TW200901876A - Thioimidate compound and use thereof for controlling pests - Google Patents

Abstract

The present invention provides a thioimidate compound having an excellent control efficacy against pests, which is represented by the formula (I): wherein R represents a C6-12 bicycloalkyl group or a C1-3 alkyl group substituted with a C6-12 bicycloalkyl group; m represents an integer of 0 to 2; n represents an integer of 0 to 2; X represents a halogen atom, a C1-3 alkyl group, a C1-3 haloalkyl group, a C1-4 alkoxy group, or a nitro group, and two X's are the same or different when m is 2; and Z represents a halogen atom, a C1-3 alkyl group, a C1-3 haloalkyl group, or a C1-4 alkoxy group, and two Z's are the same or different when n is 2.

Description

200901876 VI. Description of the Invention: TECHNICAL FIELD OF THE INVENTION The present invention relates to thioimidate compounds and their use for controlling pests. [Prior Art] A variety of compounds have been studied and actually used for the purpose of controlling pests (specifically disclosed in The Pesticide Manual (by British Crop Protection Council, 13th edition)). The thioimidate compound is disclosed in the patent document JP 9-202766. SUMMARY OF THE INVENTION The object of the present invention is to provide a compound having excellent control effects against pests. The present inventors have conducted intensive studies and found that a thioimidate compound represented by the following formula (I) has an excellent therapeutic effect against pests, and thus completed the present invention. That is, the present invention provides: (1) A thioimidate compound represented by the formula (I):

Wherein R represents a C6-12 bicycloalkyl group or an anthracene-3 alkyl group substituted by a C6-12 bicycloalkyl group; m represents an integer representing 0 to 2; η represents an integer of 0 to 2; and X represents a halogen atom. Cl-3 alkyl, Cl-3 halo, Cl-4 alkoxy or nitro, and when m is 2, two X are the same or different; and Z represents 4 320202 200901876 N, a Ci- 3 炫, Ci-3 halogen or Ci_4 alkoxy, and when n is 2, the two oximes are the same or the same (hereinafter referred to as the compound (丨)); (2) according to the above (1; And a thioimidate compound, wherein R in the formula (I) represents a C6-12 bicycloalkyl group; (3) a thioimidate compound according to the above (1), wherein R in the formula (I) represents a bicyclo[4.4.0] fluorenyl group; (4) A pest control preparation comprising the compound of any one of the above (1) to (3) as an active ingredient; The use of any of the above compounds (1) to (3) for the control of pest i (6), the use of any of the above compounds (1) to (3), for the manufacture of a pest control preparation; Any of the compounds of (1) to (3); and the like. (ΌA method for controlling pests, comprising applying the compound (I) to a pest or a pest habitat to have an excellent control effect against pests. [Embodiment] (Best aspect of the invention) Hereinafter, the present invention will be described. Specific examples of the substituent are used. Preferred examples of the C6-, 2-bicycloalkyl group include a Ce bicycloalkyl group such as a bicyclo[3.1.0]-2-hexyl group represented by the following formula:

丨"屄,双环,双环 [2.2. l]-l- 320202 200901876 % heptyl, bicyclo [2· 2. l]-2-heptyl and bicyclo [2. 2·丨卜厂庚基: 0>Χ> ^ C8 bicycloalkyl group such as the bicyclo ring of the following formula [4· 2. 〇]_3_octyl, bicyclo[3. 3. 0]-2-octyl and bicyclo[3. 3. 〇]-3-octyl Base: bo xo * , G bicycloalkyl group such as the bicyclo ring of the following formula [4. 3. 〇]_2_ fluorenyl, bicyclo [4. 3. 0]-3-fluorenyl, bicyclo [4. 3. 〇]- 7-fluorenyl and bicyclo [4· & 〇]_8-octyl: . ό〇Χχ> oi ay . w and Cm bicycloalkyl such as the bicyclo [4·4. 0]_2-fluorenyl and bicyclic ring of the following formula [4. 4. 0]-3-癸 base: : '

Preferred is a Cm bicycloalkyl group. / Cu alkyl" includes methyl, ethyl, propyl or isopropyl. Preferred examples of the Ci_3 alkyl group substituted with a CV!2 bicycloalkyl group include (bicyclo[2.2.1]-1-heptyl)methyl, (bicyclo[2·2heptyl)methyl, (bicyclo[ 2. 2. 1 ]-7-heptyl)fluorenyl, (bicyclo[4. 4. 〇]_2_fluorenyl)methyl, (dual 320202 200901876 ring [4. 4. 0]-3-indenyl) Indenyl, 1-(bicyclo[4.4.0]-2-indenyl)ethyl and 2-(bicyclo[4.4.0]-3-indenyl)ethyl. "Halogen atoms" include fluorine, chlorine, bromine or moth atoms. Preferred examples of the G-3 haloalkyl group include a linear or branched alkyl group substituted with at least one halogen atom, such as fluoromethyl, difluoroindenyl, trifluoromethyl, chloromethyl, bromomethyl, iodo Base, pentafluoroethyl, 2, 2, 2-trifluoroethyl and 2, 2, 2-trifluoro-1-(trifluoromethyl)ethyl. C!-4 alkoxy is methoxy, ethoxy, propoxy, isopropoxy, butoxy, isobutoxy, second butoxy or tert-butoxy. Preferred examples of the phenyl group substituted by (X)m include 4-fluorophenyl group, 4-chlorophenyl group, 4-bromophenyl group, 4-methylphenyl group, 4-trifluorodecylphenyl group, 4- Nonyloxyphenyl, 4-nitrophenyl, 3-fluorophenyl, 3-chlorophenyl, 3-bromophenyl, 3-methylphenyl, 3-trifluoromethylphenyl, 3-indole Oxyphenyl, 3-nitrophenyl, 2-oxylphenyl, 2-chlorophenyl, 2-formylphenyl, 2-methylphenyl, 2-triemethylphenyl, 2-methyl Oxyphenyl, 2-nitrophenyl, 3,4-difluorophenyl, 3,4-dichlorophenyl, 3,4-didecylphenyl, 3,5-difluorophenyl, 3 , 5-dichlorophenyl, 3, 5-dimethylphenyl, 2-fluoro-4-methylphenyl, 3-fluoro-4-indolylphenyl, 2-ox-4-mercaptophenyl , 3-chloro-4-mercaptophenyl, 4-fluoro-2-indolylphenyl, 2-chloro-4-trifluorodecylphenyl, 3-chloro-4-trimethylnonylphenyl, 2 - 4-methoxyphenyl, 3-1 fluorodi 4-indolyloxyphenyl and 4-chloro-3-indolylphenyl. Preferred examples of the phenyl group substituted by (Z)n include 4-fluorophenyl group, 4-chlorophenyl group, 4-bromophenyl group, 4-methylphenyl group, 4-trifluorodecylphenyl group, 4- Nonyloxyphenyl, 4-(t-butoxy)benzene, yl, 3-fluorophenyl, 3-chlorophenyl, 3-bromo 7 320202 200901876 Phenyl, 3-methylphenyl, 3-tri Fluorylphenyl, 3-methoxyphenyl, 2-fluorobenyl, 2-chlorophenyl, 2-bromophenyl, 2-nonylphenyl, 2-trifluorodecylphenyl, 2- Nonyloxyphenyl, 3,4-difluorophenyl, 3,4-diphenyl, 3,4-dimethylphenyl, 3, 5-difluorophenyl, 3, 5-dichlorobenzene , 3, 5-dimercapto, 2-fluoro-4-methylphenyl, 3-fluoro-4-methylphenyl, 2-chloro-4-methylphenyl, 3-chloro-4 -methylphenyl, 4-fluoro-2-indolylphenyl, 4-oxa-2-indolylphenyl, 2-ox-4-trifluoromethylphenyl, 3-chloro-4-tetrafluoromethyl Phenylphenyl, 2-fluoro-4-methoxyphenyl, 3-fluoro-4-nonyloxyphenyl, and 4-chloro-3-indolylphenyl. Specific examples of the compound (I) include the following: in the thioimidate compound of the formula (I), r is a Ce_12 bicycloalkyl group; and in the thioimidate compound of the formula (I), r is a C7_10 bicycloalkane. In the thioimidate compound of formula (I), R is bicyclo[3. 1.〇]hexyl, bicyclo[4.1.0]heptyl, bicyclo[3. 2·0]heptyl, bicyclo [2. 2. 1]Heptyl, bicyclo[3.3.0]octyl, bicyclo[4.2.0]octyl, bicyclo[4.3.0]indolyl or bicyclo[4.4.0]癸Wherein R is bicyclo[3. 1. 〇]-2-hexyl, bicyclo[4.1. 〇]-2-heptyl, bicyclo[4.1.0]-3 in the thioiminoacetate compound of formula (I) -heptyl, bicyclo[3.2.〇]-3-heptyl, bicyclo[2.2.1]-1-heptyl, bicyclo[2.2.1]-2-heptyl, bicyclo[2.2.1]-7-g , bicyclo[4. 2. 0]-3-octyl, bicyclo 3·0]-2-octyl, bicyclo[3·3.0]-3-octyl, bicyclo[4. 3. 0]- 2-indenyl, bicyclo[4. 3. 0]-3-indenyl, bicyclo[4. 3. 0]-7-indenyl, bicyclo[4. 3. 0]-8-indenyl, bicyclo[4 4. 0]-2-indenyl or bicyclo [4. 4. 0]-3_ fluorenyl; 320202 200901876 wherein R is a bicyclo [4.4.0] fluorenyl group in the thioimidate compound of formula (I); And the following thio An imidate compound: bicyclo[4·4.0]-3-indolyl 3-(3,5-dichlorophenylthio)-N-(.phenyl)thioimidate; 'double % [4. 4. 0]- 3-mercapto 3_(4- phenylphenylthio)(.phenyl)thio propylene imidate ( thioacrylimidate); bicyclo[4. 4. 0]-3 - mercapto 3-(4-methylphenylthio)-N-(phenyl) thiopropanthene imidate; bicyclo[4. 4. 0]-3-indolyl 3-(4- (Phenoxyphenylthio)(phenyl)thiopropenyl imidate; Bicyclo[4.4.0]-3-indolyl 3-(3-chlorophenylthio)-N-(benzene Thiopropyl imidic acid S; Bicyclo[4.4.0]-3-indolyl 3-(3-mercaptophenylthio)-N-(phenyl)thiopropene Amino acid ester; bicyclo[4.4.0]-3-indolyl 3-(3-fluorophenylthio)-n-(phenyl)thiopropenyl imidate; bicyclo[4.4. 0] 3-mercapto 3-(4-nitrophenylthio(phenyl)thiopropenyl imidate; bicyclo[4·4·0]-3-indenyl N-phenyl-3- 3-trifluoromethylphenylthio)thiopropenyl imidate; bicyclo[4·4.0]-3-indolyl N-phenyl-3-(4-trifluoromethylphenylsulfide Thiopropenyl imidate; bicyclo [4.4. 0]-3- 3-(4-fluorophenylthio)_1(4- mercaptophenyl) thiopropenyl imidate; 320202 9 200901876 Bicyclo[4. 4. 0]-3-indolyl 3-(4 -fluorophenylthio)-N-(phenyl)thiopropenyl imidate; and bicyclo[4.4.0]-3-indolyl 1^-(4-chlorophenyl)-3-(4 -|11 phenylthio)thiopropenyl imidate. The method of producing the compound (I) will be described later. Compound (I) is a compound represented by formula (II):

H-C three C-U

Among them, R, Z and η are produced by reacting with a compound represented by the formula (III) as defined above (hereinafter referred to as a compound (II)):

Among them, X and m are as defined above (hereinafter referred to as compound (I)). 2至1. 2等。 The equivalent of 0. 8 to 1. 2 equivalents. This reaction can be carried out in the presence of a base in a reaction system containing the compound (II) and the compound (III). Examples include metal alkoxides such as sodium ethoxide, sodium methoxide and potassium t-butoxide; nitrogen-containing compounds such as triethylamine, diisopropylethylamine, pyridine, 4-didecylaminopyridine And N,N-dimercaptoaniline; carbonates such as potassium carbonate, sodium carbonate, sodium hydrogencarbonate and potassium cesium carbonate; hydroxides such as sodium hydroxide and hydroxide; metal hydrides such as lithium hydride, hydrogenation Sodium and potassium hydride; and organolithium, such as butyl lithium and diiso 10 320202 200901876 propylamine chain. As long as there is no adverse effect on the reaction, the amount used is not particularly limited. The reaction can be carried out in a suitable solvent. Examples of the solvent include aliphatic hydrocarbons such as pentane, hexane, heptane and petroleum ether; aromatic hydrocarbons such as benzene, toluene and dinonylbenzene; and esters such as methyl acetate, ethyl acetate and citric acid. Ethyl ester and ethyl propionate; ketones such as acetone and methyl ethyl ketone; ethers such as diethyl mystery, dipropyl Ni, diisopropyl mystery, dibutyl bond _, tetrazole and two a decane; a nitrile such as acetonitrile and propionitrile; a guanamine such as dimethyl decylamine and dimethyl acetamide; an anthracene such as a dimethyl sulfoxide; an anthracene such as cyclobutyl hydrazine; Amidoxime, such as hexamethylenephosphonamide; i-hydrocarbons such as dichlorosilane, chloroform, 1,2-dichloroethane, and tetra-carbonated carbon; and aromatic amines, such as σ , methyl ° ratio σ, diterpene ratio σ 喧 and 喧 。. These solvents may be used singly or in combination or as a mixed solvent with water. Usually, the reaction temperature is from -50 to 150 ° C, preferably from -20 to 120 ° C, and more preferably from -10 to 60 ° C. The reaction time is usually from 0.1 to 96 hours, and preferably from 0.1 to 24 hours. After completion of the reaction, the compound (I) can be isolated by a conventional operation step, for example, concentrating the reaction mixture; or the reaction mixture can be poured into water, extracted with an organic solvent, and the extract can be concentrated. The obtained compound (I) can be purified by a conventional method such as distillation, re-sinking, recrystallization or chromatography. Hereinafter, a method for producing the starting compound used for the production of the compound (I) will be explained. Compound (11) is produced from a compound of formula (IV) by a conventional method (for example, the method disclosed in Synthes i s 11 320202 200901876 1989) (1), plOO, 1999 and Chem. Lett., P1261:

Among them, R, Z and η are as defined above (hereinafter referred to as compound (Iv)). Compound (111) is a conventional compound or can be produced by a conventional method. Compound (IV) is usually a compound of formula (v) in the presence of a base:

MesSi-C^CH (V) (hereinafter referred to as compound (V)) reacts with a compound of formula (VI) VZ)n

S=〇=iN

(VI) wherein Z and η are as defined above (hereinafter referred to as compound (vi)), and then the reaction product is reacted with a compound of the formula (VII) to prepare: RL (VII) wherein R is as The above-defined "and L" represent a leaving group (hereinafter referred to as a compound (VII)). Examples of the leaving group represented by L in the formula (VII) include a _ atom and a formula: a group represented by L2S〇3, wherein L2 represents a halogenated Cl_3, such as a fluorenyl or a trifluoromethyl group. Or a phenyl group which may be substituted by a Cm alkyl group; a reaction between the compound (V) and the compound (VI). An excess of the person (VI) may be used, but based on the compound (v), preferably yttrium. Examples of the base used in the reaction include alkali metal alkoxides such as sodium ethoxide, 320202 12 200901876 sodium decanoate and potassium t-butoxide; nitrogen-containing compounds such as triethylamine, diiso) Propyl ethylamine, pyridine, 4-dimethylaminopyridine and hydrazine, hydrazine-dimethylaniline; carbonates such as potassium carbonate, sodium carbonate, sodium cesium carbonate and hydrogencarbonate; hydroxides such as hydrogen Oxidation of sodium and potassium hydride; metal hydrides such as lithium hydride, sodium hydride and potassium hydride; and organolithium such as butyl lithium and lithium diisopropylamide. 5至1.2当量。 The compound (V) is preferably used from 0.8 to 1.2 equivalents. The reaction can be carried out in a suitable solvent. Examples of the solvent include aliphatic hydrocarbons such as pentane, hexane, heptane and petroleum ether; aromatic hydrocarbons such as benzene, toluene and xylene; and esters such as methyl acetate, ethyl acetate and hydrazine. Ethyl ethyl ester and ethyl propionate; ketones such as acetone and methyl ethyl ketone; ethers such as diethyl bond, dipropyl bond, diisopropyl mystery, dibutyl bond, tetrazine π pentane and Dioxane; nitriles such as acetonitrile and propionitrile; guanamines such as dimethylformamide and dimercaptoacetamide; sulfoxides such as dimercaptopurine; terpenoids such as cyclobutane Phosphonamides such as hexamethylphosphonium; functional hydrocarbons such as dichlorosilane, chloroform, 1,2-dichloroethane and carbon tetrachloride; and aromatic amines such as pyridine; Mercaptopyridine, lutidine and quinoline. These solvents may be used singly or in combination or as a mixed solvent with water. Usually, the reaction temperature is from -100 to 100 ° C, and preferably from -80 to 80 ° C. 1至24小时。 The reaction time is usually from 0.1 to 96 hours, preferably from 0.1 to 72 hours, and more preferably from 0.1 to 24 hours. The amount of the compound (VII) is preferably from 0.8 to 5 equivalents, based on the compound (V). The reaction can be carried out in a suitable solvent. The same solvent as shown in the reaction of the compound (V) and the compound (VI) of 13 320202 200901876 can be used. Generally, the degree of reactivity is from -5 Torr to 2 〇 〇 C, preferably from 150 〇C, and more preferably from -10 to 12 Torr. (: The reaction time is usually from 2 Torr to 96 hours, preferably from 0.1 to 72 hours, and more preferably from 〇'1 to hr. .1 to 24, after completion of the reaction, the compound (IV) can be used The conventional operation steps are single, such as concentrating the reaction mixture; or pouring the mixture into water to extract it with a solvent, and concentrating the extract. The compound (5) obtained by the machine can be purified by a conventional method, such as a crane, Re-sinking, recrystallization or chromatography. Alternatively, the reaction mixture itself can be used as a starting material for the subsequent reaction. Compound (10) is produced by a conventional method disclosed in Chem, pi26: (4) geometric isomers and substances - (4) and their mixed compounds (1) have excellent control effects on pests, such as health pests, animal parasitism, such as health Plant parasitic pests, the right ones are used to control these pests. Compounds, animals, plants, and plants, which are excellent in their control, are used as pest control systems. use Also suitable steps or even of veterinary medicine / suspension formulation to be applied through conventional insecticide, form. In other words, compound (1) is dissolved or dispersed in a suitable liquid carrier, mixed with a suitable solid carrier or adsorbed onto a suitable solid carrier prior to application, in the form of a formulation, such as an emulsion, , liquid preparation, microemulsion, flowable preparation, oily preparation, wettable powder, powder, granule, fine granule, seed coating preparation, aerosol preparation, key agent, microcapsule, aerosol, aerosol propellant, carbon dioxide Formula, heat transpiration preparation such as mosquito coil, electric mosquito and electric mosquito liquid repellent, aerosol preparation, Ew preparation, ointment, capsule, granule, injectable solution, resin formulation and The lotion may be added to the formulation such as an emulsifier, a suspending agent, a spreader, a penetrating agent, a wetting agent, a thickening agent and/or a stabilizer, and the composition can be produced according to a conventional method. Examples of the liquid carrier used in the above formulation include water, alcohols (e.g., methanol, ethanol, n-propanol, isopropanol, benzyl alcohol, and ethylene glycol), ketones (for example, acetone methyl ethyl ketone, methyl group). Isobutyl ketone and cyclohexanone), ethers (eg tetrahydro π pentane, ethylene glycol monomethyl ether, diethylene glycol monodecyl ether, diethyl, alcohol monoethyl ether and propylene glycol monomethyl Ether), aliphatic hydrocarbons (such as coal =, paraffin oil, fuel oil and motor oil), aromatic hydrocarbons (such as toluene, diterpenoids, solvent petroleum brain and methyl naphthalene), body hydrocarbons (such as two Methyl chloride, chloroform and carbon tetrachloride), amines (eg hydrazine, hydrazine-dimercaptocarboxamide, hydrazine, hydrazine :: methyl acetamide, hydrazine-methylpyrrolidone and _ _ octyl Pyrrolidone), esters (eg, ethyl acetate, butyl acetate, fatty acid glycerides, and r-butyrolactone), nitriles (eg, acetonitrile and propionitrile), carbonates (eg, propylene carbonate), and Vegetable oils (eg rapeseed oil, cottonseed oil, corn oil, safflower oil and orange oil). The liquid carriers may be used in combination with one or more (preferably one to 320202 15 200901876) in an appropriate ratio. Examples of solid carriers (diluents or extenders) used in the above formulations include vegetable powders (e.g., soy flour, tobacco powder, flour and wood flour), mineral powders (e.g., clays such as kaolin, bentonite, and acid white clay). , talc such as talc powder and pyrophyllite (pyr〇 phyllite), Shi Xishi such as chopped algae and mica), alumina, sulfur powder, activated carbon, calcium carbonate, potassium chloride, ammonium sulfate, stone acid hydrogen Sodium, lactose and urea. These solid carriers may be used by mixing one or more (preferably one to three) in an appropriate ratio. Examples of the gaseous carrier used in the above formulation include fluorocarbon, butane gas, LPG (liquefied petroleum gas), dimethyl ether and carbon dioxide. These gaseous carriers may be used in combination with one or two in appropriate proportions or in combination with a suitable liquid carrier. Examples of the ointment base used in the above preparation include polyethylene glycol, pectin, a polyol ester of a long-chain fatty acid such as glyceryl monostearate, a cellulose derivative such as decyl cellulose, sodium alginate, Bentonite, higher alcohols, polyols such as glycerin, petrolatum, white petrolatum, liquid paraffin, lard, various vegetable oils, lanolin, dehydrated lanolin, hardened oil and resin. These soft pastes; = 11] bases can be used in combination with one or more (preferably one to three), using, or _ adding a surfactant as described later. Examples of surfactants used as emulsifiers, spreaders, penetrants or dispersants in the above formulations include nonionic and anionic surfactants such as soaps, polyoxyethylidene aryl bonds (eg DA) I -1CHI N〇igen and EA142. (trade name) manufactured by K0GY0SEIYAKU; Τ0Η0 Nonnal (trade name) manufactured by CHEMICAL INDUSTRY, alkyl sulphide 16 320202 200901876 acid salt (such as Emal 10 manufactured by KAO CORPORATION) Anonymous) and Emal 40 (trade name), alkylbenzene sulfonate (for example, Neogen (trade name) and Neogen T (trade name) manufactured by DAI-ICHI K0GY0 SEIYAKU Co., Ltd.; Neoprex (trade name) manufactured by KAO CORPORATION )), polyoxyethylene ethyl ether (for example, the brand name of Noigen ET-135C manufactured by DAI-ICHI K0GY0 SEIYAKU Co., Ltd.), polyoxyethylene ethyl oxy-propyl block polymer (for example, SANYO CHEMICAL INDUSTRIES) Manufactured NEWP0LPE-64C trade name)), polyol ester (such as Tween 20 (trade name) and Tween 80 (trade name) manufactured by KAO CORPORATION), alkyl sulfosuccinate ( For example, SANM0RIN 0T 20 (trade name) manufactured by SANYO CHEMICAL INDUSTRIES; Newkalgen EX70 (trade name) manufactured by TAKEMOTO OIL & FAT, and alkenyl sulfonate (for example, Sorpol 5115 (trade name) manufactured by CHEMICAL0Η0 CHEMICAL INDUSTRY) ). These surfactants may be used by mixing one or more (preferably one to three) in an appropriate ratio. Compound (I) can also be mixed with other insecticide active ingredients, such as insecticides (eg pyrethroid insecticides, organophosphate insecticides, urethane insecticides, new final tests) (neoJQic〇tin〇id) insecticides and natural insecticides), acaricides, motor oils, nematicides, herbicides, phytohormones, plant growth regulators, fungicides (eg copper fungicides, organic Chlorine fungicides, organic sulfur fungicides and phenol fungicides, synergists, attractants, repellents, safeners, pigments, fertilizers, animal feeds (eg for Feeds for raising animals such as cattle, pigs and chickens, such as dogs and miscellaneous 320202 17 200901876 What kind of animal feed, and for captive fish such as gold grab fish (yell〇wta (1) and sea bream (sea bream) Feeds for animals), pharmaceutical supplements for animals (1) for the treatment and prevention of animals, pet animals and fish, and for nutritional supplements for animals. The content of the compound (1) of the phlegm of the tree is based on the total amount of the pest control preparation of the present invention, and is usually 〇. ι纟8〇% by weight, ::' is 1 to 2. wt%. Specifically When the compound (1) is used as the emulsification from the liquid agent or the wettable powder (for example, the water-dispersible granule), it is from 1 to 8% by weight, preferably from ～5% by weight. It is used as an oil or In the case of a powder preparation, it is usually used in an amount of 1.1.5% by weight, preferably 〇1 to 2% by weight.

In the case of granulated lions, the content is usually from 1 to 5 g% by weight, preferably from 1 to 20% by weight. I: and other active ingredients (for example, insecticides, herbicides, chlorpyrifos) It may be mixed with the pest control preparation of the present invention, and is usually used in an amount of from 0.1 to 80% by weight, preferably from 1 to 20% by weight, based on the total amount of the preparation of the present invention. The content of the additive is usually from 〇. to 99.9% by weight of 1%, preferably from j to gq of the active ingredient _ and # depending on the insecticide', more specifically in the case of the herbicide of the present invention The amount is usually (10)% by weight of the agent =, the content of the active agent is from ! to 20% by weight · ^ ^ to 15 parts by weight (iv); the flow aid is a two-component preparation such as an emulsion or wettable 320202 18 200901876 For example, water-dispersible granules, when used, are suitable to be diluted with water (100 to 5000 times). The substance (I) can be used as a pest control preparation for farmland such as dry grassland or orchard and uncultivated land. ) can control pests in the farmland of the crops listed below without causing crop damage "Crops" π agricultural crops: corn, rice, wheat, barley, rye, oats, tall wood, cotton, soybeans, peanuts, buckwheat, sugar beets, rapeseed, geranium, sugar cane and tobacco; (s〇lanaceous) vegetables (eg eggplant, tomato, green pepper, pepper and potato), cucurbitaceous vegetables (eg moon melon pumpkin, watermelon and melon), cruciferous (brassicace〇us) vegetables (eg radish) , turnip, western horseradish, kohlrabi, celery cabbage, kale, leaf fennel, broccoli and broccoli, asteraceous vegetables (eg burdock, garland chrysanthemum, radix and lettuce) , Liliaceae (1111 & (:6〇1^) vegetables (such as shallots, onions, garlic and bamboo shoots), umbelliferous vegetables (such as carrots, coriander, order vegetables and wind, grass (Parsnip )), chenopodi aceous vegetables (such as fried vegetables and chard), labiate vegetables (such as scallions, mint and basil) 'strawberry, sweet potato' yam yam and芋(ar〇id); flowers and decorative plants; foliage plants; fruit: pomaceous fruits (eg apples, pears, Japanese 320202 19 200901876 pears, Chinese quince and quince), stone fruit Stone fruit (eg peach, plum, nectarine, sauer apricot, yellow peach, apricot and medlar * orange fruit (such as Satsuma orange, ritual, gracious, lime and grapefruit) ), nuts (such as walnuts, walnuts, agrelite (called 1), almonds, pistachios, cashews and Hawaiian beans), berries (such as blue mother, cranberry, blackberry and raspberry), grapes , persimmon, olive, medlar, fragrant*, coffee, datepaim and coconut fruit. Trees other than fruit trees: tea, raspberry, flowering trees, road trees (eg white wax =, birch, hawthorn, eucalyptus, ginkgo, lilac, maple, oak, celcis, iiqUidambar, Platanus, zelkova, arborvitae, fir, heml〇ck fir, juniper tree, pine, spruce and yew. The above crops include herbicides by traditional breeding methods or genetic recombination techniques. Resistant, such herbicides include HPPD inhibitors such as isoxaflutole, ALS inhibitors such as imazethapyr and thifensulfuron-methyl, and Epsp synthetase inhibitors , bran acid synthase inhibitor, acetoin coenzyme A. carboxylase inhibitor and bromoxynil. Examples of crops that are resistant by traditional breeding methods include Clearfield®, canola, which fights against The imidazol-based herbicide of grass smoke; and STS soybean, which is resistant to sulfenilamide Als inhibitor-type herbicide such as thifensulfuron-methyl. Similarly, it provides anti-drug by the method of cultivation Examples of crops include SR corn, which is resistant to triterpene oxime and aryloxybenzene 320202 20 200901876 oxypropionic acid herbicide, acetoin coenzyme A carboxylase inhibitor, etc. Provided with acetamyl coenzyme A carboxylate Examples of enzyme inhibitor resistant crops are disclosed in The Proceeding of The National Academy of Sciences of The United States of America (Proc. Natl. Acad. Sci. USA), Vol. 87, p7175-7179, 1990. Mutation Acetyl-CoA carboxylase, which is resistant to acetaminophen coenzyme A carboxylase inhibitors, has been reported in the literature Weed

Science, Vol. 53, p728-746, 2005. Inhibition of acetaminophen coenzyme A

A resistant crop is produced by introducing a mutated acetaminophen coenzyme A carboxylase gene into a crop by genetic recombination techniques, or by introducing a ruthenium coenzyme A carboxylase associated with a mutation providing resistance into a crop. And manufacturing. V As a crop to which resistance is conferred by genetic recombination technology, there are exemplified by glyphosate and glufosinate H^liti. These have been marketed under the trade names of RoundupReady® and LibertyLink®. The above crops include those which are capable of selectively synthesizing certain types of toxins by genetic recombination techniques, known as Bacillus. Examples of insecticidal toxins which are manifested by genetically recombinant plants, including derived from waxy Bacillus cereus and Bacillus popilliae; for example, (5-endotoxin insecticidal protein, such as CrylAb, CrylAc derived from BacΠ1 us «. thuringiensis, CrylF, CrylFa2, Cry2Ab, Cry3A, Cry3Bbl and Cry9C, VIP1, VIP2, VIP3 and VIP3A; insecticidal proteins derived from nematodes; animal-derived toxins such as saxitoxin, spider toxin, brown beetle toxin and insect-specific neurotoxin 21 320202 200901876 Toxins of true & planet lectine; lectins. protease inhibitors such as trypsin inhibitors, A serine protease inhibitor, a potato storage protein (patatin), a cysteine protease inhibitor, and a papain inhibitor; rib〇some inactivation proteins (RIP) such as lysine, corn up, ' I tj, abrin, saporin, and single-stranded nuclear inactivated protein (bryodin); steroid metabolic enzymes such as 3-light steroid oxidase, ecdysteroid-UDP-sugar Base conversion enzyme and cholesterol oxidase; ecdysone inhibitor; HMG-CoA reductase; ion channel inhibitor such as sodium ion channel inhibitor and ion channel inhibitor; juvenile hormone esterase Diuretic hormone receptor; stilbene synthase; bibenzyl synthase; chitinase; and glucanase. Toxins expressed in recombinant crops of these genes 'including hybrid toxins of insecticidal proteins For example, 5-endotoxin, such as CrylAb,

CrylAc, CrylF, CrylFa2, Cry2Ab, Cry3A, Cry3Bbl and

Cry9C, VIP1, VIP2, VIP3 and VIP3A, partially defective toxins and modified toxins. Fusion toxins are formed by a new combination of different domains of such proteins by means of genetic recombination techniques. A typical example of a partially defective toxin is CrylAb, in which part of the amino acid sequence is deleted. The modified toxin can be exemplified by a natural toxin in which a single or a plurality of amino acids are substituted. Examples of toxins and recombinant plants capable of synthesizing toxins are disclosed, for example, in the patent documents EP-A-0374753, WO93/07278, W095/34656, EP-A-0427529, EP-A-451878 and W003/052073. . . . - 22 320202 200901876 Toxins contained in these genetically recombinant plants, in particular to provide resistance against pests of the order Coleoptera, diptera and Lepidoptera (butterfly and moth) Sex. It is known that genetically recombinant plants contain single or multiple insecticidal pest resistance genes and produce single or multiple toxins. Some of these are commercially available. Examples of genetically modified plants include YieldGard® (a corn variety that represents CrylAb toxin), YieldGard Rootworm® (a corn variety that represents Cry3Bbl toxin), YieldGard Plus® (a corn variety that exhibits CrylAb and Cry3Bbl toxin), Herculex I® ( It belongs to the cotton variety that expresses CrylAc toxin), Bollgard II® (belongs to the performance of glufosinate phosphinotricine N-acetyltransferase (PAT) to provide anti-CrylFa2 toxin and glufosinate resistance to corn Variety), NC0TN33B® (a cotton variety that exhibits CrylAc Qinsu), B〇ugard I® (a cotton variety that represents CrylAc toxin), Bol lgard® (a cotton variety that exhibits CrylAb and Cry2Ab toxins), VIPC0T® (belongs to performance) Cotton varieties with VIP toxins), NewLeaf® (belonging to the C. cerevisiae cultivar Cry3A toxin), NatureGard® Agrisure® GT Advantage (Glyphosate resistance trait), Agrisure® GB Advantage (BtllCorn Borer (CB)) Traits) and pr〇tecta®. Such crops include those which are capable of producing an anti-pathogenic substance (having a selective activity) by genetic recombination techniques. Anti-pathogenic substances are listed by microorganisms, such as RP proteins (PRPs, disclosed in patent document EP-A-0392225); ion channel inhibitors such as sodium ion channel inhibitors and calcium channel inhibitors (known to be diseased) 320202 23 200901876 KPl, KP4 and KP6 toxins produced by venom); purine synthase; conjugated synthase; shell multi-enzyme; glucanase; and peptide antibiotics, antibiotics with heterocycles and anti-plant disease resistance A protein factor of sex (referred to as a plant disease resistance gene' and disclosed in patent document W003/000906). Such anti-pathogenic substances and genetically modified plant lines for the production thereof are disclosed in the patent documents EP-A-0392225, W095/33818 and EP-A-0353191. The fungicides, phytohormone agents, plant growth regulators, herbicides, insecticides, acaricides and nematicides which can be formulated together with the compound (I) are as follows. Examples of insecticides include: (1) organophosphorus compound-filled aluminum, butathiofos, cadusafos, chlorethoxyfos, chlorfenvinphos, chlorpyrifos, Chlorpyrifos-methyl, cyanophos (CYAP), diazinon, DCIP (dichlorodiisopropyl scale), dephosphorus (EDC) and dichlorvos (dichlorvos; DDVP), dimethoate, dimethylvinphos, disulfoton, EPN, ethion, ethoprophos, etrimfos, fen Fenthion (MPP), fenitrothion (MEP), fosthiazate, formothion, hydrogen filling, isofenphos, isoxathion, marathion ), mesulfenfos, methidathion (DMTP), monoctophos, naled (BRP), sulphate 24 320202 200901876 (oxydeprofos; ESP), balathon (parathion) ), phosalone, Phosmet (PMP), pirimiphos-methyl, pyridafenthion, quinalphos, phenthoate (PAP), profenofos, plus pine ( Propaphos), prothiofos, pyraclorfos, salithion, sulprofos, tebupirimfos, temephos, tetrachlorvinphos, Tobufoss, thiometon, trichlorphon (DEP), vamidothion, etc.; (2) urethane compound (alanycarb), bendicarb (bendiocarb) , benfuracarb, BPMC, carbaryl, carbofuran, carbosulfan, cloethcarb, ethiofencarb, zhongdingwei (fenbucarb), fenothiocarb, fenoxycarb, furathiocarb, isoprocarb (MIPC), metolcarb, methomyl, extinction Methicarb,

• I NAC, oxamyl, pirimicarb, propoxur; PHC, XMC, thiodicarb, xylylcarb, etc.; (3) Synechto Compounds arinathrin, allethrin, benfluthrin, beta-cyfluthrin, bifenin 25 320202 200901876 (bifenthrin), cyproterrin (cycloprothrin), Saifu Cyfluthrin 1 cyhalothrin, cypermethrin, deltamethrin, esfenvalerate, ethofenprox, fenpropathrin, Fenhua (fenvalerate), flucythrinate, flufenoprox, flumethrin, fluvalinate, halfenprox, imiprothrin, baifenning (permethrin), prallethrin, pyrethrins, resmethrin, sigma-cypermethrin, silafluofen, tef luthrin ), trondomethrin, and byfun Thrin), (EZ)-(IRS, 3RS; IRS, 3SR)-2, 2-dimercapto-3-prop-1-enylcyclopropanecarboxylic acid 2, 3, 5, 6-tetrafluoro-4- (methoxy methoxy) benzyl ester, (EZ)-(IRS, 3RS; 1RS, 3SR)-2, 2-dimercapto-3-prop-cycloalkenyl carboxylic acid 2, 3, 5, 6-tetrafluoro-4-methylbenzyl ester, (1RS, 3RS; IRS, 3SR)-2, 2-dimethyl-3-(2-methyl-1-propenyl)cyclopropanecarboxylic acid 2, 3,5,6-tetrafluoro-4-(decyloxymercapto)benzoquinone, etc.; (4) Nereisetoxin compound cartap, bentsap, thiosulfan ( Thiocyclam), monosultap, insecticidal double (1^5111 7 & 0), etc.; (5) new test compound imidacloprid, nitenpyram, sub-26 320202 200901876 acetamiprid, thiamethoxam, thiacloprid, clothianidin, dinotefuran, etc.; (6) Benzamidine urea compound chlorfluazuron , bistrifluron, diafenthiuron, diflubenzuron, fluazuron, flucycloxuron, flufen (flufenoxuron), hexaflumuron, lufenuron, novaluron, noifurumuron, teflubenzuron, triflumuron, etc.; (7) benzene Pyridazole compound acetoprole, fenpini (^1)1'〇]^1), vaniliprole, π-pyridr〇le, β-fipronil ( Pyrafluprole); (8) Bt toxin insecticide derived from the active scorpion of Bacillus thuringiensis and the crystalline toxin produced therefrom, and mixtures thereof; (9) hydrazine compound circumcision ( Chromafenozide), halofenozide, methoxyfenozide, tebufenozide, etc.; (10) organochlorine compounds aldrin, dieldrin, dechlorination 27 320202 200901876 (dienochlor), endosulfan, methoxychlor, etc.; (11) natural insecticide motor oil and nicotine-sulfate; (12) other insecticides avermectin (avermectin- B), new bromopropylate, buprofezin, chlorphrenia Enapyr), cyromazine, 1,3-dichloropropene, emamectin-benzoate, fenazaquin, flupyrazofos, aphid ethyl ester (hydroprene), indoxacarb, metoxadiazone, milbemycin-A, pymetrozine, pyra: pyridalyl, balippren (pyriproxyfen), spinosad, sulfluramide, tolfenpyrad, triazamate, flubendiamide, SI-0009, cyflumetofen ), arsenic acid, benclothiaz, calcium cyanamide, calcium polysulfide, chlordane, DDT, DSP, flufeninim > flonicamide, flurimfen, formetanate, metam-ammonium, metam-sodium, nidinotefuran , dinotefuran, potassium oleate, pr〇trifenbute, spiromesifen , lepimectin, sulphur, beauty 28 320202 200901876 He is a metaflumizone, spirotetramat, 丽1-0101, chlorantraniliprole and a compound of formula (A): Formula (A).: . R2

Wherein R1 represents a methyl group, a gas atom, a bromine atom or a halogen atom; R2 represents a fluorine atom, a chlorine atom, a bromine atom, a Cl-4 halogen or a C-4 haloalkoxy group; and R3 represents a fluorine, chlorine or bromine atom; R4 represents an argon atom, a Cl-4 alkyl group, a C3-4 alkenyl group, a Cs-4 alkynyl group or a C3-5 cycloalkyl group (the G-4 alkyl group, the C3-4 alkenyl group, the C3-4 alkynyl group, and the C3 group). The -5 cycloalkyl group may be optionally substituted with one or more groups selected from the group consisting of halogen I atom, cyano group, methylthio group, decylsulfinyl group, fluorenyl sulfonyl group and methoxy group. R5 represents a hydrogen atom or a methyl group; R6 represents a hydrogen, fluorine or chlorine atom; represents a hydrogen, a worn or a gas atom. Examples of smoldering agents (active ingredients of acaricides) include: acequinocyl, amitraz, benzoximate, bifenazate, bromopropylate , chinomethionat, chlorobenzilate, PCBSC chlorfenson, clofentezine, cyflumetofen, dicofol, snail Etoxazole), fenbutatin oxide, fenothiocarb, fenpyroximate, 29 320202 200901876 fluacrypyrim, fluproxyfen, hexythiazox, guanidine Propargite (BPPS), polynactins, pyridaben, pyrimidifen, tebufenpyrad, tetradifon, spirodiclofen , amidoflumet, cyenopyrafen, and the like. Examples of nematicides (active ingredients of nematicides) include: DCIP, fosthiazate, levamisol, decyl isothiocyanate, morantel tartarate, Misicafos and so on. Examples of fungicides include: acibenzolar-S-methyl, amobam, ampropyf los, anilazine, azoxystrobin, and Benda Benalaxyl, b6nodanil, benomyl, benthiavalicarb, benthiazole, bethoxazin, bitertanol , blasticidine-S, Bordeaux mixture, boscalid, bromuconazole, Dingsett 31!1:111〇331:6), hypochlorous acid 4 bow (〇 & 1 to 11111117 (11'0〇111〇1^6), calcium polysulfide, captan, carbendazol, carboxin, Carpropamid, chlobenthiazone, chloroneb, chloropicrin, tetrachloroisophthalonitrile 30 320202 200901876 (chlorothalonil; ΤΡΝ), worm fill ( Chlorthiophos), cinnamaldehyde, clozylacon, CNA (2,6-dichloro-4-n-phenylaniline), oxyhydrogen Copper, copper sulphate, cyazofamid, cyflufenamid, cymoxanil, cyproconazole, cyprodinil, cyprofuram, mellon Dazomet), debacarb, dichlofluanid, DD (l,3-dichloropropene), diclocymet, dafengjing (<^.1〇1^21116) , dietofencarb, difenoconazole, diflumetorim, dimefluazole, dimethirimol, damethacin ((^11161; 11〇111〇11) 11), diniconazole-M, dinocap, edifenphos, epoxiconazole, dithioamino nickel citrate, etaconazole, Ethaboxam, ethirimol, etridiazole, famoxadone, fenamidone, fenarimol, fenbuconazole, fen Fen (iazosulam), fenhexamid, fenoxanii, fenpiclonil, Fenpr〇pidin, fenprop i morph, fent i azon, fentin hydroxide, ferimzone, fluazinam ), fludioxonil, flumetover, fiumorph, fluoroimide, flurazepam (f) u〇trimaz〇ie), fluorine.菌菌酉31 320202 200901876 (fluoxastrobin), flUqUinconazole, f lusilazole, flusulfamide, flutolanil, flurifaol, forsythia (fosety, Al), fthalide, fuberidazole, furaiaxyl, furametpyr, feucarbanil, furconazole -cis), hexaconazole, hymexazol, IBP, imazalil, imibenconazole, chrome-trioctylbenzene sulfonate (iminoctadine) -albesilate), iminoctadine-triacetate, iodocarb, ipconazole, iprodione, iprovalicarb, indole (isoprothiolane), accelerated kasugamycin, kresoxim-methyl, mancozeb, msineb, mepanipyrim, mepronil, extinction Metalaxyl, metalaxyl-M, Weibai, Nasdaq Methasulfocarb), mercapto bromide, metconazole, methfuroxam, metominostrobin, metrafenone, metsuflovax, mildiomycin , milneb, myclobutanil, myclozolin, nabam, orysastrobin, ofurace, oxadixyl, Oxolinic acid, oxpoconazole, oxycarboxin, oxytetracycline 32 320202 200901876 (oxytetracycline), pefurazoate, penconazole, pencycuron ), picoxystrobin, polycarbamate, polyoxin, potassium bicarbonate, probenazole, prochloraz, procymidone, puppies Propamocarb-hydrochloride, propiconazole, propineb, proquinazid, prothiocarb, prothioconazole, five Chloronitrobenzene (〇1^111:〇26116;?〇^), Shixi°celein (5111±1〇0]^111), shiimeo simeconazole, sipconazole, hydrogencarbonate Sodium, sodium hypochlorite, spiroxamine, SSF-129, ((E)-2-[2-(2, 5-dimercaptophenoxy)phenyl]-2-methoxy Amino-N-methylethylamine, streptomycin, sulfur, tebuconazole, tecloftalam, tetraconazole, thiabendazole, thiadinil ), thiram (TMTD), thifluzamide, thiophanate-methyl, tolclofos-methyl, TPN, triadimefon, three tailong ( Triadimenol), triazoxide, trilamide, tricyclaZole, tridemorph, triflumizole, trifloxystrobin, triforine ), triticonazole, validamycin, vinclozolin, viniconazole, zineb, ziram, clumsy 33 320202 200901876 Zoxamide, amisubrom, enestroburin, mandipropamid, meptyldinocap, and the like. Examples of herbicides, phytohormones, and plant growth regulators include: abscisic acid, acetochlor, acifluorfen-sodium, alachlor, and grass ( Alloxydim), ametryn, amicarbazone, amidosulfuron, aminoethoxyvinyl alanine, aminopyralid, AC94, 377, methylamine Amiproph〇s-methyl, ancymidol, asulam, atrazine, aviglycine, azimsulfuron, flufenacet (beflubutamid), benefene (benf luralin), grass sulfonate ^1^1^〇38士6), free speed (^6113111 1'〇11-methyl), ground phosphorus (bensu.lide; SAP ), bentazone, benthiocarb, benzimizole, benzfendizone, benzobicyclon, benzofenap, benzophenone Adenine, benzylamino, melon, bialaphos, bifenox, brassinolide (Brassino) Leit), bromacil, bromobutide, butachlor, butafenacil, butamifos, butarate, oxazinamide (cafenstrole), calcium carbonate, calcium peroxide, carbaryl, chlomethoxynil, chloridazon, chlorsulfuron (ethyl), chloramphenicol 320202 34 200901876 ( Chlorphthalim), chl〇rpropham, chlorsulfuron, chl〇rtha dimethyl, ch 1 orth i ami d (DCBN), choline chloride-ketone Grass esterification ^(10)- buckle heart 丄), cinmethylin, cinosuifuron, clethodim, clomeprop, cloxyfonac-sodium, gasification Chi〇rmequat chloride, 4-CPA (4-chlorophenoxyacetic acid), cloprop, clofencet, cumyiuron, cyanazine, CyCianiiide, cyclosulfamuron, cyhalofop-bu1:yl, 2, 4- Gas phenoxyacetate, 2, 4-dipropionic acid (dichlorprop; 2, 4-DP), daimuron, dalapon (DPA), dimethenamid- P), Daminozide, dazomet, n-decyl alcohol, and diced sodium ((^(^11^3-5〇(^11111;111诎8), dibenzophenonitrile (dichlobeni) 1 ; DBN), ° dif lufenican, dikegulac, dimepiperate, dimethametryn, dimethenamid, diquat ), dithiopyr, diuron, endothal, epocholeone, esprocarb, ethephon, Ethidimuron, ethoxysulfuron, ethychlozate, etobenzanid, fenarimol, fenoxaprop-ethyl 4, fentrazamide, flazasulfuron, difluorosulfonate 35 320202 200901876 amine (florasulam), ° fluazifop-butyl, isopropyl Fluazolate, flucarbazone, flufenacet, flufenpyr, flumetralin, flumioxazine, vinacic acid Flufluanate-sodium, flupyrsulfuron-methyl-sodium, flurprimidol, fluthiacet-methyl, foramsulfuron, Forchlorfenuron, formesafen, gibberellin, glufosinate, glyphosate, halosulfuron-methyl, forest grass (hexazinone), imazamox, imimazic acid, imazapyr, imazaquin, imazosulfuron, inabenf ide, °Induction of acetic acid (IAA), ° butylation of butyric acid, iodosulfuron, ioxynil-octanoate, isouron, isoxachlortole ), isoxadifen, karbutilate, lacquerine Lactofen), lenacil, lisuron, LGC-42153, maleic hydrazide, mecoprop; MCPP, 2-mercapto-4-chlorophenoxy Acetate, MCPA-thioethyl, 2-methyl-4-phenoxybutyric acid ethyl ester, mefenacet, mefluidide, atrophin (mepiqUat), mesosulfuron, mesulphurone (mes〇trione), thiol herbicide 36 320202 200901876 (methyl-daimuron), metolachlor, metribuzine, 曱Metasulfuron-methyl, rice, magnesium, naphthylacetate, 1-naphthylamine, naproanilide, napropamide, n-decyl alcohol, terminal sulphate (nicosulfuron), n-phenyl hydrazone, orbencarb, oxadiazon, oxaziclomefone, xine-sulfate, multi-effect saliva Pac 1 obutrazo 1 ), paraquat, pe 1 argon ic acid, pendimethalin, penoxsulam, ring Penoxoxazone, pethoxamid, phenmedipham, picloram, picolinafen, piperonyl butoxide, piperophos, Pretilachlor, primisulfuron-methyl, procarbazone, prodiamine, profluazol, profoxydim, Prohexadione-calcium, prohydrojasmon, prometryn, propanil, propoxycarbazone, pentazone; '0?72&;11^(16),霸草灵({7『&士11^611-61;]^1), pyrazolate, pyrazoosulfuron-ethyl, pyrazoxyfen , pyribenzoxim, pyributicarb, pyridafol, pyridate, pyrifalid, pyrimanobac-methyl, pyrimidine Ether (pyrithiobac), kekegrass 37 320202 200901876 (quinclorac), quinoclamine, ethyl oxalate ( Quizalofop-ethyl), rimsulfuron, sethoxydim, siduron, simazine, simetryn, sodium chlorate, continued Sulfosulfuron, SWEP (MCC), tebuthiuron, tepraloxydim, terbacil, terbucarb (MBMPC), thenyl chloride, ° Thiazufluron, thidiazuron, thifensulfuron-methyl, triaziflam, tribufos, triclopy, extinction Tridiphane, trifloxysulfuron, trifluralin, trinexapac-ethyl, trifluorosulfuron (t; ritosulfuron), uniconazole (tmiconazole-P) ), velocate (VPTC), fluorine 11 to flucetosulfuron, (orthosulfanuron), lindolin (pinozaden), scutellite yellow (pyrasulfotole), tefu 嗣 嗣 (tefuryltrione), post Tembotrione, thiencarbazone-methyl, and the like. Further, the pest control preparation of the present invention may be mixed with a synergist such as piperonyl butoxide, sesamex, sulfoxide, N-(2-ethylhexyl)-8, 9, 10 - Sanyuan borneol-5-ene-2, 3-dicarboxylimine imine (MGK 264), N-mercaptoimidazole, anti-WARF resistant strain, TBPT, TPP, IBP, PSCP, CM, phenyl tributyl Copper, diethyl maleate, DMC, FDMC, ETP, ETN, and the like. In addition, it can be mixed with safeners such as oxalofen 38 320202 200901876 (benoxacor), detoxified quinone (cl〇qUint〇cet-mexyl), cymetrinil, daimuron, dichloropropenylamine ( Dichlormid), fetchl〇raz〇ie-ethyl, fenclorim, flurazole, fluxofenim, furiiaz〇ie, Mefenpyr-diethy 1 (MG), MG191, naphthalic anhydride, oxabetrini 1 and the like. " Furthermore, the pest-preventing preparation of the present invention can be used in the form of a mixture with a topical parasitic arthropod controlling agent, such as a pyrethroid agent, an IGR agent (for example, a juvenile hormone mimic, such as Meth〇prene) and fenoxycarb; chitin synthesis inhibitors such as lufermron, fiufenoxuron, novaluron, hexaflumuron, defolon (teflubenzuron), diflubenzuron and trif lumuron' and insect growth regulators, such as Cyr〇mazine and pyr i proXyphen, or neonicotinoids "(7) 乜 (10) ^) (such as eneenpyram). It can also be administered internally to animals in combination with the above-mentioned IGR agent mixture or with internal insecticide control agents (such as macrolides (such as macrolides). Macrolide) compounds, such as a combination of selamectin, ivermectin, milbemycin, and moxidectin. a mixture of fungal agents for use in animals, vaccines, and treatments Animals, nutritional supplements or feeds. Examples of pests that are effective against s (I) include harmful arthropods, such as 320202 39 200901876 such as harmful insects, harmful powder worms, etc. Specific examples are as follows. Hemiptera (hemiptera) ): Delphacidae such as Laodelphax striatellus, Nilaparvata lugens, Sogatella furcifera, etc.; Deltocephalidae such as Nephotettix cincticeps, two black Nephitettixvirescensm, etc.; Aphididae such as Aphis gossypii, Myzus persicae, Brevicoryne brassicae, Macrosiphum euphorbiae, Solanum tract Aulacorthum solani, Rhopalosiphum padi, Toxoptera citricidus, etc.; Pentatomidae, such as Nezara antennata, Riptortus clavetus, Chinese spider edge Leptocorisa chinensis, Eysarcoris parvus, Halyomorpha mista, etc. Aleyrodidae such as greenhouse whitefly (Trialeurodes • - - . vaporariorum), silver leaf whitefly (Bemisiaargentifolii), tobacco whitefly (Bemisia tabaci), etc.; Coccidae such as orange red kidney shield (Aonidiella aurantii ), Comstockaspis perniciosa, Unaspis citri, Ceroplastes rubens, Icerya purchasi, etc.; Tingidae; (Psyl 1 idae); and so on. 40 320202 200901876 Lepidoptera: Lycidae (?7"1丨(186) such as Dictyophora ((:1^1〇suppressalis), Tryporyza incertulas, Rice leaf curler (Cnaphalocrocis medinalis), Notarcha derogata, Plodia _ interpunctella, Ostrinia furnacalis, Hellula undalis, turf teterrellus, etc.; Noctudidae For example, Spodoptera litura, Spodoptera exigua, Pseudaletia separate, Mamestra brassicae, Agrotis ipsilan, black spot silver Plusia nigrisigna, Trichopulsia spp., Helious spp., Hel icoverpha spp., etc.; Piperidae such as Pierisrapae ;Tortricidae, such as Adoxophyes spp., Eastern fruit moth (Grapholita molesta), bean leaf filling, . . . (Leguminivora glycinivorella), red bean roll (Matsumuraeses azukivora), Adoxophyes orana fasciata, Adoxophyes spp., Homona magnanima, Archips fuscocuprearms, Cydia pomonella, etc. (Graci 1 lari idae), for example, Calopti lia theivora, Phyllony cterringoneella, etc.; Carpos i ni dae such as Carpodendron (Carpos i na 41 320202 200901876 niponensis); Ly0netiidae such as Lyonetia spp., Lymantriidae such as Lymantria spp., Euproctis spp., etc.; Yponomeutida such as small moth ( Piutellaxylostella), etc.; Gelechi idae such as Pect inophora gossypiella, Phthorimaea operculella, Arctiidae, such as Hyphantriacunea, Mothidae (Tineidae) such as Tinea translucens, Tineola bisselliella, etc.; Thysanoptera: Thrips such as Frankliniella occidentals, Thrips parmi, Scirtothrips dorsalis, and Thripstabaci, Taiwanese flowers Lin马 (Frankliniella intonsa) and so on. Dipteria: Musca domestica, Culex pipiens pa 11 ens, Tabanus tr i gonus, Hy 1 emya antique, Hylemya platura ), Anopheles sinensis, Agromyza oryzae, Hydrellia griseola, Chlorops. > oryzae, Dacus cucurbitae, Mediterranean fruit Ceratitis capitata, Liriomyza trifolii, etc. Coleoptera: 42 320202 200901876 Ladybug 12 (11卩1111¥1£1111:1〇〇1; 0口1111(:13士&), Aulacophora femoralis, Phyllotreta striolata, Oulema oryzae, Echinocnemus squameus, Lisorhoptrus oryzophilus, Anthonomus grandis, and green bean (Callosobruchus) Chinensis), Sphenophorus venatus, Popillia japonica, Anomala cuprea, Diabrotica spp., KLeptinotarsa decemlineata, stag beetle Agriotes spp.), Lasioderma serricorne, Anthrenus verbasci, Tribolium castaneum, Lyctus brunneus, Anoplophora malasiaca, vertical pit Tipus (pinicus piniperda) and so on. Orthoptera: Locusta migratoria, Gryllotalpa africana, 〇xya yezoensis, Oxya japonica, etc. Hymenoptera: Athalia rosae, Acromyrmex spp., s〇lenopsis spp, etc. Nematode: Aphelenchoides bes.seyi, Nothotylenchus acris, etc. 43 320202 200901876 Dictyoptera ··Blatte 1 la germanica, Periplaneta fuliginosa, Periplaneta americana, Periplaneta brunnea, Blatta Orientalis) and so on. Acarina: Tetranychidae such as Tetranychus urticae, Panonychus citri, Oligonichusspp., etc.; Eriophyidae such as orange thorn Aculopspelekassi, etc.; Tarsonemidae such as Polyphagotarsonemus latus; Tenuipalpidae; Tuckerellidae; Ixodes spp. Haemaphysalis longicornis, Haemaphysalis f.lava, Taiwanese Dermacentor taiwanicus, Ixodes ovatus, Ixodes persulcatus, Boophilus Microplus), Rhipicephalus sanguineus, etc.; Acaridae such as Tyropha panthus putrescentiae, Dermatophagoides such as Dermatophago ides pteronyssinus; Carnivores Cheyletus such as Cheyletus eruditus, Cheyletus malaccensis, Cheyletus moorei, etc.; Section (Dermanyssidae spp.) And so on. 320202 200901876 Formulations comprising the compound (i) or a salt thereof of the present invention can also be used in the field of disease treatment for animal husbandry and animal husbandry, and can also be used for arthropods or parasitic parasites and/or in vitro. Insects, such vertebrates are, for example, humans, cows, sheep, goats, pigs, poultry, dogs, cats, fish, etc. to maintain public health. Examples of such harmful pests include Ixodes spp. (e.g., Ixodes scapular is), Boophilus spp. (e.g., Boophilus microplus), and flower bud (Amblyomma) Spp.), Hyalomama spp., Rhipicephalus spp. (eg Rhipicephalus sanguineus), Haemaphysalis spp. (eg, Haemaphysalis longicornis), Dermacentor spp., Ornithodoros spp. (eg Ornithodoros moubata), Dermanyssus gallinae, Ornithonyssus sylviarum, Sarcoptes spp .) (eg, Sarcoptes scabiei), cochlear (Psoroptes spp.), snail (Chorioptes spp.), snail (Demodex spp.), genus genus (£111:1'〇1111^ (:111& spp.), Aedes spp. (eg Aedes albopictus), Anopheles spp., Culex spp., Culicodes spp .), Musca spp., Hypoderma spp., Gasterophil Us spp·), Haematobia spp., Tabanus spp., Simulium spp., Triatoma spp., Phthiraptera (eg edulis) Genus (Damalinia spp.), caterpillar 45 320202 200901876 (Linognathus spp.), genus Haematopinus spp., Ctenocephalides spp.) (eg, Ctenocephalides felis), rats Xenopsylla spp., Monomorium pharaonis; and Nematode such as Trichostrongylus spp. (eg, Trichostrongylus brasi 1 iensis, Trichostrongylus axei) , Nippostrongyluscolubriformis, Trichinella spp., Trichinella spiralis, Haemonchus spp. (eg Haemonchus contortus), Nematodes (Nematodirus spp.) (eg Nematodirus battus) - Ostertagia spp. (eg Ostertagia circumcincta), Guberian line (Cooperia spp.), Tapeworm short spore membrane (Hymenolepis nana) and the like. In the pest control method of the present invention, the compound (I) or a salt thereof can be used as it is. Alternatively, the compound (I) or a salt thereof is formulated into the above-mentioned pest control preparation of the present invention' and applied to the pest or its habitat in the same manner as the conventional pest control preparation to allow the growing pest to contact or ingest the preparation. Examples of the habitat of the pest of the present invention include paddy fields, dry fields, orchards, uncultivated land, and residential areas. Examples of the application method include spray treatment, soil treatment, seed treatment, and treatment of hydroponic water. Specifically, the spraying treatment of the present invention is, for example, a method of applying the active ingredient (compound (I) or a salt thereof) to a plant surface 46 320202 200901876, such as leaf spraying and stem spraying, to visualize the control of pests effect. Soil treatment is, for example, a method of treating soil or irrigation water with an active ingredient to render the active ingredient permeable and transferable to the interior of the crop to protect it from damage, for example to prevent pests from being damaged by the roots of the roots. Specific examples of soil treatment include planting hole treatment (plant hole spraying, and soil incorporation after acupoint treatment), strain ro〇t treatment (root spraying, In the root soil mixing, root irrigation, and root treatment in the late seedling stage), planting groove treatment (1) direct groove spraying, and soil mixing in the planting), row processing (planting spray, soil mixing in planting, and planting in the growing season), planting in the sowing period (planting in the sowing period, and planting in the sowing period) Soil mixing), comprehensive treatment (comprehensive soil treatment, and integrated soil mixing), other soil spraying treatment (spraying of the granule preparations for growth, spraying under the stem or around the main stem, spraying on the surface of the soil) Sprinkling, soil surface mixing, seeding (s〇wing h〇le) treatment, ridge surface spray, and seed sprinkling), other irrigation treatments (soil irrigation, seedling irrigation, perfusion (/ Nstillati〇n) Treatment, irrigation at the base, drip irriSation, and chemical chemigation), phase treatment (Tianxiang spray, and seedling box irrigation), seedling treatment (seedling tray) Spraying 'Ling and seedlings' irrigation), nursery bed treatment (seed bed spraying, field bed irrigation, lowland seedbed spraying, and seedling infiltration), bed soil mixing (bed soil mixing, and before planting) Bed soil mixing), and other treatments (listing incorporation, plowing and application 320202 47 200901876 fertilizer, surface soil mixing, awnings only continued: soil mixing under the edge, phytosanitary, granule formula Flower cluster treatment, vertical treatment, and paste fertilizer mixing). The seeding system is, for example, a method of applying the active ingredient directly or at the level; the seed, the potato seed or the crop near the ball is poor to protect the crop from damage, for example, to avoid damage to the pest, so as to manifest the pest. Flood prevention%dan*3_ 孓哂°God fruit. Specific examples thereof include spraying, painting, impregnation, injection, coating, and granule coating. The hydroponic treatment is, for example, a method in which an active ingredient is added to hydroponic water to transfer the active ingredient permeable to the inside of the crop to protect it from damage, for example, to prevent pests from damaging the roots thereof. There are H cases including hydroponic water mixing and hydroponic water infusion. The amount of application in such methods can vary depending on when, where and how the formulation is administered. In general, it is preferred to apply the preparation such that the active ingredient (compound (I) or a salt thereof) is from 0.3 to 3, 〇〇〇g, preferably from 3 to 3, OOOg per hectare. When the pest control preparation of the present invention is a wettable powder, the preparation may be diluted at the time of application so that the active ingredient concentration becomes 〇1 to 1,00 ppm (diluted with water), preferably 10 to 5 Å. Another cancerous sample of the present invention provides a method for administering an internal (in vivo) or an external (body surface) of a pest control preparation of the present invention to a vertebrate, which is a systemic or non-invasive arthropod or parasite that inhabits a vertebrate. Systematic eradication. Internal administration methods include oral administration, rectal administration, implantation, and subcutaneous, intramuscular, and intravenous injection. External administration methods include transdermal administration. It is also possible to formulate feeding animals to eradicate unsanitary pests that appear in the refractory animals. When the pest control preparation of the present invention is applied to a pest or a pet animal in the presence of a pest, the dosage is largely changed depending on the administration method. In general, β is preferably administered as a preparation such that the active ingredient (compound (I) or a salt thereof) is 〇1 to 2, OOO mg, preferably 〇. 5 to 1, OOO mg ° per kg body weight of the animal. Further description will be made by way of examples, production examples, reference production examples, formulation examples, and test examples. However, the present invention i is not limited thereto. The scouring of the column chromatography at the respective examples, production examples and reference production examples was monitored by TLC (thin layer chromatography). Kieselgel 60F254 (70 to 230 net) manufactured by MERCK & CO., LTD by τιχ

Eye) As a TLC plate, the same solvent as the solvent used for column chromatography was used and detection was performed using a UV detector. Use of ΚΑΝΤΟ CHEMICAL CO., LTD. (spherical, particle size 63 to 210 nm) of yt 60 as a column of tannins and using FlorisilClOO to 200 mesh manufactured by WAKO PURE CHEMICAL INDUSTRIES LTD.) as magnesium silicate ) Pipe string. For medium pressure preparative hplc, Ultrapack (filler: Shiqi gum) manufactured by YAMAZENCO. was used. When a mixed solvent is used as the developing solvent, the mixing ratio is expressed by the volume in the brackets. The dirty R spectrum was determined by proton NMR using tetramethyl decane as an internal standard, and a JE〇L AL-400 (400 MHz) type and a Bruker AVANCE 400 (400 MHz) type spectrometer were used. All J values are shown in ppm. The measurement temperature is 25 unless otherwise stated. . . The abbreviations and names used in the following Preparations and Reference Preparations mean the following. 49 320202 200901876 s : single peak, br : broad peak, brs : wide single peak, d : double peak, t : triple peak ' Q · four peaks, Me : methyl, Et: ethyl, Ph: phenyl, Pr- n (or n-Pr): propyl, Pr-i (or i-Pr or ipr): isopropyl, Pr-cycl0 (or cyc 1 o-Pr): cyclopropyl, Bu-n (or n- Bu) : butyl, Bu-i (or i_Bu): isobutyl, Bu-s (or s-Bu): second butyl, Bu-t (or t-Bu): second butyl, THF: Tetrahydrofuran, DMF: dimethylformamide 'room temperature: 15 to 25. . . Specific examples of the compound (I) are as follows:

Compound 1-1 to Bu 6690, wherein R represents a bicyclo [4. 4.0] - 2 - fluorenyl group and the geometric isomers of the (X) n, (z) n & CH=CH double bond are as follows: Combination G"; Compound 2-1 to 2-6690, wherein R represents a bicyclo[4. 4.O]·^-fluorenyl group, and the geometrical differences of the (X)m, (Z)n&CH=CH double bonds The structure is the following "combination G"; compound 3-1 to 3-6690 'wherein R represents a bicyclo[4. 3. 0]-2-indenyl group, and in (X)m, (Z)n and CH = The geometric isomer of the CH double bond is the following "combination G", compound 4-1 to 4-6690, wherein R represents a bicyclo[4.3.0]-nonane-3_ group, and at (X)m, (2 And the geometrical isomer of the CH=CH double bond is the following "combination G"; compounds 5-1 to 5-6690, wherein R represents a bicyclo[4. 3. 〇]-7-fluorenyl group, and The geometric isomers of X)m, (Z)n&CH=CH double bonds are the following "combination G"; compounds 6-1 to 6-6690, wherein R represents a bicyclo[4· 3. 〇]-8- Mercapyl, 320202 50 200901876 and the geometric isomers of the (X)m, (Z)n and CH=CH double bonds are the following "combination G"; compounds 7-1 to 7-6690, where R represents a bicyclic ring [ 4 2. 0]_2_octyl, and at (X)m, (Z)n and CH=CH The geometrical isomer of the double bond is the lower 琏 "combination G"; the compound 8-1 to 8-6690, wherein R represents a bicyclo[4 2. 〇]_3_octyl group, and is at (X) m, (Z) n And the geometric isomer of 01=(:11 double bond is the following "combination 6"; compound 9-1 to 9-6690, wherein R represents a bicyclo[4 2. 〇]_7_octyl group, and (X) m, (Z) n & CH=CH double bond geometric isomer is the following "combination G"; compound 10-1 to 10-6690' wherein R represents bicyclo [4. 1 〇] _2 heptyl, and The geometric isomers of the (X)», (Z) η and CH=CH double bonds are the following "combination G"; the compound 11-1 to 11-6690' wherein R represents a bicyclo[4. 1〇]_3 The geometric isomer of the heptyl group and the (X)», (Z)n&CH=CH double bond is the following "combination G"; the compound 12-1 to 12-6690, wherein R represents a bicyclo[4. 〇] a 7-heptyl group, and the geometric isomer of the (X)m, (Z)n & CH=CH double bond is the following "combination G"; compound 13-1 to 13-6690, wherein R Indicates a bicyclo[3:3. 〇]_2_octyl group, and the geometric isomer of the (X)B, (Z)!^ CH=CH double bond is the following "combination G"; compound 14-1 to 14 -6690' where R represents a double ring [3.3. 〇]-3 The geometric isomers of the octyl group and the (X)m, (Z)n and CH=CH double bonds are the following "combination G"; the compounds 15-1 to 15-6690' wherein R represents a bicyclic ring [3.2. ]_2_heptyl, and the geometric isomer of (X%, (Z)n& CH=CH double bond is the following "combination G"; compound 16-1 to 16-6690, wherein R represents a bicyclo[3] ·2. 〇]_3_heptyl, and the geometric isomer of (X)m, (Z)d CH=CH double bond is the following "combination G"; compound 17-1 to 17-6690' where R Represents a bicyclo[3.2. 〇]-6-heptyl group, and the geometric isomer of the (X)B, (Z)n&CH=CH double bond is the following "combination G"; compounds 18-1 to 18- 6690, wherein R represents a bicyclo[3·丨·〇]_2_hexyl group, 320202 51 200901876 and the geometric isomer of the (X%, (Z)n& CH=CH double bond is the following "combination G"; 19-1 to 19-6690, wherein R represents a bicyclo[3·1〇]_3-hexyl group, and the geometric isomers of the (X)m, (Z)n and CH=CH double bonds are as follows: Compound 20-1 to 20-6690, wherein R represents a bicyclo[3. 1〇]-6-hexyl group, and the geometric isomer of the (X)B, (Z)n&CH=CH double bond is as follows "combination G"; 25-1 to 25-6690 'wherein R represents a (bicyclo[44. 〇]_2_fluorenyl)methyl group, and the geometric isomers of the (X)n, (Z)n and OJirCH double bonds are as follows: Combination G"; compound 26-1 to 26-6690, wherein β represents (bicyclo[4.4. 〇]_3_fluorenyl)methyl, and the geometrical difference of (X%, (Z)n& CH=CH double bond The structure is the following "combination G"; compound 27-1 to 27-6690, wherein R represents (bicyclo[3. 3. 〇]-2-octyl)methyl, and (X)ra, (Z) The geometric isomer of the n&CH=CH double bond is the following plant combination G"; Compound 28-1 to 28-6690, wherein R represents (bicyclo[3. 3. 〇]-3~octyl)methyl 'And the geometric isomer of (X)m, (Z)n^CH=CH double bond is as follows: "combination G"; .: compound 29-1 to 29-6690, where R represents (bicyclic [ 4.3· 〇]-7-fluorenyl)methyl' and the geometric isomers of the (X)m, (Z)n&CH=CH double bond are as follows: "combination G"; compound 30-1 to 30 -6690, wherein 1? represents a (bicyclo[4.3.0]-8-fluorenyl) fluorenyl group, and the geometric isomer of the (X)m, (Z)n&CH=CH double bond is as follows: G"; compounds 31-1 to 31-6690, which R represents (bicyclo[4. 1. 〇]-2 gh 52 320202 200901876) fluorenyl, and the geometric isomers of the (X)n, (Z)n and CH=CH double bonds are as follows: G", compound 32-1 to 32-6690, wherein R represents (bicyclo[4.1.0]-3-heptyl)fluorenyl, and is in the (X)m, (Z)n&CH=CH double bond The geometric isomers are the following "combination G"; compounds 33-1 to 33-6690 'wherein R represents (bicyclo[2. 1 · 1]-2-heptyl)fluorenyl' and at (X)m, The geometric isomers of the (Z)n and CH=CH double bonds are the following "combination G", compounds 34-1 to 34-6690 'where R is represented; i-(bicyclo[4. 4. 〇]-2- The geometric isomer of the oxime)ethyl group and the (X)», (Z)n&_CH=CH double bond is the following "combination G"; the compound 35-1 to 35-6690, wherein R represents i- (bicyclo[4. 4. 〇]-3-indenyl)ethyl, and the geometric isomer of (X%, «) „ and CH=CH double bond is the following “combination G”; compound 36-1 To 36-6690, wherein r represents ι_(bicyclo[3. 3. 〇]-2-octyl)ethyl, and the geometric isomers of the (X%, (2) „ and CH=CH double bonds are Said "combination G"; compound 37-1 to 37-6690, where r The geometrical isomer of b (bicyclo[3. & 〇]_3_octyl)ethyl and in (X)m, (2) „ and CH=CH double bond is the following “combination G”; 38-1 to 38-6690, wherein r represents 丨_(bicyclo[4. 3. 〇] 7_ fluorenyl)ethyl' and geometrical isomerism of (X)m, (Z)n&CH=CH double bond The substance is the following "combination G"; compound 39-1 to 39-6690, wherein r represents (bicyclo[4. & 〇布8_320202 53 200901876 fluorenyl) ethyl, and (X)m, (Z) The geometric isomers of n and CH=CH double bonds are the following "combination G"; compounds 40-1 to 40-6690, wherein R represents b (bicyclo[4.heptyl)ethyl' and (X)m The geometric isomer of (Z)n & CH=CH double bond is the following "combination G"; compound 41-1 to 41-6690, wherein r represents bicyclo[4.h 〇] 3_heptyl)ethyl 'And the geometric isomers of the (X)n, (Z)n&CH=CH double bonds are as follows: "Combination G"; ^ Compounds 42-1 to 42-6690, where r represents Bu (bicyclic [ 2· 2. Heptyl)ethyl, and the geometric isomers of the (X)·», (Z)n and CH=CH double bonds are the following “combination G”; compounds 43-1 to 43-6690, Where r 2_(bicyclo[4. 4. 〇]_2_ fluorenyl)ethyl, and the geometric isomer of (X%, (Z)n & CH=CH double bond is the following "combination G"; compound 44- 1 to 44-6690, wherein r represents 2_(bicyclo[4. 4. 〇]-3-indenyl)ethyl, and the geometric isomer of (X)m, (Z)n&CH=CH double bond Is the following "combination G"; compound 45-1 to 45-6690, wherein r represents 2-(bicyclo[3. 3. 〇]-2-octyl)ethyl' and in (X)mv (Z)n& The geometric isomer of CH=CH double bond is the following "combination G"; compound 46-1 to 46-6690 'where r represents 2-(bicyclo[3. 3. 〇b 3~ octyl)ethyl, The geometric isomers of (X)m, (redundant and CH=CH double bonds are the following "combination G"; compounds 47-1 to 47-6690, where R represents 2-(bicyclo[4. 3. Ο]-% 54 320202 200901876 The geometrical isomer of the ethyl group and the double bond of (X)·», 〇„ and CH=CH is the following “combination G”. Compounds 48-1 to 48- 6690, wherein r represents 2-(bicyclo[4. 3. 〇]~8-fluorenyl)ethyl, and the geometric isomers of (X)m, (ZV and CH=CH double bonds are as follows) G"; compound 49-1 to 49-6690, where r represents 2 (Bicyclo[4. 1. 〇]-2-heptyl)ethyl' and the geometrical isomer of (X%, (Z)n& CH=CH double bond is the following "combination G"' compound 50- 1 to 50-6690, wherein r represents 2-(bicyclo[4.1.0μ3_heptyl)ethyl, and the geometric isomer of the (X)n, (Z)n&CH=CH double bond is the following "combination" G"; compounds 51-1 to 51-6690, wherein r represents 2_(bicyclo[2.iihheptyl)ethyl, and the geometric isomers of (X)m, (2乂 and CH=CH double bonds are Said ... combination G"; "combination G" [number of compound branches: (x) m, (z) n, geometric isomer of ch=CH double bond] = f C-2: 4-F, H ,E] , C-3:4-F,H,z] Ύ [-4:4-C1, Η, Ε], [_ .5:4-Cl,H,Z], [-6:4- Br, H, E], [-7: 4-he], [-8: 4-Me, H, ^:] 55 320202 200901876 (Me) 2CH, H, E], [-13: 4-CF3, H, E], [-14: 4-CF3, Η, Z], [-15: 4-C2F5, H, E], [-16: 4-C3F7, H, E], [-17: 4- (CF3) 2 CF, Η, E], [-18:4-(CF3 )2CH,H,E], [-19:4-CHF2,H,E], [-20 : 4-CH2 F, Η , E], [-21:4-CF3CH2,H,E], [-22:4-Me〇,H,E], [-23:4-MeO,H,Z], [-24:4- EtO, H, E] , [-25:4-C 3H7〇,H,E] , [26: 4-(Me) 2 CHO, Η, E], [-27 :4-N02,H,E], [-28:4-N02,H,Z] , [-29:3-F,H,E], [-3〇:3-.F,H,Z], [-31:3-C1,H,E], C-32:3-Cl, H,Z], [-33:3-Br,Η,E], [-34:3-Ι,Η,Ε], [-35:3-Me,H,E], [-36:3- Me,H,Z], [-37:3-Et,H,E], [-38:3-C3H7,H,E], [-39:3-(Me)2CH,H,E], [ -40:3-CF3,H,E], [-41:3-CF3,H,Z],[-42:3-C2F5,H,E],[-43:3-C3F7,H,E] , [-44:3-(CF3)2CF,H,E], [-45:3-(CF3)2CH,H,E]., [-46:3-CHF2,H,E],[-47 :.3-CHF2,H,Z], [-4 8 :3-CH2 F, Η, E], [-49:3-CH2F,H,Z], [-50:3-CF3CH2,H,E ],[-51:3-MeO,H,E],[-52:3-MeO,H,Z], [-53:3-EtO,H,E], [-54:3-C3H7Ο,Η , E] , [-55:3- (Me)2CH0,H,E], [-56:3-N02,H,E],[-57:2-F,H,E],[-58: 2-C1,H,E],[-59:2-Br,H,E],[-60:2-I,H,E],[-61:2-Me,H,E], [- 62:2-Et,H,E], [-63:2-C3H7,H,E], [-64:2-(Me)2CH,H,E],[-65:2-CF3,H, E], [-66: 2-C2F5, H, E], [-67: 2-C3F7, H, E], [-68: 2-(CF3 ) 2CFfHrE], [-69: 2-(CF3)2CH, H, E], [-70: 2-CHF2, H, E], [-71: 2-CH2F, H, E], [-72: 2-CF3CH2,H,E],[-73:2-MeO, Η, E], [-7 4:2-EtO,H,E]., [A 75:2-03Η70γΙ1,Ε], [- 76:2- (Me) 2 CHO, Η, E], [77:2-N〇2,H,E], '[-78:2/3-F2,H,E],[-79: 2,4-F2,H,E],[-80:2,5-F2,H,E], [-81:2, 6-F2,H,E], C-82 : 3,4-F2 ,Η, E ],[- 83:3,4-F2,H,Z], [-84:3,5-F2rH,E], [-85:3,5-F2,H,Z], -86:2,3-Cl2,H,E], [-87:2,3-Cl2,H,Z], [-88:2,4-Cl2,H,E],[- 56 320202 200901876 89 :2,4-Cl2,H,Z] , C-9〇:2,5-Cl2,H,E] , [-91:2,5-Cl2,H,Z],[-92:2,6 -Cl2,H,E], [-93:3,4-Cl2,H,E], [-94:3,5-Cl2,H,E], [-95:2,3-Br2,H, E], [-96:2,4-Br2,H,E], [-97:2,5-Br2,H,E], [-98:2,6-Br2,H,E],[- 99:3,4-Br2,H,E], [-100:3,5-Br2,H,E], [-101:2,3-Me2,H,E], [-102:2,4 -Me2,H,E] , C-103:2,5-Me2, Η,E], C -104:2,6-Me2,H,E ] , ( -105:3,4-Me2, Η, E ] , 〔'106:3,5-

Me2,H,E], [-107:2,3-Et2,H,E], [-108:2,4-Et2,H,E],[-109:2,5-Et2,H,E ], [-110:2,6'Et2,H,E], [-lll:3,4-Et2,H,E], [-112:3,5-Et2,H,E],[-113 :2,3-(CF3)2,HrE],[-114:2,4-(CF3)2,H,E],[-115:2,5-(CF3>2,H,E], -116: 2r6-(CF3)2, H, E], [-117:3,4-(CF3)2,H,E], [-118:3,5-(CF3)2rH,E],. [-119:2,3-(CHF2)2,H,E], C-120:2,4-(CHF2)2,H,E], [-121:2,5-(CHF2)2,H ,E] (CHF2)2,H,E](CH2F)2,H,E](CH2F)2,H,E](CH2F)2,H,E] [-123:3,4-[-125 :2,3-C -127:2,5-C -129:3,4-[-131:2,3- [-122:2,6-(CHF2)2,H,E], [-124 :3,5-(CHF2)2,H,E] '[-126:2,4-(CH2F)2,H,E], [-128:2,6-(CH2F)2,H,E 3 , [-130:3,5-(CH2F)2,H,E )( (MeO)2,H,E], [-132:2,4-(MeO>2,H,E], [-133 :2,5-(MeO)2,H,E], [-134:2,6-(MeO)2,H,E],[-135:3,4-(MeO)2,H,E] , [-136:3,5-〇yieO)2,H,E],[-137:2,3-(EtO)2,H,E],[-138:2,4-(EtO)2, H,E], [-139:2,5-(EtO)2fH,E) f [-140:2,6-(EtO)2,HfE), (-141:3,4-(EtO)2, H, E], i-l'42: 3,5-(EtO 2,H,E],[-143:2-Cl-3-F,H,E], [-144:2-Cl-4-F,H,E], [-145:2-Cl- 5-F,H,E3 r [-14 6:2-01-6- F,H,E],[-147:3-Cl-2-F,H,E],[-148:3-Cl -4-F,H,E],[-149:3-Cl-5-F,H,E], [-15〇:4-Cl-2-F,H,E], [-151:4 -Cl-3-F,H,E],[- 57 320202 200901876 152:2-F-3-Me,H,E ], [-153:2-F-4-Me,H,E], [ -154:2-F-5-Me,H,E] , C-155:2-F-6-Me,H,E] , [-156:3-F-2-Me,Η,E ], [- 157:3-F-4-Me,H,E ) , [ -158:3-F-5-Me,H,E ], [-159:4-F-2-Me,H,E] , [-160:4-F-3-Me,H,E], [-161:2-Cl-3-Me,H,E],[-162:2-Cl-4-Me,H,E ], [-163:2-Cl-5-Me, Η, E], [-164:2-C1-6-

Me, H, E], [-165: 3-Cl-2-Me, H, E], [-166: 3-Cl-4-Me, Η, · E], [-167:3-Cl- 5-Me,H,E],[-168:4-Cl-2-Me,H,E],[-169:4-Cl-3-Me,H,E],[-170:2-F -3-CF3,H,E],[-171:2-F-4-CF3,H,E],[-172:2-F-5-CF3,H,E], [-173:2- F-6-CF3, Η, E], [ -174:3-F-2-CF3,H,E], [-175:3-F-4-CF3,H,E],[-176:3 -F-5-CF3,H,E], [-177:4-F-2-CF3,H,E], [-178:4-F-3-CF3,H,E],[-179: 2-C1-3-CF3,H,E], [-180:2-Cl-4-CF3,H,E], [-181:2-Cl-5-CF3,H,E],[-182 :2-Cl-6-CF3,H,E] , [-183:3-Cl-2-CF3, Η,E], [-184:3-01-4-CF3,H,E],[- 185:3-Cl-5-CF3,H,E],[-186:4-Cl-2-CF3,H,E],[-187i4-Cl-3-CF3,H,E], [-188 :2-Me-3-CF3,H,E], [-189:2-Me-4-CF3,H,E3,[-190:2-Me-5-CF3,H,E], (-191 :2-Me-6-CF3 , Η, E], [-192:3-Me-2-CF3,H,E], [-193:3-Me-4_CF3, Η, E], [-194: 3-Me-5-CF3,H,E], [-195:4-Me-2-CF3,H,E], [-196:4-Me-3-CF3,H,E],[- 197 :2-F-3-MeO,H,E],C-198:2-F-4-MeO,Η,E], [ -199:2-F-5- 1

MeO,H,E] r [-200:2-F-6-MeOrH,E] , [-201:3-F-2-MeO,H,E],J-202:3-F-4-MeO ,H,E], [-203:3-F-5-MeO,Η,E ] , [-204:4-F-2-

MeO, H, E], [-2〇5: '4-F-3-MeO, H, E], [-206: 2-Cl-3-MeO, Η, E], [-207:2- Cl-4-MeO,H,E) , [-208:2-Cl-5-MeO,Η,E] r [-2Q9:2-C1-6-MeO,H,E],[-210:3 -Cl-2-MeO,H,E],[-211:3-Cl-4-iieO,H,E], [-212:3-Cl-5-Me〇,H,E], [-213 :4-Cl-2-MeO,H,E] , [-214:4-C1-3- 58 320202 200901876

MeO,H,E] , [-215:2-Me-3-MeO,Η,Ε], [-216:2-Me-4-MeO,H,E],[-217:2-Me-5 -MeO,H,E], [-218:2-Me-6-MeO,H,E], [-219:3-Me-2-MeO,H,E],[-220:3-Me- 4-MeO,H,E], [-221:3-Me-5-MeO,H,E], [-222:4-Me-2-MeO,H,E), [-223:4-Me -3-MeO,Η,Ε ] , [ -224:Η,4- F.,E] , C-225:4-F, 4-F,E] , [-226: 4-F, 4-F , Ζ], [-227:4-01,4-F, E], [-228:4-Cl,4-F,Z], [-229:4-Br,4-F,Ε], [ -230: 4-1,4-F, E], [-231: 4-Me, 4-F, E], [-232: 4-Me, 4-F, Ζ], [-233:4- Et,4-F,E], ( -234 :4-C3 Η7 ,4-F,E ] , [-235 : 4-(Me) 2 CH, 4-F, Ε], [- 236: 4- CF3,4-F,E] , [-237 : 4-CF3,4-F, Ζ], [-238 : 4-C2 F5 , 4-F, Ε], [-239:4-C3F7 ,4- F, E], [-240: 4-(CF3) 2 CF, 4-F, Ε], C-241: 4-(CF3)2CH, 4-F, E], C-242: 4-CHF2, 4-F,E] , [-243 : 4-CH2 F, 4-F, Ε], [-244:4-CF3CH2,4-F,E], [-245:4-MeO,4-F, Ε] , [-246:4-MeO,4-F,Z], [-247:4-EtO,4-F,E], [-248:-4-C3H7〇,4-F,E], [-249:4-(Me)2CHO,4-F,E], [-250:4-N02,4-F,E] r [-251:4-N02/4-F,Z], [- 252:3-F,4-F,E , [-253: 3-F, 4-F, Z], [-254: 3-Cl, 4-F, E], [-255: 3-Cl, 4-F, Z], [-256: 3-Br,4-F,E], [-257:3-1,4-F,e3,[-258:3-Me,4-F,E],[-259:3-Me,4- F,Z],[-260:3-Et,4-F,E],[-261:3-C3H7,4-F,E] f [-262:3-(Me)2CH,4-F, E] , [-263 : 3-CF3 v 4-F, E], [-264: 3-CF3, 4-F, Z], [-265 : 3-C2 F5,4-F, E], [ -266:3-C3F7,4-F:E], [-267:3-(CF3)2CF, 4-F,E], [-268: 3-(CF3) 2 CH, 4-F, E] , [-269:3-CHF2,4-F,E] , [-270:3-CHF2,4-F,Z], [-271:3-CH2 F, 4-F, E〇, [一272 :3-CH2F,4-F,Z], [1-2273: 3-CF3 CH2,4-F, E], [1274:3-Me〇,4-F,E], [1275: 3- MeO, 4 — F, Z] , [ -27§: 3-EtO, 4- F, E], [-277:3-C3H70,4-F, E], [-278:3-(Me)2CHO , 4-F, E], [-279: 3-N〇2,4-F, E], [-280:2-F,4-F,E], [-281:2-C1,4- F, E], [- 59 320202 200901876 282: 2-Br, 4-F, E], [-283: 2-I, 4-F, E], [-284: 2-Me, 4-F, E], [-285: 2-Et, 4-F, E], [-286: 2-C3H7, 4-F, E], [-287: 2-(Me)2CH, 4-F, E] , [-288 : 2-CF3, 4-F, E], [-289: 2-C2F5, 4-F, E] , [-290:2-C3F7,4-F,E], [-291:2-(CF3)2CF,4-F,E], [-292 : 2-(CF3 ) 2 CH, 4-F, E] , [-293:2-CHF2,4-F,E] , [-294:2-CH2F,4-F,E], [-295:2-CF3CH2,4-F,E], [- 296:2-MeO,4-F,E], [-297:2-EtO,4-F,E], [-298:2-C3H70, 4-F,E], [-299: 2-( Me) 2 CHO, 4-F, E], C -300:2- N〇2,4-F,E] , C-301:2,3-F2 ,4-F,E] , [-302 : 2,4-F2, 4-F, E], [-303:2,5-F2,4-F,E], C-304:2,6-F2,4-F,E], C-305 : 3, 4-F2 , 4- F, E] , [-306:3,4-F2,4-F,Z] , [-307 : 3,5-F2 , 4-F, E] , [- 308:3,5-F2,4-F,Z], [-309:2,3-Cl2,4-F,E], [-310:2,3-Cl2,.4-F,Z], [-311:2,4-C12,4-F,e], [-312:2,4-Cl2,4-F,Z], t-313:2,5-Cl2,4-F,E] , [-314:2,5-C12,4-F,Z], [-315:2,6-C12,4-F,E],.[-316:3,4-CI2,4-F, E] , [-317:3,5-CI2,4-F,E] , [-318:2,3-Br2,4-F,E],[-319:2,4-Br2,4-F , E], [-320:2,5-Br2,4-F,E], [-321:2,6-Br2,4-F,E], [-322:3,4-Br2;4- F, E), [-323:3,5-Br2,4-F,E], [-324:2,3-Me2,4-F,E], [-325:2,4-Me2, 4 -F, E], [-326:2,5-Me2,4-F,E], [-327:2,6-Me2,4-F,E] , (-328:3,4-Me2, 4-F, E], 〔 -329:3,5-Me2,4-F,E], [-330 : 2,3-Et2 , 4-F, E], [- 331:2,4-Et2,4-F,E], [-332:2,5-Et2,4-F,E), [-333:2,6-Et2,4-F,E], [-334:3,4-Et2,4-F,E] , '[-335:3,5-Et2,4-F,E], [-336:2,3-(CF3)2,4-F,E], [-337:2,4-(CF3) 2,4-F,E], [-338:2,5-(CF3)2,4-F,E], C-339:2,6-(CF3)2,4-F,E]; .-340:3,4-(CF3)2,4-F,E], [-341:3,5-(CF3)2,4-F,E], [ -342:2,3-(CHF2 2,4-F,E] , [-343:2,4-(CHF2)2,4-F,E] r [-344:2,5- 60 320202 200901876 (CHF2)2,4-F, E], [-345:2, 6-(CHF2>2,4-F, E 3 r [-346:3,4- (CHF2) 2,4-F,E ], [-347:3,5 -(CHF2 )2 ,4-F,E], [-348:2,3- (CH2F)2,4-F,E], [-349:2,4-(CH2 F)2 ,4-F , E ], C -350: 2,5- (CH2F) 2,4-F, E], [-351:2,6-(CH2F)2 ,4-F,E], [-352:3, 4-(CH2F)2,4-F,E], [-353:3,5-(CH2F)2r4-F,E], [-354:2,3-(MeO)2,4-F,E ], [-355:2,4-(MeO>2,4-F,E], C-356:2,5-(MeO)2,4-F,E], [-357:2,6- (MeO)2,4-F,E 3 , [-358:3,4- (MeO)2,4-F,E], [-359:3,5-(MeO)2,4-F,E ], C -360:2,3- (EtO>2 ,4-F, E], [-361:2 ,4-(EtO)2,4-F,E ], C -362:2,5- (EtO)2,4-F,E], [-363:2,6-(EtO)2,4- F, E ), [-364:3,4- (EtOh , 4-F, E], [-365:3,5- (EtO) 2,4-F,E] , [-366:2-Cl -3-F, 4-F, E], C-367: 2-Cl-4-F, 4-F, E], [-368: 2-C1-5-F, 4-F, E], [-369:2-Cl-6-F,4-F,E], [-370:3-Cl-2-F,4-F,E], [-371:3-C1-4-F, 4-F, E], [-372:3-Cl-5-F,4-F, E], [-373:4-C1-2-F, 4-F, E], [-374:4 -Cl-3-F,4-F,E], C-375:2-F-3-Me,4-F,E3, [-376:2-F-4-Me,4-F,E] , [-377:2-F-5-Me,4二F,E], [-378:2-F-6-Me,4-F,E], [-379:3-F-2-Me ,4-F,E] , {-380:3-F-4-Mef4-F, Έ ] , [-381:3-F-5-Me,4-F,E] , [-382:4- F-2-Me,4-F,E] , [-383:4-F-3-Me,4-F,E), [-384:2-Cl-3-Me,4-F,E] , [-385:2-Cl-4-Me,4-F,E], [-386:2-Cl-5-Me,4-F,E], [-387:2-Cl-6-Me , 4-F, E], [-388: 3-Cl-2-Me, 4-F, E], [-389: 3-Cl-4-Me, 4-F, E], [-390: 3-Cl-5-Me,4-F,E], [-391:4-Cl-2-Me,4-F,E], [-392:4-Cl-3-Me,4-F, E] , [-393:2-F-3-CF3,4-F,E], [-394:2-F-4-CF3,4-F,E],[-395:2-F-5 -CF3,4-F,E], [-396:2-F-6-CF3,4-F,E], [-397:3-F-2-CF3,4-F,E], (- 398:3- F-4-CF3,4-F,E] , [-399:3-F-5-CF3,4-F,E] , C-400:4-F-2- 61 320202 200901876 CF3,4-F , E], [ -401:4-F-3-CF3, 4-F, E), [-4 02 : 2-Cl-3-CF3, 4-F, E], [-4 03:2- Cl-4-CF3,4-F,E] ,[-404 :2-Cl-5-CF3 , 4-F, E], [-4 05:2-Cl-6-CF3,4-F,E ], [-406:3-Cl-2-CF3,4-F, E], [-407:3-CI-4-CF3,4-F,E], (-408:3-Cl-5- CF3,4-F,E], [-409:4-01-2-CF3,4-F,E], [-410:4-Cl-3-CF3,4-F,E), [-411 :2-Me-3-CF3,4-F,E], [-412:2-Me-4-CF3,4-F,E],[-413:2-Me-5-CF3,4-f , E], [-414 : 2-Me-6-CF3, 4-F, E], [-415 : 3-Me-2-CF3,4-F, E]. , [-416:3-

Me-4-CF3,4-F,E], [-417:3-Me-5-CF3,4-F,E], [-418:4-Me-2-CF3,4-F,E] , [-419:4-Me-3-CF3/4-F,E], [-420:2-F-3-MeO,4-F,E], [-421:2-F-4-MeO , 4-F, E], [-422: 2-F-5-MeO, 4-F, E], [-423: 2-F-6-MeO, 4-F, E], [-424: 3-F-2-MeO, 4-F, E], C*-425: 3-F-4-MeO, 4-F, E], [-426: 3-F-5-MeO, 4-F , E], [ -427 : 4-F-2-MeO, 4-F, E], [-428:4-F-3-MeO,4-F,E], [-429:2-Cl- 3-MeO,4-F,E], [-430:2-Cl-4-MeO,4-F,E], [-431:2-Cl-5-MeO,4-F,E], [ -432:2-

Cl-6-MeO,4-F,E], [-433:3-Cl-2-MeO,4-F,E], [-434:3-C1-4-

MeO,4-F,E], [-435:3-Cl-5-MeO,4-F,E], [-436:4-Cl-2-MeO,4-F,E], [-437 :4-Cl-3-MeO, 4-F,E] , [-438 :2-Me-3-MeO, 4-F, E], [-439:2-Me-4-MeO,4-F , E] , [-440: 2-Me-5-MeO, 4-F, E], [-441:2-

Me-6-MeO, '4-F, E], [-442 : 3-Me-2-MeO, 4-F, E], [ -443: 3-Me-'4-

MeO,4-F,E] , C-444 : 3-Me-5-MeO, 4-F,E] , [-445: 4-Me-2-MeO,4-F,E], [-446 :4-Me-3-MeO,4-F,E], [-447:H,4-Cl,E], [-448:4-Ff4-C1,E], C-449:4-F, 4-Cl,Z) f [-450:4-C1,4-C1,E], [-451:4-Cl,4-Cl,Z],[-452:4-Br,4-Cl,E ], [-453: 4-I, 4-Cl, E], [-454: 4-Me, 4-Cl, E] f [-455: 4-Me, 4-C1, Z], [-456 :4-Et,4-Cl,E], [-457:4-C3H7,4-Cl,E] , [-458:4-(Me)2CH,4-Cl, E] , [-459:4 - 62 320202 200901876 CF3,4-C1,E]r[-460:4-CF3,4-Cl,Z], [-4 61: 4-C2 F5,4-C1, E], [-462:4 -C3F7,4-Cl,E ] , [-463 : 4-(CF3 ) 2 CF, 4-C1, E ] , [-464 :4-(CF3 )2CH, 4-Cl,E], [-465 :4-CHF2,4-Cl,E], C-466:4-CH2F, 4-C1,E],C-467:4-CF3CH2,4-ClfE], [-468:4-MeO, 4- C1, E ], [- 469: 4-MeO, 4-Cl, Z], [-470: 4-EtO, 4-C1, E], C-471: 4-C3H70, 4-Cl, E], [-472:4-(Me)2CHO,4-Cl,E], [-473:4-N02,4-Cl.,E], [-474:4-N〇2,4-Cl,Z] , [-475:3-F,4-C1,E], [-476:3-F,4-C1,Z], [-477:3-Cl,4-Cl,E],[-478: 3-C1,4-Cl,Z], [ -479:3-Br,4-Cl,E], [-480:3-I,4-Cl,E],[-481:3-Me,4 -Cl,E],[-482:3- Me, 4-Cl, Z], [-483: 3-Et, 4-Cl, E], [-484: 3-C3H7, 4-Cl, E], [-485: 3-(Me) 2CH, 4-Cl,E] , [-486:3-CF3,4-Cl,E] , [-487:3-CF3,4-C1,Z],[-488:3-C2F5, 4-Cl,E ], [-489 : 3-C3 F7 , 4-C1, E], [- 490:3-(CF3)2CF,4-Cl,E] , [-491:3-(CF3)2CH,4-C1 , E], [-492:3-CHF2,4-C1,E], [-493:3-CHF2,4-Cl,Z], [-494:3-CH2F,4-Cl,E], C -495:3-CH2F, 4-Cl,Z], C-496 : 3-CF3 CH2 , 4-C1, E ] , [-497:3-

MeO, 4-Cl, E], [-498: 3-MeO, 4-Cl, Z], [-499: 3-EtO, 4-Cl, E]-·, [-500:3-C3H7〇, 4-C1,E] , [-501: 3-(Me) 2 CHO, 4 - Cl, E], [-502:3-N02,4-C1,E], [-503:2-F,4 -C1,E], [-504:2-C1,4-C1,E], [-505:2-Br,4-Cl,E], [-506:2-1,4-C1,EJ, [-507:2-Me,4-C1,E]' r [-508:2-Et,4-Cl,E], [-509 :2-C3 H·? , 4-C1, E], C -510:2-(Me)2CH,4-Cl,E], [-511:2-CF3,4-Cl,E], [-512:2-C2F5,4-C1,E], C-513 :2-C3F7,4-Cl,E] , [-514:2-(CF3)2CFr4-C1,E], [-515:2-(CF3)2CH,4-Cl,E], [-516: 2-CHF2,4-C1,E],.[-517:2-CH2F,4-C1,E], C-518:2-CF3 CH2, 4-Cl,E],[-519: 2-Me 〇,4-C1, E], [-520:2-Et〇,4-Cl,E], C-521:2-C3H70,4-C1,E], C-522:2- 63 320202 200901876 ( Me) 2CHO, 4-Cl, E], [-523: 2-N02, 4-C1, E], [ -524:2,3-F2,4-

Cl, E], [-525: 2,4-F2,4-Cl, E], [-526:2,5-F2,4-Cl,E], [-527:2,6-F2,4 -Cl, E], [-528:3,4-F2,4-Cl,E], [-529:3,4-F2,4-Cl,Z], [-530:3,5-F2, 4-Cl, E], [-531:3,5-F2,4-Cl,Z], [-532:2,3-Cl2,4-Cl,E],[-533:2,3-Cl2 , 4-Cl, Z], [-534: 2,4-C12,4-C1,E], [-535:2,4-Cl2,4-Cl,Z],[-536:2,5- Cl2,.4-Cl,E], [-537:2,5-Cl2,4-Cl,Z], [-538:2,6-Cl2,4-C1,E], [-539:3, 4-C12,4-C1,E] , [-540:3,5-Cl2,4-Cl,E], [-541:2,3-Br2,4-C1,E], [-542:2 , 4-Br2,4-Cl, E], [-543:2,5-Br2,4-C1,E], [-544:2,6-Br2,4-C1,E], [-545: 3,4-Br2,4-Cl,E], [-546:3,5-Br2,4-C1,E], [-547:2,3-Me2,4-Cl,E], C-548 :2,4-Me2,4-Cl,E] ,' [-549:2,5-Me2,4-C1,E] , [-550:2,6-Me2,4-ClfE] , [-551 :3,4-Me2,4-C1,E], [-552:3,5-Me2,4-Cl,E], [-553:2,3-Et2,4-Cl,E], [- 554:2,4-Et2,4-C1,E], [-555:2,5-Et2,4-Cl,E], [-556:2,6-Et2,4-Cl,E], [ -557:3,4-Et2,4-Cl,E], [-558:3,5-Et2,4-Cl,E], [-559:2,3-(CF3)2,4-C1, E], C -560: 2,4-(CF3)2,4-Cl,E ], [-561:2,5-(CF3)2,4-C1,E], [-562:2,6 -( CF3 >2,4-Cl,E], [-563:3,4-(CF3)2,4-C1,E], [-564:3,5-(CF3)2,4-Cl,E ], C -565:2,3- (CHF2)2,4-C1,E], [-566:2,4-(CHF2)2,4-ClrE], [-567:2,5- (CHF2 2,4-C1,E], [-568:2,6-(CHF2)2,4-Cl,E], C-569:3,4-(CHF2)2,4-C1,E], [-570:3,5-(CHF2)2,4-Cl,E], [-571:2,3-(CH2F)2,4-C1,.E]., [-572:2,4- (CH2F)2,4-Cl,E], [-573:2,5-(CH2F)2,4-C1,E], [-574:2,6-(CH2F)2,4-C1/E ], [.-575:3,4-(CH2F)2,4-C1,E], [-576:3,5-(CH2F)2,4-Cl,E], [-577:2,3 - (MeO)2,4-Cl,E], [-578:2,4-(MeO)2,4-Cl,E ], C -579:2,5- 64 320202 200901876 (MeO)2,4 -Cl,E 〕 (MeO)2,4-Cl,E] (EtO)2,4-Cl,E] (EtO)2,4-Cl,E] (EtO)2,4-Cl,E] [ -580:2,6-(MeO)2,4-Cl,E], [-581:3,4. [-582:3,5-(MeO)2,4-Cl,E],[-583 :2,3-[-584:2,4-(EtO)2,4-Cl,E],[-585:2,5-[-586:2,6-(Et〇)2,4-Cl , E 〕 , [ -587:3,4-[-588:3,5-(EtO)2 r4-Cl,E], [-589:2-C1-3-F,4-C1,E], [-590:2-Cl-4-F,4-Cl,E], [-591:2-C1-5-F,4-C1,E], C-592:2-Cl-6-F, 4-Cl,E] , [-593:3-C1-2 -F,4-C1,E) , [-594:3- . > .

Cl-4-F,4-Cl,E], [-595:3-Cl-5-F,4-Cl,E], [-596:4-C1-2-F,4-C1,E] λ C-597: 4-Cl-3-F, 4-Cl, E], [-598: 2-F-3-Me, 4-C1, E], (-599: 2-F-4-Me , 4-Cl, E], [-600: 2-F-5-Me, 4-C1, E], [-601: 2-F-6-Me, 4-C1, E], [-602: 3-F-2-Me,4-Cl,E], C-603:3-F-4-Me,4-C1,E], [-604:3-F-5-Me,4-Cl, E] , [-605:4-F-2-Me,4-Cl,E], [-606:4-F-3-Me,4-Cl,E], [-607:2-Cl-3 -Me,4-C1,E] , [-608:2-Cl-4-Me,4-Cl,E3, [-609:2-Cl-5-Me,4-C1,E] r [-610 :2-Cl-6-Me,4-ClfE] , [-611:3-Cl-2-Me,4~C1,E] , [-612 : 3-Cl-4-Me,4-C1,E ), [-613:3-Cl-5-Me,4-Cl,E], C-614: 4-Cl-2-Me, 4-C1, E], [-: 615:4-Cl-3 -Me,4-Cl,E] ,[-616:2-F-3-CF3,4-C1, E],C-617:2-F-4-CF3 Λ 4-C1, E] , [- 618 : 2-F-5-CF3 , 4-C1, E] , [t-619 :2-F-6-CF3,4-C1,E] , C-620:3-F-2-CF3,4 -Cl,E] , [-621:3-F-4-CF3,4-C1,E> , [-622:3-F-5-CF3,4-Cl,E]' , [-623:4 -F-2-CF3,4-C1,E], [- 624:4-F-3-CF3,4-Cl,E], [-625:2-Cl-3-CF3,4-Cl,E ], [-626:2-Cl-4-CF3,4-Cl,E] ', [-627:2-Cl-5-CF3,4-Cl,E], [-628:2-G1-6 -CF 3,4-C1,E] , C-629:3-Cl-2-CF3r4-Cl,E], [-630:3-Cl-4-CF3,4-C1,E], [-631:3 -Cl-5-CF3,4-Cl,E], [-632:4-Cl-2-CF3,4-Cl,E], C-633:4-Cl-3-CF3,4-Cl,E ], [-634:2-Me-3-CF3,4-C1,E],[- 65 320202 200901876 635:2-Me-4-CF3,4-Cl,E], [-636:2-Me -5-CF3,4-C1,E] , [-637:2-Me-6-CF3,4_C1,E] t [-638:3~Ms—2-CF3, 4~C1,E] t C- 639: 3-Me-4-CF3,4-C1,E], [-640:3-Me-5-CF3,4-Cl,E], C-641:4-Me-2-CF3,4- C1,E], [-642:4-Me-3-CF3,4-Cl,E], [-643:2-F-3-MeO,4-Cl,E], [-644:2-F -4-MeO,4-Cl,E ] , [ -645:2-F-5-MeO,4-C1,E], [- 646:2-F-6-MeO,4-Cl,E], [-647:3-F-2-MeO,4-C1,E], [-648:3-F-4-MeO,4-Cl,E],[-649 : 3-F-5-Me〇 , 4-C1, E], [-650: 4-F-2-MeO, 4-C1, E], [-651: 4-F-3-MeO, 4-Cl, E], [-652: 2-Cl-3-MeO,4-Cl,E], C-653:2-Cl-4-MeO,4-Cl,E], [-654:2-Cl-5-MeO,4-Cl, E ] , C- 655: 2-Cl-6-MeO, 4-Cl, E], [-656: 3-Cl-2-MeO, 4-Cl, E], [-657:3-Cl-4 -MeO, 4-Cl, E], [-658 : 3-Cl-5-MeO, 4-Cl, E], [-1559: 4-C1-2-MeO, 4-Cl, E], [- 660: 4-Cl-3-MeO, 4-Cl, E], [-661: 2-Me-3-MeO, 4-C 1,E] , [-662:2-Me-4-MeO,4-Cl,E], [-663:2-Me-5-MeO,4-Cl,E], C-664:2-Me -6-MeO, 4-Cl, E 3 , [-665:3-Me-2-MeO, 4-C1, E], [- 666:3-Me-4-MeO, 4-Cl, E), [-667:3-Me-5-MeO,4-C1,E], [-668:4-Me-2-MeO, 4-Cl,E], [-669: 4-Me-3-MeO, 4-C1·, E〕r [ -670:H, 4-CF3,E], [-671:4-F,4-CF3,E], [-672:4-F,4-CF3,Z] , [-673: 4-Cl, 4-CF3, E], [-674: 4-Cl, 4-CF3., Z], [-675: 4-Br, 4-CF3, E], [-676 :4-1,4-CF3,E], [-677:4-Me,4-CF3,E], [-678:4-Me,4-CF3,Z],[-679:4-Et, 4-CF3, E], [-680: 4-C3H7, 4-CF3, E], [-681: 4-(Me)2CH/4-CF3, E], [-682: 4-CF3,4- CF3 , E ] , [ -683:4- CF3,4-CF3,Z ] , '[ -684:4-C2F5/4-CF3,E ] , [ -685 : 4-C3 F7,4- CF3,E ], [-686:4-(CF3)2CFf4-CF3,E], [-687: 4-(CF3) 2 CH, 4-CF3,E], C-688:4-CHF2,4-CF3,E r [-689: 4-CH2 F, 4-CF3, E], [- 690:4-CF3 CH2,4-CF3,E), C-691:4-MeO,4-CF3,E], [ -692:4- 66 320202 200901876

MeO,4-CF3,Z] , [ -693:4-EtO, 4-CF3 ,E ] , C -694 : 4-C3 H7 0, 4-CF3,E], [-695:4-(Me) 2CHO, 4-CF3, E], [-696 : 4-N02,4-CF3, [-697:4-N02,4-CF3,Z], [ -698 :3-F, 4-CF3 ,E ] , [ -699:3-F, 4-CF3,Z] , [-700:3-d, 4-CF3 ,E) , [-701:3-Clf 4-CF3,z) , [-702:3 -Br,4-CF3,E], C-703:3-1,4-CF3,E], [-704 : 3-Me,4-CF3,E],[-7〇5:3-Me, 4-CF3,Z], [-706:3-Et,4-CF3,E], C-707:3-C3H7,4-CF3,E],[-708:3-(Me)2CH,4- CF3, E], [-709: 3-CF3, 4-CF3, E], [-710: 3-CF3, 4-CF3, Z], [-711: 3-C2F5r4-CF3, E], [- 712: 3-C3F7,4-CF3,E], [-713:3-(CF3)2CF,4-CF3,E], [-714:3-(CF3) 2 CH, 4-CF3,E], [-715:3-CHF2,4-CF3,E], X-716:3-CHF2,4-CF3,Z], [-717:3-CH2F,4-CF3,E], [-718:3 -CH2F,4-CF3,Z]; [-719:3-CF3CH2,4-CF3,E], [-720:3-MeO,4-CF3,E],[ -721:3-MeO,4- CF3,Z], [-722:3-EtO,4-CF3,E], [-723:3-C3H70,4-CF3,E], [-724:3-(Me)2CHO,4-CF3, E ] , [-725:3-N02,4-CF3,E], C-726:2-F,4-CF3,E], [-727:2-Cl,4-CF3,E],[- 728:2-Br,4-CF3,E] [-729:2-I,4-CF3,E], [-730:2-Me,4-CF3,E], [-731:2-Et,4-CF3,E], C-732:2 -C3H7,4-CF3,E) , [-733 : 2-(Me) 2 CH, 4-CF3 , E), [-734:2-CF3,4-CF3 ,E ] , [-735 :2- C2 F5,4-CF3 , E ] , [-736 :2- C3Ft,4-CF3,E ] , [ -737:2-(CF3)2CF,4-CF3.,E] , C -738:2- (CF3)2CH,4-CF3,E], C-739:2-CHF2,4-CF3,E], C-740:2-CH2 F, 4-CF3,E],[-741:2-CF3CH2 , 4-CF3, E], [-742: 2-MeO, 4-CF3, E], [-743:2-Et〇,4-CF3,E], C-744:2-C3H70,4-CF3 , E ] , C -745:2- (Me)2CHO,4-CF3,E], [-746:2-N02,4-CF3,E],[-747;2,3-F2,4-CF3 , E], [-748: 2,4-F2,4-CF3,E], [-r49:2,5-F2,4-CF3,E], [-750:2, 6-F2, 4- CF3 , E ] , [-751:3,4-F2 , 4-CF3 ,E ] , [-752 :3,4- 67 320202 200901876 F2,4-CF3,Z] , [-753:3,5- F2,4-CF3,E] , [-754 : 3,5-F2,4-CF3 , Z], [-755:2,3-Cl2,4-CF3,E], [-756:2,3 -Cl2,4-CF3,Z],[- 757:2,4-Cl2,4-CF3,E), [-758:2,4-Cl2,4-CF3,Z],[-759:2, 5-

Cl2/4-CF3,E] , [-760:2,5-Cl2,4-CF3,Z ] , [-761: 2, 6-Cl2 , 4-CF3,E] , [-762:3, 4 -Cl2,4-CF3,E], [-763: 3,5-Cl2, 4-CF3, E), [-764:2,3-Br2,4-CF3,E], C-765:2, 4-Br2, 4-CF3, EJ, [-766:2,5-

Br2,4-CF3,E], [-767:2,6-Br2r4-CF3,E], C-768:3,4-Br2, 4-cf3,e] r [-769:3,5-Br2 , 4-CF3, E], [-770 : 2,3-Me2,4-CF3,E], [- 771:2, 4-Me2,4-CF3 ,E] , C-772 :2,5- Me2,4-CF3,E ] , [-773:2, 6- Me2 / 4-^ cf3 ,E], [-774 :3, 4-Me2,4-CF3 ,E 3 , [-775:3, 5-Μθ2,4-CF3 ,E] r [-776:2,3-Et2,4-CF3,E] , [-777 :2,4-Et2 , 4,CF3 ,E], [- 778:2 , 5-Et2,4-CF3,E], [-779:2,6-Et2,, I-CF3,E], [-780:3,4- Et2,4-CF3,E], [-781 :3,5-Et2,4-CF3,E],C-782:2,3-(CF3)2/4-CF3, E] r [-783:2,4-(CF3)2,4-CF3 , E], [-784:2,5-(CF3)2,4-CF3,E] r [-785:2,6-(CF3 )2 , 4-CF3 ,E ], [-786:3, 4-(CF3)2,4-CF3,E] t [-787:3,5-(CF3)2,4-CF3,E], [-788:2,3- (CHF2)2,4- cf3 ,e] f [-789:2,4-(CHF2)2,4-CF3,E], [-790:2,5-(CHF2)2,4-CF3, E] r [-791:2, 6-(CHF2)2,4-CF3,E], [-792:3,4-(CHF2)2,4-CF3,E] f [-793:3, 5-(CHF2)2,4-CF3 ,eD , [-794:2,3-(CH2F)2,4-CF3 ,E] r [-795:2,4-(CH2F)2,4-CF3,E], [-796:2,5 -(CH2F)2,4- cf3,e] r [-•7 97:2, 6-(CH2F)2,4-CF3,E], -798:3, 4-(CH2F)2,4- cf3,e] 9 C -799:3,5- (CH2 F)2,4-CF3 ,E ], [-800:2,3-(MeO 2,4-CF3,E] t [-801:2,4-(MeO)2,4-CF3,E], [-802:2,5T(MeO)2,4-CF3, E] t [ -803:2., 6-(MeO) 2, 4-CF3,E ], [-804:3,4-(MeO)2,4-CF3,E] r [-805:3,5-(MeO 〉2r4-CF3, E], [-806:2,3-(Et〇j2,4- 68 320202 200901876 CF3,E], [-807:2,4-(EtO)2,4-CF3,E] , [-808:2,5-(EtO)2,4-CF3,E] , [ -809:2,6-(EtO)2,4-CF3,E ] , [-810 : 3,4-( EtO) 2 , 4-CF3,E ] , [ -811:3,5-(EtO)2,4-CF3,E], C-812:2-Cl-3-F,4-CF3,E], [-813: 2-Cl-4-F, 4-CF3, E], [-814: 2-Cl-5-F, 4-CF3, E], [-815: 2-Cl-6-F, 4-CF3,E], [-816:3-C1-2-F,4-CF3,E],[- 817:3-Cl-4-F,4-CF3,E], C-818:3 -C1-5-F,4-CF3,E] , [-819:4- C1-2-F, 4-CF3 ,E ] , [-820:4-Cl-3-F,4-CF3,E 〕, 〔-821:2-F-3-

Me, 4-CF3, E], C-822: 2-F-4-Me, 4-CF3, E], [-823: 2-F-5-Me, 4-CF3, E], [-824 :2-F-6-Me,4-CF3,E] , [-825:3-F-2-Me,4-CF3,E], [-826:3-F-4-Me,4-CF3 , E 〕 , C -827: 3-F-5-Me, 4-CF3, E ), [- 828: 4-F-2-Me, 4-CF3, E] , [-829:4-F- 3-Me,4-CF3,E]·,[-830:2-C-836:3-Cl-5-Me,4-[-838:4-Cl-3-Me,4-[-840: 2-F—4-CF3,4 — [—842 :2-F—6—CF3 , 4-[—844 : 3-F-4-CF3 , 4-[-846:4-F-2-CF3, 4-[-848:2-Cl—3-CF3,4 — [-850:2-Cl-5-CF3,4-[-852:3—Cl~2—CF3,4—[-854:3- C1-5—CF3, A — [-856:4—Cl-3-CF3 t A — (-858:2-Me-4-CF3,4-

Cl-3-Me,4-CF3,E〇, [-831:2-C1-4-M6,4-CF3,E], [-832:2-C1-5-Me,4-CF3,E] , [-833:2-Cl-6-Me,4-CF3,E], C-834:3-Cl-2-Me,4-CF3,E], [-835:3-Cl-4-Me ,4-CF3,E]CF3,E], [-837:4-Cl-2-Me,4-CF3,E], CF3,E],[ -839:2-F-3-CF3,4- CF3, E), CF3, E], [-841: 2-F-5-CF3, 4-CF3, E], CF3, E], [-843:3-F-2-CF3, 4-CF3, E ], CF3, E], [ -845:3-F-5-CF3 , 4-CF3 ,E ], CF3 , E ] , [ -847: 4-F-3-CF3,4-CF3,E] , CF3, E] , [ -849:2-Cl-4-CF3 ,4-CF3 ,E ], CF3,E]., [ -851:2-Cl-6-CF3 , 4-CF3 ,E ], CF3,E], [-853:3-Cl-4-CF3, 4-CF3,E], CF3,E], [-855:4-Cl-2-CF3,4-CF3,E], CF3, E], [ -857 : 2-Me-3-CF3 , 4-CF3 , E], 69 320202 200901876 cf3,e], [-85 9 :2-Me-5-CF3,4-CF3/E]r [ ~860 :2-Me-6-CF3 f 4 — cf3,e], [-8 61: Me-2-CF3,4-CF3 ,E]f [-862:3-Me-4-CF3,4 - cf3,e], [-8 63:3-Me-5-CF3,4-CF3,E], [-864 :4-Me-2-CF3,4-CF3,E], [ -865:4 -Me-3-CF3,4-CF3,E], C-866:2-F-3-MeO,4-CF3,E], [-867:2-F-4-MeO,4-CF3,E 〕 , C -868:2-F-5 -MeO,4-CF3,E], [-869:2-F-6-MeO,4-CF3,E], [-870:3-F-2-Me〇,4-CF3,E], [ -871:3-F-4-MeO,4-CF3,E], ( -872:3-F-5-MeO,4-CF3,E), [-873:4-F-2-MeO,4 -CF3,E], [-874:4-F-3-MeO,4-cf3,e], [-875:2-Cl-3-MeO,4-CF3,E], [-876:2- Cl-4-MeO,4- cf3,e], [-877:2-Cl-5-MeO,4-CF3,E], [ -878 :2-Cl-6-MeO,4- cf3,e] , [-879:3-Cl-2-MeO,4-CF3,E ] , [-880:3-Cl-4-MeO,4-CF3,E], [-881:3-Cl-5-MeO , 4-CF3, E], [ -882:4-Cl-2-MeO,4- cf3,e], [-883:4-Cl-3-MeO,4-CF3,E], [-884: 2-Me-3-MeO,4-CF3,E]Λ [-885:2-Me-4-MeO,4-CF3,E], C-886:2-Me-5-MeO,4-C. F3, E], C-887: 2-Me-6-MeO, 4-CF3, E], C-888: 3-Me-2-MeO, 4- cf3, e], [-889: 3-Me -4-MeO,4-CF3,E], [-890:3-Me-5-MeOf4-CF3,E], [-891:4-Me-2-MeO,4-CF3,E], [- 892: 4-Me-3-MeO, 4-CF3, E], [-893: H, 4-MeO, E], [-8 94 : 4-F, 4-MeO, E], [-895: 4-F, 4-MeO,Z], [-896:4-Cl,4-MeO,E], [-897:4-Cl,4-MeO,Z], [-898:4-Br,4 -MeO,E],[-899:4-1,4-MeO,E], [-900:4-Me f 4-MeO,E],[-901:4-Me,4-MeO,Z ] , [-902:4-Et,4-MeO,E ] f C-903:4-C3H7,4-

MeO,E] , [-904:4-'(Me)2CH,4-MeO,E] , [-905:4-CF3 , 4-MeO, E],[-906:4-CF3,4-MeO , Z], [-907 : 4-C2 Fs r 4-MeO, E], C-908: 4-C3F7, 4-MeO, E], [-909:4-(CF3)2CF, 4-MeO, E ] , C -910:4- (CF3 )2CH, 4-

MeO, E], [-911:4-CHF2,4-MeO,E], [-912:4-CH2 Ff 4-MeO,E], [- 70 320202 200901876 913:4-CF3CH2,4-MeO, E 3 , [ -914:4-MeO,4-MeO,E], [ -915:4-

Me〇,4-MeO,Z], [-916:4-EtO, 4-MeO,E], [ -917:4-C3H70,4-

MeO, E], [-918 : 4- (Me)2 CHO,4-MeO,E] , [-919:4-N02,4-MeO,E], [-920:4-NOZ,4-MeO ,Z ] , [-921:3-F,4-MeO,E],[ -922:3-F,4-

MeO,Z], [-923:3-Cl,4-MeO,E], [-924:3-C1,4-MeO,Z], [-925:3-Br,4-MeO,E], [-926: 3-I, 4-MeO, E], [-927: 3-Me, 4-MeO., E], [-928: 3-Me, 4-MeO, Z], [-929: 3-Et,4-MeO,E],[ -930:3-C3H7,4-

MeO, E] , [-931: 3-(Me) 2CH, 4-MeO, E], [-932: 3-CF3, 4-MeO, E], [-933: 3-CF3, 4-MeO, Z] ., [-934 : 3-C2 F5,4-MeO, E], [-935:3-C3 F-, ,4-MeO,E ] , C -936:3- (CF3 ).2 CF , 4-MeO, E ] , [-937 : 3-(CF3 ) 2 CH, 4-

MeO, E], [-938:3-CHF2,4-MeO,E], [-939:3-CHF2,4-MeO,Z], [-940:3-CH2F,4-MeO,E], [-941:3-CH2F,4-MeO,Z], [-942:3-CF3CH2,4-MeO,E], [-943:3-MeO,4-MeO,E], [-944:3 -MeO,4-

MeO,Z], [-945:3-EtO,4-MeO,E], [-946:3-C3H70,4-MeO,E],[-947:3-(Me)2 CHO,4-MeO , E ] , [-948 :3-N02,4-MeO,E ] , [-949:2-F,4-MeO,E) , [-950:2-Cl,4-MeO,E], [ -951: 2-Br, 4-MeO, E), [-952: 2-1,4-MeO, E], [-953: 2-Me, 4-MeO, E] [ -954:2-Et , 4-

MeO,E] , [-955:2-C3H7,4-MeO,E] , [-956: 2-(Me)2CH,4-MeO,E], [-957:2-CF3,4-MeO, E ] , [-958 : 2-C2 F5,4-MeO, E ] , [-959:2- C3 F7 ,4-MeO,E 〇, [ -960:2-(CF3 ) 2CF, 4-MeO, E], [-961:2-(CF3)2CH,4-MeO,E], [-962:2-CHF2,4-MeO, E), [-963:2-CH2F,4-MeO,E] , C-964: 2-CF3CH2, 4-MeO, E], [-965: 2-MeO, 4-MeO, E], [-966: 2-EtO, 4-MeO, E], [-967: 2-C3H70, 4-MeO, E],. [-968:2-(Me)2CHO,4-MeO,E], [-969:2-NOz,4-MeO,E3, C-970:2, 3-F2,4-

MeO, E], [-971:2,4-F2,4-MeO,E], [-972:2,5-F2,4-MeO,E], [- 71 320202 200901876 973:2,6- F2,4-MeO,E ] , C -974 : 3, 4-F2 , 4-MeO, E ] , [-975:3,4-F2,4-MeO,Z], [-976:3,5 -F2,4-MeO,E], '[-977 :3, 5-F2,4-MeO,Z] [-978:2,3-Cl2,4-MeO,E], [-979:2, 3-Cl2,4-MeO,Z],[- 980:2,4-Cl2,4-MeOfE], [-981:2r4-Cl2,4-MeO,Z3, [-982:2,5-

Cl2 , 4-MeO,E ] , [ -983:2,5-Cl2,4-MeO,Z], [ -984:2,6-Cl2,4-

MeO, E], [-985:3,4-Cl2,4-MeO,E], [-986:3,5-Cl2,4-Me9,E], [-987:2,3-Br2,4 -MeO, E], [-988: 2,4-Br2,4-MeO, E], [-989:2,5-Br2,4-MeO,E], [-990:2,6-Br2, 4-MeO, E ) , [-991: 3,4-Br2 , 4-

MeO, E] , [-992:3,5-Br2,4-MeO,E] , [-993:2,3-Me2 , 4-MeO,E) , C-994 :2,4-Μβ2 , 4 -MeO,E3 ., C-995 :2,5-Μθ2 , 4-MeO,E!) , [-996:2,6-

Me2,4-MeO,E], [-997 : 3,4-Me2,4-MeO, E ] , [-998*: 3, 5-Me2 , 4-

MeO, E], [-999:2,3-Et2,4-MeO,E], [-1000:2,4-Et2,4-MeO,E], [-1001:2,5-Et2,4 -MeO,E 〕 , [ -1002:2,6-Et2,4-MeO,E],[- 1003:3,4-Et2,4-MeO,E], [ -1004:3,5-Et2, 4-MeO,E ],[- 1005:2,3-(CF3)2,4-MeO,E], [-1006:2,4-(CF3)2,4-MeO,E], [-1007 :2,5-(CF3)2,4-MeO,E],[-1008:2,6-(CF3)2,4-MeO,E], [-1009:3,4-(CF3)2, 4-MeO/E) , Cl〇l〇: 3,5-(CF3)2,4-MeO,Έ],[-1011:2,3-(CHF2)2,4-MeO,E],[- 1012:2,4-(CHF2)2,4-MeO,E],[-1013:2,5-(CHF2)2,4-MeO,E], [-1014:2,6-(CHF2)2 , 4-MeO, E], [_ 1015:3,4-(CHF2) 2,4-MeO,E] , [-1016:3,5-(CHF2)2 , 4-MeO,E],[- 1017:2,3-(CH2F)2,4-MeO,E], [-1018:2,4-(CH2F)2,4-MeO,E],[-1019:2,5-(CH2F)2 , .4-MeO, E], [-l〇20:2,6-(CH2F)2,4-MeO,E], [-1021:3/4-(CH2F)2,4-MeOrE], [ -1022 : 3, 5-(CH2 F) 2 , 4-Me〇, E], [-1023:2,3-(MeO)2,4-MeO,E], [-1024:2Λ4-(MeO) 2,4-MeO,E],[-1025:2,5-(MeO)2,4-MeO,E], [-1026:2,6-(MeO)2,4-MeO,E], - 72 320202 200901876 1027:3,4-(MeO)2,4-Me〇,E], 1029:2,3-(EtO)2,4-M eO,E], 1031:2,5-(EtO)2,4-MeO,E], 1033:3,4-(EtO)2,4-MeO,E], 1035:2-Cl-3-F , 4-MeO, E ], 1037: 2-Cl-5-F, 4-MeO, E ], 1039: 3-Cl-2-F, 4-MeO, E ], 1041: 3-Cl-5- F,4-MeO,E], 1043:4-Cl-3-F,4-MeO,E], 1045:2-F-4-Me,4-MeO,E], 1047:2-F-6 -Me,4-MeO,E], 1049:3-F-4-Me,4-MeO,E], 1051:4-F-2-Me,4-MeO,E], 1053:2-Cl- 3-Me,4-MeO,E ], 1055:2-Cl-5-Me,4-MeO,E], 1057:3-Cl-2-Me,4-MeO,E ], 1059:3-Cl -5-Me,4-MeO,E], 1061:4-Cl-3-Me,4-MeO,E], 1063:2-F-4-CF3,4-MeO,E], 1065:2- F-6-CF3 f 4-MeO, E ], 1067:3-F-4-CF3 , 4-MeO,E ], 1069:4-F-2-CF3,4-MeO,E], 1071:2 -Cl-3-CF3,4-MeO,E], 1073:2-Cl-5-CF3,4-MeO,E], 1075:3-Cl-2-CF3,4-MeO,E], 〔- 1028:3,5-(Me〇)2,4-MeO,E],[-[-1030:2,4-(EtO)2,4-MeO,E],[-[-1032:2,6 -(Et〇)2,4-MeO,E],[-[-1034:3,5-(EtO)2,4-MeO,E], [-[-1036:2-Cl-4-F, 4-MeO, E], [-[-1038:2-Cl-6-F>4-MeO, E·], [-C-1040:3-Cl-4-F,4-MeO,E], [_ [-1042: 4-Cl-2-F, 4-MeO, E], [-[-1044:2-F-3-Me,4-MeO,E],[-[-1046:2- F-5-Me,4-MeO,E ].,[-C -10 48: 3-F-2-Me, 4-MeO, E], C - [-1050: 3-F-5-Me, 4-MeO, E], [-[-1052:4-F-3- Me, 4-MeO, E 3 , C - [-1054: 2-Cl-4-Me, 4-MeO, E], [-[-1056: 2-Cl-6-Me, 4-MeO, E] , [-[-1058:3-Cl-4-Me,4-MeO,E 3 ,[- [-1060:4-Cl-2-Me, 4-MeO, E 3 ,[- [-1062:2 -F-3-CF3,4-MeO,E],[-[-1064:2-F-5-CF3,4-Me〇,E],[-[-1066:3-F-2-CF3r4- MeO, E], [-[-1068:3-F-5-CF3,4-MeO,E], [-[-1070:4-F-3-CF3,4-MeO,E), C - [ -1072: 2-Cl-4-CF3, 4-Me.O, E], [-[-1074:2-Cl-6-CF3,4-MeO,E],[-[-1076:3-Cl -4-CF3,4-MeO,E],[- 73 320202 [-1114:4-Me-2-MeO,4-MeO,E 3 ,[-1115:4-Me-3-MeO,4-MeO , E], [-1116:H,4-(Me)3CO,E], [-1117:4-F,4-(Me)3CO,E], [-1118 : 4-F, 4-(Me ) 3 CO, Z ] , [-1119:4-01,4-(Me)3CO,E ) , C -1120:4-C1,4-(Me)3C〇,Z ] , [ -1121:4- Br,4-(Me)3CO,E], [-1122:4-1,4-(Me)3CO,E] r [ -1123:4-Me,4-(Me)3CO,E ] , C - 1124: 4-Me,4-(Me)3〇〇rZ ] , C -1125:4-Et,4- 200901876 1077:3-Cl-5-CF3,4-MeO,E] 1079:4-Cl- 3-CF3,4-MeO,E] 1081:2-Me-4-CF3,4-MeO,E] 1083:2-Me-6-CF3,4-MeO,E] 1085 :3-Me-4-CF3,4-MeO,E) 1087:4-Me-2-CF3,4-MeO,E] 1089:2-F-3-MeO,4-MeO,E ] 1091:2 -F-5-MeO,4-MeO,E] 1093:3-F-2-MeOf 4-MeO,E) 1095:3-F-5-MeO,4-MeO,E ] 1097:4-F- 3-MeO,4-MeO,E] 1099:2-Cl-4-MeO,4-MeO,E] 1101:2-Cl-6-MeO,4-MeO,E] 1103:3-Cl-4- MeO, 4-MeO, E] 1105: 4-Cl-2-MeO, 4-MeO, E] 1107: 2-Me-3-MeO, 4-MeO, E] 1109: 2-Me-5-MeO, 4-MeO,E] 1111:3-Me-2-MeO,4-MeO,E] 1113:3-Me-5-MeO,4-MeO,E] C-107 8 :4-C1-2-CF3 , 4-MeO, E ], [-[-1080:2-Me-3-CF3,4-MeO,E ), [-[-1082:2-Me-5-CF3,4-MeO,E ], [-[-1084:3-Me-2-CF3,4-MeO,E] f [-[-1086:3-Me-5-CF3,4-MeO,E],[-[-1088:4- Me-3-CF3,4-MeO,.E],[-[-1090:2-F-4-MeO,4-MeO,E]., [一[-1092 : 2-F-6-MeO, 4-MeO, E], [-[-1094 : 3-F-4-MeO, 4-MeO, E ], [-[-1096:4-F-2-MeO,4-MeO,E ], [ -[-1098:2-Cl-3-MeO,4-MfeO,E], [-C-HOO: 2-Cl-5-MeO, 4-MeO, E], [-[-1102:3-Cl -2-MeO,4-MeO,E],[-[-1104:3-Cl-5-MeO,4-Me〇,E],[-[-1106:4-Cl-3-MeO,4- MeO, E], [-C-1108: 2-Me-4-MeO, 4-MeO, E] f [-[-1110: 2-Me-6-MeO, 4-MeO, E], [-[ -1112: 3-Me-4-MeO, 4-MeO ,E],[— (Me)3CO,E] Γ -1 1 4-Γ.ο . 4- 74 320202 200901876 (Me)2CH,4-(Me)3CO,E],[-1128:4-CF3r4 -(Me)3CO,E],[-1129:4-CF3,4-(Me)3CO,Z 3 , [-1130 : 4-C2 F5,4-(Me) 3 CO, E 3 ·, [- 1131:4-C3F7,4-(Me)3CO,E],[-1132:4-(CF3)2CF,4-(Me)3CO,E],[-1133:4-(CF3)2CH,4- (Me)3CO,E],,[-1134:4-CHF2,4-(Me)3CO,E], [-1135:4-CH2F,4-(Me)3CO,E], [-1136:4 -CF3CH2,4-(Me)3CO,E], [-1137:4^00/4-(Me)3C〇,E] , C-1138 :4-MeO, 4-(Me) 3 CO, Z ] , C-1139: 4-EtO, 4-(Me)3CO, E], [-1140: 4-C3H7O, 4-(Me)3CO, E], [-1141: 4-(Me)2CHO,4- (Me)3C〇,E] , [-1142:4-NOz,4-(Me)3CO,E ], [-1143:4-N〇2,4-(Me)3CO,Z], [-114 4:3-F, 4 - (Me>3 CO, E], [- 1145:3-F,4-(Me)3CO,z3, C-1146: 3-C1, 4-(Me) 3 CO, E] , [-1-147:3-Cl,4-(Me)3CO,Z] , [-1148:3-Br,4-(Me)3CO,E] · [-1149:3-1,4 - (Me)3CO,E 〕 , [ -1150:3-Me,4-(Me)3CO,E], [ -1151:3-Me,4-(Me)3CO,Z], [-1152:3 -Et,4-(Me)3CO,E], [-1153:3-C3H7,4-(Me.)3CO,E], [-1154:3-(Me)2CH,4-(Me>3CO, E], [-1155: 3-CF3, 4-(Me) 3CO , E], [ -1156: 3-CF3,4-(Me) 3 CO, Z ) , [-1157 :3-C2 F5,4- (Me)3CO,E] , [ -1158:3-C3 F7 ,4-(Me)3 CO,E] , [ -1159:3- (CF3 )2CF,4-(Me)3CO,E], C-1160:3-(CF3 )2CH,4-(Me)3CO , E], [-1161: 3-CHF2, 4-(Me) 3CO, E], [-1162: 3-CHF2, 4-(Me)3CO, Z], [-1163: 3-CH2F, 4- (Me) 3CO, E], C -1164 : 3-CH2 F, 4- (Me) 3 CO, Z ], (-1165: 3-CF3CH2, 4-(Me) 3CO, E], [-1166: 3-MeO,4-(Me),3CO,E],[-1167:3-MeO,4-(Me)3C〇,Z], [-1168 :3-EtOf 4-(Me) 3 C0,E 3, [- 1169: 3-C3H7O, 4-(Me) 3CO, E] , [-1170: 3-(Me) 2CHO, 4-(Me) 3CO, E], [-1171: 3-N02, 4 -(Me)3C0,E],[-1172:2-F,4-(Me)3CQ,E],[-1173:2-Clr4-(Me)3CO,E], C-1174:2-Br , 4-(Me)3 CO,E ], [- 1175:2-1,4-(Me)3CO,E] , [-1176:2-Me,4-(Me>3CO,E], [- 1177:2- 75 320202 200901876

