TW200529745A

TW200529745A - Plant protection compositions and use thereof

Info

Publication number: TW200529745A
Application number: TW94103448A
Authority: TW
Inventors: Taranta Claude Buckpesc Rainer
Original assignee: Bayer Cropscience Gmbh
Priority date: 2004-02-06
Filing date: 2005-02-03
Publication date: 2005-09-16
Also published as: WO2005074685A1; KR20060133594A; KR101196233B1; CN1929735B; WO2005074685A8; CN1929735A; JP2007520511A

Description

200529745 (1) 九、發明說明【發明所屬之技術領域】本發明係關於一種包含乳酸2 -乙基己酯（EHL )的植物之保護組成物之應用及及一種含有EHL之特殊的植物 . 保護組成物。【先前技術】 > 對於水稻作物而言，爲了達到令人滿意的病蟲害控制必需讓稻米植株及/或出現在水中的害蟲以直接且適時的方式與所施加的活性物質相接觸，或者必需把活性物質均勻且充份地分散在整個水稻田中。例如，在標準應用過程中係使用習知噴灑液或顆粒但如此卻十分昂貴。把處理過程中如揭露於J P - A - 1 0 1 7 5 8 0 4之置於水溶性容器如瓶中之活性物質，或者揭露於U S - 5 4 3 9 6 8 3號置於袋中之活性物質置於稻田周圍的方法則較爲經濟。在活性物質從容器 | 中釋出以後，該等活性物質在水面上的均勻散佈則與多種 • 因素有關且可藉由加入適當的添加劑來加以改善或甚至予以保證。可以使用的特殊組成物有例如揭示於JP-A-1 00 1 74 1 0之弱水溶性活性物質或者如揭示於】卩_厂 05 3 3 9 1 03、直接溶於質子惰性溶劑如酞酸（c8_Cl3 )·院基酯之非水溶性活性物質。在w 0 · A - 0 1 / 3 5 7 3 8號中，將植物油加到活性物質中，且油中的活性物質含量可藉著再加入質子惰性溶劑來進一步地提高。然後可以經由油膜的形成而促使活性成份均勻地散佈在水稻田裡。然而，油膜同樣 -4 - 200529745 (2) 地也會阻礙空氣及水之間氧氣的交換且額外地引入特定的溶解促進劑則可能會對生態有不良的影響。此外，人們還需要一種新穎的方法，其可以更容易地在水稻田中施用，效果更可靠且其操作對使用者而言更爲安全。 ¥ 【發明內容】本發明之目的係在發展一種使用方法，其可用來控制 φ 水稻作物的病蟲害同時儘可能地避免前述之經濟及生態上的問題。令人訝異地，本發明現在發現到透過將農業化學之活性物質溶於EHL中可獲得一種植物之保護組成物，其特別適合用於水稻作物之病蟲害防治上。本發明的植物之保護組成物及其應用對於使用者而言既簡單又安全，在考慮活性物質之毒性時其顯示極有利的特性且對於水稻田之病蟲害防治亦顯出可靠的效果。此外 φ ，由於EHL可經由生物徹底地分解成二氧化碳及水所以 “ 對於環境的影響也有所改善。一開始本發明之組成物會形 . 成溶劑膜，此時可促進活性物質在水稻田中均勻地散佈開來，不過接下來該膜會被分解成數千個微小的液滴，如此便不會因爲水面完全被膜覆蓋住而阻礙空氣和水之間氧氣的交換了。 WO-A-91/ 1 4 366中揭露EHL爲一種可調節葡萄生長之活性物質。在此，EHL係以固定劑量且未添加額外添加劑地直接釋入水中並在葡萄生長早期製成葉片噴灑液來使用 -5- (3) (3)200529745 在WO-A-OO/ 1 8227中描述EHL可用來作爲使不溶性農業化學之活性物質懸浮於非水性濃縮懸浮液之懸浮劑。在WO-A-03 /07 6 5 7中揭示EHL爲一種防止殺蟲劑組成物結晶之化學劑，特別是可防止含有吡咯之殺真菌組成物在施用期間結晶。在此等文獻中無一者曾建議可將含有EHL的植物之保護組成物用在稻米作物上以獲得特別的效用。所以，於本發明一態樣中係在提供一種使用如下之植物保護組成物來控制稻米作物之病蟲害之應用，其中該保護組成物包含： (a)乳酸2-乙基己酯， (b ) —或多種可溶於該組成物之農業化學之活性物質，及 (c )任意地一或多種配方助劑。本發明之再一態樣係在提供一種控制水稻作物病蟲害之方法，其中係將一種如下之植物之保護組成物施用在水田的水中或水面上，其中該保護組成物包含： (a)乳酸2-乙基己酯， (b ) —或多種可溶於該組成物之農業化學之活性物質，及 (c )任意地一或多種配方助劑。於本發明之意義中，”植物保護組成物”係指農業化學之活性物質之調合物，即，其可爲一種含有EHL及一或 200529745200529745 (1) IX. Description of the invention [Technical field to which the invention belongs] The present invention relates to the application of a plant protective composition containing 2-ethylhexyl lactate (EHL) and a special plant containing EHL. Protection组合物。 Composition. [Prior art] > For rice crops, in order to achieve satisfactory pest and disease control, rice plants and / or pests appearing in water must be brought into direct and timely contact with the applied active substance, or The active substance is evenly and well dispersed throughout the rice field. For example, the use of conventional sprays or granules in standard applications is expensive. Dispose of the active substance in a water-soluble container, such as a bottle, as disclosed in JP-A-1 0 1 7 5 8 0 4 during processing, or in US-5 4 3 9 6 8 No. 3 in a bag The method of placing the active substance around the rice field is more economical. After the active substance is released from the container | the uniform distribution of the active substance on the water surface is related to a number of factors and can be improved or even guaranteed by the addition of appropriate additives. The special composition that can be used is, for example, a weakly water-soluble active substance disclosed in JP-A-1 00 1 74 1 0 or as disclosed in 卩卩 plant 05 3 3 9 1 03, directly soluble in aprotic solvents such as phthalic acid (C8_Cl3) · Insoluble active substance of nosyl ester. In w 0 · A-0 1/3 5 7 3 8, vegetable oil is added to the active material, and the content of the active material in the oil can be further increased by adding an aprotic solvent. The formation of an oil film can then be used to encourage the active ingredients to be evenly distributed throughout the rice field. However, the oil film also -4-200529745 (2) The ground will also hinder the exchange of oxygen between air and water and the introduction of specific dissolution promoters may have adverse ecological effects. In addition, there is a need for a novel method that can be applied more easily in rice fields, the effect is more reliable, and its operation is safer for the user. [Summary of the Invention] The purpose of the present invention is to develop a method of use that can be used to control the pests and diseases of the φ rice crop while avoiding the aforementioned economic and ecological problems as much as possible. Surprisingly, the present invention has now found that a plant protective composition can be obtained by dissolving an active substance of agrochemicals in EHL, which is particularly suitable for controlling pests and diseases of rice crops. The plant protective composition and application thereof of the present invention are simple and safe for the user, show extremely advantageous characteristics when considering the toxicity of the active substance, and show a reliable effect on the control of diseases and insect pests in rice fields. In addition, φ, because EHL can be completely decomposed into carbon dioxide and water through biology, "the impact on the environment is also improved. At first, the composition of the present invention will form. A solvent film is formed, and at this time, the active substance can be promoted uniformly in the rice field It spreads, but the membrane will be broken down into thousands of tiny droplets, so that the water surface is completely covered by the membrane, which will not hinder the exchange of oxygen between air and water. WO-A-91 / 1 4 366 revealed that EHL is an active substance that can regulate the growth of grapes. Here, EHL is directly released into the water at a fixed dose without additional additives and made into a leaf spray in the early stages of grape growth to use -5- (3 (3) 200529745 described in WO-A-OO / 1 8227 EHL can be used as a suspending agent for suspending insoluble agrochemical active substances in non-aqueous concentrated suspensions. In WO-A-03 / 07 6 5 7 It was revealed that EHL is a chemical agent for preventing the crystallization of insecticide compositions, and in particular, it can prevent the fungicidal composition containing pyrrole from crystallizing during application. None of these documents has suggested that EHL-containing plants can be The protective composition is used on rice crops to obtain a special effect. Therefore, in one aspect of the present invention, an application is provided for controlling pests and diseases of rice crops using the following plant protection composition, wherein the protective composition comprises: (a) 2-ethylhexyl lactate, (b)-or agrochemical active substances soluble in the composition, and (c) any one or more formulating aids. Another aspect of the present invention The invention provides a method for controlling pests and diseases of rice crops, wherein a protective composition of a plant is applied to water or water on a paddy field, wherein the protective composition comprises: (a) 2-ethylhexyl lactate, ( b)-one or more agrochemically active substances that are soluble in the composition, and (c) any one or more formulating aids. In the sense of the present invention, "plant protection composition" means the activity of agrochemicals A blend of substances, that is, it can be a substance containing EHL and one or 200529745

多種農業化學之活性物質之活性物質濃縮液，或爲此等活性物質濃縮液與配方助劑之調合物。此等任意使用之配方助劑可爲調合技術中習知的添加劑及助劑，其爲多數不同劑型典型使用的成份，例如：乳化劑（例如可用在可乳化濃縮液（EC )及微乳液（ME )之劑型）、濕化劑如可用在即用型液體調合物（AL )之劑型）、惰性物質（例如可用在顆粒（GR )及可乳化顆粒（EG )之劑型）、分散劑 (例如可用在水包油乳液（EW )及懸浮乳液（SE )之劑型）及界面活性劑（例如可用在溶解性濃縮液（S L )之劑型），也可加入額外的溶劑、增稠劑、流動安定劑、佐劑、活性物質安定劑、保存劑、消泡劑、成膜劑及抗凍劑，且此等物質可用在多數不同的劑型中。可能需要的配方助劑如乳化劑、濕化劑、惰性物質、分散劑、界面活性劑、溶劑及額外的添加劑爲熟悉此技術者所習知，且係述於例如：Watkins，“ Handbook of Insecticide Dust Diluents and Carriers 55 5 2nd Ed.? Darland Books, Caldwell, N.J. ； H. v. Olphen, u Introduction to Clay Colloid Chemistry9% 2nd Ed.? J. Wiley & Sons, N.Y.； C. Marsden，“Solvents Guide”，2nd Ed·，Interscience，N.Y.， 1 9 6 3 ; McCutcheon's “Emulsifiers and Detergents-Concentrates of active substances for various agricultural chemistry active substances, or blends of such active substance concentrates and formulation auxiliaries. These optional additives can be conventional additives and additives in blending technology, which are typical ingredients used in most different dosage forms, such as: emulsifiers (such as can be used in emulsifiable concentrates (EC) and microemulsions ( ME)), wetting agents such as ready-to-use liquid formulations (AL), inert substances (such as granules (GR) and emulsifiable granules (EG)), dispersants (such as available In oil-in-water emulsion (EW) and suspension emulsion (SE) formulations and surfactants (such as formulations that can be used in soluble concentrates (SL)), additional solvents, thickeners, flow stabilizers can also be added , Adjuvants, active substance stabilizers, preservatives, defoamers, film formers and antifreezes, and these substances can be used in most different dosage forms. Formulation aids that may be required such as emulsifiers, wetting agents, inert substances, dispersants, surfactants, solvents, and additional additives are familiar to those skilled in the art and are described in, for example, Watkins, "Handbook of Insecticide Dust Diluents and Carriers 55 5 2nd Ed.? Darland Books, Caldwell, NJ; H. v. Olphen, u Introduction to Clay Colloid Chemistry 9% 2nd Ed.? J. Wiley & Sons, NY; C. Marsden, "Solvents Guide ", 2nd Ed ·, Interscience, NY, 1 9 6 3; McCutcheon's" Emulsifiers and Detergents-

International Ed.”，Annual, M C P u b 1. Corp., Ridgewood, N.Y. ; McCutcheon 丨 s “Emulsifiers and Detergents-North America Ed.”，Annual, MC Pub]· corp.，Ridgewood，N.Y.;International Ed. ", Annual, MC P u b 1. Corp., Ridgewood, N.Y .; McCutcheon 丨 s" Emulsifiers and Detergents-North America Ed. ", Annual, MC Pub] · corp., Ridgewood, N.Y .;

Sisley and Wood,Sisley and Wood,

Encyclopedia of Surface Active (5) 200529745Encyclopedia of Surface Active (5) 200529745

Agents’’，C h e m . P u b 1. Co. Inc.? N.Y., 1964 ； Schonfeldt, “Grenzflachenaktive Athylenoxidaddukte’’[Surface-Active ethylene oxide adducts], W i s s . V erlagsgesell. 9 Stuttgart, 1 9 7 6 ; Winnacker-Ktichler, “Chemische Technologie” [Chemical Technology]， Volume 7， C. Hanser Verlag， Munich， 4 th edition, 1 9 8 6 ； Μ o 11 e t and Grubenmann，Agents '', C hem. Pub 1. Co. Inc.? NY, 1964; Schonfeldt, “Grenzflachenaktive Athylenoxidaddukte” [Surface-Active ethylene oxide adducts], W iss. V erlagsgesell. 9 Stuttgart, 1 9 7 6; Winnacker-Ktichler, "Chemische Technologie" [Chemical Technology], Volume 7, C. Hanser Verlag, Munich, 4th edition, 1 9 8 6; Μ 11 and and Grubenmann,

“Formulierungstechnik” [Formulation Technology], Wiley-V C H - V e r 1 a g, W e i n h e i m，2 0 0 0 o 溶劑EHL，乳酸2-乙基己酯，爲一種2-乙基己醇與乳酸（較佳爲L- ( + )-乳酸）形成之酯類，其可例如從 Purac Bioquimica ( Gram Vial 19-25，0 8 1 60 Montmela-Barcelona，西班牙）或 Purac Biochem ( Gorinchem, NL )公司之Purasolv® EHL產物取得。EHL的其它名稱還有 ·· 2-乙基己基S-乳酸酯，2-乙基己基L-乳酸，L-乳酸2-乙基己基酯；CAS-No. 1 86 8 1 7-80-1 ; EC-No. 22 8 -5 03 -2。 EHL顯示出良好的溶劑特性，其在環境中可徹底地被分解成二氧化碳及水且沒有任何臭氧還原作用。此外’ EHL (在大鼠，口服）之 LD5G値爲每公斤體重超過 2 000mg，所以在毒物學上是無害的。在人體，EHL的酯鍵會很快地被分解掉且EHL會透過酵素水解而分解成二氧化碳及水。因爲此等便利的特性，所以EHL經常被用在金屬加工上來使材料脫脂且印刷工業亦把EHL用在顏料及墨水中作爲添加劑。對於把EHL用於植物之保護組成物中而言此等性質 (6) 200529745 害蟲使用 EHL 成物除。儲存物質護組的，成物定性善活、林除草劑、除劑含生具有以及蟲及是很有利的，而且還能支持農業化學之活性物質防治的活性，此外還減少了對植物的不良副作用，例如在殺蟲劑時所造成的植物傷害（植物毒害性）°使用的其它優點還有可製得具有較佳閃點之植物之保護組，如此可使得運輸及儲存時所需的限制減少或完全消此外，藉由使用EHL可使得該植物之保護組成物的安定性獲得改善。再者’ EHL可使得農業化學之活性在低溫下仍保持溶液狀態’從而確保冷凍該植物之保成物時該組成物的安定性。據此，將EHL用在活性物質之濃縮液是很有利例如其可在把農業化學之活性物質製成植物之保護組前藉由濕潤該活性物質的表面來增加該活性物質的安。此外，在製備該植物之保護組成物時EHL亦可改性物質之均質性。術語”農業化學之活性物質”包含用在農業、園藝 > 業及獸醫學領域以及居家與畜牧業之所有物質，例如 ^ 劑、殺蟲劑、殺真菌劑、殺細菌劑、殺線蟲劑、殺藻 . 殺軟體動物劑、殺病毒劑、誘生耐藥性物質、具有驅活性之物質及具有生長調節劑活性之物質、含有或不物之組成物，以及補充微量元素及營養素之肥料。以除草、殺昆蟲、殺真菌、殺細菌及殺病毒活性之物質具生長調節劑活性之物質爲較佳。以具有除草、殺昆殺真菌活性之物質爲特佳。較佳地該農業化學之活性物質在20°C下溶於EHL之 (7) 200529745 溶解度爲至少5 g/1，較佳爲至少1 0 g/1。"Formulierungstechnik" [Formulation Technology], Wiley-V CH-Ver 1 ag, Weinheim, 2 0 0 0 o Solvent EHL, 2-ethylhexyl lactate, a 2-ethylhexanol and lactic acid (preferred Is an ester formed from L-(+)-lactic acid, which can be obtained, for example, from Purac Bioquimica (Gram Vial 19-25, 0 8 1 60 Montmela-Barcelona, Spain) or Purac Biochem (Gorinchem, NL) Company's Purasolv® EHL Product obtained. Other names for EHL are ... 2-ethylhexyl S-lactate, 2-ethylhexyl L-lactic acid, L-lactic acid 2-ethylhexyl ester; CAS-No. 1 86 8 1 7-80- 1; EC-No. 22 8 -5 03 -2. EHL shows good solvent properties, it can be completely decomposed into carbon dioxide and water in the environment without any ozone reducing effect. In addition, the LD5G of EHL (in rats, orally) exceeds 2,000 mg per kg of body weight, so it is toxicologically harmless. In the human body, the ester bonds of EHL are quickly broken down and EHL is decomposed into carbon dioxide and water by hydrolysis of enzymes. Because of these convenient properties, EHL is often used in metal processing to degrease materials and the printing industry also uses EHL in pigments and inks as additives. These properties apply to the use of EHL in plant protection compositions (6) 200529745 Pests are eliminated using EHL products. The storage material protection group, the qualitative goodness of adult products, forest herbicides, herbicides containing insects and insects are very beneficial, and can also support the activity of agrochemical active substance control activities, in addition to reduce the adverse effects on plants Side effects, such as plant damage caused by pesticides (phytotoxicity) ° Other advantages of use are protection groups that can produce plants with better flash points, which can limit the transport and storage Reduced or eliminated. In addition, the stability of the plant's protective composition can be improved by using EHL. Furthermore, 'EHL can keep the activity of agrochemicals in a solution state at a low temperature', thereby ensuring the stability of the composition when the preservation of the plant is frozen. Accordingly, it is advantageous to use EHL in a concentrated solution of an active substance. For example, it can increase the safety of the active substance by moistening the surface of the active substance before making it into a plant protection group. In addition, EHL can also modify the homogeneity of the material when preparing the plant's protective composition. The term "active substances in agrochemicals" includes all substances used in the fields of agriculture, horticulture & veterinary science, and home and animal husbandry, such as agents, pesticides, fungicides, bactericides, nematicides, Algaecides. Molluscicides, bactericides, inducing drug-resistant substances, substances with repellent activity and substances with growth regulator activity, compositions with or without, and fertilizers supplemented with trace elements and nutrients. The substances having herbicidal, insecticidal, fungicidal, bactericidal and virucidal activity and those having growth regulator activity are preferred. Particularly preferred are those with herbicidal and fungicidal activities. Preferably, the agrochemical active substance is soluble in EHL (7) 200529745 at 20 ° C. The solubility is at least 5 g / 1, preferably at least 10 g / 1.

具有除草活性之物質之實例可提及的有例如：艾蔻尼芬（aclonifen)，醯胺硫芬（amidosulfuron)，艾尼羅福斯（anilofos)，黃草靈，班福賽特（befuresate)，比司培黎貝克（b y s p i r i b a c )-鈉，溴苯腈，綠麥隆，環奈特（ cyclanilide )，迪麥得奮（desmedipham)，戴闊扶（ diclofop )-甲基（二氯苯氧基苯氧基丙酸甲酯），戴陸分尼肯（diflufenican )，敵草隆，乙烯利，乙福馬賽特（ ethofumesate )，乙氧硫芬（ethoxysulfuron)，芬氧丙（ fenoxaprop) -P-乙基，芬措醯胺（fentrazamide)，氣卡本顚1 (flucarbazone)-鈉，富芬沈（flufenacet)，富塔萌 (flurtamone) ，父瑞硫芬（foramsulfuron)，糖服息內特（glufosinate)-錢，鎭草靈，碑硫芬（iodosulfuron) ，碑苯腈，異丙隆（isoproturon)，異氧富妥（ isoxaflutole )，臨紐隆（linuron)，麥分奈習特（ mefenacet)，中富佛隆（mesofulfuron)-甲基，間米挫（ metamitron )，間硫瀾（meto su 1 am )，賽克津，仰it阿給 (o x a d i a r g y 1 )，惡草靈，分米黛芬（p h e n m e d i p h a m )，羅彼卡釆隆（ropoxycarbazone)-鈉，硫氧參恩（ sulxotrione)及賽戴歐隆（thidiauron)。具有殺昆蟲活性之物質之實例可提及的有例如：乙醯米皮敵（acetamiprid)，阿梨奈松（acrinathrin)，涕天威，雙甲脒，保棉磷，貝塔-賽福辛（cyfluthrin )，西維因，克羅賽那丁（ cloth ia nidi η)，賽福辛（cyfluthrin) -10- 200529745 (8) ，氯氰菊酯，溴氰菊酯，板硫烷，愛西叵（e t h i p r ο 1 e )，滅克磷，芬那米磷（fenamiphos )，倍硫磷，銳勁特，吡蟲啉，多滅磷，滅蟲威，滅縧靈，楓吸磷，苄氯菊酯，伏殺磷，剖賽福斯（prothiofos )，希拉富芬（silafluofen ) ，螺戴克羅芬（spirodiclofen)，羅米希芬（spiromesifen )，賽克羅匹（thiacloprid)，硫雙滅多威，挫羅米辛（ tralomethrin )，三卩坐碟，敵百蟲及參附麥隆（triflumuron )°Examples of the substance having herbicidal activity may be mentioned, for example: alonifen, amidosulfuron, anilofos, yellow grass spirit, befuresate, ratio Spiribac (byspiribac)-sodium, bromobenzonitrile, green malon, cyclanilide, desmedipham, diclofop-methyl (dichlorophenoxyphenoxy) Methyl propionate), diflufenican, diurfenican, ethephon, ethofumesate, ethoxysulfuron, fenoxaprop-P-ethyl , Fentrazamide, flucarbazone-sodium, flufenacet, flurtamone, foramsulfuron, glufosinate -Qian, Lingcaoling, iodosulfuron, benzonitrile, isoproturon, isoxaflutole, linuron, mefenacet, Zhongfu Mesofulfuron-methyl, metamitron, meta-sulfur (Meto su 1 am), secketin, yangdiargy 1 (oxadiargy 1), oxadiazine, phenmedipham, ropoxycarbazone-sodium, sulxotrione And thidiauron. Examples of the substance having insecticidal activity may be mentioned, for example: acetamiprid, arinathrin, aldicarb, dimethoam, boron phosphorus, cyfluthrin ), Westin, cloth ia nidi η, cyfluthrin -10- 200529745 (8), cypermethrin, deltamethrin, sulfanil, ethipr ο 1 e ), Fenfenphos, Fenamiphos, Fenthion, Regent, Imidacloprid, Polychlorfen, Fenfencarb, Fenfen, Maple Phosphate, Permethrin, Fufenfos, Dissection Prothiofos, silafluofen, spirodiclofen, spiromesifen, thiacloprid, thiodicarb, tralomethrin ), Three crickets sitting on a plate, trichlorfon and triflumuron °

