WO2003028710A3 - Verbindungen zur reduzierung übermässiger nahrungsaufnahme - Google Patents
Verbindungen zur reduzierung übermässiger nahrungsaufnahme Download PDFInfo
- Publication number
- WO2003028710A3 WO2003028710A3 PCT/EP2002/010805 EP0210805W WO03028710A3 WO 2003028710 A3 WO2003028710 A3 WO 2003028710A3 EP 0210805 W EP0210805 W EP 0210805W WO 03028710 A3 WO03028710 A3 WO 03028710A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- food
- compounds
- excessive intake
- reducing excessive
- reducing
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/428—Thiazoles condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Engineering & Computer Science (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Obesity (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Endocrinology (AREA)
- Child & Adolescent Psychology (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Priority Applications (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2003532043A JP2005504110A (ja) | 2001-09-28 | 2002-09-26 | 食物の過剰摂取量を低減させる化合物 |
AU2002337135A AU2002337135A1 (en) | 2001-09-28 | 2002-09-26 | Compounds for reducing excessive intake of food |
EP02772350A EP1438047A2 (de) | 2001-09-28 | 2002-09-26 | Verbindungen zur reduzierung übermässiger nahrungsaufnahme |
CA002461586A CA2461586A1 (en) | 2001-09-28 | 2002-09-26 | Compounds for the reduction of excessive food intake |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10148233A DE10148233A1 (de) | 2001-09-28 | 2001-09-28 | Verbindungen zur Reduzierung übermäßiger Nahrungsaufnahme |
DE10148233.7 | 2001-09-28 |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2003028710A2 WO2003028710A2 (de) | 2003-04-10 |
WO2003028710A3 true WO2003028710A3 (de) | 2003-09-12 |
Family
ID=7700867
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/EP2002/010805 WO2003028710A2 (de) | 2001-09-28 | 2002-09-26 | Verbindungen zur reduzierung übermässiger nahrungsaufnahme |
Country Status (9)
Country | Link |
---|---|
US (7) | US20030087941A1 (de) |
EP (1) | EP1438047A2 (de) |
JP (1) | JP2005504110A (de) |
AU (1) | AU2002337135A1 (de) |
CA (1) | CA2461586A1 (de) |
DE (1) | DE10148233A1 (de) |
PE (1) | PE20030628A1 (de) |
UY (1) | UY27459A1 (de) |
WO (1) | WO2003028710A2 (de) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10148233A1 (de) * | 2001-09-28 | 2003-04-10 | Boehringer Ingelheim Pharma | Verbindungen zur Reduzierung übermäßiger Nahrungsaufnahme |
DE10312809A1 (de) * | 2003-03-21 | 2004-09-30 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Pramipexol zur Reduzierung übermäßiger Nahrungsaufnahme bei Kindern |
DE10334188B4 (de) * | 2003-07-26 | 2007-07-05 | Schwarz Pharma Ag | Verwendung von Rotigotin zur Behandlung von Depressionen |
DE10334187A1 (de) * | 2003-07-26 | 2005-03-03 | Schwarz Pharma Ag | Substituierte 2-Aminotetraline zur Behandlung von Depressionen |
NZ547152A (en) * | 2003-10-16 | 2009-12-24 | Neurosearch As | Pharmaceutical composition comprising a monoamine neurotransmitter re-uptake inhibitor and an acetylcholinesterase inhibitor |
DE10361258A1 (de) * | 2003-12-24 | 2005-07-28 | Schwarz Pharma Ag | Verwendung von substituierten 2-Aminotetralinen zur vorbeugenden Behandlung von Morbus Parkinson |
CA2553649A1 (en) * | 2004-01-22 | 2005-08-04 | Neurosearch A/S | Compounds for the sustained reduction of body weight |
EP1708707A1 (de) * | 2004-01-22 | 2006-10-11 | Neurosearch A/S | Pharmazeutische zusammensetzung mit einem monoamin-neurotransmitter-wiederaufnahmehemmer und einem n-methyl-d-aspartat (nmda)-rezeptorantagonisten |
DE102004014841B4 (de) * | 2004-03-24 | 2006-07-06 | Schwarz Pharma Ag | Verwendung von Rotigotin zur Behandlung und Prävention des Parkinson-Plus-Syndroms |
US7754770B2 (en) * | 2005-06-27 | 2010-07-13 | Mason Chemical Company | Antimicrobial composition |
TWI392670B (zh) * | 2006-06-22 | 2013-04-11 | Ucb Pharma Gmbh | 經取代的2-胺基萘滿之於製造用於預防、減緩及/或治療各種類型疼痛之藥物上的用途 |
