UY28622A1 - QUINOLONA ANTIBACTERIAL AGENTS - Google Patents
QUINOLONA ANTIBACTERIAL AGENTSInfo
- Publication number
- UY28622A1 UY28622A1 UY28622A UY28622A UY28622A1 UY 28622 A1 UY28622 A1 UY 28622A1 UY 28622 A UY28622 A UY 28622A UY 28622 A UY28622 A UY 28622A UY 28622 A1 UY28622 A1 UY 28622A1
- Authority
- UY
- Uruguay
- Prior art keywords
- antibacterial agents
- iii
- formula
- quinolona
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Abstract
Se describen compuestos de fórmula I, II, III, v, V y VI y procedimientos para su preparación. Tambie´n se describen procedimientos para fabricar compuestos biológicamente activos de fórmula I, II, III, IV, V y VI a´sí como composiciones farmacéuticamente aceptables que comprenden compuestos de fórmula I, II, III, IV, V y VI. Los compuestos de fórmula I, II, III, IV, V y VI, como se describen en este documento, pueden usarse en diversas aplicaciones incluyendo su uso como agentes antibacterianos.Compounds of formula I, II, III, v, V and VI and processes for their preparation are described. Methods for manufacturing biologically active compounds of formula I, II, III, IV, V and VI therein are also described as pharmaceutically acceptable compositions comprising compounds of formula I, II, III, IV, V and VI. The compounds of formula I, II, III, IV, V and VI, as described herein, can be used in various applications including their use as antibacterial agents.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US52307103P | 2003-11-18 | 2003-11-18 | |
US60549604P | 2004-08-31 | 2004-08-31 |
Publications (1)
Publication Number | Publication Date |
---|---|
UY28622A1 true UY28622A1 (en) | 2005-06-30 |
Family
ID=34623167
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY28622A UY28622A1 (en) | 2003-11-18 | 2004-11-17 | QUINOLONA ANTIBACTERIAL AGENTS |
Country Status (6)
Country | Link |
---|---|
AR (1) | AR046638A1 (en) |
NL (1) | NL1027545C2 (en) |
PE (1) | PE20050582A1 (en) |
TW (1) | TW200524930A (en) |
UY (1) | UY28622A1 (en) |
WO (1) | WO2005049602A1 (en) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK1666477T3 (en) | 2003-09-10 | 2013-07-29 | Kyorin Seiyaku Kk | 7- (4-TRISUBSTITUTED 3-CYCLOPROPYLAMINOMETHYL-1-PYRROLIDINYL) -QUINOLONCARBOXYLIC ACID DERIVATE |
CA2617557A1 (en) | 2005-08-04 | 2007-02-15 | Sirtris Pharmaceuticals, Inc. | Benzimidazole derivatives as sirtuin modulators |
DE102006005861A1 (en) * | 2006-02-09 | 2007-08-23 | Aicuris Gmbh & Co. Kg | Substituted quinolones III |
EP2097400B1 (en) | 2007-01-05 | 2013-07-03 | Daiichi Sankyo Company, Limited | Fused substituted aminopyrrolidine derivative |
CN101622240B (en) * | 2007-01-05 | 2014-07-23 | 第一三共株式会社 | Fused substituted aminopyrrolidine derivative |
EP2149571A4 (en) | 2007-05-24 | 2010-09-01 | Kyorin Seiyaku Kk | Mutilin derivative having heterocyclic aromatic ring carboxylic acid structure in substituent at 14-position |
DE102007036068A1 (en) * | 2007-08-01 | 2009-02-05 | Wacker Chemie Ag | Process for the preparation of alkylmethoxymethyltrimethylsilanylmethylamines |
CN102112440A (en) | 2008-05-30 | 2011-06-29 | 武田药品工业株式会社 | Heterocyclic compound |
AU2010211672B2 (en) | 2009-02-06 | 2016-08-04 | Nippon Shinyaku Co., Ltd. | Aminopyrazine derivative and medicine |
AR091858A1 (en) | 2012-07-25 | 2015-03-04 | Sova Pharmaceuticals Inc | CISTATIONIN-g-LIASA INHIBITORS (CSE) |
US10435403B2 (en) | 2015-06-09 | 2019-10-08 | Bayer Pharma Aktiengesellschaft | Positive allosteric modulators of muscarinic M2 receptor |
CN109689654A (en) * | 2016-07-11 | 2019-04-26 | 拜耳医药股份有限公司 | 1- pyridyl group-naphthyridines -3- benzamide type and application thereof that 7- replaces |
EP3296298A1 (en) | 2016-09-14 | 2018-03-21 | Bayer Pharma Aktiengesellschaft | 7-substituted 1-aryl-naphthyridin-3-carboxamides and their use |
JOP20190045A1 (en) | 2016-09-14 | 2019-03-14 | Bayer Ag | 7-substituted 1-aryl-naphthyridine-3-carboxylic acid amides and use thereof |
WO2018060073A1 (en) | 2016-09-29 | 2018-04-05 | Bayer Cropscience Aktiengesellschaft | Novel 5-substituted imidazole derivatives |
-
2004
- 2004-11-05 WO PCT/IB2004/003666 patent/WO2005049602A1/en active Application Filing
- 2004-11-16 PE PE2004001119A patent/PE20050582A1/en not_active Application Discontinuation
- 2004-11-17 UY UY28622A patent/UY28622A1/en not_active Application Discontinuation
- 2004-11-17 TW TW093135213A patent/TW200524930A/en unknown
- 2004-11-18 NL NL1027545A patent/NL1027545C2/en not_active IP Right Cessation
- 2004-11-18 AR ARP040104261A patent/AR046638A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
TW200524930A (en) | 2005-08-01 |
NL1027545A1 (en) | 2005-05-23 |
PE20050582A1 (en) | 2005-08-25 |
NL1027545C2 (en) | 2006-01-17 |
WO2005049602A1 (en) | 2005-06-02 |
AR046638A1 (en) | 2005-12-14 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20150525 |