具有殺真菌活性之物質之實例可提及的有例如：唄特醇（bitertanol)，溴慕空娜 D坐（bromuconazole)，多菌靈，卡回帕米得（carpropamid)，賽HI空娜π坐（ cyproconazole)，克瘟散，芬娜米同（fenamidone)，芬海塞米得（fenhexamid)，分丁（fentin)，富阿色挫賓 (fluoxastrobin)，富昆空娜哇（fluquinconazole)，福色提（fosetyl )-鋁，撲海因，音叵福立卡伯（ iprovalicarb )，潘塞克羅（pencycuron)，巨氯雷（ prochloraz)，丙判摩卡（propamocarb)鹽酸，甲基代森鋅，回硫空娜挫（prothioconazole)，匹梨米森尼（ pyrimethanil)，螺氧胺（spiroxamine)，太布空娜唑（ tebuconazole)，甲苯福奈得-二氯福奈得（1〇1)^1£111&]^(1-dichlofluanid)，粉銹寧，三代曼醇（triadimenol)，三氟氧挫賓（trifloxystrobin)及三泰空娜卩坐（triticonazole 較佳者爲除草及殺昆蟲之活性物質。更佳者爲殺昆蟲 -11 - 200529745 Ο) 之活性物質，特別是愛西叵及銳勁特。前述活性物質於活性物質濃縮液中之濃度，即於EHL 中之濃度變化很大且將視個別的終端用途而定。用途可決定濃度，此爲熟悉此技術人士參照活性物質濃縮液及其個 ’ 別之終端用途所習知。較佳地濃度爲0.1重量°/。到95重量 ^ %，特佳地爲0.2重量％到85重量％。於本發明較佳具體例中，該植物之保護組成物中包括 B 了一種額外的成份，其爲選自聚二甲基矽氧烷類之化合物，其被認爲可防止泡沫的形成（所以被稱爲”消泡劑”），可來自例如 Break Thru® (Goldschmidt, Essen，德國），Dow Corning® (Dow Chemicals，Wiesbaden，德國）及 Silwet® ( 〇si Specialities/Akzo Nobel，Frankfurt,德國）。該聚二甲基矽氧烷本身可改善活性物質在水表面的行爲。該聚二甲基矽氧烷之濃度變化很大且將視該植物之保 φ 護組成物所需之散佈效果而定。通常用途會決定濃度，此 - 爲熟悉此技術人士參考每次所需的散佈效果後所習知。較佳地濃度爲0.5重量％到3 0重量％，特佳地爲3重量％到 1 0重量％。聚二甲基矽氧烷較佳係用在液體調合物中，特別是用在AL劑型中（同如下所解釋般）^ 除了前面以提及的成份以外，依據該農業化學之活性物質的化學性質還可以在調合物中使用其它額外的物質。此等物質包括使該農業化學之活性物質安定之物質， -12- 200529745 (10) 如丁基化羥基甲苯（BHT )、檸檬酸或醋酸，可以選用的物質及濃度範圍很廣且將視該農業化學之活性物質之安定性而定。通常用途會決定濃度，此爲熟悉此技術人士參考每一次所需溶解之農業化學之活性物質後所習知。較佳地 • 濃度爲0.0 1重量％到1重量％，特佳地爲（K 1重量％到0.2 ‘ 重量％。類似地，在本發明之調合物中，特別是在液體調合物 φ 中，尤其是在AL劑型中（同下文所解釋般），可以包括其它選自非極性或極性及質子惰性或親質子性溶劑之額外的溶劑，例如苯甲醇、二甲基亞礪（DMSO )、苯甲酸 C12-C15 烷基酯（Pentonat DB(R))、肥酸二異丙酯（ Crodamol DA(R) ) 、N -辛基B比咯Π定酮（NOP)或二甲基乙醯胺（DMAc )。此等額外溶劑之濃度範圍變化很大且將視本發明液體AL劑型之植物之保護組成物中欲溶解之農業化學之活性物質之安定性而定。通常用途會決定濃度 φ ，此爲熟悉此技術人士參考每次所需溶解之農業化學之活一性物質後所習知。較佳地濃度爲50重量％到95重量％， V 特佳地爲75重量％到85重量％。可能的調合物劑型變化很大。關於此點，此等方法爲熟悉此技術人士一般所熟知且述於例如 Winnacker-Kuchler，“Chmische Technologie” [Chemical Technology], volume 7，C. Hanser Verlag, Munich, 4th edition, 1986 i J. W. van V alkenburg, “Pesticide Formulations”， Marcel Dekker N. Y·， 1 9 7 3 ； K. Martens, “Spray Drying -13· (11) (11)200529745Examples of substances having fungicidal activity may be mentioned, for example: bitertanol, bromuconazole, carbendazim, carpropamid, sai kona Seated (cyproconazole), Kewensan, fenamidone, fenhexamid, fentin, fluoxastrobin, fluquinconazole, Fosetyl-aluminum, puffin, iprovalicarb, pencycuron, prochloraz, propamocarb hydrochloride, methyl methanoate Zinc, prothioconazole, pyrimethanil, spiroxamine, tebuconazole, toluconide-dichlorofunaide (101) ^ 1 £ 111 &] ^ (1-dichlofluanid), fentanine, triadimenol, trifloxystrobin, and triticonazole. Preferred are herbicidal and insecticidal active substances. The better is the active substance of Insecticide-11-200529745 〇), especially Don't be Aishin and Ruijinte. The concentration of the aforementioned active substance in the active substance concentrate, that is, the concentration in the EHL varies greatly and will depend on the individual end use. The use determines the concentration, which is familiar to those skilled in the art with reference to active substance concentrates and their individual end uses. A preferred concentration is 0.1% by weight. To 95% by weight, particularly preferably 0.2 to 85% by weight. In a preferred embodiment of the present invention, the plant protective composition includes an additional component B, which is a compound selected from polydimethylsiloxanes, which is considered to prevent the formation of foam (so Known as "defoamers") and can come from, for example, Break Thru® (Goldschmidt, Essen, Germany), Dow Corning® (Dow Chemicals, Wiesbaden, Germany) and Silwet® (〇si Specialities / Akzo Nobel, Frankfurt, Germany) . The polydimethylsiloxane itself improves the behavior of the active substance on the water surface. The concentration of the polydimethylsiloxane varies greatly and will depend on the spreading effect required for the plant's φ protection composition. Normal use will determine the concentration, this-as will be familiar to those skilled in the art after referring to the required dispersion effect each time. More preferably, the concentration is from 0.5% to 30% by weight, and particularly preferably from 3% to 10% by weight. Polydimethylsiloxane is preferably used in liquid blends, especially in AL dosage forms (as explained below) ^ In addition to the ingredients mentioned above, the chemistry of the active substance according to the agrochemical Properties It is also possible to use other additional substances in the blend. These substances include those that stabilize the active substance of the agricultural chemistry, -12-200529745 (10) such as butylated hydroxytoluene (BHT), citric acid or acetic acid. The range of substances and concentrations that can be selected is wide and will depend on the The stability of active substances in agricultural chemistry depends. Normal use will determine the concentration, which is familiar to those skilled in the art after referring to the active substance of agricultural chemistry to be dissolved each time. Preferably • the concentration is from 0.01 to 1% by weight, particularly preferably (K from 1 to 0.2% by weight. Similarly, in the blends of the present invention, especially in the liquid blend φ, Especially in the AL dosage form (as explained below), it may include other additional solvents selected from non-polar or polar and aprotic or protic solvents, such as benzyl alcohol, dimethyl sulfite (DMSO), benzene C12-C15 alkyl formate (Pentonat DB (R)), diisopropyl fatty acid (Crodamol DA (R)), N-octyl B-pyridinone (NOP) or dimethylacetamide ( DMAc). The concentration range of these additional solvents varies widely and will depend on the stability of the agrochemical active substance to be dissolved in the plant's protective composition of the liquid AL dosage form of the present invention. Normal use will determine the concentration φ, this It will be familiar to those skilled in the art after referring to the agrochemical chemistry that needs to be dissolved each time. The preferred concentration is 50% to 95% by weight, and V is particularly preferably 75% to 85% by weight. The possible blend formulations vary widely. In this regard, these methods are Those familiar with this technology are generally familiar and described in, for example, Winnacker-Kuchler, "Chmische Technologie" [Chemical Technology], volume 7, C. Hanser Verlag, Munich, 4th edition, 1986 i JW van Valkenburg, "Pesticide Formulations", Marcel Dekker N. Y ·, 1 9 7 3; K. Martens, "Spray Drying -13 · (11) (11) 200529745

Handbook’’，3rd Ed” 1979，G. Goodwin Ltd., London,或 Mollet and Grubenmann, “Formulierungstechnik” [Formulation Technology]，Wiley-VCH-Verlag? W e i n h e i m ? 2000之中° 調合物劑型之實例有（每次皆採用GCPF調合物碼之縮寫及說明）：AE氣霧分粉末；AL任何其它液體；CG 包膠顆粒；CL接觸液體或凝膠；CS膠囊懸浮液；DC分散濃縮液；DP可粉碎粉末；DT直接投藥之錠劑；EC可乳化濃縮液；ED可電泳液體；EG可乳化顆粒；EO油包水乳液；EW水包油乳液；FG微細顆粒；FS種子處理用之可流動濃縮液；GG巨顆粒；GL可乳化凝膠；GP浮塵 (flo-dust ) ; GR顆粒；GW水溶性凝膠；ME微乳液； MG巨顆粒；OF油溶混性之可流動濃縮液/油溶混性懸浮液；OL油溶混性液體；OP油可分散粉末；PC凝膠或糊劑濃縮液；S E懸浮乳液；S G水溶性顆粒；S L溶解性濃縮液；S Ο散佈油；S P水溶性粉末；S T水溶性錠劑；S ϋ超低體積（ULV )懸浮液；ΤΒ錠劑；TC技術性物質；ΤΚ技術性濃縮液；UL超低體積（ULV )液體；WG水可分散顆粒；WP可濕化粉末；XX其它。較佳者爲液體劑型及固體劑型，其可透過活性物質濃縮液來製得。此等劑型包括劑型 EC (爲可乳化濃縮液之 GCPF碼）；GR (爲顆粒之 GCPF碼）；EW (爲水包油乳液之GCPF碼）；ME (爲微乳液之GCPF碼）；EG (爲可乳化顆粒之GCPF碼）；SE (爲懸浮乳液之 GCPF碼）；SL (爲可溶性濃縮液之 -14- 200529745 (12) GCPF 51 ) ; c S (爲膠囊懸浮液之GCPF碼），·及AL (立即可用液體劑型之GCPF碼）。較佳爲液體劑型，尤其是立即可用液體劑型（劑型AL )。於個別劑型中，含有EHL及一或多種農業化學之活 ^ 性物質之活性物質濃縮液之濃度範圍變化很大且將視所對 ^ 應之劑型而定。通常用途會決定濃度，此爲熟悉此技術人士參考個別劑型後所習知。較佳地濃度爲2重量％到9 5重 • 量％，特佳地爲10重量％到90重量％。本發明亦包括製備含有EHL及一或多種農業化學之活性物質之活性物質濃縮液，以及從該活性物質濃縮液來製備植物之保護組成物。相關之所用之方法爲熟悉此技術者一般所習知，且例如係述於前述不同劑型所引用之文獻 (參見上文）。在製備時一般較有利地係採用實施例中所使用之添加及混合之順序或者實施例中所代表之個別成份〇 # 本發明之活性物質濃縮液爲一種真溶液，即在室溫下 • 該濃縮液液體中之農業化學之活性物質係呈溶解的形式。 V 所有熟悉此技術者習知的方法皆可用來作爲施用的形式；可提及的有例如：噴灑、霧化、多種直接施用之特殊方法’及多種在植物附近非直接施用之特殊方法如將顆粒混入泥土中或施用在灌水稻田的水中。本發明不同劑型之植物保護組成物施用在每單位面積及/或施用在病蟲害防治之測試主體上之個別份量的變化極大。關於此點通常地，如熟悉此技術者參考個別的使用 -15- (13) (13)200529745 領域後所習知般可用多種施用媒體來給予不同的習知用量 ’例如在採用標準噴灑法時每英畝需施用數百公升的水，而在使用超低體積航空器施用時則每英畝係施用數公升的油’而採用注射法時施用量則減成數毫升的生理溶液而已。所以於對應的施用媒體中本發明植物之保護組成物的濃度會有很大的變化且將視個別的使用領域而定。通常所用的濃度爲熟悉此技術人士參考個別的使用領域後所習知。較佳地濃度爲0.01重量％到99重量％，特佳地爲0.1重量 %到9 0重量％。於本發明其它的較佳具體例中，極有利地可將本發明之活性物質濃縮液或從該濃縮液製得之不同劑型的植物之保護組成物直接與其它的植物之保護組成物/調合物混合在一體，於該其它的植物保護組成物/調合物中亦含有農業化學之活性物質及額外的配方助劑。關於此等所用的方法、可能需要的配方助劑及植物之保護組成物/調合物一般皆爲熟悉此技術者所習知且係述於例如 Watkins，“ Handbook of Insecticide Dust Diluents and Carriers，’，2nd Ed., Darland Books, Caldwell，紐約；H. v. Olphen， “Introduction to Clay Colloid Chemistry”，2nd Ed·, J. Wiley & Sons, N.Y.； C. Marsden, u Solvents Guide9% 2nd Ed·，Interscience，紐約，1963 ; McCutcheon’s “Emulsifiers and Detergents- International Ed,”， Annual, MC Publ. Corp·，Ridgewood,紐約；McCutch eon’s u Emulsifiers and Detergents-North America Ed.”，Annual，MC Publ· corp·， -16- (14) (14)200529745Handbook ", 3rd Ed" 1979, G. Goodwin Ltd., London, or Mollet and Grubenmann, "Formulierungstechnik" [Formulation Technology], Wiley-VCH-Verlag? Weinheim? 2000 Examples of blend formulations are ( Abbreviation and description of GCPF blend code are used each time): AE aerosol powder; AL any other liquid; CG encapsulated particles; CL contact liquid or gel; CS capsule suspension; DC dispersion concentrated solution; DP can be crushed Powder; DT directly administered tablets; EC emulsifiable concentrate; ED electrophoretic liquid; EG emulsifiable particles; EO water-in-oil emulsion; EW oil-in-water emulsion; FG fine particles; flowable concentrate for FS seed treatment GG giant particles; GL emulsifiable gel; GP flo-dust; GR particles; GW water-soluble gel; ME microemulsion; MG giant particles; OF oil miscible flowable concentrate / oil miscible OL oil miscible liquid; OP oil dispersible powder; PC gel or paste concentrated liquid; SE suspension emulsion; SG water-soluble particles; SL soluble concentrated liquid; S 0 dispersion oil; SP water-soluble powder ; ST water-soluble tablets; S ϋ ultra low (ULV) suspension; TB tablets; TC technical substances; TK technical concentrated liquid; UL ultra-low volume (ULV) liquid; WG water-dispersible particles; WP wettable powder; XX other. The preferred is Liquid and solid dosage forms, which can be prepared through active substance concentrates. These dosage forms include dosage form EC (GCPF code for emulsifiable concentrates); GR (GCPF code for granules); EW (oil-in-water emulsion GCPF code); ME (GCPF code for microemulsions); EG (GCPF code for emulsifiable particles); SE (GCPF code for suspension emulsions); SL (-14- 200529745 for soluble concentrated liquids) (12) GCPF 51); c S (GCPF code for capsule suspension), and AL (GCPF code for ready-to-use liquid dosage form). Liquid dosage forms are preferred, especially liquid dosage forms (dosage form AL) for immediate use. In individual dosage forms The concentration range of active substance concentrates containing EHL and one or more active substances of agrochemicals varies widely and will depend on the corresponding dosage form. Usually the concentration will be determined by the use. This is a reference for those skilled in the art Known after individual dosage forms. The preferred concentration is 2% to 95% by weight, particularly preferably 10% to 90% by weight. The present invention also includes preparing an active substance concentrate containing EHL and one or more agrochemical active substances, and extracting from the active substance The concentrate is used to prepare a plant protective composition. The methods used are generally known to those skilled in the art, and are described, for example, in the literature cited in the aforementioned different dosage forms (see above). It is generally more advantageous to use the order of addition and mixing used in the examples or the individual ingredients represented in the examples when preparing. # The active substance concentrate of the present invention is a true solution, that is, at room temperature. The agrochemical active substance in the concentrate liquid is in a dissolved form. V All methods familiar to those skilled in the art can be used as a form of application; mention can be made of, for example: spraying, atomizing, special methods of direct application 'and various special methods of indirect application near the plant, such as The granules are mixed into the soil or applied to the water irrigating the paddy field. The individual amounts of plant protection compositions of the present invention in different dosage forms applied per unit area and / or on test subjects for pest control vary greatly. In this regard, generally, as is familiar to those skilled in the art after referring to the individual use -15- (13) (13) 200529745, multiple application media can be used to give different conventional dosages, such as when using standard spraying methods. Hundreds of liters of water per acre need to be applied. When using ultra-low-volume aircraft, several liters of oil are applied per acre, and the injection amount is reduced to a few milliliters of physiological solution. Therefore, the concentration of the protective composition of the plant of the present invention in the corresponding application medium will vary greatly and will depend on the individual field of use. The concentrations usually used are familiar to those skilled in the art after referring to individual fields of use. The preferred concentration is from 0.01% to 99% by weight, particularly preferably from 0.1% to 90% by weight. In other preferred embodiments of the present invention, it is extremely advantageous that the active substance concentrated solution of the present invention or the plant protective composition of different dosage forms made from the concentrated solution can be directly combined with other plant protective compositions / blends. The ingredients are mixed together, and the other plant protection compositions / blends also contain active ingredients of agricultural chemistry and additional formulation aids. The methods used, the formulation aids and plant protection compositions / blends that may be required are generally known to those skilled in the art and are described in, for example, Watkins, "Handbook of Insecticide Dust Diluents and Carriers, ', 2nd Ed., Darland Books, Caldwell, New York; H. v. Olphen, "Introduction to Clay Colloid Chemistry", 2nd Ed ·, J. Wiley & Sons, NY; C. Marsden, Solvents Guide 9% 2nd Ed ·, Interscience, New York, 1963; McCutcheon's "Emulsifiers and Detergents- International Ed,", Annual, MC Publ. Corp., Ridgewood, New York; McCutch eon's u Emulsifiers and Detergents-North America Ed. ", Annual, MC Publ · corp ·, -16- (14) (14) 200529745

Ridgewood，紐約；Sisley and Wood, “Encyclopedia of Surface Active Agents”，Chem. Publ. Co. Inc.，紐約 5 1964 ;Schonfeldt, “Grenzflachenaktive Athylenoxidaddukte” [Surface - Active ethylene oxide adducts] ? Wi s s. V e r 1 a g s g e s e 11 · , S t u 11 g a r t，1 9 7 6。較佳的方法爲槽混法、共調合法及顆粒塗覆法。通常，係以上述的農業化學之活性物質及/或劑型作爲額外的混合夥伴爲佳。前述混合夥伴的混合比例變化很大且係依個別的終端用途而定。通常用途會決定混合比例，此爲熟悉此技術人士參考個別終端用途後所習知。混合比例可爲1 -1 〇 000 ( 含有活性物質濃縮液之植物之保護組成物/調合物）：1-1 0，0 0 0 (不含活性物質濃縮液之植物之保護組成物/調合物 );較佳爲 1-1，000: 1-1,000，特佳爲 1-100: 1-100。Ridgewood, New York; Sisley and Wood, "Encyclopedia of Surface Active Agents", Chem. Publ. Co. Inc., New York 5 1964; Schonfeldt, "Grenzflachenaktive Athylenoxidaddukte" [Surface-Active ethylene oxide adducts]? Wi s s. V er 1 agsgese 11 ·, S tu 11 gart, 1 9 7 6. The preferred methods are tank mixing, co-tuning, and particle coating. Generally, it is preferable to use the above-mentioned agrochemical active substances and / or dosage forms as an additional mixing partner. The mixing ratio of the aforementioned mixing partners varies widely and depends on the individual end use. Normal use determines the mixing ratio, which is familiar to those skilled in the art after referring to the individual end use. Mixing ratio can be 1-1 000 (protective composition / mixture of plants containing active substance concentrate): 1-1 0,0 0 0 (protective composition / mixture of plants without active substance concentrate ); Preferably 1-1,000: 1-1,000, particularly preferably 1-100: 1-100.

