WO2001090102A3 - 6-heteroclyclyl-3-oxo-3,4-dihydro-quinoxalines - Google Patents

6-heteroclyclyl-3-oxo-3,4-dihydro-quinoxalines Download PDF

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Publication number
WO2001090102A3
WO2001090102A3 PCT/EP2001/005382 EP0105382W WO0190102A3 WO 2001090102 A3 WO2001090102 A3 WO 2001090102A3 EP 0105382 W EP0105382 W EP 0105382W WO 0190102 A3 WO0190102 A3 WO 0190102A3
Authority
WO
WIPO (PCT)
Prior art keywords
quinoxalines
heterocyclyl
dihydro
oxo
relates
Prior art date
Application number
PCT/EP2001/005382
Other languages
German (de)
English (en)
Other versions
WO2001090102A2 (fr
Inventor
Hans-Georg Schwarz
Karl-Heinz Linker
Mark Wilhelm Drewes
Peter Dahmen
Dieter Feucht
Rolf Pontzen
Original Assignee
Bayer Ag
Hans-Georg Schwarz
Karl-Heinz Linker
Mark Wilhelm Drewes
Peter Dahmen
Dieter Feucht
Rolf Pontzen
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10055499A external-priority patent/DE10055499A1/de
Application filed by Bayer Ag, Hans-Georg Schwarz, Karl-Heinz Linker, Mark Wilhelm Drewes, Peter Dahmen, Dieter Feucht, Rolf Pontzen filed Critical Bayer Ag
Priority to AU65944/01A priority Critical patent/AU6594401A/en
Publication of WO2001090102A2 publication Critical patent/WO2001090102A2/fr
Publication of WO2001090102A3 publication Critical patent/WO2001090102A3/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/60—1,4-Diazines; Hydrogenated 1,4-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D249/12—Oxygen or sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

L'invention concerne des composés correspondant à la formule générale (I), dans laquelle R?1, R2, R3¿ et Z ont les significations données dans la description, ainsi qu'un procédé et de nouveaux produits intermédiaires permettant de produire ces composés, et leur utilisation comme agents phytosanitaires, en particulier comme herbicides.
PCT/EP2001/005382 2000-05-24 2001-05-11 6-heteroclyclyl-3-oxo-3,4-dihydro-quinoxalines WO2001090102A2 (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU65944/01A AU6594401A (en) 2000-05-24 2001-05-11 6-heterocyclyl-3-oxo-3,4-dihydro-quinoxalines

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE10025624 2000-05-24
DE10025624.4 2000-05-24
DE10055499A DE10055499A1 (de) 2000-05-24 2000-11-09 6-Heterocyclyl-3-oxo-3,4-dihydro-chinoxaline
DE10055499.7 2000-11-09

Publications (2)

Publication Number Publication Date
WO2001090102A2 WO2001090102A2 (fr) 2001-11-29
WO2001090102A3 true WO2001090102A3 (fr) 2002-06-20

Family

ID=26005810

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2001/005382 WO2001090102A2 (fr) 2000-05-24 2001-05-11 6-heteroclyclyl-3-oxo-3,4-dihydro-quinoxalines

Country Status (2)

Country Link
AU (1) AU6594401A (fr)
WO (1) WO2001090102A2 (fr)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BRPI0815327A2 (pt) 2007-08-31 2015-12-15 Purdue Pharma Lp "compostos de piperidina do tipo quinoxalina substituída e os usos destes"
RU2500678C2 (ru) 2008-07-21 2013-12-10 Пэдью Фарма Л.П. Замещенные хиноксалинового типа мостиковые пиперидиновые соединения и их применение
JP5872585B2 (ja) 2010-12-22 2016-03-01 パーデュー、ファーマ、リミテッド、パートナーシップ リン置換キノキサリンタイプピペリジン化合物とその使用
US9290488B2 (en) 2011-12-01 2016-03-22 Purdue Pharma L.P. Azetidine-substituted quinoxalines as opioid receptor like-1 modulators
EP2822931B1 (fr) 2012-03-09 2017-05-03 Inception 2, Inc. Composés de triazolone et leurs utilisations
US9085561B2 (en) 2012-07-30 2015-07-21 Purdue Pharma L.P. Cyclic urea- or lactam-substituted quinoxaline-type piperidines as ORL-1 modulators
EP2935228B9 (fr) 2012-12-20 2017-12-06 Inception 2, Inc. Composés de triazolone et leurs utilisations
US9090618B2 (en) 2012-12-27 2015-07-28 Purdue Pharma L.P. Substituted benzimidazole-type piperidine compounds and uses thereof
US9963458B2 (en) 2012-12-27 2018-05-08 Purdue Pharma L.P. Indole and indoline-type piperidine compounds and uses thereof
US9040533B2 (en) 2012-12-27 2015-05-26 Purdue Pharma L.P. Oxime-substituted-quinoxaline-type piperidine compounds as ORL-1 modulators
US9951038B2 (en) 2012-12-27 2018-04-24 Purdue Pharma L.P. Quinazolin-4(3H)-one-type piperidine compounds and uses thereof
CN105579440A (zh) 2013-09-06 2016-05-11 因森普深2公司 三唑酮化合物及其应用

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0311135A2 (fr) * 1987-10-09 1989-04-12 Schering Aktiengesellschaft Azoles et azines hétérocycliques substituées, procédé pour leur préparation et leur utilisation comme agents à activité herbicide
EP0597360A1 (fr) * 1992-11-12 1994-05-18 Bayer Ag N-phényle-triazolin (thi)ones substitués, procédés et produits intermédiaires pour leur préparation et leur utilisation comme herbicides, insecticides et acaricides

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0311135A2 (fr) * 1987-10-09 1989-04-12 Schering Aktiengesellschaft Azoles et azines hétérocycliques substituées, procédé pour leur préparation et leur utilisation comme agents à activité herbicide
EP0597360A1 (fr) * 1992-11-12 1994-05-18 Bayer Ag N-phényle-triazolin (thi)ones substitués, procédés et produits intermédiaires pour leur préparation et leur utilisation comme herbicides, insecticides et acaricides

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
LYGA, J.W. ET AL.: "Structural replacements for the benzoxazinone protox inhibitors", PESTICIDE SCIENCE, vol. 55, 1999, pages 281 - 287, XP002176842 *

Also Published As

Publication number Publication date
WO2001090102A2 (fr) 2001-11-29
AU6594401A (en) 2001-12-03

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