UY31642A1 - Imidazolidina-2,4.dionas sustituidas con arilo, procesos para su preparación, medicamentos que comprenden estos compuestos y uso de los mismos. - Google Patents
Imidazolidina-2,4.dionas sustituidas con arilo, procesos para su preparación, medicamentos que comprenden estos compuestos y uso de los mismos.Info
- Publication number
- UY31642A1 UY31642A1 UY031642A UY31642A UY31642A1 UY 31642 A1 UY31642 A1 UY 31642A1 UY 031642 A UY031642 A UY 031642A UY 31642 A UY31642 A UY 31642A UY 31642 A1 UY31642 A1 UY 31642A1
- Authority
- UY
- Uruguay
- Prior art keywords
- compounds
- drugs
- imidazolidina
- dionas
- arilo
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/72—Two oxygen atoms, e.g. hydantoin
- C07D233/74—Two oxygen atoms, e.g. hydantoin with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to other ring members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Diabetes (AREA)
- Addiction (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Child & Adolescent Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
La invención se refiere a Imidazolidina-2,4-dionas sustituidas con arilo de la fórmula I en la que cada uno de los radicales R y R´, A, D, E, G, L, p y R1 a R10 es como se ha definido anteriormente, y a sales fisiológicamente compatibles de los mismos. Los compuestos son adecuados, por ejemplo, como fármacos antiobesidad.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP08290130 | 2008-02-07 |
Publications (1)
Publication Number | Publication Date |
---|---|
UY31642A1 true UY31642A1 (es) | 2009-08-31 |
Family
ID=39493923
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY031642A UY31642A1 (es) | 2008-02-07 | 2009-02-06 | Imidazolidina-2,4.dionas sustituidas con arilo, procesos para su preparación, medicamentos que comprenden estos compuestos y uso de los mismos. |
Country Status (8)
Country | Link |
---|---|
US (1) | US20110053947A1 (es) |
EP (1) | EP2252591B1 (es) |
AR (1) | AR070524A1 (es) |
AT (1) | ATE513815T1 (es) |
CL (1) | CL2009000259A1 (es) |
TW (1) | TW200942528A (es) |
UY (1) | UY31642A1 (es) |
WO (1) | WO2009097999A1 (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP3159331A1 (en) | 2010-05-05 | 2017-04-26 | Infinity Pharmaceuticals, Inc. | Tetrazolones as inhibitors of fatty acid synthase |
US20130197043A1 (en) | 2010-08-31 | 2013-08-01 | Snu R&Db Foundation | Use of the fetal reprogramming of a ppar agonist |
US9981928B2 (en) | 2013-06-20 | 2018-05-29 | Bayer Cropscience Aktiengesellschaft | Aryl sulfide derivatives and aryl sulfoxide derivatives as acaricides and insecticides |
CN113024513A (zh) * | 2021-03-22 | 2021-06-25 | 中国药科大学 | 新型雄激素受体降解剂、制备方法和医药用途 |
AU2022414087A1 (en) * | 2021-12-14 | 2024-08-01 | Trustees Of Tufts College | Use of hyperpolarizing agents alone and in combination with other therapeutic agents for treating cancers including glioblastoma |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE19530298C2 (de) * | 1995-08-17 | 1999-07-22 | Woerwag Pharma Gmbh | Verwendung von Orotsäure zur Prävention und Therapie des metabolischen Syndroms |
WO2004101529A1 (ja) * | 2003-05-19 | 2004-11-25 | Ono Pharmaceutical Co., Ltd. | 含窒素複素環化合物およびその医薬用途 |
-
2009
- 2009-01-30 EP EP09707966A patent/EP2252591B1/de active Active
- 2009-01-30 WO PCT/EP2009/000592 patent/WO2009097999A1/de active Application Filing
- 2009-01-30 AT AT09707966T patent/ATE513815T1/de active
- 2009-02-05 CL CL2009000259A patent/CL2009000259A1/es unknown
- 2009-02-05 AR ARP090100401A patent/AR070524A1/es unknown
- 2009-02-05 TW TW098103591A patent/TW200942528A/zh unknown
- 2009-02-06 UY UY031642A patent/UY31642A1/es not_active Application Discontinuation
-
2010
- 2010-08-06 US US12/852,216 patent/US20110053947A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
AR070524A1 (es) | 2010-04-14 |
EP2252591B1 (de) | 2011-06-22 |
EP2252591A1 (de) | 2010-11-24 |
WO2009097999A1 (de) | 2009-08-13 |
CL2009000259A1 (es) | 2009-06-26 |
US20110053947A1 (en) | 2011-03-03 |
ATE513815T1 (de) | 2011-07-15 |
TW200942528A (en) | 2009-10-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20130206 |