本發明之一較佳具體例爲一種植物之保護組成物的用途，其中該組成物爲一種液體調合物，較佳地爲一種AL 調合物，其包含EHL，任意地一或多種選自非極性或極性質子惰性或親質子性溶劑，一或多種選自聚二甲基砂氧院類之消泡劑，一或多種農業化學之活性物質及任意地用以安定該活性物質之物質。特佳者爲 purasolv® ’ DMS0 ’ Break Thru OE 441®及愛西叵’特佳地爲含有65重量％之 Purasolv®，30 重量。/。之 DMS0’ 2 重量 °/〇之 Break Thru 0E 441©及3重量％之愛西叵。在本發明較佳具體例之製備中，一般較佳地係採用實 -17- (15) 200529745 施例中所顯示之添加及混合個別成份的順序。本發明所使用的植物之保護組成物中有一部份爲已知且有一部份則爲新穎的。所以，於本發明再一態樣中係提供一種植物之保護組成物，其包含： a)乳酸2-乙基己酯，A preferred embodiment of the present invention is the use of a plant protection composition, wherein the composition is a liquid blend, preferably an AL blend, which contains EHL, optionally one or more selected from non-polar Or polar aprotic or protic solvents, one or more antifoaming agents selected from the group consisting of polydimethyl sulfoxide, one or more active substances of agricultural chemistry, and any substance used to stabilize the active substance. Particularly preferred are purasolv® ’DMS0 ′ Break Thru OE 441® and Acetone 特 particularly preferred are 65% by weight of Purasolv®, 30% by weight. /. DMS0 ’2 weight ° / 〇 Break Thru 0E 441 © and 3% by weight of Azadirachtin. In the preparation of the preferred embodiments of the present invention, it is generally preferred to use the order of adding and mixing the individual ingredients as shown in the practical example -17- (15) 200529745. Some of the protective compositions of plants used in the present invention are known and some are novel. Therefore, in another aspect of the present invention, a plant protection composition is provided, which comprises: a) 2-ethylhexyl lactate,

b )溶於其中之一或多種農業化學之活性物質係選自如下群組： 1)艾蘧尼芬（aclonifen)，醯胺硫芬（amidosulfuron )，艾尼羅福斯（anilofos )，黃草靈，班福賽特（ befuresate)，比司培黎貝克（byspiribac)-鈉，溴苯腈，綠麥隆，環奈特（cyclanilide)，迪麥得奮（desmedipham )，戴闊扶（以(：1(^〇?)-甲基（二氯苯氧基苯氧基丙酸甲酯），戴陸分尼肯（diflufenican )，敵草隆，乙烯利，乙福馬賽特（ethofumesate)，乙氧硫芬（ethoxysulfuron) ，芬氧丙（fenoxaprop) -P-乙基，芬措醯胺（ fentrazamide)，氟卡本酮（flucarbazone)-鈉，富芬沈（ flufenacet )，富塔萌（flurtamone)，父瑞硫芬（ foramsulfuron)，糖服息內特（glufosinate)-錢，鎭草靈，碘硫芬（iodosulfuron )，碘苯腈，異丙隆（ i sopro turon )，異氧富妥（isoxaflutole)，臨紐隆（ 1 i η υ r ο n )，麥分奈習特（mefenacet)，中富佛隆（ m e s 〇 f u 1 f u r ο η )-甲基，間米挫（m e t a m i t r ο η )，間硫爛（ m e t o s u 1 a m )，賽克津，仰威阿給（o x a d i a r g y 1 )，惡草靈 -18- (16) 200529745 ，分米黛芬（phenmedipham)，羅彼卡釆隆（ ropoxy carbazone )-鈉，硫氧參恩(sulxotrione )及賽戴歐隆(thidiauron) ; 2 )乙醯米皮敵（acetamiprid )，阿梨奈松（ acrinathrin )，涕天威，雙甲脒，保棉碟，貝塔-賽福辛（耆b) the active substance dissolved in one or more of the agrochemicals is selected from the following group: 1) alonifen, amidosulfuron, anilofos, yellow grass spirit, Befuresate, bespiribac-sodium, bromobenzonitrile, green malon, cyclanilide, desmedipham, Dai Kuofu (with (: 1 (^ 〇?)-Methyl (dichlorophenoxyphenoxypropionate methyl ester), diflufenican, diuron, ethephon, ethofumesate, ethoxysulfur Ethoxysulfuron, fenoxaprop-P-ethyl, fentrazamide, flucarbazone-sodium, flufenacet, flurtamone, parent Foramsulfuron, glufosinate-money, humulose, iodosulfuron, iodosulfuron, isopro turon, isoxaflutole, Pro Nurong (1 i η υ r ο n), mefenacet, mes fu 1 fur ο η) -methyl, metamitr ο η), metosu 1 am, secketin, oxadiargy 1, oxadiazine-18- (16) 200529745, min Phenmedipham, ropoxy carbazone-sodium, sulxotrione and thidiauron; 2) acetamiprid, aprinidone ( acrinathrin), Xitianwei, Shuangjiayu, cotton discs, Beta-Syfosin (耆

cyfluthrin)，西維因，克羅賽那丁（ clothianidin)，賽福辛（cyfluthrin)，氯氰菊酯，溴氰菊酯，板硫烷，愛西回（ethiprole)，滅克磷，芬那米憐（fenamiphos)，倍硫磷，銳勁特，吡蟲啉，多滅磷，滅蟲威，滅縧靈，礪吸磷，苄氯菊酯，伏殺磷，剖賽福斯（prothiofos )，希拉富芬（silafluofen)，螺戴克羅芬（spirodiclofen)，羅米希芬（spiromesifen) ，賽克羅匹（thiacloprid)，滅縧靈，礪吸碟，予氯菊酯，伏殺憐，剖賽福斯（p r 〇 t h i 〇 f 〇 s )，希拉富芬（silafluofen )，螺戴克羅芬（ spirodiclofen)，羅米希芬（spiromesifen)，賽克羅匹（ thiacloprid)，硫雙滅多威，挫羅米辛（tralomethrin)，三唑磷，敵百蟲及參附麥隆（triflumuron) •，及 3)唄特醇（bitertanol)，多菌靈，卡叵帕米得（ carpropamid)，克癒散，芬娜米同（fenamidone)，芬海塞米得（fenhexamid)，分丁（fentin)，富阿色挫賓（ fluoxastrobin)，福色提（fosetyl)-銘，撲海因，音叵福立卡伯（iprovalicarb)，潘塞克羅（pencycuron)，丙判摩卡（propamocarb)鹽酸，甲基代森鋅，叵硫空娜挫（ p r 〇 t h i 0 C ο n a ζ ο 1 e )，匹梨米森尼（p y r i m e t h a n i 1 )，螺氧胺 -19- (17) (17)200529745 (spiroxamine)，甲苯福奈得·二氯福奈得（t〇〗ylfluanid-dichlofluanid)及三氟氧挫賓（trifl〇xystr〇bi]1); c )任意地一或多種配方助劑。較佳地，該組成物係含有一或多種選自群組i )及2 )之農業化學物質，更佳地係含有選自群組2 )之物質，特別是銳勁特及/或愛西叵。更佳地，該組成物係含有一或多種聚二甲基矽氧烷（如前所述）以作爲成份c )。再佳地，該組成物含有安定該農業化學之活性物質的物質，尤其是丁基化羥基甲苯，檸檬酸或醋酸。再佳地，該組成物還含有額外的非極性或極性質子惰性或親賓子性溶劑，特別是苯甲醇，DMS0、苯甲酸C12-C】5烷基酯、肥酸二異丙酯、N-辛基吡咯啶酮及二甲基乙醯胺。此等額外之配方助劑的較佳濃度係如前文所述。特佳地，組成物係含有兩或多種額外的配方助劑。於本發明再一態樣中係提供一種活性物質濃縮液，其含有a )乳酸2-乙基己酯及b ) —或多種選自群組1 )、2 )及/或3 )之農業化學之活性化合物。於本發明再一態樣中，係提供一種含有如上所述組成物之水溶性容器。術語”有害生物”係包含在相關使用領域中會造成經濟損失及/或有害健康之所有形式的生物。較佳地係指有害的植物及動物以及會造成疾病的生物；特佳地係指陸生及 -20- (18) 200529745 水生的雜草，包括禾本科植物、藻類、苔類；節肢動物，包括昆蟲及蛛形綱節肢動物（如蟎類）；蠕蟲，包括線蟲類；曬齒動物、真菌、細菌及病毒等。特佳地”有害生物”係指有害節肢動物包括昆蟲及蛛形綱節肢動物，以及蠕蟲包括線蟲類。cyfluthrin), sivevain, clothianidin, cyfluthrin, cypermethrin, deltamethrin, sulfanil, ethiprole, fenamiphos, fenamiphos ), Fenthion, Regent, Imidacloprid, Pirfenazone, Pyracetam, Piracetam, Phosphorus, Permethrin, Phosphos, Prothiofos, Silafluofen ), Spirodiclofen, spirodiclofen, spiromesifen, thiacloprid, mirex, rough sucker, permethrin, vomethoxamine, sacrifice prion 〇thi 〇f 〇s), silafluofen, spirodiclofen, spiromesifen, thiacloprid, thiodiphenidone, tromethine ( tralomethrin), triazophos, trichlorfon and triflumuron •, and 3) bitertanol, carbendazim, carpropamid, keyusan, fenami Same (fenamidone), fenhexamid, fentin, fluox astrobin), fosetyl-Ming, puffin, iprovalicarb, pencycuron, propamocarb hydrochloride, methyl methanozine, thorium sulfide娜 na 挫 (pr 〇thi 0 C ο na ζ ο 1 e), pirimethani 1, spiroxamine-19- (17) (17) 200529745 (spiroxamine), toluene funaide dichloride Funat (t〇 ylfluanid-dichlofluanid) and trifluorooxobin (trifloxystrobi) 1); c) any one or more formulation aids. Preferably, the composition contains one or more agrochemicals selected from groups i) and 2), and more preferably contains a substance selected from group 2), especially Ruijinte and / or Acesulfame . More preferably, the composition contains one or more polydimethylsiloxane (as described above) as the component c). Even more preferably, the composition contains a substance which stabilizes the active substance of the agrochemical, especially butylated hydroxytoluene, citric acid or acetic acid. Even more preferably, the composition also contains additional non-polar or polar aprotic or aprotic solvents, especially benzyl alcohol, DMS0, benzoic acid C12-C] 5 alkyl esters, diisopropyl ferric acid, N-octyl pyrrolidone and dimethylacetamide. The preferred concentrations of these additional formulation aids are as previously described. Particularly preferably, the composition contains two or more additional formulation aids. In yet another aspect of the present invention, an active substance concentrate is provided, which contains a) 2-ethylhexyl lactate and b)-or more agricultural chemicals selected from the group 1), 2) and / or 3) Of active compounds. In still another aspect of the present invention, a water-soluble container containing the composition as described above is provided. The term "harmful organism" includes all forms of organisms that cause economic loss and / or are harmful to health in the relevant field of use. Preferably refers to harmful plants and animals and organisms that cause disease; particularly preferred refers to terrestrial and -20- (18) 200529745 aquatic weeds, including grasses, algae, moss; arthropods, including Insects and arachnid arthropods (such as mites); worms, including nematodes; sun-toothed animals, fungi, bacteria and viruses. Particularly preferred "pests" are harmful arthropods including insects and arachnid arthropods, and worms including nematodes.

水稻作物之病蟲害的實例有（皆使用其學名及英文俗名）：剛毛棘荀果（Acanthospermun hispidum)(星刺果 );Acid ovor ax a venae淡褐亞種（細菌性白葉枯病）；瓜葉蝗（Acrida cinerea) ;無翅蝗（Acrida exaltata)； Aeneolamia contigua (牧草斑點沫蟬）；黃側沫蟬（ Aeneolamia flavilatera )(黃邊沬蟬）；異沬禪（ Aeneolamia varia)(蛙蟬）；印度合萌（Aeschynomene indica)(北方節蠶豆）；霍香蔚（Ageratum conyzoides )(山羊草）；水稻潛葉蠅（Agromyxa oryzae)(水稻小葉病）；穀夜蛾（Agrotis segetum)(蕪菁蛾）；背圓粉扁蟲（Ahasverus advena)(外國榖甲蟲）； Aleurocybotus indicus ; A 1 e u r o g 1 y p h u s o vatu s (棕足穀虫蒴 );米僞步行蟲（Alphitobius diaperinus)(少穀蟲）；長梗滿天星（Alternanthera philoxeroides)(鱷魚草）；虫彭螺菊（Alternanthera sessilis)(無柄歡樂草）；蕃節輪斑菌（Alternaria alternata f. sp. lycopersici)(葉輪斑病）；疊心葉燒菌（Alter nariapadwickii)(層燒症）；青寛（Am ar an thus retro flex us )(紅根）；朿丨J 莧（ Amaranth us spinosus ) (朿丨J 莧）；Anadastus filiform is; -21 - (19) 200529745Examples of diseases and insect pests of rice crops (both using their scientific names and common names in English): Acanthospermun hispidum (star fruit); Acid ovor ax a venae light brown subspecies (bacterial bacterial leaf blight); melons leaves Locust (Acrida cinerea); wingless locust (Acrida exaltata); Aeneolamia contigua (grass-spotted grasshopper); yellow-side grasshopper (Aeneolamia flavilatera) (yellow-winged cicada); Aeneolamia varia (frog cicada); Aeschynomene indica (Northern section broad beans); Ageratum conyzoides (Goat grass); Agromyxa oryzae (rice leaf disease); Agrotis segetum (turnip moth); Ahsverus advena (foreign cricket beetle); Aleurocybotus indicus; A 1 eurog 1 yphuso vatu s (Brown-footed worm); Alphitobius diaperinus (Lesser worm); Sky star (Alternanthera philoxeroides) (crocodile grass); insect snail (Alternanthera sessilis) (unscented happy grass); Alternaria alternata f. Sp. Lycopersici (leaf spot) Disease); Alter nariapadwickii (layer fever); Am ar an thus retro flex us (red root); 朿丨 J 苋 (Amaranth us spinosus) (朿丨 J 苋); Anadastus filiform is; -21-(19) 200529745

Anadastus scutellatus;耕地紫繁縷（Anagallis arvensis) (緋紅紫繁縷）；M馬（Anaphothripobscurus)(牧草蟲 ) ;Anaphothrip sudanesis ; Anisopteromalus cal andrae ；Anadastus scutellatus; Anagallis arvensis (Crimson Purple Stellaria); M Horse (Anaphothripobscurus) (Grasshopper); Anaphothrip sudanesis; Anisopteromalus cal andrae;

麗金龜（Anomala antiqua)(塊莖金龜子）；葡萄綠麗金龜（Anomala dimidiata)；麗金龜（Anomala pallida)；稻乾尖線蟲（A p h 1 e n c h o i d e s b e s s e y i )(水稻葉線蟲）； Arthri nium phaespermum ； Aspavia armigera ；寄生麴黴( Aspergillus parasiticus ) ；土麴黴(Aspergillus terreus) ;枯麹黴（Aspergillus ustus)；稻芒角蠅（Atherigona oryzae)(射擊蠅）；負煌（Atractomorphacrenulata); 切葉家蟻（Atta opaciceps );六孔切葉家蟻（Atta sexdens)(切葉蟻）；青稞（Avena fatua)(野燕麥） ;蠘狀芽孢桿菌（Bacillus cereus);枯草桿菌（Bacillus suvtilis);稻肉瘤菌（Balansia oryazae-sativae (烏巴塔（udbatta)症）·’二室葉禪（Balclutah abdominalis) ;大鬼鼠（Bandicotaindica)(印度大鼠）；大麥黃萎症病毒（大麥黃萎症）；鳥類的害蟲；德國蜚蠊（Blattella germanica )(巴豆蟲）·，南部麥長 _ ( Blissus insularis )(南方麥虱/);麥長蝽（Blissus leucopterus)(麥風 );黃細心（Boerhavia diffusa )(豬草）；單帶挵蝶（ Borbo cinnara )(水稻捲葉病）；鴨舌黃（Borreria latifolia )(闊葉紐釦草）；臂形草（Brachiaria paspaloides)(常單株草）；虫牙（Brevenniarehi)(食稻蟲），雀麥錶砍病母，Burkholderia glumae (細困性腐設 -22- (20) 200529745Anomala antiqua (tubular beetle); grape green beetle (Anomala dimidiata); Aleala pallida; A ph 1 enchoidesbesseyi (rice leaf nematode); Arthri nium phaespermum; Aspavia armigera; Aspergillus parasiticus; Aspergillus terreus; Aspergillus ustus; Atherigona oryzae (shooting fly); Atractomorphacrenulata; Atta opaciceps ); Six-hole leaf-cutting house ants (Atta sexdens) (leaf-cutting ants); barley (Avena fatua) (wild oats); Bacillus cereus; Bacillus suvtilis; Balansia oryazae -sativae (udbatta disease) · 'Balclutah abdominalis; Bandicotaindica (Indian rat); Barley Verticillium virus (Barley Verticillium); Pests of birds; German cricket (Blattella germanica) (croton) · Southern wheat long _ (Blissus insularis) (Southern wheat lice /); Wheat long cricket (Blissus leucopterus) ( Wind); Yellow Carefulness (Boerhavia diffusa) (Pigweed grass); Single-banded butterfly (Borbo cinnara) (rice leaf curl); Yellow-tongue (Borreria latifolia) (Broad-leaved button grass); Brachiaria paspaloides (Every single plant); Brevenniarehi (rice-eater), Bromeliad cut-off disease mother, Burkholderia glumae (Fine sleep rot-22- (20) 200529745

症）；Burkholderia plan tarii ;粉斑螟（Cadra acutella ) (葡萄乾蛾）；蘇馬（Caliothrips striatopterus)(玉米黑牧草蟲）；綠豆象（Callosobruchus chinensis)(中國象鼻蟲）；露尾甲（Carpophilus);玉米紅褐露尾甲（ Carpophilus dimidi atus )(玉米囊甲蟲）；山扁豆（ Cassia obtusifolia)(鐮形莢）；Caulopsis cuspidata (長角稻螅）；Caulopsis gracillima (長角蝗）；Caulopsis sponsa (長角蝗）；青葙（Celosia argentea)(鵪鶉草） ;漢藜草（Cenchrus echinatus (剌芒草）； Ceratobasidium cereale (穀類銳眼斑症）；金魚藻（ Ceratophyllum demersum ) ( ί完熊尾草)；Ceresa minor ；跳甲(Chaetocnema basalis)；白藜(Chenopodium album )(肥母雞草）；跳觸（Cheyletus malaccensis);禾草螟（Chiloagamemnon)(玉米東方蠢蟲）；臺灣稻螟（ Chilo auricilius )(金緣稻蠢蟲）：稻褐頭螟（Chilo diffusilineus );玉米禾螟（Chilo partellus )(斑莖蠢蟲 )•，七星稻螟（Chilo plejadellus )(美國稻桿蠢蟲）；稻多麗螺（C h i 1 ο ρ 〇 ] y c h r y s u s )(黑頭條紋蠢蟲）；蔗條螟（Chilo sacchariphagus)(斑蠢蟲）；二化螟（Chilo suppressalis)(稻莖蠢蟲）；禾草螺（Chilo zacconius) ;搖蚊（Chironomus tepperi)(紅 ί丘蚓）；虎尾草（ Chloris barbata)(紫頂虎尾草）；稻桿蠅（Chlorops oryzae)(稻莖蛆）；臺灣大螅（Chondracris rosea)( 橘螅）；白花菜（C 1 e o m e v i s c o s a )(黃 m e s a m b a y );虫舂 -23- (21) 200529745Disease); Burkholderia plan tarii; Cadra acutella (raisin moth); Calithrips striatopterus (corn black pasture grass insect); Callosbruchus chinensis (Chinese weevil); Carpophilus ); Carpophilus dimidi atus (Corn cyst beetle); Mountain lentils (Cassia obtusifolia) (Sickle pod); Caulopsis cuspidata (Longhorn rice owl); Caulopsis gracillima (Longhorn locust); Caulopsis sponsa (Long-horned locust); green cockroach (Celosia argentea) (quail grass); Chinese quinoa (Cenchrus echinatus); Ceratobasidium cereale (cereal sharp eye spot disease); Ceratophyllum demersum (ί End beartail grass) ); Ceresa minor; Chaetocnema basalis; Chenopodium album (fat hen grass); Cheyletus malaccensis; Chiloagamemnon (corn flea); Taiwan rice loquat (Chilo auricilius): Chilo diffusilineus; Chilo partellus (spotted moth) •, Chilo pl ejadellus) (American rice stalk stupid); rice snail (C hi 1 ο ρ 〇 ychrysus) (black-headed streaked stupid worm); cane stripe (Chilo sacchariphagus) (spot moth); Chilo suppressalis ) (Rice stalk worm); grass snail (Chilo zacconius); chironomus tepperi (red 红 wormworm); chloris (Chloris barbata) (purple crested grass); rice straw fly (Chlorops oryzae) ( Rice stem cricket); Taiwan cockroach (Chondracris rosea) (Tangerine cricket); white cauliflower (C 1 eomeviscosa) (yellow mesambay); insect cricket 23- (21) 200529745

(Cletus punctiger);針緣蝽（Cletus trigonus)(細米蟲）；稻縱捲葉螟（C n a p h a 1 o c r o c i s m e d i n a 1 i s )(稻捲葉蟲）；旋孢菌（Cochliobolus geniculatus )(穀根腐病） •，旋孢菌（Cochliobolus lunatus)(草、稻及高粱的頭黏菌）；旋孢菌（Cochliobolus miyabeanus)(稻褐葉斑症 );旋孢菌（Cochliobolus ravenelii)(假黑穗病）；旋孢菌（Cochliobolus sativus)(斑瘡瘡）；Cofana spectra (白葉跳蟬）；Cofana unimaculata (白葉跳禪·）; Collaria oleosa ； Colposcelis s i gnat a ；圓葉妬草（ C o m m e 1 i n a benghalensis )(鴨妬草）；白竹仔菜（ Commelina diffusa ) ( 水草 ) ； Conocephaloides obscurellus;角艎（Conocephalus cinerus)(長角綠牧草虫皇）；角煌（Conocephalus propinquus)(長角螅）；角螅（Conocephalus saltator)(長角幢）；加拿大假蓬（ Cony za canadensis)(加拿大蒿）；家白蟻（Coptotermes )(白蟻）；繩黃麻（Corchorus aestuans) ; Corcyra cephalonica (食稻蛾）；皮孔菌（Corticium rolfsii)(菌絲根腐症）；滿天飛（Crassocephalum crepidioides); 環線蟲（Criconemella )(環線蟲）；Cricotopus bicinctus ； Cricotopus sylvestris ； Cricotopus trifasciatus ;錄扁縠盜（Cryptolestes ferrugineus)(銹穀蟲）；長角扁榖盜（Cryptolestes pusillus)(扁穀蟲）；蚊（ Culicoides furens ) ; Curvularia (黑仁）；Cymoninus notabilis;狗牙草（Cynodon dactylon)(百慕達草）； -24- (22) 200529745 莎草（Cyperus brevifolius)(菅茅）；莎草（Cyperus compressus ) ( 一年生菅茅）；異花莎草 (Cyperus difformis )(小花果薹）；Cyperus esculentus (黃果薹） :碎米莎草（Cyperus iria )(蚱蜢莎草）；香附子（ Cyperus rotundus )(堅果草）；龍爪草（Dactyloctenium aegyptium)(毛莨）；Deois flavopicta (淡褐沬蟬）；葉甲（Diabrotica speciosa ) ( SI 蘆蟲）；Diasemopsis(Cletus punctiger); Cletus trigonus (fine rice worm); C napha 1 ocrocismedina 1 is (rice leaf worm); Cochliobolus geniculatus (grain root rot ) •, Cochliobolus lunatus (cephalomycetes of grass, rice and sorghum); Cochliobolus miyabeanus (rice leaf spot); Cochliobolus ravenelii (false smut) ; Cochliobolus sativus (spot sores); Cofana spectra (leafhopper); Cofana unimaculata (Collar leaf zen); Collaria oleosa; Colposcelis si gnat a; Comcel 1 ina benghalensis (Duck jealous grass); White bamboo lettuce (Commelina diffusa) (Water grass); Conocephaloides obscurellus; Conocephalus cinerus (Long-horned green herbivorous emperor); Conocephalus propinquus (Long-horned owl); Conocephalus saltator) (Long-horned building); Cony za canadensis (Artemisia canadensis); Coptotermes (termites); Corchorus aestuans; Corcyra cepha lonica (rice-eating moth); Corticium rolfsii (mycelial root rot); Skyfly (Crassocephalum crepidioides); Ringworm (Criconemella) (Cyclosphaera); Cricotopus bicinctus; Cricotopus sylvestris; Cricotopus trifasciatus; Pirate (Cryptolestes ferrugineus) (Crustworm); Cryptolestes pusillus (Plantworm); Mosquito (Culicoides furens); Curvularia (Black Kernel); Cymoninus notabilis; Cynodon dactylon (Hundred) (Muda grass); -24- (22) 200529745 Cyperus (Cyperus brevifolius) (Echidrum); Cyperus (Compressus) (Cyperus annual); Cyperus difformis (Cyperus difformis); Cyperus esculentus (Cyperus ilia) (Cyperus iria) (grass sedge); Cyperus rotundus (nut grass); Dactyloctenium aegyptium (hairy owl); Deois flavopicta (hazel brown Cicada); Leaf beetle (Diabrotica speciosa) (SI worm); Diasemopsis

macrophthalma (柄眼蠢蟲）；異草螟（Diatraea centre 11 a )(甘蔗及稻之柄眼蠢蟲）；異草螟（Diatraea lineolata )(新熱帶玉米柄蠢蟲）；Dichelops melacanthus; Dicladispa armigera (稻 hispa );升馬唐（Difitaria cillaris)(熱帶手指草）；D i m o rp h o p t e r u s ; Dinoderus minutus (竹粉後甲蟲）；突眼蠅（Diopsis apicalis);突眼蠅（Diopsis longicornis)(柄眼蠅）；Ditylenchus angustus (稻莖線蟲）；Doloessa viridis ;斑角蝽（ Dolycoris baccarum)(黑刺李甲蟲）；角_ ( Dolycoris indicus);食根金花蟲（Donacia provosti)(稻食根蟲 ) ；Draeculacephala clypeata (尖頭葉跳禪）；macrophthalma (stalk-eye stupid); Diatraea centre 11 a (sugar cane and rice-stemmed stupid); Diatraea lineolata (new tropical corn-stemmed stupid); Dichelops melacanthus; Dicladispa armigera ( Rice hispa); Difitaria cillaris (tropical finger grass); Dimo rp hopterus; Dinoderus minutus (bamboo meal beetle); Diopsis apicalis; Diopsis longicornis ); Ditylenchus angustus (rice stem nematode); Doloessa viridis; Dolycoris baccarum (sloe beetle); horn (Dolycoris indicus); Donacia provosti (rice root worm); Draeculacephala clypeata (Leaped Leaf Zen)

