PE20091176A1 - NEW CRYSTALLINE C FORM OF (2R) - (3-AMINO-2-FLUOROPROPYL) PHOSPHINIC ACID - Google Patents
NEW CRYSTALLINE C FORM OF (2R) - (3-AMINO-2-FLUOROPROPYL) PHOSPHINIC ACIDInfo
- Publication number
- PE20091176A1 PE20091176A1 PE2008002132A PE2008002132A PE20091176A1 PE 20091176 A1 PE20091176 A1 PE 20091176A1 PE 2008002132 A PE2008002132 A PE 2008002132A PE 2008002132 A PE2008002132 A PE 2008002132A PE 20091176 A1 PE20091176 A1 PE 20091176A1
- Authority
- PE
- Peru
- Prior art keywords
- fluoropropyl
- amino
- phosphinic acid
- new crystalline
- crystalline
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/14—Antitussive agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/30—Phosphinic acids R2P(=O)(OH); Thiophosphinic acids, i.e. R2P(=X)(XH) (X = S, Se)
- C07F9/301—Acyclic saturated acids which can have further substituents on alkyl
Abstract
SE REFIERE A UN COMPUESTO EN FORMA CRISTALINA C DE ACIDO (2R)-(3-AMINO-2-FLUOROPROPIL)FOSFINICO CARACTERIZADO POR UN PATRON DE RAYOS X EN POLVO QUE REPRESENTA SUSTANCIALMENTE d: 5,8 ANGSTROM. REFERIDA ADEMAS A UNA FORMULACION SIENDO UTIL EN EL TRATAMIENTO DEL ASMA RELACIONADO CON EL REFLUJO, ENFERMEDADES PULMONARES, SINDROME DE DECLIVE, TRASTORNOS GASTROINTESTINAL FUNCIONAL, ENTRE OTROSREFERS TO A COMPOUND IN CRYSTALLINE C FORM OF (2R) - (3-AMINO-2-FLUOROPROPYL) PHOSPHINIC ACID CHARACTERIZED BY A POWDERED X-RAY PATTERN THAT SUBSTANTIALLY REPRESENTS d: 5.8 ANGSTROM. ALSO REFERRED TO A FORMULATION BEING USEFUL IN THE TREATMENT OF ASTHMA RELATED TO REFLUX, PULMONARY DISEASES, DECLINE SYNDROME, FUNCTIONAL GASTROINTESTINAL DISORDERS, AMONG OTHERS
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US1583307P | 2007-12-21 | 2007-12-21 |
Publications (1)
Publication Number | Publication Date |
---|---|
PE20091176A1 true PE20091176A1 (en) | 2009-09-03 |
Family
ID=40801459
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PE2008002132A PE20091176A1 (en) | 2007-12-21 | 2008-12-18 | NEW CRYSTALLINE C FORM OF (2R) - (3-AMINO-2-FLUOROPROPYL) PHOSPHINIC ACID |
Country Status (5)
Country | Link |
---|---|
AR (1) | AR070046A1 (en) |
PE (1) | PE20091176A1 (en) |
TW (1) | TW200940560A (en) |
UY (1) | UY31555A1 (en) |
WO (1) | WO2009082348A1 (en) |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE9904508D0 (en) * | 1999-12-09 | 1999-12-09 | Astra Ab | New compounds |
SE0102057D0 (en) * | 2001-06-08 | 2001-06-08 | Astrazeneca Ab | New Salts I |
WO2009014490A1 (en) * | 2007-07-25 | 2009-01-29 | Astrazeneca Ab | Combination of (3-amino-2-fluoropropyl)phosphinic acid and omeprazole for treating tlesr, gerd, and nerd |
-
2008
- 2008-12-18 WO PCT/SE2008/051505 patent/WO2009082348A1/en active Application Filing
- 2008-12-18 PE PE2008002132A patent/PE20091176A1/en not_active Application Discontinuation
- 2008-12-19 UY UY31555A patent/UY31555A1/en unknown
- 2008-12-19 TW TW097149952A patent/TW200940560A/en unknown
- 2008-12-19 AR ARP080105599A patent/AR070046A1/en unknown
Also Published As
Publication number | Publication date |
---|---|
UY31555A1 (en) | 2009-08-03 |
AR070046A1 (en) | 2010-03-10 |
TW200940560A (en) | 2009-10-01 |
WO2009082348A1 (en) | 2009-07-02 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD | Application declared void or lapsed |