TW347388B - Oxazolidinone derivatives having adhesion receptor antagonism - Google Patents
Oxazolidinone derivatives having adhesion receptor antagonismInfo
- Publication number
- TW347388B TW347388B TW084111533A TW84111533A TW347388B TW 347388 B TW347388 B TW 347388B TW 084111533 A TW084111533 A TW 084111533A TW 84111533 A TW84111533 A TW 84111533A TW 347388 B TW347388 B TW 347388B
- Authority
- TW
- Taiwan
- Prior art keywords
- receptor antagonism
- adhesion receptor
- oxazolidinone derivatives
- group
- known amino
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
- C07D263/24—Oxygen atoms attached in position 2 with hydrocarbon radicals, substituted by oxygen atoms, attached to other ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
An oxazolidinone derivative of the formula I (I) in which R1 is (group); R2 is H, A, Ac, A-SO2-, Ar-SO2- or a known amino protective group; R3 is H or A, A being a C1-C6-alkyl; D is H2N-C(=NH)- where the primary group also can provide a known amino protective group; Ac is C1-C10-alkanoyl or C7-C11-aroyl; Ar is phenyl which is unsubstituted or mono-substituted by A, or benzyl; and physiologically unobjectionable salts thereof.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE4439110 | 1994-11-02 | ||
DE19509093A DE19509093A1 (en) | 1994-11-02 | 1995-03-16 | Adhesion receptor antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
TW347388B true TW347388B (en) | 1998-12-11 |
Family
ID=6532300
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TW084111533A TW347388B (en) | 1994-11-02 | 1995-11-01 | Oxazolidinone derivatives having adhesion receptor antagonism |
Country Status (7)
Country | Link |
---|---|
KR (1) | KR100379996B1 (en) |
AR (1) | AR005224A1 (en) |
CO (1) | CO4520228A1 (en) |
DE (2) | DE19509093A1 (en) |
TW (1) | TW347388B (en) |
UA (1) | UA54367C2 (en) |
ZA (1) | ZA959212B (en) |
-
1995
- 1995-03-16 DE DE19509093A patent/DE19509093A1/en not_active Withdrawn
- 1995-10-19 DE DE59503324T patent/DE59503324D1/en not_active Expired - Lifetime
- 1995-10-31 ZA ZA959212A patent/ZA959212B/en unknown
- 1995-11-01 TW TW084111533A patent/TW347388B/en active
- 1995-11-01 UA UA95114762A patent/UA54367C2/en unknown
- 1995-11-01 AR ARP950100002A patent/AR005224A1/en unknown
- 1995-11-02 CO CO95051975A patent/CO4520228A1/en unknown
- 1995-11-02 KR KR1019950039300A patent/KR100379996B1/en not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
UA54367C2 (en) | 2003-03-17 |
DE19509093A1 (en) | 1996-05-09 |
KR100379996B1 (en) | 2003-07-22 |
ZA959212B (en) | 1996-07-24 |
DE59503324D1 (en) | 1998-10-01 |
KR960017662A (en) | 1996-06-17 |
CO4520228A1 (en) | 1997-10-15 |
AR005224A1 (en) | 1999-04-28 |
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