Drechslera gigantea (眼斑）；爪卩圭木棉黑帶紅蝽（ Dysdercus nigrofasciatus ) ；紅蝽 ( Dy sdercus superstitiosus);薦灰粉阶（Dysmicoccus boninsis)(粉紅食蔗蟲）：埃及金鋼鑽（Earias insulana )(埃及莖蠢蟲）：芒稷（Echinochloa colonum )(叢稻）·，稗（ Echinochloa crus-galli ) (榖場草）；稻禾（ -25- (23) 200529745Drechslera gigantea (eye spots); Dysdercus nigrofasciatus; Dy sdercus superstitiosus; Dysmicoccus boninsis (pink sugar cane): Egyptian gold diamond (Earias insulana) ) (Egyptian stem worm): Echinochloa colonum (bush rice) ·, Echinochloa crus-galli (grass field); rice grass (-25- (23) 200529745

Echibocnemus oryzae ) ;稻鱗象蟲（EchinocnemusEchibocnemus oryzae); Echinocnemus oryzae

squameus )(稻株象鼻蟲）；布袋蓮（Eichhornia eras sipes )(水風信子）；小玉米螟（Elasmopalpus lignosellus)(小玉米柄蠢蟲）；牛筋草（Eleusine indica )(禽足草）；紫背草（Emilia sonchifolia )(耗草）；葉裡粉蟲（Entyloma oryzae )(稻葉黑穗病）；Eoreuma 1 〇 f t i n i ;稻水蠅（E p h y d r a m a c e Γΐ a r i a )(稻蠅）；附球（ Epicoccum nigrum )(榖紅斑症）；瓢蟲（Epi 1 achna similis)(玉米瓢蟲）；長穩鯽魚草（Eragrostis japonica )(巧愛草）；歐氏文菌（Erwinia carotovora亞種 carotovora )(地瓜的細菌性根腐症）；歐氏文菌（squameus) (rice weevil); Eichhornia eras sipes (water hyacinth); Elasmopalpus lignosellus (small corn stalk); Eleusine indica (podia) ; Emilia sonchifolia (grass); Entyloma oryzae (smut smut); Eoreuma 10ftini; rice water fly (E phydramace Γΐ aria) (rice fly); attached ball ( Epicoccum nigrum) (Erythema erythematosus); Ladybug (Epi 1 achna similis) (Corn ladybug); Eragrostis japonica (Qiaoai grass); Erwinia carotovora subspecies carotovora (sweet potato) Bacterial root rot);

Erwinia chrusanthrmi p v. chrusanthemi )(大麗花的細菌性凋萎症）；二齒犀金龜（Euetheola bidentata )(二齒聖金龜）；大戟（Euphorbia helioscopia)(日大戟）；乳仔草（Euphorbia hi rta )(園大戟）；稻黃毛白毒蛾（ Euproctis minor )；毒蛾(Euproctis virguncula )；毒蛾 (Euproctis xanthorrhoea )；菜幢(Eurydema ventralis ) ;Euscyrtus concinnus ； Eusarcori s ]ewisi ； Eusarcori s parvus (白斑刺蟲）；Eysarcoris ventralis;小飄浮草（ Fimbristylis littoralis )(小飄浮草）；薊馬（ Frankliniella intonsa)(花薊馬）；鐮刀菌（Fusariuni) ;尖鐮孢（Fusarium oxysporum);鐮刀菌（Fusarium proliferatum ) ； G a e u m a η η o m y c e s gi. a minis 品種 gram inis (冠鞘腐枯病）；牛膝菊（Galinsoga parviflora)(小花 -26- (24) 200529745Erwinia chrusanthrmi p v. Chrusanthemi) (Dahlia's bacterial wilt); Euetheola bidentata (Two-tooth holy turtle); Euphorbia helioscopia (Japanese Euphorbia); Euphorbia hi rta) (Euphorbia); Euproctis minor; Euproctis virguncula; Euproctis xanthorrhoea; Eurydema ventralis; Eucyrtus concinnus; Eusarcori s] ewisi ); Eysarcoris ventralis; Fimbristylis littoralis (floating grass); Frankliniella intonsa (thrips); Fusariuni; Fusarium oxysporum; Fusarium proliferatum G aeuma η η omyces gi. A minis gram inis (crown sheath rot); Hyssop (Galinsoga parviflora) (小花 -26- (24) 200529745

II

牛膝菊）；緖秧秧（Galium aparine)(豬狭秧）； Geoica 1 u c i f u g a ；赤黴菌(Gibberella avenacea ) (鐮刀菌枯萎病）；赤黴菌（Gibberella baccata)(咖啡根頸腐枯病）；赤黴菌（Gibberella fujikuroi)(水稻 bakanae 症）；赤黴菌（Gibberella);玉米赤黴菌（Gibberella zeae )(玉米頂穗枯萎病）；Graminella nigrifrons (黑臉葉跳蟬）；非洲螺蛄（Gryllotalpa africana )(非洲螻蛄 );黑螺蟀（G r y 11 u s a s s i m i 11 i s )(野總蟀），·稻管薊馬 (Haplothrips aculeatus )(草薊馬）；皮薊馬（ Haplothrips ganglbaueri ) ; Helicotylenchus dihystera ( 常見旋線蟲）；紫草（Heliotropium eutopaeum)(纈草 )•’ 狗尾草（Heliotropium Indicum)(印度纈草）·，長懦孢(Helminthosporium sigmoideum 品種 irregulare ) ( 稻莖腐枯症）；Helodytes foveolatus (水稻象鼻蟲）·，二星瘤蟲(Herpetogramma phaeopteralis)(草蟲);異皮線蟲（H e t e r 〇 d e r a g 1 y c i n e s )(大豆囊線蟲）；稻異皮線蟲 Heterodera oryzae )(稻囊線蟲）；稻異皮線蟲（ H e t e r o d e r a ο 1· y z i c ο 1 a )(稻囊線蟲）；甘蔗異皮線蟲（ Heterodera sacchari )(甘蔗囊線蟲）；Heteronychus licas (黑甘蔗甲蟲）；Heteronychus lioderes;等岐蔗蝗 (Hieroglyph us banian )(稻螳）；高梁蔗螅（ Hieroglyphus nigrorepletus ) ; Hirschmanniella oryze (稻根線蟲）；Hirschmanniella ;黑金龜（Holochilus brasiliensis ) •，黑金龜（Holotrichia serrata)(白虫齊螬） -27- (25) 200529745Hyssop); Galium aparine (Swine Narrow); Geoica 1 ucifuga; Gibberella avenacea (fusarium wilt); Gibberella baccata (coffee root neck rot); Gibberella fujikuroi (bakanae disease of rice); Gibberella; Gibberella zeae (corn head blight wilt); Graminella nigrifrons (Black-faced leafhopper); Gryllotalpa africana (African salamander); Black snail salamander (Gry 11 usassimi 11 is) (Wild total salamander), · Haplothrips aculeatus (thrips grass); Thrips (Haplothrips ganglbaueri); Helicotylenchus dihystera (common spins) Nematodes); Heliotropium eutopaeum (valerian) • 'Heliotropium Indicum (Herbalium spp.), Helminthosporium sigmoideum (irregulare) (rice stem rot); Helodytes foveolatus (rice elephant trunk) Insects) ·, Herpetogramma phaeopteralis (Grassworm); Heterophyllum nematode (H eter 〇derag 1 ycines) (Soybean sacral line Insects); Heterodera oryzae (rice cyst nematodes); Heterodera oryzae ο 1 · yzic ο 1 a) (sea worms); Heterodera sacchari (sugar cane worms) Heteronychus licas (black sugarcane beetle); Heteronychus lioderes; Hieroglyph us banian (rice praying); Hieroglyphus nigrorepletus; Hirschmanniella oryze (rice root nematode); Hirschmanniella; black brasilis (Holoc) •, Holotrichia serrata (White Worm Qilu) -27- (25) 200529745

;黑金龜（Holotrichia seticollis) ; Hoplolaimus indicus (茅線蟲）；Hoplolaimus seinh or sti (茅線蟲）； Hortensia s i m i 1 i s (常見綠甘蔗葉跳蟬）；水蠅（ Hydrellia deonieri )(稻潛葉蟲）·，大麥水蠅（Hydrellia griseola )(稻潛葉蟲）；菲律賓水蠅（Hy dr el 1 i a philippina)(稻潛葉蟲）；稻黑水蠅（Hydrellia sasakii )(稻莖蛆）；水蠅（Hydrellia );水蠅（Hy dr el lia tomiokai );水蠅（Hydrellia verticillata)(水草蠅）； Hydronomidius molitor ; Hylephila phyleus (稻口P 頭蟲） ;肉座菌（Hypocrea rufa)(柑橘果實枯萎病）；綠鱗象甲（Hypomeces squamosus )(綠象鼻蟲）；銹李（ Hysteroneura setariae)(腐李蚜蟲）；空心菜（Ipomoea aquatica)(水疲菜）；田間鴨嘴草（Ischaemum rugosum )(皴鴨嘴）；鴨嘴草（I s c h a e m u m t i m o r e n s e )(蜈松草 ) •’ J a v e s e 11 a pelucida ;蕃節蠢蟲（Keiferia lycopersicella)(蕃茄針蟲）；Khuskia oryzae(玉米芯腐枯病）；萊利蘭（Laelia suffusa);馬纓丹（Lantana camara )(馬纓丹）；稻灰非 SI ( Laodelphax st r i a t el 1 υ s )(小褐跳蟲）；薛草竊蠢（Lasioderma serricorne)( 蔽草甲蟲）；李氏禾（Leersiahexandra)(南方切割草） ;青萍（Lemna perpusilla )(浮萍）；網翅書蝨（ Lepinotus reticulatus )(網翅書蝨）；Leptispa pygmaea (稻某蟲）·’ Leptochloa chinensis (亞洲 sprangletop); 禾蛛緣蝽（Lept0corisa acuta )(稻籽蟲）；蛛緣蝽（ -28- (26) 200529745Black beetle (Holotrichia seticollis); Hoplolaimus indicus (Grass nematode); Hoplolaimus seinh or sti (Grass nematode); Hortensia simi 1 is (common green sugarcane leafhopper); Water fly (Hydrellia deonieri) (rice leaf miner) , Barley water fly (Hydrellia griseola) (rice leaf miner); Philippine water fly (Hydr el 1 ia philippina) (rice leaf miner); Rice black water fly (Hydrellia sasakii) (rice stalk); water fly ( Hydrellia); water flies (Hy dr el lia tomiokai); water flies (Hydrellia verticillata); Hydronomidius molitor; Hylephila phyleus (rice mouth P head worm); Hypocrea rufa (citrus fruit fusarium wilt) ; Green scale weevil (Hypomeces squamosus) (Green Weevil); Hysteroneura setariae (Prunus aphid); Ipomoea aquatica (Water weed); Ischaemum rugosum (皴 uck beak) ; I schaemumtimorense (蜈松草) • 'J avese 11 a pelucida; Keiferia lycopersicella (tomato needles); Khuskia oryzae (corn cob rot ); Laelia suffusa; Lantana camara (Lantana); rice ash non-SI (Laodelphax st riat el 1 υ s) (small brown jumping worm); Lasioderma serricorne ) (Seal beetle); Leersiahexandra (Southern cutting grass); Lemna perpusilla (Lemna); Lepinotus reticulatus (Lepinotus reticulatus); Leptispa pygmaea (rice) Insects) · Leptochloa chinensis (Asian sprangletop); Leptochora acuta (Rice seed insect); Arachnid (-28- (26) 200529745

Leptocorisa chine n sis ) ( corbett 稻，昆蟲）；蛛緣蝽(Leptocorisa chine n sis) (corbett rice, insect);

Leptocorisa oratorius ) (細稻蟲）；足緣蝽（ Leptoglossus gonagra )(瓜緣蝽）·，褐毛金龜（ Leucopholis irrorata ) (玩具蟲）；金龜(Leucopholis lepidophora)(檳榔白鱭螬）；金門見風紅（Lindernia) ;心葉母草(Lindernia anagallis )；泥花草(Lindernia antipoda ) ; Lindernia ciliata; Lindernia Crustacea;陌上Leptocorisa oratorius) (fine rice worm); Leptoglossus gonagra (melon margin puffer), brown hair beetle (Leucopholis irrorata) (toy bug); gold beetle (Leucopholis lepidophora) (betel nut white beetle); Golden Gate sees the wind red (Lindernia); Lindernia anagallis; Lindernia antipoda; Lindernia ciliata; Lindernia Crustacea; Mo Shang

菜（Lindernia procumbens)(常見僞紫蘩縷）；書虱（ Liposcelis bostrychophila )(書 1¾ );書風（L i p o s c e 1 i s entomophila)(穀嚅蟲）；書風（Liposcelis paeta)(穀曬蟲）·’ 象甲（Lissorhoptrus brevirostris);象甲（ Lissorhoptrus isthmicus ) ；象甲 ( Lissorhoptrus oryzophilus )(美國水薊馬）；螟蛉（Lithacodia distinguenda )(稻僞尺蠖）；飛幢（Locusta migratoria )(遷移性蝗蟲）；Lonchura punctulata (斑點 munia) ;Lonchura ； Longula m a1 a c a ; Lophocateres p u s i 11u s (尼加拉瓜穀蟲）；白花水龍（Ludwigia adscendens)(水月見草）；細葉水丁香（Ludwigia hyssopifo】ia)(水月見草）；水丁香（Ludwigia octovalvis )(月見柳）；殻球孢（Macrophomina phaseolina)(豆類或薛草的炭枯病） ;長針葉蜂（Macrosteles quqdrilineatus)(翠菊葉跳禪 );長針葉蜂（Macrosteles striifrons) ； Magnaporthe grisea (稻癒）；Magnaporthe salvinii (莖腐病）； M a 1 i a r p h a separatella (稻白蠹蟲);Maras mia e x i g u q ( -29- (27) 200529745 稻捲葉蟲）；Marasmia patnalis (稻捲葉蟲）；Marasmia ruralis (稻捲葉蟲）；Marasmia trapezalis (玉米結網毛蟲）·’田字草（Marsilea minuta )(輕飄胡椒草）；稻眼蝶（Melanitis leda ismene )(稻蝶）·，稻蝶（MelanitisVegetables (Lindernia procumbens) (common pseudo-purple wisteria); Book lice (Liposcelis bostrychophila) (Book 1¾); Book wind (L iposce 1 is entomophila) (Valley); Book wind (Liposcelis paeta) (Valley Sunworm) · 'Weevil (Lissorhoptrus brevirostris); Weevil (Lissorhoptrus isthmicus); Weevil (Lissorhoptrus oryzophilus) (American thrips); Lithacodia distinguenda (Rice pseudochimonis); Flying locust (Locusta migratoria) ); Lonchura punctulata (spot munia); Lonchura; Longula m a1 aca; Lophocateres pusi 11u s (Valley of Nicaragua); White flower water dragon (Ludwigia adscendens) (Water primrose); Ludwigia hyssopifoia) (Water primrose ); Water cloves (Ludwigia octovalvis) (Seventh month willow); Macrosporum (Macrophomina phaseolina) (Leguria or Xuecao's charcoal blight); Macrosteles quqdrilineatus (Aster leaf jumping zen); (Macrosteles striifrons); Magnaporthe grisea (Inulin); Magnaporthe salvinii (Stem rot); M a 1 iarpha sepa ratella (rice beetle); Maras mia exiguq (-29- (27) 200529745 rice leaf roller); Marasmia patnalis (rice leaf roller); Marasmia ruralis (rice leaf roller); Marasmia trapezalis (corn netting caterpillar) · 'Tianzi grass (Marsilea minuta) (light pepper grass); rice-eye butterfly (Melanitis leda ismene) (rice butterfly) ·, rice butterfly (Melanitis

suyadana);野路葵（Melochia corchori folia)(紅草） •，根節線蟲（M e 1 o i d o g y n e a r e n a r i a )(花生根節線蟲）；根節線蟲（M e 1 o i d o g y n e e x i g u a )(咖啡根節線蟲）；根節線蟲（Meloidogyne graminicola )(稻根節線蟲）；根節線蟲（Mel oi do gyne incognita )(根節線蟲）； Memnoniella echinata ；曼蝽(Menida histrio )；菊小頭蘇馬(Microcephalothriops abdominalis )(菊萷馬);含羞草（Mimosa pigra)(巨大含羞草）；含羞草（Mimosa pudica )(含羞草）；Mocis frugalis; Mocis latipes (草尺蠖）；鴨舌草（Monochoria vaginalis)(狗魚草）； Mo n ographella albescens (葉灼枯病）；Monographella nivalis (穀類根腐病）；Mormidea angustata ; Mormidea g u e r i n i ； Mormidea picti ventris (惡臭蟲) ；Mormidea ypsilon(惡臭蟲）；小鼠（Mus musculus domesticus)( 小鼠）；蛇目蝶（Mycalesis hors fieldi);球腔菌（ Mycosphaerella holci )(穎片枯萎症）；球腔菌（ Mycosphaerella tassiana )(胡椒果實腐枯病）； Mycovellosiella oryzae (白葉條斑病）·，粉綠狐尾藻（ Myriophyllum aquaticum ) (鸚羽草）；聚藻（suyadana); Melochia corchori folia (red grass) •, Root-knot nematode (M e 1 oidogynearenaria) (Peanut root-knot nematode); Root-knot nematode (M e 1 oidogyneexigua) (Coffee root-knot nematode); Root-knot Nematodes (Meloidogyne graminicola) (Rhizomatidae); Mel oi do gyne incognita (Rhizobial Nematode); Memnoniella echinata; Menida histrio; Microcephalothriops abdominalis (Horse); Mimosa pigra (Migsa mimosa); Mimosa pudica (Mimosa); Mocis frugalis; Mocis latipes (grassworm); Monochoria vaginalis (dogfish grass); Mo n ographella albescens (leaf blight); Monographella nivalis (cereal root rot); Mormidea angustata; Mormidea guerini; Mormidea picti ventris (mite bug); Mormidea ypsilon (mice bug); Mouse (Mus musculus domesticus) (mouse ); Mycalesis hors fieldi; Mycosphaerella holci (Mycelium fusarium wilt); Mycosphaerella tassiana) (Pepper Fruit rot blotch); Mycovellosiella oryzae (white leaf streak) -, light green foxtail (Myriophyllum aquaticum alginate) (parrot feathers grass); Synechococcus (

Myriophyllum spicatum )(尖水狐尾藻）；黏蟲（ -30- 200529745 (28)Myriophyllum spicatum) (Myriophyllum spicatum); slimeworm (-30- 200529745 (28)