Et,4-(Me)3CO,E ] , [-1178 :2-C3 H7,4-(Me) 3 CO, EJ , [-1179:2- (Me)2CH,4-(Me)3CO,E ], [-1180: 2-CF3,4-(Me)3CO, E]., [-1181: 2-C2F5,4-(Me)3CO, E], [-1182:2-C3F7,4-( Me) 3CO, E], [-1183: 2-(CF3)2CF, 4-(Me)3CO, E], [-1184: 2-(CF3)2CH, 4-(Me)3CO, E], -1185: 2-CHF2,4-(Me)3CO,E], [-1186:2-CH2F,4-(Me)3CO,E3,[- 1187:2-CF3CH2,4-(Me)3CO,E ], C-1188: 2-MeO, 4-(Me)3CO, E], [-1189: 2-EtO, 4-(Me>3CO, E], [-1190: 2-C3H7O, 4-(Me ) 3CO, E], [-1191: 2-(Me)2CHO, 4-(Me)3C〇, E], [-1193:2,3-F2/4-(Me)3CO,E], [- 1195: 2,5-F2,4-(Me)3CO,E], C -1197:3,4-F2,4-(Me) 3 C〇, E], [-1199:3,5-F2, 4-(Me)3CO,E], [-1201:2,3-Cl2,4-(Me)3CO,E] r [-1203:2,4-Cl2,4-(Me)3C〇,E] , [-1205:2,5-Cl2,4-(Me)3C〇,E), [-1207:2,6-Cl2,4-(Me)3CO,E], [-1209:3,5- Cl2,4-(Me)3CO,E], [-1211:2,4-Br2,4-(Me>3CO,E], [-1213:2,6-Br2,4-(Me)3CO,E ], [-1215:3,5-Br2,4-(Me)3CO,E], [-1217:2,4-Me2,4-(Me)3CO,E], [-1219:2,6- Me2,4-(Me)3CO,E], [-1221:3,5-Me2,4-(Me)3CO,E], [-1223:2,4-Et2,4-(Me) 3CO,E], [-1225:2,6-Et2,4-(Me)3CO,E], [-1192:2-N02,4-(Me)3C〇,E], [-1194:2, 4-F2,4-(Me)3C〇,E], [-1196:2,6-F2,4-(Me)3C〇,E], [-1198:3,4-F2,4-(Me ) 3CO, Z], [-1200:3,5-F2,4-(Me)3 CO,Z], [-1202:2,3-Cl2,4-(Me)3C〇,Z], [- 1204: 2,4-Cl2,4-(Me)3CO,Z], [-1206:2,5-CI2,4-(Me)3CO,Z], [-1208:3,4-Cl2,4- (Me)3CO,E], [-1210:2,3-Br2,4-(Me)3CO,E] r [-1212:2,5-Br2,4-(Me)3CO,E], C- 1214:3,4-Br2,4-(Me)3CO,E} r [-1216:2,3-Me2,4-(Me)3C〇,E〇, [-1218:2,5-Me2,4 -(Me)3C〇,E], [-1220:3,4-Me2,4-(Me)3CO,E], [-1222:2,3-Et2,4-(M^)3CO,E] , [-1224:2,5-Et2,4-(Me)3CO,E] f [-122 6:3, 4-Et2 , 4- (Me) 3C〇,E], 76 320202 200901876 [-1227: 3,5-Et2,4-(Me>3CO,E], [ -1228:2,3-(CF3)2,4- (Me>3CO,E], [-1229:2, 4-(CF3) 2,4-(MehCO,E],.[-1230:2,5-(CF3)2,4-(Me)3C〇,E], C-1231: 2,6-(CF3) 2 , 4- (Me) 3 CO, E ], [- 1232:3,4-(CF3)2,4-(Me)3CO,E], [ -1233:3,5-(CF3)2,4- (Me) 3CO,E] , [-1234:2,3- (CHF2)2,4-(Me)3 CO,E] r [-1235:2, 4- (CHF2)2,4-(Me)3CO,E ] , C-1236: 2,5-(CHF2) 2,4-(Me)3C〇:E],[-1237:2,6-(CHF2)2,4-(Me)3CO,E], [-1238:3,4-(CHF2)2,4 - (Me)3CO,E] , [-1239:3,5-'(CHF2)2,4-(Me)3CO,E] , [-1240:2,3- (CH2F)2 ,4-(Me ) 3C〇,E] , C-1241: 2,4-(CH2 F) 2 , 4-(Me) 3 CO, E],[-1242:2,5-(CH2F)2,4-(Me) 3CO,E] , C -1243:2,6-(CH2 F) 2,4-(Me)3CO,E] , [-1244:3, 4-(CH2F)2,4-(Me)3CO,E ] , (-1245:3,5- (CH2F)2 ,4-(Me)3CO,E] , [-1246:2,3-(MeO) 2,4-(Me) 3 CO, E ],[ - 1247: 2,4-(Me〇)2,4-(Me)3CO,E 〕. , [ -1248:2,5-(MeO) 2,4- (Me)3CO,E], [-1249 :2,6-(MeO)2,4-(Me)3CO,E], [ -1250:3, 4- (MeO)2,4-(Me)3CO,E ] , [-1251:3,5 -(MeO)2,4-(Me)3CO,E],[- 1252:2,3-(EtO}2,4-(Me)3 CO,E], [ -1253:2,4-(EtO ) 2,4- < · , * (Me) 3CO,E ] , [-1254:2,5-(EtO)2r[(Me)3CO,E]r C -1255:2,6- (EtO) 2,4-(Me)3CO,E],[-1256:3,4-(EtQ)2,4-(Me)3CO,E],[-1257:3,5-(EtO)2,4- (Me)3C〇,E] , [-1258:2-C1-3-F,4-(Me)3 CO,E], C -1259:2-Cl-4-F,4-(Me)3 CO,E 〕 , 〔 -1260:2-C1-5-F,4-(Me)3CO,E] , C-1261:2-Cl-6-F,4-(Me)3CO,E] , C -1262:3-C1-2-F, 4-(Me) 3C〇,E],'[-12 63 : 3-C1- 4-F, 4- (Me) 3 CO, E] , [-1264:3-d-5-F,4-(Me)3CO,E] , [-1265:4-C1-2-F,4 -(Me)3CO,E],.[-1266:4-Cl-3-F,4-(Me)3CO,E],[ -1267:2-F-3-Me,4-(Me)3CO , E], [-1268: 2-F-4-Me, 4-(Me)3CO, E), [-1269: 2-F-5-Me, 4-(Me)3CO, E], 77 320202 200901876 [-1270:2-F-6-Me,4-(Me)3CO,E], [ -1271:3-F-2-Me,4-(Me)3CO,E], [-1272:3 -F-4-Me,4-(Me)3CO,E],〇1273:3-F-5-

Me, 4-(Me) 3C〇, E], [-1274 : 4-F-2-Me, 4-(Me) 3 CO, E] , [-1275.-4-F-3-Me, 4 -(Me)3〇〇,E), [ -1276:2-Cl-3-Me,4-(Me)3CO, E ] , C - 1277:2-Cl-4-Me,4- (Me) 3CO,E] , [-12 78:2-Cl-5-Me,4-(Me)3COfE), [-1279:2-Cl-6-Mer4-(Me)3CO,E], C -1280: 3-Cl-2-Me,4-(Me)3CO,E], [-1281:3-Cl-4-Me,4-(Me)3CO,E], [-1282:3-Cl-5- Me,4-(Me)3CO,E) , [-1283:4-Cl-2-Me,4-(Me)3CO,E) , [-1284:4-Cl-3-Me,4-(Me ) 3CO, E ] , [-1285: 2-F-3-CF3 , 4-(Me) 3CO, E] · [- 1286: 2-F-4-CF3,4-(Me)3CO, E], [-1287: 2-F-5-CF3,4-(Me)3CO, E], [-1288: 2-F-6-CF3,4-(Me) 3 CO, E ] , [ -1289 : 3 *-F-2-CF3, 4-(Me)3CO,E] r [-1290:3-F-4-CF3,4-(Me)3CO,E], [-1291:3-F-5- CF3,4-(Me)3CO,E) f [-1292:4-F-2-CF3,4-(Me)3CO,E] , [-1293:4-F-3-CF3,4-(Me ) 3 CO,E] , [-1294:2-Cl-3-CF3,4-(Me)3 CO,E ], [- 1295:2-Cl-4-CF3,4-(Me)3CO,E ], [ -1296:2-Cl-5-CF3,4-(Me)3CO,E], [-1297:2-Cl-6-CF3,4-(Me)3CO,E], C-1298: 3-C1-2-CF3,4-(Me)3 CO,E ] , [ -1299:3-Cl-4-CF3,4-(Me)3CO,E],[- 1300:3-Cl-5 -CF3,4-(Me)3C〇,E , [ -1301:4-Cl-2-CF3,4-(Me)3C〇,E], [-1302:4-Cl-3-CF3,4-(Me)3CO,E], [-1303: 2-Me-3-CF3,4-(Me)3CO,E], [-13CM: 2-Me-4-CF3,4-(Me) 3 CO,E],[- 1305:2-Me-5 -CF3,4-(Me)3 CO,E ] , [ -1306:2-Me-6-CF3,4- (Me)3CO,E] , [-1307:3-Me-2-CF3,4- (Me)3CO,E] , [-1308:3-Me-4-CF3,4-(Me)3CO,E ] r [ -1309:3-Me-5-CF3,4-(Me)3〇〇 , E ), [-1310:4-Me-2-CF3,4-(Me)3CO,E], [ -1311:4-Me-3-CF3,4-(Me)3C〇,E3, [- 1312: 2-F-3-MeO, 4-(Me)3 CO, E), [-1313: 2-F-4- 78 320202 200901876

MeO,4-(Me)3CO,e3, [-1314:2-F-5-MeO,4-(Me)3CO,E], [-1315:2-F-6-MeO,4-(Me) 3CO, E], C-1316: 3-F-2-MeO, 4-(Me)3CO, E],, [-1317: 3-F-4-MeO, 4-(Me>3CO, E], [-1318: 3-F-5-MeO, 4-(Me)3CO, E], [-1319: 4-F-2-MeO, 4-(Me)3CO, E], 〔 -1320:4- F-3-MeO,4-(Me)3CO,E], [-1321:2-Cl-3-MeO,4-(Me)3CO,E], [-1322:2-Cl-4-MeO, 4-(Me) 3 C〇,E ) , [ -1323 :2-Cl-5-MeO, 4-(Me) 3 CO, E ·], [- 1324:2-Cl-6-MeO,4- (Me) 3 CO, E 〕 , [ -1325:3 diCl-2-MeO,4-(Me)3CO,E] , [-1326:3-Cl-4-MeO,4-(Me)3 CO , Ej , [-1327: 3-Cl-5-MeO, 4-(Me) 3CO, E ] , [ -1328: 4-Cl-2-MeO, 4-(Me) 3CO, E], [- 1329 :4-Cl-3-MeO,4-(Me)3CO,E ] , C -1330:2-Me-3-MeO,4-(Me)3CO,E],[-1331:2-Me-4 -MeO,4-(Me)3CO,E],[-1332:2-Me-5-MeO,4-(Me)3 CO,E], [-1333:2-Me-6-MeO,4- (Me)3 CO, E], [- 1334: 3-Me-2-MeO, 4-(Me) 3 CO, E 〕 , 〔 -1335: 3-Me-4-MeOr 4- (Me) 3CO, E], [-1336: 3-Me-5-MeOr4-(Me)3CO, E], [-1337: 4-Me-2-MeO, .4-(Me.)3CO, E], [-1338 :4-Me-3-MeO, 4-(Me) 3CO, E], [-1339:H,3-F,E], [-13 40:4-F,3-F,E], [-1341:4-F,3-F,Z], [-1342:4-C1,3-F,E], [-1343:4-C1 , 3-F, 2] , [-1344: 4-Br, 3-F, El·, [-1345: 4-1,3-F, E], [-1346: 4-Me, 3-F, E], [-1347: 4-Me, 3-F, Z], [-1348 : 4-Et, 3-F, E ] / C -1349: 4-C3 H7,3-F, E !1 , [-1350: 4-(Me)2CH, 3-F, E], [-1351: 4-CF3, 3-F, E], [-1352: 4-CF3, 3-F, Z], C- 1353:4-C2F5,3-F,E ] , C-1354 : 4-C3 F7,3-F, E ] , [-1355:4-(CF3)2CF,3-F,E].,C - 1356: 4-(CF3)2CH, 3-F, E], C-1357: 4-CHF2,3-F, E], [-1358:4-CH2F, 3-F, E], [-i359: 4-CF3Cii2r3-F, E], . [-1360:4-MeO,3-F,E], [-1361:4-MeO,3-F,Z], [-1362:4-EtO,3- F, E], [-1363: 4-C3H7〇, 3-F, E], [-1364: 4-(Me)2CHO, 3-F, E],. [- 79 320202 200901876 1365:4-N 〇2,3-F,E], [-1366: 4-N02,3-F, Z], [-1367 : 3-F, 3-F, E]r C-1368:3-F,3- F,Z] , [-1369:3-C1, 3-F, E] , [-1370 :3-C1,3-F, Z] [-1371:3-Br,3-F,E] , [ -1372: 3-1,3-F, E], [-1373: 3-Me, 3-F, E], [-1374: 3-Me, 3-F, Z], [-1375: 3- Et,3-F,E], [-1376:3-C3H7,3_F,E], [-1377:3-(Me)2CH,3-F, E], [-1378: 3-CF3, 3-F, E], [-1379: 3-CF3/3-F, Z], C-1380: 3-C2 Fs, 3-F, E), [ -1381: 3-C3 F7,3-F,E], [-1382:3-(CF3)2CF,3-F,E], [-1383:3-(CF3)2CH,3-F,E] , [-1384: 3-CHF2, 3-F, E], [-1385: 3-CHF2, 3-F, Z], [-1386: 3-CH2F, 3-F, E], [-1387: 3-CH2F,3,F,Z], [-1388:3-CF3CH2,3-F,E], C-1389:3-MeOf3-F,E], [-1390:3-MeO,3-F ,Z] , (-1391:3-EtO,3-F,E], [-1392:3-C3H70,3-F,E], [-1393:3-(Me)2CHO/3-F,E ], [-1394: 3-N02, 3-F, E], [-1395: 2-F, 3-F, E], [-1396: 2-C1,3-F, E], [-1397 :2-Br,3-F,E], [-1398:2-1,3-F,E], [-1399:2-Me,3-F,E], [-1400:2-Et, 3-F, E], [-1401: 2-C3H7, 3-F, E], [-1402: 2-(Me> 2CH, 3-F, E], [-1403: 2-CF3, 3- F, E], [-1404: 2-C2F5, 3-F, E], C-1405: 2-C3F7, 3-F, E), [-1406 : 2-(CF3 ) 2 CF, 3-F , E] , [-1407:2-(CF3)2CH,3-F,E], [-1408:2-CHF2,3-F,E], [-1409:2-CH2F,3-F,E ], [-1410: 2-CF3CH2, 3-F, E], [-1411: 2-Me〇, 3-F, E], [-1412: 2-EtO, 3-F, E], [- 1413 :2-C3 H7 O', 3-F, E ] , C -1414:2- (Me)2C HO,3-F,E], [-1415:2-N〇2,3-F,E], [-1416:2,3-F2,3-F,E], [-1417:2,4 -F2,3-E:,E],[-1418:2,5-F2,3-F,E], [-1419:2,6-F2,3-F,E'], [-1420: 3, 4-F2,3-F, E], [, 1421: 3, 4-F2, 3-F, Z], [-1422: 3, 5-F2, 3-F, E], [-: U23:3,5-F2,3-F.,Z], [-1424:2,3-CI2,3-F,E], C-1425:2,3-Cl2,3-F,Z], [-1426: 2,4-C12,3-F,E], [-1427:2,4-C12,3-F,Z], [-1428:2,5-C12,3-F,E] , 80 320202 200901876 [-1429: 2,5-C12,3-F,Z], [-1430:2,6-C12,3-F,E], [-1431:3,4-C12,3- F, E], [-1432:3,5-Cl2,3-F,E], [-1433:2,3-Br2,3-F,E], [-1434:2,4-Br2,3 -F, E], [-1435:2,5-Br2,3-F,E], [-1436:2,6-Br2/3-F,E], [-1437 : 3,4-ΒΓ2 / 3-F, E] , [-1438 : 3, 5-Br2 ^ 3-F, E], [-1439:2,3-Me2,3-F,E] , [-1440:2,4-Me2 ,3-F,E] , [-1441:2,5-Me2,3-F,E], [-1442:2,6-Me2,3-F,E],[-1443:3,4- Me2,.3-F,E], [-1444:3,5-Me2,3-F,E]r[-1445:2,3-Et2,3-F,E], [-1446:2, 4-Et2,3-F,E], [-1447:2,5-Et2,3-F,E], [-1448:2,6-Et2,3-F,E], [-1449: 3,4-Et2,3-F,E], [-1450:3,5-Et2,3-F,E], [-1451:2,3-(CF3)2,3-F,E], [ -1452:2,4-(CF3)2,3-F,E], [ -1453:2, 5-(CF3)2,3-F,E], [-1454:2,6-(CF3>;2,3-F,E],[* -1455:3, 4-(CF3)2,3-F,E], [-1456:3,5-(CF3)2,3-F,E] , [ -1457:2,3- (CHF2)2,3-F,E], [-1458:2,4-(CHF2h,3-F,E], [-1459:2,5-(CHF2) 2,3-F,E ) , [ -1460:2,6-(CHF2) 2,3-FfE ] , [-1461:3,4- (CHF2) 2,3-F,E], [-1462 :3,5-(CHF2)2,3-F,E], [-1463:2,3-(CH2F)2,3-F,E], [-1464:2,4-(CH2F)2, 3-F, E], [.-1465:2,5-(CH2F)2,3-F,E], [-1466:2,6-(CH2F)2,3-F,E], [- 1467:3,4-(CH2F)2,3-F,E ] , [ -1468:3,5-(CH2F)2,3-F,E ] , [-1469:2,3- (MeO)2 , 3-F, E 〕 , [ -1470:2,4-(MeO)2,3-F,E ] , [ -1471:2,5- (MeO)2,3-F,E], 〔 1472:2,6-(MeO)2,3-F,E], [ -1473:3,4-(MeO)2,3-F,E], [-1474:3,5-(MeO)2 , 3-F, E 〕 , [ -1475:2,3- (Et〇) 2,3-F,E 〕 , . 〔 -1476:2,4-(EtO)2,3-F,E 〕 , [-1477:2,5- (EtO)2,3-F,E ] , [ -1478:2,6-(EtO)2,3-F,E], [ -1479:3,4- (Et 〇) 2,3-F, E], -1480:3,5-(EtO)2,3-F,E], [-1481:2-Cl-3-F,3-F,E], [-1482:2-Cl-4-F, 3-F,E] , [-1483:2-C1-5-F,3-F,E], 81 320202 200901876 C-1484:2-Cl-6-F,3-F,E] , 〔- 1485: 3-C1-2-F, 3-F, E], [-1486: 3-Cl-4-F, 3-F, E], [-1487: 3-Cl-5-F, 3- F, E], [-1488: 4-Cl-2-F, 3-F, E], [-1489: 4-Cl-3-F, 3-F, E], [-1490: 2-F -3-Me,3-F,E], [-1491: 2-F-4-Me, 3-F, E], [-1492: 2-F-5-Me, 3-F, E], [-1493: 2-F-6-Me, 3-F, E], [-14 94: 3-F-2-Me, 3-F, E], C-1495: 3-F-4-Me , 3-F, E], [-1496: 3-F-5-Me, 3-F, E], [-1497: 4-F-2-Me, 3-F, E], [-1498: 4-F-3-Me,3-F,E], [-1499:2-Cl-3-Me,3-F,E], [-1500:2-Cl-4-Me,3-F, E]r [ -1501:2-Cl-5-Me,3-F,E ] , [ -1502:2-C1-6-

Me, 3-F, E], . [ -1503:3-Cl-2-Me,3-F,E ) , [ -1504:3-Cl-4-Me,3- F,E], [- 1505: 3-Cl-5-Me, 3-F, E], [-1506: 4-Cl-2-Me, 3-F, E], [-1507: 4-Cl-3-Me, 3- F, E] , [-1508 : 2-F-3-CF3,3-F, E]*, [-1509:2-F-4-CF3,3-F,E) , [-1510:2- F-5-CF3,3-F,E 3 , [-1511:2-F-6-CF3,3-F,E], [-1512:3-F-2-CF3,3-F,E) , [-1513 : 3-F-4-CF3,3-F, E], [-1514:3-F-5-CF3,3-F,E], [-1515:4-F-2-CF3 , 3-F, E], [-1516: 4-F-3-CF3, 3-F, E], [-1517: 2-Cl-3-CF3, 3-F, E], [-1518: 2-Cl-4-CF3,3-F,E], [-1519:2-Cl-5-CF3,3-F,E], [-1520:2-C1-6-CF3,3-F, E], [-1521: 3-Cl-2-CF3, 3-F, E], [-1522: 3-Cl-4-CF3, 3-F, E], [-1523: 3-Cl-5 -CF3,3-F,E], [-1524:4-Cl-2-CF3,3-F,E], [-1525:4-Cl-3-CF3,3-F,E], [- 1526: 2-Me-3-CF3, 3-F, E], [-1527: 2-Me-4-CF3, 3-F, E 3 , [ -1528: 2-Me-5-CF3, 3- F, E 〕, [- 1529: 2-Me-6-CF3, 3-F, E], [-1530: 3-Me-2-CF3, 3-F, E], [- 1531: 3-Me -4-CF3,3-F,E], [-1532:3-Me-5-CF3,3-F,E], [- 1533:4-Me-2-CF3,3-F,E], [-1534:4-Me-3-CF3,3-F,E],[- 1535:2-F-3-M eO,3-FfE], [-1536: 2-F-4-MeO, 3-F, E], [-1537: 2-F-5-Me〇, 3-F, E], [-1538: 2-F-6-MeO,3-F,E ] , [-1539:3-F-2- 82 320202 200901876

MeO, 3_F, E], (-1540: 3-F-4-MeO, 3-F, E], C-1541: 3-F-5-MeO, 3-F, E], [-1542:4 -F-2-MeO,3-F,E], [-1543:4-F-3-MeO,3-F,E], [- 1544:2-Cl-3-MeO,3-F,E 1546: 2-Cl-5-MeO, 3-F, E] 1548: 3-Cl-2-MeO, 3-F, E] 1550: 3-Cl-5-MeO, 3-F, E] 1552 :4-Cl-3-MeO,3-F,E] 1554:2-Me-4-MeO,3-F,E) 1556:2-Me-6-MeO,3-F,E ] 1558:3 -Me-4-MeO,3-F,E ) 1560:4-Me-2-MeO,3-F,E] [-1545:2-Cl-4-Me〇,3-F,E]., [-[-1547:2-Cl-6-MeOf3-F,E ],-[-1549:3-Cl-4-MeO,3-F,E ] , C - [-1551:4-Cl-2 -MeO,3-F,E.],[-[-1553:2-Me-3-MeO,3-F,E], [-[-1555:2-Me-5-MeO,3-F, E], [-[-1557:3-Me-2-MeO,3-F,E], [-[-1559:3-Me-5-MeO,3-F,E),[-[-1561 :4-Me-3-MeO,3-F,E], [-1562:H,3-C1,E], [-1563:4-Fr3-C1,E], [-1564:4-F, 3-C1,Z],[-1565:4-C1,3-C1,E ] , [-1566:4-C1,3-C1,Z],[ -1567:4-Br,3- C1,E ], [-1568: 4-I, 3-C1, E], [-1569: 4-Me, 3-C1, E], [-1570: 4-Me, 3-Cl, Z], [-1571 :4-Et,3-Cl,E], [-1572:4-C3H7,3-C1,E], [-1573:4-(Me)2CH,3-Cl,E], [-1574:4 -CF3,3-C1,E], [-1575: 4-CF3,3-C1,Z], [-157 6:4-C2F5,3-C1,E], [-1577:4-C3F7,3-C1,E], [-1578:4-(CF3 2CF,3-ClrE], [-1579:4-(CF3)2CH,3-Cl,E], [-1580:4-CHF2,3-Cl,E], C-1581:4-CH2F,3 -C1,E ] , C -1582:4-CF3CH2,3-Cl,E 3 , [ -1583:4-MeO,3-Cl,E ], C -1584:4-MeO,3-

Cl,Z], [-1585:4-EtO,3-Cl,E], [-1586:4-C3H70,3-Cl,E], [-1587:4-(Me)2CHO,3-Cl, E] , [-1588 : 4-N02,3-Clf E , [-1589:4-N02,3-C1,Z], [-1590:3-F,3-C1,E], [-1591: 3-F,3-Q1,Z], [-1592:3-C1,3-C1,E], [-1593:3-C1,3-C1,Z], [-1595:3-Br,3 - C1, E] , [-1595: 3-1,3-Cl, E], [-1596: 3-Me, 3-C1, E], [-1597: 3- 83 320202 200901876

Me,3-Cl,Z], [-1598:3-Et,3-C1,E], [-1599:3-C3H7,3-C1,E], [-1600:3-(Me)2CH/ 3-Cl,E ] , [-1601:3-CF3,3-C1,EJ , [-1602:3-CF3,3-C1,Z].,[-1603:3-C2F5,3-C1,E ], [-1604:3-C3F7,3-C1,E], [-1605:3-(CF3)2CF,3-C1,E], [-1606:3-(CF3)2CHr3-C1,E] , [-1607:3-CHF2,3-Cl,E], [ -1608:3-CHF2,3-C1,Z ], [ -1609:3-CH2F,3-C1/E], [-1610: 3-CH2F,3-C1,Z], C-1611: 3-CF3 CH2,3-C1,E], [-1612:3-MeO,3-Cl,E], [-1613:3-MeO, 3-C1,Z],[- 1614:3-EtO,3-Cl,E 3 ,C -1615:3-C3H7〇, 3-C1,E ] , [-1616:3- (Me)2CH0,3 -Cl, E], [-1617: 3-N02, 3-Cl, E], [-1618: 2-F, 3-Cl, E], [-1619: 2-Cl, 3-Cl, E] , [-1620: 2-Br, 3-Cl, E], [-1621: 2-I, 3-Cl, E], [-1622: 2-Me, 3-Cl, E], [-1623: 2-Et, 3: Cl, E], [-1624: 2-C3H7, 3-Cl, E], [-1625: 2-(Me) 2CH, 3-Cl, E], [-1626: 2- CF3,3-C1,E], [-1627:2-C2F5,3-C1,E], [-1628:2-C3F7,3-C1,E], C-1629:2-(CF3)2CF, 3-C1,E] , C-1630:2-(CF3)2CH,3-C1,E],[-1631:2-CHF2,3-Cl,E ], [ -1632:2-CH2F,3- C1,E ) f [-1633:2- GF3CH2,3-Cl,E ] , C -1 634: 2-MeOr3-Cl, E-], [-1635:2-EtOf 3-C1,E], [-1636:2-C3H70,3-C1,E], [-1637:2-(Me) 2CHO, 3-Cl, E], [-1638: 2-N〇2; 3-Cl, E], [-1639 : 2,3-F2,3-C1, E ] [-1640:2,4- F2,3-C1,E], [-1641:2,5-F2,3-C1,E], [-1642.:2,6-F2,3-C1,E], [-1643:3, 4-F2,3-Cl,E], [-1644:3,4-F2,3-ClrZ], [-1645:3,5-F2,3-C1,E], [-1646:3,5 -F2,3-Cl,Z], [-1647:2,3-Cl2,3-Cl,E], C-1648:2,3-C12,3-Cl,Z), [-1649:2, 4-Cl2,3-C1,E],[- 1650:2,4-CI2^3-C1,Z3, C-1651:2,5-CI2^3-C1,E], (-1652:2, 5-C12,3-C1,Z) , X-1653:2,6-Cl2,3-Cl,E ] , [ -1654:3, 4-Cl2,3- C1,E] , [-1655:3 , 5-CI2, 3-Cl, E], [-1656: 2r3-Br2, 3-C1, E], [- 84 320202 200901876 1657: 2, 4-Br2, 3-C1, e3, [-1658: 2,5-Br2,3-C1,E], [-1659:2,6-Br2,3-C1,E], [-1660:3, 4-Br2,3-C1,E]., [- I661: 3,5-Br2,3-C1,E], [-1662:2,3-Me2,3-C1,E], [-1663:2,4-Me2,3-C1,E], -1664: 2,5-Me2,3-Cl,E], [-1665:2,6-Me2,3-C1,, [-1666:3,4-Me2,3-C1,E], [- 1667:3,5-Me2,3-Cl,E ] , [ -1668 : 2,3-Et2,3-C1,E] , [-1669:2,4-Et2,3-C l, Ej, [-1670:2,5-Et2,3-C1,E), [-1671:2,6-Et2,3-Cl,E], [-1672:3,4-Et2,3- Cl,E] r [-1673:3,5-Et2,3-C1,E], [-1674:2,3-(CF3)2,3-Cl,E], [-1675:2,4- (CF3)2,3-Cl,E ] , [-1676:2,5-(CF3 )2,3-Cl,E ] , [-1677:2,6-(CF3)2,3-C1,E ], [-1678:3,4-(CF3)2,3-C1,E], [-1679:3, 5-(CF3)2,3-C1,E], [-1680:2,3- (CHF2) 2,3-C1,E], [-1681:2,4-(CHF2h,3-Cl,E], [-1682:2,5-(CHF2)2,3-Cl,E], [-1683:2,6-(CHF2)2,3-C1,E] , [-1684:3,4-(CHF2)2/3-Cl,E] , [-1685:3,5-(CHF2 2,3-C1,E],[-1686:2,3-(CH2F)2,3-C1,E], [-1687:2,4-(CH2F)2/3-Cl/E], [-1688:2,5-(CH2F)2,3-Cl,E] , [-1689:2,6-(CH2F)2,3-Cl,E] , [-1690:3,4-(CH2F 2,3-Cl,E] , [-1691:3,5-(CH2 F) 2,3-Cl,E 3 ,[-1692:2,3-(MeO)2 ,3-Cl,E] , C -1693: 2,4-(Me〇)2,3-Cl,E], [-1694:2,5-(Me〇>2,3-Cl,E], [-1695:2,6 -(MeO)2,3-Cl,E], [-1696:3, 4-(MeO)2,3-C1,E], [-1697:3,5-(MeO)2,3-Cl, E 3 , C-1698: 2,3-(EtO) 2,3-C1,E3 , [-1699:2,4-(EtO) 2,3-Cl,E], C-1700:2,5- (EtO)2,3-Cl,E], [-1701:2,6-(Et〇)2,3-Cl,E],'[ -1702:3,4-(Et〇)2,3-Cl,E],[-1703:3,5-(EtO)2,3-ClfE3, C-1704:2-Cl-3-F,3 -Cl, Ej, [-17〇5:2-C1-4-F,3-Cl,E], [-1706:2-Cl-5-F,3-Cl,E], [-1707:2 -Cl-6-F,3-C1,E], [-1708:3-Cl-2-F,3-Cl,E], [-1709:3-C1-4-F,3-C1ΓE], 85 320202 200901876 [-1710:3-Cl-5-F,3-Cl,E ] , [ -1711:4-C1-2-F,3-C1,E ], [- 1712:4-Cl-3 -F,3-Cl,E], [-1713:2-F-3-Me,3-ClrE]., [-1714:2-F-4-Me,3-Cl,E], [-1715 :2-F-5-Me,3-C1,E],[ -1716:2-F-6-

Me, 3-C1, E], [-1717: 3-F-2-Me, 3-Cl, E], [ -1718: 3-F-4-Me, 3-C1, E], [-1719 :3-F-5-Me,3-Cl,E] , [-1720:4-F-2-Me,3-Cl,E], [-1721:4-F-3-Me,3-Cl , E] , [-1722: 2-Cl-3-Me, 3-Cl, E] r [, 1723: 2-Cl-4-Me, 3-Cl, E], 1725: 2-Cl-6- Me, 3-Cl, E], 1727: 3-Cl-4-Me, 3-Cl, E], 1729: 4-Cl-2-Me, 3-Cl, E], 1731: 2-F-3 -CF3,3-Cl,E], 1733:2-F-5-CF3r3-Cl,E], 1735:3-F-2-CF3,3-Cl,E], 1737:3-F-5- CF3,3-Cl,E], 1739:4-F-3-CF3,3-Cl,E], 1741:2-Cl-4-CF3,3-Cl,E], 1743:2-Cl-6 -CF3,3-Cl,E], 1745:3-Cl-4-CF3,3-Cl,E], 1747:4-Cl-2-CF3,3-Cl,E], 1749:2-Me- 3-CF3,3-Cl,E], 1751:2-Me-5-CF3,3-Cl,E], 1753:3-Me-2-CF3,3-Cl,E], 1755:3-Me -5-CF3,3-Cl,E], 1757:4-Me-3-CF3,3-Cl,E], 1759:2-F-4-MeO,3-Cl,E], [-1724: 2-Cl-5-Me,3-Cl,E ],-[-1726:3-Cl-2-Me,3-Cl,E], [-[-1728:3-Cl-5-Me,3 -Cl, E], [-[-1730:4-Cl-3-Me,3-Cl,E], [-[-1732:2-F-4-CF3,3-CI,E], C - [-1734: 2-F-6-CF3,3-Cl, E]r[-[-1736:3-F-4-CF3,3-Cl, EJ,-[-1738:4-F-2- CF3,3-Cl,E ) r 〔-[-1740:2-Cl- 3-CF3,3-Cl,E],[-[-1742 :2-C1-5-CF3,-3_Cl, E],[—[-1744:3-Cl-2-CF3,3-Cl,E ], [-[-1746:3-Cl-5-CF3,3-Cl,E], [-[-1748:4-Cl-3-CF3,3-Cl,E],[-[-175Q: 2-Me-4-CF3,3-Cl,E], [-[-1752:2-Me-6-CF3,3-Cl,E], [-[-1754:3-Me-4-CF3, 3-Cl,E],[-[-1756 : 4-Me-2-CF3,3-Clv E ], [-C -1758:2-F-3-MeO,3-Cl,E ] , C - [-1760: 2-F-5-MeO, 3-Cl, E], [- 86 320202 200901876 1761: 2-F-6-MeO, 3-Cl, E], 1763: 3-F-4-MeO , 3-Cl, E 〕, 1765: 4-F-2-MeO, 3-Cl, E ), 1767: 2-Cl-3-MeO, 3-Cl, E ], 1769: 2-Cl-5- MeO, 3-Cl, E], 1771: 3-Cl-2-MeO, 3-Cl, E], 1773: 3-Cl-5-MeO, 3-Cl, E], 1775: 4-Cl-3 -MeO,3-Cl,E], 1777 :2—Me-4-Me〇,3-Cl,E]., 1779:2-Me-6-MeO,3-Cl,E ], 1781:3- Me-4-MeO,3-Cl,E ), C -1762:3-F-2-MeO,3-Cl,E 3 ,C - [-1764:3-F-5-MeO,3-Cl, E], [-[-1766:4-F-3-MeO,3-Cl,E], [-[-1768:2-Cl-4-MeO,3-Cl,E],[-[-1770 :2-Cl-6-MeO,3-Cl,E],[-[-1772:3-Cl-4-MeO,3-Cl,E],[-[-1774:4-Cl-2-MeOr3 -Cl, E], [- [-1776: 2-Me-3-MeO, 3-Cl, E], [- [-1778: 2-Me-5-MeO, 3- Cl, E], [-[-1780:3-Me-2-MeO, 3-Cl, E], [-[-1782:3-Me-5-MeO, 3-Cl,E], [- 1783 :4-Me-2-MeO,3-Cl,E], [-1784:4-Me-3-MeO,3-C1,E], [- 1785:H,3-CF3,E], C- 1786: 4-F,3-CF3,E] f [-1787:4-F,3-CF3,Z], [-1788:4-C1,3-CF3,E], [-1789:4-C1 , 3-CF3, Z], [ -1790:4-

Br,3-CF3,E], [-1791:4-I,3-CF3,E], [-1792:4-Me,3-CF3,E], [-1793:4-Me,3-CF3 ,Z], [-1794:4-Et,3-CF3,E], [-1795:4-C3H7,3-CF3,E],[-1796:4-(Me)2CH,3-CF3, [ -1797 : 4-CF3 r 3-CF3 , E), C-1798: 4-CF3,3-CFs ,Z] , [-17 99 : 4-C2 F5,3-CF3 , E ] , [-1800: 4-C3F7,3-CF3,E ] , [ -1801:4-(CF3 )2CF,3-CF3,E],[ -1802:4- (CF3 )2CH,3-CF3,E], [ -1803 :4-CHF2,3-CF3,E], [-1804:4-CH2F,3-CF3,E], [-1805:4-CF3CH2,3-CF3,E], [-1806: 4-MeO, 3-CF3, E], [-1807: 4-MeO, 3-CF3, Z], [-1808: 4-EtO, 3-CF3, E], [-1809: 4-C3H7〇, 3-CF3, E ] , [ -1810 : 4-(Me) 2 CHO, 3-CF3 fcE], [- 1811:4-N02,3-CF3,E], [-1812:4-N02,3-CF3,Z] , [-1813:3-F,3-CF3,E], [-1814:3-F,3-CF3,Z], [-1815: 3-C1, 3-CF3 Λ E], [- 87 320202 200901876 1816: 3-Cl, 3-CF3, Z], [-1817: 3-Br, 3-CF3, E], [-1818: 3-I, 3-CF3, E], [-1819: 3- Me, 3-CF3, E], [-1820: 3-Me, 3-CF3, Z], [-1821: 3-Et, 3-CF3, E], [-1822: 3-C3H7, 3-CF3 , E 〕 , [-1823: 3-(Me) 2CH, 3-CF3 , E] , [-1824 : 3~CF3 , 3-CF3, E ] f C-1825: 3-CF3, 3-CF3, Z], [-1826: 3-C2F5, 3-CF3, E], [-1827: 3-C3F7, 3-CF3, E], [-1828: 3-(CF3)2CF, 3-CF3, E], [-1829: 3-(CF3)2CH, 3-CF3,.E], [-1830: 3-CHF2, 3- CF3, E], [-1831: 3-CHF2, 3-CF3, Z], [-1832: 3-CH2F, 3-CF3, E], [-1833: 3-CH2F, 3-CF3, Z], [-1834: 3-CF3CH2, 3-CF3, E], [-1835: 3-MeO, 3-CF3, [-1836: 3-MeO, 3-CF3, Z], [-1837: 3-EtO, 3-CF3,E], [-1838:3-C3H70,3-CF3,E], [-1839:3-(Me)2CHO,3-CF3,E], [-1840: 3-N02,3- CF3, E], [ -1841:2-F,3-CF3,E]., [-1842:2-Cl,3-CF3,E], [-1843:2-Br,3-CF3,E] , [· 1844: 2-1,3-CF3 , E ] , [-1845: 2-Me, 3-CF3, E] , [-184 6: 2-Et, 3- CF3, E], [-1847 :2-C3H7,3-CF3,E]r[-1848 :2-(Me) 2 CH, 3-CF3, E], C-1849:2-CF3,3-CF3,E] , [-1850: 2-C2F5,3-CF3,E] f [-1851:2-C3F7,3-CF3,E } , [ -1852:2-(CF3)2CF,3-CF3,E], [ -1853:2- (CF3>2CH,3-CF3,E], [-1854:2-CHF2,3-CF3,E], [-1855:2-'CH2F,3-CF3,E], [-1856:2-CF3CH2 , 3-CF3, E], [-1857: 2-MeO, 3-CF3, E], [-1858: 2-EtO, 3-CF3, E], [-185 9 : 2-C3 H7 O, 3-CF3 , E], [-1860: 2-(Me) 2CHOr3-CF3 , E] , [ -1861: 2-N02, 3-CF3 , E], [- 1862: 2,3-F2,3-CF3,E], [-1863:2,4-F2,3-CF3,E], [-1864:2,5-F2f3-CF3/E], [-1865:2 , 6-F2,3-CF3,E ] , C -1866: 3,4-F2,3-CF3,E], [-1867:3, 4-F2,3-CF3,Z], [-1868: 3,5-F2,3-CF3,E], [-1869:3,5-F2,3-CF3,Z], [-1870:2,3-Cl2,3-CF3,E], [-1871 :2,3-C12,3-CF3,Z] , [-1872:2,4-Cl2/3-CF3/E] , C-1873:2,4-Cl2,3- 88 320202 200901876 CF3,Z] , [-1874: 2,5-Cl2,3-CF3,E], [-1875:2,5-Cl2,3-CF3,Z], [-1876:2,6-C12,3-CF3,E ], [-1877:3,4-C12,3-CF3,E], [-1878:3,5-Cl2,3-CF3,E], C-1879:2,3-Br2,3-CF3, E ],[- 1880:2,4-Br2,3-CF3,E] r [-1881:2,5-Br2,3-CF3,E], [-1882:2,6-Br2,3-CF3 , E 〕 , [-1883:3,4-Br2,3-CF3,E], [- 1884:3,5-Br2,3-CF3,E], [-1885: 2,3-Me2,3- CF3, E]., [- 1886: 2,4-Me2,3-CF3,E], [-1887:2,5-Me2,3-CF3,E], [- 1888:2,6-Me2, 3-CF3,E ] , [-1889:3,4-Me2,3-CF3,E], [- 1890:3,5-Me2,3-CF3,E], [-1891:2,3-Et2 , 3-CF3, E , [- 1892:2,4-Et2,3-CF3,E], [-1893:2,5-Et2,3-CF3,E], [- 1894:2, 6-Et2,3-CF3 3 , C -1895: 3,4-Et2,3-CF3/E ],[- 1896:3,5-Et2,3-CF3,E], [-1897:2,3-(CF3)2,3-CF3 , E], [-1898:2,4-(CF3 )2 f3-CF3 ,E] , [-1899 :2,5-(CF3 ) 2,3-CF3 , E ) r [- 1900:2,6 -(CF3)2,3-CF3,E] , [-1901: 3,4-(CF3 ) 2,3-CF3 , E ],[- 1902:3,5-(CF3)2,3-CF3, E] , [-1903:2,3-(CHF2)2,3-CF3,E],[-1904:2,4-(CHF2)2,3-CF3,E], [-1905:2,5 -(CHF2)2,3-CF3,E],[-1906:2,6-(CHF2)2,3-CF3,E), [-1907 :3,4-(CHF2) 2 / 3-CF3 , E], [-1908:3, 5-(CHF2)2,3-CF3,E], [-1909:2,3-(CH2F)2,3-CF3,E], [-, 1910:2, 4-(CH2F)2,3-CF3,E] , [-1911:2,5-(CH2 F) 2 f 3-CF3 r E) , C- 1912:2,6-(CH2F)2,3- CF3, E], [-1913:3,4-(CH2F)2,3-CF3,E], [-1914:3,5-(CH2F)2,3-CF3,E], [-1915:2 ,3-(MeO)2,3-CF3,E], [-1916:2,4-(MeO)2,3-CF3/E], [-1917 :2,5-(MeO) 2,3- CF3 , E ], [- 1918:2,6-(MeO) 2,3-CF3,E], [-1919:3,4-(MeO)2,3-CF_3,E], [-1920:3 , 5-(MeO)2,3-CF3,E], [-1921:2,3-(EtO)2,3-CF3,E], [-1922:2,4-(EtO)2,3- CF 3,E] , [-1923:2,5-(EtO>2,3-CF3,E], [- 89 320202 200901876 1924:2,6-(EtO)2,3-CF3,E] 1926:3 ,5-(EtO)2,3-CF3,E] 1928:2-Cl-4-F,3-CF3,E], 1930:2-Cl-6-F,3-CF3,E], 1932: 3-Cl-4-F,3-CF3,E]( 1934:4-Cl-2-F,3-CF3,E ) ' 1936:2-F-3-Me,3-CF3,E 〕 · 1938 :2-F-5-Me,3-CF3,E], 1940:3-F-2-Me,3-CF3,E], 1942:3-F-5-Me,3-CF3,E], 1944: 4-F-3-Me, 3-CF3, E], 1946: 2-Cl-4-Me, 3-CF3, E] 1948: 2-Cl-6-Me, 3-CF3, E] 1950 :3-Cl-4-Me,3-CF3,E] 1952:4-Cl-2-Me,3-CF3,E 3 1954 :2-F-3-CF3,3-CF3 ,E ]-1956: 2-F-5-CF3,3-CF3,E] 1958: 3-F-2-CF3,3-CF3,E] 1960:3-F-5-CF3,3-CF3,E] 1962:4- F-3-CF3,3-CF3,E], 1964:2-Cl-4-CF3,3-CF3,E] 1966:2-Cl-6-CF3,3-CF3,E] 1968:3-Cl -4-CF3,3-CF3/E] 1970: 4-C1-2-CF3,3-CF3, E ] 1972:2-Me-3-CF3,3-CF3,E] 90 ,[-1925:3 , 4-(EtO)2,3-CF3,E],[- ,[-1927:2-C1-3-F,3-CF3,E ),[- * [-1929:2-Cl-5- F,3-CF3,E],[-[-1931:3-Cl-2-F,3-CF3,E],[-[-1933:3-Cl-5-F,3-CF3,E] , [-[-1935:4-Cl-3-F,3-CF3, E.], [-[-1937:2-F-4-Me,3-CF3,E],[-[-1- 939 :2- F-6-Me, 3-CF3, E], -[-1941:3-F-4-Me,3-CF3,E], [-[-1943:4-F-2-Me,3-CF3 , E ], [-[-1945:2-Cl-3-Me,3-CF5,E ], [-r [-1947:2-Cl-5-Me,3-CF3 ,E3 , C - r [ -1949: 3-Cl-2-Me, 3-CF3, E], [-r [-1951: 3-Cl-5-Me, 3-CF3, E], [-r [-1953: 4-Cl -3-Me,3-CF3,E3, C - r [-1955:2-F-4-CF3,3-CF3,E],-[-r C-1957:2-F-6-CF3,3 -CF3,E],[-r [-1959:3-F-4-CF3,3-CF3,E], [-r C -1961: 4-F-2-CF3,3-CF3, E ), [-[-1963:2-Cl-3-CF3,3-CF3,E], [-,[-1965:2-Cl-5-CF3,3-CF3,E],[-,[-1967: 3-Cl-2-CF3,3-CF3,E],[-,[-1969:3-Cl-5-CF3,3-CFs,E],[-,[-1971:4-Cl-3- CF3,3-CF3,E],[-,[-1973:2-Me-4-CF3,3-CF3,E],[-320202 200901876 [-1975:2-Me-6-CF3,3-CF3 , E], [-[-1977:3-Me-4-CF3,3-CF3,E], [-C-1979:4-Me-2-CF3,3-CF3,E],[-[- 1981: 2-F-3-MeO, 3-CF3, E], [-[-1983: 2-F-5-MeO, 3-CF3, E], C-[-1985: 3-F-2- MeO,3-CF3,E],[-[-1987 : 3-F-5-MeO, 3-CF3 , E ], [-[-1989:4-F-3-MeO,3-CF3,E] , [-[-1991:2-Cl-4-MeO,3-CF3,E],[-[-1993:2-Cl-6-MeO,3-CF3,E],[-[-1995:3 -Cl-4-MeO,3-CF3,[-[-1997:4-Cl-2-MeO,3- CF3, E), [-[-1999: 2-Me-3-MeO, 3-CF3, E], [-[-2001: 2-Me-5-MeO, 3-CF3, E], [-[ -2003: 3-Me-2-Me, 3-CF3, E], [-[-2005: 3-Me-5-MeO, 3-CF3, E] r [- 1974 : 2-Me-5- CF3,3-CF3, e3 197 6:3-Me-2-CF3,3-CF3,E] 1978:3-Me-5-CF3,3-CF3,E] 1980:4-Me-3-CF3, 3-CF3,E] 1982:2-F-4-MeO,3-CF3,E] 1984:2-F-6-MeO,3-CF3,E) 1986:3-F-4-MeO,3- CF3, E] 1988: 4-F-2-MeO, 3-CF3, E] 1990: 2-Cl-3-MeO, 3-CF3, E] 1992: 2-Cl-5-MeO, 3-CF3, E] 1994: 3-Cl-2-MeO, 3-CF3, E] 1996: 3-Cl-5-MeO, 3-CF3, E] 1998: 4-Cl-3-MeO, 3-CF3, E] 2000: 2-Me-4-MeO, 3-CF3, E] 2002: 2-Me-6-MeO, 3-CF3, E] 2004: 3-Me-4-MeO, 3-CF3, E] 2006: 4-Me-2-Me〇,3-CF3, E] [-2007:4-Me-3-MeO,3-CF3,E] 2008:H,3-MeO,E] , [-2009:4- F,3-MeO,E] , [-2010:4-F,3-MeO,z], C-2011:4-Cl,3-MeO,E3 , [-2012:4-C1,3-MeO, Z ] , [-2013:4-

Br,3-MeO,E],[-2014:4-I,3-MeO,E],[-2015:4-Me,3-MeO,E],[-2016:4-Me,3-MeO , Z] , [-2017:4-Et,3-MeO,E] , C-2018:4-C3H7,3-MeO,E] , [-2019:4-(Me)2CH,3-MeO,E ), [-2020:4-CF3,3-MeO,E], C-2021:4-CF3,3-MeO,Z], [-2022:4-C2F5,3-MeO,E] ,.[- 2023:4-C3F7f3-MeO,E ] , [ -2024:4-(CF3)2CF,3-MeO,E ] , [-2025:4- (CF3)2CH,3-MeO,E ] r 〔 -2026 :4-CHF2,3-MeO,E], [-2027:4- 91 320202 200901876 CH2F, 3-MeO,E], C-202 8:4-CF3 CH2,3-MeO,E ] , [-2029 :4-MeO,3-

MeO, E], C-2030: 4-MeO, 3-MeO, Z], [-2031: 4-EtO, 3-MeO, E), [-2032: 4-C3H7O, 3-MeO, E], [-2033: 4-(Me)2CHO, 3-MeO, E], [- 2034: 4-NO2, 3-MeP, E], [-2035: 4-N〇2, 3-MeO, Z], [-2036: 3-F, 3-MeO, E], [-2037: 3-F, 3-MeO, Z], [-2038: 3-Cl, 3-MeO, E], [-2039:3 -Cl,3-MeO,Z ) , C-2040:3-Br,3-MeO,E ) , [-2041:3-1,3-

MeO, E], [-2042: 3-Me, 3-MeO, E], C-2043: 3-Me, 3-MeO, Z), C-2044: 3-Et, 3-MeO, E], [-2045:3-C3H7,3-MeO,E ] , [-2046:3-(Me)2CH,3-MeO,E] , [-2047:3-CF3,3-MeO,E] , C- 2048: 3-CF3, 3-

MeO, Z], [-2049: 3-C2F5, 3-MeO, E], [-2050: 3-C3F7, 3-MeO, E], [-2051: 3-(CF3)2CF, 3-MeO, E], [-2052: 3-(CF3)2CH, 3-MeO, E], [-2053: 3-CHF2, 3-MeO, E], C-2054: 3-CHF2, 3-MeO, Z) , [-2055:3-CH2F,3-MeO,E}, [-2056:3-CH2F,3-MeO,Z], [-2057:3-CF3CH2,3-MeO,E], [-2058: 3-MeO,3-MeO,E], [-2059:3-MeO,3-Me〇,Z], [- 2060:3-EtO,3-MeO,E3, [-2061:3-C3H7〇, 3-MeO,E ] r [-2062:3-(Me)2CH〇,3-MeO,E],[-2063:3-N02,3-MeO,E ] , [-2064:2-F,3 -

Me〇, E], [-2065: 2-Cl, 3-MeO, E], [-2066: 2-Br, 3-MeO, E], [- 2067: 2-1,3-Me〇, E ], [-2068:2-Me,3-MeOfE ] , [-2069:2-Et,3-

MeO, E], [-2070: 2-C3H7, 3-MeO, E], [-2071: 2-(Me) 2CH, 3-MeO, E], [-2072: 2-CF3, 3-MeO, E], [-2073: 2-C2F5, 3-MeO, E], [-2074: 2-C3F7, 3-MeO, E 3 , [ -2075: 2-(CF3 ) 2 CF, 3-MeO, E ] , [-2076:2-(CF3 )2〇H,3-MeO,E ') , [ -2077 :2-CHF2,3-MeO, E ] , [-2078:2-CH2F, 3-Me〇, E] , [-207 9 : 2-CF3 CH2,3-MeO, E ] , C-2080:2-MeO, 3-

MeO, E], [-2081: 2-EtO, 3-MeO, E], [-2082: 2-C3H7 0,3-MeO, E], [-2083: 2-(Me)2CHO, 3-MeO , E 〕 , 〔 -2084:2-N02r3-MeO,E 〕,[- 92 320202 200901876 2085:2,3-F2,3-MeO,E] , [-2086:2,4-F2,3-MeO ,E] , [-2087:2,5-F2,3-MeO,E] , [ -2088:2,6-F2,3-MeO,E ] , [ -2089 : 3,4-F2,3-

MeO,E] , [-2090:3, 4-F2 r 3-MeO, Z] , [-2091: 3,5-F2,3-MeO, E],[-2092:3, 5-F2,3 -MeO,Z] , [-2093:2,3-Cl2,3-MeO,E] , [-2094:2,3-Cl2,3-MeO,Z] , [-2095:2,4-Cl2, 3-MeO,E] , [-2096:2,4-Cl2,3-

