compounds
- formula
- treatment
- methods
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Epidemiology (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Obesity (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Transplantation (AREA)
- Hematology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La présente invention concerne un composé pur du point de vue énantiomère, de formule I, ainsi que des formulations pharmaceutiques le contenant, et des procédés pour l'utiliser pour le traitement de maladies auto-immunes.
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US80890606P | 2006-05-26 | 2006-05-26 | |
US80877006P | 2006-05-26 | 2006-05-26 | |
US60/808,906 | 2006-05-26 | ||
US60/808,770 | 2006-05-26 | ||
US81561706P | 2006-06-22 | 2006-06-22 | |
US60/815,617 | 2006-06-22 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2007139948A2 WO2007139948A2 (fr) | 2007-12-06 |
WO2007139948A3 true WO2007139948A3 (fr) | 2008-01-24 |
Family
ID=38649936
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/US2007/012516 WO2007139948A2 (fr) | 2006-05-26 | 2007-05-25 | Composés d'imidazo-azépinone |
Country Status (1)
Country | Link |
---|---|
WO (1) | WO2007139948A2 (fr) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2217242A1 (fr) * | 2007-11-15 | 2010-08-18 | Eisai R&D Management Co., Ltd. | Procédés d'utilisation |
WO2011011494A1 (fr) * | 2009-07-21 | 2011-01-27 | Eisai R&D Management Co., Ltd. | Composés imidazoazépinones |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0385489A1 (fr) * | 1989-03-03 | 1990-09-05 | Eisai Co., Ltd. | Composés d'azacyclooctadiènes et leur usage pharmaceutique |
EP1619193A1 (fr) * | 2003-04-18 | 2006-01-25 | Ono Pharmaceutical Co., Ltd. | Compose de spiropiperidine et son utilisation medicinale |
WO2006128143A2 (fr) * | 2005-05-27 | 2006-11-30 | Eisai Co., Ltd. | Composes a base d'hydantoine |
-
2007
- 2007-05-25 WO PCT/US2007/012516 patent/WO2007139948A2/fr active Application Filing
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0385489A1 (fr) * | 1989-03-03 | 1990-09-05 | Eisai Co., Ltd. | Composés d'azacyclooctadiènes et leur usage pharmaceutique |
EP1619193A1 (fr) * | 2003-04-18 | 2006-01-25 | Ono Pharmaceutical Co., Ltd. | Compose de spiropiperidine et son utilisation medicinale |
WO2006128143A2 (fr) * | 2005-05-27 | 2006-11-30 | Eisai Co., Ltd. | Composes a base d'hydantoine |
Also Published As
Publication number | Publication date |
---|---|
WO2007139948A2 (fr) | 2007-12-06 |
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