WO2006106244A3 - PROCEDE DE PREPARATION DE β-AMINOESTERS OU α-, β-DIAMINOESTERS DERIVES DE LA SERINE - Google Patents
PROCEDE DE PREPARATION DE β-AMINOESTERS OU α-, β-DIAMINOESTERS DERIVES DE LA SERINE Download PDFInfo
- Publication number
- WO2006106244A3 WO2006106244A3 PCT/FR2006/000780 FR2006000780W WO2006106244A3 WO 2006106244 A3 WO2006106244 A3 WO 2006106244A3 FR 2006000780 W FR2006000780 W FR 2006000780W WO 2006106244 A3 WO2006106244 A3 WO 2006106244A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- esters
- preparing
- serine
- diamino
- amino
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C247/00—Compounds containing azido groups
- C07C247/02—Compounds containing azido groups with azido groups bound to acyclic carbon atoms of a carbon skeleton
- C07C247/04—Compounds containing azido groups with azido groups bound to acyclic carbon atoms of a carbon skeleton being saturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C253/00—Preparation of carboxylic acid nitriles
- C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/26—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of esters of sulfonic acids
- C07C303/28—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of esters of sulfonic acids by reaction of hydroxy compounds with sulfonic acids or derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D295/145—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/15—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
L'invention concerne un procédé de préparation d'un composé de formule (I), dans laquelle R1, R2, R3 identiques ou différents sont des groupements protecteurs et Nu est un groupe nucléophile, procédé dans lequel on fait réagir un composé nucléophile sur un composé (II), dans laquelle R1, R2, R3 sont tels que définis ci-dessus et Y représente un groupe partant.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0503537A FR2884249A1 (fr) | 2005-04-08 | 2005-04-08 | Procede de preparation de beta-aminoesters ou alpha-, beta-diaminoesters derives de la serine |
FR0503537 | 2005-04-08 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2006106244A2 WO2006106244A2 (fr) | 2006-10-12 |
WO2006106244A3 true WO2006106244A3 (fr) | 2007-09-13 |
Family
ID=35544328
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/FR2006/000780 WO2006106244A2 (fr) | 2005-04-08 | 2006-04-07 | PROCEDE DE PREPARATION DE β-AMINOESTERS OU α-, β-DIAMINOESTERS DERIVES DE LA SERINE |
Country Status (2)
Country | Link |
---|---|
FR (1) | FR2884249A1 (fr) |
WO (1) | WO2006106244A2 (fr) |
-
2005
- 2005-04-08 FR FR0503537A patent/FR2884249A1/fr active Pending
-
2006
- 2006-04-07 WO PCT/FR2006/000780 patent/WO2006106244A2/fr active Application Filing
Non-Patent Citations (2)
Title |
---|
P. GMEINER, A. KÄRTNER AND D. JUNGE: "Practical EPC Synthesis of 1,2- and 1,3-diamino alcohols", TETRAHEDRON LETTERS, vol. 34, no. 27, 1993, Great Britain, pages 4325 - 4326, XP002365984 * |
SOMEKH, L. AND SHANZER, A.: "Facile Stereospecific Synthesis of alpha-fluoro-beta-amino Acids", J. AM. CHEM. SOC., vol. 104, 1982, pages 5836 - 5837, XP002365983 * |
Also Published As
Publication number | Publication date |
---|---|
FR2884249A1 (fr) | 2006-10-13 |
WO2006106244A2 (fr) | 2006-10-12 |
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