MeO,z) , (-2097:2,5-Cl2,3-MeO,E] , [-2098:2,5-Cl2,3-MeO, z), [-2099:2,6-CI2,3 -MeO,E], [ -2100 : 3,4-Cl2,3-MeO,E], [- 2101:3,5-Cl2,3-Me〇,E], [-2102:2,3-Br2 , 3-MeO, E 〕, [- 2103: 2, 4-Br 2 , 3-MeO, E ] , { -2104: 2,5-Br2f3-MeO, E ), [- 2105:2,6-Br2, 3-MeO, E], [ -2106:3,4-Br2,3-MeO,E], [- 2107:3,5-Br2,3-MeO,E], [-2108:2,3-Me2 , 3-MeO,.E], [- 2109:2,4-Me2,3-Me〇,E], [ -2110:2,5~Me2,3-MeO,E 3 , C - 2111:2, 6-Me2,3-MeO,E] , C -2112:3,4-Me2,3-MeO,E ],[- 2113:3,5-Me2,3-MeO,E ], [ -2114:2 , 3-Et2,3-MeO, E 3, [- 2115:2,4-Et2,3-MeO,E], [-2116:2,5-Et2,3-MeO,E], [- 2117: 2,6-Et2,3-MeO,E), [-2118:3,4-Et2,3-MeO,.E], [- 2119:3,5-Et2,3-MeO,E], [- 2120: 2,3-(CF3)2,3-MeO,E], [-2121:2,4-(CF3)2,3-MeO,E], [-2122:2,5-(CF3)2 , 3-MeO, E ], [- 2123:2,6-(CF3>2,3-MeO,E], [-2124:3,4-(CF3)2,3-MeO,E], (- 2125:3,5-(CF3)2,3-MeO,E] , [-2126:2,3-(CHF2)2r3-MeO,E],[-2127:2,4-(CHF2)2.3-ΜθΟ ,Ε], [-2128:2,5-(CHF2)2,3-MeO,E],[-2129:2,6-(CHF2)2,3- MeO, E], [-2130:3,4-(CHF2)2,3-MeO,E], [-2131:3,5-(CHF2)2.3-MeO,Ej, [-2132:2,3- (CH2F)2,3-ΜβΟ,E],[-2133:2,4-(CH2F)2,3-MeO,E3, [-2134:2,5-(CH2F)2,3-MeO,E] , [-2135:2,6-(CH2F)2,3-MeO,E], [-2136:3,4-(CH2F)2,3-MeO,E], [-93 320202 [-2138:2 ,3-(MeO)2,3-MeO,E],[-[-2140:2,5-(MeO)2,3-MeO,E],[-[-2142:3,4-(MeO) 2,3-MeO,E] r [-[-2144:2,3-(EtO)2,3-MeO,E], [-[-2146:2,5-(EtO)2,3-MeO, E] , C-[-2148:3,4-(EtO)2,3-MeO,E], [-[-2150:2-C1-3-F,3-MeO,E ϋ ,[- 〔- 2152: 2-Cl-5-F, 3-Me〇, E], [-[-2154:3-Cl-2-F,3-MeO, E], [-[-2156:3-Cl-5 -F,3-MeO,E 3 ,- C -2158:4-Cl-3-F,3-MeO,E ] , C - [-2160:2-F-4-Me,3-MeO,E] , [-[-2162:2-F-6-Me,3-MeO,E] r [-[-2164:3-F-4-Me,3-MeO,E 3 ,[- [-2166:4 -F-2-Me,3-MeO,E], [-[-2168:2-Cl-3-Me,3-MeO,E],[-[-2170:2-Cl-5-Me,3 -MeO,E ),[-[-2172 : 3-Cl-2-Me, 3-MeO, E], [-[-2174 : 3-Cl-5-Me, 3-MeO, E ], [- [-2176:4-Cl-3-Me,3-MeO,E],[-[-2178 : 2-F-4-CF3,3-MeOf E ], [-[-2180:2-F-6 -CF3,3-MeO,E],[-[- 2182: 3-F-4-CF3,3-MeO/E], [-[-2184: 4-F-2-CF3,3-MeO, E), [-[-2186:2-Cl-3- CF3,3-MeO,E],[- 200901876 2137:3,5-(CH2F)2,3-MeO,E], 2139:2,4-(MeO)2,3-MeO,E] 2141:2 ,6-(MeO)2,3-MeO,E] 2143:3,5-(MeO)2,3-MeO,E] 214 5:2,4-(EtO)2,3-MeO,E] 2147 :2,6-(Et〇)2,3-MeO,E] 214 9:3,5-(Et〇)2,3-MeO,E] 2151:2-Cl-4-F,3-MeO, E 〕 2153: 2-Cl-6-F, 3-MeO, E] 2155: 3-Cl-4-F, 3-MeO, E] 2157: 4-Cl-2-F, 3-MeO, E] 2159: 2-F-3-Me, 3-MeO, E 3 2161: 2-F-5-Me, 3-MeO, E] 2163: 3-F-2-Me, 3-MeO, E] 2165: 3-F-5_Me,3-MeO,E] 2167:4-F-3-Me,3-MeO,E] 2169:2-Cl-4-Me,3-MeO,E] 2171:2-Cl- 6-Me,3-MeO,E] 2173:3-Cl-4-Me,3-MeO,E] 2175:4-Cl-2-Me,3-MeO,E 3 2177:2-F-3- CF3,3-MeO,E] 2179:2-F-5-CF3,3-MeO,E] 2181:3-F-2-CF3,3-MeO,E] 2183:3-F-5-CF3, 3-MeO,E] 2185:4-F-3-CF3,3-MeO,E] 94 320202 200901876 2187:2-Cl-4-CF3,3-Me〇,E] 2189:2-Cl-6- CF3,3-MeO,E] 2191:3-Cl-4-CF3,3-Me〇,E] 2193:4-Cl-2-CF3,3-MeO,E] 2195:2-Me-3-CF3 , 3-Me〇,E] 2197:2-Me-5-CF3,3-MeO,E] 2199:3-Me-2-CF3,3-MeO,E] 2201:3-Me-5-CF3, 3-MeO,E] 2203: 4_Me-3-CF3,3-MeO,E] 2205:2-F-4-MeO,3-MeO,E] 2207:2-F-6-MeO,3-MeO, E ] 2209: 3-F-4-MeO, 3-Me〇, E] 2211: 4-F-2-MeO, 3-MeO, E ] 2213: 2-Cl-3-MeO, 3-MeO, E 2215: 2-Cl-5-MeO, 3-MeO, E] 2217: 3-Cl-2-MeO, -3-Me〇, E] 2219: 3-Cl-5-MeO, 3-MeO, E ] 2221: 4-Cl-3-MeO, 3-MeO, E] 2223: 2-Me-4-MeO, 3-Me〇, E] 2225: 2-Me-6-MeO, 3-MeO, E] 2227: 3-Me-4-MeO, 3-MeO, E] 2229: 4-Me-2-MeO, 3-MeOf E] [-2188: 2-Cl-5-CF3, 3-MeO, E] [ -2190:3-Cl-2-CF3,3-MeO,E] C-2192:3-C1-5-CF3,3-MeO,E] [-2194:4-Cl-3-CF3,3-MeO ,E] [-2196:2-Me-4-CF3,3-MeO,E] [-2198 :2-Me-6-CF3,3-MeO,.E] [-2200:3-Me-4- CF3,3-MeO,E] [-22〇2:4-Me-2-CF3,3-MeO,E] [-2204:2-F-3-MeO,3-MeO,E] [-2206: 2-F-5-MeO,3-MeO,E] [-2208:3-F-2-MeO,3-ΜβΟ,Ε ] [-2210:3-F-5-MeO, 3-MeO,E 3 [-2212: 4-F-3-MeOf3-MeO, E) [-2214: 2-Cl-4-MeO, 3-MeO, E] (-2216: 2-Cl-6-MeO, 3-MeO, E) C-2218: 3-Cl-4-MeO, 3-MeO, E]· [-2220:4-Cl-2-MeO,3-MeO,E] [-2222:2-Me-3-Me 〇,3-MeO,E] [-2224:2-Me-5-MeO,3-MeO,E ] [-2226:3-Me-2-MeO,3-MeO,E] [-2228:3- Me-5-MeO,3- Me〇, E] [- 〔- 〔-[-[-[-[-[-[-[-[-[-[-[-[-[-[-[- 3-MeO,3-MeO,E] 2231:H,3-(Me)3CO,E], [-2232 : 4-F, 3-(Me) 3 CO, E],. [-2233:4- F,3-(Me)3 CO, Z] , [-2234:4-C1,3-(Me)3COfE3 , [-2235:4-01,3-(Me)3CO,Z], [-2232: 4-Br,3-(Me)3CO,E], 〔 -2237:4-1,3- « 95 320202 200901876 (Me)3CO,E ] , C -2238:4-Me,3-(Me)3CO , E ) , [ -2239: 4-Me, 3- (Me) 3CO, Z], [-2240: 4-Et, 3-(Me) 3CO, E], [-2241: 4-C3H7, 3- (Me) 3CO, E], [-2242: 4-(Me) 2CH, 3-(Me) 3CO, E], [-2243: 4-CF3, 3-(Me) 3CO, E], [-2244 :4-CF3,3-(Me)3CO,Z], [-2245:4-C2F5,3-(Me)3CO,E], [-2246:4-C3F7,3-(Me)3CO,E] , [ -2247:4-(CF3)2CF,3-(Me)3CO,E], [-2248:4-(CF3>2CH,3-(Me)3CO,E], [-2249:4-CHF2 , 3-(Me)3CO, E], [-2250: 4-CH2F, 3-(Me)3CO, E], [-2251: 4-CF3CH2, 3-(Me)3C〇, E], [- 2252:4-MeO,3-(Me)3CO,E],[-2253':4-MeO,3-(Me)3C〇,Z ] , [-2254 : 4-EtO, 3-(Me) 3 CO, E ], [- 2255: 4-C3H70, 3-(Me) 3C0, E], [-2256: 4-(Me) 2CHO, 3-(Me) 3CO, E], C-2257 :4-N02,3-(Me)3CO,E] , [-2258:4-N02,3-(Me)3 CO,Z],[-2259:3-F,3-(Me)3CO,E ], [-2260:3-F,3-(Me)3CO,Z],[-2261:3-01,3-(Μθ)3〇Ολε3 , [-2262:3-Cl,3-(Me) 3C〇,Z], C-2263:3-Br,3-(Me)3C〇,E], [ -2264:3-1,3-(Me)3CO,E ] , C -2265:3-Me , 3- (Me) 3CO, E], [-2266: 3-Me, 3-(Me) 3CO, Z], [-2267: 3-Et, 3-(Me) 3CO, E], 〔 -2268 :3-C3H7,3-(Me)3.CO,E] , [ -2269:3- (Me)2CH,3-(Me)3CO,E],[-2270:3-CF3,3-(Me ) 3CO, E], [-2271: 3-CF3, 3-(Me) 3CO, Z], [-2272: 3-C2F5, 3-(Me) 3CO, E], [-2273: 3-C3F7, 3-(Me)3CO,E ] , [ -2274 :3-(CF3 ) 2 CF, 3-(Me) 3 CO, E], [- 2275:3-(CF3)2CH,3-(Me)3CO , E], [-2276: 3-CHF2, 3-(Me)3CO, E], [-2277: 3-CHF2, 3-(Me) 3CO, Z], C-2278: 3-CH2F, 3- (Me)3 CO,E ] r [-2279:3-CH2F,3-(Me)3CO,Z], [-2280:3_CF3CH2,3-(Me)3CO,E], (-2281:3-MeO ,3-(Me)3CO,E] , [-2282:3-MeO,3-(Me)3CO,Z],[-2283:3-EtO,3-(Me)3CO,E],[-2284 :3-C3H7〇,3-(Me)3CO,E],[-2285:3-(Me)2CHO,3-(Me)3C〇,E] , C-2286:3-N02,3-(Me ) 3 CO,E], 96 320202 200901876 [-2287:2-F,3-(Me)3C O, E 3 , C-2288 : 2-C1,3-(Me) 3 CO, E ], [- 2289: 2-Br, 3-(Me) 3CO, E], [-2290: 2-I, 3-(Me)3CO, E], [-2291: 2-Me, 3-(Me)3CO, E), [ -2292: 2-Et, 3-(Me)3CO, E], [-2293: 2-C3H7,3-(Me)3CO,E], [ -2294:2-(Me)2CH,3-(Me)3CO,E],[- 2295:2-CF3,3-(Me)3CO, E], [-2296 : 2-Cz F5,3-(Me) 3 CO, E ], [- 2297:2-C3F7,3-(Me)3CO,E] , [-22 98 : 2-(CF3 2 CF, 3-(Me) 3 CO, E ], [-2299:2-(CF3)zCH,3-(Me)3CO,E], [-2300:2-CHF2,3-(Me)3CO , E], C-2301: 2-CH2F, 3-(Me)3 CO, E], [-2302: 2-CF3CH2, 3-(Me)3CO, E], [-2303: 2-MeO, 3 -(Me)3CO,E],[-2304:2-EtO,3-(Me)3CO,E], [-2255:2-C3H70,3-(Me)3 CO,E], [-2306: 2-(Me)2CHO,3-(Me)3CO,E) 2308:2,3-F2,3-(Me)3CO,E], 23X0:2,5-F2,3-(Me)3CO,E ], 2312:3,4-F2,3-(Me)3C〇,E], 2314:3,5-F2,3-(Me)3CO,E], 2316:2,3-C12,3-( Me)3CO,E], 2318:2,4-Cl2,3-(Me)3CO,E], 2320:2,5-CI2,3-(Me)3CO,E], 2322:2,6-Cl2 , 3-(Me)3CO, E], 2324:3,5-Cl2,3-(Me)3C〇,E], 2326:2,4-Br2,3-(Me)3CO,E], 2328: 2,6-Br2,3-(Me)3CO,E], 2330:3,5-Br2,3-(Me)3CO,E], 2332:2,4-Me2, 3-(Me)3CO,E], 2334:2,6-Me2,3-(Me)3CO,E], [-2307:2-NO2,3-(Me)3C0,E],[-[- 2309:2,4-F2,3-(Me) 3 CO, E],[-[-2311:2,6-F2,3-(Me)3COfE],[-[-2313:3r4-F2,3 -(Me)3CO,Z],[-[-2315:3,5-F2,3-(Me)3CO,Z],[-,[-2317:2,3-Cl2,3-(Me)3CO ,Z],[--· ,[-2319:2,4-CI2,3-(Me)3CO,Z],[-r [-2321:2,5-Cl2,3-(Me)3CO,z3 , [-, [-2323:3,4-Cl2,3-(Me)3CO,E],.[-,[-2325:2,3-Br2,3-(Me)3COfE],[-.[ -2327: 2,5-Br2,3-(Me)3CO,E],[-,[-2329:3,4-Br2,3-(Me)3CO,E],[-.[-2331:2 , 3-Me2,3-(Me)3COfE],[-,[-2333:2,5-Me2,3-(Me)3CO,E],[-C-2335:3,4-Me2,3- (Me)3CO, E], [- 97 320202 200901876 2336:3,5-Me2,3-(Me)3CO,E], [-2337:2,3-Et2,3-(Me)3CO,E] , [-2338: 2,4-Et2,3-(Me)3C〇,E], [-2339:2,5-Et2,3-(Me)3CO,E],[-2340:2,6- Et2,3-(Me)3CO,E],[-2341: 3,4-Et2,3-(Me)3CO,E],[-2342:3,5-Et2,3-(Me)3CO,E ], [-2343:2,3-(CF3)2,3-(Me)3CO,E], [-2344:2,4-(CF3)2,3-(Me)3CO,E], 〔 2345:2,5-(CF3)2,3-(Me)3CO,E],[-2346:2,6-(CF3)2,3-(Me)3CO,E), [-2347:3, 4- (CF3>2,3-(Me)3CO,E , [-2348:3,5-(CF3)2,3-(Me)3CO,E], [-2349:2,3-(CHF2)2,3-(Me)3CO,E], C-2350 :2,4-(CHF2) 2,3-(Me)3CO,E],[-2351:2,5-(CHF2)2,3-(Me)3C〇,E],[-2352:2, 6-(CHF2)2,3-(Me)3CO,E],[-2353:3, 4-(CHF2)2,3-(Me)3CO,E],[-2354:3,5-(CHF2 2,3-(Me)3CO,E], C-2355:2,3-(CH2F) 2,3-(Me)3CO,E],[-2356:2, 4-(CH2F)2, 3-(Me)3CO,E],[-2357:2,5-(CH2F)2,3-{Me)3CO,E] , [-2358:2,6-(CH2F)2,3-(Me ) 3CO, E), [-2359:3, 4-(CH2F)2,3-(Me)3CO,E] , [ -2360 : 3,5-(CH2 F) 2,3- (Me)3C〇 , E] , [-2361:2,3-(MeO)2,3-(Me)3C0,E ] , [-2362:2,4- (MeO)2;3-(Me)3CO,E] , [-2363: 2,5-(MeO)2,3-(Me)3CO,E],[- 2364:2, 6-(MeO)2,3-(Me)3 CO, E 〕 , 〔 -2365 :3, 4-(MeO)2,3-(Me)3CO,E],[-2366:3,5- (MeO) 2,3- (Me) 3 CO, E ] , [-2367:2, 3-(EtO)2,3-(Me)3CO,E], [-236.8 :2,4-(EtO) 2,3-(Me) 3CO, E], [- 2369:2,5-(EtO 2,3-(Me)3C〇,E 〕 , [ -2370:2,6-(EtO)2,3-(Me)3CO,E], C-2371:3, 4-(EtO)2, 3-(Me)3CO,E] , [-2372:3, 5- (EtO) 2,3-(Me)3CO,E],, [ -2373 :2-C1-3-F, 3-( Me) 3 CO, E], [- 2374: 2-Cl-4-F, 3-(Me)3C〇, E], [-2375: 2-C1-5-F, 3-(Me)3〇 〇,E), C -2376:2-Cl-6-F,3-(Me)3CO,E ] r [ -2377:3-C1-2-F,3-(Me)3CO,E] , 〔 -2378: 3-Cl-4-F, 3-(Me)3CO, E], [-2379: 3-Cl-5- 98 320202 200901876 F,. 3-(Me)3C〇, E], [- 2380 : 4-C1-2-F, 3-(Me) 3 CO, E], [-2381:4-C1-3-F,3-(Me)3CO,E] , [-2382:2-F -3-Me,3-(Me)3CO, E) , [-2383:2-F-4-Me,3-(Me)3CO,E ] , [ -2384:2-F-5-Me,3 -(Me)3CO,E],[- 2385:2-F-6-Me,3-(Me)3C0,E) , [-2386:3-F-2-Me,3-(Me)3CO, E], [-2387: 3-F-4-Me, 3-(Me)3C〇, E], [-2388:3-F-5-Me,3-(Me)3CO,E], [- 238 9:4-F-2-Me,3- (Me)3COfE] , [ -2390:4-F-3-

Me,3-(Me)3C〇,E] , [-2391:2-Cl-3-Me,3-(Me)3CO, E] , [-2392:2-Cl-4-Me,3-( Me) 3CO, E ] , [-2393: 2-Cl-5-Me, 3-(Me) 3CO, E], [- 2394: 2-Cl-6-Me, 3-(Me) 3CO, E] , [-2395:3-Cl-2-Me,3-(Me)3CO,E], [-2396:3-Cl-4-Me,3-(Me)3 CO,E], 〔 -2397: 3-Cl-5-Me,3-(Me)3CO,E],[-2398:4-Cl-2-Me,3-(Me)3 CO,E],[-2399:4-Cl-3 -Me,3-(Me)3CO,E] , [-2400:2-F-3-CF3,3-(Me)3CO,E] , [-2401:2-F-4-CF3,3-( Me)3CO,E], [-2402 :2-F-5-CF3,3-(Me) 3 CO, E],[- 2403:2-F-6-CF3,3-(Me)3CO,E ],[-2404:3-F-2-CF3,3-(Me) 3 CO, E], [-2405:3-F-4-CF3,3-(Me)3CO,E], [ -2406 :3-F-5-CF3,3-(Me)3CO,E],[-2407:4-F-2-CF3,3-(Me)3CO,E], (-2408:4-F-3 - CF3,3-(Me)3C〇,E ] , C -2409:2-Cl-3-CF3,3-(Me)3CO,E ],[- 2410:2-Cl-4-CF3,3- (Me)3CO,E], [-2411:2-Cl-5-CF3,3-(Me)3CO,E], [-2412:2-Cl-6-CF3,3-(Me)3C〇, E] Λ C-2413: 3-Cl-2-CF3, 3-(Me)3C〇, E 〕 , C -2414: 3-Cl-4-CF3, 3-(Me)3CO, E ]r[- 2415: 3-Cl-5-CF3, 3-(Me)3CO, E], [-2416:4-Cl-2-CF3,3-(Me)3CO, E], [-2417:4-Cl- 3-CF3,3-(Me)3CO,E], [-2418: 2-Me-3-CF3,3-(Me)3CO,E], [ -2419:2-Me-4-CF3,3-(Me)3CO,E ), [- 2420:2- Me-5-CF3,3-(Me)3C〇,E], [ -2421:2-Me-6-CF3,3-(Me)3CO,E], [-2422:3-Me-2-CF3 ,3-(Me)3CO,E] , [-2423:3-Me-4- 99 320202 200901876 CF3,3-(Me)3CO,E] , [ -2424:3-Me-5-CF3,3- <Me>3CO, E], [- 2425: 4-Me-2-CF3, 3-(Me)3CO, E], [ -2426:4"Me-3-CF3,3-(Me)3C〇 , E],. [2427:2-F-3-MeO,3-(Me)3CO,E], C-2428:2-F-4-

MeO, 3-(Me)3CO, E], [-2429: 2-F-5-MeO, 3-(Me)3CO, E], [_2430: 2-F-6-MeO, 3-(Me) 3CO, E ] , I > 2431: 3-F-2-MeO, 3-(Me) 3 CO, E], [- 2432: 3-F-4-MeO, 3-(Me)3CO, E], [-2433:3-F-5-MeO,3-(Me)3CO,E], [-2434:4-F-2-MeO,3-(Me)3CO,E], [-2435:4- F-3-MeO,3-(Me)3CO,E], [-2436:2-Cl-3-MeO,3-(Me)3CO,E], [-2437:2-Cl-4-MeO, 3-(Me>3CO,E], [-2238:2-Cl-5-MeO,3-(Me)3CO,E],[- 2439:2-Cl-6-MeO,3-(Me)3CO , E 〕 , [ -2440: 3-Cl-2-MeO, 3- (Me) 3CO, E], [-2441: 3-Cl-4-MeO, 3-(Me) 3CO, E], C- 2*442: 3-Cl-5-MeO, 3-(Me)3CO, E], [-2443: 4-Cl-2-MeO, 3-(Me)3CO, E], [- 2444:4- Cl-3-MeO,3-(Me)3C〇/E ) , [ -2445:2-Me-3-MeO,3-(Me)3CO,E],[-2446:2-Me-4-MeO ,3-(Me)3CO,E] ·[-2447:2-Me-5-MeO,3-(Me)3COrE ) , C -2448:2-Me-6-MeO,3-(Me)3CO, E 3 ,[- 2449:3-Me-2-MeO,3-(Me)3CO,E], [ -2450:3-Me'4-MeO,3-(Me)3CO,E],[-2451 :3-Me-5-MeO,3-(Me)3CO,E],[-2452:4-Me-2-MeO,3-(Me)3CO,E ] , [ -2453:4-Me-3 -MeO,3-(Me)3CO,E ] , C - 2454:H,2-F,E] , C-2455:4-F,2-F,E] , C-2456 :4-F,2-F,Z3 ,(-2457:4-Cl,2-F,E] , [-2458:4-Cl,2-F,Z] , [-2459:4-Br,2 -F,E], [-2460:4-1,2-F,E] , [-24 61: 4-Me, 2-F, E] , [-2462 : 4-Me, 2-F, Z ], C -2463:4-Et,2-F,E ] , [ -2464 : 4-C3H7,2-F,E ] , [-2465:4- (Me)2CH,2-F,E], [-2466: 4-CF3., 2-F, E], [-2467: 4-CF3, 2-F, Z], [-2468: 4-C2F5, 2-F, E], C-2469: 4-C3 F7,2-F, E ] , [-2470:4-(CF3>2CF,2-F,E], [-2471:4-(CF3)2CH,2-F,E], [- 2472:4-100 320202 200901876 CHF2,2-F,E], [-2473:4-CH2F,2-F,E], [-2474:4-CF3CH2r2-F,E], [-2475:4- MeO,2-F,E] , [-2476:4-MeO,2-F,Z) , [-2477:4-EtO,2-F,E],[-2478:4-C3H70,2-F , E], [-2479: 4-(Me) 2CHO, 2-F, E], [-2480: 4-NO2, 2-F, E], [-2481: 4-N〇2, 2-F , Z], [-2482: 3-Fr2-F, E], [-2483: 3-F, 2-F, Z], [-2484: 3-Cl, 2-F, E], [-2485 :3-Cl,2-F,Z], [-2486:3-Br,2-F,E], [-2487:3-1,2-F,E). , [-2488:3-Me , 2-F, E], [-2489: 3-Me, 2-F, Z], [-2490: 3-Et, 2-F, E], [-2491: 3-C3H7, 2-F, E], [-2492: 3-(Me) 2CH, 2-F, E], [-2493: 3-CF3, 2-F, E], [-2494: 3-CF3, 2-F, Z], [-2495: 3-C2F5, 2-F, E], [-2496: 3-C3F7, 2-F, E], [-2497:3 -(CF3)2CF,2-F,E], [-2498:3-(CF3)2CH,2-F,E], [-2499:3-CHF2,2-F,E], [-2500: 3-CHF2r2-F,Z],.[-2501:3-CH2F,2-F,.E], [-2502:3-CH2F,2-F,Z], [-2503:3-CF3CH2,2 -F,E], C-2504:3-Me0,2-F,E] , [-2505:3-MeO, 2-F, Z] , C-2506:3-EtO,2-F,E] , [-2507:3-C3H7O,2-F,E], [-2508:3-(Me)2CHO,2-F,E], [-2509:3-NO2,2-F,E], [ -2510:2-F,2-F,E], [-2511:2-C1,2-F,E], [-2512:2-Br,2-F,E],[-2513:2- 1,2-F,E], [-2514:2-Me,2-F,E], [-2515:2-Et,2-F,E], [ -2516:2-C3H?,2- F, E ] , [-2517:2- (Me)2.CH,2-F,E], [-2518:2-CF3,2-F,E],[-2519:2-C2F5,2- F,E], [-2520:2-C3F7,2-F,E] , [-2521:2-(CF3 ) 2 CF, 2-F, E] f [-2522:2-(CF3)2CH, 2-F, E], [-2523: 2-CHF2, 2-F, E], [-2524: 2-CH2F, 2-F, E], [-2525: 2-CF3CH2, 2-F, E ], [-2526: 2-MeO, 2-F, E], [-2527: 2-EtO, 2-F, E], [-2528: 2-C3H70, 2-F, E], [-2529 :2-(Me>2CHO,2-F,E], [-2530:2-NO2,2-F,E], [-2531:2,3 -F2,2-F,E], [-2532:2, 4-F2,2-F,E], [-2533:2,5-F2,2-F,E], [-2534:2, 6-F2,2-F,E], [-2535:3,4-F2,2-F,E], [-2536:3,4-F2,2-101 320202 200901876 F,Z],[- 2537 :3, 5-F2,2-F,E], [-2538 : 3,5-F2,2-F, Z], [- 2539:2,3-Cl2,2-F,E], -2540: 2,3-Cl2,2-F,Z], [-2541:2,4-Cl2,2-F,E], [-2542:2, 4-Cl2,2-F,Z], [-2543:2,5-Cl2,2-F,E], 〇2544:2,5-Cl2,2-F,Z], [-2545:2,6-Cl2,2-F,E], [-2546:3, 4-C12,2-F,E], [-2547:3,5-Cl2,2-F,E], [-2548:2,3-Br2,2-F,E] , [-2549:2,4-Br2,2-F,E], [-2550:2,5-Br2,2-F,E], [-2551:2,6-Br2,2-F,E ], [-2552:3,4-Br2,2-F,E], [-2553:3,5-Br2,2-F,E], [-2554:2,3-Me2,2-F, E] , [-2555:2,4-Me2,2-F,E] , [-2556:2,5-Me2,2-F,E] , [-2557:2,6-Me2,2-F , E], [-2558:3,4-Me2,2-F,E], [-2559:3,5-Me2,2-F,E] f [-2560:2,3-Et2,2- F,E] , [-2561:2,4-Et2,2-F,E] , [-2562:2,5-Et2,2-F,E] , C-2563 : 2,6-ETt2,2 -F, E], [-2564:3,4-Et2,2-F,E], [-2565:3,5-Et2,2-F,E], [-2566:2,3- (CF3 ) 2,2-F, E] [-2567:2,4-(CF3)2,2-F,E], [-2568:2,5-(CF3)2,2-F,E], [-2569:2,6-(CF3>; 2,2-F,E], [-2570:3,4-(CF3)2,2-F,E], [-2571:3,5-(CF3)2,2-F,E], [-2572:2,3-(CHF2)2,2-F,EJ r [ -2573:2,4-(CHF2)2,2-F,E ), (-2574:2,-5- (CHF2 ) 2,2-F,E ], [-2575:2,6-(CHF2)2,2-F,E], [-2576:3,4-(CHF2)2,2-F,E], [-2577:3,5-(CHF2)2,2-F,E], C-2578:2,3-(CH2F)2,2-F,E], [-2579:2,4-(CH2F ) 2,2-F,E ], [-2580:2,5- (CH2F) 2,2-F,E], C -2581:2,6- (CH2F)2,2-F,E ], [-2582:3,4-(CH2F)2,2-F,E], [-2583:3,5-(CH2F)2,2-F,E], [-2584:2,3- (Me 〇)2,2-F,E], [-2585:2,4-(MeO)2,2-F,E], [-2586:2,5- (Me〇) 2,2-F,E ],, (-2587:2,6-(MeO)2,2-F,E ], [-2588:3, 4- (Me〇)2,2-F,E], [-2589:3,5 -(MeO)2,2-F,E], [-2590:2,3- (Et〇)2,2-F,E], [-2591:2,4-(EtO)2,2-F , E], C -2592: 2,5- 102 320202 200901876 (EtO)2,2-F,E 〕 , [ -2593:2,6-(EtO)2,2-F,E], [-2594 :3,4- (EtO)2,2-F,E ] , C-2595:3,5-(EtO)2,2-FfE ) , C-2596:2-C1-3-F,2-F ,E] , [-2597:2-C1-4-F , 2-F, E], [-2598: 2-C1-5-F, 2-F, E], [-2599: 2-Cl-6-F, 2-F, E], [-2600: 3-C1-2-F,2-F,E] , [-2601:3-Cl-4-F,2-F,E] , C-2 602:3-Cl-5-F,2-F , E), [-2603: 4-C1-2-F, 2-F, E], [-2604: 4-Cl-3-F, 2-F, E], [-2605: 2-F- 3-Me,2-F,E], [-2606:2-F-4-Me,2-F,E], [-2607:2-F-5-Me,2-F,E], [ -2608: 2-F-6-Me, 2-F, E], [-2609: 3-F-2-Me, 2-F, E], [ -2610: 3-F-4-Me, 2 -F,E], [-2611:3-F-5-Me,2-F,E], [-2612:4-F-2-Me,2-F,E], [-2613:4- F-3-Me,2-F,E], [-2614:2-Cl-3-Me,2-F,E], [-2615:2-

Cl-4-Me,2-F,E], [ -2616:2-Cl-5-Me,2-F,E] , C-2B17:2-C1-6-

Me, 2-F, E], [ -2618: 3-Cl-2-Me, 2-F, E ], [-2619: 3-Cl-4-Me, 2-F, E], [-2620 :3-Cl-5-Me,2-F,E], [-2621:4-Cl-2-Me,2-F,E], [-2622:4-Cl-3-Me,2-F , E], [-2623: 2-F-3-CF3, 2-F, E], [-2624: 2-F-4-CF3, 2-F, E], [ -2 625:2-F -5-CF3,2-F,E ) , [ -2626:2-F-6- CF3-,2-F,E],C-2627:3-F-2-CF3,2-F,E] , [-2628 : 3-F-4-CF3,2-F, E], [-2629:3-F-5-CF3,2-F,E], [-2630:4-F-2-CF3 , 2-F, E], [-2631: 4-F-3-CF3, 2-F, E], [-2632: 2-Cl-3-CF3, 2-F, E], [-2633: 2-CI-4-CF3,2-F,E], [-2634:2-Cl-5-CF3,2-F,E], C-2635:2-C1-6-CF3,2-F, E] , (-2636:3-Gl-2-CF3,2-F,E] , [-2637:3-Cl-4-CF3,2-F,E] , [-2638:3-Cl-5 -CF3,2-F,E], [-2639:4-Cl-2-CF3,2-F,E], [-2640:4-Cl-3-CF3,2-F,E], [- 2641: 2-Me-3-CF3, 2-F, E], '[-2642: 2-Me-4-CF3, 2-F, E], [-2643: 2-Me-5-CF3, 2 -F,E 〕,[- 2644:2-Me-6-CF3,2-F,E ] , [ -2645:3-Me-2-CF3,2-F,E ],[- 2646:3- Me-4-CF3,2-F,E 3 ,[ -2647:3-Me-5-CF3,2-F,E],[- 103 320202 200901876 2648:4-Me-2-CF3,2-F , E ] , [ -2649:4-Me-3-CF3,2-F,E ], [- 2650:2-F-3-MeO,2-F,E] , [-2651: 2-F-4-MeO, 2-F, E], [-2652: 2-F-5-Me〇, 2-F, E], [1-2653:2-F-6- Me〇, 2-F, E], [ -2654:3-F-2-

MeO, 2-F, E], [ -2 655:3-F-4-MeO, 2-F, E 3 , C-2656: 3-F-5-MeO, 2-F, E], [- 2657: 4-F-2-MeO, 2-F, E], [-2658: 4-F-3-MeO, 2-F, E], [-2659: 2-Cl-3-MeO, 2- F, E ] , [-2660: 2-Cl-4-MeO, 2-F, E], [- 2661: 2-Cl-5-MeO, 2-FrE] 2663: 3-Cl-2-MeO, 2-F,E ) 2665:3-Cl-5-MeO,2-F,E ] 2667:4-Cl-3-MeO,2-F,E ] 2669:2-Me-4-MeO,2- F,E 〕 2671:2-Me-6-MeO,2-F,E] 2673:3-Me-4-Me〇,2-F,E] 2675:4-Me-2-MeO,2-F , E ] [-2662:2-Cl-6-MeO,2-F,E ],[-[-2664:3-Cl-4-MeO,2-F,E ),-[-2666:4- Cl-2-MeO,2-F,E],[-[-2668:2-Me-3-MeO,2-F,E],[-[-2670:2-Me-5-MeO,2- F, E], [-[-2672:3-Me-2-MeO,2-F,E], [-[-2674:3-Me-5-MeO,2-F,E 3 ,[- 〔 -2676: 4-Me-3-MeO, 2-F, E], [-2677: H, 2-C1, E], [-2678: 4-F, 2-C1, E], [-2679: 4-F, 2-C1, Z], [-2680: 4-Cl, 2-Cl, E], [-2.681: 4-C1, 2-C1, Z], [-2682: 4-Br, 2 -

ClrE] r [-2683:4-1,2-Cl,E], [-2684:4-Me,2-C1,E], [-2685:4-Me,2-Cl,Z], [- 2686: 4-Et, 2-Cl, E], [-2687: 4-C3H7, 2-Cl, E], [-2688: 4-(Me) 2CH, 2-Cl, E], [-2689: 4-CF3,2-C1,E],C-2690:4-CF3,2-C1,Z], C-2691:4-C2F5,2-C1,E) , [-2692 : 4-C3 F7, 2-C1, E], [-2693:4-(CF3)2CF,2-C1,E] , (-2694 : 4-(CF3 ) 2 CH, 2-C1, EJ , [-2695:4-CHF2 , 2-Cl, E], [ -2696: 4-CH2F, 2-C1, E], [ -2697: 4-CF3CH2, 2-Cl, E 3 , [ -2698 : 4-MeO, 2-Cl, E ] , C -2699: 4-MeO,2- C1,Z] , [-2700:4-Et0,2-C1,E] , C-2701:4-C3H70,2-C1,E],[- 2702: 4-(Me)2CHO, 2-Cl, E], [-2703: 4-N02, 2-ClrE], [-2704: 4-104 320202 200901876 N〇2, 2-C1, Z], [ -2705: 3-F, 2-C1, E], [-2706: 3-F, 2-C1, Z], [-2707: 3-Cl, 2-Cl, E], [-2708: 3- Cl, 2-Cl, Z], [-2709: 3-Br, 2-C1, E], [-2710: 3-I, 2-C1, E], [-2711: 3-Me, 2-C1 , E], [-2712: 3-Me, 2-Cl, Z], [-2713: 3-Et, 2-Cl, E], [-2714: 3-C3H7, 2-Cl, E], [ -2715: 3-(Me)2CH, 2-C1, E], C-2716: 3-CF3, 2-C1, E], [-2717: 3-CF3, 2-C1, Z], [-2718 :3-C2F5,2-C1,E],[-2719:3-C3F7,2- C1,E], [-2720:3-(CF3)2CF,2-Cl,E], [-2721:3-(CF3)2CH,2-Cl,E], [-2722:3-CHF2,2 -Cl,E] , [-2723:3-CHF2,2-Cl,Z], [-2724:3-CH2F,2-C1,E], [-2725:3-CH2F,2-Cl,Z] , [ -2726:3-CF3CH2,2-

Cl, E], [-2727: 3-MeO, 2-Cl, E], [-2728: 3-MeO, 2-Cl, Z], [-2729: 3-EtO, 2-Cl, E], [-2730:3-C3H7O,2-Cl,E]/[-2731:3-(Me)2CHO,2-C1,E], C -2732:3-N〇2,2-C1,E] f C -2133:2-F,2-

Cl, E], [-2734: 2-Cl, 2-Cl, E], [-2735: 2-Br, 2-Cl, E], [-2736: 2-I, 2-Cl, E], [-2737: 2-Me, 2-Cl, E]., [-2738: 2-Et, 2-Cl, E], [-2739: 2-C3H-7, 2-Cl, E), [- 2740: 2-(Me)2CH, 2-Cl, E], [-2741: 2-CF3, 2-C1, E], [-2742: 2-C2F5, 2-Cl, E], [-2743: 2-C3F7,2-Cl,E], [-.2744:2-(CF3)2CF,2-'Cl,E], [-2745:2-(CF3)2CH,2-Cl,E], -2746: 2-CHF2, 2-Cl, E], [-2747: 2-CH2F, 2-Cl, E], [-2748: 2-CF3CH2, 2-Cl, E], [-2749:2- MeO, 2-Cl, E], [-2750: 2-EtO, 2-C1, E], [-2751: 2-C3H70, 2-C1, E], [-2752: 2-(Me)2CHO, 2-Cl, E], [-2753: 2-N02, 2-Cl, E], [-2754: 2, 3-F2, 2-Cl, E], [-2755: 2, 4-F2, 2 -C1,E] , C-2756:2,5-F2,2-Cl,E] , [-2757:2,6-F2,2-C1,E], [-2758:3,4-F2f2- Cl, Ej, [-2759:3,4-F2,2-C1,Z], [-2760:3,5-F2,2-C1,E],[-2761:3, 5-F2,2- Cl,Z], [-2762:2,3-Cl2,2-Cl,E], C-2763:2,3-Cl2,2-ClrZ], [ -2764:2,4-Cl2,2-C1 , E 3 , [- 105 320202 200901876 2765: 2, 4-Cl 2 , 2-Cl, Z] , C-2766: 2, 5-Cl 2 , 2-ClfE] , [-2767: 2, 5-C12, 2 -C1,Z) , [-2768:2,6-Cl2,2-Cl,E ] , C-2769 : 3,4-Cl 2,2-Cl,E], [-2770:3,5-Cl2,2-Cl,E], [-2771:2,3-Br2,2-Cl,E], [-2772:2,4 -Br2,2-Cl,E], C-2773:2,5-Br2,2-C1,E], [-2774:2,6-Br2,2-C1,E], [-2775:3, 4-Br2,2-Cl,E], [-2776: 3,5-Br2,2-Cl,E], [-2777:2,3-Me2,2-Cl,E], [-2778:2 , 4-Me2,2-Cl,E], [-2779:2,5-Me2,2-Cl,E] r [-2780:2,6-Me2,2-C1,E], [-2781: 3,4-Me2,2-Cl,E ] , [-2782:3,5-Me2,2-Cl,E], C-2783:2,3-Et2,2-Cl,E],[-2784 : 2,4-Et2,2-Cl,E], [-2785:2,5-Et2,2-Cl,E], [-2786:2,6-Et2,2-Cl,E], [- 2787:3,4-Et2,2-C1,E], [-2788:3,5-Et2,2-C1,E], [-2789:2,3-(CF3)2,2-Cl,E ], [.-2790:2, 4-(CF3)2,2-Cl,E], [-2791:2,5-(CF3)2,2-Cl,E], [-2792:2,6 -(CF3)2,2-Cl,E ] , [-2793:3, 4-{CF3 )2,2-Cl,E ] , [-2794:3,5-(CF3 ) 2,2-Cl, E ] , [-2795:2,3-(CHF2) 2,2-Cl,E] , [-2796:2,4-(CHF2) 2,2-Cl,E] , [-2797:2,5 -(CHF2)2,2-Cl,E] , [-2798:2,6-(CHF2)2,2-Cl,E3, [-2799:3,4-(GHF2)2,2-Cl,E ), [-2800:3,5-(CHF2)2/2-Cl,E] , [-2801:2,3-(CH2F)2,2-Cl,E] , [-2802:2,4- (CH2F)2,2-Cl,E] , [-2803:2,5-(CH2F)2,2-Cl,E] , [-2804:2, 6- (CH2F)2,2-C1,E] , [-2805:3,4-(CH2F)2,2-Cl,E] , [-2806:3,5-(CH2F)2,2-C1,E r [-2807:2,3-(MeO)2,2-ClfE] , [-2808:2,4-(MeO)2,2-Cl,E], [-2809 :2,5-(MeO 2,2-C1, E 3 , [-2810:2,6-(MeO)2,2-Cl,E ] , [-2811:3,4-(MeO)2,2-Cl,E], [-2812:3,5-(MeO)2,2-Cl,E], [-2813:2,3-(Et〇)2,2-C1, E],[-2814:2,4-( EtO)2,2-Cl,E ] , (-2815:2,5-(EtO)2,2-Cl,E ] , [-2816:2,6-(Et〇)2,2-C1,E ], [-2817:3,4-(Et〇)2,2-Cl,E], [-2818:3,5-106 320202 200901876 (Et〇)2,2-C1,E], [-2819 :2-Cl-3-F,2-Cl,E] , [-2820:2-Cl-4-F,2-C1,E], ( -2821:2-Cl-5-F,2-Cl , E ) , C -2822: 2-C1-6-F, 2-C1, E], [-2823: 3-Cl-2-F, 2-Cl, E], [-2824: 3-C1- 4-F,2-C1,E] ,· C-2825:3-Cl-5-F,2-Cl,E. ] , [ -2826 : 4-C1-2-F, 2-C1, EJ , [- 2827: 4-Cl-3-F, 2-Cl, E], [-2828: 2-F-3-Me, 2-Cl, E], [-2829: 2-F-4-Me, 2-Cl,E ] , [-2830:2-F-5-Me,2-C1,E ) , [-2831:2-F-6-

Me, 2-Cl, E], [-2832: 3-F-2-Me, 2-Cl, E], [-2833: 3-F-4-Me, 2-C1, E], [-2834 :3-F-5-Me,2-Cl,E], [-2835:4-F-2-Me,2-Cl,E], C-2836:4-F-3-Me,2-Cl , E ] , [-2837: 2-Cl-3-Me, 2-Cl, E] / C- 2838: 2-Cl-4-Me, 2-Cl, E], [-2839: 2-Cl- 5-Me,2-Cl,E] /C - 2840:2-Cl-6-Me,2-Cl,E], [-2841:3-Cl-2-Me,2-CI,E] tc - 2842: 3-Cl-4-Me, 2-Cl, E], [-2843: 3-Cl-5-Me, 2-Cl, E] fc - 2844: 4-Cl-2-Me, 2-Cl , E 〕, [-2845: 4-Cl-3-Me, 2-Cl, E] r 〔- 2846: 2-F-3-CF3, 2-Cl, E ], C -2847:2-F- 4-CF3,2-Cl,E 3 t [- 2848:2-F-5-CF3,2-Cl,E], [-2849:2-F-6-CF3,2-Cl,E] tc - 2850: 3-F-2-CF3, 2-Cl, E], [-2851: 3-F-4-CF3, 2-Cl, E] } [- 2852: 3-F-5-CF3,2- Cl,E 〕, [-2853:4-F-2-CF3,2-Cl,E] rc - 2854:4-F-3-CF3,2-Cl,E], [-2855:2-Cl- 3-CF3,2-Cl,E ] r [- 2856:2-Cl-4-CF3f2-Cl, E3, [-2857:2-Cl-5-CF3,2-Cl,E] t [- 2858: 2-Cl-6-CF3,2-Cl,E], [-2859:3-Cl-2-CF3,2-Cl,E] r c- 2860:3-Cl-4-CF3,2-Cl, E ], [-2861:3-C1-5-CF3,2_C1,E] r c- 2862:4-Cl-2-CF3,2-Cl,E ], [-2863:4-C l-3-CF3,2-Cl,E ] r [- 2864:2-Me-3-CF3,2-Cl,E], [-2865:2-Me-4-CF3,2-Cl,E ] r [- 2866:2-Me-5-CF3,2-Cl,E ], [-2867:2-Me-6-CF3,2-Cl,E] t [- 2868:'3-Me-2- CF3,2-Cl,E], [-28 69:3-Me-4-CF3,2-Cl,E] t c- 107 320202 200901876 2870:3-Me-5-CF3,2-Cl,E ] 2872: 4-Me-3-CF3,2-C1,E] 2874:2-F-4-MeO,2-Cl,E] 2876:2-F-6-MeO,2-Cl,E] 2878: 3-F-4-MeO,2-Cl,E] 2880:4-F-2-MeO,2-Cl,E] 2882:2-Cl-3-MeO,2-Cl,E] 2884:2- Cl-5-MeO, 2-Cl, E] 2886: 3-Cl-2-Me〇, 2-Cl, E] 2888: 3-Cl-5-MeO, 2-Cl, E] 2890: 4-Cl -3-MeO, 2-Cl, E] 2892: 2-Me-4-MeO, 2-Cl, E] 2894: 2-Me-6-MeO, 2-Cl, E] 2896: 3-Me-4 -MeO,2-Cl,E] 2898:4-Me-2-MeO,2-Cl,E] [-2871:4-Me-2-CF3,2-Cl,E] [-2873:2-F -3-MeO,2-Cl,E ] [-2875:2-F-5-MeO,2-Cl,E] (-2877:3-F-2-MeO,2-Cl,E ] [-2879 :3-F-5-MeO,2-Cl,E] [-2881:4-F-3-Me〇,2-Cl,E] [-2883:2-Cl-4-MeO,2-Cl, E ] [-2885: 2-Cl-6-MeO, 2-Cl, E] [-2887: 3-Cl-4-MeO, 2-Cl, E] [-2889: 4-Cl-2-MeO, 2-Cl,E ] [-2891:2-Me-3-MeO,2-Cl,E] [-2893:2-Me-5-MeO,2-Cl,E] [-2895:3-Me- 2-MeO, 2-Cl, E 〕 [-2897: 3-Me-5-MeO, 2-Cl, E] C- [- [ 〔- 〔-[- [- [- c [-2899:4-Me-3-MeO, 2-Cl , E], [-2900: H, 2-CF3, E], C-2901: 4-F, 2-CF3/ [-2902: 4-F, 2-CF3, Z] [-2903: 4-Cl , 2-CF3 , E ] , C-2904 : 4-C1,2-CF3 , Z ] , [-2905:4-Br,2-CF3,E], [-2906:4-I,2-CF3, E], [-2907: 4-Me, 2-CF3, E], [-2908: 4-Me, 2-CF3, Z], [-2909: 4-Et, 2-CF3, E], [- 2910:4-C3H7,2-CF3,E], [-2911:4-(Me)2CH,2-CF3,E], [-2912: 4-CF3,2-CF3, E], C-2913: 4-CF3,2-CF3,Z3, C-2914 : 4-C2 Fs , 2-CF3 , E ] , [-2915:4- C3F7,2-CF3 ,E ] , ( -2916:4-(CF3 ) 2CF, 2-CF3, E], [-2917:4-(CF3), 2CHf 2-CF3, E], [ -2918:4-CHF2,2-CF3,E ], [ -2919:4-CH2F, 2-CF3, E], C-2920: 4-CF3CH2, 2-CF3, E], [-2921: 4-MeO, 2-CF3, E], [-2922: 4-Me〇, 2-CF3, Z], [-2923:4-EtO,2-CF3,E], [- 108 320202 200901876 2924:4-C3H70,2-CF3,E], [-2925:4-(Me)2CHO,2-CF3 , E], [-2926: 4-N〇2, 2-CF3, E], [-2927: 4-N02, 2-CF3, Z], [-2928: 3-F, 2-CF3, E] , [-2929: 3-F, 2-CF3, Z], [-2930: 3-Cl, 2-CF3, E], [-2931: 3-Clf2-CF3, Z 3, [-2932:3-Br,2-CF3fE ] f [-2933:3-1,2-CF3,E].,[-2934.:3-Me,2-CF3,E],[-2935 :3-Me,2-CF3,Z], [-2936:3-Et,2-CF3,E), C-2937: 3-C3 H7,2-CF3, E), [-2938:3- ( Me) 2CH, 2-CF3, E], [-2939: 3-CF3, 2-CF3, E], [-2940: 3-CF3, 2-CF3, Z], [-2941: 3-C2F5, 2 -CF3, E], [-2942: 3-C3F7, 2-CF3, E], [-2943: 3-(CF3)2CF, 2-CF3, E], [-2944:3, (CF3)2CH, 2-CF3, E], [-2945: 3-CHF2, 2-CF3, E], [-2946: 3-CHF2, 2-CF3, Z], [-2947: 3-CH2F, 2-CF3, E ], C-2948: 3-CH2F, 2-CF3, Z], [-294 9:3-CF3 CH2,2-CF3,E], [-2950:3-MeO,2-CF3,E], -2951: 3-MeO, 2-CF3, Z], [-2952: 3-EtO, 2-CF3, E], [-2953: 3-C3H70, 2-CF3, E], [-2954: 3- (Me)2CHO,2-CF3,E], [-2955:3-N〇2,2-CF3,E],[ -2956:.2-F,2-CF3,E],[,2957:2 -Cl,2-CF3,E], [-2958:2-Br,2-CF3,E], [-2959:2-I,2-CF3,E], [-2960:2-Me,2- CF3,E], C-2961:2-Et,2-·CF3,E], C-2 962:2-C3H-7,2-CF3,e3 r [-2963:2- (Me) 2 CH, 2-CF3, E], C-2964: 2-CF3, 2-CF3, E], [-2965: 2-C2 F5, 2-CF3, E], [-2966: 2-C3F7, 2-CF3, E] , [ -2967:2-(CF3 )2CF,2-CF3 ] , [-2968:2- (CF3 )2CH,2-CF3 ,E ] , [ -2969:2-CHF2,2-CF3 ,E], C -2970:2-CH2F,2-CF3,E] , [-2971:2-CF3CH2,2-CF3,E] , [-2972 :2-MeO, 2-CF3fE] , [-2973:2-EtO , 2-CF3, E], [-2974: 2-C3 H·, 0, 2-CF3, E], [-2975: 2-(Me)2CHO, 2-CF3., E], C-297 6 : 2-N02,2-CF3 , E ], [- 2977:2,3-F2,2-CF3 ,E) , [-2978 : 2,4-F2,2-CF3 , E) , [-2979: 2,5-F2,2-CF3,E] , [ -2980:2,6-F2,2-CF3 ,E ] , C -2981: 3,4-F2,2- 109 320202 200901876 CF3,E) f [-2982: 3,4-F2,2-CF3,Z], [-2983: 3,5-F2,2-CF3, E), [-2984:3,5-F2,2-CF3, Z] , C-2985 : 2,3-Cl2,2-CF3 , E] , [-2986:2,3-C12,2-CF3,Z] , [-2987:2, 4-Cl2,2-CF3,E ], [-2988 : 2f 4-Cl2, 2-CF3, Z], [-2989: 2, 5-Cl2, 2-CF3, E], [-2990: 2, 5-Cl2, 2-CF3, Z ], [-2991:2,6-Cl2,2-CF3,E], [-2992:3,4-Cl2,2-CF3,E], c-2993:3,5-Cl2,2-CF3, E], [-2994: 2,3-Br2,2-CF3,E), (- 2995:2,4-Br2,2-CF3,E], [-2996:2,5-Br2,2-CF3 , E 〕, c - 2997: 2,6-Br2,2-CF3,E], [-2998:3,4-Br2,2-CF3,E], c - 2999:3,5-Br2,2- CF3, E 〕, 〔-3000:2,3-Me2, 2-CF3rE 〕, c - 3001: 2, 4-Me2,2-CF3,E], [-3002:2,5-Me2,2-CF3,E], [- 3003:2,6-Me2,2 -CF3,E 〕, [-3004:3, 4-Me2,2-CF3,.E] r (- 3005:3,5-Me2,2-CF3,E ], [-3006:2,3-Et2 , 2-CF3, E], [- 3007:2,4-Et2,2-CF3,E], [-3008:2,5-Et2,2-CF3,E], [- 3009:2,6- Et2,2-CF3,E], [-3010:3,4-Et2,2-CF3,E], [- 3011:3,5-Et2,2-CF3,E ], [-3012:2,3 -(CF3)2,2-CF3,E], [- 3013:2., 4- (CF3 )2,2-CF3,E], [-3014:2,5-(CF3)2.,2- CF3, E], [- 3015:2, 6-(CF3)2,2-CF3,E], [-3016:3r4-(CF3)2,2-CF3,E], [- 3017:3,5 -(CF3)2,2-CF3,E], [-3018:2,3-(CHF2)2,2-CF3,E], [- 3019:2,4-(CHF2)2,2-CF3, E3 , [-3020 : 2,5-(CHF2 ) 2,2-CF3 , E), 3021:2, 6-(CHF2 ) 2,2-CF3 ,E) , [-3022 : 3,4-(CHF2 ) 2 λ 2-CF3 , E], [-3023:3,5-(CHF2 ) 2,2-CF3 ,E] , [-3024 : 2,3-(CH2 F) 2,2-CF3 , E) , [-3025:2,4-(CH2F)2,2-CF3,E], [-3026:2,5-(CH2 F) 2,2-CF3, E],[-3027:2,6- (CH2F)2,2-CF3,E] f [-3028 : 3,4-(CH2 F) 2,2-CF3 , E], [-3029:3,5-(CH2F)2,2-CF3, E] , [-3030 : 2,3-(MeO) 2,2-CF3 , E] , [-3031:2,4-(MeO)2,2-CF3/E], [-3032 :2,5-(MeO) 2,2-CF3 , E ), [- 110 320202 200901876 3033:2, 6-(MeO)2,2-CF3,Ε] 3035:3,5-(MeO)2,2-CF3,E] ' 3037:2,4-(EtO)2,2-CF3,E] 3039: 2,6-(EtO)2,2-CF3,E] 3041:3,5-(EtO)2,2-CF3,E 3 3043:2-Cl-4-F,2-CF3,E], 3045 :2-Cl-6-F,2-CF3,E], 3047:3-Cl-4-F,2-CF3,E, 3049:4-Cl-2-F,2-CF3,E], 3051 :2-F-3-Me,2-CF3,E 3 , 3053:2-F-5-Me,2-CF3,E], 3055:3-F-2-Me,2-CF3,E], 3057: 3-F-5-Me, 2-CF3, E] r 3059: 4-F-3-Me, 2-CF3, E], 3061: 2-Cl-4-Me, 2-CF3, E] , 3063: 2-Cl-6-Me, 2-CF3, E], 3065: 3-Cl-4-Me, 2-CF3, E], 3067: 4-Cl-2-Me, 2-CF3, E ], 3069: 2-F-3-CF3, 2-CF3, E], 3071: 2-F-5-CF3, 2-CF3, E) 3073: 3-F-2-CF3, 2-CF3, E ], 3075: 3-F-5-CF3, 2-CF3, E 3 , 3077: 4-F-3-CF3, 2-CF3, E], 3D79: 2-Cl-4-CF3, 2-CF3, E]( 3081:2-Cl-6-CF3,2-CF3,E], [-3034:3,4-(MeO)2,2-CF3,E],[-[-3036:2,3- (EtO)2,2-CF3,E],[-[-3038:2,5-(EtO)2,2-CF3,E] , C- [-3040:3, 4-(EtO)2,2 -CF3, E], [-[-3042:2-Cl-3-F,2-CF3,E], C -[-3044:2-Cl-5-F,2-CF3,E],[- [-3046: 3-Cl-2-F, 2-CF3, E], [-[-3048:3-Cl-5-F,2- CF3, E 3 , [- [-3050:4-Cl-3-F,2-CF3,E], [-[-3052:2-F-4-Me,2-CF3,E], C - 〔 -3054: 2-F-6-Me, 2-CF3., E], [-[-3056:3-F-4-Me,2-CF3,E],[-[-3058:4-F- 2-Me,2-CF3,E],-[-3D60:2-Cl-3-Me,2-CF3,E],[-[-3062:2-Cl-5-Me,2-CF3,E ), [-[-3064:3-Cl-2-Me,2-CF3,E ] , C - [-3066:3-Cl-5-Me,2-CF3,E], [-[-3068: 4-Cl-3-Me,2-CF3,E],[-[-3070:2-F-4-CF3,2-CF3,E],[-[-3072:2-F-6-CF3, 2-CF3,E],[-[-3074:3-F-4-CF3,2-CF3,E],[-[-3076:4-F-2-CF3,2-CF3,E], -[-3078:2-Cl-3-CF3r2-CF3,E], [-[-3080:2-Cl-5-CF3,2-CF3,E],[-[-3082:3-Cl-2 -CF3,2-CF3,E]r [- 111 320202 200901876 3083:3-Cl-4-CF3,2-CF3,Ε], [-3084 : 3-Cl-5-CF3,2-CF3 , E ] , [- 3085: 4-Cl-2-CF3, 2-CF3/E), [-3086: 4-Cl-3-CF3, 2-CF3, E]., [- 3087: 2-Me-3- CF3,2-CF3,E], [-3088 :2-Me-4-CF3,2-CF3, E ],[- 3089:2-Me-5-CF3,2-CF3 ,E] , [-3090 :2-Me-6-CF3,2-CF3, E],[-3091:3-Me-2-CF3,2-CF3,E], [-3092 : 3-Me-4-CF3,2-CF3 , E ], [- 3093 : 3-Me-5-CF3,2-CF3 , E ] , [-3094 : 4-Me-2-CF3,2-CF3 , E], [-3 95:4-Me-3-CF3,2-CF3,E], [-3096: 2-F-3-MeO, 2-CF3, E], [-3097:2-F-4-MeO,2- CF3, E], [-3098: 2-F-5-MeO, 2-CF3, E], [- 3099: 2-F-6-MeO, 2-CF3, E], [-3100: 3-F -2-MeO, 2-CF3, E], [- 3101: 3-F-4-MeO, 2-CF3, E], [-3102: 3-F-5-MeO, 2-CF3, E], [- 3103 : 4-F-2-MeO, 2-CF3 , E ] , C -3104 : 4-F-3-MeO, 2-CF3 , E ], [-3105: 2-Cl-3-MeO, 2-CF3, E], C-3106: 2-Cl-4-MeO, 2-CF3, EJ, [-3107: 2-Cl-5-MeO, 2-CF3, E), [-3108:2- Cl-6-MeO,2-CF3, E] r [- 3109:3-Cl-2-MeO,2-CF3,E], [-3110:3-Cl-4-MeO, 2-CF3, E] , [-3111:3-Cl-5-MeO,2-CF3,E], [-3112:4-Cl-2-MeO,2-CF3,E], [-3113:4-Cl-3-MeO ,2-CF3, E], C-3114:2-Me-3-MeO,2-CF3> E] r[-3115:2-Me-4-MeO,2-CF3,EJ, C-3116:2 -Me-5-MeO, 2-CF3, E), C-3117: 2-Me-6-MeO, 2-CF3, E], [-3118: 3-Me-2-MeO, 2-CF3, E ], [-3119: 3-Me-4-MeOr2-CF3, E], [-3120: 3-Me-5-MeO, 2-CF3, E] r (- 3121: 4-Me-2-MeO, 2-CF3,E],[-3122:4-Me-3-MeO,2-CF3,E]f[-3123:H,2-MeO,E], [-3124:4-F,2-MeO ,E] , [-3125:4-F,2-MeO,Z], [-3126:4-Cl, 2-MeO, E],. [-3127 : 4, C1, 2-MeO, Z], C -3128: 4-Br, 2-MeO, E], [-3129:4-1f2-MeO, E] , [-3130:4-Me,2-MeO,E], [-3131:4-Me,2-Me〇,Z], [-3132:4-Et,2-MeO,E], [-3133 :4-C3H7,2-MeO,E] , [-3134:4-(Me)2 CH,2-MeO,E) , (-3135:4-CF3,2-MeO,E], 112 320202 200901876 C -3136: 4-CF3,2-MeO,Z], [-3137:4-C2F5,2-MeO,E], [-3138:4-C3F7,2-MeO,E], [-3139:4- (CF3)2CF,2-MeO,E ] [-3140:4- (CF3)2CH,2-Me〇,E], [ -3141:4-CHF2,2-MeO,E ] r [ -3142:4 - CH2F, 2-MeO, E], .[-3143 : 4-CF3 CH2,2-MeO, E ] , [-3144 : 4-MeO, 2-

MeO, E], [-314 5:4-MeO, 2-MeO, Z], [-3146:4-EtO, 2-Me〇, E], [-3147:4-C3H70,2-Me0,E ], 〔一3148:4-(Me)2CHO,2-MeO,E],[一3149:4-N02,2-MeO,E], [-3150:4-N02,2-MeO,Z3, [ -3151:3-F,2-MeO,E ) , [ -3152:3-F,2-MeO,Z] , [ -3153:3-C1r2-MeO,E ],[- 3154:3-Cl, 2-MeO,Z ] , [-3155:3-Br,2-MeO,E ] , [-3156:3-1,2-

Me〇, E], [-3157:3-Me,2-MeO,E], [-3158:3-Me,2-MeO,Z], [- 3159:3-Et,2-MeO,E ] , [ -3160:3-C3H7,2-MeO,E ] , C -3161:3- (Me)2CH,2-lXIeO,E],[ -3162 : 3-CF3,2-MeO, E ] , [ -3163 : 3-CF3,2-

MeO,Z] , [-3164 :3-C2 F5,2-ΜθΟ,Ε), [-3165 : 3-C3 F7,2-MeO, E], [-3166:3-(CF3 )2CF,2- MeO, E], [-3167: 3-(CF3) 2 CH, 2-MeO, E], [-3168: 3-CHF2, 2-MeO, E], [-3169: 3-CHF2, 2-MeO , Z ] , C-3170: 3-CH2F, 2-MeO, E], [-3171: 3-CH2 F, 2-MeO, Z], [-3172: 3-CF3CH2, 2-MeO, E], [-3173: 3-MeO, 2-MeO, E], [-3174: 3-MeO, 2-MeO, Z], [-3175: 3-Et〇, 2-Me〇, E], C-3176 :3-C3H7〇,2-MeO,E 3 , C-3177:3-(Me)2CHO,2-MeO,E], [-3178:3-N02,2-MeO,E], [-3179: 2-F,2-

MeO, E], [-3180: 2-Cl, 2-MeO, E], [-3181: 2-Br, 2-MeO, E], [-3182: 2-I, 2-Me〇, E] , [-3183:2-Me,2-MeO,E], [-3184:2-Et,2-

MeO, E] , [-3185: 2-C3H7, 2-MeO, E], [-3186: 2-(Me) 2CH, 2-MeO, E], [-3187: 2-CF3, 2-MeO, E] , [-3188:2-C2F5,2-MeO,E] f [-3189:2-C3F7,2-Me〇,E], [ -3190:2-(CF3 )2CF,2-MeO,E ],, ( -3191:2-(CF3)2CH,2-Me〇,E], [ -3192:2-CHF2,2-MeO,E ], [ -3193:2- 113 320202 200901876 CH2F,2-MeO , E], [-3194: 2-CF3CH2, 2-MeO, E], C-3195: 2-MeO, 2-

Me〇, E], [-3196: 2-EtO, 2-MeO, E], [-3197: 2-C3H7〇, 2-MeO, E], [-3198: 2-(Me)2CHO, 2- MeO, E 〕 , 〔 -3199:2-N02,2-MeO,E ],[- 3200:2,3-F2,2-MeO,E] , [-3201:2,4-F2,2-MeO , E] , [-3202:2,5-F2,2-MeO,E ] , C -3203:2,6-F2,2-MeO,E ] , [ -3204 : 3, 4-F2,2-