Mythimna)(地蠶）；黏蟲（Mythimna latiuscula);勞氏黏蟲（Mythimna loreyi)(玉米毛蟲）；東方黏蟲（ Mythimna separata )(稻田粟蠶蛾幼蟲）；美洲黏蟲（ Mythimna unipuncta)(稻粟蠶蛾幼蟲），·白脈黏蟲（ Mythimna ve n alba);拂尾藻（Naj as graminea)(草狀茨藻）；大茨藻（Naj as marina)(冬青葉茨藻）；小茨藻 (Naj as minor )(針葉茨藻）；螟鈴（N ar an g a d i f f u s a ) (稻綠半尺蠖）；叢刺殻（Nectria haematococca品種 brevicona )(蕃節乾腐症）；叢刺殼（Nectria rigidiuscula )(綠點癭）；Neoconocephalus m ax i 11 o s u s ( 長角蝗）；葉禪（Nephotettix);黑尾葉蟬（Nephotettix cincticeps ),(稻綠葉跳蟬）；葉蟬（Nephotettix malayanus );葉蟫（Nephotettix nigropictus)(稻綠葉跳禪）；葉禪（Nephotettix parvus);葉蟬（Nephotettix virescens)(綠稻葉跳蟬）；稻綠蝽（Nezara viridula) (綠惡臭蟲）；褐飛風（Nilaparvata bakeri);稻褐飛風 (Nilaparvata lugnes )(褐背稻跳蟲，ΒΡΗ )； Nilaparvata maeander ； Nisaga simplex ;粉風（Nisia nervosa )(灰幢）；紅翅煌（Nomadacris septemfasciata )(紅蝗）：盾蝽（Oebalus insularis )(稻惡臭蟲）；盾蝽（Oebalus ornatus)(稻惡臭蟲）：盾蝽（Oebalus p o e c Π u s );美洲稻盾 _ ( 0 e b a 1 u s p u g n a x )(稻惡臭蟲） •，盾蝽（Oebalus ypsiloinoides)(稻蟲）：盾蝽（ Oebalus ypsilongriseus ) ；稻小爪· Ο 1 i g ο n y c h υ s oryzae -31 - (29) 200529745Mythimna) (Groundworm); Mythimna latiuscula; Mythimna loreyi (Corn caterpillar); Mythimna separata (Paddy field millworm larva); Mythimna unipuncta (rice) Larvae of millet silkworm moth), Mythimna ve n alba; Naj as graminea (Ceratium spp.); Naj as marina (C. holly); C. aeruginosa (Naj as minor) (Nana as gaffer); Nar an gadiffusa (Rice green half-footed owl); Nectria haematococca variety brevicona (Vanilla dry rot); Nectria rigidiuscula ) (Green-pointed cricket); Neoconocephalus m ax i 11 osus (Long-horned locust); Yechan (Nephotettix); Black-tailed leafhopper (Nephotettix cincticeps), (rice leafhopper); Leafhopper (Nephotettix malayanus); Leafhopper (Nephotettix nigropictus) (rice green leaf jumping zen); leaf zen (Nephotettix parvus); leafhopper (Nephotettix virescens) (green rice leaf jumping cicada); rice green magpie (Nezara viridula) (green bug); Nilaparvata bakeri ); Rice brown flying wind (Nilaparvata lu gnes) (Brownback rice hopper, ΒΗ); Nilaparvata maeander; Nisaga simplex; Nisia nervosa (grey building); Nomadacris septemfasciata (red locust): Oebalus insularis (rice stench) Oebalus ornatus (rice bug): Oebalus poec Π us; American rice shield _ (0 eba 1 uspugnax) (rice bug) •, Oebalus ypsiloinoides (rice bug) ): Oebalus ypsilongriseus; rice claws 〇 1 ig ο nych υ s oryzae -31-(29) 200529745

；O m a 1 ο n y x felina (鼻涕蟲）；Orphulella punctata ; Orseolia oryzae (稻莖癭蚋）；Orseolia oryzivora (非洲稻癭納）；稻（O r y z a 1 ο n g i s t a m i n a t a )(多年生野稻）；稻（Oryza rufipogon)(紅稻）；鋸榖盜（Oryzaephilus suri namensis )(鋸齒穀蟲）；Oryzophagus oryzae ；稻負泥蟲（Oulema oryzae)(稻葉蟲）·，酢醬草（Oxalis corni cul ata )(蔓生木酸模（USA));酢醬草（Oxalis latifolia )(酸模）；中華稻蝗 Oxy a chinensi s (稻蝗）；曰本稻艎（Oxya japonica) ; Oxya nitidula;稻幢（稻田螅）；北海道稻蝗Oxy a yezoensis (日本蝗蟲）；小眼穀盜（Palorus ratzeburgi)(小眼擬榖盜）；舖地黍（ P a n i c u m repens ) (魚雷草）；P a r a 1 ο n g i d o r u s australis ( 針線蟲);Parapoynx fluctuosalis ； Parapoynx stgnalis ( 稻盒結子木）；兩色綠刺蛾（Parasa bicolor);直紋稻苞蟲（Parnara guttatus (稻跳蟲）；稻苟蟲（Parnara nas〇 );兩耳草（Paspalum conjugatum)(酸草）：雙穗雀稗 (Paspalum distichum)(節草）；蔗飛風(Perkinsiella saccharicida )(甘蔗葉跳蟬）；廣布盤多毛孢（ Pestalotia disseminata )(桉樹葉斑病）；潛岩虫菌 Petrobia latens (褐麥);天社蛾（Phalera combusta) ;Phlugis mantispa (長角螅）；Phlugis teres;莖點黴（ Phoma leveillei )(鞘疙瘩）；稻擬莖點黴（P h o m o p s i s oryzae-sativae)(根頸腐枯症）；澳洲蘆葦（Phragmites australis )(蘆葦）；Phthia obscura ; Phthia picta (黑蟲 -32- (30) 200529745 );庭園葉麗跋（Phyllopertha horticola )(歐洲蕨鐘） ;總角金龜（Phyllophaga helleri )；大萍（Pistia stratiotes )(大藻）；文鳥（Ploceus cucullatus)(稻織布鳥）：印度蠢蛾（Plodia interpunctella)(印度粉蛾）、 ;早熟禾（Poa annua )(—年生牧草）·，金花蟲屬（ Podontia quattuordecimpunctata ) ; 蓼（ Polygonum; O ma 1 ο nyx felina (snot); Orphulella punctata; Orseolia oryzae (rice stem borer); Orseolia oryzivora (african rice borer); rice (O ryza 1 ο ngistaminata) (perennial wild rice); rice (Oryza) rufipogon) (red rice); Oryzaephilus suri namensis (Oryzaephilus surinamensis); Oryzophagus oryzae; Oulema oryzae (rice leaf insect) ·, Oxalis corni cul ata Rumex (USA)); Oxalis latifolia (Ramex); Oxy a chinensi s (Rice locust); Oxya japonica; Oxya nitidula; Rice house (Rice field); Hokkaido rice Locust Oxy a yezoensis (Japanese locust); Palorus ratzeburgi (small-eyed pupae); Panicum repens (torpedo grass); Para 1 ο ngidorus australis (Paratoynx); Parapoynx fluctuosalis; Parapoynx stgnalis (rice box knotwood); two-color green spiny moth (Parasa bicolor); rice grain bud (Parnara guttatus); rice gougworm (Parnara nas〇); Paspalum conjugatum (acid grass): Paspalum distichum (knotweed); Perkinsiella saccharicida (cane leafhopper); Pestalotia disseminata (eucalyptus leaf spot) ; Petrobia latens (brown wheat); Pheraras combusta; Phlugis mantispa (Longhorn owl); Phlugis teres; Phoma leveillei (Shell maggot); P. oryzae (P homopsis oryzae-sativae); Phragmites australis (Phragmites); Phthia obscura; Phthia picta (Black Worm-32- (30) 200529745); Phyllopertha horticola (Europe) Fern bell); total horn beetle (Phyllophaga helleri); daping (Pistia stratiotes) (large algae); wen bird (Ploceus cucullatus) (rice weaver bird): Indian moth (Plodia interpunctella) (Indian meal moth),; precocious Poa annua (—annual forage) ·, Podontia quattuordecimpunctata; Polygonum

aciculare )(節草）；毛蓼（Polygonum barbatum)(節草）；水蓼（Polygonum hydropiper)(沼地胡椒）；多黏黴（Polymyxa graminis )(小麥條狀嵌紋病毒）；多足搖蚊（Polypedilym cultellatum) ； Pomacea canaliculata (金蝸牛）；Pomacea glauca ;馬齒寛（Portulaca oleracea )(馬齒寛）；草地墊刃線蟲（Pratylenchus brachyurus )(根病變線蟲）；刃線蟲（Pratylenchus penetrans)(北美根病變線蟲）；刃線蟲（Pratylenchus zeae)(根病變線蟲）；Psalis pennatula (多毛稻毛蟲）；Psammotettix striatus ； Pseudocochliobolus eragrostidis (玉米葉斑病）；綠膿桿菌（Pseudomonas aeruginosa) •，螢光假單孢菌（Pseudomonas fluorescens)(馬鈴薯粉紅眼斑症）；假單孢菌（Pseudomonas fuscovaginae)( 鞘褐腐枯病）；惡臭假單孢菌（Pseudomonas putida)( 生物防治：歐文氏菌）；丁香假單孢菌稻小種（ Pseudomonas syringae p v. oryzae )(暈圈枯萎病）；丁香假單孢菌丁香小種（Pseidomonas syringae ρν· syringae) (細菌性黑腐倂或瘟病（核果及假果））；丁香假單孢菌 -33- (31) 200529745aciculare) (Arthropoda); Polygonum barbatum (Arthropoda); Polygonum hydropiper (Marsh pepper); Polymyxa graminis (Wheat stripe mosaic virus); Polypedilym cultellatum); Pomacea canaliculata (gold snail); Pomacea glauca; Portulaca oleracea (purslane); Pratylenchus brachyurus (root disease nematode); Pratylenchus penetrans (North American root) Disease nematodes); Pratylenchus zeae (root disease nematodes); Psalis pennatula (hairy caterpillars); Psammotettix striatus; Pseudocochliobolus eragrostidis (maize leaf spot disease); Pseudomonas aeruginosa (Pseudomonas aeruginosa) Pseudomonas fluorescens (Potato pink eye spot); Pseudomonas fuscovaginae (Sheath brown rot); Pseudomonas putida (Biological control: Erwinia); Pseudomonas lilac Pseudomonas syringae p v. Oryzae (Halo wilt); Pseudomonas syringae Race (Pseidomonas syringae ρν · syringae) (bacterial black rot or blast (drupe and pseudofruit)); Pseudomonas syringae -33- (31) 200529745

玉米 /」、種(Pseudomonas s y r i n g a e p v zizania )(細菌性葉條紋病）；丁香假單孢菌（Pseudomonas syringae);紫斑穀螟（Pyralis farinalis )(粉蛾）；腐黴（Pythium arrhenomanes )(榖根腐病）；禾生腐黴（Pythium graminicola )(禾苗枯萎病）；畸雌腐黴（Pythium irregulare)(黑：甜菜管狀枯斑病）；刺腐黴（Pythium spinosum)(根腐病，觀賞植物）；終極腐黴（Pythium ultimum );家鼠（Rattus argentiventer)(稻田野鼠）；緬鼠（Rattus exulans )(灌叢大鼠）；褐家鼠（Rattus norvegicus)(褐鼠）；黑家鼠（Rattus rattus)(黑鼠） ;家鼠（Rattus rattus diardii)(馬來西亞家鼠）；家鼠 (Rattus rattus mindanensis)(常見、菲律賓野鼠）；電光葉蟬（Recilia dorsalis ) ( Z形葉跳蟬）；絲核菌（Maize / ", species (Pseudomonas syringaepv zizania) (bacterial leaf streak); Pseudomonas syringae; Pyralis farinalis (Pink moth); Pythium arrhenomanes (Root rot Disease); Pythium graminicola (grass blight); Pythium irregulare (black: beet tuber leaf spot); Pythium spinosum (root rot, ornamental plants); Pythium ultimum; Rattus argentiventer (rice field rat); Rattus exulans (shrub rat); Rattus norvegicus (brown rat); Rattus rattus ) (Black rat); house rat (Rattus rattus diardii) (Malaysian house rat); house rat (Rattus rattus mindanensis) (common, Philippine wild rat); electro-optic leafhopper (Recilia dorsalis) (Z-leafhopper); silk nucleus bacteria(

Rhizoctonia);稻枯斑絲核菌（Rhizoctonia oryzae)(鞘點病）；根蟎（Rhizoglyphus robini ) •，玉米既（Rhizoctonia); Rhizoctonia oryzae (Sheath spot disease); Rhizoglyphus robini • Corn both (

Rhopalosiphum maidis)(玉米Φ牙蟲）；禾穀縊管Φ牙（ Rhopalosiphum padi )(燕麥赔蟲）；紅腹溢管Φ牙（ Rhopalosiphum rufiabdominale )(稻根 $牙蟲）；稻蠢（ Rhyzopertha dominica)(美國大麥象鼻蟲）；稻黑線矮小病毒；稻小株病毒（稻矮小症）；稻癭矮小病毒；稻草狀矮株病毒；稻hoja blanca病毒（稻白葉症）；稻零亂矮株病毒稻條狀壞死 fur 〇 virus ;稻條狀病毒；稻條狀 tenuWirus ;稻暫時黃化棒狀病毒（稻黃化矮株病毒）；稻t u n g 1· 〇桿狀病毒；稻t u n g r 〇病（稻t u η g r 〇病毒）；稻 -34- (32) 200529745 tiingro球狀病毒；稻黃化矮小植物原漿；稻黃化斑病毒；波狀吐根（R i c h a r d i a b r a s i 1 i e n s i s )(澳洲白眼症）；Rhopalosiphum maidis) (Maize Φ toothworm); Hegulosiphum Φ tooth (Rhoopalosiphum padi) (oat worm); Red-bellied overflow pipe Φ tooth (Rhopalosiphum rufiabdominale) (rice root $ toothworm); Rice stupid (Rhyzopertha dominica) (American barley weevil); rice black dwarf virus; rice small virus (rice dwarf disease); rice dwarf dwarf virus; rice straw dwarf virus; rice hoja blanca virus (rice leaf disease); Rice strip necrosis fur 0 virus; rice strip virus; rice strip tenuWirus; rice transient yellow bar virus (rice yellow stunt virus); rice tung 1.0 baculovirus; rice tungr 0 disease (rice tu η gr 〇 virus); rice-34- (32) 200529745 tiingro globular virus; rice yellowing dwarf plant syrup; rice yellow spot virus; Richardiabrasi 1 iensis (Australia white eye);

Rivula atimeta (綠毛蟲）；羅氏草（Rottboellia cochinchinensis)(搔癢草）；Rupela albinella(稻南美白蠢蟲）；甜子根草（Saccharum spontaneum)(野甘蔗 );野慈姑（8&§以&1^§11>^1^113丨5)(小箭頭）；槐葉蘋 (S alvinia molesta) (卡里巴草）；S arocladium oryzae (稻鞘腐枯病）；螻蛄（Scapteriscus )(螻蛄）；螻蛄 (Scapteriscus didactylus ) (波多黎加螻蛄）； Scaptocoris castaneus (隱藏惡臭蟲）；昨猛（ Schistocerca pallens)(美國煌）；麥二叉虫牙（Schizaphis graminum )(春綠虫牙);白禾螟(Scirpophaga incertulas )(黃莖蠢蟲）；稻白禾膜（Scirpophagainnotata)(白稻莖蠢蟲）；橙尾白禾螺（Scirpophaga nive 11a )(白稻蠢蟲）；Scirpus grossus (大香蒲）；莎草（Scirpus juncoides ) (大燈心草） » 莎草(Scirpus maritimus ) ( 鹽沼燈心草）；指疫黴（Sclerophthora macrospora)(霜黴病）；灰色小核菌（Sclerotium fumigatum);喜水小核菌(Sclerotium hydrophilum ) ; S co tinophara cinerea ; S cotinophara ； S cotinophara coarctata (黑稻蟲) ；Rivula atimeta (green caterpillars); Roche's grass (Rottboellia cochinchinensis) (pruritic grass); Rupela albinella (rice leaf white stupid bug); Saccharum spontaneum (wild sugarcane); Ye Cigu (8 & § to & 1 ^ §11 > ^ 1 ^ 113 丨 5) (small arrow); Salvinia molesta (Kariba grass); Sarocladium oryzae (rice sheath blight); Scapteriscus (蝼蛄)蝼蛄 (Scapteriscus didactylus) (Puerto Rican 蝼蛄); Scaptocoris castaneus (Hidden Stink Bug); Schistocerca pallens (US Huang); Schizaphis graminum (Spring Green Worm); White Wo Scirpophaga incertulas) (yellow-stemmed stink bug); rice white grass (Scirpophagainnotata) (white rice-stem stupid); orange-tailed white grass snail (Scirpophaga nive 11a) (white rice stupid); Scirpus grossus (large cattail); sedge (Scirpus juncoides) (Brush rushes) »Scirpus maritimus (Salt marsh rush); Sclerophthora macrospora (downy mildew); Sclerotium fumigatum; Sclerotium hydrophilum); S co tinophara cinerea; S cotinophara; S cotinophara coarctata (black rice worm);

Scotinophara 1 a t i u s c υ 1 a ；稻黑虫春(Scotinophara lurida) (黑稻蟲）；大螟（Sesamia calalmistis )(非洲粉紅莖蠢蟲）；高梁蛀莖夜蛾（Sesamia cretica)(大甘蔗蠢蟲 );大螟（Sesamia inferens )(紫莖蠹蟲）：大螟（ -35- (33) 200529745 S e s a m i a η ο n a g r i o i d e s )(地中海玉米桿蠹蟲）；大螟（ Sesamia nonagrioides botanephaga ) ；大螟(SesamiaScotinophara 1 atiusc υ 1 a; Scotinophara lurida (Black rice worm); Sesamia calalmistis (African pink-stemmed moth); Sorghum stalk-spotted night moth (Sesamia cretica) (large sugarcane moth) ; Great borer (Sesamia inferens) (Purple stem borer): Great borer (-35- (33) 200529745 S esamia η ο nagrioides) (Mediterranean corn stalk borer); Great borer (Sesamia nonagrioides botanephaga); Large borer (Sesamia

uniformis)(鑽銷毛蟲）；狗尾草（Setaria parviflora) (節根狐尾）；狗尾草（Setaria pumila)(黃狐尾）；倒剌狗尾草（Setaria verticillata)(剛毛狐尾）；狗尾草（ Setaria viridis)(綠狐尾）·，透高蛾（Setomorpha rutella );Setosphaeria holmii; Setosphaeria rostrata(草斑葉病）；細葉金午時草（Sida acuta )(掃帚草）；棉鼠（ Sigmodon )(野鼠）；米象（Sitophilus oryzae)(小穀萷馬）；玉米象Sitophilus zeamais (大穀象鼻蟲）；麥蛾 (Sitotroga cerealella)(穀蛾）；Sogata wallicci ;白背飛風（Sogatella furcifera)(白背螅；WBPH);飛鼠（ Sogatella vibix )(白背蝗）；詹森草（Sorghum halepense )(詹森草）；稻亞球殼菌（Sphaerulina oryzina)(窄褐葉斑病）；尖瓣草（Sphenoclea zeylanica )(模草）·，灰翅夜蛾（Spodoptera culium)(草地毛蟲 );灰翅夜蛾（Spodoptera exempta)(黑粟蠶蛾幼蟲） ;灰翅夜蛾（Spodoptera exigua)(甜菜粟蠶蛾幼蟲）；灰翅夜蛾（Spodoptera frugiperda)(秋粟蠶蛾幼蟲）·，海灰翅夜蛾（Spodoptera littoralis)(埃及棉葉蟲）；灰翅夜蛾（Spodoptera litura)(芋頭毛蟲）；稻灰翅夜蛾 (Spodoptera mauritia )(稻群聚毛蟲）；頂眉紋夜蛾（ Spodoptera mauritia acronyctoides)(粟蠶蛾幼蟲）；鳥灰翅夜蛾（Spodoptera or nit hogal]i)(黃條粟蠶蛾幼蟲） -36- (34) 200529745 ;藥材甲（Stegobium p a n i c e u m ) (姓蟲）；uniformis) (Drill Pin Caterpillar); Setaria parviflora (node root foxtail); Setaria pumila (yellow foxtail); Setaria verticillata (bristle foxtail); Setaria viridis (setaria viridis) ( Green foxtail) ·, Setomorpha rutella; Setosphaeria holmii; Setosphaeria rostrata (grass leaf blight); Sida acuta (broom grass); Cotton rat (Sigmodon) (wild rat); Rice Elephant (Sitophilus oryzae) (Otani 萷); Corn elephant Sitophilus zeamais (Otani weevil); Wheat moth (Sitotroga cerealella) (Cotella); Sogata wallicci; Sogatella furcifera (White-backed Owl) WBPH); Sogatella vibix (white-backed locust); Sorghum halepense (Jensen grass); Sphaerulina oryzina (narrow brown leaf spot); Sphenoclea zeylanica) (mould grass), Spodoptera culium (grass caterpillar); Spodoptera exempta (black moth larva); Spodoptera exigua (beet millet moth larva) Gray-winged Spodoptera Spodoptera frugiperda), Spodoptera littoralis (Egyptian cotton leafworm); Spodoptera litura (Taro caterpillar); Spodoptera mauritia (Spodoptera mauritia) ( Caterpillars of rice swarms); Spodoptera mauritia acronyctoides (Spodoptera moth larvae); Spodoptera or nit hogal] i) (Spodoptera or nit hogal) i-36- (34) 200529745; Medicinal A (Stegobium paniceum) (surname worm);

S tenchaetothrips biform is (稻萷馬）；Stenopola dorsalis ;Stenotus rubrovittatus (高梁蟲）；獨腳金（Striga angustifolia )(獨腳金）；獨腳金（Striga aspera)(獨腳金）；獨腳金（Striga hermonthica)(獨腳金）；獨腳金（Striga lutea)(獨腳金）；金腰箭（Synedrella nodi flora)(金腰箭);Tagosodes cubanus (稻蝗); Tagosodes orizicolus (稻 delphacid ) ; Tagosodes pusanus ;Tarbinskiellus portentosus (稻螻蛄）；跗線鱗（ Tarsonemus fuzhouensi s ) ;跗線蠘(T arsonemus talpae ) ;ί弄蝶（Telicota augias) ; T enebroi des mauritanicus ( 大榖盜）；四脈綿呀（Tetraneura nigriabdominalis)(稻根虫牙蟲）；Tetranyshus urticae (雙點 _ 蛛輸）；Thaia oryzivora (橘稻葉跳禪）；Thaia subrufa; Thanatephorus cucumeris (多種名稱，視宿主而定）；Thioptera botyoides;棕櫚馬（Thrips palmi)(瓜薊馬）；肩蝽 (Thyanta perditor )(褐莖蟲);Tibraca limbativentris (惡臭蟲）；腥黑粉菌（Tilletia barclayana)(稻黑穗病 );稻大蚊（Tipula aino )(稻大蚊）；黃邊黃脊非虱（ Toya propinqua ) ；假海馬齒寛（Triant hema portulacastrum )(馬齒莧）；赤擬榖盜（Tribolium castaneum)(紅粉蟲）；雜擬穀盜（Tribolium confusum )(混粉蟲）；T r i c h i s p a s e r i c e a (硬毛稻）； Trichodorus (粗短根線蟲）；蚤螻（Tridactylus minutus -37- (35) 200529745 );紅鬚盲蝽（Trigonotylus coelestialium)(稻葉蟲）S tenchaetothrips biform is (Rice Horse); Stenopola dorsalis; Stenotus rubrovittatus (Sorghum); Striga angustifolia (Stroke gold); Striga aspera (Stroke gold); Stroke gold (Strike aspera) Striga hermonthica) (Striga lutea) (Striga lutea) (Single-leg gold); Synedrella nodi flora (Golden waist arrow); Tagosodes cubanus (rice locust); Tagosodes orizicolus (rice delphacid); Tagosodes pusanus; Tarbinskiellus portentosus (rice magpie); tarsal scale (Tarsonemus fuzhouensi s); tarsal magpie (T arsonemus talpae); Telicota augias; T enebroi des mauritanicus (big pirate); (Tetraneura nigriabdominalis) (rice root worm toothworm); Tetranyshus urticae (double dot _ spider lose); Thaia oryzivora (orange rice leaf jumping zen); Thaia subrufa; Thanatephorus cucumeris (various names, depending on the host); Thioptera botyoides; palm horse (Thrips palmi) (Thrips palmi); Thyanta perditor (Brown Stem); Tibraca limbativentris (Bad bug); Tilletia barclayan a) (Smut of rice); Tipula aino (Rice mosquito); Yellow edge yellow ridge non-lice (Toya propinqua); Triant hema portulacastrum (purslane); Tribolium castaneum (Trichomonas molitor); Tribolium confusum (Trichomonas); T richispasericea (Sclerotium); Trichodorus (Stubby root nematode); Tridactylus minutus -37- ( 35) 200529745); Trigonotylus coelestialium (rice leaf insect)

