WO2000063176A3 - Disubstituierte Pyridine und Pyrimidine als Herbizide und Fungizide - Google Patents

Disubstituierte Pyridine und Pyrimidine als Herbizide und Fungizide Download PDF

Info

Publication number
WO2000063176A3
WO2000063176A3 PCT/EP2000/002979 EP0002979W WO0063176A3 WO 2000063176 A3 WO2000063176 A3 WO 2000063176A3 EP 0002979 W EP0002979 W EP 0002979W WO 0063176 A3 WO0063176 A3 WO 0063176A3
Authority
WO
WIPO (PCT)
Prior art keywords
substituted alkyl
possibly substituted
cycloalkyl
pyrimidines
fungicides
Prior art date
Application number
PCT/EP2000/002979
Other languages
English (en)
French (fr)
Other versions
WO2000063176A2 (de
Inventor
Otto Schallner
Kristian Kather
Ernsrt Rudolf F Gesing
Mark Wilhelm Drewes
Dieter Feucht
Rolf Pontzen
Ingo Wetcholowsky
Gerd Haenssler
Astrid Mauler-Machnik
Original Assignee
Bayer Ag
Otto Schallner
Kristian Kather
Gesing Ernst Rudolf F
Mark Wilhelm Drewes
Dieter Feucht
Rolf Pontzen
Ingo Wetcholowsky
Gerd Haenssler
Astrid Mauler-Machnik
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag, Otto Schallner, Kristian Kather, Gesing Ernst Rudolf F, Mark Wilhelm Drewes, Dieter Feucht, Rolf Pontzen, Ingo Wetcholowsky, Gerd Haenssler, Astrid Mauler-Machnik filed Critical Bayer Ag
Priority to AU45427/00A priority Critical patent/AU4542700A/en
Publication of WO2000063176A2 publication Critical patent/WO2000063176A2/de
Publication of WO2000063176A3 publication Critical patent/WO2000063176A3/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/26—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/34—One oxygen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/38—One sulfur atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)

Abstract

Die Erfindung betrifft neue jeweils disubstituierte Pyridine und Pyrimidine der allgemeinen Formel (I), in welcher A für N oder CH steht; R1 für Hydroxy, Mercapto, Amino, Cyano, Carboxy, Carbamoyl, Thiocarbamoyl, Halogen, oder für jeweils gegebenenfalls substituiertes Alkyl, Alkoxy, Alkoxycarbonyl, Alkylthio, Alkylsulfinyl, Alkylsulfonyl, Alkylamino, Dialkylamino, Alkenyloxy, Alkenylthio, Alkenylamino, Alkinyloxy, Alkinylthio, Alkinylamino oder Cycloalkyl steht; R2 für Wasserstoff, Hydroxy, Formyloxy, Halogen, oder für gegebenenfalls substituiertes Alkyl, Alkoxy, Alkylcarbonyloxy, Alkoxycarbonyloxy, Alkylaminocarbonyloxy, Dialkylaminocarbonyloxy, Alkenyloxy oder Alkinyloxy steht; R3 für jeweils gegebenenfalls substituiertes Alkyl, Alkenyl, Cycloalkyl, Cycloalkylalkyl, Aryl oder Arylalkyl steht; und R4 für jeweils gegebenenfalls substituiertes Alkyl, Alkenyl, Cycloalkyl, Cycloalkylalkyl, Aryl oder Arylalkyl steht, sowie Verfahren zu ihrer Herstellung und ihre Verwendung als Pflanzenbehandlungsmittel, insbesondere als Herbizide und als Fungizide.
PCT/EP2000/002979 1999-04-16 2000-04-04 Disubstituierte pyridine und pyrimidine als herbizide und fungizide WO2000063176A2 (de)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU45427/00A AU4542700A (en) 1999-04-16 2000-04-04 Disubstituted pyridines and pyrimidines

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE1999117160 DE19917160A1 (de) 1999-04-16 1999-04-16 Disubstituierte Pyridine und Pyrimidine
DE19917160.2 1999-04-16