MeO, E] , [-3205:3, 4-F2,2-MeO,z] , [-3206: 3,5-F2 , 2-MeO, E], [-3207:3,5-F2,2 -MeO,Z] , [-3208:2,3-Cl2,2-MeO,E] , [-3209:2,3-Cl2,2-MeO,Z] , [-3210:2,4-Cl2, 2-MeO,E], [-3211:2,4-Cl2,2-MeO,Z], [-3212:2,5-Cl2,2-MeO,E], [-3213:2,5-Cl2 , 2-MeO, Z], [-3214:2,6-Cl2,2-MeO,E], [ -3215:3,4-Cl2,2-MeO,E ),[- 3216:3,5- Cl2,2-MeO,E], [-3217:2,3-Br2,2-MeO/E], [- 3218:2,4-Br2,2-MeO,E], [-3219:2,5 -Br2,2-MeO,E], [- 3220:2,6-Br2,2-MeO,E], [-3221:3,4-Br2,2-MeO,E],[- 3222:3, 5-Br2,2-MeO,E], [-3223:2,3-Me2,2-MeO,E], [- 3224:2,4-Me2,2-Me〇,E], [ -3225: 2,5-Me2,2-MeO,E],[- 322 6:2, 6-Me2,2-MeO,-E], [ -3227 : 3, 4-Me2,2-MeO, E] , [ · - 3228: 3r5-Me2, 2-Me〇, E 〕 , [ -3229:2,3-Et2,2-MeO,E ], [- 3230:2,4-Et2,2-MeO,E], [ -3231:2,5-Et2,2-MeO,E],[- 3232:2,6-Et2,2-MeO,E ] , [ -3233 : 3,4-Et2,2-MeO, E] , [.- 3234:3,5-Et2,2-MeO,E], [-3235:2,3-(CF3)2,2-MeO,E], [-3236:2, 4-(CF3) 2,2-MeO,E] , [-3237:2,5-(CF3)2,2-M eO, E3, [-3238:2,6-(CF3)2,2-MeO,E], [-3239:3, 4-(CF3)2,2-MeO,E3, C- 3240:3,5 -(CF3)2,2-MeO,E] , [-3241:2,3-(CHF2)2,2-MeO,E],[-3242:2,4-(CHF2)2,2-MeO, E] , [-3243:2,5-(CHF2)2,2-MeO,E],[-3244:2,6-(CHF2)2,2-MeO,E], [-3245:3,4 -(CHF2)2,2-MeO,E],[- 114 320202 200901876 324 6:3,5- (CHF2 )2,2-MeO,E] 3248:2,4- (CH2 F)2,2- MeO, E] 3250: 2,6-(CH2F)2,2-MeO,E] 3252:3,5-(CH2F)2 r2-Me〇,E] 3254:2,4-(MeO)2, 2-MeO,E] 3256:2,6-(MeO)2,2-MeO,E] 3258:3,5-(MeO)2,2-Me〇,E] 3260:2, 4- (Et- 〇) 2,2-MeO,E] 3262:2,6-(EtO)2,2-MeO,E] 3264:3,5-(EtO)2,2-MeO,E] 3266:2-Cl- 4-E,2-MeO,E], 3268:2-Cl-6-F,2-MeO,E], 3270:3-Cl-4-F,2-MeO,E], 3272:4-Cl -2-F,2-MeO,E], 3274:2-F-3-Me,2-MeO,E], 327-6:2-F-5-Me, 2-MeO, E], 3278: 3-F-2-Me,2-MeO,E 〕 r 3280:3-F-5-Me,2-MeO,E ], 3282:4-F-3-Me,2-MeO,E 〕, 3284 :2-Cl-4-Me,2-Me〇,E], 3286:2-Cl-6-Me,2-MeO,E], 3288:3-Cl-4-Me,2-MeO,E ] f 3290: 4-Cl-2-Me, 2-MeO, E], 3292: 2-F-3-CF3, 2-MeO, E 3 , 3294: 2-F-5-CF3, 2-MeO, E ], 115 , C-3247: 2, 3 -<CH2F)2,2-ΜθΟ,Ε],[-,C-3249:2,5-(CH2F)2,2-MeO,E],[-,[-3251:3,4-(CH2F 2,2-MeO,E],[-,[-3253:2,3-(MeO)2,2-Me〇,E], [-, [-3255:2,5-(MeO)2, 2-MeO,E],[-,[-3257:3,4-(MeO)2,2-MeO,E],[-,[-3259:2,3-(EtO)2,2-MeO, E], [-, [-3261: 2, 5-{EtO) 2, 2-MeO, E], [-, [-3263: 3, 4-(Et〇) 2, 2-MeO, E], [-, [-3265: 2-Cl-3-F, 2-MeO, E], C - [-3267: 2-Cl-5-F, 2-MeO, E], [-[-3269:3 -Cl-2-F,2-MeO,E],[-[-3271:3-Cl-5-F,2-MeO,E],[-[-3273:4-Cl-3-F,2 -MeO, E], [-[-3275:2-F-4-Me,2-MeO,E], [-[-3277:2-F-6-Me,2-MeO,E],[- [-3279: 3-F-4-Me, 2-MeO, E], [-[-3281:4-F-2-Me,2-MeO,E], C - [-3283:2-Cl- 3-Me,2-MeO,E],[-[-3285:2-Cl-5-Me,2-MeO,E),[-[-3287:3-Cl-2-Me,2-Me〇 , E], [-[-3289:3-Cl-5-Me,2-MeO,E], [- [-3291:4-Cl-3-Me,2-MeO,E],[-[- 3293: 2-F-4-CF3, 2-Me〇, E], [-[-3295: 2-F-6-CF3, 2-MeQ, E], [- 320202 200901876 3296: 3-F-2 -CF3,2-Me〇,E] 3298:3-F-5-CF3,2-MeO,E] 3300:4-F-3-CF3,2-Me〇,E] 3302:2-Cl-4 -CF3,2-MeO,E] 3304:2-Cl-6-CF 3,2-MeO,E] 3306:3-Cl-4-CF3,2-MeO,E] 3308:4-Cl-2-CF3,2-MeO,E] 3310:2-Me-3-CF3, 2-MeO,E] 3312:2-Me-5-CF3,2-MeO,E], 3314:3-Me-2-CF3,2-MeO,E] 3316:3-Me-5-CF3,2 -MeO,E] 3318:4-Me-3-CF3,2-Me〇,E] 3320:2-F-4-MeO,2-Me〇,E] 3322:2-F-6-MeO,2 -MeO,E ] 3324:3-F-4-MeO,2-MeO,E ] 3326:4-F-2-MeO,2-MeO, E ] 3328:2-Cl-3-MeOf2-MeO,E ] 3330: 2-Cl-5-Me〇, 2-Me〇, E] 3332: 3-Cl-2-MeO, 2-MeO, E] 3334: 3-Cl-5-MeO, 2-MeO, E ] 3336: 4-Cl-3-MeO, 2-MeOrE] 3338: 2-Me-4-MeO, 2-MeO, E) 3340: 2-Me-6-Me〇, 2-MeO, E] 3342: 3-Me-4-MeO,2-MeO,E] 3344:4-Me-2-MeO,2-MeO,E] [-3297 : 3-F-4-CF3,2-MeO, E ], -C -3299:4-F-2-CF3,2-MeO,E j ,[-[-3301:2-Cl-3-CF3,2-MeO,E],[-[-3303:2-Cl -5-CF3,2-MeO,E],[-[-3305:3-Cl-2-CF3,2-MeO,E],[-[-3307:3-CI-5-CF3,2-MeO , E ), [-[-3309:4-Cl-3-CF3,2-MeO,E], [-[-3311:2-Me-4-CF3,2-MeO,E],[-[- 3313: 2-Me-6-CF3, 2-MeO, E], [-C-3315: 3-Me-4-CF3, 2-MeO, E] r [-[-3317:4-Me-2- CF3,2-MeO,E],[-[-3319:2-F-3-MeO,2-MeO,E],[-[-3321:2-F-5-Me〇/2-MeO,E ),[-[-332 3:3-F-2-MeO,2-MeO,E], [-[-3325:3-F-5-MeO,2-MeO,E],[-[-3327:4-F-3- MeO, 2-MeO, E], [-C-3329: 2-Cl-4-MeO, 2-MeO, E) r [-C-3331: 2-Cl-6-MeO, 2-MeO, E] , [-C-3333:3-Cl-4-MeO,2-MeO,E 3 ,(-[-3335:4-Cl-2-MeO,2-MeO,EJ,[-[-3337:2- Me-3-MeO,2-MeO,E] f [-[-3339: 2-Me-5-MeO,2-MeO,E 3 ,[-C-3341:3-Me-2-MeO,2- MeO, E ], [-[-3343:3—Me-5-MeO, 2~MeO, E), [-[-3345:4-Me-3-MeO,2-MeO,E],[- 116 320202 200901876 3346:H,2-(Me)3C〇,E ] , C-3347:4-F,2-(Me)3 CO,E ] , [-3348:4-F,2-(Me)3C 〇,Z] , C-3349:4-Cl,2-(Me)3CO,E] , [-3350:4-C1,2-(Me)3CO,Z ] , [ -3351:4-Br,2 -(Me)3CO,E), [ -3352:4-1,2-(Me)3C〇,E], [ -3353:4-Me,2-(Me)3CO,E], [-3535: 4-Me,2-(Me)3CO,Z ] , [-3355:4-Et,2-(Me)3CO,E], C-3356:4-C3H7,2-(Me)3CO,E], [-3357: 4-(Me)2CH, 2-(Me)3CO, E], [-3358: 4-CF3, 2-(Me)3CO, E], [-3359: 4-CF3, 2-( Me)3CO,Z],[-3360:4-C2F5,2-(Me)3CO.,E], [ -3361:4-C3F7,2-(Me)3C〇,E ) r C -3362:4 - (CF3)2CF,2-(Me)3CO,E) , [-3363 : 4-(CF3 ) 2 CH, 2-(Me) 3 CO, E],[- , 3364:4-CHF 2,2-(Me)3CO,E] , [-3365:4-CH2F,2-(Me)3COrE), [- '1.. 3366:4-CF3CH2,2-(Me)3C〇,E] , [-3367:4-MeO,2-(Me)3 CO,E],[-3368:4-MeO,2-(Me)3C0,Z], [-3369:4-EtO,2-(Me ) 3CO, E], [- 3370: 4-C3H7O, 2-(Me) 3CO, E], [-3371: 4-(Me) 2CHO, 2-(Me) 3CO, E], [-3372: 4 -N〇2,2-(Me)3CO,E], [-3373:4-N〇2,2-(Me)3CO,Z], [-3374:3-F,2-(Me)3C0, E] , [-3375:3-F,2-(Me)3CO,Z] , [-3376:3-Cl,2-(Me)-3 CO,E] , C-3377 : 3-C1,2 -(Me) 3 C〇, Z3 , C-3378 : 3-Br, 2-(Me)3CO,E 〕 , [ -3379:3-1,2-(Me)3CO,E 〕 , C -3380: 3-Me,2-(Me)3CO,E], [-3381:3-Me,2-(Me)3CO,Z], [-3382:3-Et,2-;,. (Me)3CO, E] , [ -3383:3-C3H7,2-(Me)3CO,E] , C -3384:3- (Me)2CH,2-(Me)3C〇,E] , [-3385:3-CF3 ,2-(Me)3C〇,E] , C-3386:3-CF3,2-(Me)3CO,Z],[-3387:3-C2F5,2-(Me)3CO,E],[- 3388:3-C3F7,2-(Me)3CO,E], C-3389:3-(CF3)2CF,2-(Me)3CO,E], C-3390:3-(CF3)2CH,2- (Me)3CO,E], [-3391:3-CHF2,2-(Me)3CO,E], [-3392.:3-CHF2,2-(Me)3CO,Z], [-3393 :3 -CH2 F, 2-(Me) 3 C〇, E ], C-3394: 3-CH2F, 2-(Me)3CO, Z], [ -3395 : 3-CF3 CH2,2-(Me) 3 〇〇, E), 117 320202 200901876 [-3396:3-MeO,2-(Me)3CO,E] , C-3397:3-MeO,2 -(Me)3CO,Z],[-3398:3-EtO,2-(MehC〇,E], [-3399:3-C3H7〇,2-(Me)3CO,E],[-3400:3 -(Me)2CHO,2-(Me)3CO,E], [-3401:3-N02,2-(Me)3CO,E], [-3402:2-F,2-(Me)3CO,E ], [-3403: 2-C1, 2-(Me)3CO, E], C-3404: 2-Br, 2-(Me)3CO, E], [-3405: 2-I, 2-(Me ) 3CO, E], [-3406: 2-Me, 2-(Me)3CO, E], C-3407: 2-Et, 2-(Me)3CO, E), [-3408: 2-C3H7, 2-(Me)3CO, E.], [-3409: 2-(Me)2CH, 2-(Me)3CO, E], [- 3410: 2-CF3, 2-(Me)3CO, E], [-3411: 2-C2 F5,2-(Me) 3 CO, E ], [- 3412:2-C3F?,2-(Me)3CO,E] , [-3413 :2-(CF3 ) 2CF, 2-(Me) 3CO,E], [-3414 :2-(CF3)2CH,2-(Me)3〇〇,E], [ -3415:2-CHF2,2-(Me)3CO,E] , [-3416: 2-CH2F, 2-(Me)3CO, E], [-3417: 2-CF3 CH2, 2-(Me)3CO, E], [-3418: 2-MeO, 2-(Me ) 3CO, E], [-3419: 2-EtO, 2-(Me)3CO, E], [ -3420: 2-C3H7O, 2-(Me)3CO, E], C -3421: 2- (Me 2CHO,2-(Me)3CO,E ] , C -3422:2-N02,2-(Me)3CO,E 3 ,[- 3423:2,3-F2,2-(Me)3CO,E] , [-3424:2,4-F2,2-(Me)3 CO, E], [-3425: 2, 5-F2, 2-(Me) 3C〇, E3, C-3426: 2, 6-F2, 2-(Me) 3 CO, E ], [-3427: 3, 4-F2,2-(Me) 3CO,E) , [-3428 : 3,4-F2,2-(Me) 3CO, Z ],[-3429:3,5-F2,2-(Me ) 3C〇, E], [-3430:3,5-F2,2-(Me)3CO,Z], [-3431:2,3-Cl2,2-(Me)3COrE], [-3432:2 ,3-Cl2,2-(Me)3C〇,Z),[-3433:2,4-Cl2f2-(Me)3CO,E] , [-3434:2,4-Cl2,2-(Me)3CO ,Z],[-3435:2,5-Cl2,2-(Me)3CO,E], C-3436:2,5-Cl2,2-(Me)3CO,Z],[-3437:2, 6-Cl2,2-(Me)3C〇,E] f [-3438:3,4-Cl2,2-(Me)3CO,E],[-3439:3,5-Cl2,2-(Me) 3CO,E] , C-3440:2,3-Br2,2-(Me)3CO,E],[-3441:2,4-Br2,2-(Me)3CO,E] , [-3442:2 ,5-Br2,2-(Me)3CO,E],[-3443:2,6-Br2,2-(Me)3C〇,E], [-3444:3,4-Br2,2-(Me )3CO,E] , C- 118 320202 200901876 3445:3,5-Br2,2-(Me)3CO,E] , [-3446:2,3-Me2,2-(Me)3C〇,E], [-3447: 2,4-Me2,2-(Me)3CO,E], [-3448:2,5-Me2,2-(Me)3CO,E],[-3449:2,6-Me2, 2-(Me)3CO,E] , [-3450:3,4-Me2Λ2-(Me)3CO,E],[-3451:3,5-Me2,2-(Me)3CO,E], [- 3452:2,3-Et2,2-(Me)3CO,E],[-3453:2,4-Et2,2-(Me)3C〇,E], [-3454:2,5-Et2,2 -(Me)3CO,E],[-3455:2, 6-Et2,2-(Me)3C〇,E] , [-3456:3, 4~Et2,2-(Me)3CO,E), [-3457: 3,5-Et2,2-(Me)3CO,E],[-3458:2,3-(CF3)2,2-(Me>3CO,E], [-3459:2,4-(CF3) 2,2-(Me)3CO,E 〕 , [ -3460:2,5-(CF3)2,2-(Me)3CO,E],.[-3461:2,6-(CF3 )2,2 -(Me)3CO,E],[ -3462:3,4-, (CF3)2,2-(Me)3CO,E],[-3463:3,5-(CF3)2,2-(Me&gt ;3CO,E],[- 3464:2,3-(CHF2)2,2-(Me)3CO,E] , C -34 65 :2, 4~ (CHF2 ) 2,2- (Me)3CO, E) , [-3466:2,5-(CHF2 )2.2-(Me)3CO,E] , [-3467:2,6- (CHF2)2r2-(Me)3CO,E], [-3468:3 , 4-(CHF2)2,2-(Me)3CO, E], [-3469:3,5-(CHF2)2,2-(Me)3CO,E], [-3470:2,3-( CH2F)2,2-(Me)3CO,E] , [-3471:2,4-(CH2F)2,2-(Me)3CO,E) , [-3472:2,5- (CH2F)2, 2-(Me)3CG,E] , [-3473 :2, 6-(CH2 F) 2,2-(Me) 3〇〇,ε3-,(-3474 :3,4-(CH2F)2,2 -(Me)3CO,E] , [ -3475 :3, 5-(CH2 F) 2,2- (Me)3CO,E] , [-3476:2,3-(MeO)2,2-(Me ) 3C〇, E], [-3477:2,4-, (MeO)2,2-(Me)3CO,E], [-3478:2,5-(MeO)2,2-(Me)3CO , E], [- 3479: 2,6-(MeO) 2,2-(Me)3CO,E], [-3980:3,4-(MeO)2,2-(Me)3CO,E], [-3481:3,5-(MeO)2,2-(Me)3C〇,E], [ -3482:2,3-(EtO)2,2-(Me) 3CO,E],[-3483 :2,4-(EtO)2,2-(Me) 3CO,E 3 ,[-3484:2,5-(EtO)2,2-(Me)3CO,E], C-3485:2,6 -(EtO)2,2-(Me)3CO,E],[-3486:3,4-(EtO)2,2-(Me)3CO,E],[-3487:3,5-(EtO) 2,2-(Me)3CO,E ] , C -3488:2-C1-3-F,2-(Me)3C〇,E ],[- 119 320202 200901876 3489:2-Cl-4-F, 2-(Me)3CO, E], [-3490: 2-C1-5-F, 2-(Me)3C〇, E], [-3491: 2-Cl-6-F, 2-(Me) 3CO, E 〕 , [ -3492: 3-C1-2-F, 2-(Me)3CO, E], [-3493: 3-Cl-4-F, 2-(Me)3C〇, E], [-3494:3-01-5- F,2-(Me)3CO,E],[-3495:4-Cl-2-F,2-(Me)3CO,E],[-3496:4- Cl-3-F,2-(Me)3C〇,E], [-3497:2-F-3-Me,2-(Me)3CO,E], [-3498:2-F-4-Me ,2-(Me>3C0,E],[ -3499:2-F-5-Me,2-(Me)3C〇, E j , C -3500:2-F-6-Me,2-(Me ) 3CO, E], [-3501: 3-F-2-Me, 2-(Me) 3CO, E], [-35〇2: 3-F-4-Me, 2-(Me)3C〇, E 〕 , 〔 -3503:3-F-5-Me,2- (Me)3C〇,E],[-3504:4-F-2-Me,2-(Me)3C〇,E ], [ -3505:4-F-3-

Me,2-(Me)3CO,E], [-3506:2-Cl-3-Me,2-(Me)3CO,E] , [-3507:2-Cl-4-Me,2-(Me ) 3CO, E], [-3508: 2-Cl-5-Me, 2-(Me)3C〇, E], [- 3509: 2-Cl-6-Me, 2-(Me)3CO, E] , [-3510: 3-Cl-2-Me, 2-(Me)3CO, E], [-3511: 3-Cl-4-Me, 2-(Me)3CO, E], [-3512:3 -Cl-5-Me,2-(Me)3C〇,E] , [-3513:4-Cl-2-Me,2-(Me)3CO,E] r [-3514:4-Cl-3- Me, 2-(Me)3C〇, E], [-3515: 2-F-3-CF3, 2-(Me)3CO, E], [-3516: 2-.F-4-CF3,2- (Me)3CO, E], [-3517: 2-F-5-C.F3, 2-(Me) 3 CO, E], [-3518: 2-F-6-CF3, 2-(Me) 3CO, E], [-3519: 3-F-2-CF3, 2-(Me)3CO, E], [-3520: 3-F-4-CF3, 2-(Me)3CO, E], [ -3521:3-F-5-CF3,2-(Me)3CO,E] , [-3522:4-F-2-CF3,2-(Me)3CO,E],[ -3523:4-F -3- CF3,2-(Me)3CO,E], [-3524:2-Cl-3-CF3,2-(Me)3CO,E],[- 3525:2-Cl-4-CF3,2 -(Me)3CO,E], [ -3526:2-Cl-5-CF3,2-(Me)3CO,E], [-3527:2-Cl-6-CF3,2-(Me)3CO, E], [-3528: 3-Cl-2-CF3, 2-(Me) 3 CO, E ] , [ -3529: 3-Cl-4-CF3, 2-(Me) 3 CO, E], C - 3530: 3-Cl-5-CF3, 2-(Me)3CO, E], [ -3531: 4-Cl-2-CF3, 2-(Me)3C〇, E], C-3532: 4-Cl-3-CF3, 2-(Me)3CO, E], [-3533: 2-Me-3- 120 320202 200901876 CF3, 2-(Me)3 CO, E 3 , [ - 3534: 2-Me-4-CF3, 2-(Me)3CO, E], [- 3535: 2-Me-5-CF3, 2-(Me)3C〇, E]. , C -3536:2- Me-6-CF3,2-(Me)3CO,E], [-3537:3-Me-2-CF3,2-(Me)3CO,E], [-3538:3-Me-4-CF3, 2-(Me)3C〇,E], [-3395:3-Me-5-CF3,2-(Me)3C〇,E],[- 3540:4-Me-2-CF3,2-(Me ) 3CO, E 〕 , [ -3541: 4-Me-3-CF3, 2-(Me)3CO, E], [-3542: 2-F-3-MeO, 2-(Me)3CO, E), [-3543:2-F-4-

MeO, 2-(Me)3C〇, E], [-3544: 2-F-5-MeO, 2-(Me)3CO, E], [-3545: 2-F-6-MeO, 2-( Me)3 C〇,E ] , [-3546:3-F-2-Me〇,2-(Me)3CO,E], [- 3547:3-F-4-MeO,2-(Me)3CO , E] , [-3548: 3-F-5-MeO, 2-(Me)3CO, e3, [-354 9:4-F-2-MeOr 2-(Me)3CO, E], [-3550 :4-F-3-Me〇,2-(Me)3CO,E],[-3551:2-Cl-3-MeO,2-(Me)3CO,E],[-3B52:2-Cl- 4-MeO,2-(Me)3C〇,E], [ -3553:2-Cl-5-MeO,2-(Me)3CO, E ],[- 3554:2-Cl-6-MeO,2 -(Me)3C〇,E 〕 , [ -3555:3-Cl-2-MeO,2-(Me)3CO,E] , [-3556:3-Cl-4-MeO,2-(Me>3CO , E] , [-3557:3-01-5-MeO,2-(Me)3C〇,E], [-3558:4-Cl-2-MeO,2-(Me)3 CO, E], [- 3559: 4-Cl-3-MeO, 2- (Me) '3CO, E 〕 , 〔 -3560: 2-Me-3-MeO, 2- (Me)3CO, E) , C-3561:2 -Me-4-MeO,2-(Me)3CO,E], C-3562:2-Me-5-MeO,2-(Me)3C〇,E], [ -3563:2-Me-6- MeO,2-(Me)3CO,E],[- 3564:3-Me-2-MeO,2-(Me)3CO,E ] , [ -3565:3-Me-4-MeO,2-- ( Me) 3CO, E], [-3566: 3-Me-5-Me〇, 2-(Me)3CO, E], [-3567: 4-Me-2-MeO, 2-(Me)3 CO, E ] , C -3568: 4-Me-3-MeO, 2-(Me)3CO, E ), [- 3569:H,2,3-F2,E], [-35.70 :4-F,2,3-F2,E], [-3571:4-F,2,3-F2,Z], [-3572:4-Cl,2,3-F2,E]r[- 3573: 4-Cl, 2,3-F2, Z], [-3574: 4-Br, 2, 3-F2, E], [ -3575: 4-1, 2, 3-F2, E], [ -3576:4-

Me,2,3-F2,E] , C -3577:4-Me,2,3-F2,Z ] , C -3578:4-Et,2,3- 121 320202 200901876 F2,E],[- 35"79:.4-C3H7,2,3-F2,E], [-3580:4-(Me)2CH,2,3-Fs,E], [-3581:4-CF3,2,3- F2, E], [-3582: 4-CF3, 2, 3-F2, Z], [-3583: 4-C2F5, 2, 3-F2, E], [-3584: 4-C3F7, 2, 3 -F2,E], [-3585:4-(CF3)2CF,2,3-F2, C-3586:4-(CF3)2CH,2,3-F2,E], [-3587:4-CHF2 , 2,3-F2 ,E]., [ -3588:4-CH2F,2,3-F2>E 3 , C -3589:4- CF3CH2,2, 3-F2 ,E]r [ -3590:4 -MeO,2,3-F2,E], C -3591:4-MeO, 2, 3-F2, Z] , [-3592:4-EtO,2,3-F2,E] , [-3593 : 4-C3 H7 0, 2,3-F2, E], [-3594: 4-(Me}2CHO, 2,3-F2, E], [-3595:4-N02,2,3-F2,E ], [-3596: 4-N02, 2, 3-F2, Z], [-3597: 3-F, 2, 3-F2, E], [-3598: 3-F, 2, 3-F2, Z], [-3599: 3-Cl, 2, 3-F2, E], [-3600: 3-C1, 2, 3-F2, Z], [-3601: 3-Br, 2, 3-F2rE ], [-3602: 3-r, 2, 3-F2, E], [-3603: 3-Mef2, 3-Fz, E), C-3604: 3-Me, 2, 3-F2, Z] , [-3605:3-Et,2,3-F2,E] , [ -3606:3-C3H7,2,3-F2,E] , C -3607:3- (Me)2CH,2,3- F2, E], [ -3608: 3-CF3, 2r3-F2, E], C - 3609: 3-CF3, 2, 3-F2, Z], [-3610: 3-C2F5, 2, 3-F2, E], [-3611: 3-C3F7, 2, 3-F2, E]. > [-3612: 3-(CF3)2CF, 2,3-F2,E],[-3613:.3-(CF3)2CH,2,3-F2,E], [-3614:3-CHF2,2,3-F2,E], [-3615 :3-CHF2,2,3-F2,Z], [-3616:3-CH2F,2,3-F2,E], [-3617:3-CH2F,2,3-F2,Z], [- 3618: 3-CF3CH2, 2,3-F2, E], [-3619: 3-MeO, 2,3-F2, E], [-3620: 3-MeO, 2, 3-F2, Z], [ -3621:3-EtO,2,3-F2,E], [-3622:3-C3H*7〇,2,3-F2,E], [ -3623:3-(Me)2CHO,2,3 -F2 ,E ] , C -3624 : 3-N02,2,3- F2,E] , C-3625:2-F,2,3-F2,E) , [-3626:2-C1,2, 3-F2 , E ], [- 3627:2-Br,2,3-F2,E ] , [ -3628 :2-1f2,3-F2rE ] , [-3629:2-

Me, 2, 3-F2, E], [-3630: 2-Et, 2, 3-F2, E], [-3631: 2-C3H7, 2, 3-F2, E], [-3632: 2 -(Me)2CH,2,3-F2,E],[-3633:2-CF3,2,3-F2,E]Λ 122 320202 200901876 [-3634:2-C2F5,2,3-F2,E ] , [ -3 635 :2-C3 F7 , 2,3-F2 , E ], [-3636:2-(CF3 )2CF/2,3-F2 ,E] , [-3637 :2-(CF3 ) 2 CH, 2,3-F2 , E], [-3638:2-CHF2,2,3-F2 ,E] , [-3639 : 2-CH2 F, 2,3-F2 , E] , [-3640 :2-CF3CH2,2,3-F2 ,E ] , [ -3641:2-MeO,2,3-F2 ,E ] , [ -3642:2-EtO, 2, 3-F2 ,E],[ - 3643:2-C3H7〇,2,3-F2,E], C-3644:2-(Me)2CHO,2,3-F2,E3, C-3645 : 2-N02,2,3-F2 , E ] , [-3646:2,3- F2,2,3-F2,E] , [-3647:2,4-F2,2,3-F2 ,E] , [-364 8 : 2,5-F2 , 2,3-F2,E] , [-3649:2,6-F2,2,3-F2 ,E] , [-3650: 3,4-F2,2 f 3-F2 , E], [- 3651:3,4-F2,2,3-F2,Z ] , [ -3652 : 3,5-F2,2,3-F2 , E ] , C- ( 3653:3,5-F2,2,3 -F2,Z], [-3654:2,3-Cl2,2,3-F2,E], [- 3655:2,3-Cl2,2,3-F2,Z], [-3656:2, 4-Cl2,2,3-F2.,E],[-3657:2,4-Cls,2,3-F2,Z~} f 〔-3658:2,5-Cl2,2,3-F2, E], [-3659:2,5-Clz,2,3-F2,Z ] , [ -3660:2,6-Cl2,2,3-Fs,E ],[- 3661:3,4-C12 ,2,3-F2 ,E , [ -3662 : 3,5-Cl2,2,3-F2 , E], [- 3663:2,3-Br2,2,3-F2 ,E ] , C -3664 : 2,4-Br2,2 , 3-F2 , E ), [- 3665:2,5-Br2,2,3-F2 ,E ) , C -3666: 2,6-Br2,2,3-F2 , E ],[- 3667: 3, 4-Br2 r2,3-F2, E], [-3966: 3,5-Br2,2,3-F2, E], [- 3669:2,3-Me2,2,3-F2,E ] , [ -3670 : 2,4-Me2,2,3-F2 , E], [- , 3671:2,5-Me2,2,3-F2,E } , [ -3672:2,6-Me2 , 2,3-F2 , E], [.- 3673:3,4-Me2,2,3-F2 ,E ] , C -3674 : 3,5-Me2,2,3-F2 , E ],[ - 3675: 2,3-Et2,2,3-F2,E ] , [-3676:2,4-Et2,2,3-F2,E], [- 3677:2,5-Et2,2,3 -F2,E ] , [ -3678:2,6-Et2,2,3-F2,E], [- 3679:3,4-Et2,2,3-F2,E], [ -3680: 3, 5-Et2,2,3-F2 , E ],[-3681:2,3-(CF3 )2,2,3-F2 ,E] , [-3682 : 2,4-(CF3 ) 2,2, 3-F2 , E], [-3683:2,5-(CF3 )2,2,3-F2 ,E] , [-3684 : 2,6-(CF3 ) 2,2,3-F2 , E] , [- 123 320202 200901876 3685:3, 4-(CF3)2,2,3-F2,E] , [-368 6:3,5-(CF3 ) 2,2,3-F2 , E],[ -3687: 2,3-(CHF2)2,2,3-F2,E], [-3688:2,4-(CHF2)2,2,3-F2,E], [-3689:2,5 -(CHF2)2,2,3-F2,E] , [ -3690:2, 6-(CHF2)2,2,3-F2,E]., [ -3691:3,4-(CHF2 ) 2,2,3-F2,E] , [ -3692:3,5- (CHF2 )2,2,3-F2 ,E] , [ -3693:2,3-(CH2F)2,2,3 -F2 , E ], [- 3694:2,4-(CH2F) 2,2,3-F2,E] , [-3695 : 2,5-(CH2 F) 2,2,3-F2 , EJ , [-3696:2, 6-(CH2F)2,2,3-F2,E], [-3697:3,4-(CH2F) 2,2,3-F2,E], [-3998:3 , 5-(CH2F)2,2,3-F2,E] , [ -3699:2,3-(MeO)2,2,3-F2,E) , [-3700:2,4-(MeO) 2,2,3-F2,E] , [-3701:2,5-(MeO)2,2,3-F2,E], [-3702:2,6-(MeO)2,2,3- F2, E], [-3703:3,4-(MeO)2,2,3-F2,E), [-3704:3,5-(MeO)2,2,3-F2,E], 1 -3705: 2,3-(Et〇)2,2,3-F2,E], [-3706:2,4-(EtO>2,2,3-F2,E], [-3707:2, 5-(EtO)2,2,3-F2,E] , [-3708:2,6-(EtO)2,2,3-F2,E] , [-3709:3,4-(EtO)2 , 2,3-F2,E] , C-3710:3,5-(EtO)2,2,3-F2/E3 , [-3711:2-

Cl-3-F, 2,3-F2, E], [-3712: 2-Cl-4-F, 2,3-F2, E], [-3713: 2-Cl-5-F, 2, 3-F2, E}, [-3714: 2-C1-6-F, 2, 3-F2, E], [-3715: 3-C1-2-F, 2, 3-F2, E], [ -3716:3-Cl-4-F,2,3-F2 rE ) , [ -3717 :3-C1-5-

Fr2,3-F2,E], [-3718:4-Cl-2-F,2,3-F2,E], [-3719:4-Cl-3-F, 2r3-F2,E], [ -3720: 2-F-3-Me, 2, 3-F2, E], [ -3721: 2-F-4-

Me,2,3-F2,E ] , [-3722:2-F-5-Me,2,3-F2,E], [ -3723:2-F-6-

Me,2,3-F2,E] , [-3724:3-F-2-Me,2,3-F2,E ] , [-3725:3-F-4-

Me,2,3-F2,E ] , [-3726:3-F-5-Me,2,3-F2 ,E], [-3727:4-F-2-

Me,2,3-F2,E] , [-3728 : 4-F-3-Me, 2,3-F2 , E 3 , [-3729:2-01-3-

Me, 2, 3-FZ, E], [-3730: 2-Cl-4-Me, 2, 3-F2, E), [-3731: 2-C1-5-

Me,2,3-F2 ,E] , [-3732:2-Cl-6-Me,2,3-F2 ,E] , [-3733:3-01-2- 124 320202 200901876

Me, 2, 3-F2, E], [-3734: 3-Cl-4-Me, 2, 3-F2, E],

Me,2,3-F2,E] , [-3736: 4-Cl-2-Me, 2,3-F2 , E ] r Me,2,3-F2,E], [-3738:2-F -3-CF3,2,3-F2,E] CF3,2,3-F2, C-3740:2-F-5-CF3,2,3-F2,E] CF3,2,3-F2,E ],[-3742:3-F-2-CF3,2,3-F2,E] CF3,2,3-F2,E], [-3744:3-F-5-CF3,2,3-F2 , E] CF3,2,3-F2,E], [-3746:4-F-3-CF3,2,3-F2,E], CF3,2,3-F2.,E],[-3748 :2-Cl-4-CF3,2,3-F2,E], CF3,2,3-F2,E], [-3750:2-Cl-6-CF3,2,3-F2,E], CF3,2,3-F2,E]r[-3752:3-Cl-4-CF3,2,3-F2,E], CF3,2,3-F2,E],[-3754:4-Cl -2-CF3,2,3-F2,E], CF3,2,3-F2,E], [-3756:2-Me-3-CF3,2,3-F2,E], CF3,2, 3-F2, E], [-3758: 2-Me-5-CF3, 2, 3-F2, E], CF3, 2, 3-F2, E], [-37 60: 3-Me-2- CF3,2,3-F2,E], CF3,2,3-F2,E] , [-3762:3-Me-5-CF3,2,3-F2,E], CF3,2,3-F2 , E], [-3764: 4-Me-3-CF3, 2; 3-F2, E] Me〇, 2, 3-F2, E], [-37 66: 2-F-4-MeO, 2 Λ 3-F2 ,E] ' MeO,2,3-F2 ,E) , C-37 68 : 2-F-6-MeO, 2,3-F2 , E ], MeO,2,3-F2 ,E ], [-3770 : 3-F-4-MeO, 2,3-F2 , E ], MeO, 2,3-F2, E], [-3772:4-F-2-MeO,2,3- F2, E], MeO, 2, 3-F2, E], [-3774: 2-Cl-3-MeO, 2, 3-F2,E], MeO,2,3-F2,E], [-3776:2-Cl-5-MeO,2,3-F2,E], MeO,2,3-F2,E], [-3778: 3-Cl-2-MeO, 2,3-F2, E], MeO, 2,3-F2, E], [-3780: 3-Cl-5-MeO, 2, 3-F2, E], MeO, 2,3-F2, E], [-3782: 4-Cl-3-MeO, 2, 3-F2, E], [-3735: 3-01-5-C-3737: 4 -Cl-3-,[-3739:2-F-4-, C-3741:2-F-6-, [-3743:3-F-4-, C-3745:4-F-2-C -3747: 2-Cl-3-[-3749:2-01-5-[-3751:3-01-2-[-3753:3-01-5-[-3755:4-01-3-[ -3757: 2-Me-4-[-3759:2-Me-6-C-3761:3-Me-4-C-3763:4-Me-2-,[-3765:2-F-3- , [-3767: 2-F-5-, C-3769: 3-F-2-.C-3771: 3-F-'5- C-3773: 4-F-3-C-3775: 2- Cl-4-[-3777:2-01-6-[-3779:3-01-4-[-3781:4-01-2-C-3783:2-Me-3- 125 320202 200901876

MeO, 2,3-F2, E], [-3784: 2-Me-4-MeO, 2, 3-F2, E], [-3785: 2-Me-5-MeO, 2, 3-F2, Ε] , [-3786:2-Me-6-MeO,2,3-F2,Ε], C-3787:3-Me-2-Me〇,2,3-F2,E], [-3788: 3-Me-4-MeO, 2,3-F2, E], 〇3789: 3-Me-5-Me〇, 2,3-F2, E], [-3790:4-Me-2-MeO, 2,3-F2,E], [-3791:4-Me-3-MeO,2,3-F2,E], [-3792:H,2,4-F2,E], [-3793:4 -F,2,4-F2,E], C-3794:4-F,2,4-F2,Z], C-3795: 4-C1, 2, 4-F2, E 3 , [-3796: 4-Clr2,4-F2,Z], [-3797:4-Bit,2,4-F2,E], [-3798:4-I,2,4-F2,E], [-3799:4 -Me,2,4-F2,E], [-3800:4-Me,2,4-F2,Z], [-3801:4-

Et,2,4-F2,E ] , [ -3802:4-C3H7,2,4-F2,E], C -3803:4- (Me)2CH,2,4-F2,E],[- 3804: 4-CF3, 2, 4-F2, E], [-3805: 4-CF3, 2, 4-F2, Z], [-3806: 4-C2F5, 2, 4-F2, E], [ -38O7r4-C3F7,2,4-F2,E], [-3808: 4-(CF3)2CF,2,4-F2,E), C-3809: 4-(CF3) 2 CH, 2, 4- F2, E], [-3810: 4-CHF2, 2, 4-F2, E], [-3811: 4-CH2F, 2, 4-F2, E], [-3812: 4-CF3CH2, 2, 4 -F2rE], [-3813:4-MeOr2,4-F2,E], [-3814:4-MeO,2,4-F2,ZJ, [-3815:4-EtO,2,4-F2,E3 , [-3816:4- C3H7〇,2,4-F2,e3,C-3817:4-(Me)2CHO,2,4-F2,E3, [-3818:4-N02,2,4-Fs , E 3 , [ -3819:4-N02,2,4-F2 ,Z ] , C -3820 : 3-F, 2,4- F2,E], [-3821:3-F,2,4_F2, Z], [-3822: 3-Cl, 2, 4-F2, E], [-3823: 3-Cl, 2, 4-F2, Z], [ -3824: 3-Br, 2, 4-F2 , E ] , C -3825:3- I,2,4-F2,E] , C-3826:3-Me,2,4-F2,El , C-3827:3-Me,2,4-F2 , Z] [-3828: 3-Et, 2, 4-F2, E], [-3829: 3-C3H7, 2, 4-F2, E], [-3830: 3_ (Me) 2CH, 2, 4 -F2./E ] , C -3831:3-CF3,2,4-F2 ,E 3 [ -3832:3-CF3,2,4-F2,Z], [-3833:3-C2F5,2, 4-F2,E], [-3834:3-C3F7,2,4-F2,E], [-3835:3-(CF3)2CF,2,4- F2, E], [-3836: 3-(CF3)2CH, 2, 4_F2, E], [-3837: 3-CHF2, 2, 4-F2, E], [-3838: 3-CHF2, 2 , 4-F2, Z], 126 320202 200901876 [-3839: 3-CH2: F, 2, 4-F2, Ε], [-3840: 3-CH2 F, 2,4-F2, Z], [- 3841: 3-CF3CH2, 2,4-F2, E], [-3842: 3-MeO, 2, 4-F2, E], [-3843: 3-MeO, 2, 4-F2, Z], [ -3844 : 3-EtO, 2,4-F2 , E] , [-3845 :.3-C3 H7 〇, 2,4-F2,E], [ -3846:3-(Me)2CHO,2,4 -F2, E], C -3847 : 3-N02,2,4-F2,E], [-3848:2-F,2,4-F2,E], [-3849:2-Cl,2, 4-F2, E], [-3850: 2-Br, 2, 4-F2, E], [ -3851: 2-1, 2, 4-F2, E], C -3852: 2-

Me, 2, 4-F2, E], [-3853: 2-Et, 2, 4-F2, E], [-3854: 2-C3H7, 2, 4-F2, E], [-3855: 2 -(Me)2CH,2,4-F2,E], [-3856:2-CF3,2,4-F2,E], [-3857:2-C2F5,2,4-F2,E], -3858: 2-C3F7,2,4-F2,E], [-3859:2-(CF3)2CF, 2,4-F2,E], [-3860:2-(CF3)2CH,2,4 -F2,E], [-3861:2-CHF2,2,4-F2,E], [-3862:2-CH2F,2,4-F2,E] ; [-3863:2-CF3CH2,2, 4-F2,E], [ -3864:2-MeO,2,4-F2,E], C -3865:2-

EtO,2,4-F2,E] , [ -3866:2-C3H70,2,4-F2,E] , C -3867:2- (Me)2CHO,2,4-F2 ,E] , [- 3868 :2-N02,2,4-F2 r E 3 , [-3869:2,3- F2,2,4-F2fE] , C-3870:2,4-F2/2,4-F2 ,E] , [-3871: 2,5-F2,2,4-F2,e3, [-3872:2,6-F2,2,4-F2,E], [-3873: 3> 4-F2,2, 4-F2 f E], [-3874:3,4-F2,2,4-F2,Z ] , C -3875: 3, 5-F2,2,4-F2 , E ] , C- 387 6: 3,5-F2,2,4-F2,Z 3 ,C -3877 : 2,3-Cl2,2,4-F2 , E 3,C-3878:2,3-Cl2,2,4-F2, Z 〕 , [ -3879:2,4-Cl2,2,4-F2,E ], C -3880:2,4-Cl2,2,4-F2,Z], [-3881:2,5-Cl2 , 2,4-F2,E], [-3882:2,5-CI2,2,4-F2,Z ] , ( -3883:2, 6-Cl2,2,4-F2,E ] , C- 3884: 3,4-Cl2,2,4-F2,E ] , ( -3885:3, 5-Cl2,2,4-F2 , E ],[- 3886:2,3-Br2,2,4- F2, E], [-3889:2,4-Br2,2,4-F2,E], [-3888:2,5-Br2,2,4-F2,E], [-3889:2, 6 -Br2,2,4-F2,E], [-3890:3,4-Br2,2,4-F2,E], [-3891:3,5-Br2,2,4-F2,E], 〔- 127 320202 200901876 3892:2,3-Me2,2,4-F2 ,Ε ] , 〔 -3893: 2,4-Me2,2,4-F2 , E], [- 3894:2,5-Me2 , 2,4-F2,E ] , [ -3895: 2,6-Me2,2,4-F2 , E], [- 3896:3,4-Me2,2,4-F2 ,E ] , 〔 3 897 : 3,5-Me2,2,4-F2 , E] , C - 3898:2,3-Et2,2,4-F2,E ] , [-3899:2,4-Et2,2,4- F2, E], [- 3900:2,5-Et2,2,4-F2,E], [ -3901: 2,6-Et2,2,4-F2, E ] , C - 3902:3, 4 -Et2,2,4-F2,E ] , [ -3903: 3,5-Et2,2,4-F2 , E].,[- .3904:2,3-(CF3)2,2,4- F2, E] , [-3905 : 2,4-(CF3 ) 2,2,4-F2 , E], [-3906:2,5-(CF3 )2 r2,4-F2 ,E] , [- 3907 : 2,6-(CF3 ) 2,2,4-F2 , E], [-3908:3, 4-(CF3) 2,2,4-F2,E] , [-3909 : 3,5- (CF3 ) 2,2,4-F2 , E],[-3910:2,3-(CHF2 )2,2,4-F2 ,E] , [-3911: 2,4-(CHF2 ) 2,2 , 4-F2 , E], [-3912:2,5-(CHF2)2,2,4-F2,E] , [ -3913:2,6- (t:HF2 ) 2,2,4- F2 , E], [ -3914:3,4-(CHF2>2,2,4-F2,E], '[ -3915:3,5- (CHF2)2,2,4-F2,E], [ -3916:2,3-(CH2F)2,2,4-F2,E],[- 3917:2,4-(CH2F)2,2,4-F2/E], [-3918 : 2,5 -(CH2 F) 2,2,4-F2 , E], [-3919:2,6-(CH2F)2,2,4-F2,E ] , [ -3920 : 3, 4-(CH2 F) 2,2,4- F2,E] , [ -3921:3, 5-(CH2F)2,2,4-F2/E ] , [ -3922:2,3- (MeO)2,2,4- F2 , E] , [-3923 : 2,4-(MeO) 2,2,4-F2 , E] , [-3924:2,5-(MeO)2,2,4-F2,E] , [ -3925:2,6-(MeO)2,2,4-F2,E) , [-3926:3,4-(MeO ) 2,2,4-F2 ,E] , [-3927 : 3,5-(MeO) 2,2,4-F2 , E] , [-3928:2,3-(EtO)2,2,4 -F2,E], [-3929:2,4-(EtO)2,2,4-F2,E], [-3930:2,5-(EtO)2,2,4-F2,E], [-3931: 2,6-(EtO)2,2,4-F2,E], [-3932:3,4-(EtO)2,2,4-F2,E], [-3933:3/ 5-(EtO)2,2,4-F2,E) , [-3934:2-

Cl-3-F, 2f4-F2, E], [-3935:2-Cl-4-F, 2,4-F2, E], [-3936:2-01-5-F,2,4- F2, E], [-3937: 2-Cl-6-F, 2, 4-F2, E], [-3938: 3-C1-2-

Fr2,4-F2,E], [ -3939:3-Cl-4-F,2,4-F2 ,E ] , [ -3940:3-C1-5- 128 320202 200901876 F,2,4-F2 ,Ε] r 〔-3941:4-C1-2-F,2,4-F2,E] r [-3942:4-01-3-F,2,4-F2,Ε] / [-3943: 2-F-3-Me,2,4-F2,E ] r [-3944:2-F-4-Me, 2,4-F2,Ε] t [—3945 :2-F-5~Me, 2,4 —F2,E] r [-3946:2 — F—6~ Me,2,4-F2 ,Ε] r [-3947:3-F-2-Me,2,4-F2,E ] r [-394 8:3 —F—4- Me,2,4-F2 ,E] ' 〔394 9:3-F-5-Me,2,4-F2 ,E〕 r 〔-3950:4 -F-2- Me,2,4-F2,E] t C -3951:4-F-3-Me,2,4-F2,E] r [-3952:2-Cl-3-' Me, 2,4-F2,E] f [-3953:2-Cl-4-Me,2,4-F2,E] t [-3954:2-01-5- Me,2,4-F2,E] t C-3955: 2-Cl-6-Me, 2,4-F2, E] t C-3956: 3-Cl-2- Me, 2,4-F2, E] r [—3957 : 3-Cl -4-Me,2,4-F2 / E] t C-3958:3-Cl-5- Me,2,4-F2 ,E] t [-3959:4-Cl-2-Me,2,4 -F2,E] r [-3960:4-01-3- Me,2,4-F2,E] f [-3961:2-F-3-CF3,2,4-F2,E] r [- 3962: 2-F-4-CF3,2,4-F2,E] t [-3963:2-F-5-CF3,2,4-F2,E] f C-3964:2-F-6- CF3,2,4-F2, E ] r C-3965:3-F-2-CF3,2,4-F2,E] t [-3966:3-F-4-CF3,2,4-F2, E] r C-3967: 3-F-5-CF3, 2, 4-F2, E] r [-3968:4-F— 2-CF3,2,4-F2,E] r [-3969:4-F-3-CF3,2,4-F2,E] t C-3970:2 -Cl-3-CF3,2,4-F2>E] r [-3971:2-Cl-4-CF3,2,4-F2,E] r [-3972:2-01-5- CF3,2 ,4-F2,E] r [-3973:2-Cl-6-CF3,2,4-F2,E] f [-3974:3-01-2-CF3,2,4-F2,E] r [-3975:3-Cl-4-CF3,2,4-F2,E] r [-3976:3-01-5- CF3,2,4-F2,E] t C-3977 : 4-CI- 2-CF3,2,4-F2, E] ,[-3978:4-01-3-CF3,2r4-F2,E] r [-3979:2-Me-3-CF3,2,4-F2, E] r C-3980: 2-Me-4-CF3,2,4-F2,E] r [-3981:2-Me-5-CF3,2,4-F2,E] r [-3982:2 -Me-6- CF3,2,4-F2 ,E] r [-3983:3-Me-2-CF3,2,4-F2,E] t C-3984:3-Me-4-CF3,2 ,4-F2,E] r C-3985:3-Me-5-CF3,2,4-F2,E] r [-3986:4-Me-2-CF3,2,4-F2,E] r C-3987: 4-Me-3-CF3,2,4-Fz,E] r [-3988:2_F-3- Me〇,2,4-F2,E] r [-3989:2-F-4 -MeO,2,4-F2,E] r C-3990:2-F-5- 129 320202 200901876

MeO, 2,4-F2, E], [-3991: 2-F-6-MeO, 2, 4-F2, E], [-3992: 3-F-2-MeO, 2, 4-F2, E], [-3993: 3-F-4-MeO, 2, 4-F2, E], 〇 3994: 3-F-5-MeO, 2, 4-F2, e3, [-3995: 4-F -2-MeO,2,4-F2,E], [-3996:4-F-3-MeO,2,4-F2,E], [-3997:2-Cl-3-MeO,2,4 -F2,E],.[-3998:2-Cl-4-MeO,2,4-F2,E], [-3999:2-Cl-5-MeO,2,4-F2,E], [ -4000:2-01-6-MeO,2,4-F2,E], [-4001:3-Cl-2-MeO,2,4-F2,E], [-4002:3-Cl-4 -MeO,2,4-F2,E], [-4003:3-Cl-5-MeO,2,4tF2,E], [-4004:4-Cl-2-MeO,2,4-F2,E ], .C-4005: 4-Cl-3-MeO,2,4-F2,E], [-4006:2-Me-3-MeO,2,4-F2,E], [-4007 :2 -Me-4-MeO,2,4-F2,E], [-4008:2-Me-5-MeO, 2,4-F2,E], [-4009:2-Me-6-MeO,2 , 4-F2, E], [-4010:3-Me-2-MeO/2,4-F2,E], C-4011:3-Me-4-MeO,2,4-F2,E3, [ -4012:3-Me-5-MeO,2,4-F2,E], [-4013:4-Me-2-MeO,2,4-F2,E], [-4014:4-Me-3 -MeO,2,4-F2,E], C-4015:H,2,5-F2, [-4016:4-F,2,5-F2,E] , [-4017:4-F,2 , 5-F2, Z], [-4018: 4-gi, 2, 5-F2, E], [-4019: 4-Cl, 2, 5-F2, Z], [-4020: 4-Br, 2,5-F2, E], [ -4 021:4-1,2,5-F2,E], [-4022:4-Me ,2,5-F2,E] r C -4023:4-Me,2,5-F2,Z ] , C -4024:4-Et,2,5- F2,E) , [ -4025:4- C3H7,2,5-F2,E) , C -4026: 4-(Me) 2 CH, 2,5- F2,E], [-4027:4-CF3,2,5-F2.,E], [-4028:4-CF3,2,5-F2,Z], [-4029:4-C2F5,2,5-F2,e3, [-4030: 4-C3 F7,2,5-F2,E] , [-4031: 4-(CF3)2CF, 2,5-F2, E], [-4032: 4-(CF3)2CH, 2,5-F2, E], [-4033: 4-CHF2, 2 ,5-F2/e ] , c -4034:4-CH2F,2,5-F2 rE ) , [ -4035:4- CF3CH2,2,5-F2,E], [ -4036:4-MeO,2 ,5-F2,E],[ -4037:4-MeO,2,5-F2,Z],〇4038:4-EtO,2,5-F2,E],[-4039:4-C3H7O,2 , 5-F2, E], [-4040: 4-(Me) 2CHO, 2, 5-F2, E], [-4041: 4-N〇2, 2, 5-130 320202 200901876 F2/E], C-4042: 4-N〇2,2,5-F2,z] , C-4043:3-F, 2,5-F2 , E 3 , C-4044:3-F,2,5-F2, Z], [-4045: 3-Cl, 2, 5-F2, E], [-4046: 3-C1, 2, 5-F2, Z], [-4047: 3-Br, 2, 5-F2 , E], [-4048: 3-I, 2, 5-F2, E], [-4049: 3-Me, 2, 5-F2, E], [-4050: 3-Me, 2, 5- F2,Z], [-4051:3-Et,2,5-F2,E], [ -4052:3-C3H7,2,5-F2,E], [ -4053:3- (Me)2CH, 2,5-F2,E], [-4054:3-CF3,2,5-F2,E], [-4055:3-CF3,2,5~F2 ^ z ] , C — 4056 : 3~ 〇 2 F5, 2, 5 — F2 , E] , C — 4057 : 3—C3 F7, 2/5~ F2, E], [-4058: 3-(CF3)2CF, 2,5-F2,E],[-4D59:3-(CF3)2CH,2,5-F2,E] f C-4060:3-CHF2,2,5-F2,E] , [-4 061 : 3-CHF2,2,5-F2 , Z ], [-4062:3-CH2F,2,5-F2,E], [-4063:3-CH2F,2,5-F2,Z], [- 4064: 3-CF3CH2, 2,5-F2, E], C-4065: 3-MeO, 2,5-F2, Ej *, [-4066:3-MeO,2,5-F2,Z], -40.67:3-EtO,2,5-F2,E], [-4068:3-C3H7O,2,5-F2,E], [ -4069:3-(Me)2CHO,2,5-F2/ E ] , C -4070:3-N02,2,5- F2,E] , C-4071:2-F,2,5-F2,E] , [-4072 :2-C1, 2,5-F2 , E 3 , [-4073:2-Br,2,5-F2,E ] , [ -4074:2-1,2,5-F2 ,E 3 , [-4075:2-

Me, 2,5-F2, E], [-407 6:2-Et, 2,5-F2, E], [-4077:2-C3H7,2,5-F2,E], [-4078: 2-(Me)2CH.,2,5-F2,E], [-4079:2-CF3,2,5-F2,E], C -4080:2-C2F5,2,5-F2,E 3 , [ -4 081:2-C3 F7,2,5-F2 , E ], [- 4082:2-(CF3)2CF,2,5-F2,E], [-4083:2-(CF3)2CH , 2,5-F2,E], [-4084:2-CHF2,2,5-F2,E],.[-4085:2-CH2F,2,5-F2,E], [-4086:2 -CF3CH2,2,5-Fs,E], [ -4087:2-MeO,2,5-F2,E 3 , C -4088:2-

EtO,2,5-F2,E], [ -4089:2-C3H7O,2,5-F2,E], C -4090:2-(Me)2CHOr2,5-F2,E] , [-4091: 2-N02 r 2,5-F2 , E ] , [-4092:2,3- F2,2,5-F2,E] , [-4093:2,4-F2,2,5-F2,E] , [-4094 : 2,5-F2,2,5-F2,E], [-4095:2,6-F2,2,5-F2,E],[-4096:3,4-F2,2 ,5-F2,E], 131 320202 200901876 [-4097:3,4-F2,2,5-F2,Z], [-4098:3,5-F2,2,5-F2,E], -4099:3,5-F2,2,5-F2,Z) , [ -4100 : 2,3-Cl2,2,5-F2 , E], C - 4101:2,3-Cl2,2,5 -F2,Z ] , [ -4102:2,4-Cl2,2,5-F2,E], [- 4103:2,4-Cl2,2,5-F2,Z], [-4104:2, 5-Cl2,2,5-F2, E], [-4105:2,5-C1Z,2,5-F2,Z ], [ -4106:2, 6-Cl2,2,5-F2,E ] , [- 4107:3,4-Cl2,2,5-F2,E ] , [ -4108:3,5-Cl2,2,5-F2,E ] , C - 4109:2,3-Br2,2 , 5-F2, E], [-410:2,4-Br2,2,5-F2,E], [-4111:2,5-Br2,2,5-F2,E], [-4112: 2,6-Br2,2,5-F2,E],[- 4113:3,4-Br2,2,5-F2,E], [-4114:3,5-Br2,2,5-F2, E], [- 4115:2,3-Me2,2,5-F2,E 3 , [ -4116:2,4-Me2,2,5-F2,E],[- 4117:2,5-Me2 , 2,5-F2 , E ] , [ -4118 : 2,6-Me2,2, 5-F2*, E ), [- 4119:3,4-Me2,2,5-F2,E], -4120:3,5-Me2,2,5-F2,E],[-4121:2,3-Et2,2,5-F2,E], [-4122:2,4-Et2,2,5 -F2,E ],[- 4123:2,5-Et2,2,5-F2 ,E], [ -4124 :2,6-Et2,2,5-F2 , E ],[- 4125:3, 4-Et2,2,5-F2,E 3 , [ -4126: 3,5-Et2,2,5-F2, E], [- 4127:2,3-(CF3)2,2,5-F2 , E] , [-4128 : 2,4-(-CF3 ) 2,2,5-F2 , E], [-4129:2,5-(CF3)2,2,5-F2,E], [ -4130 : 2,6-(CF3 ) 2,2,5-F2 , E3 ,[-4131:3,4-(CF3)2,2,5-F2,E] , [-4132 : 3,5- (CF3) 2,2,5-F2, E], [-4133:2,3-(CHF2)2,2,5-F2,E], [-4134:2,4-(CHF2)2,2 ,5-F2,E]·, [-4135:2,5-(CHF2)2,2,5-F2,E], [-4136:2,6-(CHF2)2,2,5-F2, E] , 〔 -4137:3,4-(CHF2)2,2,5-F2,E] , C -4138:3,5- (CHF2)2,2,5-F2,E], 〔 -4139 :2,3-(CH2F)2,2,5-F2,E],[- 4140:2r4-(CH2F)2,2,5-F2,E] , [-4141:2,5-(CH2 F ) 2,2,5-F2 , E], [-4142:2,6-(CH2F)2,2,5-F2,E] r [ -4143 : 3,4-(CH2 F) 2,2, 5-F2,E] r 〔 -4144:3,5-(CH2F)2,2,5-F2,E] , C -4145:2,3- 132 320202 200901876 (MeO)2,2,5-F2 ,Ε), C-4146:2,4-(MeO)2,2,5-F2,E] , [-4147:2,5-(MeO)2,2,5-F2,E], [- 4148:2, 6-(MeO)2,2,5-F2,E], [-414 9:3,4-(MeO)2,2,5-F2,E] , (-4150 : 3, 5-(MeO) 2,2,5-F2 , E] , [-4151:2,3- (EtO)2,2,5-F2,E] , [-4152:2,4-(EtO)2,2,5-F2,E] , [-4153:2,5-(EtO)2,2 ,5-F2,E] , [-4154:2,6-(EtO)2,2,5-F2,E] , [-4155:3,4-(Et〇)2,2,5-F2, E], [-4156:3,5-(EtO)2,2,5-F2,E], [-4157:2-Cl-3-F, 2,5-F2, E], [-4158: 2-Cl-4-F,2,5-F2,E], [-4159:2-Cl-5-Fr2,5-F2,E], [-4160:2-Cl-6-F, 2, 5-F2,E], [-4161:3-Cl-2-F,2,5-F2,E], [-4162:3-Cl-4-F,2,5-F2,E], -4163:3-Cl-5-F,2,5-F2,E), [-4164:4-Cl-2-Fr2,5-F2,E), { -4165 : 4-C1-3- F , 2,5-F2 ,E ) , [ -4166:2-F-3-Me,2,5-F2 rE ] , ( -*4167:2-F-4-

Me,2,5-F2,E] , [ -4168:2-F-5-Me,2,5-F2 ,E ] , [-4169:2-F-6-

Me, 2,5-F2, E], [-4170: 3-F-2-Me, 2, 5-F2, E], [-4171: 3-F-4-Me, 2, 5-F2, E], [-4172: 3-F-5-Me, 2, 5-F2, E], [-4173: 4-F-2-Me, 2, 5-F2, E], [-4174: 4 -F-3-Me,2,5-F2,E], [-4175:2-Cl-3-Me,2,5-F2,E], [-4176:2-:Cl-4-Me, 2,5-F2,E], [-4177:2-Cl-5-Me,2,5-F2,E], C-4178:2-Cl-6-Me,2,5-F2,E ] , [-4179:3-01-2-Me,2,5-F2,E], C-4180:3-Cl-4-Me,2,5-F2,E], [-4181:3-01 -5-Me,2,5-F2,E] , C-4182:4-Cl-2-Me,2,5-F2,E3, C-4183:4-C1-3-Me,2,5- F2, E], [-4184: 2-F-3-CF3, 2, 5-F2, E], [-4185: 2-F-4-CF3, 2, 5-F2, E], [-4186 :2-F-5-CF3,2,5-F2,E] , [-4187:2-F-6- CF3,2,5-F2,E) , (-4188:3-F-2-CF3 , 2,5-F2,E) , [-418 9:3-F-4-CF3,2,5-F2,E], [-4190:3-F-5-CF3,2,5-F2, E], [-4191: 4-F-2-CF3, 2, 5-F2, E], C-4192: 4-F-3-CF3, 2, 5-F2, E], [-4193: 2 -01-3-CF3,2,5-F2,E], [-4194:2-Cl-4-CF3,2,5-F2,E], [-4195:2-Cl-5- 133 320202 200901876 CF3,2,5-F2,Ε], [-4196:2-Cl-6-CF3,2,5-Fz,Ε], [-4197:3-Cl-2-CF3,2,5-F2, E], [-4198: 3-Cl-4-CF3, 2, 5-F2, E], [-4199: 3-Cl-5-CF3, 2, 5-F2, E], [-4200: 4 -Cl -2-CF3,2,5-F2,E],.[-4201:4-Cl-3-CF3,2,5-F2,E], [-4202:2-Me-3-CF3,2, 5-F2, E], [-4203: 2-Me-4-CF3, 2, 5-F2, E], [-4204: 2-Me-5-CF3, 2, 5-F2, E], [ -4205: 2-Me-6-CF3, 2,5-F2, E], [-4206: 3-Me-2-CF3, 2, 5-F2, E], [-4207: 3-Me-4 -CF3,2,5-F2,E], [-4208:3-Me-5-CF3,2,5-F2,E], [-4209:4-Me-2-CF3,2,5-F2 , E], [-4210: 4-Me-3-CF3, 2, 5-F2, E], [-4211: 2-F-3-MeO, 2, 5-F2, E], [-4212: 2-F-4-Me〇,2,5-F2, E], [-4213:2-F-5-Me〇,2,5-F2,E], [-4214:2-F-6- MeO, 2,5-F2, E], [-4215: 3-F-2-Me〇, 2,5-F2, E], C-4216: 3-F-4-MeO, 2,5-F2 , E ] , [-*4217:3-F-5-MeO>2,5-F2,E] , [-4218:4-F-2-MeO,2,5-F2 , E] , [-4219 :4-F-3-MeO,2,5-F2,E] , [-4220:2-Cl-3-MeO,2,5-F2,E] , [-4221:2-Cl-4-MeO ,2,5-F2,E] , [-4222:2-Cl-5-MeO,2,5-F2 ,E) , [-4223:2-01-6-MeO,2,5-F2,E ], [-4224: 3-Cl-2-MeO, 2, 5-F2, E], [-4225: 3-Cl-4-MeO, 2, 5-F2, E], [-4226: 3- Cl-5-MeO,2,5-F2,E]r[-4227:4-Cl-2-MeO, 2,5-F2,.E] f [-4228 : 4-Cl-3-MeO, 2 ,5-F2,E] , C-4229:2-Me-3-MeO,2,5-F2,E] , [-4230:2-Me-4-MeO ,2,5-F2,E] , [-4231:2-Me-5-MeO,2,5-F2,E], [-4232:2-Me-6-MeO,2,5-F2,E ], [-4233: 3-Me-2-MeO, 2,5-F2, E]r [-4234:3-Me-4-MeO, 2,5-F2, E], [-4235:3- Me-5-MeO, 2,5-F2, E], [-4236: 4-Me-2-MeO, 2,5-F2, E], [-4237: 4-Me-3-MeO, 2, 5-F2, E], [-4238:H,3,4-F2,E], [-4239:4-F,3,4-F2,E], [-4240:4-F,3,4 -F2,Z], [-4241:4-Cl,3,4-F2,E], [-4242:4-C1,3,4-F2,Z3, [-4243: 4-Br,3,4 -F2 , E] , C-4244 : 4-1,3,4-F2 , E] r [-4245: 4-Me,3,4-F2,E], [-4246:4-Me,3, 4-F2, Z], [-4247: 4-, 134 320202 200901876

Et,3,4-F2/E '3 , [ -4248 :4-C3H7,3,4-F2,E] , i -4249:4- (Me)2CH,3,4-F2 ,E], -4250: 4-CF3,3,4-F2,E], [-4251:4-CF3,3,4-F2,Z], C-4252:4-C2F5,3,4-F2,E], [-4253: 4-C3 F7,3,4-F2,E], [-4254:4-(CF3)2CF,3,4-F2,E], [.-4255:4-(CF3)2CH, 3,4-F2,E], [-4256:4-CHF2,3,4-F2,E], [-4257:4-CH2F,3,4-F2,E], [-4258:4-CF3CH2 ,3,4-F2 ,E ] , C-4259 : 4-MeO, 3, 4-F2 , E 3 , C~ 4260:4-MeO,3,4-F2,Z],[-4261:4- EtO, 3,4-F2, E], [-4262:4-C3H70,3,4-F2/E], [-4263:4-(Me)2CHO,3,4-F2,E], [- 4264:4-N〇2,3,4-F2,E], C-4265:4-N02,3,4-F2,Z], C-4266:3-F, 3,4-F2,E] , [-4267: 3-F, 3, 4-F2rZ], [-426 &: 3-Cl, 3,4-F2, E], [-4269: 3-Cl, 3, 4-F2, Z] , [-4270: 3-Br, 3, 4-F2, E], [-4271: 3-I, 3, 4-F2, E], [-4272: 3-Me, 3, 4-F2, E], [-4273: 3-Me, 3, 4-F2rZ], [-4274: 3-Et, 3, 4-F2, E], [-4275: 3-C3H7, 3, 4-F2, E ], [-4276: 3-(Me) 2CH, 3, 4-F2, E], [-4277: 3-CF3, 3, 4-F2, E], [-4278: 3-CfF3, 3, 4 -F2,Z], [-4279:3-C2F5,3,4-F2,E], [-4280:3-C3F7,3,4-F2,E], [-4281: 3-(CF3)2CF, 3,4-F2, E], [-4282: 3-(CF3) 2 CH, 3,4-F2, E], [-4283:3-CHF2,3 , 4-F2 , E) , [-4284 : 3-CHF2,3, 4-F2 , Z], [-4285:3-CH2F,3,4-F2,E], [-4286:3-CH2F, 3,4-F2,Z], [-4287:3-CF3CH2,3/4-F2,e3[-4288:3-MeO, 3,4-F2, E], [-4289:3-MeO,3 , 4-F2, Z], [-4290: 3-EtO, 3, 4-F2, E], [-4291: 3-C3H7O, 3, 4-F2, E], [ -4292: 3-(Me ) 2CHO,3,4-F2 ,E ] , C -4293 : 3-N02,3,4- F2,E], [-4294:2-F,3,4-F2?E], [-4295: 2-Cl,3,4-F2,E], [-4296:2-Br,3,4-F2,E], C-4297:2-Ir3,4-F2,E 3 , [-4298:2 -

Me,3,4-F2,E], [-4299:2-Et,3,4-F2,E], [-4300:2-C3H7,3,4-F2,E], [-4301:2 -(Me)2CH,3,4-F2,E],[-4302:2-CF3,3,4-F2,E], 135 320202 200901876 [-4303:2-C2F5,3,4-F2 ,Ε ], C -4304:2-C3F7,3,4-F2,e] , C- 4305:2-(CF3 )2CF,3,4-F2 ,E] , [-4306 : 2-(CF3 ) 2 CH , 3, '4-F2 , E], [-4307:2-CHF2,3a4-F2 ,E] , [-4 308 : 2-CH2 F, 3,4-F2 , E] f [-4309:2 -CF3CH2,3, 4-F2,E], [ -4310:2-MeO,3,4-F2,E ], [ -4311:2-EtO,3,4-F2,E], [ -4312: 2-C3H7〇,3,4-F2,E 3 , [ -4313:2- (Me)2CHO,3,4-F2,E] , [-4314 :2-N02,3,4-F2 , E ] , [ -4315:2,3- F2,3,4-F2,E] , [-4316:2,4-F2,3,4-F2 ,E] , C-4317 :2,5-F2,3 , 4-F2, E], [-4318: 2, 6-F2, 3, 4-F2, E], [-4319: 3, 4-F2, 3, 4-F2, E], [-4320: 3,4-F2,3,4-F2,: 2] ,[-4321:3,5-F2,3,4-F2,E ] r [- 4322:3,5-F2,3,4-F2 ,Z] r [-4323:2,3-CI2,3,4-F2,E ] t C - 4324:2,3-Cl2,3,4-F2,Z ] t [-4325:2,4- Cl2,3,4-F2.,E] f [- 4326:2,4-Cl2,3,4-F2,Z] t [-4327:2,5-Cl2,3,4-F2,E] r C - 4328: 2,5-GI2,3,4-F2,Z ] r C -4329:2,6-Cl2,3,4-F2,E ] r [- 4330:3,4-Cl2,3, 4-F2 , E 〕 f 〔-4331:3,5-Cl2,3,4-F2,E] r [- 4332:2,3-Br2,3,4-F2,E] r [-4333:2,4- Br2,3,4-F2,E] t [- 4334:2,5-Br2,3,4-F2,E] r [-4335:2, 6-Br2,3, 4-F2,E ] f 〔 - 4336:3,4-Br2,3,4-F2,E 〕 r 〔-4337:3,5-Br2,3,4-F2,E 〕 r 〔- 4338:2,3-Me2,3,4 -F2,E 〕 r 〔-4339:2,4-Me2,3,4-F2,E 〕 t 〔- 4340:2,5-Me2,3, 4-F2 ,E ] r [-4341:2, 6-Me2,3,4-F2,E ] rc - 4342:3,4-Me2,3,4-F2 ,E] r [-4343:3,5-Me2,3,4-F2,E ] r [- 4344:2,3-Et2,3,4-F2,E ) r [-4345:2,4-Et2,3,4-F2,E ] r [- 4346:2,5-Et2,3, 4-F2,E] r C -4347:2,6-Et2,3,4-F2,E ] f [- 4348:3,4-Et2,3,4-F2,E ] r [-4349:3 ,5-Et2,3,4-F2,E 〕 r 〔- 4350:2,3-(GF3)2,3,4-F2,E] , [-4351: 2,4-(CF3 ) 2,3 , 4-F2 , E) , C-4352: 2,5-(CF3)2,3,4-F2,e3 , [-4353 : 2,6-(CF3 ) 2,3,4-F2 , E] , [- 136 320202 200901876 4354:3,4-(CF3)2,3,4-F2,E] , [-4355 : 3,5-(CF3 ) 2,3,4-F2 , E],[- 4356:2,3-(CHF2)2,3,4-F2,E],[-4357:2,4-(CHF2)2/3,4-F2,E], [-4358':2,5 -(CHF2)2,3,4-F2,E] , [-4359:2,6-(CHF2)2,3,4-F2,E]., [ -4360:3, 4-(CH F2) 2,3,4-F2,E ) , [ -4361:3, 5- (CHF2) 2,3,4-F2,E], [-4362:2,3-(CH2F)2,3, 4-F2,E],[- 4363:2,4-(CH2F)2,3,4-F2,E], [-4364:2,5-(CH2F)2,3,4-F2,E] , [-4365:2, 6-(CH2 F)2,3,4-F2,E], [ -4366: 3,4-(CH2 F) 2,3,4-F2,E], [ -4367 :3,5-(CH2F)2,3,4-F2,E 3 , [ -4368:2,3- (iyieO)2,3,4-F2,E],[-4369:2,4-( Me〇)2,3,4-F2,E],[-4370:2,5-(MeO)2,3,4-F2, [-4371: 2,6-(MeO) 2,3 f 4- F2 , E] , [-4372:3,4- (MeO) 2,3,4-F2,e3 , [-4373:3,5-(MeO) 2,3,4-F2 , E] , [- 4374:2,3-(EtO)2,3,4-F2,E], [-4375:2,4-(EtO)2,3,4-F2,E], [-4376:2,5- (Et〇) 2,3,4-F2,E], [-4377:2, 6-(EtO)2,3,4-F2,E], [-4378:3, 4-(Et〇)2 ,3,4-F2rE], [-4379:3,5-(Et〇)2,3,4-F2rE], [-4380:2-Cl-3-F,3,4-F2,E), C-4381: 2-Cl-4-F, 3,4-F2, E], [-4382: 2-01-5-F, 3, 4-F2, E], [-4383: 2-Cl- 6-F,3,4-F2,E], [-4384:3-01-2-F,3,4-F2,E], [-4385:3-Cl-4-F,3,4- F2 , E]r [ -438 6: 3-C1-5-F,3, 4-F2 ,E ] , [ -4387:4-Cl-2-F,3,4-.F2 ,E], [ -4388: 4-Cl-3-F,3,4-F2,E], [-4389:2-F-3-Me,3,4-F2,E], [-4390:2-F-4-

