UA91350C2 - Производные 3-фенилпиразола как модуляторы 5-нт2а серотонинового рецептора, полезные для лечения расстройств, связанных с этим рецептором - Google Patents
Производные 3-фенилпиразола как модуляторы 5-нт2а серотонинового рецептора, полезные для лечения расстройств, связанных с этим рецептором Download PDFInfo
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- UA91350C2 UA91350C2 UAA200706860A UAA200706860A UA91350C2 UA 91350 C2 UA91350 C2 UA 91350C2 UA A200706860 A UAA200706860 A UA A200706860A UA A200706860 A UAA200706860 A UA A200706860A UA 91350 C2 UA91350 C2 UA 91350C2
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- Prior art keywords
- methyl
- phenyl
- pyrazol
- compound
- ylethoxy
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- 238000011282 treatment Methods 0.000 title claims abstract description 94
- OEDUIFSDODUDRK-UHFFFAOYSA-N 5-phenyl-1h-pyrazole Chemical class N1N=CC=C1C1=CC=CC=C1 OEDUIFSDODUDRK-UHFFFAOYSA-N 0.000 title abstract description 15
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Abstract
Данное изобретение касается некоторых 3-фенилпиразольных производных формулы (Иа) и их фармацевтических композиций, которые модулируют активность 5-НТсеротонинового рецептора.Соединения и их фармацевтические композиции направлены на лечение агрегации тромбоцитов, заболевания коронарных артерий, инфаркта миокарда, приступа транзиентной ишемии, стенокардии, удара, мигающей аритмии предсердия, для снижения риска образования сгустков крови, астмы или ее симптомов, тревожного возбуждения или его симптома, поведенческих расстройств, лекарственного психоза, психоза возбуждаемости, синдрома Туретта,
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
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US62977404P | 2004-11-19 | 2004-11-19 |
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UA91350C2 true UA91350C2 (ru) | 2010-07-26 |
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UAA200706860A UA91350C2 (ru) | 2004-11-19 | 2005-11-17 | Производные 3-фенилпиразола как модуляторы 5-нт2а серотонинового рецептора, полезные для лечения расстройств, связанных с этим рецептором |
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UA (1) | UA91350C2 (ru) |
ZA (1) | ZA200703885B (ru) |
Cited By (1)
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CN115554290A (zh) * | 2021-07-01 | 2023-01-03 | 中国科学院分子细胞科学卓越创新中心 | 五羟色胺或其受体激动剂在治疗ilc2细胞介导的免疫性疾病中的应用 |
-
2005
- 2005-11-17 UA UAA200706860A patent/UA91350C2/ru unknown
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2007
- 2007-05-14 ZA ZA200703885A patent/ZA200703885B/xx unknown
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
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CN115554290A (zh) * | 2021-07-01 | 2023-01-03 | 中国科学院分子细胞科学卓越创新中心 | 五羟色胺或其受体激动剂在治疗ilc2细胞介导的免疫性疾病中的应用 |
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ZA200703885B (en) | 2009-11-25 |
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