TW201713342A - 以吡嗪羧醯胺化合物為有效成分之醫藥組成物 - Google Patents

以吡嗪羧醯胺化合物為有效成分之醫藥組成物 Download PDF

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Publication number
TW201713342A
TW201713342A TW105113124A TW105113124A TW201713342A TW 201713342 A TW201713342 A TW 201713342A TW 105113124 A TW105113124 A TW 105113124A TW 105113124 A TW105113124 A TW 105113124A TW 201713342 A TW201713342 A TW 201713342A
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TW
Taiwan
Prior art keywords
bmx
cancer
compound
pharmaceutical composition
pharmaceutically acceptable
Prior art date
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TW105113124A
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English (en)
Chinese (zh)
Inventor
Satoshi Konagai
Hiroko Yamamoto
Hideki Sakagami
Original Assignee
Astellas Pharma Inc
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Publication date
Application filed by Astellas Pharma Inc filed Critical Astellas Pharma Inc
Publication of TW201713342A publication Critical patent/TW201713342A/zh

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
TW105113124A 2015-04-28 2016-04-27 以吡嗪羧醯胺化合物為有效成分之醫藥組成物 TW201713342A (zh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2015092301A JP2018104290A (ja) 2015-04-28 2015-04-28 ピラジンカルボキサミド化合物を有効成分とする医薬組成物

Publications (1)

Publication Number Publication Date
TW201713342A true TW201713342A (zh) 2017-04-16

Family

ID=57198305

Family Applications (1)

Application Number Title Priority Date Filing Date
TW105113124A TW201713342A (zh) 2015-04-28 2016-04-27 以吡嗪羧醯胺化合物為有效成分之醫藥組成物

Country Status (3)

Country Link
JP (1) JP2018104290A (ja)
TW (1) TW201713342A (ja)
WO (1) WO2016175252A1 (ja)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2019014653A (ja) * 2015-11-27 2019-01-31 アステラス製薬株式会社 がん免疫を介したがん治療方法
US20190282569A1 (en) 2016-10-26 2019-09-19 Astellas Pharma Inc. Stable pharmaceutical composition
TW202340177A (zh) 2021-12-30 2023-10-16 美商拜歐米富士恩股份有限公司 作為 flt3抑制劑之吡嗪化合物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX360970B (es) * 2008-06-27 2018-11-23 Avila Therapeutics Inc Compuestos de heteroarilo y usos de los mismos.
AR089727A1 (es) * 2012-01-17 2014-09-10 Astellas Pharma Inc Compuesto de pirazin-carboxamida
ES2618007T3 (es) * 2012-08-06 2017-06-20 Acea Biosciences, Inc. Nuevos compuestos de pirrolopirimidina como inhibidores de proteína cinasas

Also Published As

Publication number Publication date
WO2016175252A1 (ja) 2016-11-03
JP2018104290A (ja) 2018-07-05

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