Me, 3,4-F2, E], [-4391: 2-F_5-Me, 3, 4_F2, E], C — 4392: 2 — F—6 — Me, 3, 4-F2, E ] , 〔 -4393: 3-F-2-Me, 3,4-F2, E], C-4394: 3-F-4-

Me,3/4-F2,E] , C-4395:3-F-5-Me,3,4-F2 ,E ] , [-4396: 4-F-2-

Me,3,4-F2,E] , [-4397 : 4-F-3-Me, 3,4-F2 , E ] , [-4398:2-01-3-Me,3,4-F2, E], C-4399: 2-Cl-4-Me, 3f4-F2, E], [-4400: 2-01-5-Me, 3, 4-F2, E], C-4401: 2-Cl -6-Me,3,4-F2,E ] , [-4402:3-Cl-2- 137 320202 200901876

Me,3,4-F2,Ε], [-4 403:3-Cl-4-Me,3,4-F2,E],

Me,3,4-F2,E] , [-4405:4-Cl-2-Me,3,4-F2,E], Me., 3,4-F2,E],[ -4 4 07 : 2-F-3-CF3,3,4-F2,E]CF3,3,4-F2,E],[-4409:2-F-5-CF3,3,4-F2,E] CF3,3 ,4-F2,E],[-4411:3-F-2-CF3,3,4-F2,E] CF3,3,4-F2,E], [-4413:3-F-5-CF3 ,3,4-F2 ,E] CF3,3,4-F2,E],[-4415:4-F-3-CF3,3,4-F2,E], CF3,3,4-F2,E ], [-4417: 2-Cl-4-CF3,3,4-F2,E]·CF3,3,4-F2,E],[-4419:2-Cl-6-CF3,3,4- F2, E], CF3,3,4-F2,E], [-4421:3-Cl-4-CF3,3,4-F2,E], CF3,3,4-F2,E],[- 4423: 4-Cl-2-CF3,3,4-F2,E], CF3,3,4-F2,E], C-4425:2-Me-3-CF3,3,4-F2,E] , CF3,3,4-F2,E], [-4427:2-Me-5-CF3,3,4-F2,E], CF3,3,4-F2,E], C-4429:3- Me-2-CF3,3,4-F2,E3, CF3,3,4-F2,E], [-4431:3-Me-5-CF3,3,4-F2,E], CF3,3, 4-F2,E],[-4433:4-Me-3-CF3,3,4-F2,E] Me〇,3,4-F2,E],[-4435:2-F-4-MeO ,3,4-F2,E] MeO, 3, 4-F2 ,E] , [-4437:2-F-6-Me〇,3,4-F2,E]

Me〇,3,4_F2,E], [a 4439:3-F-4-Me〇,3, 4-F2,E]

Me〇,3,4-F2,E] , [-4 441: 4-F-2-MeO, 3,4-F2 ,E ] MeO, 3, 4-F2 ,E) , [-4 443 : 2 -Cl-3-MeO, 3,4-F2, E], MeO,3,4-F2,E], [-4445:2-Cl-5-MeO,3,4-F2,E], MeO, 3,4-F2,E] , [-4 447 : 3-Cl-2-MeO, 3,4-F2 , E], MeO, 3,4-F2, E] , [-4449:3-Cl- 5-MeO,3,4-F2,E], MeO,3,4~F2,E] , [-4451:4-Cl-3-Me〇,3,4-F2,E] r [-4404: 3-01-5-[-4406:4-Cl-3-r [—4408:2-F-4-r [—4410:2—F—6—, [-4412:3-F-4-, C-4414: 4-F-2-[-4416:2-01-3-.[-4418:2-Cl-5-^ C-4420:3-Cl-2-C-4422:3-Cl- 5-[-4.424:4-Cl-3-[-4426:2-Me-4-[-4428:2-Me-6-C-4430:3-Me-4-[-4432:4-Me- 2-, C-4434: 2-F-3-, C-4436: 2-F-5-r C-4438: 3-F-2-, C-4440: 3-F-5-, C-4442 :4-F-3-[-4444:2-01-4-[-4446:2-Cl-6-[-4448:3-01-4-[-4450:4-01-2-[-4452 :2-Me-3- 138 320202 200901876

MeO,3,4-F2,Ε],.[-4453:2-Me-4-Me〇,3,4-F2,E],[-4454:2-Me-5-MeO,3,4- F2, E], [-4455: 2-Me-6-MeO, 3, 4-F2, E), [-4456: 3-Me-2-MeO, 3, 4-F2, E], [-4457 :3-Me-4-MeO,3,4-F2,E] , [-4458:3-Me-5-MeO,3,4-F2,E], [-4459:4-Me-2-MeO ,3,4-F2,E] , [-4460:4-Me-3-MeO,3,4-F2,E] , [-4461:H,3,5-C12,E] , [-4462: 4-F,3,5-Cl2,E], [-4463:4-F,3,5-Cl2,Z], [-4464:4-Cl,3,5-Cl2,E], [-4465 :4-Cl,3,5-Cl2,Z], [-4466:4-Br,3,5-Cl2,E], [-4467:4-I,3,5-C12,E], [- 4468: 4-Me,3,5-Cl2,E), [-4469: 4-Me, 3,5-Cl2, Z], [-4470:4-Et,3,5-Cl2,E], -4471: 4-C3H7,3,5-Cl2,E], [-4472:4-(Me)2CH,3,5-Cl2,E], [-4473:4-CF3,3,5-Cl2, E] , [-4474:4-CF3,3,5-C12,Z], [ -4475:4-C2 F5,3,5-Cl2,E], * [ -4476:4- C3F7,3,5 -Cl2, E], C-4477: 4-(CF3)2CF, 3,5-C12, E], [-4478:4-(CF3)2CH,3,5-Cl2,E], [-4479: 4-CHF2,3,5-Cl2,E], [-4480:4-CH2F,3,5-C12,E], [ -4481:4-CF3CH2,3,5-Cl2,E), [-4482 :4-

MeO,3,5-Cl2,E) , [-4483:4-MeO,3,5-Cl2,Z] , [-4484 : 4-EtO, 3, 5-C12,E] , C-4485:4 -C3H70,3f5-Cl2,E], [-4486: 4-(Me)2CHO,3,5-C12,E], [-4487:4-N02,3,5-Cl2,E], [-4488 :4-N02,3,5-Cl2,Z], [-4489:3-F,3,5-Cl2,E], C-4490:3-F, 3,5-Cl2,Z], [- 4491:3-C1,3,5-C12,E],[ -4492:3-d, 3,5-Cl2,Z ] , [ -44 93 : 3-Br, 3,5-

Cl2, E], [-4494: 3-I, 3, 5-Cl2, E], [-4495: 3-Me, 3, 5-Cl2, E], [-4496: 3-Me, 3, 5 -Cl2,Z), [-4497:3-Et,3,5-Cl2,E], [-4498:3-C3H7,3,5-Cl2,E), [-4499:3-(Me)2CH , 3,5-Cl2 , EJ , [-4500:3-CF3,3,5-Cl2,E ) , [ -45〇1:3-CF3,3,5-Cl2,Z], [ -4502:3 -C2F5 ,3,5-Cl2 ,E ] , [ -4503:3-C3F7,3,5-Gl2 ,E ] , C -4504:3-(CF3hCF,3,5-Cl2,E], [-4505 :3-(CF3>2CH,3,5-Cl2,E],[- 139 320202 200901876 4506:3-CHF2,3,5-Cl2,Ε], [-4055 : 3-CHF2,3,5-Cl2 , Z], [- 4508: 3-CH2F, 3,5-Cl2, E], C-4509: 3-CH2F, 3,5-Cl2, Z], [- 4510:3-CF3CH2,3,5- Cl2, E], C -4511: 3-MeO, 3,5-Cl2, E], [-4512:3-MeO,3,5-Cl2,z], (-4513:3-EtO,3f5-Cl2 , E] , [-4514:3-C3H70,3,5-C12,E] , [-4515:3-(Me)2CHO,3,5-Cl2,E], [-4516:3-N〇2 , 3r5-C12, E], [-4517: 2-F, 3, 5-C12, E], [-4518: 2-Cl, 3, 5-Cl2, E], [-4519: 2-Br, 3,5-Cl2,E],[-4520:2-I,3,5-Cl2,E], [-4521:2-Me,3,5-Cl2,E] r [-4522:2-Et ,3,5-Cl2,E], [-4523:2-C3H7,3,5-Cl2,E], [-4524:2-(Me)2CH,3,5-Cl2, EJ, [-4525: 2-CF3,3,5-Cl2,E],[-4 526: 2-C2F5,3,5-Cl2,E], C-4527:2-C3F7,3,5-C12,E], [-4528:2-(CF3)2CF,3,5-Cl2,E ]; [-4529:2-(CF3)2CH,3,5-C12 r E] , [-4530:2-CHF2,3,5-Cl2,E], [-4531:2-CH2 F,3, 5-C12, E], [-4532: 2-CF3CH2, 3, 5-Cl2, E], [-4533: 2-MeO, 3, 5-Cl2, E], [-4534: 2-EtO, 3 ,5-Cl2,E], [-4535:2-C3H7O, 3,5-Cl2,E], [-4536:2-(Me)2CHO,3,5-Cl2,E], [-4537:2 - N02,3,5-Cl2,E], [-4538:2,3-F2,3,5-Clz,E], [-4539:2, 4-F2,3,5-C12,E], [-4540:2,5-F2,3,5-Cl2,E], C-4541:2,6-F2,3,5-CI2, E], [-4542:3, 4-F2,3, 5-Cl2rE 3 , (-4543:3,4-F2,3,5-C12,Z], [-4544:3,5-F2,3,5-Cl2,E], [-4545:3,5 - F2,3,5-C12,Z], C -4546:2,3-CI2,3,5-Cl2,E ] f [-4547:2, 3- C12,3,5-C12,Z ], [-4548 : 2,4-Cl2,3,5-Cl2,E], [-4549:2,4-C12,3,5-C12,Z], [-4550:2,5-CI2,3, 5-CI2,E], [-4551:2,5- CI2,3,5-CI2 'Z], [-4552:2, 6-Cl2,3,5-Cl2,E], [-4553:3 , 4- C12,3,5-C12,E], [-4554:3,5-CI2,3,5-Cl2,E ], C-4555:2,3-Br2,3,5-C12,E ], [-4556:2,4-Br2,3,5-Cl2,E], [-4557:2,5-140 320202 2 00901876

Br2,3,5-C12,E ] , [ -4558:2,6-Br2,3,5-Cl2 , E ] , [-4559:3,4-

Br2,3,5-Cl2,E], [-4560:3,5-Br2,3,5-Cl2,E], [-4561:2,3-Μθ2 a 3 ^ 5-C12 ^ E ] , [ -4562 : 2,4-Me2,3,5-CI2 , E ] , [-4563:2,5- Μβ2 / 3 f 5-CI2 , E ] , C -4564 :2,6-Μθ2,3, 5 -CI2 , E ] , [-4565:3,4- Μθ2,3,5-CI2^E ] , [ -4 566:3,5-Μθ2,3,5-CI2 ,E ) , [-4567:2 , 3-

Et2,3,5-Cl2,E], [ -4568:2,4-Et2,3,5-Cl2,E ] , [-4569:2,5-

Et2,3,5-Cl2,E], [-4570:2,6-Et2,3,5-Cl2,E], [-4571:3,4-Et2,3,5-Cl2,E], [ -4572:3,5-Et2,3,5-Cl2,E ] , [-4573:2,3- (CF3)2,3,5-C12,E], [ -4574 :2,4-(CF3 ) 2,3,5-Cl2,E ),[- 4575:2,5-(CF3)2,3,5-Cl2,E] , [-4576:2, 6-(CF3)2,3,5 -Cl2,E], [-4577:3,4-(CF3)2,3,5-Cl2,E], [ -4578 : 3, 5-'(CF3 ) 2,3,5- C12,E] , [ -4579:2,3-(CHF2)2,3,5-Cl2,E], [ -45-80:2,4- (CHF2)2,3,5-C12,E], [-4581 :2,5-(CHF2)2,3,5-C12,E],[-4582:2,6-(CHF2)2,3'5-Cl2,E],[-4583:3,4-( CHF2) 2,3,5-Cl2,E], [-4584:3,5-(CHF2)2,3,5-CI2,E], [-4585:2,3-(CH2F)2,3, 5- C12,E] ,· [ -4586:2,4-(CH2F)2,3,5-Cl2,E ] , -[ -4587:2,5- (CH2F)2,3,5-Cl2 , E ] , [ -4588:2, 6-(CH2F)2,3,5-Cl2 ,E ],[- 4589:3, 4-(CH2'F)2,3,5-Cl2,E], -4590:3,5-(CH2F)2,3,5-Cl2,E], [-4591:2,3-(MeO)2,3,5-Cl2,E], [-4592: 2,4 -(MeO) 2,3, .5- C12,E 〕 , [ -4593:2,5-(MeO)2,3,5-Cl2,E], [ -4594:2,6- (Me〇) 2,3,5-Cl2,E], [ -4595:3,4-(MeO)2,3,5-Cl2, E),[- 4596:3,5-(MeO)2,3,5- CI2/E] , [-4597:2,3-(EtO)2,3,5-C L2,E] f [-4598:2,4-(EtO)2,3,5-Cl2,E ] , [ -4599:2,5-(EtO)2,3,5-C12,E 3 , [ -4600:2,6-(EtO)2,3,5-Cl2,E], [ -4601:3,4-(EtO)2,3,5-Cl2,E] , [-4602:3,5 -(EtO)2,3,5-Cl2,E] , [-4603:2- 141 320202 200901876

Cl-3-F,3,5-Cl2,Ε], [-4604:2-Cl-4-F,3,5-Cl2,Ε], [-4605:2-Cl-5-F:;3 , 5-Cl2, E], [-4606: 2-Cl-6-F, 3,5-Cl2, E]., [-46〇7:3-Cl-2-F,3,5-Cl2, E3, C-4608: 3-Cl-4-F, 3,5-Cl2, Ε], [-4609: 3-Cl-5-F, 3,5-Cl2, E], [-4610:4- Cl-2-F,3,5-Cl2,E],.[-4611:4-Cl-3-F,3,5-Cl2,E], [-4612:2-F-3-Me,3 , 5-Cl2, E], [-4613: 2-F- 4-Me, 3, 5-Cl2, E], [-4614: 2-F-5-Me, 3, 5-Cl2, E], [-4615: 2-F-6-Me, 3,5-Cl2, E], [-4616: 3-F-2-Me, 3r5-Cl2, E], [-4617: 3-F-4- Me,3,5-Cl2,E] , [-4618:3-F-5-Me,3,5-Cl2,E ] , [-4 619:4-F-2-Me,3,5-Cl2 , E], [-4620: 4-F-3-Me, 3, 5-Cl2, E], [-4621: 2-Cl-3-Me, 3, 5-Cl2, E], [-4622: 2-Cl-4-Me,3,5-Cl2,E], [-4623:2-Cl-5-Me,3,5-Cl2,E], [-4624:2-Cl-6-Me, 3,5-Cl2,E], [-4.625:3-Cl-2-Me,3,5-Cl2,E], [-4626:3-Cl-4-Me,3,5-Cl2,E] , [-4627: 3-Cl-5-Me, 3, 5-Cl. 2, E], [-4628: 4-Cl-2-Me, 3, 5-Cl2, E], [-4629: 4 -Cl-3-Me,3,5-Cl2,Ej, [-4630:2-F-3-CF3,3,5-Cl2,E], [-4631:2-F-4-CF3,3, 5-Cl2,E], [-4632:2-F-5-CF3,3,5-Cl2,E], [-4633:2-F-6-CF3,3,5-Cl2, E], [-4634: 3-F-2-CF5, 3, 5-Cl2, E], [-4635: 3-F-4-CF3, 3, 5-Cl2, E], C-4636:3 -F-5-CF3,3,5-Cl2,E3, [-4637:4-F-2-CF3,3,5-C12,eD, [-4638:4-F-3-CF3,3,5 -Cl2,E], [-4639:2-Cl-3-CF3,3,5-Cl2,E], C-4640:2-Cl-4-CF3,3,5-Cl2,E], [- 4641: 2-Cl-5-CF3,3,5-Cl2,E]r C -4642:2-Cl-6-CF3,3,5-Cl2,E],[-4643:3-Cl-2- CF3,3,5-Cl2,E], [-4644:3-Cl-4-CF3,3,5-Cl2,E], [-4645:3-Cl-5-CF3,3,5-Cl2, E 〕 , [ -4646:4-Cl-2-CF3,3,5-C12,E ], [ -4647:4-Cl-3-CF3,3,5-Cl2,E ] , [ -4648:2 -Me-3-CF3,3f5-Cl2,E3 f C-4649:2-Me-4-CF3,3,5-Cl2,E] , C-4650:2-Me- 5-CF3,3,5- Cl2, C-4651: 2-Me-6-CF3,3,5-Cl2, [-4652:3- 142 320202 200901876

Me-2-CF3,3f5-Cl2,Ε], [ -4653:3-Me-4-CF3,3,5-Cl2,E], [- 4654:3-Me-5-CF3,3,5- Cl2,E] ., [-4 655 : 4-Me-2-CF3,3,5-Cl2 , E], [-4656:4-Me-3-CF3,3,5-Cl2,E], [ -4657: 2-F-3-MeO,3,5-Cl2,E], [-4658:2-F-4-MeO,3,5-Cl2,E], [-4659:2-F-5 -Me〇,3,5-Cl2,E], [-4660:2-F-6-MeO,3,5-Cl2,E], [-4661:3-F-2-MeO,3,5- Cl2,E], [-4662:3-F-4-MeO,3,5-Cl2,E], [-4663:3-F-5-MeO,3,5-Cl2,E], [-4664 :4-F-2-MeO,3,5-Cl2,E],[-4665:4-F-3-Me〇,3,5-Cl2,E], [-4666:2-Cl-3- MeO,3,5-Cl2,E], [-4667:2-Cl-4-MeOf3,5-C12,E], [-4266:2-Cl-5-MeO,3,5-Cl2,E] , [ -4669:2-Cl-6-MeO, 3,5-CI2, E3 f [-4670:3-Cl-2-MeO,3,5-Cl2,E], [-4671:3-01- 4-MeO,3,5-Cl2,E], [-4672:3-Cl-5-MeO,3,5-Cl2,E]; [-4673:4-Cl-2-MeO,3,5- Cl2, E] , C -4674: 4-Cl-3-MeO, 3,5-Cl2, E), [- 4675: 2-Me-3-MeO, 3,5-Cl2, E), [-4676 :2-Me-4-MeO,3,5-Cl2,E], [-4677:2-Me-5-MeO,3,5-Cl2,E], C-4678:2-Me-6-MeOf3 , 5-

Cl2, E], [ -4679:3-Me-2-MeO,3,5-Cl2,E], [ -4680:3-Me-4-MeO,3,5-Cl2,E],·- 4681: 3-Me-5-MeO, 3,5-Cl2, E), [-4682·: 4-Me-2-Me〇, 3,5-Cl2, E], [-4683:4-Me- 3-MeO, 3,5-Clz, E], [- 4684:H,3-Cl-4-F,E], [-4685:4-F,3-Cl-4-F,E], [ -4686:4-F,3-Cl-4-F,Z]r C — 4687 :4-Cl,3-Cl-4-F,E] , (—4688 : 4-Cl, 3-Cl—4 - F,Z] , C-4689:4-Br,3-€l-4-F,E] , [-4690:4-1,3-C1-4-F,E],[-4691:4 -Me,3-Cl-4-F,E] , [-4692:4-Me,3-C1-4-F,Z] , [-4693:4-Et,3-Cl-4-F,E ], [ -4694:4-C3H7,3-Cl-4-F, E 0 , [-4695:4-(Me)2CH,3-Cl-4-F,E], [-4696:4-CF3 , 3-C1-4-F, E], [-4697:4-CF3,3-Cl-4-F/Z ] , [ -4698 :4-C2F5,3-Cl-4-F,E 3 , [ -4699:4-C3F7,3-Cl-4-F,E], [-4700:4- (CF3 )2CF, 3-Cl-4-F,E] , [-4701:4- 143 320202 200901876 (CF3)2CH,3-Cl-4-F,E], [-4702:4-CHF2,3-Cl-4-F,E], [-4703:4-CH2F,3-Cl-4-F , E], [-4704: 4-CF3CH2, 3-Cl-4-F, E]·, [-4705: 4-MeO, 3-Cl-4-F, E], [-4706: 4-MeO , 3-C1-4-F, Z]/ [-4707:4-EtO,3-Cl-4-F,E], [-4708:4-C3H7O,3-Cl-4-F,E], C -4709:4- (Me)2CH Q,3-Cl-4-F,E] , [-4710:4-N02,3-C1-4-F,E] r [-4711:4-N〇2,3-Cl-4-F, Z], C-4712: 3-F, 3-C1-4-F, E], [-4713: 3-F, 3-C1-4-F, Z], [-4714: 3-Cl, 3 -Cl-4-F, E], [-4715: 3-Cl, 3-Cl-4-F, Z], [-4716: 3-Br, 3-Cl-4-F, E 3 , [ - 4717: 3-1,3-C1-4-F, E 3 , [- 4718: 3-Me, 3-Cl-4-F, E] , [-4719: 3-Me, 3-C1-4- F,Z] , [-4720:3-Et,3-Cl-4-F,E ] r 〔 -4721:3-C3H7,3-Cl-4-FrE 〕 , [ -4722:3- (Me) 2CH,3-Cl-4-F,E] , [-4723:3-CF3,3-C1-4-F,E] ; [-4724:3-CF3,3-Cl-4-F,Z] , [-4725: 3-C2F5, 3-Cl-4-F, E], [-4726: 3-C3F7, 3-Cl-4-F, E), [-4727: 3-(CF3)2CF, 3-Cl-4-F,E) , [-4728:3-(CF3)2CH,3-Cl-4-F,E], C-4729:3-CHF2,3-Cl-4-F,E ], [-4730:3-CHF2,3-Cl-4-F,Z], [ -4731:3-CH2F,3-Cl-4-F,E ] ., [ -4732:3-CH2F,3 -Cl-4-F,Z] , [-4733:3-CF3CH2,3-Cl-4-F,E] , [-4734:3-

MeO, 3-Cl-4-F, E], [-4735: 3-MeO, 3-C1-4-F, Z], [-4736: 3-EtO, 3-

Cl-4-F,E] [-4737:3-C3H70,3-Cl-4-F,E) [-4738:3-(Me)2CHO,3-Cl-4-F,E], [- 4739:3-N02,3-Cl-4-F,E], [-4740:2-F,3-Cl-4-F,E], [-4741:2-01,3-Cl-4- F, E], C-4742: 2-Br, 3-C1-4-F, E], [-4743: 2-1,3-Cl-4-F, E], [-4744: 2-Mer3 -C1-4-F,E], [-4745:2-Et,3-Cl-4-F,E ) , [-4746:2-C3H7,3-C1-4-F,E ],[- 4747: 2-(Me)2CH, 3-Cl-4-F, E], C-4748: 2-CF3, 3-C1-4-F, E], [-474 9: 2-C2 Fs, 3 -Cl-4-F,E ] , [ -4750:2-C3F7,3-C1-4-F,E],[-4751:2-(CF3)2CF/3-Cl-4-F,E] , [-4752: 2-(CF3)2CH, 3-C1-4-F, E], 144 320202 200901876 [-4 753: 2-CHF2, 3-Cl-4-F, E], [-4754: 2-CH2F, 3-C1-4-F, E], [-4755: 2-CF3CH2, 3-Cl-4-F, E], [-4756: 2-MeO, 3-C1-4-F, E], [- 4757: 2-EtO, 3-Cl-4-F, E ] r [ -4758: 2-C3H70, 3-C1-4-F, E], [-4759: 2-(Me) 2CH〇,3-Cl-4-F,E], [-4760:2-NO2,3-Cl-4-F,E], [-4761:2,3-F2,3-Cl-4-F , E ] , [ -4762 : 2,4-F2,3-C1-4-F, E ], [- 4763:2,5-F2,3-Cl-4-F,E], [-4764: 2f6-F2,3-Cl-4-F,E],[- 4765:3,4-F2,3-Cl-4-F,E ] , [-4766 : 3, 4-F2,3-C1- 4-F, Z ], [- 4767:3,5-F2,3-Cl-4-F,E ] , (-4768 : 3,5-F2,3-C1-4-F , Z ], [- 4769: 2,3-Cl 2,3-Cl-4-F, E], [-4770:2,3-Cl 2,3-Cl-4-F,Z], [-4771: 2,4-Cl2,3-Cl-4-F,E], [-4772:2,4-Cl2,3-Cl-4-F,Z], [-4773:2,5-Cl2,3- Cl-4-F/E] , [-4774:2,5-Cl2,3-C1-4-F,Z],[- 4775:2, 6-Cl2,3-Cl-4-F,E] , C-4776: 3,4-Cl2,3-C1-4-F, E], [-4777:3,5-Cl2,3-Cl-4-F,E], C-4778:2,3 -Br2,3-C1-4-F,E] r [-4779:2,4-Br2,3-Cl-4-F,E] , C-4780:2,5-Br2,3-C1-4 -F,E],[-4781:2,6~Bx2/3—Cl-4—F, E ] , [ —4782:3,4-Br2^3-Cl—4-F, EJ, [-4783 :3,5-Br2,3-Cl-4-F,E] , [-4784:2,3-Me2,3-C1-4-F,EJ,[- 4785:2,4-Me2f3-Cl- 4-F,E] , [-4786:2,5-Me2,3-C1-4-F,E3,[- 4787:2,6-Me2,3-Cl-4-F,E), [- 4788:3,4-Me2/3-C1-4-F,E],[-4789:3,5-Me2,3-Cl-4-F,E], [-4790:2,3-Et2, 3-C1-4-F, E], [- 4791:2,4-Et2,3-Cl-4-F,E], C-4792:2,5-Et2,3-C1-4-F, E], [-4793: 2, 6-Et2, 3-Cl-4-F, E], C-4794: 3, 4-Et2, 3-C1-4-F, E) ./ [-4795: 3,5-Et2,3-Cl-4-F,E] ,[-4796:2,3-(CF3)2,3-C1-4-F,E], (-4797:2,4-( CF3) 2,3-Cl-4-FfE] , ' C-4798 : 2,5-(CF3 ) 2,3-C1-4-F,E] ., [-4799:2, 6-(CF3) 2,3-C1-4-F,e3, (-4800 : 3, 4-(CF3 ) 2,3-Cl-4-F,E], [ - 4801:3,5-(CF3)2,3-Cl-4-F,E ] f [ -4802:2,3- 145 320202 200901876 (CHF2)2,3-Cl-4-F,E], 〔 -4803 : 2,4-(CHF2)2,3-Cl-4-F,E], [- 4804:2,5-(CHF2)2,3-Cl-4-F,E], [-4805 :2,6-(CHF2)2,3-C1-4- F,E] , C -4806:3,4-(CHF2)2 , 3-Cl-4-F,E ) , C -4807:3 ,5-(CHF2)2,3-Cl-4-F,E] , (-4808:2,3-(CH2F)2,3-Cl-4-F,E],[- 4809:2, 4 -(CH2F)2,3-C1-4-F,E], [ -4810:2,5-(CH2F)2,3-C1-4-F,E], [-4811:2,6-( CH2F) 2,3-Cl-4-F,E], [ -4812:3,4-(CH2F)2,3-Cl-4-F,E], [-4813:3,5-(CH2: F) 2,3-Cl-4-F, E], [-4B14:2,3-(Me〇)2,3-Cl-4-F,E], [a 4815:2,4-(Me 〇)2,3-C1-4-F,E], [-4816:2,5-(MeO)2,3-Cl-4-F,E], [-4817:2,6-(MeO) 2,3-C1-4- F,E],[-4818:3,4-(MeO)2,3-Cl-4-F,E], [-4819:3,5-(MeO)2, 3-Cl-4-F,E],[ -4820:2,3-(EtO)2,3-Cl-4-F,E ] , C~4821:2, 4- (Et〇)2,3 -Cl-4-F,E 〕 , [ -4822:2,5-(EtO)2,3-Cl-4-F,E],[- 4823:2,6-(EtO)2,3-Cl -4-F, E], [-4824:3,4-(Et〇>2,3-Cl-4-F,E], [-4825:3,5-(EtO>2,3-Cl -4-F,E 〕 , [ -4826:2-C1-3-F,3-C1-4- F,E], [-4827:2-C1- 4-F,3-Cl-4-F,E] , [-4828:2-C1-5-F, 3-C1-4-F,E] ·, -[-4829:2-01-6- Γ,3-01-4-Ε,Ε], [-4 830 : 3'-Cl-2-F, 3-C1-4-F, E], [-4 831:3-Cl-4-F ,3-Cl-4-F,E] , [-4 832:3-C1-5-F, 3-C1-4-F,E) , C-4833:4-Cl-2-F,3- Cl-4-F, E] , C-4834: 4-C1-3-F, 3-C1-4-F, E], [-4835: 2 —F-3-Me, 3-Cl-4 — F,E] , [-4836:2-F—4—Me, 3~Cl-4-F, E〇, [-4837:2-F-5-Me,3-Cl-4-F,E] , [-4838:2-F-6-Me,3-C1-4-F, E], [— 4 839:3~F—2—Me, 3-Cl—4-F, e3, [—4840 :3-F—4—Me, 3~Cl—4—. F, E], [-4841: 3-F-5-Me, 3-Cl-4-F, E], [-4842:4- F-2-Me,3-Cl-4-F,E] f [—4843:4—F~3~Μθ,3-Cl—4-FfE), [—4844:2-Cl-3-Me, 3-Cl-4-F,E] , C-4845:2-Cl-4-Me,3-Cl-4-F,E) , [-4846:2-Cl-5-Me,3-Cl- 4-F, E], [-4847: 2-Cl-6-Me, 3-Cl-4-F, E], [-4848: 3-C1-2- 146 320202 200901876

Me, 3-Cl-4-F, E],. [-484 9 : 3-Cl-4-Me, 3-C1-4-F, E], [-4850: 3-d-5-Me, 3-Cl-4-F,E] , [-4851:4-Cl-2-Me,3-Cl-4-F,E] , [-4852:4-Cl-3-Me,3-Cl- 4-F,E ] , [ -4853:2-F-3-CF3,3-C1-4-F, E], [- 4B54:2-F-4-CF3,3-Cl-4-F, E], [-4855: 2-F-5-CF3, 3-Cl-4-F, E], C-4856: 2-F-6-CF3, 3-Cl-4-F, E], [ -4857: 3-F-2-CF3,3-C1-4-F,E],[-4 858:3-F-4-CF3,3-Cl-4-F,E], [-4859: 3-F-5-CF3,3-C1-4-FrE]r [-4860:4-F-2-CF3,3-Cl-4-F,E] , [-4861:4-F-3- CF3,3-Cl-4-F,E] , [-4862:2-Cl-3-CF3,3-Cl-4-F,E] , [-4863:2-C1-4-CF3,3- Cl-4-F,E] , C-4864:2-Cl-5-CF3,3-Cl-4-F,E] , [-4865:2-CI-6-CF3,3-Cl-4- F,E] , [ -4866:3-Cl-2-CF3,3-Cl-4-F,E ], [- 4867:3-Cl-4-CF3,3-Cl-4-F/E] , [-4868:3-Cl-5-CF3, J-C1-4-F, E], C-4869:4-C1-2-CF3 f3-C1-4 —F,E ] t [-4870: 4-Cl-3—CF3,3-Cl—4 — F,E] , [-4871:2-Me-3-CF3,3-Cl-4-F,E] , [-4872:2-Me- 4-CF3,3-Cl-4-F,E], C-4873:2-Me-5-CF3,3-Cl-4-F,E], C~4874:2-Me-6-CF3, 3-Cl-4-F,E] , [-4875:3-Me-2-CF3,3-Cl-4-F,E] r [-4876:3-Me-4-CF3,3-Cl- 4-F, E], [-4877: 3-Me-5-CF3, 3-C1-4-F, E , [- 4 87 8 : 4-Me-2-CF3,3-Cl-4-F, E] , [-4879: 4-Me-3-CF3,3-C1-4-F, E], [ -4880: 2-F-3-MeO, 3-Cl-4-F, E], [-4881: 2-F-4-MeO, 3-C1-4-F, E], C-4882:2 -F-5-MeO,3-Cl-4-F,E] , [-4883:2-F-6-MeO,3-C1-4-F,E], C-4884:3-F-2 -MeO,3-Cl-4-F,E] , [-4885:3-F-4-Me〇,3-Cl-4-F,E] r [-4886:3-F-5-Me〇 , 3-Cl-4-F, E], [-4887: 4-F-2-

MeO, 3-Cl-4-F, E], [-4 888 : 4-F-3-MeO, 3-C1-4-F, E ) , [-4889:2-

Cl-3-MeO,3-C1-4-F, E] , [-4890:2-Cl-4-Me〇,3-Cl-4-F,E], [- 4891:2-Cl-5 -MeO,3-Cl-4-F,E) , [-4892 :2-Cl-6-MeO, 3-C1-4-F,E], C-4 8 93:3-Cl-2-MeO ,3-Cl-4-F,E ] , C-4 8 94:3-Cl-4-MeO,3-C1-4- 147 320202 200901876 F,E],[-4895:3-Cl-5- MeO, 3-Cl-4-F, E], [-4896: 4-Cl-2-MeO, 3-Cl-4-F, E], C-4897: 4-Cl-3-MeO, 3- Cl-4-F, E] , C-4898: 2-Me-3-

MeO, 3-Cl-4-F, E], [-4899: 2-Me-4-MeO, 3-Cl-4-F, E], [-4900: 2-Me-5-MeO, 3- C1-4-F, E ] , [-4901: 2-Me-6-MeO, 3-C1-4-F, E], [- 4902: 3-Me-2-MeO, 3-Cl-4- F, E] , [-4903: 3-Me-4-MeO, 3-C1-4-F, E], [-4904: 3-Me-5-MeO, 3-C1-4-F, E] , C-4905: 4-Me-2-MeO, 3-C1-4-F, E], C-4906: 4-Me-3-MeO, 3-Cl-4-F, E], [-4 907.: H, 4-C1-3-F, E), [-4908: 4-F, 4-Cl-3-F, E], [-4909: 4-F, 4-C1-3-F , Z], [-4910: 4-Cl, 4-Cl-3-F, E], [-4911: 4-01,4-Cl-3-F, Z], [-4912: 4-Br, 4-C1-3-F, E], [-4 913: 4-Ί, 4-Cl-3-F, E], [-4914: 4-Me, 4-C1-3-F, E], C -4915:4-Me,4-C1-3-F,Z ] , [ -4916:4-Et,4-C1-3-F,E ),[- 4917:4-C3H7,4-Cl- 3-F, E], [-4918: 4-(Me) 2CH, 4-C1-3-F, E], [-4919: 4-CF3, 4-Cl-3-F, E], [- 4920: 4-CF3,4-C1-3-F,Z ], [- 4921:4-C2F5,4-Cl-3-F,E ] , [ —4922 : 4-C3 F7,4-Cl-3 —F, EJ ,[— 4923:4-(CF3)2CF,4-Cl-3-F,E] , [-4924 : 4-(CF3 ) 2 CH, 4-C1-3-F, E], C-4925: 4-CHF2,4-Cl-3-F, E), [-4926:4-CH2F,4-C1-3-F,E], (-4 927:4-CF3CH2,4-Cl -3-F,E ] , [ -4 928:4-MeO, 4-Cl-3-F,E ], [- 4929:4-MeO,4-Cl-3-F,Z ], [ -4930 :4-EtO,4-C1-3-F , E 〕, [- 4 931: 4-C3H70/4-Cl-3-F, E], [-4932: 4-(Me) 2CHO, 4-C1-3-F, E], [-4933: 4-N02,4-Cl-3-F,E], [ -4934 :4-N02,4-C1-3-F, Z ], [- 4935:3-F,4-Cl-3-F, E], [-4936: 3-F, 4-Cl-3-F, Z], [-4937: 3-Cl, 4-Cl-3-F, E], [-4938: 3-Cl, 4 -Cl-3-F,Z], [-4939:3-Br,4-C1-3-F,E], [-4940:3-1,4-Cl-3-F,E), [- 4941: 3-Me, 4-C1-3-F, E), [-4942: 3-Me, 4-Cl-3-F, Z], C-4943: 3-Et, 4-C1-3- F,E ],[- 4944:3-C3H7,4-Cl-3-F,E] , [-4945:3-(Me)2CH,4-C1-3-F,E],[- 148 320202 200901876 4946: 3-CF3,4-Cl-3-F,E 〕 r 〔 -4947:3-CF3,4-C1-3-F,Z 〕,[-4948:3-C2F5,4-Cl-3 -F,E], C -4 94 9:3-C3 F7,4-C1-3-F, E ], [-4 950:3-(CF3)2CF,4-Cl-3-F,E] , [-4951: 3-(CF3)2CH, 4-C1-3-F, E], [-4952: 3-CHF2, 4-Cl-3-F, E], [-4953: 3-CHF2, 4-Cl-3-F, Z], [-4954: 3-CH2F, 4-Cl-3-F, E 3 , C -4955 : 3-CH2 F, 4-C1-3-F, Z 3 , [- 4956: 3-CF3CH2, 4-Cl-3-F, E], C-4957: 3-MeO, 4-C1-3-F, E], [-4958: 3-MeO, 4-Cl- 3-F,Z ] , C -4959:3-EtO,4-C1-3-F,E 3,(- 4960:3-C3H7O,4-Cl-3-F,E], [-4961:3 -(Me)2CHO,4-C1-3-F,E], [-4962:3-N〇2,4-Cl-3-F,E ], [ -4963:2-F,4-C1-3-F,E ], [-4964:2-Cl,4-Cl-3-F,E^ , [-4965:2-Br,4- C1-3-F, E), [-4966: 2-I, 4-Cl-3-F, E], C-4967: 2-Me, 4-Cl-3-F, E], [-4968 :2-Et,4-C1-3-F,E] , [-4969:2-C3H7,4-Cl-3-F,E] , [-4970:2-(Me)2CH,4-C1- 3-F, E], [-4971: 2-CF3, 4-Cl-3-F, E], [-4972: 2-C2F5, 4-Cl-3-F, E], [-4 973: 2-C3 F7 , 4-C1-3-F, Ej , [-4 974 : 2-(CF3 ) 2 CF, 4-C1-3-F, E], [-4975: 2-(CF3 ) 2CH, 4-Cl-3-F,E], [-4976:2-CHF2,4-C1-3-F,E], C-4977:2-CH2F,4-Cl-3-F,E]· , C-4 97 8 : 2-CF3 CH2 , 4-C1-3-F, E] , [-4979: 2-MeO, 4-Cl-3-F, E], [-4980: 2-EtOr4-C1 -3-F,E], C-4981:2-C3H7〇,4-Cl-3-FrE], [-4982:2-(Me)2CHO,4-C1-3-F,E], [- 4983: 2-N〇2,4-C1-3_F,E],[—4984:2,3-F2,4—Cl-3—F,E ] r [-4985:2,4-F2 f4-Cl -3-FrE ] , [-4986: 2,5-F2 , 4-Cl-3-F, E ], [- 4987:2,6-F2 ,4-Cl-3-F,E ] , [- 4 988 : 3,4-F2 , 4-C1-3-F, E ] , C- 4989:3, 4-F2 ,4-Cl-3-F,Z ] , [-4 990 : 3,5- F2, 4-C1-3-F, E), [- 4991:3,5-F2,4-Cl-3-F,Z] , C-4992:2,3-Cl2,4-C1-3- F, E3, [-4993: 2, 3-CI2, 4-Cl-3-F, Z], [-4994: 2, 4-Cl2, 4-C1-3-F, E3, C-4995: 2,4-CI2,4-Cl-3-F,Z}, [-4996:2,5-Cl2,4-C1-3-F, E3,[- 149 320202 200901876 4997:2, 5-Cl2,4-Cl-3-F,Z], [-4998:2,6-Cl2,4-C1-3-F,E), C-4999:3,4-Cl2,4-Cl- 3-F,E] , C-5000:3,5-Cl2,4-C1-3-F,E],[-5001:2,3-Br2,4-Cl-3-F,E), -5002: 2., 4-Br2,4-C1-3-F, E], [-5003:2,5-Br2r4-C1-3-F,E), [-5004:2,6-Br2, 4-Cl-3—F, E], [-5005:3,4-Br2,4-Cl-3-F,E], C-5006:3,5-Br2r4-C1-3-F,E] , [-5007: 2,3-Me2,4-Cl-3-F, E], [-5008: 2,4-Me2,4-C1-3-F, E], [-5009:2,5 -Me2,4-Cl-3-F,E] f C-5010:2,6-Me2,4-C1-3-F,E],[-5011:3,4-Me2,4-Cl-3 -F,E] f C-5012:3,5-Me2,4-C1-3-F,E3,C-5013:2,3-Et2,4-Cl-3-F,E] r C-5014 :2,4-Et2,4-C1-3-F,E3 Λ [-5015:2,5-Et2,4-Cl-3-F,E] , [-5016:2r6-Et2 , 4-C1- 3-F, E3, [-5017:3,4-Et2,4-Cl-3-F,E], [-5018:3,5-Et2, 4-C1-3-F, E], [- 5019:2,3-(CF3)2,4-Cl-3-F,E], [-5020:2,4-(CF3)2,4-Cl-3-F,E], [-5021: 2,5-(CF3)2,4-Cl-3-F,E], [-5022:2,6-(CF3)2,4-C1-3-F,E], [-5023:3, 4-(CF3)2,4-Cl-3-F,E], [-5024:3,5-(CF3)2,4-Cl-3-F,E], [-5025:2,3- (CHF2)2,4-Cl-3-F,E], -5026:2,4-(CHF2)2,4-Cl-3-F>E]r C-5027:2,5-(CHF2)2,4-Cl-3-F,E] ·, C~ 5028:2,6-(CHF2>2,4-Cl-3-F,E], [-5029:3,4-(CHF2)2,4-C1-3-F,E], [-5030: 3,5-(CHF2)2,4-Cl-3-F,E], [ -5031:2,3- (CH2F)2, 4-Cl-3-F,E], [-5032:2, 4-(CH2F)2,4-Cl-3-F,Έ], [- 5033:2,5-(CH2F)2,4-Cl-3-F,E],[ -5034:2, 6- (CH2F)2,4-C1-3-F,E], [-5035:3,4-(CH2F)2,4-Cl-3-F,E], C -5036:3,5- (CH2F ) 2,4-Cl-3-F,E ] , C-5037:2/3-(MeO)2,4-Cl-3-F,E ],[- 5038:2,4-(MeO)2 , 4-Cl-3-F, E], [-5039:2,5-(MeO)2,4-Cl-3-F,E], [-5040:2,6-(MeO)2,4 -Cl-3-F,E] , C-5041:3,4-(MeO)2,4-C1-3-F,E] , [-5042:3,5-(MeO)2,4-Cl -3-F,E] , [-5043:2,3-(EtO)2,4- 150 320202 200901876

Cl-3-F, E], [ -5044:2,4-(EtO)2,4-Cl-3-F,E ] , [ -5045:2,5- (Et〇) 2,4-Cl -3-F,E] , [ -5046:2, 6-(EtO)2 ,4-Cl-3-F,E ], [- 5047:3,4-(EtO)2,4-Cl-3 -F,E], [-5049:2-Cl-3-F,4-Cl-3-F,E], [-5051:2-C1-5-F, 4-Cl~3-F, E ], [-5053: 3-Cl-2-F, 4-Cl-3-F, E], C-5055: 3-Cl-5-F, 4-Cl-3-F, E], C- 5057: 4-Cl-3-F, 4-Cl-3-F, E], [-5048:3,5-(EtO)2,4-Cl-3-F,E], [-5050:2 -Cl-4-F,4-C1-3-F,e], [-5052:2-Cl-6-F, 4-C1-3-F, e3, [-5054:3-Cl-4- Ff 4-Cl-3-F, E], [-5056:4-Cl-2,F, 4-Cl-3—F, e3, [-5058:2-F-3-Me,4-Cl- 3-F,E] r C-5059:2-F-4-Me,4-Cl-3-F,E] , [-5060:2-F-5-Me,4-C1-3-F, E], C-5061: 2-F-6-Me, 4-Cl-3-F, E], [-5062: 3-F-2-Me, 4-C1-3-F, E], [ -5063: 3-F-4-Me, 4-Cl-3-F, E], [-5064: 3-F-5-Me, 4-Cl-3-F, E], [-5065: 4 -F-2-Me,4-Cl-3-F,E], [-5066:4-F-3-Me,4-C1-3-F,E], [-5067:2-Cl-3 -Me, 4-Cl-3-F,E), [ -5068 : 2-Cl-4-Me,4-C1-3- F,E] , [-5069:2-Cl-5-Me,4 -Cl-3-F,E] , [-5070:2-Cl-6-Me,4-C1-3-F,E], [-5071:3-Cl-2-Me,4-Cl-3 -F,E] , [-5072:3-Cl-4-Me,4-Cl-3-F,E], [-5073:3-Cl-5-Me, 4-Cl-3 -F,.E],[-5074 : 4-C1-2-

Me, 4-Cl-3-F, E], [-5075: 4-Cl-3-Me, 4-C1-3-F, E] r [-5076: 2-F-3-CF3,4- Cl-3-F,E] r C-5077:2-F-4-CF3,4-Cl-3-F,E] , [-5078:2-F-5-CF3,4-Cl-3- F,E ) r C -5079:2-F-6-CF3,4-Cl-3-FfE ], [-5080:3-F-2-CF3,4-Cl-3-F,E] , -5081: 3-F-4-CF3, 4-C1-3-F, E], C -5082: 3-F-5-CF3, 4-C1-3-F, E], [ -5083 : 4 -F-2-CF3,4-C1-3- F,E) f C-5084;4-F-3-CF3,4-Cl-3-F,E] f [-5085: 2-Cl-3 -CF3,4-C1-3-F,E],[-5086:2-Cl-4-CF3,4-Cl-3-F,E], [ -5087:2-C1-5-CF3,4 -Cl-3-F, E], [-5088: 2-Cl-6-CF3, 4-Cl-3-F, E], [-5089: 3-CI-2-CF3, 4-Cl-3 -F, E 3 , [ -5090:3-Cl-4-CF3,4-Cl-3-F,E ], [- 151 320202 200901876 5091:3-Cl-5-CF3,4-Cl-3- F,E] , [-5092:4-Cl-2-CF3,4-C1-3-F,E], [-5093:4-Cl-3-CF3,4-Cl-3-F,E] , [ -5094:2-Me-3-CF3,4-C1-3-F,E) , C-5095:2-Me-4-CF3,4-Cl-3-F,E] , (-5096 :2-Me-5-CF3,4-Cl-3-F,E] , [-5097:2-Me-6-CF3,4-Cl-3-F,E] , [-5098:3-Me -2- CF3,4-Cl-3-F,E) , C-5099:3-Me-4-CF3,4-Cl-3-F,E) , [-5100:3-Me-5-CF3 , 4-C1-3-F, E ] , [-5101: 4-Me-2-CF3, 4-C1-3-F, E], [-5102: 4-Me-3-CF3, 4-Cl -3-F,E] , [-5103:2-F-3-MeO,4-C1-3-F,E], [ -5104: 2-F-4-MeO, 4-Cl-3-F, E] · C -5105: 2-F-5-MeO, 4-C1-3-F, E], C-5106:2 -F-6-MeO,4-Cl-3-F,E] , [-5107:3-F-2-MeO,4-C1- 3-FrE] , [-5108:3-F-4-MeO ,4-Cl-3-F,E] , C-5109:3-F-5-MeO,4-

Cl-3-F,E ] , C-5110:4-F-2-MeO,4-Cl-3-F,E ] , [ -5lll:4-F-3-

MeO,4-Cl-3-F,E] , [-5112:2-Cl-3-MeO, 4-C1-3-F,E] , [-5113:2-Cl-4-MeO,4- C1-3-F, E ] , [ -5114: 2-Cl-5-MeOr4-C1-3-F, E ], [- 5115: 2-Cl-6-MeO, 4-Cl-3-F, E] , C-5116: 3-Cl-2-MeO, 4-C1-3-F, E], [-5117: 3-Cl-4-MeO, 4-Cl-3-F, E], C -5118:3-Cl-5-MeO,4-C1-3-F,E]r [-5119:4-Cl-2-MeO,4-Cl-3-F,E], [-5120:4 -Cl-3-Me〇,4-Cl-3-F,E] , [-5121:2-Me-3-MeO,4-C1-3-F,E] , C-5122:2-Me- 4-

MeO,4-Cl-3-F,E] , [-5123:2-Me-5-MeO,4-C1-3-F,E] , [-5124:2-Me-6-MeO,4- C1-3-F, E 3 , C-5125: 3-Me-2-MeOr 4-Cl-3-F, E ], 512 6:3-Me-4-MeO, 4-Cl-3-F, E] , [-5127:3-Me-5-MeO,4-C1-3-F,E], [-5128:4-Me-2-MeO,4-Cl-3-F,E], C -5129: 4-Me-3-MeO, 4-C1-3-F, E], [ -5130:H,3-F-4-(Me)3C〇,E], [ -5131:4-F ,3-F-4-(Me)3CO,E] r C-5132:4-F,3-F-4-(Me)3CO,Z] f [-5133:4-C1,3-F- 4 - (Me)3CO,E] , [-5134:4-Cl,3-F-4-(Me)3CO,Z] , [-5135:4-Br,3-F-4-(Me)3C〇 , E], [ -5136:4-1,3-F-4-(Me)3CO, E 3 , [ -5137:4- 152 320202 200901876

Me, 3-F-4-(Me)3CO, E], [-5138:4-Me,3-F-4-(Me)3CO,Z],[- 5139:4-Et,3-F- 4-(Me)3CO,E] , [-5140:4-C3H7.3-F-4-(Me)3CO,E], [-5141:4-(Me)2CH,3-F-4-( Me)3C〇,E ] , C -5142:4-CF3,3-F-4-(Me)3CO,E 〕 . , [ -5143:4-CF3,3-F-4-(Me)3COrZ ] , [-5144:4-C2F5,3-F-4-.(Me)3CO,E], [-5145:4-C3F7,3-F-4-(Me)3CO,E],[a 514 6 :4-(CF3)2CF,3-F-4-(Me)3C〇,E] ,[-5147 : 4-(CF3 ) 2 CH, 3-F-4-(Me)3CO,E] , [ -5148: 4-CHF2,3-F-4-(Me>3C〇,E], [-5149:4-CH2F,3-F-4-(Me)3CO,E]f[-5150 : 4- CF3CH2,3-F-4-(Me) 3CO, E], [-5151:4-MeO,3-F-4-(Me)3CO,E ) , , [ -5152:4-MeO,3-F -4- (Me)3CO,Z 〕 , [ -5153:4-EtO,3-F-4-(Me)3CO,E ] , C -5154:4-C3H70,3-F-4-(Me) 3CO,E], [-5155:4-(Me)2CHO,3-F-4-(Me)3CO,E], [-5156:4-N〇2,3-F-4-(Me)3CO , E ] , C -5157:4-N02,3-F-4- (Me)3CO,Z] , C-5158:3-F,3-F-4-(Me)3CO,E] , [- 5159: 3-F, 3-F-4-(Me)3CO, Z] r [-5160:3-Clr3-F-4-(Me)3CO,E], [-5161:3-C1,3- F-4-(Me)3CO,Z],.[-5162:3-Br,3-F-4-(Me)3CO,E],[-5163:3-1,3-F-4-( Me) 3-C〇, E], [-516 4 : 3-Me, 3-F-4-(Me) 3CO, E ] , [-5165:3-

Me,3-F-4-(Me)3CO,Z ] , C -5166:3-Et,3-F-4-(Me)3CO,E 3 ,[- 5167:3-C3H7,3-F- 4-(Me)3CO,E], C-5168:3-(Me)2CH,3-F-4-(Me)3CO,E],[-5169:3-CF3,3-F-4-( Me) 3CO, E], [-5170: 3_CF3, 3-F-4-(Me)3CO, Z], C-5171: 3-C2F5, 3-F-4-(Me)3CO, E], [ -5172: 3-C3F7, 3-F-4-(Me)3CO, E], [-5173: 3-(CF3)2CF, 3-F-4-(Me)3CO, E], [-5174: 3-(CF3)2CH,3-F-4-(Me)3CO, E3, [-5175:3-CHF2,3-F-4-(Me)3CO,E], [ -5176:3-CHF2, 3-F-4-(Me)3CO,Z ] , [-5177:3-CH2F,3-F-4-(Me)3CO,E],[-5178:3-CH2F,3-F-4- (Me)3CO,Z],[-5179:3-CF3CH2,3-F-4-(Me)3CO,E], [ -5180:3-MeO,3-F-4- 153 320202 200901876 (Me) 3CO, .E], [-5181: 3-MeO, 3-F-4-(Me)3CO, Z], [-5182: 3-EtO, 3-F-4-(Me)3CO, E], C-5183: 3-C3H7〇, 3-F-4-(Me)3CO, E], [-5184: 3-(Me)2CHO, 3-F-4-(Me)3C〇, E], [ -5185:3-N02,3-F-4-(Me)3CO,E], C-5186:2-F,3-F-4-(Me)3〇〇,Ej, C-5187:2- C1, 3-F-4-(Me)3CO, E], [-5188: 2-Br, 3-F-4-(Me)3CO, E], [-5189: 2-1,3-F- 4-(Me)3CO,E], [-5190:2-Me,3-F-4-(Me)3CO,E 3 · { -5191:2-Et,3-F-4-(Me)3CO , E], [-5192: 2-C3H7, 3-F_4-(Me) 3CO, E],.[-5193:2-(Me)2CH,3-F-4-(Me)3CO,E] f C-5194 :2-CF3,3-F-4-(Me) 3 CO, E 3,. [-5195:2-C2F5,3-F-4-(Me)3CO,E], [-5196:2-C3F7,3-F-4-(Me)3CO,E], [-5197 :2-<CF3>2CF, 3-F-4-(Me)3CO, E], [-5198: 2-(CF3)2CH, 3-F-4-(Me)3CO, E], [- 5199:2-CHF2r3-F-4-CMe)3CO,E], [-5200:2-CH2F,3-F-4-(Me)3CO,E] , C -5201:2-CF3 CH2,3- F-4-(Me)3CO, E], [-5202: 2-MeO, 3-F-4-(MehC〇, E], [-5203: 2-EtO, 3-F-4-(Me) 3CO, E], [-52D4: 2-C3H7〇, 3-F-4-(Me)3CO, E], [-5205: 2-(Me)2CHO, 3-F-4-(Me)3 CO , E] , [-5206: 2-N〇2,3-F-4-(Me)3 CO, EJ , [-5207:2,3-F2,3-F-4-(Me)3CQrE ] , [ -5208:2,4-F2,3-F-4-(Me)3CO,E], [-5209:2,5-F2,3-F-4-(Me)3CO,E],[- 5210:2,6-F2,3-F-4-(Me)3CO,E] , [-5211: 3, 4-F2,3-F-4-(Me) 3 C〇, E ],[- 5212:3,4-F2,3-F-4-(Me)3 C〇,Z 〕 , [ -5213:3,5-F2,3-F-4-(Me)3〇〇,E) , C-5214: 3,5-F2,3-F-4-(Me)3CO/z3, [-5215:2,3-CI2^3-F-4-(Me)3〇0,ε], [ -5216:2,3-CI2,3-F-4-(Me)3CO,Z], C-5217:2,4-Cl2,3-F-4-(Me)3CO,E], [ -5218 :2,4-Cl2,3-F-4-(Me)3CO,Z],[-52 19:2,5-Cl2,3-F-4-(Me)3CO, E], [.-5220:2,5-CI2^3-F-4-(Me)3CO,Z], [-5221 :2,6-CI2,3-F-4-(Me)3〇0,E] , C-5222:3,4-CI2,3-F-4-(Me)3CO,E ] , [ -5223 :3,5-Cl2,3-F-4- 154 320202 200901876 (Me)3C〇,E] ·[-5224:2,3-Br2,3-F-4-(Me>3CO,E], [ -5225: 2,4-

Br2,3-F-4-(Me)3CG,E), [-5226:2,5-Br2,3-F-4-(Me)3CO, EJ, [-5227:2,6-Br2,3 -F-4-(Me>3CO,E], [-552:3, 4-Br2,3-F-4-(Me)3CO,E], [-5229:3,5-Br2,3-F -4-(Me)3CO,E] , [-5230:2,3-Me2,3-F-4-(Me)3CO,E] , C-5231:2,4-Me2,3-F-4 -(Me)3CO,E),[-5232:2,5-Me2,3-F-4-(Me)3CO,E], [-5523:2,6-Me2,3-F-4- ( Me) 3C〇, E], [-5234:3, 4-Me2,3-F-4-(Me)3C〇, E], [-5235:3, 5-

Me2,3-F-4-(Me)3C〇,E] , [-5236:2,3-Et2,3-F-4-(Me)3CO,E] f [-5237:2, 4-Et2 , 3-F-4-(Me)3CO, E] · [ -5238:2,5-Et2,3-F-4-(Me)3CO,E] , [-5239:2,6-Et2,3 -F-4-(Me)3C〇,E] , [-5240:3,4-Et2,3-F-4-(Me)3CO,E] , [-5241:3,5-Et2,3- F-4-(Me)3 CO,E],[-5242:2,3-(CF3)2,3-F-4-(Me)3CO,E],[-5243:2,4-(CF3 2,3-F-4-(Me)3CO,E], [-5244:2,5-(CF3)2,3-F-4-(Me)3CO,E], [- 5245:2, 6-(CF3)2,3-F-4-(Me)3CO,E], [-5246:3,4-(CF3)2,3-F-4-(Me)3CO,E], [- 5247:3,5-(CF3)2,3-F-4-(Me)3C〇,E], C-5248:2,3-(CHF2)2,3-F-4-(Me)3 CO , E], [-524 9 : 2,4- (CHF2.) 2,3-F-4-(Me)3CO, E 3 , [ -5250:2,5-(CHF2)2,3-F- 4-(Me)3CO,E],[- 5251:2,6-(CHF2)2,3-F-4-(Me)3CO,E] , C-5252:3,4-(CHF2)2, 3-F-4-(Me)3CO,E), [-5253:3,5-(CHF2)2,3-F-4-(Me>3C〇,E],[- 5254:2,3- (CH2F)2,3-F-4-(Me)3C0,E],[-5255:2,4-(CH2F)2,3-F-4-(Me) 3C〇,E], [-556 :2,5-(CH2F) 2,3-F-4-(Me) 3C〇,E],[- 5257:2,6-(CH2F)2,3-F-4-(Me)3C0,E ], [-5258:3, 4-(CH2F)2,3-F-4-(Me) 3CO,E ] , [ -5259:3,5-(CH2F)2,3-F-4- (Me)3C〇, E], [- 5260:2,3-(MeO>2,3-F-4-(Me)3CO,E], [-5261:2,4-(MeO)2,3 -F-4-(Me)3C〇,E], [ -5262:2,5-(MeO)2,3-F-4-(Me)3 CO, EJ, [- 155 320202 200901876 5263:2, 6-(MeO)2,3-F-4-(Me)3CO,E] , [-5264:3,4-(MeO)2,3-F-4-(Me)3C〇,E], [ -5265:3,5-(Me〇)2,3-F-4-(Me)3CO,E],[- 5266:2,3-(EtO)2,3-F-4-(Me)3CO , E], [-5267:2,4-(EtO)2,3-F-4-(Me)3CO,E], [-5268:2,5-(EtO)2,3-F-4- (Me)3CO,E 〕 , C - 5269:2,6-(EtO)2,3-F-4-(Me)3CO,E] , [-5270:3,4-(EtO)2,3- F-4-(Me)3CO, E], [-5271:3, 5-(EtO)2,3-F-4-(Me)3CO,E) , [-5272 :2-C1-3-F , 3-F-4-(Me)3 CO, E] , [-5273: 2-C1-4-F, 3-F-4-(Me>3CO, E], [-527 4:2-Cl -5-F,3-F-4-(Me)3CO, E 3 , C-5275:2-C1-6-F,3-F-4-(Me)3CO,E] , C-5276:3 -Cl-2-F,3-F-4-(Me)3CO,E] , [-5277:3-Cl-4-F,3-F-4-(Me)3CO,E] , [-5278 :3-C1-5-F,3-F-4-(Me)3CO,E],[-5279:4-Cl-2-F,3-F-4-(Me)3CO,E], [ -5280: 4-C1-3-F, 3-F-4-(Me)3CO, E], [-5281: 2-F-3-Me, 3-F-4-(Me)3CO, E] , [-5282: 2-F- 4- Me, 3-F-4-(Me)3CO, E3, [-5283 : 2-F-5-Me, 3-F-4-( Me) 3 C〇, E ],.

