UY29587A1 - AMINOQUINOLINE AND AMINOQUINAZOLINE QUINASA MODULATORS - Google Patents

AMINOQUINOLINE AND AMINOQUINAZOLINE QUINASA MODULATORS

Info

Publication number
UY29587A1
UY29587A1 UY29587A UY29587A UY29587A1 UY 29587 A1 UY29587 A1 UY 29587A1 UY 29587 A UY29587 A UY 29587A UY 29587 A UY29587 A UY 29587A UY 29587 A1 UY29587 A1 UY 29587A1
Authority
UY
Uruguay
Prior art keywords
compounds
aminoquinoline
aminoquinazoline
trkb
flt3
Prior art date
Application number
UY29587A
Other languages
Spanish (es)
Inventor
Michael David Gaul
Guozhang Xu
Christian Andrew Baumann
Nand Baindur
Kevin Douglas Kreutter
Alexander J Kim
Bao-Ping Zhao
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Priority to UY29587A priority Critical patent/UY29587A1/en
Publication of UY29587A1 publication Critical patent/UY29587A1/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La invención está dirigida a compuestos aminoquinolina y aminoquinazolina de Fórmula I: en la cual R1, R2, R3, B, Z, Q, p, q y X son tal como se han definido aquí, el uso de dichos compuestos como moduladores de la proteína tirosinquinasa, particularmente inhibidores de FLT3 y/o TrKB, al uso de dichos compuestos para reducir e inhibir la actividad de quinasa de FLT3 y/o TrKB en una célula o un sujeto, y al uso de dichos compuestos para prevenir o tratar en un sujeto, un desorden y/o desórdenes proliferativos de células relacionados con FLT3 y/o TrKB. La presente invención está además dirigida a composiciones farmacéuticas que comprenden los compuestos de la presente invención y a los métodos para tratar los trastornos tales como cánceres y otros desórdenes proliferativos de células.The invention is directed to aminoquinoline and aminoquinazoline compounds of Formula I: in which R1, R2, R3, B, Z, Q, p, q and X are as defined herein, the use of said compounds as protein modulators tyrosine kinase, particularly inhibitors of FLT3 and / or TrKB, to the use of said compounds to reduce and inhibit the kinase activity of FLT3 and / or TrKB in a cell or a subject, and to the use of said compounds to prevent or treat in a subject , a disorder and / or proliferative disorders of cells related to FLT3 and / or TrKB. The present invention is further directed to pharmaceutical compositions comprising the compounds of the present invention and to methods for treating disorders such as cancers and other proliferative cell disorders.

UY29587A 2006-06-08 2006-06-08 AMINOQUINOLINE AND AMINOQUINAZOLINE QUINASA MODULATORS UY29587A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
UY29587A UY29587A1 (en) 2006-06-08 2006-06-08 AMINOQUINOLINE AND AMINOQUINAZOLINE QUINASA MODULATORS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
UY29587A UY29587A1 (en) 2006-06-08 2006-06-08 AMINOQUINOLINE AND AMINOQUINAZOLINE QUINASA MODULATORS

Publications (1)

Publication Number Publication Date
UY29587A1 true UY29587A1 (en) 2006-10-02

Family

ID=38813183

Family Applications (1)

Application Number Title Priority Date Filing Date
UY29587A UY29587A1 (en) 2006-06-08 2006-06-08 AMINOQUINOLINE AND AMINOQUINAZOLINE QUINASA MODULATORS

Country Status (1)

Country Link
UY (1) UY29587A1 (en)

Similar Documents

Publication Publication Date Title
ECSP077998A (en) AMINOQUINOLINE AND AMINOQUINAZOLINE KINASE MODULATORS
NI200700313A (en) AMINOPIRIMIDINS AS MODULATORS OF THE KINASE.
NI200700316A (en) AMINOPIRIMIDINS AS MODULATORS OF THE KINASE
ECSP088573A (en) TRIAZOLOPIRIDAZINAS AS MODULATORS OF THYROSINE KINASE
UY29588A1 (en) KINASE MODULATORS WITH ALQUILQUINOLINA AND ALQUILQUINAZOLINA STRUCTURES
UY29590A1 (en) TIENOPIRIMIDINE AND TIENOPIRIDINE QUINASA MODULATORS
EA201100425A1 (en) PIKOLINAMIDA DERIVATIVES AS KINASE INHIBITORS
EA201100580A1 (en) IMIDAZOPIRIDAZINCARBONITRILE USED AS KINASE INHIBITORS
EA200901144A1 (en) PIM KINASE INHIBITORS AND METHODS OF THEIR APPLICATION
GT200800202A (en) QUINAZOLINS FOR THE INHIBITION OF PDK1
ECSP109953A (en) DERIVATIVES OF PIRIDAZINONA
CR20120510A (en) DERIVATIVES OF PIPERIDIN-4-IL AZETIDINE AS INHIBITORS OF JAK1
NI200800060A (en) BENCIMIDAZOLS REPLACED AS CINASA INHIBITORS.
EA201170288A1 (en) OXABICYCLOPTANES AND OXABICYCLOPTENS
EA201170680A1 (en) ACTIVE AND P70 S6 KINASE INHIBITORS
CL2012003637A1 (en) Compounds derived from substituted quinazoline or triazolopyridine, selective tyrosine kinase inhibitors; medicine; pharmaceutical composition; and its use to treat, prevent or improve retinal / macular edema, age-related macular degeneration and retinal vascular effusion related to ischemia, among others.
EA200702136A1 (en) COMPANIES OF STANNSOPORFIN AND THEIR APPLICATION
GT200600250A (en) KINASE MODULATORS WITH ALQUILQUINOLINA AND ALQUILQUINAZOLINA STRUCTURES CROSSED REFERENCE WITH RELATED APPLICATIONS
ATE548364T1 (en) AMINOPYRAZOLE KINASE INHIBITORS
UY29587A1 (en) AMINOQUINOLINE AND AMINOQUINAZOLINE QUINASA MODULATORS
UY29592A1 (en) AMINOPIRIMIDINS AS KINASE MODULATORS
UA105483C2 (en) Isoquinolinone derivatives, compositions based thereon and use thereof as pi3k inhibitors
CR9238A (en) PIRROLOPIRAZOLES, POWERFUL INHIBITORS OF CINASA