;盲蝽（Trigonotylus ruficornis );穀斑皮蠹（ Trogoderma granarium )(榖斑皮蠢蟲）：皮蠹（ Trogoderma variabile )(穀皮蠢）；Tylenchorhynchus annulatus (短線蟲）；Tylenchorhynchus brevilineatus ( 莢痂線蟲）；毛覃甲（Typhaea stercorea)(有毛覃蟲） •，核線菌（Typhula ishikariensis )(小點穀白黴）；腐食酪虫蔭（Tyrophagus putrescentiae)(榖觸）；Ulomoides dermestoides;單孢銹菌（Uromyces coronatus)(稻錄病 );擬黑粉菌（Ustilaginoidea virens)(假黑穗病）；黃花狸藻（Utricularia aurea)(狸藻）；黃單胞菌（ Xanthomonas campestris)(十字花科黑腐病）；稻黃單胞菌稻小種（Xanthomonas oryzae pv. oryzae)(稻葉枯萎病）；Xiphinema (匕首線蟲）；Xiphinema americanum (匕首線蟲）；Xiphinema ifacolum (匕首線蟲）；Zeros o r i e n t a 1 i s ; Z u 1 i a entreriana o 本發明之其它態樣還包括施用本發明液體AL劑型之植物之保護組成物之方法。此等適當的標準方法爲熟悉此技術者所習知。一般，有利地可以把該植物之保護組成物裝於水溶性瓶罐、薄囊袋或其它容器中並置於稻田邊緣如此從特殊的搖動容器中逐滴加入，或者使用後背式噴灑器或類似的裝置來施用到水稻田的水面上來施用。【實施方式】 -38- (36) 200529745 本發明係使用如下實施例來顯示，但其內容不限於此等實例。 1 ·製備實例：AL (任何其它液體；立即可用溶液）劑型之植物之保護組成物-變化型1 ( AL1 ) 關於此點，係先製備活性物質濃縮液且然後將該活性物質濃縮液與該等溶劑及濕化劑混合在一起。; Trigonotylus ruficornis; Trogoderma granarium (trogoderma variabile); Tylenchorhynchus annulatus (short-line nematode); Tylenchorhynchus brevilineatus (Viburnum nematode) ; Typhaea stercorea (Hydrophyllum) •, Typhaula ishikariensis (White mold of P. spp.); Tyrophagus putrescentiae (Snake); Ulomoides dermestoides; Monospore rust (Uromyces coronatus) (rice disease); Ustilaginoidea virens (pseudosmut); Utricularia aurea (Utricularia); Xanthomonas campestris (Cruciferae) Black rot); Xanthomonas oryzae pv. Oryzae (rice leaf blight); Xiphinema (dagger nematode); Xiphinema americanum (dagger nematode); Xiphinema ifacolum (dagger nematode); Zeros orienta 1 is Z u 1 ia entreriana o Other aspects of the invention include a method of applying a plant protective composition of the liquid AL dosage form of the invention. These appropriate standard methods are known to those skilled in the art. Generally, it is advantageous to pack the plant protection composition in water-soluble bottles, thin sachets, or other containers and place them on the edge of the rice field so that they are added dropwise from a special shaking container, or using a back sprayer or similar The device is applied to the water surface of the rice field. [Embodiment] -38- (36) 200529745 The present invention is shown using the following examples, but the contents are not limited to these examples. 1 · Preparation example: AL (any other liquid; ready-to-use solution) dosage form of plant protection composition-Variation 1 (AL1) In this regard, an active substance concentrated solution is first prepared and then the active substance concentrated solution and the Wait for the solvent and wetting agent to mix together.

表1 . .1-製備：活性物質濃 ^縮液AL1 成份組成（g) 解說 Purasolv®EHL 650.00 乳酸2-乙基己酯愛西叵 30.00 (農業化學之）活性物質表1.2-製僱 ί :植物之保護組成物AL1 成份組成（g ) 解說活性物質濃縮液AL1 680.00 DMSO 3 00.0 溶劑 Break Thru OE 441® 20.00 濕化劑 2 .製備實例：AL (任何其它液體；立即可用溶液）劑型之植物之保護組成物-變化型2 ( AL2 ) 關於此點，係先製備活性物質濃縮液且然後將該活性物質濃縮液與該等溶劑及濕化劑混合在一起。 -39- (37) 200529745 表2.卜製備:活性物質濃縮液AL2 成份組成（g ) 解說 Purasolv®EHL 625.00 乳酸2 -乙基己酯 BPMC 200.00 (農業化學之）活性物質愛西叵 20.00 (農業化學之）活性物質表2.2-製備：植物之保護組成物AL2 成份組成（g ) 解說活性物質濃縮液AL2 845.00 DMSO 113.30 溶劑 Break Thru OE 44 1® 20.00 濕化劑 3 .製備實例：AL (任何其它液體；立即可用溶液）劑型之植物之保護組成物-變化型3 ( A L 3 ) 關於此點’係先製備活性物質濃縮液且然後將該活性物質濃縮液與該等溶劑及濕化劑混合在一起。表丄.1-製備丄活性物質濃縮液AL3 成份組成（g ) 解說 Purasolv®EHL 100.00 乳酸2-乙基己酯硫雙滅多威 25.00 (農業化學之）活性物質 -40- (38) 200529745 表3.2 -製備：植物之保護組成物A L 3 成份組成（g ) 解說活性物質濃縮液AL3 125.00 ---------- 苯甲醇 861.60 溶劑 Break Thru OE 440® 50.00 濕化劑 • 4·製備實例：AL (任何其它液體；立即可用溶液）劑型之植物之保護組成物-變化型4 ( AL4 ) 關於此點，係先製備活性物質濃縮液且然後將該活个生物質濃縮液與該等溶劑及濕化劑混合在一起。Table 1. .1-Preparation: Concentrated active substance ^ Shrinkage AL1 Ingredient composition (g) Explanation Purasolv® EHL 650.00 2-Ethylhexyl lactate Acetamine 30.00 (of agricultural chemistry) Active substance Table 1.2- Manufacturing employment: Plant Protective composition AL1 Ingredient composition (g) Explanation active substance concentrate AL1 680.00 DMSO 3 00.0 Solvent Break Thru OE 441® 20.00 Humidifier 2. Preparation example: AL (any other liquid; ready-to-use solution) dosage form of plant protection Composition-variant 2 (AL2) In this regard, an active substance concentrated solution is first prepared and then the active substance concentrated solution is mixed with these solvents and a wetting agent. -39- (37) 200529745 Table 2. Preparation: Ingredient composition of active substance concentrated liquid AL2 (g) Explanation of Purasolv® EHL 625.00 2-Ethylhexyl lactate BPMC 200.00 (of agricultural chemistry) Active substance azepam 20.00 (Agrochemical Of) Active Substances Table 2.2-Preparation: Plant protection composition AL2 Ingredient composition (g) Interpretation of active substance concentrate AL2 845.00 DMSO 113.30 Solvent Break Thru OE 44 1® 20.00 Humidifier 3. Preparation example: AL (Any other liquid ; Ready-to-use solution) plant protection composition of dosage form-Variation 3 (AL 3) In this regard, 'the active substance concentrate is first prepared and then the active substance concentrate is mixed with these solvents and wetting agents . Table 丄 .1- Preparation 丄 Active Substance Concentrate AL3 Ingredient Composition (g) Explain Purasolv® EHL 100.00 2-Ethylhexyl Lactate Thiodifencarb 25.00 (Agrochemical) Active Substances 40- (38) 200529745 Table 3.2 -Preparation: Plant protection composition AL 3 Ingredient composition (g) Interpretation of active substance concentrate AL3 125.00 ---------- Benzyl alcohol 861.60 Solvent Break Thru OE 440® 50.00 Humidifier • 4 · Preparation examples : AL (any other liquid; ready-to-use solution) plant protection composition in a dosage form-Variant 4 (AL4) In this regard, the active substance concentrate is first prepared and then the living biomass concentrate and the solvents are prepared And humidifier.

表4.1-製備：活性物質濃 [縮液AL4 成份組成（g ).. 解說 Purasolv®EHL 100.00 乳酸2 -乙基己酯硫雙滅多威 30.00 (農業化學之）活性物質表4.2-製備：植物之保護組成物AL4 成份組成（g ) 解說活性物質濃縮液AL4 130.00 苯甲醇 863.50 溶劑 Break Thru OE 440® 50.00 濕化劑 -41- (39) 200529745 5 ·製備實例：AL (任何其它液體；立即可用溶液）劑型之植物之保護組成物-變化型5 ( AL 5 ) 關於此點’係先製備活性物質濃縮液且然後將該活性物質濃縮液與該等溶劑及濕化劑混合在一起。表5.1-製備：活性物質濃【縮液AL5 成份組成（g ) 解說 Purasol v®EHL 100.00 乳酸2-乙基己酯硫雙滅多威 30.00 (農業化學之）活性物質愛西叵 7.50 (農業化學之）活性物質表5.2-製備：植物之保護組成物AL 5 成份組成（g ) 解說活性物質濃縮液A L 5 137.50 苯甲醇 854.00 溶劑 Break Thru 0E 440® 50.00 濕化劑Table 4.1-Preparation: Concentrated active substance [Condensate AL4 Ingredient composition (g) .. Explain Purasolv® EHL 100.00 2-Ethylhexyl lactate Thiopenthol 30.00 (agrochemical) Active substance Table 4.2-Preparation: Plant Protective composition AL4 Ingredient composition (g) Explanation of active substance concentrate AL4 130.00 Benzyl alcohol 863.50 Solvent Break Thru OE 440® 50.00 Humidifier-41- (39) 200529745 5 · Preparation example: AL (Any other liquid; ready-to-use solution ) Protective composition of plants in a dosage form-Variant 5 (AL 5) In this regard, an active substance concentrated solution is first prepared and then the active substance concentrated solution is mixed with the solvent and the wetting agent. Table 5.1- Preparation: Concentrated active substance [condensed AL5 Ingredient composition (g) Explanation Purasol v® EHL 100.00 2-Ethylhexyl lactate thiodifendicarb 30.00 (of agricultural chemistry) Active substance Azadirachtin 7.50 (of agricultural chemistry) Active Substances Table 5.2-Preparation: Plant Protection Composition AL 5 Ingredient Composition (g) Explanation of Active Substance Concentrate AL 5 137.50 Benzyl Alcohol 854.00 Solvent Break Thru 0E 440® 50.00 Humidifier

6 ·製備實例：AL (任何其它液體；立即可用溶液）劑型之植物之保護組成物-變化型6 ( AL6) 關於此點，係先製備活性物質濃縮液且然後將該活性物質濃縮液與該等溶劑及濕化劑混合在一起。 -42 - (40) 200529745 表6 · 1 •製備：活性物質濃 E縮液AL6 成份組成（g ) 解說 Purasolv®EHL 1 00.00 乳酸2-乙基己酯硫雙滅多威 20.00 (農業化學之）活性物質愛西叵 5.00 (農業化學之）活性物質表6.2-製備：植物之保護組成物AL6 成份組成（g ) 解說活性物質濃縮液AL6 125.00 苯甲醇 861.20 溶劑 Break Thru OE 440® 50.00 濕化齊!！ 7 ·製備實例：GR (顆粒）劑型之植物之保護組成物_ 變化型1 ( GR1 ) 關於此點，係先製備活性物質濃縮液且然後將該活性物質濃縮液吸附到一種惰性物質上。 -43- (41) 200529745 表7.1-製備：活性物質濃縮液GR1 成份濃度（重量％ ) 解說 Purasolv®EHL 16.7 乳酸2-乙基己酯愛西叵 6.7 (農業化學之）活性物質 Hallcomid M8-1 0⑧ 76.6 溶劑表7.2-製備：植物之保護組成物GR1 成份濃度（重量％ ) 解說活性物質濃縮液GR1 15 Sepiolite 3 0/60 篩孔 ® 85 惰性物質6 · Preparation Example: AL (Any other liquid; ready-to-use solution) plant protection composition in a dosage form-Variant 6 (AL6) In this regard, an active substance concentrated solution is first prepared and then the active substance concentrated solution and the Wait for the solvent and wetting agent to mix together. -42-(40) 200529745 Table 6 · 1 • Preparation: Concentrated active substance AL6 Condensate AL6 Ingredient composition (g) Explain Purasolv® EHL 1 00.00 2-Ethylhexyl lactate thiodifendicarb 20.00 (of agricultural chemistry) Activity Substance Acetone 5.00 (of agricultural chemistry) Active substance table 6.2-Preparation: Plant protection composition AL6 Ingredient composition (g) Explain active substance concentrated liquid AL6 125.00 Benzyl alcohol 861.20 Solvent Break Thru OE 440® 50.00 Humidification !!!! 7 · Preparation example: GR (granular) dosage form of plant protection composition _ Variation 1 (GR1) In this regard, the active substance concentrate is first prepared and then the active substance concentrate is adsorbed onto an inert substance. -43- (41) 200529745 Table 7.1- Preparation: Concentration of Active Material Concentrate GR1 (% by weight) Explanation of Purasolv® EHL 16.7 2-Ethylhexyl Lactate Acetyl 6.7 (Agrochemical) Active Substance Hallcomid M8-1 0⑧ 76.6 Solvents Table 7.2-Preparation: Plant Protection Composition GR1 Ingredient Concentration (% by Weight) Interpretation of Active Material Concentrate GR1 15 Sepiolite 3 0/60 Sieve® 85 Inert Substance

8 .製備實例：GR (顆粒）劑型之植物之保護組成物-變化型2 ( GR2 ) 關於此點，係先製備活性物質濃縮液且然後將該活性物質濃縮液吸附到一種惰性物質上。表8.1-製' 備：活性物質濃縮液GR2 成份濃度（重量％) 解說 Purasol v®EHL 50 乳酸2-乙基己酯愛西叵 5 (農業化學之）活性物質 DMS0 45 溶齊!1 -44 - (42) 200529745 孝8.2-製備：植物之保護組成物GR2 成份濃度（重量％) 解說活性物質濃縮液GR2 2 單丙二醇 4 佐劑 Biodac載體20/10篩孔⑧ 94 惰性物質 9 .製備實例：EC (可乳化濃縮液）劑型之植物之保護組成物關於此點’係先製備活性物質濃縮液且然後將該活性物質濃縮液與乳化劑混合在一起。8. Preparation example: GR (granular) dosage form of plant protection composition-variant 2 (GR2) In this regard, an active substance concentrated solution is first prepared and then the active substance concentrated solution is adsorbed onto an inert substance. Table 8.1- Preparation: Preparation: Active ingredient concentrated solution GR2 Ingredient concentration (% by weight) Explanation of Purasol v®EHL 50 2-ethylhexyl lactate Azadirachtin 5 (of agricultural chemistry) Active substance DMS0 45 Soluble! 1 -44- (42) 200529745 Xiao 8.2- Preparation: Plant protection composition GR2 component concentration (% by weight) Interpretation of active substance concentrate GR2 2 Monopropylene glycol 4 Adjuvant Biodac carrier 20/10 sieve ⑧ 94 Inert substance 9. Preparation example: EC (Emulsifiable concentrate) The protective composition of the plant in this dosage form is to prepare an active substance concentrate and then mix the active substance concentrate with the emulsifier.

表9 · 1 -製備：活性物質濃縮液£ C 成份組成（g ) 解說 Purasolv®EHL 150.0 乳酸2·乙基己酯溴氰菊酯 25.00 (農業化學之）活性物質 Solvesso 10 0® 645.9 溶劑 -45- (43) 200529745Table 9 · 1-Preparation: Concentrated active substance £ C Composition (g) Explanation Purasolv® EHL 150.0 2. Ethylhexyl lactate Deltamethrin 25.00 (agrochemical) Active substance Solvesso 10 0 645.9 Solvent-45 -(43) 200529745

表9.2 -製備：植物之保護組成物E C 成份組成（g ) 解說活性物質濃縮液EC 820.9 醋酸 0.1 活性物質安定劑 BHT 1.0 活性物質安定劑 Emulsogen EL 3 60® 2 1.0 非離子性乳化劑十二烷基苯-磺酸鈣 49.0 陰離子性乳化劑 1 〇·製備實例：EW (水包油乳液）劑型之植物之保護組成物關於此點’係先製備活性物質濃縮液且然後將該活性物質濃縮液於水中乳化。然後把該濃縮之乳液安定化。Table 9.2-Preparation: Plant protection composition EC Ingredient composition (g) Explain active substance concentrate EC 820.9 Acetic acid 0.1 Active substance stabilizer BHT 1.0 Active substance stabilizer Emulsogen EL 3 60® 2 1.0 Nonionic emulsifier dodecane Benzene-calcium sulfonate 49.0 Anionic emulsifier 1 〇 · Preparation Example: Plant protection composition of EW (oil-in-water emulsion) dosage form In this regard, an active substance concentrate is first prepared and then the active substance concentrate is prepared Emulsified in water. The concentrated emulsion is then stabilized.

表1 0.1-製赛：活性物質濃縮液EW 成份組成（g ) 解說 Purasol v ⑧ EHL 50.0 乳酸2 -乙基己酯溴氰菊酯 12.50 (農業化學之）活性物質環己酮 125.00 溶劑苯甲酸苯甲酯 125.00 溶劑 -46- (44) (44)200529745 表10.2-製備 i :植物之保護組成物EW 成份組成（g) 解說活性物質濃縮液EW 3 12.50 Methyl paraben® 0.1 保存劑 Propyl paraben® 0.1 保存劑 Empiphos 03 D® 10.00 陰離子性乳化劑 Witconol NS 500K® 17.50 非離子性乳化劑 Genapol X060® 17.50 非離子性乳化劑聚乙烯吡咯啶酮 15.00 流動安定劑 K90® 檸檬酸 0.20 活性物質安定劑 Rhodorsil 416® 0.20 消泡劑 Rhodorsil 426R® 0.20 消泡劑單丙二醇 120.00 抗凍劑水 525.00Table 1 0.1-Making: Composition of active substance concentrated solution EW (g) Explanation Purasol v ⑧ EHL 50.0 2-Ethylhexyl lactate deltamethrin 12.50 (of agricultural chemistry) Active substance cyclohexanone 125.00 Solvent benzoate Methyl ester 125.00 Solvent-46- (44) (44) 200529745 Table 10.2- Preparation i: Plant protection composition EW Ingredient composition (g) Interpretation of active substance concentrate EW 3 12.50 Methyl paraben® 0.1 Preservative Propyl paraben® 0.1 Preservation Empiphos 03 D® 10.00 Anionic emulsifier Witconol NS 500K® 17.50 Nonionic emulsifier Genapol X060® 17.50 Nonionic emulsifier Polyvinylpyrrolidone 15.00 Flow stabilizer K90® Citric acid 0.20 Active substance stabilizer Rhodorsil 416® 0.20 Antifoam Rhodorsil 426R® 0.20 Antifoam Monopropylene Glycol 120.00 Antifreeze Water 525.00

1 1 ·製備實例：ME (微乳液）劑型之植物之保護組成物關於此點，係先製備活性物質濃縮液且然後將該活性物質濃縮液於水中乳化以形成微乳液。 -47- (45) 2005297451 1 Preparation example: ME (microemulsion) plant protection composition in dosage form In this regard, an active substance concentrate is first prepared and then the active substance concentrate is emulsified in water to form a microemulsion. -47- (45) 200529745

表11.卜製備：活性物質濃縮液ME 成份組成（g ) 解說 P11 r a S ο 1 V ⑧ E H L 50.0 乳酸2-乙基己酯溴氰菊酯 12.50 (農業化學之）活性物質茴香醚 236.00 溶劑環己酮 139.00 溶劑Table 11. Preparation: ME composition of active substance concentrate (g) Explanation P11 ra S ο 1 V ⑧ EHL 50.0 2-ethylhexyl lactate deltamethrin 12.50 (of agricultural chemistry) active substance anisole 236.00 solvent ring Hexone 139.00 solvent

表1 1 . 2 -製備··植物之保護組成物Μ E 成份組成（g ) 解說活性物質濃縮液Μ E 445.00 _ 檸檬酸 0.20 活性物質安定劑 — 己二醇 130.00 抗凍劑 S 〇 p r 〇 p h 〇 r B S U ® 144.00 非離子性乳化劑 Soprophor 4D384® 36.00 陰離子性乳化劑一水 254.80 1 2 ·製備實例：EG (可乳化顆粒）劑型之植物之保護組成物關於此點，係先製備活性物質濃縮液。接著在一粒化裝置中將該活性物質濃縮液之乳液噴在惰性物質上。 -48 - (46) 200529745Table 1 1.2-Preparation · Plant protection composition M E Ingredient composition (g) Interpretation of active substance concentrated solution M E 445.00 _ Citric acid 0.20 Active substance stabilizer-Hexanediol 130.00 Antifreeze S 〇pr 〇ph 〇r BSU ® 144.00 Nonionic emulsifier Soprophor 4D384® 36.00 Anionic emulsifier monohydrate 254.80 1 2 · Preparation example: EG (emulsifiable granule) dosage form of plant protection composition In this regard, the active substance is first concentrated liquid. The emulsion of the active substance concentrate is then sprayed onto an inert substance in a granulating device. -48-(46) 200529745

表12.1-製備：活性物質濃縮液EG 成份組成（g ) 解說 Purasol v®EHL 3.3 乳酸2-乙基己酯溴氰菊酯 11.0 (農業化學之）活性物質 S ο 1 v e s s 〇 2 0 0® 45.1 溶劑磷酸三丁酯 40.7 溶劑表12.2-製備〖：植物之保護 [組成物EG 成份濃度（重量％) 解說活性物質濃縮液E G 45.50 Mowiol 3-83® 27.50 惰性物質 Mowiol 4-88® 13.50 惰性物質分散劑 1 494® 11.00 分散劑十二烷基苯-磺酸鈣 0.55 陰離子性乳化劑檸檬酸 0.35 活性物質安定劑 Rhodorsil 4 16® 0.30 消泡劑 Rhodorsil 426R® 0.30 消泡劑水 525.00 濕化 1 3 ·製備實例：SE (懸浮乳液）劑型之植物之保護組成物關於此點’係先製備活性物質濃縮液。然後將該活性物質濃縮液之乳液於含有一種第二農業化學之活性物質之 -49- (47) 200529745 水性組成物中微粒化，從而分散其固態顆粒。Table 12.1-Preparation: Active Ingredient Concentrated Liquid EG Ingredient Composition (g) Explanation of Purasol v® EHL 3.3 2-ethylhexyl lactate deltamethrin 11.0 (of agricultural chemistry) Active substance S ο 1 vess 〇 2 0 0® 45.1 Solvent Tributyl Phosphate 40.7 Solvent Table 12.2-Preparation :: Plant protection [Composition EG Ingredient Concentration (% by weight) Explanation of active substance concentrate EG 45.50 Mowiol 3-83® 27.50 Inert substance Mowiol 4-88® 13.50 Inert substance dispersion Dispersant 1 494® 11.00 Dispersant dodecylbenzene-calcium sulfonate 0.55 Anionic emulsifier citric acid 0.35 Active substance stabilizer Rhodorsil 4 16® 0.30 Antifoam Rhodorsil 426R® 0.30 Antifoam water 525.00 Humidity 1 3 · Preparation example: SE (suspension emulsion) dosage form of plant protection composition. In this regard, the active substance concentrate is first prepared. The emulsion of the active substance concentrate is then micronized in an aqueous composition containing -49- (47) 200529745, a second agrochemical active substance, thereby dispersing its solid particles.

