TW202308631A - 用於治療mpnst之化合物和組成物 - Google Patents
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- Chemical & Material Sciences (AREA)
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- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202163184422P | 2021-05-05 | 2021-05-05 | |
| US63/184,422 | 2021-05-05 |
Publications (1)
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|---|---|
| TW202308631A true TW202308631A (zh) | 2023-03-01 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| TW111116420A TW202308631A (zh) | 2021-05-05 | 2022-04-29 | 用於治療mpnst之化合物和組成物 |
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| US (1) | US20240238284A1 (https=) |
| EP (1) | EP4333847A1 (https=) |
| JP (1) | JP2024517788A (https=) |
| CN (1) | CN117177752A (https=) |
| TW (1) | TW202308631A (https=) |
| WO (1) | WO2022234409A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2025510572A (ja) | 2022-03-08 | 2025-04-15 | レボリューション メディシンズ インコーポレイテッド | 免疫不応性肺癌を治療するための方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SI1761528T1 (sl) | 2004-06-11 | 2008-06-30 | Japan Tobacco Inc | 5-amino-2,4,7-triokso-3,4,7,8-tetrahidro-2H-pirido(2,3-D)pirimidinski derivati in sorodne spojine za zdravljenje raka |
| ES2522346T3 (es) | 2008-08-22 | 2014-11-14 | Novartis Ag | Compuestos de pirrolopirimidina como inhibidores de CDK |
| JO3517B1 (ar) | 2014-01-17 | 2020-07-05 | Novartis Ag | ان-ازاسبيرو الكان حلقي كبديل مركبات اريل-ان مغايرة وتركيبات لتثبيط نشاط shp2 |
| EP4302834A3 (en) | 2016-07-12 | 2024-07-17 | Revolution Medicines, Inc. | 2,5-disubstituted 3-methyl pyrazines and 2,5,6-trisubstituted 3-methyl pyrazines as allosteric shp2 inhibitors |
| EP3923941B1 (en) * | 2019-02-12 | 2025-12-03 | Novartis AG | Pharmaceutical combination comprising tno155 and ribociclib |
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2022
- 2022-04-28 CN CN202280029051.XA patent/CN117177752A/zh active Pending
- 2022-04-28 WO PCT/IB2022/053970 patent/WO2022234409A1/en not_active Ceased
- 2022-04-28 US US18/558,756 patent/US20240238284A1/en active Pending
- 2022-04-28 EP EP22722574.5A patent/EP4333847A1/en active Pending
- 2022-04-28 JP JP2023567063A patent/JP2024517788A/ja active Pending
- 2022-04-29 TW TW111116420A patent/TW202308631A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2022234409A1 (en) | 2022-11-10 |
| CN117177752A (zh) | 2023-12-05 |
| US20240238284A1 (en) | 2024-07-18 |
| JP2024517788A (ja) | 2024-04-23 |
| EP4333847A1 (en) | 2024-03-13 |
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