WO2003042189A1 - Procede de preparation d'un ester de l'acide 1-h-1,2,4-triazole-3-carboxylique - Google Patents

Procede de preparation d'un ester de l'acide 1-h-1,2,4-triazole-3-carboxylique Download PDF

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Publication number
WO2003042189A1
WO2003042189A1 PCT/JP2002/011981 JP0211981W WO03042189A1 WO 2003042189 A1 WO2003042189 A1 WO 2003042189A1 JP 0211981 W JP0211981 W JP 0211981W WO 03042189 A1 WO03042189 A1 WO 03042189A1
Authority
WO
WIPO (PCT)
Prior art keywords
triazole
compound
carboxylic acid
producing
acid ester
Prior art date
Application number
PCT/JP2002/011981
Other languages
English (en)
French (fr)
Inventor
Sumio Shimizu
Yutaka Nishino
Kazuhiro Yoshida
Original Assignee
Shionogi & Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co., Ltd. filed Critical Shionogi & Co., Ltd.
Priority to JP2003544025A priority Critical patent/JPWO2003042189A1/ja
Publication of WO2003042189A1 publication Critical patent/WO2003042189A1/ja

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • AIDS & HIV (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PCT/JP2002/011981 2001-11-15 2002-11-15 Procede de preparation d'un ester de l'acide 1-h-1,2,4-triazole-3-carboxylique WO2003042189A1 (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2003544025A JPWO2003042189A1 (ja) 2001-11-15 2002-11-15 １−ｈ−１，２，４−トリアゾール−３−カルボン酸エステルの製造法

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2001350843 2001-11-15
JP2001-350843 2001-11-15

Publications (1)

Publication Number Publication Date
WO2003042189A1 true WO2003042189A1 (fr) 2003-05-22

Family

ID=19163258

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/JP2002/011981 WO2003042189A1 (fr) 2001-11-15 2002-11-15 Procede de preparation d'un ester de l'acide 1-h-1,2,4-triazole-3-carboxylique

Country Status (3)

Country Link
JP (1) JPWO2003042189A1 (ja)
TW (1) TW200407132A (ja)
WO (1) WO2003042189A1 (ja)

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4639266A (en) * 1984-09-11 1987-01-27 Hoechst Aktiengesellschaft Plant protection agents based on 1,2,4-triazole derivatives and also new derivatives of 1,2,4-triazole
DE4225778A1 (de) * 1992-08-04 1994-02-17 Hoechst Ag 1,2,4-Triazolyl-3-carbonsäure-4-aminopiperidide, Verfahren zu ihrer Herstellung, sie enthaltende Mittel und ihre Verwendung als Schädlingsbekämpfungsmittel, insbesondere Fungizide
WO2000039086A1 (fr) * 1998-12-25 2000-07-06 Shionogi & Co., Ltd. Composes heterocycliques aromatiques possedant des activites inhibitrices de l'integrase du vih

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4639266A (en) * 1984-09-11 1987-01-27 Hoechst Aktiengesellschaft Plant protection agents based on 1,2,4-triazole derivatives and also new derivatives of 1,2,4-triazole
DE4225778A1 (de) * 1992-08-04 1994-02-17 Hoechst Ag 1,2,4-Triazolyl-3-carbonsäure-4-aminopiperidide, Verfahren zu ihrer Herstellung, sie enthaltende Mittel und ihre Verwendung als Schädlingsbekämpfungsmittel, insbesondere Fungizide
WO2000039086A1 (fr) * 1998-12-25 2000-07-06 Shionogi & Co., Ltd. Composes heterocycliques aromatiques possedant des activites inhibitrices de l'integrase du vih

Also Published As

Publication number Publication date
JPWO2003042189A1 (ja) 2005-03-10
TW200407132A (en) 2004-05-16

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