[-5284 : 2 — F-6—Me,3 — F—4 —(Me)3 CO,E 3 , [ —5285:3—F—2-Me,3-F—4-(Me)3CO, E], [-5286: 3-F-4-Me, 3-F-4-(Me)3CO, E], [-5287: 3-F- 5- Me, 3-F-4-(Me) 3CO, E], [-5288: 4-F-2-Me, 3-F-4-(Me)3CO, E], C-528 9:4-F-3-Me, 3-F-4- (Me)3 C〇,E] , [-5290:2-Cl-3-Me,3-F-4-(Me)3C〇,E], [-5291:2-Cl-4-Me,3 -F-4-(Me)3 CO,E] ,[-5292:2-Cl-5-Me, 3-F-4-(Me) 3CO,E], [-5293:2-Cl-6- Me, 3-F-.4-(Me)3CO,E], C-5294:3-Cl-2-Me,3-F-4-(Me)3 CO, E 3 , [-5295:3-

Cl-4-Me,3-F-4-(Me)3C〇,E], [ -5296:3-Cl-5-Me,3-F-4-(Me)3COfE], [-5297:4 -Cl-2-Me,3-F-4-(Me)3CO, E], [-5298:4-Cl-3-Me,3-F-4-(Me)3 CO, E 3 , [ 5299 12-F—3-CF3,3-F-4-(Me)3C〇rE], [-5300:2-F-4-CF3,3-F-4-(Me)3CO,E], [ -5301:2-F-5-CF3,3-F-4-(Me)3CO,E] , (-5302:2-F-6-CF3,3-F-4-(Me)3 CO,E ], 156 320202 200901876 C-5303: 3-F-2-CF3, 3-F-4-(Me)3C〇, E], [-5304: 3-F-4-CF3, 3-F-4- (Me)3CO,E], [-5305:3-F-5-CF3,3-F-4-(Me)3CO,E],.[-5306:4-F- 2-CF3,3-F -4-(Me)3 CO,E] , [-5307:4-F-3-CF3,3-F-4-(Me) 3 CO, E], [-5308:2-Cl-3-CF3 , 3-F-4-(Me)3CO, E] , [-5309:2-Cl-4-CF3,3-F- 4-(Me)3CO,E ] , [ a 5310:2-Cl-5 —CF3,3-F-4-(Me)3C〇,E],[5311:2-Cl-6-CF3,3-F-4-(Me)3CO,E],[-5312:3- Cl-2-CF3,3-F-4-(Me)3C〇,E], [-5313:3-Cl-4-CF3,3-F-4-(Me)3CO,E], (-5314 :3-CI-5-CF3,3-F-4-(Me)3 CO, E 〕 , 〔 -5315: 4-Cl-2-CF3,3-F-4-(Me)3C〇,E] , [-5316: 4-Cl-3-CF3, 3-F-4-_3CO, E], [-5317: 2-Me-3-CF3, 3-F-4-(Me)3CO, E], [ -5318 :2-Me-4-CF3,3-F-4- (Me)3C〇,E], [-5319:2-Me-5-CF3,3-F-4-(Me)3CO,E] ; [-5320:2-Me-6-CF3,3-F -4-(Me)3C〇,E], [-5321:3-Me-2-CF3,3-F-4-(Me)3CO,E], [-5322:3-Me-4-CF3, 3-F-4-(Me)3CO,E] r [-5323:3-Me-5-CF3,3-F-4-(Me)3 CO, E], [-5324:4-Me-2 -CF3,3-F-4-(Me)3C〇,E) , [-5325:4-Me-3-CF3,3-F-4-(Me)3 CO,E] , [-5326:2 -F-3-MeO, 3-F-4-(Me)-3 CO, E 〕 , 〔 -5327 : 2-F-4-MeO, 3-F-4- (Me)3C〇,E] , [5328:2-F-5-Me〇, 3-F-4-(Me)3CO, E] r C-5329: 2-F-6-MeO, 3-F-4-(Me)3CO, E] , [-5330: 3-F-2-MeO, 3-F-4-(Me)3CO, E], [-5331: 3-F-4-MeOf3-F-4-(Me)3CO, E] r C-5332: 3-F-5-MeO, 3-F-4-(Me)3CO, E], [-5333: 4-F-2-MeO, 3-F-4-(Me) 3 CO, E] , C~5334:4-F- 3-MeO,3-F-4-(Me)3 CO,E] , [-5335:2-Cl-3-MeO, 3-F-4 - (Me)3CO,E], [-5336:2-Cl-4-MeO,3-F-4-(Me)3C〇,E], [-5337:2-Cl-5-MeO,3- F- 4-(Me)3CO,E], C-5338:2-Cl-6-MeO/3-F-4-(Me)3CO,E],[- 5339:3-Cl-2-MeO, 3-F-4-(Me)3CO,E] , C-5340:3-Cl-4-MeO,3-F-4-(Me)3CO,E] , [-5341:3-Cl-5- MeO, 3-F-4-(Me)3〇〇, E], [-5342:4- 157 320202 200901876

Cl-2-MeO,.3-F-4-(Me) 3CO,E], (Me)3CO,E], [-5344:2-Me-3-MeO Me-4-MeO,3-F- 4-(Me)3CO,E], (Me)3CO,E], [-5347:2-Me-6-MeO Me-2-MeO,3-F-4-(Me)3CO,E], [ -5343: 4-Cl-3-MeO, 3-F-4-3-F-4-(Me)3CO, E]', [-5345:2-[-534 6:2-Me-5-MeO , 3-F-4-3-F-4-(Me)3CO, E] , [-5348:3-[-5349:3-Me-4-MeO,3-F-4-(Me)3CO, E], C-5350: 3-Me-5-MeO, 3-F-4-(Me)3CO, E], [-5351: 4-Me-2-MeO, 3-F-4-(Me) 3CO, E 〕 , [ -5352: 4-Me-3-MeO, 3-F-4-(Me)3CO, E], [-5353:H,4-Me,E], [-5354:4- F,4-Me,E], [-5355:4-F,4-Me,Z], [-5356:4-Cl,4-Me,E],[-5357:4-Cl,4-Me , Z], [-5358: 4-Br, 4-Me, E], [-5359: 4-I, 4-Me, E], [-5360: 4-Me, 4-Me, E], [ -5361: 4-Me, 4-Me, Z], [-5362: 4-Et, 4-Me, E], [-5363: 4-C3H7, 4-Me, E], [-5364: 4- (Me) 2CH, 4-Me, E], [-5365: 4-CF3, 4-Me, E], [-5366: 4-CF3, 4-Me, Z], [-5367: 4-C2F5, 4-Me, E], [-5368: 4-C3F7, 4-Me, E], [-5369: 4-(CF3)2CF, 4-Me, E], [-5370: 4-(CF3)2CH , 4-Me, E], [-5371: 4-CHF2, 4-Me, E], [-5372: 4-CH2F, 4-Me, E], [-5373: 4-CF3CH2, 4-Me, E , [-537-4 : 4-MeO, 4-Me, E ] , C -5375 : 4-MeO, 4-Me, Z 3 , C -5376: 4-EtO, 4-Me, E], [- 5377:4-C3H70,4-Me,E], [-5378:4-(Me)2CHO,4-Me,E], [-537 9:4-N〇2,4-Me,E],[ -5380: 4-NO2,4-Me,Z], [-5381:3-F,4-Me,E], [-5382:3-Fr 4-Me,Z], [-5383:3-C1 , 4-Me, E], [-5384: 3-Cl, 4-Me, Z], C-5385: 3-Br, 4-Me, E]f[-538 6:3-1,4-Me , E], [-5387: 3-Me, 4-Me, E], [-5388: 3-Me, 4-Me, Z], [-5389: 3-Et, 4-Me, E], [ -5390: 3-C3H7,4-Me, E], [-5391: 3-(Me}2CH, 4-Me, E], [-5392: 3-CF3, 4-Me, E], [-5393 :3-CF3,4-Me,Z], [-5394:3-C2F5,4-Me,E], [-5395:3-C3F7,4-Me,E], [-5396:3-(CF3 2CF,4-Me,E], [-5397:3-(CF3)2CH,4-Me,E], [-5398:3-CHF2,4-Me,ED, C-5399:3-CHF2, 4-Me,Z] , C-5400:3-CH2 F, 4- 158 320202 200901876

Me, E], [-5401: 3-CH2F, 4-Me, Z], [-5402: 3-CF3CH2, 4-Me, E], [- 5403: 3-MeO, 4-Me, E], C-5404: 3-MeO, 4-Me, Z], [-5405: 3-EtO, 4-

Me, E], [-5406: 3-C3H7O, 4-Me, E], [-5407: 3-(Me) 2CHO, 4-Me, E], [- 5408: 3-NO2, 4-Me, E], [-5409: 2-F, 4-Me, E], [-5410: 2-Cl, 4-Me, E], [- 5411: 2-Br, 4-Me, E], [- 5412: 2-I, 4-Me, E], [-5413: 2-Me, 4-Me, E], [- 5414: 2-Et, 4-Me, E], [-5415: 2-C3H7 , 4-Me, E], [-5416: 2-(Me) 2CH, 4-

Me, E], [-5417: 2-CF3, 4-Me, E], [-5418: 2-C2F5, 4-Me, E], [-5419: 2-C3F7r4-Me, E], [- 5420: 2-(CF3)2CF, 4-Me, E]., [-5421: 2-(CF3)2CH, 4-

Me, E], [-5422: 2-CHF2, 4-Me, E], [-5423: 2-CH2F, 4-Me, E], [-5424: 2-CF3CH2, 4-Me, E], [-5425: 2-MeO, 4-Me, E], [-5426: 2-EtO, 4-Me, E], [- 5427: 2-C3H70, 4-Me, E], C-5428:2 -(Me)2CHO,4-MefE V, C-5429:2-N〇2,4-Me,E], [-5430:2,3-F2,4-Me,E], [-5431:2 , 4-F2,4-Me,E], [- 5432:2, 5-F2,4-Me,E], [-5433:2, 6-F2,4-Me,ED, C-5434 : 3f 4-F2,4-

Me, E], [ -5435:3, 4-F2,4-MerZ], [ -5436: 3,5-F2,4-Me, E], [- 5437:3,5-F2,4-Me ,Z ] , C -5438:2,3-Cl2,4-Me,E ] , C -5439:2,3-

Cl2,4-Me,Z], [-5440:2,4-Cl2_,4-Me,E], [-5441:2,4-Cl2,4-Me,Z],[· 5442:2,5 -Cl2,4-Me,E], [-5443:2,5-Cl2,4-Me-rZ], [-5444:2,6-

Cl2,4-Me,E], [-5445:3,4-Cl2,4-Me,E], [-5446:3,5-Cl2,4-Me,E],[- 5447:2,3 -Br2,4-Me,E 3 , [ -5448:2,4-Br2,4-Me,E ) , X -5449:2,5-

Br2,4-Me,E], [-5450:2,6-Br2,4-Me,E], [-5451:3,4-Br2,4-Me,E],[- 5452:3,5 -Br2,4-Me,E ] , C -5453:2,3-Μθ2,4-Me,E ] , C -5454:2/4-

Me2 r4-Me, E], C-5455: 2,5-ΜΘ2, 4-Me, E], [-5456:2,6-ΜΘ2 f 4-Me,E], C~ 5457:3,4- Μβ2,4-Me,E 3 , C -5458:3,5-Μβ2, 4-Me,E ] , [ -5459:2,3-

Et2,4-Me,E], [-5460:2,4-Et2,4-Me,E], [-5461:2,5-Et2,4-Me,E], [- 5462:2,6 -Et2/4-Me,E ] , C -5463:3,4-Et2,4-Me,E ] , C -5464:3,5- 159 320202 200901876

Et2,4-Me,E], [-54 65:2,3-(CF3)2,4-Me,E], [-5466:2,4-(CF3)2,4-Me,E], [-5467:2,5-(CF3)2,4-Me,E], [-5468:2,6-(CF3)2,4-Me,E],[-5469:3,4-(CF3 ) 2,4-Me, E], [-5470:3,5-(CF3)2,4-Me,E], [-5471:2,3-(CHF2)2,4-Me,E], [-5472:2,4-(CHF2)2,4-Me,E], [-5473:2,5-(CHF2)2,4-Me,E], C-5474:2,6-(CHF2 ) 2 , 4-Me, E ], [-5475:3,4-(CHF2) 2,4-Me,E ], C -5476:3,5-(CHF2)2,4-Me,E ], C-5477: 2,3-(CH2F)2,4-Me,E], C-5478:2,4-(CH2F)2,4-Me,E 5479:2,5-(CH2F)2,4 -Me,E], [-5480:2,6-(CH2F)2,4-Me,E], [-5481:3, 4-(CH2F)2,4-MerE], [-5482:3, 5-(CH2F)2,4-Me,E],[-5483:2,3-(MeO)2,4-Me,E],[-5484:2,4-(MeO)2,4-Me , E], [-5485: 2,5-(MeO) 2,4-Me, E ] , C -5486: 2,6-(MeO) 2,4-Me,E ], [-5487:3, 4-(MeO)2,4-Me,E], [-5488:3,5-(Me〇)2,4-Me,E], [-5489:2,3-(EtO)2,4- Me,E ] , C -5490:2,4-(EtO)2,4-Me,E ],[-5491:2, 5-(EtO)2,4-Me,E ) , C -5492:2 , 6-(EtO)2,4-Me,E],[-5493:3,4-(EtO)2,4-Me,E], [-5494:3,5-(EtO)2,4- Me, E], [-5495: 2-C1-3-F, 4-Me, E3, C-5496: 2-C1-4-F, 4- Me, E] , [-5497: 2-C1-5-F, 4-Me, ED, C-5498: 2-Cl-6-F, 4-Me, E], C-54 99: 3-C1 -2-F, 4-Me, E ], [-5500:3-Cl-4-F,4-Me,E] , C-5501: 3-C1-5-F, 4-Me,E] , [-5502: 4-01-2-F, 4-Me, E], [-5503: 4-C1-3-F, 4--Me, E], [-5504: 2-F-3-Me , 4-Me, E], [-5505: 2-F-4-Me, 4-Me, E], [-5506: 2-F-5-Me, 4-Me, E], [-5507: 2-F-6-Me, 4-Me, E], [-5508: 3-F-2-Me, 4-Me, E], [ -5509: 3-F-4-Me, 4-Me, E], [-5510: 3-F-5-Me, 4-Me, E], [-5511: 4-F-2-Me, 4-Me, E], [-5512: 4-F-3 -Mef 4-Me,E],C-5513:2-Cl-3-Me,4-Me,E),[-5514:2-C1-4-Me,4-Me,E], [-5515 :2-Cl-5-Me,4-Me,E], [-5516:2-Cl-6-Me,4-Me,E], [-5517:3-Cl-2-Me,4-Me , E], [-5518: 3-Cl-4-Me, 4-Me, E], [- 160 320202 200901876 5519: 3-Cl-5-Me, 4-Me, E3, C-5520: 4- Cl-2-Me,4-MerE ] f [-5521:4-Cl-3-Me,4-Me,E 3 ,[ -5522:2-F-3-CF3,4-Me,E], C -5523: 2-F-4-CF3,4-Me,E], [-5524:2-F-5-CF3,4-Me,E], [-5525:2-F-6-CF3,4 -Me, E], [-5526: 3-F-2-CF3, 4-Me, E], [-5527: 3-F-4-CF3, 4-Me, E], [-5528: 3- F-5-CF3,4-Me,E],[-5529:4-F-2-CF3,4-Me,E],[- 5530: 4-F-3-CF3,4-Me,E], [-5531:2-Cl-3-CF3,4-Me,E], C-5532:2-C1-4-CF3,4- Me, E], [-5533: 2-Cl-5-CF3, 4-Me, E], [-5534: 2-Cl-6-CF3, 4-Me, E], [-5535: 3-Cl -2-CF3,4-Me,E], [-5536:3-Cl-4-CF3,4-Me,E], [-5537:3-Cl-5-CF3,4-Me,E], [-5538: 4-Cl-2-CF3,4-Me, E], [-5539: 4-Cl-3-CF3, 4-Me, E], [-5540: 2-Me-3-CF3, 4-Me, E], [-5541: 2-Me-4-CF3, 4-Me, E], [-5542: 2-Me-5-CF3, 4-Me, E], [-5543: 2 -Me-6-CF3,4-Me,E], [-5544:3-Me-2-CF3,4-Me,E], [-5545:3-Me-4-CF3,4-Me,E ], [-5546: 3-Me-5-CF3, 4-Me, E], [-5547: 4-Me-2-CF3, 4-Me, E], [-5548: 4-Me-3- CF3,4-Me,E], [ -5549:2-F-3-MeO,4-Me,E], C-5550:2-F-4-MeO,4~Me,E], C-5551 :2-F-5-MeO,4-Me,E ] , C-5552:2-F-6-MeO,4-Me,E],[-5553:3-F-2-MeO,4-Me , E], [-5554: 3-F-4-MeO, 4-Me, E], [-5555: 3-F-5-Me〇, 4-Me, E], [-5556: 4-F -2-MeOr 4-Me,E], [-5557:4-F-3-MeO,4-Me,E], [-5558:2-Cl-3-MeO,4-Me,E], [ -5559: 2-C1-4-MeO, 4-Me, E], [-5560: 2-Cl-5-MeO, 4-Me, E], [-5561: 2-Cl-6-Me〇, .4-M e, E], [-5562: 3-Cl-2-MeO, 4-Me, E], [-5563: 3-Cl-4-Me〇, 4-Me, E], [-5564: 3- Cl-5-MeO, 4-Me, E3, C-5565: 4-Cl-2-MeO, 4-Me, E], [-5566: 4-Cl-3-MeO, 4-Me, E], [-5567: 2-Me-3-MeO, 4-Me, E], C-5568: 2-Me-4-MeO, 4-Me, E], [-5569: 2-Me-5-Me〇 , 4-Me, E], [-5570: 2-Me-6-Me〇, 4-Me, E], [-5571: 3-Me-2-MeO, 4-Me, E], [-5572 :3-Me-4-MeO,4-Me,E], [-5573:3-Me-5-MeO,4-Me,E],[-5574:4-Me-2-MeO,4-Me ,E],[-5575:4- 161 320202 200901876

Me-3-MeO, 4-Me, E], [-5576: H, 3-Me, E], [-5577: 4-F, 3-Me, E], [-5578: 4-F, 3 -Me,Z], [-5579:4-Cl,3-Me,E], [-5580:4-Cl,3-Me,Z], [-5581:4-Br,3-Me,E] , [-558.2: 4-1,3-Me, E], [-5583: 4-Me, 3-Me, E], [-5584: 4-Me, 3 II Me, Z], [-5585: 4-Et,3-Me,E], [-5586:4-C3H7,3-Me,E], [-5587:4-(Me)2CH,3-Me,E], [-5588:4- CF3,3-Me,E], [-5589:4-CF3f3-Me,Z], [-5590:4-C2F5,3-Me,E], [-5591:4-C3F7,3-Me,E ], [-5592: 4-(CF3)2CF, 3-Me, E], C-5593: 4-(CF3)2CH, 3-Me, E), [-5594: 4-CHF2, 3-Me, E], [-5595: 4-CH2 F, 3-Me, E], [-5596: 4-CF3 CH2, 3-Me, E], C-5597: 4-MeO, 3-Me, E], C-5598: 4-MeO, 3-Me, ZD, C-5599: 4-EtO, 3-Me, E], [-5600: 4-C3H7O, 3-Me" E], [-5601: 4- (Me) 2CHO, 3-Me, E], [-5602: 4-N〇2, 3-Me, E], [-5603: 4-N〇2, 3-Me, Z], [-5604: 3:^,3-Me,E], [-5605:3-F,3-Me,Z], [-5606:3-Cl,3-Me,E], [-5607:3-Cl,3 -Me,Z], [-5608:3-Br,3-Me,E], [-5609:3-1,3-Me,E], [-5610:3-Me,3-Me,E] , C -5611: 3-Me, 3-Me, Z ] , [·-5612 :3- Et, 3-Me, E ] , C -5613 :3-C3 H7,3-Me,E "} , C -5614:3-(Me)2CH,3-Me,E 3 , C -5615 : 3 -CF3,3-Me, ED,C-5616:3-CF3,3-Me,z3, C-5617 : 3-C2 F5,3-Me, E ] , C-5618:3-C3F7v3-Me,E ], [-5619: 3-(CF3)2CF, 3-Me, E], [-5620: 3-(CF3)2CH, 3-Me, E], [-5621: 3-CHF2, 3-Me, E], C-5622: 3-CHF2, 3-Me, ZD, C-5623: 3-CH2F, 3-Me, E], [-5624: 3-CH2F, 3-Me, Z], [-5625 :3-CF3CH2,3-Me,E], [-5626:3-MeO,3-Me,E ] , [-5627:3-MeO,3-Me,Z ] , [ -5628:3-EtO, 3-Me, E], [-5629: 3-C3H7O, 3-Me, E], [-5630: 3-(Me) 2CHO, 3-Me, E], [-5631: 3-N02, 3- Me, E], [-5632: 2-F, 3-Me, E], [-5633: 2-Cl, 3-Me, E], [-5634: 2-Br, 3-Me, E], [-5635: 2-I, 3-Me, E], [-5636: 2-Me, 3-Me, E], [-5637: 2-Et, 3-Me, E], C-5638: 2 -C3H7,3-Me,E], [-5639:2-(Me)aCH,3-Me,E], [-5640:2-CF3,3-Me,E], [-5641:2-C2F5 ,.3-Me,E],[-5642:2- 162 320202 200901876 C3F7,3-Me,E], [-5643:2- (CF3 ) 2 CF, 3-Me, E] , [-5644 : 2-(CF3)2CH,3-Me,E],C-5645:2-CHF2,3-Me,E],[-5646:2-CH2F,3-Me,E],[-5647:2- CF3CH2,3-Me,E],C-5648:2-MeO,3-Me,E],C- 5649: 2-EtO, 3-Me, E], C-5650: 2-C3H7O, 3-Me, E3, [-5651: 2-(Me)2CHO, 3-Me, E], C-5652: 2-N02,3-Me,E], [-5653:2,3-F2,3-Me,E], [-5654:2,4-F2,3-Me,E], [-5655:2 ,5-F2,3-Me,E),C-5656:2,6-F2,3-Me,E],C-5657:3,4-F2,3-Me,E],[ -5658: 3,4-F2,3-Me,Z], [-5659:3,5-F2,3-Me,E], [-5660:3,5-F2,3-Me,Z "} , C -5661: 2,3-Cl2,3-Me, E ] , [ -5662:2,3-Cl2,3-Me,Z], [-5663:2,4-Cl2,3-Me,E], C-5664: 2,4-Cl2,3-Me,Z], C-5665: 2,5-Cl2,3-Me,ED, C-5666:2,5-Cl2,3-Me/Z 3 , [-5667: 2,6-Cl2,3-Me,E], [-5668:3,4-Cl2,3-Me,E], [-5669:3, 5-Cl2',3-Me,E ], [-5670: 2,3-Br2,3-Me, E], [-5671:2,4-Br2,3-Me,E], [-5672:2,5-Br2,3-Me, E], [-5673: 2,6-Br2,3-Me, E], [-5674:3,4-Br2,3-Me,E], [-5675:3,5-Br2,3-Me , E 〕 , 〔 -5676:2,3-Me2,3-Me,E 〕 , C -5677:2/4-Me2,3-Me,E], [-5678:2,5-Me2,3- Me, E], [-5679: 2, 6-Me2, 3-Me, E], [-5680: 3, 4-^Me2, 3-Me, E], C -5681: 3, 5-Me2, 3-Me, E ] -, [ -5682:2,3-Et2,3-Me,E], [-5683:2,4-Et2,3-Me,E], [-5684:2,5- Et2,3-Me,E], -5685:2,6-Et2,3-Me,E 3 ,C -5686:3,4-Et2,3-MefE ] f C-5687:3,5-Et2,3-Me,E],[- 5 688: 2,3-(CF3)2,3-Me,E], [-5689:2,4-(CF3)2,3-Me,E], [-5690:2,5-(CF3) 2,3-Me,E], [-5691:2,6-(CF3)2,3-Me?E], [-5692:3,4-(CF3)2,3-Me,E], -5693:3,5-(CF3)2,3-Me,E], [-5694:2,3-(CHF2)2,3-Me,E], [-5695:2,4-(CHF2) 2,3-Me,E], [-5696:2,5-(CHF2)2,3-Me,E]., [-5697:2,6-(CHF2)2,3-Me,E], [-5698:3,4-(CHF2)2,3-Me,E], [-5699:3,5-(CHF2)2,3-Me,E], [-5700:2,3-(CH2F 2,3-Me,E]r[ -5701: 2,4-(CH2F)2,3-Me,E], [- 163 320202 200901876 5702:2,5-(CH2F)2,3-Me, E], C -5703 : 2, 6-(CH2 F) 2,3-Me, E ], C-5704:3, 4-(CH2F>2,3-Me, E.], [-5705:3 ,5-(CH2F)2,3-Me,E], [-5706:2,3-(MeO)2,3-Me,E], [-5707:2,4-(MeO)2,3- Me, E], [-5708: 2, 5-(MeO) 2, 3-Me, E ] , C - 5709: 2, 6-(MeO) 2, 3-MerE ], [-5710: 3, 4 -(MeO)2,3-Me,E], [-5711:3,5-(MeO)2,3-Me,E], [-5712:2,3-(EtO)2,3-Me, E], [-5713: 2,4-(EtO) 2,3-Me, E], [-5714:2,5-(EtO)2,3-Me, E 3 , C -5715:2,6 -(EtO)2,3-Me,E ] , C-5716: 3,4-(EtO)2,3-Me,E], [-5717:3,5-(EtO)2,3-Me,E], [-5718:2-Cl-3 -F,3-Me,E] , C-5719:2-C1-4-F,3-Me,E], C-5720:2-C1-5-F,3-Me,E],[- 5721: 2-Cl-6-F, 3-Me, E], [-5722: 3-Cl-2-F, 3-Me, E], [-5723: 3-Cl-4-F, 3- Me, E] , [-5724 : 3-C1-5-F, 3-Me, E ] , C'-5725: 4-Cl- 2- F, 3-Me, E], [-5726:4- Cl-3-F,3-Me,E], [-5727:2-F-3-Me,3-Me,E], C-5728:2-F-4-Me,3-Me,E] , [-5729: 2-F-5-Me, 3-Me, E), C-5730: 2-F-6-Mef3-Me, E), C -5731: 3-F-2-Me, 3 -Me,E ] , C -5732:3-F-4-Me,3-

Me, E], [-5733: 3-F-5-Me, 3-Me, E], [-5734: 4-F-2-Me, 3-Me, E], [- 5735: 4-F -3-Me,3-Me,E], [-5736:2.-Cl-3-Me,3-Me,E], [-5737:2-Cl- 4-Me,3-Me,E3, C-5738: 2-Cl-5-Me, 3-Me, E], C-5739: 2-Cl-6-Me, 3-

Me, E], [-5740: 3-Cl-2-Me, 3-Me, E], [-5741: 3-Cl-4-Me, 3-Me, E], [- 5742: 3-Cl -5-Me, 3-Me, E], [-5743: 4-Cl-2-Me, 3-MerE], [-5フ44:4-

Cl-3-Me,3-Me,E], [-5745:2-F-3-CF3,3-Me,E], C-5746:2-F-4-CF3,3-Me,E] , [-5747 : 2-F-5-CF3, 3-Me, E], [-5748: 2-F-6-CF3, 3-< - -. Me, E], [-5749: 3- F-2-CF3,3-Me,E], [-5750:3-F-4-CF3,3-Me,E], [- 5751:3-F-5-CF3,3-Me,E] , [-5752:4-F-2-CF3,3-Me, ,[-5753:4-F- 3-CF3,3-Me,E], [-5754:2-Cl-3-CF3,3 -Me,E 〕 , C -5755:2-C1-4-CF3,3-Me,E], [-5756:2-Cl-5-CF3,3-Me,E], [-5757:2- Cl-6-CF3,3-. 164 320202 200901876

Me, E], [-5758: 3-Cl-2-CF3, 3-Me, E], [-5759: 3-Cl-4-CF3, 3-Me, E], [-57 60:3- Cl-5-CF3,3-Me,E],[-57 61: 4-Cl-2-CF3,3-Me,E],[-57 62:4-CI-3-CF3,3-Me, E], C-5763: 2-Me-3-CF3, 3-Me, E], C-57 64: 2-Me-4-CF3, 3-Me, E], [-5765: 2-Me- 5-CF3,3-Me,E], [-5766:2-Me-6-CF3,3-Me,E], [-57 67:3-Me-2-CF3,3-Me,E], [-57 68:3-Me-4-CF3,3-Me,E], [-5769:3-Me-5-CF3,3-Me,E], [-5770:4-Me-2-CF3 , 3-Me, E], [-5771: 4-Me-3-CF3, 3-Me, E], [-5772: 2-F-3-MeO, 3-Me, E], C-5773: 2-F-4-Me〇,3-Me,E], [a 5774:2-F-5-Me〇,3-Me,E], [1-575:2-F-6-Me〇,3 -Me, E], [-5776: 3-F-2-MeO, 3-Me, E], [-5777: 3-F-4-MeO, 3-Me, E], [-5778: 3- F-5-Me〇,3-Me,E], [-5779:4-F-2-MeO, 3-Me,E], [-5780:4-F-3-MeO,3-Me,E ], [ -5781:2-Cl-3-MeO,3-Me,E] r C -5782:2-C1-4-MeO,3-Me,E],[-57B3:2-Cl-5- MeO, 3-Me, E], [-57 84 : 2-Cl-6-MeO, 3-Me, E], [-5785: 3-Cl-2-Me〇, 3-Me, E], -5786: 3-Cl-4-MeO, 3-Me, E], [-5787: 3-Cl-5-MeO, 3-Me, E], [-5788: 4-Cl-2-MeO, 3 -Me, E], [-5789: 4-Cl-3-MeO, 3-Me, E], C-5790: 2-Me-3-MeOf3-Me, ED, C-5791: 2-Me-4-MeO, 3-Me, E], [-.5792: 2-Me-5-MeO, 3-Me, E], [-57 93: 2-Me-6-MeO, 3-Me, E], [-57 94 : 3-Me-2-MeO, 3-Me, E], [-57 95:3-Me-4-Me〇, 3-Me, E], [-5796: 3-Me-5-MeOr 3 -Me,E],[-5797:4-Me-2-MeO, 3-Me,E],C-57 98 : 4-Me-3-MeO,3-Me,E], [-5799:H , 2-Me, E], [-5800: 4-F, 2-Me, E], [-5801: 4-F, 2-Me, Z], [-5802: 4-Cl, 2-Me, E], [-5803: 4-Cl, 2-Me, Z], [-5804: 4-Br, 2-Me, E], [-5805: 4-I, 2-Me, E], [- 5806: 4-Me, 2-Me, E], [-5807: 4-Me, 2-Me, Z], [-58 08: 4-Et, 2-Me, E], [-5809: 4 -C3H7,2-Me,E], [-5810:4-(Me)2CH,2-Me,E], C-5811:4-CF3,2-Me,E 3 ,C-5812:4-CF3 , 2-Me, Z], [-5813: 4-C2F5, 2-Me, E], [-5814: 4-C3F7, 2-Me, E], [-5815: 4-(CF3)2CF, 2 -Me,ED,[-5816:4-(CF3)2CH, 2-Me,,[-5817: 4- 165 320202 200901876 CHF2,2-Me,E], [-5818:4-CH2F, 2-Me , E], [-5819: 4-CF3CH2, 2-Me, E], [-5820: 4-MeO, 2-Me, E], [-5821: 4-MeQ, 2-Me, Z], -5822: 4-EtO, 2-Me, E], [-5823: 4-C3H7〇, 2-Me, E] [-5824: 4-(Me)2CHO, 2-Me, E], [-5825: 4-N〇2, 2-Me, E], [-5826: 4-N〇2, 2-Me, Z ], [-5827: 3-F, 2-Me, E], [-5828: 3-F, 2-Me, Z], [-5829: 3-Cl, 2-Me, E], [-5830 : 3-Cl, 2-Me, Z], [-5831: 3-Br, 2-Me, E], [-5832: 3-1, Hui-Me, E], [-5833: 3-Me, 2-Me, E], C-5834: 3-Me, 2-Me, Z], C-5835: 3-Et, 2-Me, E], C-5836: 3-C3H7, 2-Me, E ], [-5837: 3-(Me) 2CH, 2-Me, E], [-5838: 3-CF3, 2-Me, E], [-5839: 3-CF3, 2-Me, Z], [.-5840:3-C2F5,2-Me,E], [-5841:3-C3F7,2-Me,E], [-5842:3-(CF3)2CF,2-Me,E], -5843: 3-(CF3)2CH, 2-Me, E], [-5844: 3-CHF2, 2-Me, E3, [-5845: 3-CHF2 f 2-Me, Z ] , [-584* 6:3-CH2 F, 2-MerE], [-5847: 3-CH2F, 2-Me, Z], [-5848: 3-CF3CH2, 2-Me, E], [-5849: 3-MeO, 2-Me, E], [-5850: 3-MeO, 2-Me, Z], [-5851: 3-EtO, 2-Me, E], [-5852: 3-C3H70, 2-Me, E ], [-5853: 3-(Me) 2CHO, 2-Me, E], [-5854: 3-N02, 2-Me, E], [-5855: 2-F, 2-Me, E], [-5856: 2-Cl, 2-Me, E], [--5857: 2-Br, 2-Me, E], C-5858: 2-1, 2^^3/C-5859:2- Me, 2-Me, E], C-5860: 2-Et, 2-Me, E], [-5861: 2-C3H 7,2-Me, E3, C-5862: 2-(Me)2CH, 2-Me, E], [-58 63: 2-CF3, 2-Me, E], [-5864: 2-C2F5, 2-Me,E], [-5865:2-C3 F7,2-Me, E], [-58 66:2-(CF3 ) 2 CF, 2-Me, E] , [-5867:2- ( CF3 ) 2 CH/2-Me, E), [-5868: 2-CHF2, 2-Me, E], [-5869: 2-CH2F, 2-Me, E], [-5870: 2-CF3CH2, 2-Me, E], [-5871: 2-MeO, 2-Me, E], [-5872: 2-EtO, 2-Me, E], [-5873: 2-C3H7〇, 2-Me, E] , C-5874: 2-(Me)2CHO, 2-Me, EI, [-5875 : 2-N02, 2-Me, Ej, [-5876: 2, 3-F2, 2-Me, E] , [-5877 : 2,4-F2,2-Me, E 3 , C-5878:2,5-F2,2-Me,E],[-587 9:2,6-F2,2-Me, E], [-5880:3,4-F2,2-Me,E ] , C -5881:3,4-F2,2-Me,Z ] , C -5882:3,5-F2,2-Me , E ] , C - 166 320202 200901876 5883: 3,5-F2,2-Me,Z], [-5884:2,3-Cl2,2-Me,E], [-5885:2,3-Cl2 , 2-Me, Z], [-5886: 2, 4-Cl2, 2-Me, E], [-5887: 2, 4-Cl2, 2-Me, Z], [-5888: 2, 5- Cl2,2-Me,E ] , C -5889:2,5-Cl2,2-Me,Z 3 ,C -5890:2,6-Cl2,2-Me,E], [-5891:3, 4 -Cl2,2-Me,E], [-5892:3,5-Cl2,2-Me,E], [-5893:2,3-Br2,2-Me,E], [ -5 894:2 , 4-Br2, 2-Me, E], [ -5895:2,5-Br2,2-Me,E], [-5896:2,6-Br2,2-Me,E], [-5897: 3,4-Br2,2-Me , E], [-5898:3,5-Br2,2-Me,E ] , C -5899:2,3-Me2,2-Me,E ] f [ -5900:2,4-Me2,2- Me, E], [-5901: 2, 5-Me2, 2-Me, E], [-5902: 2, 6-Me2, 2-Me, E], [-5903: 3, 4-Me2, 2 -Me,E ] , C -5904:3,5-Me2,2-Me,E ] , ί -5905:2,3-Et2,2-Me,E], [-5906:2,4-Et2, 2-Me, E], [-5907: 2, 5-Et2, 2-Me, E], [-5908: 2, 6-Et2, 2-Me, E 3 , C - 5909: 3, 4-Et2 , 2-Me, E 3 , C -5910:3,5-Et2,2-Me,E], [-5911:2,3-(CF3)2,2-Me,E], [-5912:2 , 4-(CF3)2,2-Me,E], [-5913:2,5-(CF3)2,2-Me,E], [-5914:2,6-(CF3)2,2- Me, E], [-5915:3,4-(CF3)2,2-Me,E], [-5916:3,5-(CF3)2,2-Me,E], [-5917:2 ,3-(CHF2)2,2-Me,E], [-5918:2,4-(CHF2)2,2-Me,E], [-5919:2,5-(CHF2)2,2- Me', E], [ -5920:2, 6-(CHF2)2,2-Me,E], [二5921:3, 4-(CHF2)2,2-Me,E], C-5922: 3,5-(CHF2)2,2-Me,E],C-5923:2,3-(CH2F)2,2-Me,E],[-5924:2,4-(CH2F)2,2 -Me,E],[-5925:2,5-(CH2F)2,2-Me,E], [-5926:2,6-(CH2F)2,2-Me,E], [-5927: 3,4-(CH2F)2,2-Me,E ] , C -5928 : 3,5-(CH2 F) 2,2-Me, E 3,C-5929:2,3-(Me〇)2 , 2-Me, E], [-593 0:2,4-(MeO)2,2-Me,E],[-5931:2,5-(MeO)2,2-Me,EI, C-5932:2,6-(MeO)2, 2-Me,E ],[-5933:3,4-(MeO)2,2-Me,E], [-5934:3,5-(MeO)2,2-Me,E], [-5935 :2,3-(EtO)2,2-Me,E 3 , C -5936:2,4-(EtO)2,2-Me,E 5937:2,5-(EtO)2,2-Me, E 〕 r 〔 -5938:2,6-(EtO)2,2-Me,E],[- 167 320202 200901876 5939:3,4-(EtO)2,2-Μβ,Ε], [-5940: 3,5-(EtO)2,2-Me,E],[-5941:2-Cl-3-F,2-Me,E] , C-5942:2-Cl-4-F/2-Me , E 3 , C-5 943: 2-C1-5-F, 2-Me, E], C-5944: 2-Cl-6-F, 2-Me, E], [-5945: 3-C1 -2-F, 2-Me, E], [-5946: 3-Cl-4-F, 2-Me, E], [-5947: 3-Cl-5-F, 2-Me, E], [-5948: 4-Cl- 2-F, 2-Me, E], [-5949: 4-C1-3-F, 2-Me, E], [-5950: 2-F-3-Me, 2-Me, E], C-5951: 2-F-4-Me, 2-Me, E], C-5952: 2-F-5-Me, 2-MerE], [-5953: 2-F -6-Me, 2-Me, E], [-5954: 3-F-2-Me, 2-Me, E], [-5955: 3-F-4-Me, 2-Me, E], [-5956: 3-F-5-Me, 2-Me, E], [-5957: 4-F-2-Me, 2-Me, E], [-5958: 4-F-3-Me, 2-Me, E], [-5959: 2-Cl-3-Me, 2-Me, E], [-5960: 2-Cl-4-Me, 2-Me, E], [-5961: 2 -Cl-5-Me, 2-Me, E], [-5962: 2-Cl-6-Me, 2-Me, E], [-5963: 3-Cl-2-Me, 2-Me, E , [-5964: 3-Cl-4-Me; 2-Me, E], [-5965: 3-Cl-5-Me, 2-Me, E], [-5966: 4-Cl-2-Me , 2-Me, E], [-5967: 4-Cl-3-Me, 2-Me, E], [-5968: 2-F-3-CF3, 2-Me, E], C-5969: 2-F-4-CF3,2-Me,E], [-5970:2-F-5-CF3,2-Me,E], [-5971:2-F-6-CF3,2-Me, E], [-5972: 3-F-2-CF3, 2-Me, E], [-5973: 3-F-4-CF3, 2-Me, E], [-5974: 3-F-5 -CF3,2-Me,E], [-5975:4-F-2-CF3,2-Me,E], [-5976:4-F- 3-CF3,2-Me,E], 〔 5977: 2-Cl-3-CF3, 2-Me, E], C-5978: 2-Cl-4-CF3, 2-Me, E], [-5979: 2-Cl-5-CF3,2- Me, E], [-5980: 2-Cl-6-CF3, 2-Me, E], [-5981: 3-Cl-2-CF3, 2-Me, E], [>5982:3- Cl-4-CF3,2-Me,E], [-5983:3-Cl-5-CF3,2-Me,E'], [-5984:4-Cl-2-CF3,2-Me,E ], [-5985: 4-Cl-3-CF3, 2-Me, E], C-598 6: 2-Me-3-CF3, 2-Me, ED, [-598.7: 2-Me-4- CF3,2-Me,E], [-5988:2-Me-5-CF3,2-Me,E], [-5989:2-Me-6-CF3,2-Me,E], [-5990 :3-Me-2-CF3,2-Me,E], [-5991:3-Me-4-CF3,2-Me,E], [-5992:3-Me-5-CF3,2-Me , E], C-5993: 4-Me-2-CF3, 2-Me, E], [-5994: 4-Me-3-CF3, 2-Me, E], [ -5995: 2-F- 3-MeO, 2-Me, E] , [ -5996:2-F-4- 168 320202 200901876

MeO, 2-Me, E], C-5997: 2-F-5-MeO, 2-Me, E], C-5998: 2-F-6-MeO, 2-Me, E], [-5999 :3-F-2-MeO,2-Me,E],[-6000:3-F-4-MeO,2-Me,E],[-6001:3-F-5-MeO,2-Me , E], [-6002: 4-F-2-MeO, 2-Me, E], [-6003: 4-F-3-MeO, 2-Me, E], [-6004: 2-Cl- 3-Me〇,2-Me,E 〕 , C -6005:2-C1-4-Me〇,2-Me,E], [1-66:2-Cl-5-MeO,2-Me,E] , [a 6007: 2-Cl-6-Me〇, 2-Me, E], [-6008: 3-Cl-2-MeO, 2-Me, E], [-6009: 3-Cl-4- Me〇, 2-Me, E], [-6010: 3-Cl-5-MeO, 2-Me, E], [-6011: 4-Cl-2-MeO, 2-Me, E], [- 6012: 4-Cl-3-MeO, 2-Me, E], C-6013: 2-Me-3-MeO, 2-Me, E], C-6014: 2-Me-4-MeO, 2- Me, ED, C ~ 6015: 2-Me-5-MeO, 2-Me, E}, C - 6016: 2-Me-6-MeO, 2-Me, 'E], [-6017: 3-Me -2-Me〇, 2-Me, E], [-6018: 3-Me-4-MeO, 2-Me, E],, [-6019: 3-Me-5-MeO, 2-Me, Ej , [-6020: 4-Me-2-MeO, 2-Me, eD, [-6021: 4-Me-3-MeO, 2-Me, E], [-6022: H, 3, 4-Me2, E], [-6023: 4-F, 3, 4-Me2, E], [-6024: 4-F, 3, 4-Me2, Z], C - 6025: 4-C1, 3, 4-Me2 , E ] , C -6026:4-Clf 3,4-Me2,Z], [-6027:4-Br,3,4-Me2,E],[-6028:4-1,3,4-Me2 , E], [ -6029:4-Me,3,4-Me2,ED, C-6030:4-Me,3,4-Me2,Z 3 ,C-6031:4-Et,3f4-Me2,E ] , C -6032 :-4-C3 H7,3,4-Me2 , E ] , C -6033:4- (Me)2CHr3,4-Me2,E ] , C -6034:4-CF3,3,4-Me2,E 3 , [ -6035:4-CF3 ,3r 4-Me2 ,ZD , C-6036:4-C2F5,3,4-Me2 ,E] , C-6037 : 4-C3 F7 ,3,4-Me2 , C- 6038 :4-(CF3 ) 2 CF, 3,4-Me2 , E3 , C-6039 : 4- (CF3 )2CH,3, 4-Me2,E],C-6〇40:4-CHF2,3, 4-Me2, [-6041:4-CH2F,3,4-Me2,E], C~ 6042:4-CF3CH2,3,4-Me2,E],[-6043:4-MeO,3,4- Me2, E], [-6044: 4-MeO, 3, 4-Me2, C-6045: 4-EtO, 3, 4-Me2 fE], C-6046: 4-C3H70, 3, 4-Me2, E ], [-6047: 4-(Me> 2CHO, 3, 4-Me2, E], [-6048: 4-NO2, 3, 4-Me2, E], [-6049: 4-N〇2, 3 , 4-Me2, Z], [-6050: 3-F, 3, 4-Me2, E], [-6051: 3-F, 3, 4-Me2, Z], [-6052: 3-Cl, 3,4-Me2,E], [-6053:3-C1,3,4-Me2 ΓZ], 169 320202 200901876 [-6054:3-Br,3,4-Me2,Ε], [-6055: 3-work, 3,4-Me2, E], C -6056:3-Me,3,4-Me2,E], [-6057:3-Me,3,4-Me2,Z],[-6058 :3-Et,3,4-Me2,E], C-605 9:3-C3H7,3,4-Me2,E ] , C -6060:3-(Me)2CH,3,4-Me2,E ], C-6061: 3—CF3, 3, 4_Μβ2 / E 3 f C -6062 : 3—CF3,3, 4-Μβ2 f 2 D , C -6063:3-C2FS ,3, 4-Me2 ,E ] , C -6064 : 3-C3 F7,3, 4- Me2 , E ) , C -6065:3-(CF3 )2CF,3,4-Me2,E] , C-6066: 3-(CF3 )2CH,3,4-Me2 ,eD , [-6067 :3- CHF2,3,4-Me2,E], [-6068:3-CHF2,3,4-Me2,Z], [-6069:3-CH2F,3,4-Me2,E], [-6070:3 -CH2F,3,4-Me2,Z], [-6071:3-CF3CH2,3,4-Me2,E], [-6072:3-MeO,3,4-Me2,E], [-6073: 3-MeO,3,4-Me"Z], [-6074:3-EtO,3,4-Me2,E], [-6075:3-C3H70,3,4-Me2,E], [-6076 :3-(Me)2 CHO,3,4-Me2,eD,[-6077:3-N02,3,4-Me2,E],[-607 8:2-F,3,4-Me2,E ], [-6079: 2-Cl, 3, 4-Me2, E], [-6080: 2-Br, 3, 4-Me2, E] r [-6081: 2-1, 3, 4-Me2, E], C-6082: 2-Me, 3, 4-Me2, E], [-6083: 2-Et, 3, 4-Me2, E], [-6084: 2-C3H7, 3, 4-Me2 , E], [-6085: 2-(Me) 2CH, 3, 4-Me2, E], [-608 6: 2-CF3, 3, 4-Me2, E], [-6087: 2-C2F5, 3,4-Me2,E],[-6088:2-C3F7,3,4-Me2,E], C-6089: 2-(CF3) 2 CF, 3,4-Me2, E],· [ - 6090: 2-(CF3 >2CH,3,4-Me2,E], [ -6091: 2-CHF2,3,4-Me2, E], [-6092:2-CH2F,3,4-Me2, E], [ -6093 : 2-CF3 CH2,3,4-Me2, E], [ -6094:2-Me〇,3,4-Me2,E], [-6095:2-EtO,3,4-Me2,E], -6096: 2-C3H7O,3,4-Me2,E], [-6097:2-(Me)2CHO,3,4-Me2,E], [-6098:2-N02,3,4-Me2, E], C -6099: 2,3-F2 ,3,4-Me2 ,E ] , [ -6100:2,4-F2,3,4-Me2 , E ]fC-6101:2,5-F2, 3,4-Me2[-6102:2,6-F2,3,4-Me2,E],[-6103:3,4-F2,3,4-Me2,E], [-6104:3,4 -F2,3,4-Me2,Z], [-6105:3,5-F2,3,4-Me2,E], [-6106:3,5-F2,3,4,Me2,Z], [-6107: 2,3-Cl2,3,4-Me2,E], [-6108:2,3-Cl2,3,4-Me2,Z], [-6109:2,4-Cl2,3, 4-Me2,E 〕,[- 170 320202 200901876 6110:2,4-Cl2,3,4-Me2,Ζ ] , C -6111:2,5-Cl2,3,4-Me2,ED,[-6112 :2,5-Cl2,3,4-Me2,Z], [-6113:2,6-Cl2,3,4-Me2,E], [-6114:3,4-Cl2,3,4-Me2 , E ) r [ -6115:3,5-Cl2,3,4-Me2,E ], C~ 6116:2,3-Br2,3,4-Me2,E 3 ,C -6117:2,4- Br2,3,4-Me2,E],C-6118:2,5-Br2,3,4-Me2,E], C-6119:2,6-Br2,3,4-Me2,E],[ -6120: 3,4-Br2,3,4-Me2,E], [-6121:3,5-Br2,3,4-Me2,E], [-6122:2,3-Me2,3,4 -Me2, E 3 , C -6123: 2,4-Me2,3,4-Me2,E ], C-6124:2,5-Me2,3,4-Me2,E], [-6125:2, 6-Me2, 3 , 4-Me2, E], [-6126:3,4-Me2,3,4-Me2,E], [_6127:3,5-Me2,3,4-Me2,E], [-6128:2 ,3-Et2,3,4-Me2,E],[-6129:2,4-Et2,3,4-Me2,E],[-6130:2,5-Et2,3,4-Me2,E ], [-6131:2,6-Et2,3,4-M02,E], [-6132:3,4-Et2,3,4-Me2,E), C-6133:3,5-Et2, 3,4-Me2,E 3,C-6134:2,3-(CF3)2,3,4-Me2,E],[-6135:2,4-(CF3)2,3,4-Me2, E] , C-6136: 2,5-(CF3)2,3,4-Me2,E], [-6137:2,6-(CF3)2,3,4-Me2,E], [-6138 :3,4-(CF3 )2,3,4-Me2 , [-6139:3,5- (CF3 )2,3, 4-Me2 ,E] , C- 6140:2,3-(CHF2 )2 ,3,4-Me2 ,E] , [-6141:2,4- (CHF2 ) 2 r 3,4-Me2 , E ], [-6142:2,5-(CHF2)2,3,4-Me2 , E], [-6143:2,6-(CHF2)2,3,4-Me2,E], [-6144:3,4-(CHF2)2,3,4-Me2,E], [- 6145:3,5-(CHF2)2,3,4-Me2,E], [-614 6:2,3-(CH2 F)2,3,4-Me2,E], [-6147:2, 4-(CH2 F)2,3,4-Me2,E], [-6148:2,5-(CH2F)2,3,4-Me2,E],[-614 9:2, 6- (CH2F ) 24-Me2 , E ], [-6150:3,4- (CH2F) 2,3,4-Me2 ,E],[-6151:3,5- (CH2F) 2,3,4-Me2 ,E ], [-6152:2,3-(MeO)2,3,4-Me2,E], [-6153:2,4-(MeO)2r3,4-Me2,E], [-6154:2, 5-(MeO)2,3,4-Me2,E],C-6155:2,6 -(MeO)2,3,4-Me2,E), C-6156:3,4-(MeO)2,3,4-Me2,E],[-6157:3,5-(MeO)2, 3,4-Me2,E], [-6158:2,3-(EtO)2,3,4-Me2,E],[-6159:2,4-(EtO)2,3,4-Me2, E], [- 171 320202 200901876 616D: 2,5-(EtO) 2,3,4-Me2,E], [-6161:2,6-(EtO)2,3,4-Me2,E], [-6162:3,4-(EtO)2,3,4-Me2,E], [-6163:3,5-(Et〇)2,3,4-Me2,E], [-6164:2 -C1-3-F,3,4-Μθ2/E ] , C -6165:2-C1-4-F,3,4-Μβ2,ED,[-6166:2-Cl-5-F,3, 4-Me2,E ] , C -6167:2-C1-6-F,3,4-Me2,ED,[-6168:3-Cl-2-F,3,4-Me2,E], [- 6169: 3-Cl-4-F, 3,4-Me2, E], [-6170: 3-Cl-5-F, 3,4-Me2, E 3 , C -6171: 4-C1-2- F,3,4-Me2,ED,C~ 6172:4-Cl-3-F,3,4-Me2,E],[-6173:2-F-3-Me,3,4-Me2,E ], [-6174: 2-F-4-Me, 3, 4-Me2, E], [-6175: 2-F-5-Me, 3, 4-Me2, E], [-6176: 2- F-6-Me,3,4-Me2,E],[-6177:3-F-2HMe,3,4-Me2,E]., [-6178:3-F-4-Me,3,4 -Μβ2,ED , C -6179:3-F-5-Me,3,4-Μθ2,ED,C-6180 : 4-F-2-Me, 3,4-Μβ2 , E )1 , C -6181 : 4-F-3-Me, 3, 4-Ηβ2 , EH , C -6182:2-Cl-3-Me,3,4-Μθ2/E ] , C-6183:2-Cl-4-Me, 3,4-Μθ2 λΕ ], [-6184:2-Cl-5-Me,3,4-Me2,E], [-6185:2- Cl-6-Me,3,4-Me2,E], [-6186:3-Cl-2-Me,3,4-Me2,E], [-6187:3-Cl-4-Me,3, 4-Me2,E], [-6188:3-Cl-5-Me,3,4-Me2,E], [-6189:4-Cl-2-Me,3,4-Me2,E], -6190: 4-Cl-3-Me, 3., 4-Me2, E], [-6191: 2-F-3-CF3, 3, 4-Me2, E], [-6192: 2-F- 4-CF3,3, 4-Me2 ,E ) , C -6193:2-F-5-CF3,3,4-Me2 , ED,C-6194:2-F-6-CF3,3,4-Me2 , E], [-6195: 3-F-2-CF3, 3, 4-Me2, E], [-6196: 3-F-4-CF3, 3, 4-Me2, E], [-6197: 3-F-5-CF3,3,4-Me2,E], [-6198:4-F-2-CF3,3,4-Me2,E], [-6199:4-F-3-CF3, 3,4-Me2,E], [-6200:2-Cl-3-CF3,3,4-Me2,E], [-6201:2-Cl-4-CF3,3,4-Me2,E] , [-6202 : 2-C1-5-CF3,3,4-Me2 ,E ) , C -6203:2-CI-6-CF3,3,4-Me2 ,E],C-6204 :3-Cl -2-CF3,3,4-Me2,E] , C-6205: 3-Cl-4-CF3,3,4-Me2,E],[-6206:3-Cl-5-CF3,3,4 -Me2, C-6207: 4-Cl-2-CF3,3, 4-Me2,E ] f C-6208:4-Cl-3-CF3,3,4-Me2,E],[-6209:2 -Me-3-CF3,3,4-Me2,E],[- 172 320202 200901876 6210:2-Me-4-CF3,3,4-Me2,E3, C-6211:2-Me-5-CF3 ,3,4-Me2 , E ], [-6212:2-Me-6-CF3,3,4-Me2,E], [-6213:3-Me-2-CF3,3,4-Me2,E ], [-6214:3-Me-4-CF3,3,4-Me2,E], C-6215: 3-Me-5-CF3,3,4-Me2,E], C~ 6216:4-Me-2-CF3,3,4-Me2,E],[-6217:4-Me- 3-CF3,3,4-Me2,E], [-6218:2-F-3-MeO,3,4-Me2,E], [-6219:2-F-4-MeO,3,4- Me2, E], [-6220: 2-F-5-MeO, 3, 4-Me2, E], C-6221: 2-F-6-MeO, 3, 4-Me2, E 3, C~ 6222 :3-F-2-MeO,3,4-Me2,E], [-6223:3_F-4-MeO,3,4-Me2,E], [-6224:3-F-5-MeOf 3, 4-Me2 , E ] , C -6225 : 4-F-2-MeO, 3,4-Me2 ,E ] , C-6226:4-F-3-MeO,3,4-Me2, C-6227: 2-Cl-3-MeO,3,4-Me2,E), C~6228:2-Cl-4-MeO,3,4-Me2,E], C-6229:2-Cl-5-MeO, 3,4-Me2,E],[-6230:2-Cl-6-MeO,3,4-Me2,E], [-6231:3-Cl-2-MeO,3,4-Me2,E] , [-6232:3-Cl-4-MeO,3,4-Me2,E], [-6233:3-Cl-5-MeO,3,4-Me2,E], [-6234:4-Cl -2-MeO,3,4-Me2,E], [-6235:4-Cl-3-MeO,3,4-Me2,E], [-6236:2-Me-3-MeO,3,4 -Me2,E] , C-6237:2-Me-4-MeO,3,4-Me2,E], C-6238:2-Me-5-MeO,3,4-Μθ2,E] , C- 6239: 2-Me-6-MeO, 3,4-Me2/E], C -6240: 3-Me-2-Me〇, 3,4-Me2, E], [-6241: 3-Me.- 4-MeO,3,4-Me2,E],[-6242:3-Me-5-MeO,3,4-Me2,E], [-6243:4-Me-2-MeO,3,4- Me2, E], [-6244: 4-Me-3-Me〇, 3,4-Me2, E], [-6245: H , 3-F-4-Me, E], [-624 6:4-Ff3-F-4-Me, E 3 , C -6247:4-F,3-F-4-MerZ ] f C -6248 :4-C1,3-F-4-Me,E], [-6249:4-Cl,3-F-4-Me,Z], [-6250:4-Br,3-F-4-Me , E], [-6251: 4-1,3-F-4-Me, E}, [-6252: 4-Me, 3-F-4-Me, E], C-6253: 4-Me, 3-F-4-Me,Z], [-6254:4-Et,3-F-4-Me,E], [-6255:4-C3H7,3-F-4-Me,E], C -6256:4-(Me)2CH,3-F-4-Me,E ] , C -6257 : 4-CF3,3-F-4-Me, E ] , C-6258:4-CF3,3- F-4-Me,Z] , C-6259 : 4-C2 F5,3-F-4-Me, E ] , [-6260:4-C3F7,3-F+Me,E], [ -6261: 4-(CF3)2CF,3-F-4-Me,E],[ -6262:4- 173 320202 200901876 (CF3 )2CH,3-F-4-Me,E 3 ,C-6263: 4-CHF2 , 3-F-4-Me, E ] , [-6264:4-CH2F,3-F-4-Me,E], C -6265 :4-CF3 CH2,3-F-4-Me, E ' i , C -6266: 4-MeO, 3-F-4-Me, E], [-6267: 4-MeO, 3-F-4-Me, Z], [-6268: 4-EtO, 3- F-4-Me, E] , C-6269: 4-C3H7Of 3-F-4-Me,E] , [-627.0 : 4- (Me) 2 CHO, 3-F-4-Me,E], [-6271:4-N02,3-F-4-Me,E], [-6272:4-N〇2,3-F-4-Me,Z], [-6273:3-F,3- F-4-Me, E], [-6274: 3-F, 3-F-4-Me, Z], [-6275: 3-Cl, 3-F-4-Me, E], C-6276 :3-Cl,3-F-4-Me,ZD, [-6277:3-Br,3-F-4-Me, E], [-6278: 3-I, 3-F-4-Me, E], [-6279: 3-Me, 3-F-4-Me, E], [-6280: 3-Me, 3 -F-4-Me,Z], [-6281:3-Et,3-F-4-Me,E], [-6282:3-C3H7,3-F-4-Me,E], [- 6283:3-(Me)2CH,3-F-4-Me,E !J , C-6284 :3-CF3,3-F-4-Me, E 3 , C-6285:3-CF3,3- F-4-Me, ZD, C-6286:3-C2 F5,3-F-4-Me,E) , [-6287:3-C3F7,3-F-4-Me,E ] , C -6288 :3-(CF3 ) 2 CFf 3-F-4-Me, E ] r C -6289:3-(CF3 )2CH, 3-F-4-Me,E ) , C-6290:3-CHF2,3 -F-4-Me, E 3 , [-6291:3-CHF2,3-F-4-Me,Z], [-6292:3-CH2F,3-F-4-Me,E], [- 6293: 3-CH2Fr3-F-4-Me, Z], [-6294: 3-CF3CH2, 3-F-4-Me, E], [-6295: 3-MeO, 3-F-4-Me, E], [-6296: 3-MeO, 3-F-4-Me, Z], [-6297: 3-EtO, 3-F-4-Me, E], [-62 98: 3-C3H70, 3-F-4-Me, E], [-6299: 3-(Me) 2CHO, 3-F-4-Me, E], [-63DD: 3-NO2, 3-F-4-Me, E ], [-6301: 2-F, 3-F-4-Me, E], [-6302: 2-Cl, 3-F-4, Me, E], [-6303: 2-Br, 3- F-4-Me, E], [-6304: 2-I, 3-F-.4-Me, E], C-6305: 2-Me, 3-F-4-Me, ED, [-6306 :2-Et,3-F-4-Me,E],[-6307:2-C3H7,3-F-4-Me,E 3 ,C -6308:2-(Me)2CH,3-F- 4-Me,E ] , C-6309:2-CF3,3-F-4-Me,E), C-6310 :2-C2 F5,3- F-4-Me, E3, [-6311:2-C3F7/3-F-4-Me,E ] , [ -6312:2-(CF3)2CF,3-F-4-Me,E ] , C -6313: 2-(CF3)2CH, 3-F-4-Me, E], C-6314: 2-CHF2, 3-F-4-Me, E], C-6315: 2-CH2F, 3- F-4-Me,E ] , C -6316:2-CF3CH2,3-F-4-Me,E ] , [ -6317:2- 174 320202 200901876