表1 3 . 1 -製備：活性物質濃縮液S E 成份組成（g ) 解說 Purasol v® EHL 150.00 乳酸2-乙基己酯溴氰菊酯 10.00 (農業化學之）活性物質乙醯苯 50.00 溶劑Table 1 3.1-Preparation: Active substance concentrate S E Ingredient Composition (g) Explanation Purasol v® EHL 150.00 2-Ethylhexyl lactate Deltamethrin 10.00 (of agrochemical) Active substance Acetylbenzene 50.00 Solvent

表13.2-製備：植物之保護組成物SE 成份組成（g ) 解說活性物質濃縮液S E 2 10.0 愛西叵 100.00 (農業化學之）第二活性物質 Soprophor FLK® 50.00 分散劑 Rhodopol G® 2.75 增稠劑 Proxel GXL® 1.00 保存劑 Rhodorsil 416® 5.00 消泡劑單丙二醇 60.00 抗凍劑 Geropon SDS® 15.00 濕化劑醋酸 0.10 活性物質安定劑 ΒΗΤ 0.40 活性物質安定劑 Soprophor BSU® 25.00 非離子性乳化劑水 540.75 -50- (48) 200529745 1 4 ·製備實例·· S L (可溶性濃縮液）劑型之植物之保護組成物關於此點，係先製備活性物質濃縮液且然後將該活性物質濃縮液與該等溶劑及界面活性劑混合在一起。Table 13.2-Preparation: Plant protection composition SE Ingredient composition (g) Interpretation of active substance concentrated liquid SE 2 10.0 Acetone 100.00 (of agricultural chemistry) Second active substance Soprophor FLK® 50.00 Dispersant Rhodopol G® 2.75 Thickener Proxel GXL® 1.00 Preservative Rhodorsil 416® 5.00 Defoamer Monopropylene glycol 60.00 Antifreeze Geropon SDS® 15.00 Humidifier Acetic acid 0.10 Active substance stabilizer BΗΤ 0.40 Active substance stabilizer Soprophor BSU® 25.00 Nonionic emulsifier water 540.75 -50 -(48) 200529745 1 4 · Preparation examples ·· SL (Soluble Concentrate) dosage form of plant protection composition In this regard, the active substance concentrate is first prepared and then the active substance concentrate and these solvents and interfaces The active agents are mixed together.

表14.1-製備：活性物質濃縮液SL 成份組成（g ) 解說 Purasol v®EHL 25.00 乳酸2-乙基己酯乙醯米皮敵 125.00 (農業化學之）活性物質表14.2-製備：植物之保言| 1組成物SL 成份組成（g ) 解說活性物質濃縮液SL 150.0 DMSO 3 20.00 溶劑 7 -丁內酯 115.00 溶劑苯甲醇 3 00.00 溶劑 Synperonic A3 ® 120.00 界面活性劑 Soprophor DSS 15® 80.00 界面活性劑Table 14.1-Preparation: Active ingredient concentrate SL Ingredient composition (g) Explanation Purasol v® EHL 25.00 2-Ethylhexyl lactate Ethylpyridine 125.00 (of agricultural chemistry) Table 14.2-Preparation: Plant guarantee 1 Composition SL Ingredient Composition (g) Interpretation of active substance concentrate SL 150.0 DMSO 3 20.00 Solvent 7-butyrolactone 115.00 Solvent benzyl alcohol 3 00.00 Solvent Synperonic A3 ® 120.00 Surfactant Soprophor DSS 15® 80.00 Surfactant

於如上實施例中係使用如下成份：Purasolv® EHL ( 乳酸 2 -乙基己醋；Purac Biochem, Gorinchem，紐西蘭或巴賽隆納，西班牙），愛西叵（通稱），DMSO ( Kuhn -51 - (49) 200529745In the above example, the following ingredients were used: Purasolv® EHL (2-ethylhexyl lactate; Purac Biochem, Gorinchem, New Zealand or Barcelona, Spain), Ezekiel (general name), DMSO (Kuhn-51 -(49) 200529745

C h e m i e / Interorgana，漢堡，德國）’ Break Thru OE 441® (聚二甲基矽氧烷；Goldschmidt，Essen，德國）， BPMC (通稱），硫雙滅多威（通稱），苯甲醇（不同供應商），Break Thru OE 440® (聚二甲基砂氧燒； Goldschmidt，Essen,德國），H a 11 c o m i d Μ 8 - 1 0 ® ( C P H a 11 ，芝力口哥，美國），Sepiolite 30/60 mesh® (Tolsa SA，馬德里，西班牙），單丙二醇（Sigma-aldrich， Taufdirchen，德國），Biodax Carrier 20/40 mesh® (芳香族烴流體；Exxon，Co longue，德國），醋酸（不同供應商 )，：BHT (丁基化羥基甲苯；Fluka，德國），Emulsogen EL 3 6 0® (脂肪酸聚二醇酯；Clariant，法蘭克福，德國），十二烷基苯-磺酸鈣（化學基團；如Akzo Novel，Duren ，德國），環己酮（Sigma-Aldrich，Taufkirchen，德國），苯甲酸苯甲酯（Sigma-Aldrich，Taufkirchen，德國）， Methyl paraben® ( Chemag，法蘭克福，德國），Propyl paraben® ( Chemag，法蘭克福，德國），Empiphos 03D® (複合有機磷酸醋；Huntsman，Neu-Isenbur，德國），Witconol NS 500 K® (聚氧乙烯聚氧丙烯嵌段共聚物； Osi/Akzo Nobel，法蘭克福，德國），Genapol X060® (乙氧基化醇；Clariant，法蘭克福，德國），聚乙烯吡咯啶嗣 K 90 ⑧（syn. Luviskol K 9 0 i BASF，Ludwigshafen，德國），醋酸（不同供應商），Rhodorsil 4 1 6® (消泡劑； Rhodia，法蘭克福，德國），Rh o d o r s i 1 4 2 6 ® (消泡劑； Rhodia，法蘭克福，德國），茴香醚（如 Rh o d i a s ο 1 v -52- (50) 200529745C hemie / Interorgana, Hamburg, Germany) 'Break Thru OE 441® (Polydimethylsiloxane; Goldschmidt, Essen, Germany), BPMC (general name), thiodicarb (general name), benzyl alcohol (different suppliers ), Break Thru OE 440® (Polydimethyl Sand Oxygen Burning; Goldschmidt, Essen, Germany), Ha 11 comid Μ 8-1 0 ® (CPH a 11, Zerichot, USA), Sepiolite 30/60 mesh® (Tolsa SA, Madrid, Spain), monopropylene glycol (Sigma-aldrich, Taufdirchen, Germany), Biodax Carrier 20/40 mesh® (aromatic hydrocarbon fluids; Exxon, Co longue, Germany), acetic acid (different suppliers) : BHT (butylated hydroxytoluene; Fluka, Germany), Emulsogen EL 3 6 0® (fatty acid polyglycol ester; Clariant, Frankfurt, Germany), dodecylbenzene-calcium sulfonate (chemical group; eg Akzo Novel, Duren, Germany), cyclohexanone (Sigma-Aldrich, Taufkirchen, Germany), benzyl benzoate (Sigma-Aldrich, Taufkirchen, Germany), Methyl paraben® (Chemag, Frankfurt, Germany), Propyl para ben® (Chemag, Frankfurt, Germany), Empiphos 03D® (complex organic phosphate vinegar; Huntsman, Neu-Isenbur, Germany), Witconol NS 500 K® (polyoxyethylene polyoxypropylene block copolymer; Osi / Akzo Nobel, Frankfurt, Germany), Genapol X060® (ethoxylated alcohol; Clariant, Frankfurt, Germany), polyvinylpyrrolidine 嗣 K 90 ⑧ (syn. Luviskol K 9 0 i BASF, Ludwigshafen, Germany), acetic acid (different suppliers ), Rhodorsil 4 1 6® (defoamer; Rhodia, Frankfurt, Germany), Rh odorsi 1 4 2 6 ® (defoamer; Rhodia, Frankfurt, Germany), anisole (such as Rh odias ο 1 v -52- (50) 200529745

MPE® ; Rhodia，法蘭克福，德國），己二醇（Sigma-Aldrich，T aufkir chen，德國)，S opropho r BSU® (三苯乙細酉分+16 EO，Rhodia’法蘭克福’德國），Solvesso 2 0 0 ® (芳香族煙流體；Ε χ χ ο η，C ο 1 ο n g n e，德國），磷酸三丁酯（如Merck (默克）或Bayer (拜耳），德國）， Mowiol 3-83®(Kuraray，法蘭克福，德國），Mowiol4-88® ( Kuraray，法蘭克福，德國），分散劑 1 494® ( Clariant;法蘭克福’德國）’乙酸苯（Haarmann & Reimer，Holzminden，德國），Soprophor FLK® (聚芳基烷氧基磷酸酯鉀鹽；Rhodia，法蘭克福，德國）， Rhodopol G® ( Rhodia，法蘭克福，德國），Proxel GXL® (A vecia，法蘭克福，德國），G e r ρ ο n S D S ® (硫琥珀酸二辛酯；Rhodia，法蘭克福，德國），醋酸（不同供應商 )，乙醯米皮敵（通稱），7 -丁內酯（Sigma-Aldrich， Taufkirchen，德國），Synperonic A3® (合成性初級醇環氧乙烯縮合物；Uniqema，Everberg，比利時）， Soprophor DSS 15® (乙氧基二苯乙嫌酣；Rhodia，法蘭克福，德國）。 1 5 ·生物性實施例1 :溫室實驗結果步驟：測試調合物AL 1及AL2 (其製備及組成參見製備例1 及 2 )。所防治之水稻田害蟲爲稻蟬：稻褐飛虱（ Nil ap arv ata lu gens )(褐背稻跳蟲；BPH )。 -53- (51) (51)200529745 每次，在實驗開始以前以每盆4 0 - 5 0株稻苗（水稻、（ Oryza sativa ;品種；Balilla ))之密度將稻苗置於標準土 (ED73)中先培養10天。在施藥前一天，先用石英砂覆蓋土壤表面且把盆器放置到夠深的容器中，接著加λ自來水使水深高於土壤表面（盆器頂緣）。然後在每盆中置入約5 0隻稻蟬（發育期：蛹後期到成蟲初期）。接著把所有的東西用有孔的塑膠袋覆蓋。在稻蟬移居到植物體後，逐漸地用水加滿容器直到水超過土壤表面（盆器頂緣）。當水的總面積量達到既定的面積値（平方公分）時則已達到實驗所需之水量。施藥的方法係吸取固定份量的組成物然後加到水面上來進行。測試的劑量相當於3、4及5公升/公頃（1/ha) 。如下個別結果係用4個含有稻株之盆器重覆實驗兩次後所得結果。在施用後第1、4、7及13天（DA A )進行評估。關於此點，係測量活的稻蟬數目且然後（使用 Henderson-Tilton公式）計算有效度（％ )。結果 -54- (52) 200529745 表1 5 -防治稻褐飛虱的活性（BPH ) 調合劑量評估後物 1/ha 〇DAA(§) 1 DAA 4 DAA 7 DAA 13 \A Φ NO. Φ Φ % Φ φ % Φ Φ % φ NO. Φ % NO· NO. NO. 未處 - 290 290 0.0 285 0.0 148 0.0 800(*) 0.0 理 AL1 5 242.5 10 95.9 0 100.0 0 100.0 0 100.0 4 295 85 71.8 0 100.0 0 100.0 0 100.0 3 250 97.5 61.0 0 100.0 0 100.0 0 100.0 AL2 5 255 1.5 99.4 0 100.0 0 100.0 0 100.0 4 270 6 97.8 0 100.0 0 100.0 0 100.0 3 305 10 96.7 0 100.0 0 100.0 0 100.0MPE®; Rhodia, Frankfurt, Germany), Hexylene glycol (Sigma-Aldrich, Taufkirchen, Germany), Sopropho r BSU® (triphenylethyl trioxide +16 EO, Rhodia 'Frankfurt' Germany), Solvesso 2 0 0 ® (aromatic smoke fluid; Ε χ χ ο η, C ο 1 ο ngne, Germany), tributyl phosphate (such as Merck or Bayer, Germany), Mowiol 3-83® ( Kuraray, Frankfurt, Germany), Mowiol4-88® (Kuraray, Frankfurt, Germany), dispersant 1 494® (Clariant; Frankfurt 'Germany)' benzene acetate (Haarmann & Reimer, Holzminden, Germany), Soprophor FLK® (Polymer Aryl alkoxy phosphate potassium salt; Rhodia, Frankfurt, Germany), Rhodopol G® (Rhodia, Frankfurt, Germany), Proxel GXL® (Avecia, Frankfurt, Germany), Ger ρ ο n SDS ® (sulfur amber Dioctyl Ester; Rhodia, Frankfurt, Germany), Acetic Acid (different suppliers), Etomidate (general name), 7-Butyrolactone (Sigma-Aldrich, Taufkirchen, Germany), Synperonic A3® (Synthetic Primary Alcohol epoxy Ethylene condensates; Uniqema, Everberg, Belgium), Soprophor DSS 15® (ethoxydiphenylethylsulfanyl; Rhodia, Frankfort, Germany). 1 5 · Biological Example 1: Greenhouse Experiment Results Steps: Test the blends AL 1 and AL 2 (for preparation and composition, see Preparation Examples 1 and 2). The rice field pests to be controlled are rice cicadas: rice brown planthoppers (Nil ap arv ata lu gens) (Brownback rice hopper; BPH). -53- (51) (51) 200529745 Each time, before the beginning of the experiment, the rice seedlings were placed in a standard soil (at a density of 40-50 rice seedlings (rice, (Oryza sativa; variety; Balilla)) per pot. ED73). One day before the application, cover the soil surface with quartz sand and place the pot in a sufficiently deep container, and then add lambda tap water to make the water depth higher than the soil surface (top edge of the pot). Then about 50 rice cicadas were placed in each pot (development stage: late pupal stage to early adult stage). Then cover everything with a perforated plastic bag. After the rice cicada migrates to the plant body, gradually fill the container with water until the water exceeds the soil surface (top edge of the pot). When the total area of water reaches a predetermined area 値 (cm 2), the amount of water required for the experiment has been reached. The application method is to take a fixed amount of the composition and add it to the water surface. Tested doses are equivalent to 3, 4 and 5 liters per hectare (1 / ha). The following individual results are obtained by repeating the experiment twice with four pots containing rice plants. Evaluation was performed on days 1, 4, 7, and 13 (DA A) after administration. At this point, the number of live rice cicadas is measured and then (using the Henderson-Tilton formula) the validity (%) is calculated. Results-54- (52) 200529745 Table 1 5-Activity against rice brown planthopper (BPH) After the assessment of the mixed dose 1 / ha 〇 DAA (§) 1 DAA 4 DAA 7 DAA 13 \ A Φ NO. Φ Φ% Φ φ% Φ Φ% φ NO. Φ% NO · NO. NO. Not treated-290 290 0.0 285 0.0 148 0.0 800 (*) 0.0 Physical AL1 5 242.5 10 95.9 0 100.0 0 100.0 0 100.0 4 295 85 71.8 0 100.0 0 100.0 0 100.0 3 250 97.5 61.0 0 100.0 0 100.0 0 100.0 AL2 5 255 1.5 99.4 0 100.0 0 100.0 0 100.0 4 270 6 97.8 0 100.0 0 100.0 0 100.0 3 305 10 96.7 0 100.0 0 100.0 0 100.0

(§)=施藥前數目；Φ No. =平均數；Φ % =平均有效度 (* )有稻蟬後代出現(§) = number before application; Φ No. = average; Φ% = average effectiveness (*) There are offspring of rice cicada

解說：可以得知在兩種AL調合物中該農業化學之活性物質愛西叵防治害蟲稻褐飛虱的快速效果（1 DAA後）及長期效果（於13 DAA )。】6.生物性實例2 :關於植物損害之溫室實驗結果步驟（參考生物性實例1 ); 植物的損害係在施用後第7及1 3天（DAA )後測定 -55- 200529745 (53) 。係以稻株的生長及外表型狀態來評估植物損害的％ (關於此點，高％値係表示有嚴重的植物損害）。表16-植物損害％調合物劑量 7DAA後的評分 13 DAA後的評分 1/ha Rep.A Rep.B Φ% Rep.A Rep.B Φ% 未處理 20 15 17.5 (§) 25 25 25 (§) AL1 5 2 1 1.5 2 1 1.5 4 3 2 2.5 3 2 2.5 3 0 1 0.5 0 1 0.5 AL2 5 5 3 4 4 6 5 4 1 2 1.5 1 2 1.5 3 0 2 1 0 2 1Commentary: We can know the rapid effect (after 1 DAA) and long-term effect (after 13 DAA) of the active substance of agrochemicals in two AL blends on the control of the pest rice brown planthopper. [6] Biological Example 2: Results of greenhouse experiments on plant damage (refer to Biological Example 1); Plant damage was measured after 7 and 13 days (DAA) after application -55- 200529745 (53). The percentage of plant damage was evaluated based on the growth and phenotypic status of rice plants (at this point, a high% indica line indicates severe plant damage). Table 16-Plant damage% Blend dose 7DAA score 13 DAA score 1 / ha Rep.A Rep.B Φ% Rep.A Rep.B Φ% Untreated 20 15 17.5 (§) 25 25 25 (§ ) AL1 5 2 1 1.5 2 1 1.5 4 3 2 2.5 3 2 2.5 3 0 1 0.5 0 1 0.5 AL2 5 5 3 4 4 6 5 4 1 2 1.5 1 2 1.5 3 0 2 1 0 2 1

Rep ·=重覆實驗；φ % =諸重覆實驗的平均値；（§ )=可偵測的生長抑制量在溫室實驗中兩種測試的AL調合物被證明對於測試稻作具有良好的耐受性。 1 7 ·生物性實驗3 :田野實驗結果步驟：調合物AL1 (其製備及組成可參考製備例1 )係與標準E C調合物進行比較來測試：A L 1含有3重量％的愛西叵且分別以每公頃5 0克（劑量1 )，8 3克（劑量2 )、 -56- 200529745 (54) 117克（劑量3)及150克（劑量4)來施用，而標準ec 則含有1 〇重量％愛西叵且分別以每公頃1 5克（劑量1 ) 、25克（劑量2 ) 、35克（劑量3 )及45克（劑量4 )來施用，在每組劑量1到4中皆含有同樣份量之農業化學之 * 活性物質愛西叵。，田野實驗的位置係在中國的江蘇（JiangSu) -RF，Rep · = repeated experiments; φ% = average 値 of repeated experiments; (§) = detectable growth inhibition. In the greenhouse experiments, the two tested AL blends proved to be well tolerant to the tested rice crops. Accepted. 17 · Biological Experiment 3: Field Experiment Results Steps: The blend AL1 (the preparation and composition can be referred to Preparation Example 1) is compared with the standard EC blend to test: AL 1 contains 3% by weight of azepam and 50 g (dose 1), 83 g (dose 2), -56- 200529745 (54) 117 g (dose 3) and 150 g (dose 4) per hectare are applied, while the standard EC contains 10% by weight Izepam is administered at 15 grams (dose 1), 25 grams (dose 2), 35 grams (dose 3), and 45 grams (dose 4) per hectare, and contains the same amount in each group of doses 1 to 4. Of Agricultural Chemistry * Active Substance Azadirachta. The location of the field experiment is in Jiangsu (JiangSu) -RF,

HuN-IPP及Xinshan-CQ。含有活性物質的調合物係以後背，式噴灑器用手噴灑來施用在水稻田中。實驗區塊的規格係採用RC B的方法每次以3 0平方米的實驗區塊來進行。如下每個位置的個別實驗結果皆是重覆3次的結果。所防治的水稻田之害蟲爲稻褐飛虱（Nilaparvata lugens )(褐背稻跳蟲；BPH )及白背飛虱（Sogatella furcifera )(白背跳蟲；WBPH )，其本來就在該等實驗位置處自然地大量存在著。此外，還檢測其對常見蜘蛛的次級作用。HuN-IPP and Xinshan-CQ. The blend containing the active substance is applied to the paddy field by spraying with a hand sprayer. The specification of the experimental block is carried out using the RC B method with 30 square meters of experimental block at a time. The results of the individual experiments at each of the positions below are repeated three times. The pests of rice fields to be controlled are rice brown planthopper (Nilaparvata lugens) (Brownback rice planthopper; BPH) and whiteback planthopper (Sogatella furcifera) (Whiteback planthopper; WBPH). Locations naturally exist in large numbers. In addition, secondary effects on common spiders were tested.