US20080254118A1 (en) * | 2007-04-11 | 2008-10-16 | Hans-Werner Wernersbach | Process for preparing pramipexole dihydrochloride tablets |
US20080254117A1 (en) * | 2007-04-10 | 2008-10-16 | Noel Cotton | Process for preparing pramipexole dihydrochloride tablets |
EP2193024A4 (de) * | 2007-09-25 | 2013-11-06 | Entrotech Inc | Farbersatzfilme, verbundstoffe daraus und verwandte verfahren |
CA2622696A1 (en) * | 2007-11-05 | 2009-05-05 | Diane Mcintosh | Methods and compositions for retarding weight gain associated with use of atypical antipsychotic drugs |
WO2010030887A1 (en) | 2008-09-11 | 2010-03-18 | Catholic Healthcare West | Nicotinic attenuation of cns inflammation and autoimmunity |
US20130045987A1 (en) * | 2010-05-03 | 2013-02-21 | Dignity Health | Novel methods of use of tetrahydroberberine (thb) |
RU2665134C2 (ru) * | 2012-05-07 | 2018-08-28 | Омерос Корпорейшн | Лечение зависимости и расстройств побуждений с применением ингибиторов фдэ7 |
KR102309836B1 (ko) | 2013-07-18 | 2021-10-12 | 에스케이바이오팜 주식회사 | 비만의 치료 |
Citations (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4855306A (en) * | 1987-04-10 | 1989-08-08 | Sandoz Ltd. | Uses of dopamine receptor agonists |
WO1990013294A1 (en) * | 1989-05-09 | 1990-11-15 | Whitby Research, Inc. | A method of reducing body weight and food intake using a dopamine d2 receptor agonist |
WO1999025328A1 (en) * | 1997-11-14 | 1999-05-27 | Warner-Lambert Company | (+)-ephedrine as a sympathomimetic drug |
WO1999059563A2 (en) * | 1998-05-15 | 1999-11-25 | Pharmacia & Upjohn Company | Cabergoline and pramipexole for treating cns diseases, especially parkinson's disease |
EP1051971A1 (de) * | 1999-05-10 | 2000-11-15 | Pierce Management, L.L.P. | Pflaster und Verfahren zur transdermalen Verabreichung von Bupropion als freie base |
EP1099441A2 (de) * | 1999-11-10 | 2001-05-16 | Pfizer Products Inc. | Zusammensetzungen enthaltend Apo-B-Sekretion/MTP Inhibitoren und Mittel gegen Fettleibigkeit und deren Verwendung |
WO2001041763A1 (en) * | 1999-12-10 | 2001-06-14 | University Of Cincinnati | Treatment of addiction disorders |
US20010016582A1 (en) * | 1997-04-28 | 2001-08-23 | Anthony H. Cincotta | Method and composition for the treatment of lipid and glucose metabolism disorders |
WO2002060423A2 (en) * | 2001-01-29 | 2002-08-08 | Otsuka Pharmaceutical Co., Ltd. | Substituted carbostyril derivatives as 5-ht1a receptor subtype agonists |
WO2002069974A1 (en) * | 2001-03-05 | 2002-09-12 | Andrew Holman | Administration of sleep restorative agents |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6004990A (en) * | 1994-06-03 | 1999-12-21 | Zebra Pharmaceuticals | Meta substituted arylalkylamines and therapeutic and diagnostic uses therefor |
DE10148233A1 (de) * | 2001-09-28 | 2003-04-10 | Boehringer Ingelheim Pharma | Verbindungen zur Reduzierung übermäßiger Nahrungsaufnahme |
-
2001
- 2001-09-28 DE DE10148233A patent/DE10148233A1/de not_active Withdrawn
-
2002
- 2002-09-26 EP EP02772350A patent/EP1438047A2/de not_active Withdrawn
- 2002-09-26 JP JP2003532043A patent/JP2005504110A/ja active Pending
- 2002-09-26 CA CA002461586A patent/CA2461586A1/en not_active Abandoned
- 2002-09-26 WO PCT/EP2002/010805 patent/WO2003028710A2/de active Application Filing
- 2002-09-26 AU AU2002337135A patent/AU2002337135A1/en not_active Abandoned
- 2002-09-27 US US10/259,118 patent/US20030087941A1/en not_active Abandoned
- 2002-09-27 UY UY27459A patent/UY27459A1/es not_active Application Discontinuation
- 2002-09-27 PE PE2002000959A patent/PE20030628A1/es not_active Application Discontinuation
-
2004
- 2004-09-07 US US10/935,508 patent/US20050032812A1/en not_active Abandoned
- 2004-09-07 US US10/935,507 patent/US20050032843A1/en not_active Abandoned
-
2005
- 2005-10-06 US US11/244,806 patent/US20060030607A1/en not_active Abandoned
-
2006
- 2006-06-26 US US11/423,159 patent/US20060223869A1/en not_active Abandoned
-
2007