MeO, 3-F-4-Me, E], [-6318: 2-EtO, 3-F-4-Me, E], [-6319: 2-C3H7〇, 3-F-4-Me, E ], [-6320: 2-(Me) 2CHO, 3-F-4-Me, E], [-6321: 2-NO2, 3-F-4-Me, E], [-6322: 2, 3 -F2,3-F-4-Me,E], [-6323:2,4-F2,3-F-4-Me,E], [-6324:2,5-F2,3-F-4 -Me,E],[-6325:2,6-F2,3-F-4-Me,E], [-6326:3,4-F2,3-F-4-Me,ED,C -6327 :3, 4-F2,3-F-4-Me,Z ],C-6328:3,5-F2,3-F-4-Me,E],[-6329:3,5-F2,3 -F-4-Me,Z],[-6330:2,3-Cl2,3-F-4-Me,E ], [ -6331:2,3-Cl2,3-F-4-Me,Z 3, C-6332: 2, 4-CI2, 3-F-4-Me, E], C -6333: 2, 4-Cl2, 3-F-4-Me, Z], [-6334: 2, 5-Cl2,3-F-4-Me,E], [-6335:2,5-Cl2,3-F-4-Me,Z], [-6336:2,6-Cl2,3-F- 4-Me,E 〕 , [-6337:3,4-Cl2,3-F-4-Me,E], [-6338:3,5-Cl2,3-F-4-Me,E],[ -6339: 2,3-Br2,3-F-4U], [-6340:2,4-Br2,3-F-4-Me,E], C-6341:2,5-Br2,3-F -4-Me,E ],[-6342:2,6-Br2,3-F-4-Me,E ] , [-6343:3,4-Br2,3-F-4-Me,E], [-6344:3,5-Br2,3-F-4-Me,E], [-6345:2,3-Me2,3-F-4-Me,E], [-6346:2,4- Me2,3-F-4-Me,E } , [-6347:2,5-Me2,3-F-4-Me,E], [-6348:2,6-Me2,3-F-4- Me, E], [-6349:3, 4-Me2,3-F-4-Me,E],[-6350:3,5-Me2,3-F-4-Me,E 3 f [-6351:2,3-Et2,3-F- 4-Me,E],[-6352:2,4-Et2,3-F-4-Me,E ] f [-6353:2,5-Et2,3-F-4-Me,E], -6354:2,6-Et2,3-F-4-Me,E],[-6355:3,4-Et2,3-F-4-Me,E],[-6356:3,5-Et2 , 3-F-4-Me, E], [-6357:2,3-(CF3)2,3-F-4-Me,E], [-6358:2, 4-(CF3)2,3 -F-4-Me,E],[-6359:2,5-(CF3)2, 3-F-4-Me,E], [-6360:2, 6-(CF3)2,3-F -4-Me, E], [-6361:3,4-(CF3)2,3-F-4-Me,E], C-6362:3,5-(CF3)2,3-F-4 -Me,E ] , [ -6363:2,3-(CHF2)2,3-F-4-Me,E], [-6364 :2,4- (CHF2 )2,3-F-4-Me ,E],[-6365:2,5-(CHF2)2,3-F-4-Me,E],C -6366:2, 6-(CHF2)2,3-F-4-Me,E ], [ -6367:3, 4- 175 320202 200901876 (CHF2) 2,3-F-4-Me,E], [-6368:3,5-(CHF2)2,3-F-4-Me, E], [-6369:2,3-(CH2F) 2,3-F-4-Me,E], [-6370:2,4-(CH2F) 2,3-F-4-Me,E] , C -6371:2,5-(CH2F)2,3-F-4-Me,E 3 ,C -6372 : 2,6-(CH2 F) 2,3-F-4-Me,E], [-6373:3, 4-(CH2F)2,3-F-4-Me,E], [-6374:3,5-(CH2F)2,3-F-4-Me,ED Λ C -6375 :2,3-(MeO)2,3-F-4-Me,E ] f [ -6376:2,4-(MeO 2,3-F-4-Me,E]r[-6377:2,5-(MeO)2,3-F-4-Me,E], [-6378:2,6-(MeO)2 , 3-F-4-Me, E], [-637 9:3,4-(MeO)2,3-F-4-Me,E], [-6380:3,5-(MeO)2, 3-F-4-Me,E], [-6381:2,3-(EtO)2,3-F-4-Me,E], [-6382:2, 4-(EtO)2,3- F-4-Me, E], [-6383: 2,5-(EtO)2,3-F-4-Me, E], C-6384: 2,6-(EtO)2,3-F- 4-Me,E],[-6385:3r4-(EtO)2,3-F-4-Me,E], [-638 6:3,5-(EtO)2,3-E-4-Me , E3, C-6387: 2-C1-3-F, 3-F-4-Me, E], [-6388: 2-Cl-4-F, 3-F-4-Me, E], [ -6389: 2-Cl-5-F, 3-F-4-Me, E], [-6390: 2-Cl-6-F, 3-F-4-Me, E], C-6391:3 -C1-2-F,3-F-4-Me,E],[-6392:3-Cl-4-F,3-F-4-Me,E ] , C-6393:3-C1-5 -F,3-F-4-Me,ED,C-6394:4-Cl-2-F,3-F-4-Me,E],[-6395:4-Cl-3-F,3- F-4-Me, E], [-6396: 2-F-3-Me, 3-F-4-Me, E], [.-6397: 2-F-4-Me, 3-F-4 -Me,E],[-6398 :2—F-5—Me, 3-F-4-Μθ,E], [-6399: 2-F-6—Me, 3-F-4-Me, E 3 fC-6400: 3-F-2-Me, 3-F-4-Me/E3, C-6401: 3-F-4-Me, 3-F-4-Me, E], C~ 6402: 3-F-5—Me, 3-F-4—Me, E ] , C ~6403: 4-F-2—Me, 3—F—4—Me, ED f C-6404:4-F-3 -Me,3-F-4-Me,E ] , [-6405:2-Cl-3-Me,3-F-4-Me,E],[- 6406: 2-Cl-4-Me, 3-F-4-Me, E], [-6407: 2-Cl-5-Me, 3-F-4-Me, E], [-6408:2- Cl-6-Me, 3-F-4-Me, E], [-6409: 3-Cl-2-Me, 3-F-4-Me, E], [-6410: 3-Cl-4- Me, 3-F-4-Me, E], [-6411: 3-Cl-5-Me, 3-F-4-Me, E], [-6412: 4-Cl-2-Me, 3- F-4-Me, E], [-6413: 4-Cl-3-Me, 3-F-4-Me, E], [-6414: 2-F-3-CF3, 3-F-4- Me, E], [-6415: 2-F-4-CF3, 3-F-4-Me, E], [- 176 320202 200901876 6416: 2 —F-5-CF3,3-F-4-Me , E], C~6417:2—F—6—CF3,3-F-4-Me, eD, C~ 6418:3-F-2-CF3,3-F-4-Me,E], -6419: 3-F-4-CF3, 3-F.-4-Me, E], [-6420: 3-F-5-CF3, 3-F-4-Me, E], [-6421: 4-F-2-CF3,3-F-4-Me,E], [-6422:4-F-3-CF3,3-F-4-Me,E], [-6423:2-Cl- 3-CF3,3-F-4-Me,E], [-6424:2-Cl-4-CF3,3-F-4-Me,E], [-6425:2-Cl-5-CF3, 3-F-4-Me, E], [-6426: 2-Cl-6-CF3, 3-F-4-Me, E], [-6427: 3-Cl-2-CF3, 3-F- 4-Me, E], [-6428: 3-Cl-4-CF3, 3-F-4-Me, E], [-6429: 3-Cl-5-CF3, 3-F-4-Me, E], C-5430: 4-Cl-2-CF3, 3-F-4-Me, E], [-6431: 4-CI-3-CF3, 3-F-4-Me, E], C -6432: 2-Me~3-CF3,3-F-4-Me,E],[-6433:2-Me-4-CF3,3-F-4—Me,E], [-6434:2 -Me -5-CF3,3-F-4-Me,E],[-6435:2-Me-6-CF3,3-F-4-Me,, [-6436:3-Me-2-CF3,3 -F-4-Me,E], [-6437:3-Me-4-CF3,3-F-4-Me,E], C-6438:3-Me-5-CF3,3-F-4 -Me,E],C-6439:4-Me-2-CF3,3-F-4-Me,E], [-6440:4-Me_3_CF3,3-F-4-Me,E], [- 6441: 2-F-3_Me〇, 3-F_4-Me, E], C-6442: 2-F-4-MeO, 3-F-4-Me, E], [-6443: 2-F-5 -MeO,3-F-4-Me,E], [-6444:2-F-6-MeO,3-F-4-Me,E], [-6445:3-F-2_MeO,3-F_4 -Me,E], [1-64:3—F-4_Me〇, 3_F_4-Me, E], [1-64:3_F—5—Me〇, 3-F “4—Me, E], C-6448: 4-F-2-MeO,3-F-4-Me,E], [-6449:4-F-3-MeO,3-F-4-Me,ED, [-6450:2-Cl-3 -Me〇,3-F-4-Me,E], [-6451:2-Cl-4-Me〇, 3-F-4-Me,E], [-6452:2-Cl-5-MeO , 3-F-4-Me, E], [-6453: 2-Cl-6-MeO, 3-F-4-Me, E], C-6454: 3-Cl-2-MeO, 3-F -4-Me,E],[-6455:3-Cl-4-MeO,3-F-4-Me,E], [-6456:3-Cl-5-MeO,3-F-4-Me , E], [-6457: 4-Cl-2-MeO, 3-F-4-Me, E], [-6458: 4-Cl-3-MeO, 3-F-4-Me, E], [-6459: 2-Me-3-MeO, 3-F-4-Me, E], [-64 60: 2-Me-4-MeO, 3-F-4-Me, E], [-6461 :2-Me-5-MeO,3-F-4-Me,E], f-6462:2-Me-6—MeO,3-F—4—Me, El, C—6463 :3—Me-2-MeO,3-F—4-Me, ED ^ [-64 64:3-Me-4—Me〇, 3-F_4 —Me, E], [-6465:3-Me- 5-MeO,3-F-4—Me, E], 177 320202 200901876 C-64 66:4-Me-2-MeO,3-F-4-Me, E] , C-64 67:4-Me -3-MeO,3-F-4-Me,E], [-6468:H,4-F-3-Me,E],[-6469:4-F,4-F-3-Me,E ], [-6470: 4-F, 4-F-3-Me, Z], [-6471: 4-Cl, 4-F-3-Me, E], [-6472: 4-Cl, 4- F-3-Me,Z], [-6473:4-Br,4-F-3-MefE], [-6474:4-1,4-F-3-Me, E], [-6475:4 -Me,4-F-3-Me,E],C-6476:4-Me,4-F-3-Me,Z], C-6477:4-Et,4-F-3-Me,E ],[-6478:4-C3H7,4-F-3-MerE 3 , C -6479:4-(Me)2CH,4-F-3-Me,E ] f C-6480:4-CF3,4 -F-3-Me,E], [-6481:4-CF3,4-F-3-Me,Z], [-6482:4-〇2 F5> 4-F-3-Me, E], [ -6483 : 4-C3 F7,4-F-3-Me, E], C -6484: 4-(CF3)2CF, 4-F-3-Me, E], [-6485:4-(CF3 ) 2CH., 4-F-3-Me, E], [-6486: 4-CHF2, 4-F-3-Me, E], [-6487: 4-CH2F, 4-F-3-Me, E3, [-6488: 4-CF3CH2, 4-F-3-Me, E], C-6489: 4-MeO, 4-F-3-Me, E], [-6450: 4-MeO, 4- F-3-Me,Z], [-6491:4-EtO,4-F-3-Me,E], C-64 92 : 4-C3 H7 0, 4-F-3-Me,E], [ -6493:4-(Me)2CHO, 4-F-3-Me,E ] , C -6494 :4-N02,4-F-3-Me,E , [-6495: 4-N02, 4-F-3-Me, Z], [-6496: 3-F, 4-F-3-Me, E], [-6497: 3-F, 4-F -3-Me,Z], [-6498:3-Cl,4-F-3-Me,E], [-6499:3-Cl,4-F-3-Me,Z], [-6500: 3-Br,4-F-3-Me,E], [-6501:3-I,4-F-3-Me,E], [-6502: 3-Me, 4-F-3-Me, ED , C -6503 : 3-Me, 4-F-3-Me, Z 3 / C -"6504:3-Et,4-F-3-Me,E ] , [ -6505:3-C3H7, 4-F-3-Me,E ] , C -6506:3-(Me)2CH, 4-F-3-Me,E ] , [ -6507 : 3-CF3,4-F-3-Me,E "} , C -6508 :3-CF3 f 4-F-3—Me, z], [-6509: 3-C2 F5,4-F-3-Me , C~6510: 3—C3 F7,4 —F-3-Me,E ] r C -6511:3-(CF3)2CF,4-F-3-Me,E ] , C -6512:3-(CF3)2CH,4-F-3-Me , ED, C-6513: 3-CHF2, 4-F-3-Me, E], C-6514: 3-CHF2, 4-F-3-Me, Z], C-6515: 3-CH2 F, 4-F-3-Me, E], C-6516: 3-CH2 F, 4-F-3-Me, Z], C-6517: 3-CF3CH2, 4-F-3-Me, E], C-6518 : 3-MeO, 4-F-3-Me, E], [-6519: 3-MeO, 4-F-3-Me, Z], [-6520: 3-EitO, 4-F- 3-Me,E],[- 178 320202 200901876 6521:3-C3H70,4-F-3-Me,E] , [-6522 : 3-(Me) 2 CHO, 4-F-3-Me, E 3 f [-6523:3-N〇2,4-F-3-Me,E], C -6524:2-F,4-F-3-Me,E } , C -6525:2-Cl, 4-F-3-Me, E], [-6526 :2-Br,4-F-3-Me,E], [-6527:2-I,4-F-3-Me,E], [-6528:2-Mer4-F-3-Me,E ], [-6529: 2-Et, 4-F-3-Me, E], [-6530: 2-C3H7, 4-F-3-Me, E], C-6531: 2-(Me)2CH , 4-F-3-Me, E 3 , C -6532: 2-CF3,4-F-3-Me,E] , C-6533:2-C2F5,4-F-3-Me,E], C-6534: 2-C3 F7,4-F-3-Me,E], C-6535:2-(CF3)2CFr4-F-3-Me,E], C-6536:2-(CF3)2CH , 4-F-3-Me, E ] , C-6537: 2-CHF 2,4-F-3-Me, E ] , [ -6538:2-CH 2 F, 4-F-3-Me, E ], [-6539: 2-CF3CH2, 4-F-3-Me, E], C -6540: 2-MeO, 4-F-3-Me, E], C-6541: 2-EtO, 4-F- 3-Me,E] , C-6542:2-C3H7Of4-F-3-Me,E],[-6543:2- (Me )2 CHO, 4-F-3-Me,E],[-654 4 :2.-N02 r 4-F-3-Me,E], [-6545:2,3-F2,4-F-3-Me,E], [-6546:2,4-F2,4 -F-3-Me,E],[-6547:2,5-F2,4-F-3-Me,E ] , C -6548:2,6-F2,4-F-3-Me,E ], C-6549: 3,4-F2,4-F-3-Me, E], [-6550:3,4-F2,4-F-3-Me,Z], [-6551:3, 5-F2,4-F-3-Me,E ] , [ -6552:3,5-F2,4-F-3-Me,Z ], C-6553:2,3-Cl2,4-F- 3-Me,E ] , [ -6554 :2,3-Cl2,4-F-3-Me, Z 6555:2,4-Cl2,4-F-3-Me,E ], [ -6556:2 , 4-Cl2,4-F-3-Me, Z 6557: 2,5-Cl2,4-F-3-Me,E], [-6558:2,5-Cl2,4- F-3-Me,Z]r[-6559:2, 6-Cl2,4-F-3-Me,E], [ -6560:3, 4-Cl2,4-F-3-Me,E ] , C-6561: 3,5-Cl2,4-F-3-Me, E 3 , [-6562:2,3-Br2,4-F-3-Me,E], [-6563:2,4 -Br2,4-F-3-Me,E], [-6564:2,5-Br2,4-F-3-Me,E],[-6565 : 2, 6-Br2 / 4-F-3 -Me, ED, [ -6566: 3,4-Br2,4-F-3-Me, E !3,C -6567:3,5-Br2,4-F-3-Me,E ] , 〔- 6568: 2,3-Me2,4-F-3-Me,E], [-6569:2,4-Me2,4-F-3-Me/E 3 , C -6570 :2,5-Me2, 4-F-3-Me, E !], [-6571:2,6-Me2,4-F-3-Me,E], [ -6572:3,4-Me2,4-F-3-Me , E 3 ,- 179 320202 200901876 6573:3,5-Me2,4-F-3-Me,E], [-6574:2,3-Et2,4-F-3-Me,E], [- 6575:2,4-Et2,4-F-3-Me,E 3 ,C -6576:2,5-Et2f4-F-3-Me,E Jri~ 6577:2,6-Et2,4-F- 3-Me, E], [-6578:3,4-Et2,4-F-3-Me,E], [-6579:3,5-Et2,4-F-3-Me,E], -6580:2, 3-(CF3)2,4-F-3-Me,E], [-6581:2,4-(CF3)2,4-F-3-Me,E], [-6582 :2,5-(CF3 )2 ,4-F-3-Me,E], [-6583:2,6-(CF3)2,4-F-3-Me,E], [-6584:3 , 4-(CF3)2,4-F-3-Me,E], [-6585:3,5-(CF3)2,4-F-3-Me,E], [-6586:2,3 -(CHF2)2,4-F-3-Me,E],[-6587:2,4-(CHF2)2,4-F-3-Me,E],[-65 88:2,5-(CHF2)2,4-F-3-Me,E], [-6589:2,6-(CHF2)2,4-F-3-Me,E], [-6590: 3,4-(CHF2)2,4-F-3-Me,E], [-6591:3,5-(CHF2)2,4-F-3-Me,E], [-6592:2, 3-(CH2F) 2 , 4-F-3-Me, E], [-6593 : 2,4-(CH2F) 2 ,.4-F-3-Me, E], [-6594:2,5 -(CH2F)2,4-F-3-Me,E],[ -6595 :2,6-(CH2 F) 2 , 4-F-3-Me,E] , [-6596:3,4- (CH2 F) 2 , 4-F-3-Me, E] , [-6597:3,5- (CH2F)2 , 4-F-3-Me,ED , [ -6598:2,3-(MeO ) 2,4-F-3-Me/E "} , C -6599:2, 4-(MeO)2,4-F-3-Me,E], [-6600:2,5-(MeO 2,4-F-3-Me,E],[-6601:2,6-(MeO)2,4-F-3-Me,E] , [-6602:3,4-(MeO)2 ,4-F-3-Me,E], [-6603:3,5-(MeO)2,4-F-3-Me,E],C-6604:2,3-(EtO)2,4 -F-3-Me,E], [-6605:2,(EtO)2,4-F-3-Me,E],[-6606:2,5-(EtO)2,4-F-3 -Me,E], [-6607:2,6-(EtO)2,4-F-3-Me,E], [-6608:3,4-(EtO)2,4-F-3-Me , E], [-6609:3,5-(EtO)2,4-F-3-Me,E], C-6610:2-C1-3-F,4-F-3-Me,E] , [-6611: 2-Cl-4_F, 4_F_3_Me, E], [-6612: 2_Cl_5-F, 4-F_3_Me, E], [-6613: 2-Cl-6-F, 4-F-3-Me ,E] , C -6614 :3-C1-2-F,4-F-3-Me, E] , C -6615:3_Cl_4_F,4_F-3_Me,E],[-661 6:3-Cl-5-F, 4_F_3-Me, E], [-6617: 4-Cl-2-F, 4-F-3-Me, E], C-6618: 4-C1-3- F,4-F-3-Me, E ], [-6619:2-F-3-Me,4-F-3-Me,E], [-6620:2-F-4-Me,4- F-3-Me, E], [- 180 320202 200901876 6621: 2-F-5-Me, 4-F-3-Me, E], [-6622: 2-F-6-Me, 4-F -3-Me, E], [-6623: 3-F-2-Me, 4-F-3-Me, E], [-6624: 3-F-4-Me, 4-F-3-Me , E], [-6625: 3-F-5-Me, 4-F-3-Me, E], [-6626: 4-F-2-Me, 4-F-3-Me, E], [-6627: 4-F-3-Me, 4-F-3-Me, E], [-6628: 2-Cl-3-Me, 4-F-3-Me, E], [-6629: 2-Cl-4-Me,4-F-3-Me,E], [-6630:2-Cl-5-Me,4-F-3-Me,E], [-6631:2-Cl- 6-Me, 4-F-3-Me, E], [-6632: 3-Cl-2-Me, 4-F-3-Me, E], [-6633: 3-Cl-4-Me, 4-F-3-Me,E] , C-6634:3-Cl-5-Me,4-F-3-Me,E], C-6635:4-Cl-2-Me,4-F- 3-Me, E], [-6636: 4-Cl-3-Me, 4-F-3-Me, E], [-6637: 2-F-3-CF3, 4-F-3-Me, 6638:2 —F-4-CF3,4-F-3-Me, E],C-6639:2-F-5-CF3,4-F-3-Me,E] , C-6640 :2- F-6-CF3,4-F-3-Me, E3, [-6641:3-F-2-CF3,4-F-3-Me,E], [-6642:3-F-4-CF3 ,4-F-.3-Me,E], [-6643:3-F-5-CF3,4-F-3-Me,.E], C-6644 : 4-F-2-CF3 , 4 -F-3-Me, E ] , C~ 6645:4-F -3-CF3,4-F-3-Me,E], [-6646:2-Cl-3-CF3,4-F-3-Me,E], [-6647:2-Cl-4-CF3 /4-F-3-Me,E] , C-6648:2-Cl-5-CF3,4-F-3-Me,E], [-6649:2-Cl-6-CF3,4-F -3-Me,E],[-6650:3-Cl-2-CF3,4-F-3-Me,E], [-6651:3-Cl-4-CF3,4-F-3-Me , E], [-6652: 3-Cl-5-CF3, 4-F-3-Me, E], [-6653: 4-Cl-2-CF3, 4-F-3-Me, E], [-6654: 4-Cl-3-CF3,4-F-3-Me, E], [-6655:2_Me_3_CF3,4_F-3-Me,E], [-6656:2_Me_4_CF3,4_F_3-Me,E] , C-6657: 2-Me-5-CF3, 4-F-3-Me, E], [-6658: 2-Me-6-CF3, 4-F-3-Me, E], [-6659 :3-Me-2-CF3,4-F-3-Me,E], [-6660:3-Me-4-CF3,4-F-3-Me,E], [-6661:3-Me -5-CF3,4-F-3-Me,E], [-6662:4-Me-2-CF3,4-F-3-Me,E], [-6663:4-Me_3-CF3,4_F_3 -Me, E], [-6664: 2_F_3_Me〇, 4_F-3_Me, E], [-6665: 2-F-4-MeO, 4-F_3-Me, E], [-6666: 2_F-5-Me 〇, 4_F-3-Me r E], C-6667: 2-F-6-MeO, 4-F-3-Me, E], C-6668: 3-F-2-MeO, 4-F- 3-Me,E ], C-6669:3-F-4-MeO,4-F-3-Me,E] , C-6670:3-F-5-MeO,4-F-3-Me, E], 181 320202 200901876 [-6671: 4-F-2-MeO/· 4-F-3-Me, E], [ -6672 : 4~F-3-MeO, 4-F-3, m ® ' E〕 C-6673 :2-Cl-3-MeO,4-F-3-Me,E),C-6674:2~Cl-4-MeO [-6675:2-Cl-5-MeO, 4-F-3-Me , E], [-6676: 2-ci-6-MeO 4K ', for example, C-6677: 3-Cl-2-MeO, 4-F-3-Me/E), C-6678: 3- Ci-4-MeO,4-F~^ C-6679:3-Cl-5-MeO,4-F-3-Me,E), C-6680:4-ci-2-MeO 4-F -3⁄4 'Heart', le'E], [-6681:4-Cl-3-Me〇,4-F-3-Me,E], [-6682:2-Me-3-MeO,4-F-3 m [-6683:2-Me-4-MeO,4-F-3-Me,E], [-6684:2-Me-5-MeO,4-F-3,m [-6685:2- Me-6-MeO, 4-F-3-Me, E], [-6686: 3-Me-2-MeO 4-F*o C-6687: 3-Me-4-MeO, 4-F-3 -Mef E],[-6688:3~Me-5-MeO 4-F-^ ' C-6689:4-Me-2-MeO, 4-F-3-Me,E], C-6690: 4 -Me_3-MeO 4-F--5 In the above "combination G", 'for example, «) „ is “h” means m = 〇(X)m is “4-F” means m=l and X is fluorine. The atom is substituted with 4~only, (χ) is "2,3-(CF3)2" means m=2 and one X is trifluoromethyl substituted for / and the other X is trifluoromethyl substituted for 3 - bit; (2) „ is “Hj yellow finger n= 0 '(Z)4 “.4-MeO” means n=l and Z is methoxy substituted in 4_ bit '(Z)n is “3- F-4-(Me)3C0" means n=2 and one Z is a gas atom substituted for the 3-position and another Z The third butoxy group is substituted at the 4-position; the geometric isomer of the CH=CH double bond is "E" means that the isoform of the CH=CH double bond in the formula (I) is E (the entgegen) The isomer, and the geometric isomer of the cH=CH double bond is "Z" means that the isomer of the CH=CH double bond in the formula (I) is a Z (samem) isomer. Example 1 Compound 2-94: Bicyclo[4.4.0]-3-indolyl 3-(3,5-dichlorophenylthio)-indole-(phenyl)thiopropene imidate 182 320202 200901876

Bicyclo[4.4.0]-3-mercapto N-(phenyl)thiopropyneimide (0.11 bogey) was dissolved in decyl alcohol (1〇1111〇, and it was added at room temperature 3 , 5-dichlorothiophenol (0. 05g), followed by stirring for 4 hours. The reaction mixture was concentrated under reduced pressure. The residue obtained was subjected to silica gel column chromatography (hexane / ethyl acetate = 30/1), followed by medium pressure Preparative HPLC (hexane/ethyl acetate = 99.2/0.8) to give bicyclo[4.4.0]-3-indolyl 3-(3,5-dichlorophenylthio)- N-(phenyl) thioacrylic acid imidate (0.07g). NMR (CDC13) δ (ppm): 1.23-2.16 (16H, m), 3.67-3.74 (0.7H, m), 3.95 (0.2H, br), 4.31 (0.1H, br), 6.14 (1H, d, J= 15.5 Hz), 6.72-6.74 (2H, m), 7.03-7.07(1H, m), 7.20-7.34 (6Η m) Example 2 _ Compound 2-4: Bicyclo[4.4.0]-3-indolyl 3-(4-chlorophenylthio)-N-(phenyl)thiopropene imidate ester

Bicyclo[4. 4. Q]-3-indolyl N-(phenyl)-3-(tridecyldecylalkyl) thiopropyneimidate (0.40 g) was dissolved in methanol (10 mL). A small amount of potassium carbonate was added thereto at room temperature, followed by stirring for 1 hour. Then, 4-chlorothiophenol (0.087 g) was added to the mixture at room temperature, followed by stirring for 4 hours. After concentrating the reaction under reduced pressure 183 320202 200901876, the mixture was subjected to a column chromatography (hexane/ethyl acetate = 30/1), followed by medium pressure preparative HPLC (hexane / ethyl acetate = 99.2 / 0.8) Preparation of bicyclo[4.4.0]-3-indolyl 3-(4-chlorophenylthio)-N-(phenyl)thiobis-sodium imidate (10 g). 3.65-3.73 (0.7H, (1H, d, J= 15.2 7.23-7.28 (7H, 1H NMR (CDC13) δ (ppm): 1.22-2.15 (16H, m) m), 3.94 (0.2H, br), 4.30 (0.1H, br), 6·〇2

Hz), 6.69-6.71 (2H, m), 7.01-7.05 (iH, m) m) The following compound was prepared in the same manner as in Example 2: Compound 2-8: Bicyclo[4.4·0]-3-癸Base q, (phenyl) thiopropylene oxime imine coffee 3~(4'methylphenylthio)♦

3.64-3.72 (0.7H, m), 3·93 (0.2H, br) (1H,d, J= 15.4 Hz)f 6.69-6·7ΐ .(2g compound 2-8 坩), 2.31 (3H, s ), 4*28 (0.1H, br), 5.97 is called 'β.98~7.〇9 (3H m) 7.21-7.25 (4H, m), 7.32 (1H, d, lc ( ? 丄Hz) Compound 2 -22: Bicyclo[4·4·0]~3~癸0 π-signed d-(4-methylchlorofu 1; ε* group)-N-(phenyl) thiopropionimide vinegar Soil

HaCO

320202 184 200901876 ^NMR (CDC13) δ (ppm): 1.21-2.14 (16H, τη), 3.63-3.71 (0.7H, m), 3.77 (3H, S), 3.92 (0.2H, br), 4.28 (0.1 H, br), 5.86 (1H, d, J= 15.4 Hz) f e.67-6.69 (2H, m), 6.78-6.80 (2H, m), 6.97-7.01 (in, m), 7.20-7.33 ( 5H, m) Compound 2-31: Bicyclo[4.4.0]-3-indolyl 3-(3-chlorophenylthio)-N-(phenyl)thiopropene imidate

Compound 2-31

IjiNMR (CDCI3) δ (ppm): 1.26-2.15 (16H, in), 3.67-3.73 (0.7H, 3.94 (〇.2H, br), 4.30 (0.1H, br}, 6.10 (1H, d, J= 15.4Hz), 6.72-6.73 (2H, m), 7.01-7.05 (1ΗΓ m) , 7.21-7.34 (7H, m) Compound 2-35: Bicyclo[4.4. 0]_3-indolyl 3-(3-曱Phenylthio)-N-(phenyl)thiopropene imidate

Compound 2-35 3.65-3.72 (0.7H, m), 3.93 (0.2H, br), 4.29 (0.1H, br), 6.05 (1H, d, J = 15.6 Hz), 6.71-6.73 (2H, m) , 7.00-7.39 (8H, m) Compound 2-36: Bicyclo[4.4.0]-3-indolyl 3-(4-mercaptophenylthio)-N-(phenyl)thiopropene oxime Imidate 185 320202 200901876

^NMR (CDC13) δ (ppm): 1.20-2.00 (16H, m), 2.34 (3H, s), 3.18 (0.6H, br), 3.40 (0.2H, br), 3.81 (0.2H, br), 6.39-6.41 (1H, m), 6.97-7.33 (10H, m) Compound 2-29: Bicyclo[4. 4.0]-3-indolyl 3-(3-fluorophenylthio)-N-(phenyl Thiopropenyl imidate

S-CH^CH~C==N—Compound 2-29 ^NMR (CDCI3) δ (ppm) : 1.22-2.02 (16Η, m) , 3.66-3.74 (0.7Η, m), 3.94, (.0.2Η , br), 4.30 (0.1Η, br), 6.11 (1Η,. d, J= 15.6 Hz), 6.72-6.74 (2H, m), 6.94-7.12 (4H, m), 7.23-7.35 (4H, m Compound 2-27: Bicyclo[4.4.0]-3-indolyl 3-(4-nitrophenylthio)-N-(phenyl)thiopropene imidate

^NMR (CDCI3) δ (ppm): 1.26-2.19 (16H, m), 3.69-3.76 (0.7H, m), 3.98 (0.2H, br), 4.33 (0.1H, br), 6.31 (1H, d , J= 15.4 Hz), 6.74-6.76 (2H, m), 7.04-7.08 (1H, m), 7.25-7.34 (3H, m) , 7.42 (2H, dr J= 8.9 Hz), 8.15 (2H, d , J= 8.9 Hz) 186 320202 200901876 Compound 2-40: Bicyclo[4.4.0]-3-indolyl N-phenyl-3-(3-trifluoromethylphenylthio)thiopropene oxime Imidate

Compound 2-4 0 NMR (CDC13) δ (ppm): 1.22-2.15 (16H, m), 3.67-3.74 (0.7H, m) f 3.95 (0.2H, br), 4.31 (0.1H, br) , 6.08 (1H, d, J = 15.4 Hz)f 6.70-6.72 (2H, m), 7.00-7.04 (1H, m)f 7.23-7.61 (7H, m). Compound 2-13: Bicyclo[4.4. 0] -3-decyl N-phenyl-3-(4-trifluoromethylphenylthio)thiopropenyl imidate

XHNMR (CDCI3) δ (ppm): 1.23-2.14 (16H, m), 3.68-3.75 (0.7H, m), 3.96 (0.2H, br), 4.31 (0.1H, br), 6.15 (1H, d, J = 15.6 Hz), 6.72-6.73 (2H, m), 7.02-7.06 (1H, m), 7.24-7.55 (7H, m) Example 3 Compound 2-5354: Bicyclo[4.4. 0]-3-癸3-(4-fluorophenylthio)-N-(4-methylphenyl)thiopropene imidate

187 Compound 2-5354 320202 200901876 Ethyl tridecylamine (0.7 mL) was dissolved in anhydrous THF (i〇mL), and n-butyl hexane was added dropwise at -78 °C. 157 m〇i/L: 3.4 mL), and the resulting mixture was heated to 〇 °C. A solution of 4-mercaptophenyl isothiocyanate (〇.75 mL) in THF (3 mL) was added dropwise to the mixture, followed by stirring for 30 minutes under ice cooling. A solution of bicyclo [4 4. 〇]_3_ mercaptomethanesulfonate (1.3 g) in THF (2 mL) was then added to the reaction mixture and the mixture was stirred for 6 hours under hot reflux. A saturated aqueous solution of sodium hydride (15 mL) and water (1 mL) were added to the mixture, and then extracted twice with n-butyl methyl ether (2 mL). The obtained organic layer was washed with saturated aqueous sodium sulfate (2 mL). The oil was subjected to column chromatography on florisil (hexane/ethyl acetate = 3 〇/1) to obtain bicyclo[4.4.0]-3-indenyl N-(4-methylbenzene). Base)-3-(trimethylsulfonic acid) thioacrylic acid imidate. • The resulting bicyclo [4.4·0]-3-indolyl-(·4-mercaptophenyl)-3-(tridecylfluorenyl) thiopropyne imidate is dissolved in sterol (l〇 (mL), and a small amount of potassium carbonate was added to the solution at room temperature, followed by stirring for 30 minutes. Then, 4-chlorothiophenol (〇. 〇 8 mL) was added thereto at room temperature, followed by stirring for 2 hours. The reaction mixture was concentrated under reduced pressure. The residue obtained was subjected to a column chromatography (hexane/acetic acid ethyl acetate = 30/1), followed by medium pressure preparative jjPLC (hexane/ethyl acetate = 99 2 / 0.8). 4. 〇]-3-mercapto 3-(4-fluorophenylthio)-N-(4-nonylphenyl) thiopropenyl imidate (0.16 g). 320202 188 94 200901876

^NMR (CDC13) δ (ppm): 1.20-2.14 (ifiM,m), 2.30 (3H, s), 3.64-3.72 (0.7H, m), 3.93 (0.2H, :br, Λ 4.30 (〇·ΐΗ , br), 5. (1H, d, J= 15.5 Hz), 6.59 (2H, df ja R . _ Hz)f 6.95-6,99 (2H, 7.03 (2H, d, J= 8.0 Hz), 7.24 nH ′′ is d, 15.5 Hz), 7.28-7.33 (2H, m) The following compounds were prepared in the same manner as in Example 3: Compound 2-2: Bicyclo [4.4. 0]-3-indenyl (phenyl) Thiopropenyl imidate 3~(4-fluorophenylthio)_N_

W (CDCI3) δ (ppm): 1.22-2.16 (l6H.rm), 3.64-3.72 (0.8H, m), 4.29 (0.2H, br), 5.92 (1H, d, j* 15.4 Hz>, 6.68_6 .7〇(2H, m), 6.96-7.04 (3H, m), 7.22-7.34 (5h, compound 2-448. Bicyclo[4.4.0]-3-indolyl N-(4-chlorophenyl) )-3-(4-fluorophenylthio)thiopropenyl imidate

Compound 2-448 t) , 3.61-3.69 (0.7H, m), 3.90 (0.2H, br), 4.26 (0.1H, br), 5.82 (1H, d, j= 15,4 Hz), 6.62 (2H , d, J = 8·5 Hz), 6.98-7.02 (2ΙΪ, m), 7.19 (2H, d, J= 8.5 Hz), 7.24-7.33 (3H, m) Compound 2-894: _ double ring [4. 4. 0]·~3-mercapto 3-(4-fluorophenylthio)-N-(decyloxyphenyl)thiopropene imidate 189 320202 200901876

Compound 2-894 ^NMRiCDCls) δ (ppm): 1.18-1.89 (16Η, m), 3.64-3.71 (1H, m), 3.80 (3H, s), 5.98 (1H, d, J = 15.4Hz), 6.65 (2H, d, J = 8.5Hz), 6.80 (2H, d, J = 8.5Hz), 6.96-7.03 (2H, m), 7.25 (1H, d, J = 15.4Hz), 7.33-7.37 (2H, m) Compound 2-1786: Bicyclo[4.4. 0]-3-indolyl 3-(4-fluorophenylthio)_N-(trimethyldecylphenyl)thiopropene succinimide

^NMRiCDCls) δ (ppm): 1.22-1.85 (16H, m), 3.63-3.68 (1H, m), 5.64 (1H, d, J= 15.4Hz), 6.82-6.98 (4H, m) , 7.2 6- 7.33, (5H, m) Compound 2-6023: Bicyclo[4. 4. 0]-3-indenyl N-(3,4-dimercaptophenyl)-3-(4-fluorophenylthio) Thiopropene broiled imiline vinegar

^NMRiCDCls) δ (ppm): 1.21-1.89 (16H, m), 2.20-2.22 (6H, m), 3.63-3.71 (0.7H, m), 3.92 (0.2H, br), 4.28 (0.1H, br ), 5.97 (1H, d, J = 15.4Hz), 6.43 (1H, d, J = 7.8Hz), 6.48 (1H, s), 6.95-7.00 (3H, m), 7.20-7.25 (1H, m) 7.31-7.34 (2H, m) 190 320202 200901876 Next, a description will be given of a production example of the starting compound of the compound (i). Production Example 1 Bicyclo[4·4·0]-3-indolyl N-(phenyl)-3-(trimethyldecyl)thiopropenyl imide

The ethynyl trimethyl sulphate (4·1 mL) was dissolved in anhydrous THF (80 mL), and a solution of n-butyl oxime in hexane (1. 57 mol/L: 20 mL) was added dropwise at -78 ° C, and the obtained The mixture was warmed to 0 °C. To the mixture was added dropwise a solution of phenyl isothioate (3.7 mL) in THF (5 mL), followed by ice-cooled sandalwood for 3 min. A solution of the bicyclo[4.4.0]-3-indolylmethyl sulphonate (7. 74 g) in THF (3 mL) was then added to the reaction mixture and the mixture was stirred under hot reflux for 6 hours. A saturated aqueous solution of sodium chloride (8 mL) and water (20 mL) were then added to the mixture, and then extracted twice with n-butylmethyl ether (8 mL and 40 mL). The organic layer was washed with a saturated aqueous solution of sodium sulfate (8 mL). The oil was subjected to alumina column chromatography (hexane/ethyl acetate = 3 〇 /1) to give bicyclo[4·4.0]-3-indolyl N-(phenyl)-3-( Trimethyl decyl) thiopropenyl imidate (4.22 g). ^HNMR (CDC13) δ(ρρπι): 0.09 (5H, s), 〇·29 (4H, s), um 9〇(16Η, m), 3.50-3.58 (0.4Η, m), 3.70-3.77 (0.6 Η, m) ^ 6.88-6.91 (1Η, ία), 7.02-7.05 (1Η, m), 7.08-7.14 (1Η, eg, 7.28_ 7.36 (2H, m). 191 320202 200901876 Manufacturing Example 2 Double loop [4· 4. 0]-3-mercapto (local) thiopropynyl imidate 酉t

Dissolving bicyclo[4.4.0]-3-indolyl-(phenyl)-3-(trimethyldecyl) thiopropene imidate (〇.18g) in decyl alcohol (1〇mL) And - a small amount of potassium carbonate was added to the solution, followed by stirring for 1 hour. The reaction mixture was concentrated under reduced pressure and extracted with water (10 mL) and chloroform. The organic layer was dried, and the solvent was evaporated to give bicyclo[4.</RTI>> ^NMR (CDC13) δ (ppm): 1.24-1.86 (16H, m) q ,, ' (0.7H, s), 3.38 (0.3H, s), 3.53-3.61 (0.3H, m) , 3.72-- 3⁄4 an 3'8〇(0.7H, m), 6.90-7.14 (3H, m), 7.31-7.37 (2H, m) Next, the formulation example will be described. Parts are parts by weight. Formulation Example 1 Compound 2-2, Compound 2-4, Compound 2-8, Compound 2-13, Compound 2-22, Compound 2-27, Compound 2-29, Compound 2-31, Compound 2-35, Compound 2-36, Compound 2-40, compound 2_94, compound 2-48 and compound 2-5354 were each dissolved in a mixture of milk xylene and 35 N,N-monodecylamine. To this was added 14 parts of polyoxyethylidene phenyl ether and 6 parts of calcium dodecylbenzenesulfonate, and the mixture was uniformly stirred to obtain a 1% by mass emulsifiable concentrate. Formulation Example 2 320202 192 200901876 Compound 2-2, Compound 2-4, Compound 2-8, Compound 2-13, Compound 2-22, Compound 2-27, Compound 2-29, Compound 2-31, Compound 2-35 20 parts of each of compound 2-36, compound 2-40, compound 2-94, compound 2-48 and compound 2-5354, added to 4 parts of sodium lauryl sulfate, 2 parts of lignin sulfate 1 bow, 20 parts of synthetic hydration Oxide fine powder and 54 parts diaraonite. The mixture was uniformly stirred to obtain a 20% wettable powder. Formulation Example 3 1 part of synthetic hydrated cerium oxide fine powder, 2 parts of lignin calcium sulfate, 30 parts of bentonite, and 65 parts of kaolin clay were added to each of 2 parts of compound 2-2, compound 2-4, and compound_2-8. , compound 2-13, compound 2-22, compound 2-27, compound 2-29, compound 2-31, compound 2-35, compound 2-36, compound 2-40, compound 2-94, compound 2-448 And compound 2-5354. A suitable amount of water is added to the mixture. The resulting mixture was further stirred, granulated by a granulator, and air-dried by a circulating dryer to prepare a formulation of 2% granules. Formulation Example 4 Compound 2-2, Compound 2-4, Compound 2-8, Compound 2-13, Compound 2-22, Compound 2-27, Compound 2-29, Compound 2-31, Compound 2-35, Compound 1-36, each of the compound 2-40, the compound 2-94, the compound 2-48, and the compound 2-5354 is dissolved in an appropriate amount of acetone. 5份福basami粘土。 5 parts of hydrated cerium oxide fine powder, 0.3 parts of PAP and 93.7 parts of Fubasami clay. After uniformly mixing the mixture, each formulation of 1% powder was prepared by evaporation to remove the fainting. 193 320202 200901876 Formulation Example 5 /1⁄2 compound 1 2, compound 2-4, compound 2 8 compound 2-13, compound 2-22, compound 2-27, compound 2 to 29, compound 2 -31, compound 2-35, compound 2-36, compound 2~4〇 compound 2-94, compound 2-448 and compound 2-53545, 35 parts of white stone mountain (containing 50 parts of polyoxyethyl ether ether sulfate) Ammonium) and 55 parts of _ scouring by pulverization by wet milling to obtain 1% by flow of each concentrate. Formulation Example 6 Compound 2-2, Compound 2-4, Compound 2-8, Compound 2 to 13, Compound 2-22, Compound 2-27, Compound 2-29, Compound 2-31, Compound 2-35, Compound 2_36, compound 2_4 oxime, compound 2n compound 2-48 and compound 2-5354 each 0.1 part, dissolved in 5 parts of xylene and 5 parts of trichloroethane. The mixture was combined with 89. 9 parts of deodorized kerosene to prepare a 0.1% oily formula. Formulation example 7

10 parts each of compound 2-2, compound 2-4, compound 2-8, compound 2-13, compound 2-22, compound 2-27, compound 2-29, compound 2 31, compound 2-35, compound 2 36. Compound 2-40, compound 2-94, compound 2-448, and compound 2-5354, dissolved in mL. 5 mL of acetone. This solution is added to 5g of animal solid feed powder (Breeding)

Solid Feed Power CE-2, trade name, manufactured by JAPAN CLEA CO., LTD) and uniformly mixed. The acetone is then evaporated to produce a poison bait. Group A: Examples of insecticides include: 194 320202 200901876 (1) Organic broken compound filling Ming, butathiofos, cadusafos, chlorethoxyfos, chlorfenvinphos , chlorpyrifos, chlorpyrifos-methyl, cyanophos (CYAP), diazinon, DCIP (dichlorodiisopropyl ester), deticulate structure (dichlofenthion; ECP), Dichlorvos (DDVP), dimethoate, dimethylvinphos, disulfoton, EPN, ethion, ethoprophos, yiduo Etrimfos, fenthion (MPP), fenitrothion (MEP), fosthiazate, formothion, phosphine, isofenphos, plusfusone Isoxathion), marathion, mesulfenfos, methidathion (DMTP), monoctophos, naled (BRP), oxydeprofos (ESP), para Parathion, phosal One), phosmet (PMP), pirimiphos-methyl, pyridafenthion, quinalphos, phenthoate (PAP), profenofos , propaphos, prednisolone 1*〇1; 1^〇£〇5), pyraclorfos, salithion, sulprofos, tebupirimfos, Temephos, tetrachlorvinphos, terbufos, thiometon, trichlorphon (DEP), vamidothion; 195 320202 200901876 (2) Amino Formate compound, cotton ring (alanycarb), bendiocarb, benfuracarb, BPMC, carbaryl, carbofuran, carbosulfan, line Cloethcarb, ethiofencarb, fenbucarb, fenothiocarb, fenoxycarb, furathiocarb, isoprocarb (MIPC), speed Metalcarb, methodom, methiocarb, NA C, oxamyl, pirimicarb, propoxur; PHC, XMC, thiodicarb, xylylcarb; (3) synthetic pyrethroid compound anagin (acrinathrin), allethrin, benfluthrin, beta-cyfluthrin, bifenthrin, cypermethrin, deltamethrin, Yihuali (esfenvaierate), ethofenprox, cyanidin g (CyCi〇pr〇thrin), cyfluthrin, Cyhai〇thrin, fenpropathrin, Fenicide ( Fenvaierate), flucythrinate, fiufenoprox, flumethrin, fiuvaiinate, halfenprox, imipr〇thrin, baifen Permethrin, prauethrin, pyrethrins, resmethrin, arsenin 196 320202 200901876 (sigma-cypermethrin), silafluofen, safford Tefluthrin, trolomethrin, transf luthrin, (EZ)-(IRS,3RS; IRS, 3SR)-2, 2-Dimercapto-3-prop-1-enylcyclopropanecarboxylic acid 2, 3, 5, 6-tetrafluoro-4-(methoxy Benzoyl) benzyl ester, (EZ)-(IRS, 3RS; 1RS, 3SR)-2, 2-dimethyl-3-propenyl...p-alkenylcyclopropanecarboxylic acid 2, 3, 5, 6-four Fluoro-4-methylbenzyl ester, (IRS, 3RS; 1RS, 3SR)-2,2-dimethyl-3-(2-indolyl-I-propyl)cyclopropanone 2, 3 , 5,6-tetrafluoro-4-(decyloxymethyl)benzoquinone S; (4) Nereisetoxin compound cartap, bensultap, thiocyclam ), monosultap and bisultap; (5) neonicotinoids imidacloprid, nitenpyram, acetamiprid, acesulfan Thiamethoxam), thiacloprid, clothianidin, and dinotefuran; (6) Benzamidine urea compound chlorfluazuron, bistrifluron, rifampin Diafenthiuron, diflubenzuron, fluazuron, flucycloxuron, flufenoxuron, hexafl Umuran), lufenuron, novaluron, noviflumuron, teflubenzuron and triflumuron; 197 320202 200901876 (7) phenyl oxazole compound Acetoprole, fipronil, vaniliprole, pyriprole and pyrafluprole; (8) Bt toxin insecticide derived from Sacillus (Bacillus) Active spores of thuringiensis) and the crystalline toxins produced therefrom, and mixtures thereof; (9) the diaamine compounds chromafenozide, halofenozide, methoxyfenozide, and fenfen (tebufenozide); (1 〇) organochlorine compounds aldrin, dieldrin, dienochlor, endosulfan and methoxychlor; (11) Natural insecticide motor oil and alkali release-sulfate; (12) other insecticides avermectin-B, bromopropylate, buprofezin, chlorphenapyr, Cyromazine, 1,3-dichloropropene, cause Emamectin-benzoate, fenazaquin, flupyrazofos, hydroprene, indoxacarb, metoxadiazone, Mebemycin 198 320202 200901876 A (milbemycin-A), pymetr〇zine, pyridalyl, pyripr〇xyfen, spinosad, flubenzamide ( Sumuramide), tolfenpyrad, triazamate, flubendiamide, SI-〇〇〇9, cyflumet〇fen, arsenic acid, benzene Chlorhexidine (bencl〇thiaz), calcium cyanamide, caicium p〇iySUif ide, chlordane, DDT, DSP, flufenerim, fluniin ( Flonicamide), flurimfen, formetanate, metam-ammonium, metam-sodium, methyl bromide, dinotefuran, potassium oleate , protrifenbute, spiromesifen, lepimectin, sulphur, and metopine (Metaf lumizone), de la give (spirotetramat), NNI-0101, chlorantraniliprole Amides (chlorantrani 1 iprole) and Formula (A) a compound: of formula (A):

Wherein R1 represents a fluorenyl group, a chlorine atom, a bromine atom or a fluorine atom; R2 represents a fluorine atom, a gas atom, a bromine atom, a C!-4 haloalkyl group or a G-4 haloalkoxy group; and R3 represents a fluorine, gas or bromine atom. R4 represents a nitrogen atom, a Cl-4 alkyl group, a C3-4 dilute group, a C3-4 fast group or a C3-5 cycloalkyl group (the Cl-4 alkyl group, the C3-4 base group, the C3-4 fast group and C3-5 199 320202 200901876 A cycloalkyl group may be optionally substituted with one or more groups selected from the group consisting of a halogen atom, a cyano group, a methylthio group, a decylsulfinyl group, a methylsulfonyl group and an anthracene. Alkyl; R5 represents a hydrogen atom or a methyl group; R6 represents a hydrogen, fluorine or chlorine atom; and R7 represents a hydrogen, fluorine or chlorine atom. Examples of acaricides (active ingredients of acaricides) include: acequinocyl, amitraz, benzoximate, bifenazate, bromopropylate ), chinomethionat, chlorobenzilate, PCBS (chlorfenson), clefentezine, cyflumetofen, dicofol, kill Etoxazole, fenbutatin oxide, fenothiocarb, fenpyroximate, fluacrypyrim, fluproxyfen, hexythiazox, sputum Propargite (BPPS), polynactins, pyridaben, pyrimidifen, tebufenpyrad, tetradifon, spirodiclofen , amidoflumet, cyenopyrafen, and the like. As a nematicide (active ingredient of nematicidal agents): DCIP, fosthiazate, levamisol, mercapto isothiocyanate, morantel tartarate, emisene Fu (imicyafos) and so on. As a fungicide: 200 320202 200901876 Acibenzolar-S-methyl, amobam, ampropyf los, ani lazine, azoxystrobin , benalaxyl, benodanil, benomyl, benthiavalicarb, bethithiazole, bethoxazin, bitertanol , blasticidine-S, Bordeaux mixture, boscalid, bromuconazole, cesium bate, (buthiobate), calcium hydrochlorite, Calcium polysulfide, captain, carbendazol, carboxin, carpropamid, chlobenthiazone, diclofenac Chloronib), chloropicrin, chlorothalonil (TPN), chlorthiophos, cinnamaldehyde, clozylacon, CNA (2,6-dichloro -4-nitroaniline), copper hydroxide, copper sulfate, racemodium (cya Zofamid), cyflufenamid, cymoxanil, cyproconazole, cyprodinil, cyprofuram, dazome, debacarb ), dichlof luanid, DD (l,3-dichloropropene), diclocymet, diclomezine, diethofencarb, difenoconazole, two Diflumetorim, dimefluazole, dimethirimol, dimethomorph, Dakli 201 320202 200901876 (diniconazole-M), dinocap, edfen (edifenphos), ep〇xic〇naz〇ie, nickel dithiocarbamate, etaconazole, ethaboxam, ethirimol, edi Etridiazole, famoxadone, fenamid〇ne, fenarimol, fenbuconaz〇ie, fendazosulam, cycloheximide Fenhexamid), fenoxanil, seed dressing (fenpici〇njj), fenprop (fenprop Idin), fenpr〇pimorph, fentiazon, fentinhydroxide, ierimzone, fiuazinam, fludioxonil , flumetover, flumorph, fiuor〇imide, fluotrimazole, fluorosis vinegar (fiu〇xastrobin), fluquinconazole, 护Flusilazole, flusulfamide, flutolanil, flutriafol, fosetyl-Al, fthalide, fuberidazole ,furalaxyl, furametpyr, difurfurylamine (|611〇&1^&1111), biting 嗤(|111*〇011&2〇16-(^3 ), hexaconazole, hymexazol, IBP, imazalil, imibenconazole, gram-net-trioctyl benzoate (iminoctadine- Albesilate), ichotox-triacetate, iodocarb, ioconcarb, 202 320202 200901876 ipconazole, Iprodione, iprovalicarb, isoprothiolane, kasugamycin, kresoxim-methyl, mancozeb, manganese nucleus (maneb), mepanipyrim, mepronil, metalaxyl, metalaxyl-M, methadine, methasulfocarb, methyl desert, Metaconazole, methfuroxam, metominostrobin, phenoxylinone (1^廿8 [611〇]16), bactericidal amine (metsuflovax), and mildiomycin ), mi lneb, myclobutani 1, myclozolin, nabam, orysastrobin, ofurace, beta cream Oxadixyl, oxo 1 inic acid, opcon. Oxpoconazole, oxycarboxin, oxytetracycline, 'pefurazoate, penconazole, pencycuron, picoxystrobin, dysen Polycarbamate, polyoxin, potassium bicarbonate, probenazole, prochloraz, procymidone, propamocarb-hydrochloride, pk (propiconazolej, propineb, proquinazid, prothiocarb, prothioconazole, quintozene; PCNB) Si lthiopham, simeconazole, sipconazole, sodium bicarbonate, sodium hypochlorite, fusarium 203 320202 200901876 (spiroxamine), SSF-129, ( (E)-2-[2-(2,5-dimethylphenoxyindolyl)phenyl]-2-methoxyimino-N-mercaptoacetamide>, streptomycin, Sulfur, tebuconazole, teci〇ftaiam, tetraconazole, thiabe Ndazole), thiadinil, thiram (TMTD), thifluzamide, thiophanate-methyl, tolclofos-methyl, TPN, three Triadimefon, triadimenol, triazoxide, triclamide, tricyclazole, tridemorph, triflumizole, trifluoro-sensitive (trifloxystrobin), triforine, triticonazole, validamycin, vinclozolin, viniconazole, zineb, thiram ( Ziram), zoxamide, amisubrom, enestroburin, mandipropamid, meptyldinocap, and the like. As a herbicide, phytohormone and plant growth regulator: abscisic acid, acetochlor, acifluorfen-sodium, alachlor, alloxydim , ametryn, amicarbazone, amidosulfuron, amino ethoxy vinyl alanine, aminopyralid, AC94, 377, methylamine Amiprophos-methyl, ancymid〇l, asulam, atrazine, aviglycine, tetrazincsulfuron 204 320202 200901876 (azimsulfuron), fluoride Beflubutamid, benfluralin, benfuresate, bensulfuron-methyl, bensilide (SAP), bentazone, benthiocarb ), benzamizole, benzfendizone, benzobicyclon, benzofenap, benzyl adenine, benzoguanamine guanidine, dipropylamine (bialaphos), bifenox, brassinolide ( Brassinolide), bromacil, bromobutide, butachlor, butafenacil, butamifos, butarate, oxazinamide (cafenstrole), calcium carbonate, calcium peroxide, carbaryl, chlomethoxynil, chloridazon, chlorimuron-ethyl, chlorphthalim, Chlorpropham., chlorsulfuron, chlorthal-dimethyl, chlorthiamid (DCBN), choline chloride, cinidon-ethyl, cycloheptin Cinmethylin, cinosulfuron, cleavage • clethodim, ci〇mepr〇p, ci〇Xyfonac-sodium, chionuequat chloride ), 4-CPA (4-chlorophenoxyacetic acid), cloprop, clofencet, cumyluron, Cyanazine, cyclanilide , Cycsulfuron (CyCi〇suifamuron), cyhalofop-butyl, 2, 4-dichlorophenoxyacetic acid Class, 2, 4-Dippropionic acid (dichlorprop; 2,4-DP), daimuron, dalapon 205 320202 200901876 (dalapon; DPA), dimethenamid-P, Daminozide, dazomet, n-decyl alcohol, dicamba-sodium (MDBA), dichlorobenzil (DBN), diflufenican, and pericin ( Dikegulac), dimepiperate, dimethametryn, dimethenamid, diquat, dithiopyr, diuron, Neisseria Endothal, epocholeone, esprocarb, ethephon, ethidimuron, ethoxysulfuron, sulphuric acid Ethychlozate), etobenzanid, fenarimol, fenoxaprop-ethyl, fentrazamide, flazasulfuron, double Florasulam, fluazifop-butyl, fluazolate, fluoroketone huanglong (f lucarbazone), flufenacet, flufenpyr, flumetralin, fluroxazine ' ^ 13⁄4 ^.#9 (f lupropanate-sodium) &gt ; 0 flurinrsulfuron-methy1-sodium, σ 啸 传 (f lurprimidol), flu omethoate (f luthiacet-methyl), foramisulfuron, forfufenuron (forchlorfenuron) ), fluorescein (formesafen), gibberellin, glufosinate, glyphosate, halosulfuron-methyl, hexazinone, alfalfa Oxygen 11 m grass smoke (imazamox), yoghurt imazapic, imazapyr, 206 320202 200901876 imazaquin, imazosuifuron, inabenfide, Indoleacetic acid (IAA), indolebutyric acid, iodosulfuron, benzoic acid vinegar (i〇Xynii-octanoate), isouron, isoxachlor (isoxachl〇rt〇le) ), isoxadifen, karbutilate, lactofen, cyclohexane (lenacil), liguron (linuron), LGC-42153, maleic hydrazide, tetrachloropropionic acid (mec〇prop; MCPP), 2-methyl-4-chlorophenoxyacetate MCPA-thioethyl, 2-mercapto-4-chlorophenoxybutyrate ethyl acetate, mefenacet, mefluidide, mepiquat, Mesosulfuron, mesotrione, methyl-daimuron, metolachlor, chlorfenapyr (age 1:1 '11211^), continued Long (1116士3111『111'011-11161±71), rice, magnesium, naphthylacetate, 1-naphthylamine, naproanilide, napropamide, n-decyl alcohol , nicosulfuron, n-phenyl glutamate, orbencarb, oxadiazon, oxaziclomefone, oxine-sulfate, Multi-effect ^ (paclobutrazol), paraquat, pelargonic acid, pendimethalin, penoxsulam, pentoxazone, acetochlor (pethox) Amid), phenmedipham, picloram, picolinafen, piperonyl butoxide, piperophos, pretilachlor, fluoride Continuation 207 320202 200901876 (primisulfuron-methyl), procarbazone, prodiamine, profluazol, profoxydim, cyclamate salt Prohexadione-calcium), prohydrojasmon, prometryn, propanil, propoxycarbazone, propyzamide, pyraflufen-ethyl ), pyrazolate, pyrazoosulfuron-ethyl, py.razoxyfen, pyribenzoxim, pyributicarb, pyridafol, up to Pyridate, pyrifalid, pyriminobac-methyl, pyrithiobac, quinclorac, quinoclamine, ethylquine Quizalofop-ethyl, rimsulfuron ), sethoxydim, siduron, simazine, simetryn, sodium chlorate, sulfosulfuron, SWEP (MCC), Tebuthiuron, tepraloxydim, terbacil, terbucarb (MBMPC), thenylchlor, 0 thiazafluron, sputum Thidiazuron, thifensulfuron-methyl, triaziflam, tribufos, triclopyr, tridiphane, trifluoro Trifloxysulfuron, trifluralin, trinexapac-ethyl, tritosulfuron, uniconazole-P, and velocate (PPTC) . 208 320202 200901876 As a synergist: piperonine scales, sesamex, sulfoxides, N-(2-ethylhexyl)-8, 9, 10-triazole borneol-5-ene-2, 3-dicarboxylimine imine (MGK 264), anti-WARF resistant strain and diethyl maleate. As a safener: benoxacor, cloquintocet-mexyl, cyometrinil, daimuron, dichlormid, fenchlorazole-ethyl ), fenclorim, flurazole, fluxofenim, furilazole, mepyrazin®, MG191, liver And oxabetrinil. Formulation Example 8 10 parts of the compound 2-2 and 1 part are listed in the above group a insecticide, acaricide, nematicide, fungicide, herbicide, plant hormone agent, plant growth regulator, synergist Or a safener, added to 4 parts of lauryl sulfonate, 2 lignin% acid 26'20 parts of synthetic hydrated oxidized _ fine powder and 54 diatomaceous earth mixture. The mixture is uniformly stirred and mixed to obtain von Hezhi Wettable powder. Formulation Example 9 10 parts of compound 2-13 and 1G parts are listed in the above group A, killing insecticide, nematicide, killing _, herbicide, phytohormone, = growth regulator a synergist or a safener, added to 4 parts of a lauryl pot = 2 parts of woody material, 2 2 parts of a mixture of synthetic hydrated oxygen-cut fine powder and earthworm soil. The resulting mixture is uniformly transferred and mixed to obtain 320202 209 200901876 Mixed wettable powder. Formulation Example 1 10 10 parts of compound 2-29 and 10 parts of the above-mentioned group A insecticide, sputum, nematicide, fungicide, herbicide, phytohormone, Plant growth regulator, synergist or safener, added A mixture of 4 parts of sodium lauryl sulfonate, 2 parts of calcium lignin sulfonate, 20 parts of synthetic hydrated cerium oxide fine powder and 54 parts of diatomaceous earth. The resulting mixture was uniformly stirred and mixed to obtain a mixed wettable powder. Formulation Example 11 10 parts of the compound 2-40 and 10 parts listed in the above group A insecticide, sputum, nematicide, fungicide, herbicide, phytohormone, plant growth regulator, synergist or a safener, added to 4 parts of sodium lauryl sulfonate, 2 parts of calcium lignin sulfonate, 20 parts of a synthetic hydrated cerium oxide fine powder and 54 parts of a mixture of diatomaceous earth. The resulting mixture is uniformly stirred and mixed to obtain a Mixed wettable powder. Formulation Example 12 10 parts of the compound 2-5354 and 10 parts of the above-mentioned group A insecticide, acaricide, nematicide, fungicide, herbicide, phytohormone, plant A growth regulator, synergist or safener is added to a mixture of 4 parts of sodium sulphate, 2 parts of lignin citrate #5, 20 parts of synthetic hydrated oxidized dream powder and 54 parts of diatomaceous earth. Mix and mix to make a mixture Wettable powder. Formulation Example 13 10 parts of the compound 2-22 and 10 parts of the insecticide of the above group A 210 320202 200901876 agent, acaricide 'nematicidal agent, fungicide, herbicide plant growth adjustment sword, Synergist or safener, add ^, phytohormone, sodium sulphate, 2 parts of lignin, 2G parts, 4 parts of laurel base, 54 parts of the present compound. The mixture obtained is evenly = chopped powder and Mixed moisturizable powder. Formulation prepared by sputum and abusiveness Example 14 10 parts of compound 2-36 and 1 part are listed as topping agent, acaricide, nematicide, fungicide, weeding '2 killing Insect plant growth regulator, synergist or safener, add u-agent 'sodium sulphate, 2 parts of lignin, 2 〇 合成 知 月 月 续 54 54 54 54 54 54 54 54 54 54 54 54 54 54 54 54 54 54 54 54 54 54 54 、 、 、 Powder and X of the injured soil. The resulting mixture was uniformly stirred and kneaded to wet the powder. The following test examples will demonstrate that the present invention is effective for the control of pests. In Test Examples 丨8, the mixture was pulverized by wet grinding by mixing 1 G of the compound (1), milk = carbon (containing 50 parts of polyoxyethylene ethyl __), and 55 parts of water. The resulting formulation was diluted to give an active ingredient concentration of 5 GGPPm. The resulting solution was used as a test solution. Test Example 1 (Spodoptera litura) Place a filter paper of the same size at the bottom of a 5.5 cm diameter polyethylene cup. Insecta LF (NIH0N NOSAN K0YG0 C0.) slice is 6 mm thick and further cut in half and placed on it' And 2 mL of the above test solution was poured. After air drying, five fourth instar Spodoptera litura larvae were released and the cup was sealed. 6 Calculate the number of dead larvae after sputum. Mortality is calculated by the following formula: 320202 211 200901876 Mortality (%) = (number of dead larvae / number of test larvae) χ 100 and assessed by the following indices: 4: 100%, 3: 80-90%, 2: 60 -79%: 1 : 30-59% and 0: 0-29% (mortality). Compound 2-2, Compound 2-4, Compound 2-8, Compound 2-22_, Compound 2-29, Compound 2-31, Compound 2-35, Compound 2-36, Compound 2-40, Compound 2-448, Any of Compound 2-894, Compound 2-5354, and Compound 2-6023 was evaluated as an index of 3 or more. Test Example 2 (Adoxophyes orana) A filter paper of the same size was placed on the bottom of a polyethylene cup having a diameter of 5.5 cm. Silkmate S (NIH0N NOSAN KOYGO C0.) was sectioned 2 mm thick and placed thereon, and 1 mL of the above test solution was poured. After air drying, a 5. 5 cm diameter filter paper was placed thereon, and 30 four-instar Spodoptera litura larvae were released, and the cup was sealed. The number of dead larvae was counted after 7 days. _ Mortality is calculated by the following formula: Mortality (%) = (number of dead larvae / number of test larvae) χ 100 and assessed by the following indices: 4: 100%, 3: 80-90%, 2: 60-79 %: 1 : 30-59% and 0: 0-2S% (mortality). Compound 2-2, Compound 2-4, Compound 2-8, Compound 2-13, Compound 2-22, Compound 2-27, Compound 2-29, Compound 2-31, Compound 2-35, Compound 2-36, Any of Compound 2-40, Compound 2-94, Compound 2-48, Compound 2-894, Compound 2-5354, and Compound 2_6023 was evaluated to have an index of 3 or more. 212 320202 200901876 Test Example 3 (Aphis gossypii) Release 30 one-year-old cotton aphid larvae on leaves of a leaf cucumber planted in an ounce cup. The next test solution was sprayed 20 (mL) the next day. The number of survivors was calculated after 6 weeks. The survival rate relative to the untreated cup was calculated by the following formula: Survival rate (%) = (number of surviving larvae / number of test larvae) χ 100 and evaluated by the following index: 4: 0%, 3: Bu 10%, 2 : 11-40% : 1 : 4 Bu 70% and 0 : > 70% (survival rate). . Compound 2-2, Compound 2-4, Compound 2-8, Compound 2-22, Compound 2-31, Compound 2-35, Compound 2-894, Compound 2-5354, and Compound 2-6023 The assessment is index 3 or greater. Test Example 4 (Nilaparvata lugens) Rice was cultivated in a 90 mL plastic cup, and 5 cm or more of two- or three-leaf rice was cut from the top of the root. 20 mL of the above test solution was sprayed per pot. After air drying, 30 larvae of the first to second instar larvae were released. Seal the cup. The number of surviving larvae was calculated after 6 days. The survival rate relative to the untreated cup was calculated by the following formula: Survival rate (%) = (number of surviving larvae / number of test larvae) χ 100 and evaluated by the following index: 4 : 0%, 3 : 1-10% 2: 11-40% : 1 : 41-70% and 0 : > 70% (survival rate). Compound 2-2, Compound 2-13, Compound 2-22, Compound 2-29, Compound 2-31, Compound 2-35, Compound 2-448, Compound 2-894, 213 320202 200901876 North Compound 2-5354 and Either of the compounds 2-6023 was evaluated as an index of 3 or more. Delta test case 5 (Musca domestica) Place the same size filter paper on the bottom of a 5.5 cm polyethylene cup. The above test solution (0.7 mL) was added dropwise to the filter paper, and 30 mg of the sugar was uniformly placed as _. Release the iq only female adult. The cup is sealed. The number of dead adults was counted after 24 hours. Mortality is calculated by the following formula: Mortality (%) = (number of dead adults / number of tested adults) xl〇〇 and evaluated by the following indices: 4: 100%, 3: 70-99%, 2: 40 -69%: 1 : 10-39% and 〇: 0-9% (mortality). Compound 2-2 was evaluated as an index of 3 or more. Test Example 6 (Blattella gernranica) A filter paper of the same size was placed on the bottom of a polyethylene cup having a diameter of 5.5 cm. The above test solution (〇.7 mL) was added dropwise to the filter paper, and 30 mg of granulated sugar was uniformly placed as a bait. Release 2 German cockroaches adults. The cup is sealed. After 6曰, the number of dead adults was counted. Mortality is calculated by the following formula: Mortality (%) = (number of dead adults / number of tested adults) xl〇〇 and assessed by the following indices: 4: 100%, 2: 50% and 〇: 〇% (death rate). Compound 2-2 was evaluated as index 4. Test Example 7 (Cul ex pi pi ens pal lens) 214 320202 200901876 The above test solution (0.7 mL) was added to 100 mL of ion-exchanged water (concentration of active ingredient: 3.5_). In this solution, 20 larvae of the light color in the later age were released, and the mortality was calculated after the next day by the following correction: mortality (%) = (number of dead larvae / number of test larvae) xl Measures. Evaluated by the following indices: 4: 9 Bu 1_, 2: 1 Bu and Q: (Death rate). Compound 2-2, Compound 2-4, Compound 2-8, Compound 2-22, Compound 2-27, Compound 2-29, Compound 2_31, Compound 2_35, Taxoline 2-40, and Compound 2-894 were evaluated as Index 4. Test Example 8 (piuteiia xylostella) 3 〇 mg of the compound was dissolved in a mixture of mL.〇75 mL of dioxan and N,N-dimethylformamide CDMF) (mixing volume ratio of xylene: N , N- " dimethylformamide = 1: 1:). Add 〇. 〇 4 mL of xylene and s〇rp〇1 3005X (trademark, manufactured by TOHOCHEMICAL INDUSTRY CO., LTD. (mixed volume ratio is So卬〇1 3005X4: 9). The mixture is diluted with ion-exchanged water. Prepare a test solution (5 〇〇ppm) of the test compound. Spray 20 mL of the test solution in the four-leaf stage of Bmssica oleracea. After the test solution is dried, the ground part is cut and 5 second-instar Plutella xylostella Larvae were placed together in a polyethylene cup (1 〇〇mL volume). The cup was stored at 25 ° C. The number of dead larvae was calculated after 5 。. Mortality was calculated by the following formula: Mortality (%) - (number of dead larvae / The number of test larvae was χ1〇〇 and evaluated by the following index: 320202 215 200901876 4 : 100%, 3: 80-99%, 2: 60-79%, 1: 30-59% and 0: 0-29% (mortality) Compound 2-2, Compound 2-4, Compound 2-8, Compound 2-13, Compound 2-22, Compound 2-27, Compound 2-29, Compound 2-31, Compound 2-35, Compound 2 -36, compound 2-40, compound 2-94, compound 2-448, compound 2-894, compound 2-5354, and compound 2-602 3Evaluated as index 3 or greater. Test Example 9 (Bemisia tabaci) 40 mg of compound (I) was dissolved in hydrazine. imL organic solvent (diphenylbenzene: N,N-dimethylformamide =1 : 1) and 〇.〇 4 mL of xylene and Sorpol 3005X (trademark, manufactured by TOHO CHEMICAL INDUSTRY Co., Ltd. (mixed volume ratio is Sorpol 3005X = 1: 9). The mixture was diluted with 80 mL of ion-exchanged water. 5 〇〇ppm compound solution. 30 mL of this solution was diluted with 45 mL of ion-exchanged water to prepare a 20Qppm compound solution. 20 mL of this 200 ppm compound solution was diluted with 6 〇mL of ion-exchanged water to prepare a 50 ppm compound solution, and 20 mL of this 50 ppm compound solution was further 60 mL. The ion exchange water was diluted to prepare an i2.5 ppm compound solution. Dine (registered trademark, manufactured by TAKEDA PHARMACEUTICAL CO., LTD.) was added to each compound solution to dilute Dine by 3,000 times to prepare a test solution. Cymbidum kanran was used. Incubate for 3 weeks in 3 oz cups. Remove all leaves except the second true leaves. Release the whitefly of the whitefly and let it lay eggs for 3 days. Remove the adult worm and keep the cup in warm 8 to the culture plate. 20mL above test spray solution, and within 7 days of each survey Cup mortality. 216 320202 200901876 Based on the 5 rating of the index below, the effect is evaluated. Index 4: 100% mortality 'index 3: 90-99% mortality (larvae attachment area is 1 to 10% of untreated group) ' 2 : 60-89% mortality (larvae attachment area is untreated group 11 Up to 40%), index 1: 30-59% mortality (41 to 70% of the larvae area is untreated) and 0: 0-29% death rate (the larval attachment area is 71% of the untreated group) Or more). In the case of 12.5 ppm, the compound 2-2, the compound 2-4, the compound 2-31, the compound 2-894, the compound 2-5354, and the compound 2-6023 were evaluated to have an index of 3 or more. Test Example 10 (Haemaphysalis l〇ngicornis) Compound (1) (0.5 mg) was dissolved in imL acetone, and uniformly applied to one side of a filter paper (TOYO No. 2; 5 x 1 Ocm). After drying, the filter paper was folded in half and the two sides were clamped to make a pouch. The test sputum (long-horned blood sputum, not blood-sucking scorpion scorpion, 10 groups) was placed therein. The opening of the pouch is clamped and sealed. The fatal ratio was observed after sputum. 'Compound 2-2 and Compound 2-29 show a mortality rate of 90% or more. As described herein, the compound (1) has an excellent control effect against pests, and has an active ingredient for use as a pest control preparation. [Simple description of the diagram] None [Key component symbol description] None 320202 217

Claims (1)

200901876 VII. Scope of Application: 1. A thioimine vinegar compound is represented by formula (I): ("W rR S-CH=CH-C=N- (I) wherein R represents Cm bicycloalkyl or substituted by c6-12 bicycloalkyl.: alkyl; m represents an integer from 〇 to 2; η represents 0 An integer up to 2;) i represents a halogen atom, a G-3 alkyl group, a Cw haloalkyl group, a C!-4 alkoxy group or a nitro group, and when m is 2, the two Xs are the same or different; and z Represents a halogen atom, a Cm alkyl group, a Cm haloalkyl group or a g-4 alkoxy group, and when η is 2, the two oximes are the same or different. 2' is a thioimidate compound according to claim 1, wherein R in the formula (I) represents a bicycloalkyl group. 4. The thioimidate compound of the first aspect of the invention, wherein R in the formula (1) represents a bicyclo [4. 4.0] fluorenyl group. A pest control preparation comprising the compound of any one of claims 1 to 3 as an active ingredient. A use of a compound of any one of claims 1 to 3 is for controlling pests. The use of the compound of any one of items 1 to 3 of the patent application of the Japanese patent: , = for the preparation of a pest control preparation. The method for controlling thieves' includes the application of a compound of the first patent range from the first patent to the pests or pest habitats in the range of 1 $ q β + y to 3 . 218 320202 200901876 IV. Designated representative map: There is no schema in this case (1) The representative representative figure of this case is: ( ). (2) A brief description of the symbol of the representative figure: 5. If there is a chemical formula in this case, please disclose the chemical formula that best shows the characteristics of the invention: ^(Z)n (I) 320202