Publications (2)

Publication Number Publication Date
WO2000063176A2 WO2000063176A2 (de) 2000-10-26
WO2000063176A3 true WO2000063176A3 (de) 2001-08-23

Family

ID=7904750

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2000/002979 WO2000063176A2 (de) 1999-04-16 2000-04-04 Disubstituierte pyridine und pyrimidine als herbizide und fungizide

Country Status (3)

Country Link
AU (1) AU4542700A (de)
DE (1) DE19917160A1 (de)
WO (1) WO2000063176A2 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20160145640A (ko) 2014-04-15 2016-12-20 다우 아그로사이언시즈 엘엘씨 살진균제로서의 금속효소 억제제 화합물
US10781177B2 (en) 2016-03-09 2020-09-22 Nippon Soda Co., Ltd. Pyridine compound and use thereof

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1770288A1 (de) * 1967-04-27 1972-04-13 Fil Lilly And Co Substituierte 5-Pyrimidinverbindungen
EP0058347A2 (de) * 1981-02-14 1982-08-25 Bayer Ag Benzyl-pyrimidinylalkyl-ether, Verfahren zu ihrer Herstellung, ihre Verwendung als Pflanzenwachstumsregulatoren und Fungizide sowie Zwischenprodukte und deren Herstellung
EP0069330A1 (de) * 1981-07-08 1983-01-12 BASF Aktiengesellschaft Pyridincarbinole, Verfahren zu ihrer Herstellung und diese enthaltende Fungizide
EP0359077A1 (de) * 1988-09-15 1990-03-21 Bayer Ag Substituierte Pyrimidyl- bzw. Pyridylalkinole, Verfahren zu ihrer Herstellung und ihre Verwendung in Schädlingsbekämpfungsmitteln
EP0713872A1 (de) * 1993-08-10 1996-05-29 Nissan Chemical Industries, Limited Neues pyrimidinderivat, herbizid und pflanzenwachstums-regulator

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1770288A1 (de) * 1967-04-27 1972-04-13 Fil Lilly And Co Substituierte 5-Pyrimidinverbindungen
EP0058347A2 (de) * 1981-02-14 1982-08-25 Bayer Ag Benzyl-pyrimidinylalkyl-ether, Verfahren zu ihrer Herstellung, ihre Verwendung als Pflanzenwachstumsregulatoren und Fungizide sowie Zwischenprodukte und deren Herstellung
EP0069330A1 (de) * 1981-07-08 1983-01-12 BASF Aktiengesellschaft Pyridincarbinole, Verfahren zu ihrer Herstellung und diese enthaltende Fungizide
EP0359077A1 (de) * 1988-09-15 1990-03-21 Bayer Ag Substituierte Pyrimidyl- bzw. Pyridylalkinole, Verfahren zu ihrer Herstellung und ihre Verwendung in Schädlingsbekämpfungsmitteln
EP0713872A1 (de) * 1993-08-10 1996-05-29 Nissan Chemical Industries, Limited Neues pyrimidinderivat, herbizid und pflanzenwachstums-regulator

Non-Patent Citations (3)

* Cited by examiner, † Cited by third party
Title
D.J.BROWN: "The Dimroth Rearrangement. Part XVI. A New General Synthesis and Rearrangement of C-Alkylated 1,6-Dihydro-6-imino-1-methylpyrimidines", JOURNAL OF THE CHEMICAL SOCIETY, PERKIN TRANSACTION I, 1974, pages 372 - 378, XP002154127 *
E.C. TAYLOR: "Heterocyclic Synthesis from o-Aminonitriles. A New Synthesis of 5-Substituted Pyrimidines.", JOURNAL OF ORGANIC CHEMISTRY, vol. 32, 1967, pages 2376 - 2378, XP002154126 *
T.M. BARGAR: "A Comparative Molecular Field Analysis Study of Obtusifoliol 14alpha-methyl Demethylase Inhibitors", PESTICIDE SCIENCE, vol. 55, 1999, pages 1059 - 1069, XP002154128 *

