UA109736C2 - Поліморфна форма мезилатної солі 2-(2,4,5-заміщеного аніліно)піримідину (варіанти) - Google Patents

Поліморфна форма мезилатної солі 2-(2,4,5-заміщеного аніліно)піримідину (варіанти)

Info

Publication number
UA109736C2
UA109736C2 UAA201403622A UAA201403622A UA109736C2 UA 109736 C2 UA109736 C2 UA 109736C2 UA A201403622 A UAA201403622 A UA A201403622A UA A201403622 A UAA201403622 A UA A201403622A UA 109736 C2 UA109736 C2 UA 109736C2
Authority
UA
Ukraine
Prior art keywords
compounds
salts
mutant
pyrimidine
substituted anilino
Prior art date
Application number
UAA201403622A
Other languages
English (en)
Ukrainian (uk)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of UA109736C2 publication Critical patent/UA109736C2/ru

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/10Spiro-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
UAA201403622A 2011-07-27 2012-07-25 Поліморфна форма мезилатної солі 2-(2,4,5-заміщеного аніліно)піримідину (варіанти) UA109736C2 (uk)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201161512061P 2011-07-27 2011-07-27

Publications (1)

Publication Number Publication Date
UA109736C2 true UA109736C2 (uk) 2015-09-25

Family

ID=53675818

Family Applications (3)

Application Number Title Priority Date Filing Date
UAA201403622A UA109736C2 (uk) 2011-07-27 2012-07-25 Поліморфна форма мезилатної солі 2-(2,4,5-заміщеного аніліно)піримідину (варіанти)
UAA201403623A UA108954C2 (xx) 2011-07-27 2012-07-25 Сполуки 2-(2,4,5-заміщеного аніліно)піримідину
UAA201312949A UA106710C2 (uk) 2011-07-27 2012-07-25 Сполука 2-(2,4,5-заміщеного аніліно)піримідину та її застосування для лікування раку

Family Applications After (2)

Application Number Title Priority Date Filing Date
UAA201403623A UA108954C2 (xx) 2011-07-27 2012-07-25 Сполуки 2-(2,4,5-заміщеного аніліно)піримідину
UAA201312949A UA106710C2 (uk) 2011-07-27 2012-07-25 Сполука 2-(2,4,5-заміщеного аніліно)піримідину та її застосування для лікування раку

Country Status (2)

Country Link
AR (1) AR115019A2 (ru)
UA (3) UA109736C2 (ru)

Also Published As

Publication number Publication date
UA106710C2 (uk) 2014-09-25
AR115019A2 (es) 2020-11-18
UA108954C2 (xx) 2015-06-25

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