- 2007-09-18 US US11/857,038 patent/US20080051444A1/en not_active Abandoned
- 2007-09-18 US US11/857,016 patent/US20080051443A1/en not_active Abandoned
Patent Citations (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4855306A (en) * | 1987-04-10 | 1989-08-08 | Sandoz Ltd. | Uses of dopamine receptor agonists |
WO1990013294A1 (en) * | 1989-05-09 | 1990-11-15 | Whitby Research, Inc. | A method of reducing body weight and food intake using a dopamine d2 receptor agonist |
US20010016582A1 (en) * | 1997-04-28 | 2001-08-23 | Anthony H. Cincotta | Method and composition for the treatment of lipid and glucose metabolism disorders |
WO1999025328A1 (en) * | 1997-11-14 | 1999-05-27 | Warner-Lambert Company | (+)-ephedrine as a sympathomimetic drug |
WO1999059563A2 (en) * | 1998-05-15 | 1999-11-25 | Pharmacia & Upjohn Company | Cabergoline and pramipexole for treating cns diseases, especially parkinson's disease |
EP1051971A1 (de) * | 1999-05-10 | 2000-11-15 | Pierce Management, L.L.P. | Pflaster und Verfahren zur transdermalen Verabreichung von Bupropion als freie base |
EP1099441A2 (de) * | 1999-11-10 | 2001-05-16 | Pfizer Products Inc. | Zusammensetzungen enthaltend Apo-B-Sekretion/MTP Inhibitoren und Mittel gegen Fettleibigkeit und deren Verwendung |
WO2001041763A1 (en) * | 1999-12-10 | 2001-06-14 | University Of Cincinnati | Treatment of addiction disorders |
WO2002060423A2 (en) * | 2001-01-29 | 2002-08-08 | Otsuka Pharmaceutical Co., Ltd. | Substituted carbostyril derivatives as 5-ht1a receptor subtype agonists |
WO2002069974A1 (en) * | 2001-03-05 | 2002-09-12 | Andrew Holman | Administration of sleep restorative agents |
Non-Patent Citations (7)
Title |
---|
DOMINO EDWARD F ET AL: "Talipexole or pramipexole combinations with chloro-APB (SKF 82958) in MPTP-induced hemiparkinsonian monkeys.", EUROPEAN JOURNAL OF PHARMACOLOGY, vol. 325, no. 2-3, 1997, pages 137 - 144, XP001121783, ISSN: 0014-2999 * |
EMILIEN G ET AL: "DOPAMINE D3 AGONISTS", EXPERT OPINION ON THERAPEUTIC PATENTS, ASHLEY PUBLICATIONS, GB, vol. 11, no. 11, 2001, pages 1713 - 1728, XP001057496, ISSN: 1354-3776 * |
FERNANDEZ-LOPEZ J-A ET AL: "PHARMACOLOGICAL APPROACHES FOR THE TREATMENT OF OBESITY", DRUGS, ADIS INTERNATIONAL LTD, AT, vol. 62, no. 6, 2002, pages 915 - 944, XP009001892, ISSN: 0012-6667 * |
IHARA T ET AL: "SINGLE AND REPEATED ORAL DOSE TOXICITY STUDIES WITH TALIPEXOLE DIHYDROCHLORIDE (B-HT 920 CL2) IN CYNOMOLGUS MONKEYS", OYO YAKURI - PHARMACOMETRICS, XX, XX, vol. 46, no. 6, 1993, pages 401 - 416, XP009001922, ISSN: 0300-8533 * |
NAGASHIMA MARIKO ET AL: "Hyperthermia induced by the dopamine D-1 receptor agonist SKF 38393 in combination with the dopamine D-2 receptor agonist talipexole in the rat.", PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, vol. 43, no. 4, 1992, pages 993 - 997, XP009003332, ISSN: 0091-3057 * |
TERRY P ET AL: "DOPAMINE RECEPTOR SUBTYPE AGONISTS AND FEEDING BEHAVIOR", OBESITY RESEARCH, BATON ROUGE, LA,, US, vol. 3, no. SUPPL 4, November 1995 (1995-11-01), pages 515S - 523S, XP001062494, ISSN: 1071-7323 * |
WILLNER P ET AL: "Reversal of stress-induced anhedonia by the dopamine receptor agonist, pramipexole.", PSYCHOPHARMACOLOGY. GERMANY AUG 1994, vol. 115, no. 4, August 1994 (1994-08-01), pages 454 - 462, XP009003272, ISSN: 0033-3158 * |
Also Published As
Publication number | Publication date |
---|---|
AU2002337135A1 (en) | 2003-04-14 |
US20030087941A1 (en) | 2003-05-08 |
PE20030628A1 (es) | 2003-07-15 |
EP1438047A2 (de) | 2004-07-21 |
WO2003028710A2 (de) | 2003-04-10 |
US20060223869A1 (en) | 2006-10-05 |
US20060030607A1 (en) | 2006-02-09 |
US20080051444A1 (en) | 2008-02-28 |
US20080051443A1 (en) | 2008-02-28 |
DE10148233A1 (de) | 2003-04-10 |
US20050032843A1 (en) | 2005-02-10 |
JP2005504110A (ja) | 2005-02-10 |
UY27459A1 (es) | 2003-04-30 |
CA2461586A1 (en) | 2003-04-10 |
US20050032812A1 (en) | 2005-02-10 |
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