• 害蟲防制結果或次級作用係在施藥不同天數後（DAT • )以防治％ (=與未經施藥的對照組比較後害蟲減少的數目 . )或次級作用％來表示。結果 · -57- (55) 200529745• Pest control results or secondary effects are expressed as% of control (= number of pest reductions compared to a non-applied control group) or% of secondary effects after different days of application (DAT). Results -57- (55) 200529745

表 17.1-位置：HuN-IPP 劑量調合物在以ΒΡΗ處理ί 麦之害蟲防治率 1 DAT 3DAT 7DAT 1 4DAT 21DAT 28DAT 1 AL1 78.1 96.7 92.1 98.0 99.2 97.6 標準EC 5 1.5 68.9 83.6 97.1 96.3 88.7 2 AL1 8 1.8 97.2 96.2 98.1 99.1 98.7 標準EC 64.0 76.9 90.7 97.8 97.4 96. 3 AL1 89.4 98.9 100 100 100 99.0 標準EC 76.9 89.6 96.8 99.2 97.6 96.2 4 AL1 90.9 100 100 100 100 99.7 標準EC 79.2 92.1 97.8 99.4 98.5 96.9 在2001年9月13日施藥；在以BPH處理以前的感Table 17.1-Position: HuN-IPP dose blends treated with ΒΡΗ wheat pest control rate 1 DAT 3DAT 7DAT 1 4DAT 21DAT 28DAT 1 AL1 78.1 96.7 92.1 98.0 99.2 97.6 Standard EC 5 1.5 68.9 83.6 97.1 96.3 88.7 2 AL1 8 1.8 97.2 96.2 98.1 99.1 98.7 Standard EC 64.0 76.9 90.7 97.8 97.4 96. 3 AL1 89.4 98.9 100 100 100 100 99.0 Standard EC 76.9 89.6 96.8 99.2 97.6 96.2 4 AL1 90.9 100 100 100 100 99.7 Standard EC 79.2 92.1 97.8 99.4 98.5 96.9 In 2001 Application on May 13; feeling before treatment with BPH

染平均値：3 23隻昆蟲/20堆土墩（=稻株群組） -58- 200529745 (56) 表17.2-位置：又丨115 1:^11??3-€(^ 劑量調合物在以WBPH處理後的害蟲防治率 1DAT 3DAT 7D AT 1 4DAT 21DAT 28DAT 1 AL1 43.9 52.2 75.5 68.1 49.1 33.2 標準EC 28.5 43.5 53.4 68.3 53.0 46.9 2 AL1 44.8 6 1.8 75.3 80.4 7 1.6 74.6 標準EC 30.1 49.9 72.5 75.8 58.9 65.1 3 AL1 45.6 62.4 79.1 80.6 61.9 5 1.9 標準EC 33.3 5 1.1 74.0 83.9 66.0 65.9 4 AL1 5 1.4 70.3 86.6 87.3 70.5 7 1.6 標準EC 36.9 5 1.1 8 1.1 8 1.7 75.0 69.8Dye average: 3 23 insects / 20 piles of mounds (= rice plant group) -58- 200529745 (56) Table 17.2-Position: again 丨 115 1: ^ 11 ?? 3- € (^ Dose blend in Pest control rate after treatment with WBPH 1DAT 3DAT 7D AT 1 4DAT 21DAT 28DAT 1 AL1 43.9 52.2 75.5 68.1 49.1 33.2 Standard EC 28.5 43.5 53.4 68.3 53.0 46.9 2 AL1 44.8 6 1.8 75.3 80.4 7 1.6 74.6 Standard EC 30.1 49.9 72.5 75.8 58.9 65.1 3 AL1 45.6 62.4 79.1 80.6 61.9 5 1.9 Standard EC 33.3 5 1.1 74.0 83.9 66.0 65.9 4 AL1 5 1.4 70.3 86.6 87.3 70.5 7 1.6 Standard EC 36.9 5 1.1 8 1.1 8 1.7 75.0 69.8

在2001年7月6日施藥；在以WB PH處理以前的感染平均値：9 8 3隻昆蟲/20堆土墩（=稻株群組） -59- 200529745 (57)Applied on July 6, 2001; average infection before treatment with WB PH: 9 8 3 insects / 20 mounds (= rice plant group) -59- 200529745 (57)

表 17.3 -位置：Jiang Su-RF 劑量調合物在以WBPH處理後的害蟲防治率 1DAT 3DAT 7DAT 1 4DAT 2 1 DAT 28DAT 1 AL1 37.8 47.2 61.3 70.2 63.8 標準EC 18.2 23.6 46.9 62.6 59.5 2 AL1 29.0 56.4 65.4 73.2 86.3 83.7 標準EC 4.6 25.9 36.4 38.6 58.3 53.9 3 AL1 19.4 42.8 49.6 73.8 83.8 76.6 標準EC 4.3 33.2 38.5 53.5 65.2 60.5 4 AL1 15.7 48.3 55.0 7 0.4 79.3 84.0 標準EC 7.8 43.2 45.1 6 1.8 68.3 75.3 在2001年8月8日施藥；在以WBPH處理以前的感Table 17.3-Location: Jiang Su-RF Dose Blends Pest Control Rate after Treatment with WBPH 1DAT 3DAT 7DAT 1 4DAT 2 1 DAT 28DAT 1 AL1 37.8 47.2 61.3 70.2 63.8 Standard EC 18.2 23.6 46.9 62.6 59.5 2 AL1 29.0 56.4 65.4 73.2 86.3 83.7 Standard EC 4.6 25.9 36.4 38.6 58.3 53.9 3 AL1 19.4 42.8 49.6 73.8 83.8 76.6 Standard EC 4.3 33.2 38.5 53.5 65.2 60.5 4 AL1 15.7 48.3 55.0 7 0.4 79.3 84.0 Standard EC 7.8 43.2 45.1 6 1.8 68.3 75.3 August 8, 2001 Daily application; feeling before treatment with WBPH

染平均値：3128隻昆蟲/20堆土墩（=稻株群組） -60 - 200529745 (58)Average pupae: 3128 insects / 20 piles of mounds (= rice plant group) -60-200529745 (58)

表17.4-三個位置之平均値劑量調合物在以WBPH處理後的害蟲防治率 1 DAT 3DAT 7DAT 1 4D AT 2 1 DAT 28D AT 1 AL1 32.6 46.0 60.9 64.5 57.0 49.5 標準EC 26.1 42.9 52.3 64.6 63.2 53.9 2 AL1 40.2 58.0 68.6 75.8 73.9 73.7 標準EC 30.5 48.9 64.5 65.8 64.7 63.1 3 AL1 38.0 54.3 66.1 77.4 72.8 67.0 標準E C. 32.7 53.2 67.0 74.9 7 1.1 67.2 4 AL1 39.7 60.9 73.1 80.0 75.5 77.3 標準EC 36.0 57.6 72.8 78.6 76.4 76.3 在2 0 0 1年施藥 -61 - 200529745 (59)Table 17.4-The average pest control rate of the three pupal dose blends after treatment with WBPH 1 DAT 3DAT 7DAT 1 4D AT 2 1 DAT 28D AT 1 AL1 32.6 46.0 60.9 64.5 57.0 49.5 Standard EC 26.1 42.9 52.3 64.6 63.2 53.9 2 AL1 40.2 58.0 68.6 75.8 73.9 73.7 Standard EC 30.5 48.9 64.5 65.8 64.7 63.1 3 AL1 38.0 54.3 66.1 77.4 72.8 67.0 Standard E C. 32.7 53.2 67.0 74.9 7 1.1 67.2 4 AL1 39.7 60.9 73.1 80.0 75.5 77.3 Standard EC 36.0 57.6 72.8 78.6 76.4 76.3 Application in 2001 -61-200529745 (59)

表5-位置·· HuN-IPP 劑量調合物在施藥後對常見蜘蛛的次級防治率 1DAT 3DAT 7DAT 1 4D AT 21DAT 28D AT 1 AL1 10.5 15.0 14.6 28.0 24.3 13.4 標準EC 10.9 15.2 15.2 29.8 25.4 14.7 2 AL1 12.4 16.7 16.6 29.3 25.5 15.8 標準EC 13.4 17.3 17.1 3 1.1 26.7 15.8 3 AL1 15.1 18.5 18.0 30.8 27.1 17.5 標準EC 14.6 19.1 18.0 3 1.8 27.5 17.4 4 AL1 15.2 17.7 17.2 32.3 27.9 1 8.9 標準EC 16.1 20.2 18.1 33.5 29.3 19.8 在2001年9月13日施藥Table 5-Location · Secondary control rate of HuN-IPP dose blends on common spiders after application 1DAT 3DAT 7DAT 1 4D AT 21DAT 28D AT 1 AL1 10.5 15.0 14.6 28.0 24.3 13.4 Standard EC 10.9 15.2 15.2 29.8 25.4 14.7 2 AL1 12.4 16.7 16.6 29.3 25.5 15.8 Standard EC 13.4 17.3 17.1 17.1 3 1.1 26.7 15.8 3 AL1 15.1 18.5 18.0 30.8 27.1 17.5 Standard EC 14.6 19.1 18.0 3 1.8 27.5 17.4 4 AL1 15.2 17.7 17.2 32.3 27.9 1 8.9 Standard EC 16.1 20.2 18.1 33.5 29.3 19.8 Application on September 13, 2001

說明：相較於標準EC調合物，於AL1調合物中該農業化學之活性物質愛西叵防治這兩種害蟲之活性平均來說明顯地增加了。不過相較於標準EC調合物，使用AL 1調合物對於常見蜘蛛的次級活性並沒有升高。 1 8 ·密度、pH値、水面散佈率及安定性步驟代表性標準法的使用結果 -62- 200529745 (60)Note: Compared with the standard EC blend, the active ingredient of Azadirachta in the AL1 blend has a significantly increased activity in controlling these two pests on average. However, compared with standard EC blends, the use of AL 1 blends did not increase the secondary activity of common spiders. 1 8 · Density, pH, water surface spread rate and stability Procedure Use of representative standard method Result -62- 200529745 (60)

表1 8-調合物類型AL1至AL6所測得的數據調合物類型密度安定性（括弧內的數據係於50°C下儲存6週後所測得的數據） pH値水面上散佈情形- 評估（§) 0小時 (h)後 1小時 (h )後 2 4小時 (h)後 AL1 1.0006 3.6 3 5/6 (3.8 ) (3 ) (5/6 ) AL2 0.9912 4.0 1/3 3 2 (4.0 ) (3 ) (2 ) (6) AL3 1 .0403 4.6 1 6 (4.2 ) (1 ) (6 ) AL4 1.041 4.5 1 5 6 (4.0 ) (1 ) (1/5 ) (1 ) AL5 1.042 4.4 1 6 6** (4.4 ) (1 ) (1 ) (6) * AL6 1.039 4.4 1 1 6" (4.4 ) (1 ) (1 ) (6)* 縮寫：h =小時；（§ )於培養皿內測試，在儲存期間有加蓋；關於此項，係使用如下評分法·· 1 ·在水面上有均質膜，於表面可看到分光色彩，2 ·有均質膜但無分光色彩’ 3 · 具有小凸起之非均質膜，4·具有大凸起之非均質膜’ 5.撕裂的膜，覆蓋面積〉5 〇 °/。’ 6 .撕裂的膜’覆室面積〈5 〇 % ( * 無結晶，* *稍有結晶）’ 7及8 ·滴狀物形成’ 9 ·未觀察到散佈的情形。 -63- 200529745 (61) 此等數據顯示所有測試之調合物類型皆具有適當的密度。全部的受測調合物類型在每一個測試時間下都具有令人滿意至優良程度的水面散佈率。所有的受試調合物類型在勉強的儲存條件下（於5 0 °C下達6週）仍可具有良好的安定性。除了此等數據以外，該等調合物AL1至AL6於-1(TC 下儲存後並無任何結晶形成的跡象故而證明此等調合物類型在冷凍下仍很安定。此外，該等調合物類型具有有利的閃點性質如AL 1爲 95°C且 AL3爲96°C，由於此種特性可以消除或減少特殊的安全性考量之需求，故而可讓該等植物之保護組成物的儲存更爲容易。 -64-Table 1 8- Measured data for blend types AL1 to AL6 Blend type density stability (data in parentheses are measured after storage at 50 ° C for 6 weeks) pH 値 Spread on water-Evaluation (§) 0 hours (h), 1 hour (h), 24 hours (h), AL1 1.0006 3.6 3 5/6 (3.8) (3) (5/6) AL2 0.9912 4.0 1/3 3 2 (4.0 ) (3) (2) (6) AL3 1.0403 4.6 1 6 (4.2) (1) (6) AL4 1.041 4.5 1 5 6 (4.0) (1) (1/5) (1) AL5 1.042 4.4 1 6 6 ** (4.4) (1) (1) (6) * AL6 1.039 4.4 1 1 6 " (4.4) (1) (1) (6) * Abbreviation: h = hour; (§) in a petri dish The test is stamped during storage. For this item, the following scoring method is used: · 1 · There is a homogeneous film on the water surface, and the spectroscopic color can be seen on the surface; 2 · There is a homogeneous film but no spectroscopic color '3 · Has Heterogeneous film with small bulges, 4. Heterogeneous film with large bulges' 5. Tearing film, covering area> 50 ° /. '6. Torn film' Covering area <50% (* no crystal, * * slightly crystalline) '7 and 8 · Drop formation' 9 · No scattering was observed. -63- 200529745 (61) These data show that all blend types tested have proper density. All tested compound types have satisfactory surface spread rates at each test time. All test compound types have good stability under marginal storage conditions (up to 6 weeks at 50 ° C). In addition to these data, the blends AL1 to AL6 did not show any signs of crystal formation after storage at -1 ° C, which proves that these blend types are still stable under freezing. In addition, these blend types have Beneficial flash point properties, such as AL 1 at 95 ° C and AL3 at 96 ° C. This feature can eliminate or reduce the need for special safety considerations, making it easier to store the protective composition of these plants -64-

Claims

200529745 (1) 10. Scope of patent application1. A method for controlling pests and diseases of rice crops, which is a plant protection composition containing the following composition: (2-ethylhexyl lactate, (b)-or more The active substance of agricultural chemistry dissolved in the composition, and (c) any one or more formulating aids; applied to the water or water surface of the rice field. 2 · The method according to item 1 of the patent application range, wherein the agriculture The chemical active substance is selected from the group: 〇 alonifen, amidosulfuron, anilofos, huangcaoling, befuresate, bis Byspiribac · sodium, bromobenzonitrile, green malon, cyclanilide, desmedipham, dilo fop-methyl (dichlorophenoxyphenoxy) Methyl propionate), diflufenican, diurfenican, ethephon, ethofumesate, ethoxysulfuron, fenoxaprop-P-ethyl , Fentrazamide, Flucar Ketone (flucarbazone)-sodium, flufenacet, f 1 urt am ο ne, foramsulfuron, glufosinate. Qian Qiang Iodosulfuron, acenaphthonitrile, isoproturon, isoxaflutole, linuron, mefenacet, Zhongfufurong (-65- 200529745 ( 2) mesofu 1 fur ο η) -methyl, metami 11 (meta 11 ο η), metosulam, secketin, oxadiargyl, oxadiazine, fenamidifene (Phenmedipham), ropoxycarbazone-sodium, sulxotrione and thidiauron;

2) acetamiprid, arinathrin, adicarb, double armor, cotton bud, cyfluthrin, saviin, clothianidin ), Cyfluthrin, cypermethrin, deltamethrin, thiomethanine, ethiprole, gram scale, fenamiphos, fenthion, ricinte, imidacloprid, polychlorin Phosphorus, chlorfencarb, chlorpheniramine, maple-sucking phosphorus, permethrin, fenfosin, prothiofos, silafluofen, spirodiclofen, romich Spiromesifen, thiacloprid, thiodicarb, tralomethrin, tri-D sitting phosphorus, trichlorfon and tr i flumuron; and 3) Bitertanol, carbendazim, carpropamid, keyusan, fenamidone, fenhexamid, fentin, fusarium (Fluoxastrobin), fosetyl-aluminum, puffin, iprovalicarb, poncecro (PenCyCUron), propamocarb hydrochloride, zinc methenoate, prothioconazole, pirimethanil, spiroxamine, tolufenad-dichlorofur (T0) yifiuanid · -66- 200529745

dichlofluanid) and trifloxystrobin. 3. The method according to item 2 of the scope of patent application, wherein the active substance of the agricultural chemistry is selected from the following group 2): C

2) acetamiprid, arinathrin, aldicarb, dimethypam, cotton wool, cyfluthrin, sivevain, clothianidin ), Cyfluthrin, cypermethrin, deltamethrin, sulfanil, ethiprole, fenfosin, fenamiphos, fenthion, ricinte, imidacloprid, doxorubicin Phosphorus, chlorfendicarb, carbendazim, phosphine, permethrin, fenfosin, prothiofos, silafluofen, spirodiclofen, romich Spiromesifen, thiacloprid, thiodifendicarb, tralomethrin, trisinophos, trichlorfon and triflumuron ° 4 · If the scope of patent application The method according to item 3, wherein the active chemical substance of the agricultural chemistry is selected from the group consisting of Ruijinte and Aisein. 5. The method according to item 1 of the patent application scope, wherein the plant protection composition contains a polydimethylsiloxane as a formulating aid c). 6. A plant protection composition comprising: (a) 2-ethylhexyl lactate, (b)-or more agrochemical active substances soluble in the composition 'and the agrochemical active substance system From the following groups: 1) alonifen, amidosulfuron, anilofos, Huangcaoling, Banforset (-67- 200529745 (4) befuresate) , Byspiribac-sodium, bromobenzonitrile, green malon, cyclanilide, desmedipham, dichloro fop-methyl (dichlorophenoxy) Methylphenoxypropionate), diflufenican, diuronic, ethephon, ethofumesate, ethoxysulfuron, fenoxaprop -P -Ethyl, fentrazamide, flucarbazone, sodium, flufenacet, flutamone, foramsulfuron, glufosinate )-Qian, yarrow, bowl of iodosulfuron, benzonitrile, isoprom (isop roturon), isoxaflutole, linuron, mefenacet, mesofulfuron-methyl, metamitron, metosulam 'Sekjin, oxadiargy 1, evil spirit

, Phenmedipham, ropoxycarbazone-sodium, suixotrione and thidiauron 2) acetamiprid, Arinathasson (acrinathrin), aldicarb, dimethyam, cotton wool, cyfluthrin, sivain, clothianidin, cyfUthrin, cypermethrin, Deltamethrin, sulfanil, ethiprole 'fencloxacin, fenam iphοs, fenthion, ricinte, imidacloprid, polychlorfen, fendicarb, fendicarb Spirits, crushing the pity 'suffering chrysanthemum vinegar' and killing the pity phosphine, pr 0 thi 〇f 〇s, Sheila-68- 200529745 (5) Fulafen (silafluofen), spirodicrofen (spi ι * odic 1 ofe η), spiro mesifen, thiacloprid, thiodicarb, dolosulfam, tralomethrin, triwaphos, trichlorfon and triflumuron ); Η

3) bitertanol, carbendazim, carpropamid, keyusan, fenamidone, fenhexamid, fentin, rich Axatrobin (fluoxastrobin), fosetyl-Ming, puffin, tone [1; iprovalicarb, pencycuron, propamocarb hydrochloride, a Gideson zinc, prothioconazole, pirimethanil, spiroxamine, tolylfluanid-dichlofluanid and trifluorooxetine (Trifloxystrobin); and (c) any one or more formulating aids 7 · The plant protection composition according to item 6 of the patent application, wherein the active substance of the agricultural chemistry is selected from the following group 2): 2) Acetamiprid, acrinathri η, aldicarb, dimethypam, cotton boron phosphate, cyfluthrin, sivevain, clothianidin , Cyfluthrin, cypermethrin, deltamethrin, sulfanil, Ethiprole, fenamiphos, fenamiphos, fenthion, ricinte, imidacloprid, polychlorfen, fendicarb, fenfen, phosphine, permethrin, voltam Phosphoric acid kill, pr 〇thi 〇f 〇s, silafluofen, spirodiclofen, Luo-69- 200529745 (6) spiromesifen, SEC Thiacloprid, thiodifendicarb, tralomethrin, triazophos, trichlorfon, and tr ifl umur on. 8. The plant protection composition according to item 7 of the patent application scope, wherein the " agrochemical active chemical substance is selected from the group consisting of Ruijinte and Aixin. • 9 • The plant protection composition according to item 7 of the scope of patent application, wherein the plant protection composition contains a polydimethylsiloxane as a formulating aid η 〇〇1 〇 Plant protection composition, further comprising a member selected from the group consisting of benzyl alcohol, dimethyl sulfoxide (DMSO), C12-C15 alkyl benzoate, diisopropyl ferrate, N-octyl pyrrolidone and dimethyl Solvent of acetamide. 1 1. An active substance concentrate comprising: (a) 2-ethylhexyl lactate, (b)-or more agrochemical active substances soluble in the concentrate, and the agrochemical The active substance is selected from the following groups:-1) alonifen, amidosulfuron., Anilofos, yellow grass, befuresate, Byspiribac-sodium, bromobenzonitrile, green wheat, cyclanilide, desmedipham, diclofop-methyl (dichlorophenoxybenzene) Methyl propionate), diflufenican, diurfenican, ethephon, ethofumesate, ethoxysulfuron, fenoxaprop-P-ethyl Fentrazamide (-70- 200529745 (7) fentrazamide), flucarbazone-sodium, flufenacet, flurtamone, foramsulfuron, sugar Glufosinate-money, scopolamine, iodosulfuron, iodobenzene , Isoproturon, isoxaflutole, -linuron, mefenacet, mesofulfuron-methyl, metamitron , Thiosulfan (, metosulam), secketin, oxadiargyl, oxadiline, phenmedipham, ropoxycarbazone-sodium, sulx 〇trione) and thidiauron; 2) acetamiprid, arinathrin 'Tiatianwei' Shuangjiamai 'cotton swabs, beta-cyfluthrin , Silvein, clothianidin, cyfluthrin 'cypermethrin, deltamethrin, sulfanil, ethethrole, fenflufen, fenaniiphos , Fenthion ^, Regent, Imidacloprid, Polychlorfen, Chlorphene, Methylim, Phosphorus, • Permethrin, Phosphos, Prothiofos, Girafufen ( silafluofen), spirodiclofen, spiromesifen Luopi (thiac 1 oprid), thiodifendicarb, tralomethrin, triazophos, trichlorfos and tri flumuron; 3) bitertanol, polybacteria Ling, Carpropamid, Kewensan, Fenaniidone, Fenhai-71-200529745 (8) fenhexamid, fen tin, Fusaid Fluoxastrobin, Fosetyl Lu, Po Haiin, Iprovalicarb, Pencycuron, Propamocarb Hydrochloride, Methyl Zinc Methylate, Rhenium R prothioconazole, pirimethanil, spiroxamine, tolufenad-dichlorofunad (10.1 > ^ 1 £ '11 ^ 1 ^ ( 3. dichlofluanid) and trifloxystrobin. ^ 1 2. A water-soluble container containing a plant protection composition as described in item 7 of the patent application. -72- 200529745 VII. Designated representative map: (1). The designated representative map in this case is ... None (2). The component representative symbols of this representative map are simply explained: None 4

8. If there is a chemical formula in this case, please disclose the chemical formula that best shows the characteristics of the invention: None