TW202416984A - 化合物i或其鹽的固體形式 - Google Patents

化合物i或其鹽的固體形式 Download PDF

Info

Publication number
TW202416984A
TW202416984A TW112130830A TW112130830A TW202416984A TW 202416984 A TW202416984 A TW 202416984A TW 112130830 A TW112130830 A TW 112130830A TW 112130830 A TW112130830 A TW 112130830A TW 202416984 A TW202416984 A TW 202416984A
Authority
TW
Taiwan
Prior art keywords
compound
salts
solid forms
trifluoromethyl
5methyl
Prior art date
Application number
TW112130830A
Other languages
English (en)
Inventor
李海軍
陳明明
康迪
黨超杰
李阿敏
王燕萍
龍偉
Original Assignee
大陸商北京加科思新藥研發有限公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 大陸商北京加科思新藥研發有限公司 filed Critical 大陸商北京加科思新藥研發有限公司
Publication of TW202416984A publication Critical patent/TW202416984A/zh

Links

Abstract

本發明涉及一種化合物I的新形式、其製備方法、或其鹽的固體形式,以及包含該化合物I的新形式的藥物組合物,其中,所述化合物爲(S)-5-((1-(3-(5-甲基-3-(三氟甲基)-8,9-二氫吡啶并[3',2':4,5]吡咯并[1,2-a]吡𠯤-7(6H)-基)-3-氧代丙氧基)丙-2-基)胺基)-4-(三氟甲基)嗒𠯤-3(2H)-酮。
TW112130830A 2022-08-17 2023-08-16 化合物i或其鹽的固體形式 TW202416984A (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
WOPCT/CN2022/112917 2022-08-17

Publications (1)

Publication Number Publication Date
TW202416984A true TW202416984A (zh) 2024-05-01

Family

ID=

Similar Documents

Publication Publication Date Title
CN101671336B (zh) 芳杂环并嘧啶衍生物和类似物及其制备方法和用途
NZ593033A (en) 4,5,7,8-tetrahydro-(optionally 4-oxo, 4-thioxo or 4-imino)-2H-imidazo[1,2-a]pyrrolo[3,4-e]pyrimidine and 4,5,7,8,9-pentahydro-(optionally 4-oxo, 4-thioxo or 4-imino)-2H-pyrimido[1,2-a]pyrrolo[3,4-e]pyrimidine derivatives as PDE1 Inhibitors
NO20054085L (no) Substituerte heksahydropyrazino [1,2-a]pyrimidin-4,7-dionderivater, fremgangsmater for fremstilling og anvendelse derav som medikamenter
GR3031500T3 (en) NOVEL 9-HYDROXY-PYRIDO [1,2-a]PYRIMIDIN-4-ONE ETHER DERIVATIVES
WO2003000695A8 (en) Pyrrolopyrimidines as protein kinase inhibitors
IL115185A0 (en) Pyrimido (5,4-d) pyrimidines pharmaceutical compositions containing them their use and processes for their preparation
GEP20063784B (en) Optical Resolution of (1-Benzyl-4- Methylpiperidin-3-Yl) -Methylamine Enantiomers and Use Thereof for Preparation of Pyrrolo 2,3-Pyrimidine Derivatives as Protein Kinases Inhibitors
MA29437B1 (fr) Compose d'imidazopyridazine
MXPA05001581A (es) Algunas imidazopiridinas novedosas y su uso.
HRP20070534T3 (en) Phosphoric acid salt of a dipeptidyl peptidase-iv inhibitor
MX2010001677A (es) Derivados de 4-(9-(3,3-difluorociclopentil)-5,7,7-trimetil-6-oxo-6 ,7,8,9-tetrahidro-5h-pirimido[4,5-b][1,4]diazepin-2-ilamino)-3-me toxibenzamida como inhibidores de las proteinas cinasas humanas plk1 a plk4 para el tratamiento de enfermedades proli
IL147280A0 (en) Quinazoline derivatives
MX2007004250A (es) Derivados de imidazo[1,5-a]triazolo[1,5-d]benzodiazepina para el tratamiento de trastornos cognitivos.
CA2517774A1 (en) Substituted 8-perfluoroalkyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one derivatives
CA2071273A1 (en) Tetrahydropyrrolo[1,2-a]pyrazine-4-spiro-3'-pyrrolidine derivatives, processes for the preparation thereof and pharmaceutical compositions containing the same
AU1428801A (en) Novel (1,2,3)-triazolo(4,5-D)pyrimidine compounds
DE69030616D1 (de) Pharmazeutische Zusammensetzungen zur Hemmung der Maillardreaktion
TW202416984A (zh) 化合物i或其鹽的固體形式
WO2007080324A3 (fr) Derives de pyrido-pyrimidone, leur preparation, leur application en therapeutique.
KR930019676A (ko) 약제 화합물
AU7425801A (en) Guanidine derivatives of quinazoline and quinoline for use in the treatment of autoimmune diseases
AU5539899A (en) Novel triazolo(4,5-(d))pyrimidine compounds
WO2006010568A3 (de) Substituierte pyrido [3',2':4,5]thieno[3,2-d]pyrimidin-2,4(1 h,3h)-diones und -4(3h)-one sowie pyrido [3',2' :4,5] furo[3,2-d]pyrimidin -2,4(1 h,3h)-dione und -4(3h)-one zur verwendung als inhibitoren der tnf-allpha freisetzung
CN103554111A (zh) 芳杂环并嘧啶衍生物和类似物及其制备方法和用途
DE69512419T2 (de) IMIDAZO[1,2-a]INDENO[1,2-e]PYRAZIN-2-CARBONSÄURE DERIVATE, IHRE HERSTELLUNG UND SIE ENTHALTENDE ARZNEIMITTEL