Also Published As

Publication number Publication date
DE19917160A1 (de) 2000-10-19
AU4542700A (en) 2000-11-02
WO2000063176A2 (de) 2000-10-26

Similar Documents

Publication Publication Date Title
MXPA04012214A (es) Insecticidas de pirazolcarboxamida.
IL143157A (en) Anilinotriazines and triazinylbenzimidazole derivatives and agricultural/horticultural fungicides containing them
HUT57728A (en) Herbicidal compositions comprising carboxamide derivatives as active ingredient and process for producing the carboxamide derivatives
MX9700132A (es) Uso de 2-((dihidro) pirazolil-3'-oximetilen)-anilidas como agentes de control de plagas y fungicidas.
WO2004046129A3 (en) Novel anthranilamide insecticides
WO2001014376A8 (en) Novel spiro compounds
CA2194502A1 (en) 2-[1',2',4'-triazol-3'-yloxymethylene]anilides, their preparation and their use
RS52225B (en) SYNERGETIC HERBICIDE PROCEDURES AND MIXTURES
MXPA97001953A (en) Employment of ariluracils in the semi-selective and non-selective field of the fight against bad hier
WO2003029243A3 (de) 2-aryloxy-6-pyrazolyl-pyridine
AU8816791A (en) Herbicidal carboxamide derivatives
UA84724C2 (ru) Производные пиримидина, гербицидные смеси и композиции на их основе, способ контроля роста нежелательной растительности
TWI349674B (en) Derivatives of [2-(8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)alkyl]phosphonic acid and methods of use thereof
MX2007000240A (es) Derivados de [1.2]-oxazin-3,5-diona y dihidropirona sustituidos con fenilo.
FR07C0036I2 (fr) Derive de pyrazole, agent pour la lutte contre les parasites le comprenant comme ingredient actif et leur procede de production
WO2005053402A3 (en) The use of n-arylhydrazine derivatives for combating pests in and on animals
WO2002028853A1 (fr) Compose de benzylamine, son procede de production et produit intermediaire correspondant
WO2002048122A3 (en) Benzamidine derivatives
EP1431299A4 (de) IMIDAZO(1,2-a)PYRIMIDINE UND DIESE ENTHALTENDE FUNGIZIDZUSAMMENSETZUNGEN
WO2000063176A3 (de) Disubstituierte Pyridine und Pyrimidine als Herbizide und Fungizide
WO2001053275A3 (de) Substituierte arylketone
WO2002042280A3 (en) Pyrimidine derivatives
JP2001342186A5 (de)
AU2573800A (en) Percutaneous absorption preparations of compound having angiotensin ii receptor antagonism
MXPA04007048A (es) Derivados de amidoacetonitrilo.

Legal Events

Date Code Title Description
AK Designated states

Kind code of ref document: A2

Designated state(s): AE AG AL AM AT AU AZ BA BB BG BR BY CA CH CN CR CU CZ DE DK DM DZ EE ES FI GB GD GE GH GM HR HU ID IL IN IS JP KE KG KP KR KZ LC LK LR LS LT LU LV MA MD MG MK MN MW MX NO NZ PL PT RO RU SD SE SG SI SK SL TJ TM TR TT TZ UA UG US UZ VN YU ZA ZW

AL Designated countries for regional patents

Kind code of ref document: A2

Designated state(s): GH GM KE LS MW SD SL SZ TZ UG ZW AM AZ BY KG KZ MD RU TJ TM AT BE CH CY DE DK ES FI FR GB GR IE IT LU MC NL PT SE BF BJ CF CG CI CM GA GN GW ML MR NE SN TD TG

DFPE Request for preliminary examination filed prior to expiration of 19th month from priority date (pct application filed before 20040101)
121 Ep: the epo has been informed by wipo that ep was designated in this application
REG Reference to national code

Ref country code: DE

Ref legal event code: 8642

122 Ep: pct application non-entry in european phase
NENP Non-entry into the national phase

Ref country code: JP