WO2002062803A1 - Thienopyrimidine derivative - Google Patents
Thienopyrimidine derivative Download PDFInfo
- Publication number
- WO2002062803A1 WO2002062803A1 PCT/JP2002/001008 JP0201008W WO02062803A1 WO 2002062803 A1 WO2002062803 A1 WO 2002062803A1 JP 0201008 W JP0201008 W JP 0201008W WO 02062803 A1 WO02062803 A1 WO 02062803A1
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- thienopyrimidine derivative
- derivative
- thienopyrimidine
- medicine
- salt
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Abstract
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2001-32121 | 2001-02-08 | ||
JP2001032121 | 2001-02-08 |
Publications (1)
Publication Number | Publication Date |
---|---|
WO2002062803A1 true WO2002062803A1 (en) | 2002-08-15 |
Family
ID=18896101
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/JP2002/001008 WO2002062803A1 (en) | 2001-02-08 | 2002-02-07 | Thienopyrimidine derivative |
Country Status (1)
Country | Link |
---|---|
WO (1) | WO2002062803A1 (en) |
Cited By (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2004029060A1 (en) * | 2002-09-26 | 2004-04-08 | Nihon Nohyaku Co., Ltd. | Novel herbicides, usage thereof, novel thienopyrimidine derivatives, intermediates of the same, and process for production thereof |
WO2006002051A1 (en) * | 2004-06-15 | 2006-01-05 | Schering Corporation | Tricyclic compounds and their use as mglur1 antagonists |
WO2007024593A1 (en) * | 2005-08-19 | 2007-03-01 | Schering Corporation | Fused tricyclic mglur1 antagonists as therapeutic agents |
WO2007072090A1 (en) * | 2005-12-20 | 2007-06-28 | Richter Gedeon Nyrt. | Thienopyridine derivatives as modulators of metabotropic glutamate receptors |
US7482360B2 (en) | 2005-09-23 | 2009-01-27 | Schering Corporation | Fused tetracyclic mGluR1 antagonists as therapeutic agents |
US7598259B2 (en) | 2004-06-15 | 2009-10-06 | Schering Corporation | mGluR1 antagonists as therapeutic agents |
US7939657B2 (en) * | 2003-10-29 | 2011-05-10 | Elan Pharmaceuticals, Inc. | N-substituted benzene sulfonamides |
US8691833B2 (en) | 2007-02-23 | 2014-04-08 | Merck Sharp & Dohme Corp. | Heterocyclic aspartyl protease inhibitors |
WO2015056771A1 (en) | 2013-10-17 | 2015-04-23 | アステラス製薬株式会社 | Sulfur-containing bicyclic compound |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1998006724A1 (en) * | 1996-08-09 | 1998-02-19 | Yamanouchi Pharmaceutical Co., Ltd. | Metabotropic glutamate receptor agonists |
JPH11189596A (en) * | 1997-12-25 | 1999-07-13 | Yamanouchi Pharmaceut Co Ltd | Metabotropic glutamate receptor agonist and new imidazobenzothiazole derivative |
WO2000059913A1 (en) * | 1999-04-06 | 2000-10-12 | Yamanouchi Pharmaceutical Co., Ltd. | Novel thiazolobenzimidazole derivatives |
-
2002
- 2002-02-07 WO PCT/JP2002/001008 patent/WO2002062803A1/en active Application Filing
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1998006724A1 (en) * | 1996-08-09 | 1998-02-19 | Yamanouchi Pharmaceutical Co., Ltd. | Metabotropic glutamate receptor agonists |
JPH11189596A (en) * | 1997-12-25 | 1999-07-13 | Yamanouchi Pharmaceut Co Ltd | Metabotropic glutamate receptor agonist and new imidazobenzothiazole derivative |
WO2000059913A1 (en) * | 1999-04-06 | 2000-10-12 | Yamanouchi Pharmaceutical Co., Ltd. | Novel thiazolobenzimidazole derivatives |
Cited By (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2004029060A1 (en) * | 2002-09-26 | 2004-04-08 | Nihon Nohyaku Co., Ltd. | Novel herbicides, usage thereof, novel thienopyrimidine derivatives, intermediates of the same, and process for production thereof |
US7939657B2 (en) * | 2003-10-29 | 2011-05-10 | Elan Pharmaceuticals, Inc. | N-substituted benzene sulfonamides |
WO2006002051A1 (en) * | 2004-06-15 | 2006-01-05 | Schering Corporation | Tricyclic compounds and their use as mglur1 antagonists |
US7989464B2 (en) | 2004-06-15 | 2011-08-02 | Schering Corporation | mGluR1 antagonists as therapeutic agents |
US7485648B2 (en) | 2004-06-15 | 2009-02-03 | Schering Corporation | mGluR1 antagonists as therapeutic agents |
US7598259B2 (en) | 2004-06-15 | 2009-10-06 | Schering Corporation | mGluR1 antagonists as therapeutic agents |
WO2007024593A1 (en) * | 2005-08-19 | 2007-03-01 | Schering Corporation | Fused tricyclic mglur1 antagonists as therapeutic agents |
US7767815B2 (en) | 2005-08-19 | 2010-08-03 | Schering Corporation | Fused tricyclic mGluR1 antagonists as therapeutic agents |
US7482360B2 (en) | 2005-09-23 | 2009-01-27 | Schering Corporation | Fused tetracyclic mGluR1 antagonists as therapeutic agents |
WO2007072090A1 (en) * | 2005-12-20 | 2007-06-28 | Richter Gedeon Nyrt. | Thienopyridine derivatives as modulators of metabotropic glutamate receptors |
US8691833B2 (en) | 2007-02-23 | 2014-04-08 | Merck Sharp & Dohme Corp. | Heterocyclic aspartyl protease inhibitors |
US8691831B2 (en) | 2007-02-23 | 2014-04-08 | Merck Sharp & Dohme Corp. | Heterocyclic aspartyl protease inhibitors |
WO2015056771A1 (en) | 2013-10-17 | 2015-04-23 | アステラス製薬株式会社 | Sulfur-containing bicyclic compound |
US9051339B2 (en) | 2013-10-17 | 2015-06-09 | Astellas Pharma Inc. | Sulfur-containing bicyclic compound |
CN105636965A (en) * | 2013-10-17 | 2016-06-01 | 安斯泰来制药株式会社 | Sulfur-containing bicyclic compound |
KR20160071408A (en) | 2013-10-17 | 2016-06-21 | 아스텔라스세이야쿠 가부시키가이샤 | Sulfur-containing bicyclic compound |
US9642852B2 (en) | 2013-10-17 | 2017-05-09 | Astellas Pharma Inc. | Sulfur-containing bicyclic compound |
CN105636965B (en) * | 2013-10-17 | 2017-11-24 | 安斯泰来制药株式会社 | The ring type compound of sulfur-bearing two |
EA029075B1 (en) * | 2013-10-17 | 2018-02-28 | Астеллас Фарма Инк. | Sulfur-containing bicyclic compound |
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