TW202333773A - Glp-1受體和gip受體雙重激動劑的醫藥組成物及其用途 - Google Patents
Glp-1受體和gip受體雙重激動劑的醫藥組成物及其用途 Download PDFInfo
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- TW202333773A TW202333773A TW111143259A TW111143259A TW202333773A TW 202333773 A TW202333773 A TW 202333773A TW 111143259 A TW111143259 A TW 111143259A TW 111143259 A TW111143259 A TW 111143259A TW 202333773 A TW202333773 A TW 202333773A
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- pharmaceutically acceptable
- sodium
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- A61P3/06—Antihyperlipidemics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Endocrinology (AREA)
- Molecular Biology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Biochemistry (AREA)
- Gastroenterology & Hepatology (AREA)
- Zoology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biophysics (AREA)
- Emergency Medicine (AREA)
- Toxicology (AREA)
- Child & Adolescent Psychology (AREA)
- Genetics & Genomics (AREA)
- Inorganic Chemistry (AREA)
- Immunology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN202111341752 | 2021-11-12 | ||
| CN202111341752.0 | 2021-11-12 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW202333773A true TW202333773A (zh) | 2023-09-01 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW111143259A TW202333773A (zh) | 2021-11-12 | 2022-11-11 | Glp-1受體和gip受體雙重激動劑的醫藥組成物及其用途 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20250115654A1 (https=) |
| EP (1) | EP4431522A4 (https=) |
| JP (1) | JP2024546026A (https=) |
| KR (1) | KR20240109258A (https=) |
| CN (1) | CN118103391A (https=) |
| AU (1) | AU2022386489A1 (https=) |
| CA (1) | CA3237796A1 (https=) |
| MX (1) | MX2024005663A (https=) |
| TW (1) | TW202333773A (https=) |
| WO (1) | WO2023083301A1 (https=) |
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| CN116693652B (zh) * | 2023-08-02 | 2024-01-05 | 北京惠之衡生物科技有限公司 | 一种glp-1/gip受体双重激动剂衍生物及其制备方法和应用 |
| TW202529797A (zh) * | 2023-12-12 | 2025-08-01 | 大陸商江蘇恆瑞醫藥股份有限公司 | Ｇｌｐ－１類似物治療代謝疾病的方法及醫藥用途 |
| WO2025149039A1 (zh) * | 2024-01-12 | 2025-07-17 | 杭州中美华东制药有限公司 | 长效glp-1/gip双激动剂的药物组合物 |
| WO2025252197A1 (zh) * | 2024-06-07 | 2025-12-11 | 江苏恒瑞医药股份有限公司 | 药物组合物 |
| WO2026037397A1 (zh) * | 2024-08-16 | 2026-02-19 | 江苏恒瑞医药股份有限公司 | Glp-1类似物的医药用途 |
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| CN101987868B (zh) * | 2009-07-30 | 2013-09-04 | 江苏豪森医药集团有限公司 | Glp-1类似物的衍生物或其可药用盐和用途 |
| WO2012088379A2 (en) * | 2010-12-22 | 2012-06-28 | Marcadia Biotech, Inc. | Methods for treating metabolic disorders and obesity with gip and glp-1 receptor-active glucagon-based peptides |
| US9453062B2 (en) * | 2011-06-10 | 2016-09-27 | Beijing Hanmi Pharmaceutical Co., Ltd. | Glucose dependent insulinotropic polypeptide analogs, pharmaceutical compositions and use thereof |
| IN2014MN02304A (https=) * | 2012-05-03 | 2015-08-07 | Zealand Pharma As | |
| AU2013366692B2 (en) * | 2012-12-21 | 2017-11-23 | Sanofi | Dual GLP1/GIP or trigonal GLP1/GIP/Glucagon agonists |
| EP3642238A1 (en) * | 2017-06-21 | 2020-04-29 | Amgen Inc. | Method of treating or ameliorating metabolic disorders using antagonistic binding proteins for gastric inhibitory peptide receptor (gipr)/glp-1 receptor agonist fusion proteins |
| SG11202103137WA (en) * | 2018-10-26 | 2021-04-29 | Novo Nordisk As | Stable semaglutide compositions and uses thereof |
| CN112351994B (zh) * | 2019-04-11 | 2024-06-07 | 江苏豪森药业集团有限公司 | 一种多受体激动剂及其医药用途 |
| US20220372072A1 (en) * | 2019-09-19 | 2022-11-24 | Dr. Reddy's Laboratories Limited | Improved purification processes for liraglutide |
| EP4086277A4 (en) * | 2019-12-30 | 2024-02-14 | Gan & Lee Pharmaceuticals Co., Ltd. | Long-acting glp-1 compound |
| CN114222755B (zh) * | 2020-05-29 | 2024-06-11 | 北京拓界生物医药科技有限公司 | Glp-1和gip受体双重激动剂化合物及其应用 |
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2022
- 2022-11-11 US US18/709,004 patent/US20250115654A1/en active Pending
- 2022-11-11 EP EP22892094.8A patent/EP4431522A4/en active Pending
- 2022-11-11 TW TW111143259A patent/TW202333773A/zh unknown
- 2022-11-11 AU AU2022386489A patent/AU2022386489A1/en active Pending
- 2022-11-11 MX MX2024005663A patent/MX2024005663A/es unknown
- 2022-11-11 CN CN202280069025.XA patent/CN118103391A/zh active Pending
- 2022-11-11 JP JP2024527503A patent/JP2024546026A/ja active Pending
- 2022-11-11 KR KR1020247018683A patent/KR20240109258A/ko active Pending
- 2022-11-11 CA CA3237796A patent/CA3237796A1/en active Pending
- 2022-11-11 WO PCT/CN2022/131375 patent/WO2023083301A1/zh not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| MX2024005663A (es) | 2024-05-28 |
| JP2024546026A (ja) | 2024-12-17 |
| EP4431522A1 (en) | 2024-09-18 |
| EP4431522A4 (en) | 2025-03-26 |
| KR20240109258A (ko) | 2024-07-10 |
| AU2022386489A1 (en) | 2024-05-23 |
| CA3237796A1 (en) | 2023-05-19 |
| US20250115654A1 (en) | 2025-04-10 |
| WO2023083301A1 (zh) | 2023-05-19 |
| CN118103391A (zh) | 2024-05-28 |
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