UY27324A1 - NEW NAPSILATE SALTS I - Google Patents
NEW NAPSILATE SALTS IInfo
- Publication number
- UY27324A1 UY27324A1 UY27324A UY27324A UY27324A1 UY 27324 A1 UY27324 A1 UY 27324A1 UY 27324 A UY27324 A UY 27324A UY 27324 A UY27324 A UY 27324A UY 27324 A1 UY27324 A1 UY 27324A1
- Authority
- UY
- Uruguay
- Prior art keywords
- napsilate
- salts
- new
- solvates
- stereoisomers
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/01—Sulfonic acids
- C07C309/28—Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C309/33—Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton of six-membered aromatic rings being part of condensed ring systems
- C07C309/34—Sulfonic acids having sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton of six-membered aromatic rings being part of condensed ring systems formed by two rings
- C07C309/35—Naphthalene sulfonic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/48—Phosphonous acids R—P(OH)2; Thiophosphonous acids including RHP(=O)(OH); Derivatives thereof
- C07F9/4808—Phosphonous acids R—P(OH)2; Thiophosphonous acids including RHP(=O)(OH); Derivatives thereof the acid moiety containing a substituent or structure which is considered as characteristic
- C07F9/4816—Acyclic saturated acids or derivatices which can have further substituents on alkyl
Abstract
Novedosas sales napsilato de fórmula I, o solvatos de las mismas y estereoisómeros de las mismas, así como también un proceso para la preparación de los mismos, composiciones farmacéuticas que contienen la sal de napsilato terapéuticamente activa y el uso de los mencionados compuestos activos en tratamientos.Novel napsilate salts of formula I, or solvates thereof and stereoisomers thereof, as well as a process for the preparation thereof, pharmaceutical compositions containing the therapeutically active napsilate salt and the use of said active compounds in treatments .
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0102057A SE0102057D0 (en) | 2001-06-08 | 2001-06-08 | New Salts I |
Publications (1)
Publication Number | Publication Date |
---|---|
UY27324A1 true UY27324A1 (en) | 2003-02-28 |
Family
ID=20284432
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY27324A UY27324A1 (en) | 2001-06-08 | 2002-06-07 | NEW NAPSILATE SALTS I |
Country Status (3)
Country | Link |
---|---|
SE (1) | SE0102057D0 (en) |
UY (1) | UY27324A1 (en) |
WO (1) | WO2002100869A1 (en) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2006050472A2 (en) * | 2004-11-03 | 2006-05-11 | Xenoport, Inc. | Acyloxyalkyl carbamate prodrugs of 3-aminopropylphosphonous and -phosphinic acids |
WO2006050471A2 (en) | 2004-11-03 | 2006-05-11 | Xenoport, Inc. | Acyloxyalkyl carbamate prodrugs of sulfinic acids, methods of synthesis, and use |
US20060160777A1 (en) * | 2004-12-27 | 2006-07-20 | Anders Lehmann | New use of GABAbeta receptor agonists |
WO2006071186A1 (en) * | 2004-12-27 | 2006-07-06 | Astrazeneca Ab | Use of gabab receptor agonists |
WO2008033572A1 (en) | 2006-09-15 | 2008-03-20 | Xenoport, Inc. | Acyloxyalkyl carbamate prodrugs, methods of synthesis and use |
CN101743011A (en) * | 2007-07-25 | 2010-06-16 | 阿斯利康(瑞典)有限公司 | The use of (3-amino-2-fluoropropyl) phosphinic acid for treatment of nerd |
PE20091176A1 (en) * | 2007-12-21 | 2009-09-03 | Astrazeneca Ab | NEW CRYSTALLINE C FORM OF (2R) - (3-AMINO-2-FLUOROPROPYL) PHOSPHINIC ACID |
PE20091311A1 (en) * | 2007-12-21 | 2009-09-30 | Astrazeneca Ab | NEW PROCESS TO PREPARE FORM A OF (2R) - (3-AMINO-2-FLUOROPROPYL) PHOSPHINIC ACID |
WO2009082345A1 (en) * | 2007-12-21 | 2009-07-02 | Astrazeneca Ab | Novel crystalline form b of (2r)-(3-amino-2-fluoropropyl)phosphinic acid |
WO2012009646A1 (en) | 2010-07-15 | 2012-01-19 | Xenoport, Inc. | Methods of treating fragile x syndrome, down's syndrome, autism and related disorders |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE9603408D0 (en) * | 1996-09-18 | 1996-09-18 | Astra Ab | Medical use |
-
2001
- 2001-06-08 SE SE0102057A patent/SE0102057D0/en unknown
-
2002
- 2002-06-04 WO PCT/SE2002/001083 patent/WO2002100869A1/en not_active Application Discontinuation
- 2002-06-07 UY UY27324A patent/UY27324A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
WO2002100869A1 (en) | 2002-12-19 |
SE0102057D0 (en) | 2001-06-08 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
DESI | Application deemed to be withdrawn |
Effective date: 20111129 |