UY26964A1 - DERIVATIVES OF ERYTHROMYCIN 6-0-REPLACED WITH GREATER GASTROINTESTINAL TOLERANCE - Google Patents

DERIVATIVES OF ERYTHROMYCIN 6-0-REPLACED WITH GREATER GASTROINTESTINAL TOLERANCE

Info

Publication number
UY26964A1
UY26964A1 UY26964A UY26964A UY26964A1 UY 26964 A1 UY26964 A1 UY 26964A1 UY 26964 A UY26964 A UY 26964A UY 26964 A UY26964 A UY 26964A UY 26964 A1 UY26964 A1 UY 26964A1
Authority
UY
Uruguay
Prior art keywords
erythromycin
derivatives
replaced
gastrointestinal tolerance
greater gastrointestinal
Prior art date
Application number
UY26964A
Other languages
Spanish (es)
Inventor
Zhenkun Ma
Souming Zhang
Ly Tam Phan
Stevan Djuric
Rick F Clark
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of UY26964A1 publication Critical patent/UY26964A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

Compuestos de fórmula I son útiles para el tratamiento de infeciones bacterianas pero sin producir el efecto colateral de intolerancia gastrointestinal. También se revelan composiciones que contienen los compuestos y métodos de tratamiento que los utilizan.Compounds of formula I are useful for the treatment of bacterial infections but without producing the side effect of gastrointestinal intolerance. Compositions containing the compounds and methods of treatment that use them are also disclosed.

UY26964A 2000-10-16 2001-10-12 DERIVATIVES OF ERYTHROMYCIN 6-0-REPLACED WITH GREATER GASTROINTESTINAL TOLERANCE UY26964A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24077700P 2000-10-16 2000-10-16

Publications (1)

Publication Number Publication Date
UY26964A1 true UY26964A1 (en) 2002-06-20

Family

ID=22907903

Family Applications (1)

Application Number Title Priority Date Filing Date
UY26964A UY26964A1 (en) 2000-10-16 2001-10-12 DERIVATIVES OF ERYTHROMYCIN 6-0-REPLACED WITH GREATER GASTROINTESTINAL TOLERANCE

Country Status (9)

Country Link
EP (1) EP1328534A2 (en)
JP (1) JP2004529857A (en)
AU (1) AU2002213267A1 (en)
BR (1) BR0109946A (en)
CA (1) CA2420012A1 (en)
MX (1) MXPA03003311A (en)
PE (1) PE20020522A1 (en)
UY (1) UY26964A1 (en)
WO (1) WO2002032919A2 (en)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR0214748A (en) 2001-12-05 2004-11-23 Ortho Mcneil Pharm Inc Erythromycin 6-oacyl ketolide derivatives useful as antibacterials
JP2005529143A (en) * 2002-04-30 2005-09-29 アボット・ラボラトリーズ Antibacterial compounds with improved pharmacokinetic profiles
US6727229B2 (en) * 2002-08-19 2004-04-27 Enanta Pharmaceuticals, Inc. 11,12-substituted lactone ketolide derivatives having antibacterial activity
WO2004078771A1 (en) * 2003-03-07 2004-09-16 Taisho Pharmaceutical Co., Ltd. 2-fluoro-6-o-substituted ketolide derivative
JP2007223900A (en) * 2004-02-03 2007-09-06 Taisho Pharmaceut Co Ltd 6-o-substituted ketolide derivative
JP2007254285A (en) * 2004-03-16 2007-10-04 Taisho Pharmaceut Co Ltd 2-fluoro-6-o-substituted ketolide derivative
JP5015016B2 (en) 2006-02-07 2012-08-29 大正製薬株式会社 10a-azalide compounds
US8293715B2 (en) 2007-08-06 2012-10-23 Taisho Pharmaceutical Co., Ltd. 10a-Azalide compound crosslinked at 10a- and 12-positions
WO2009139181A1 (en) 2008-05-15 2009-11-19 大正製薬株式会社 10a-azalide compound having 4-membered ring structure
CN102234302B (en) * 2010-05-07 2014-05-07 北京理工大学 Novel ketolide derivatives, and preparation method and medicinal compositions thereof
AR085286A1 (en) 2011-02-21 2013-09-18 Taisho Pharmaceutical Co Ltd MACROLIDO DERIVATIVE REPLACED IN POSITION C-4
AR102810A1 (en) 2014-08-18 2017-03-29 Taisho Pharmaceutical Co Ltd MACROLID DERIVATIVE REPLACED IN POSITION C-4

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6054435A (en) * 1999-03-19 2000-04-25 Abbott Laboratories 6-O-substituted macrolides having antibacterial activity

Also Published As

Publication number Publication date
CA2420012A1 (en) 2002-04-25
JP2004529857A (en) 2004-09-30
MXPA03003311A (en) 2003-09-10
WO2002032919A3 (en) 2002-09-19
PE20020522A1 (en) 2002-06-25
AU2002213267A1 (en) 2002-04-29
WO2002032919A2 (en) 2002-04-25
BR0109946A (en) 2005-08-02
EP1328534A2 (en) 2003-07-23

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20150126