TR200002757T2 - Indol derivatives with an anti-virus activity - Google Patents

Indol derivatives with an anti-virus activity

Info

Publication number
TR200002757T2
TR200002757T2 TR2000/02757T TR200002757T TR200002757T2 TR 200002757 T2 TR200002757 T2 TR 200002757T2 TR 2000/02757 T TR2000/02757 T TR 2000/02757T TR 200002757 T TR200002757 T TR 200002757T TR 200002757 T2 TR200002757 T2 TR 200002757T2
Authority
TR
Turkey
Prior art keywords
optionally substituted
hydrogen
lower alkyl
virus activity
compound
Prior art date
Application number
TR2000/02757T
Other languages
Turkish (tr)
Inventor
Fujishita Toshio
Yoshinaga Tomokazu
Original Assignee
Shionogi & Co., Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co., Limited filed Critical Shionogi & Co., Limited
Publication of TR200002757T2 publication Critical patent/TR200002757T2/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

R1'in hidrojen, alt alkyl, veya tercihe göre ikameli arylsulfonyl, veya benzeri, R2'nin hidrojen, alt alkyl, veya tercihe göre ikameli aralkyl, veya benzeri, Herbir R3,R4,R5, ve R6'nin ayri ayri hidrojen, halojen, trihalojenatli alt alkyl, veya benzeri, X'in hydroxy veya tercihe göre ikameli amino; Y'nin COOR (R, hidrojen veya bir ester kalintisi), tercihe göre ikameli aryl, veya tercihe göre ikameli heteroaryl, oldugu bir formül (I): bilesiminin integraz inhibisyon aktivitesi olup, bir anti-HIV ilaç olarak kullanilabilir.R1 is hydrogen, lower alkyl, or optionally substituted arylsulfonyl, or the like, R2 is hydrogen, lower alkyl, or optionally substituted aralkyl, or the like, Each R3, R4, R5, and R6 are separately hydrogen, halogen trihalogenated lower alkyl, or the like, X is hydroxy or optionally substituted amino; A compound of formula (I) wherein Y is COOR (R, hydrogen or an ester residue), optionally substituted aryl, or optionally substituted heteroaryl, is the integrase inhibition activity of the compound, which can be used as an anti-HIV drug.

TR2000/02757T 1998-03-26 1999-03-26 Indol derivatives with an anti-virus activity TR200002757T2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP82031998 1998-03-26

Publications (1)

Publication Number Publication Date
TR200002757T2 true TR200002757T2 (en) 2000-12-21

Family

ID=18528443

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2000/02757T TR200002757T2 (en) 1998-03-26 1999-03-26 Indol derivatives with an anti-virus activity

Country Status (1)

Country Link
TR (1) TR200002757T2 (en)

Similar Documents

Publication Publication Date Title
EP1069111A4 (en) Indole derivatives with antiviral activity
CA2396738A1 (en) Thiazole derivatives as active superoxide radical inhibitors
BR0110404A (en) Imidazopyrimidine derivatives and triazolpyrimidine derivatives
BR0013237A (en) Antibacterial heterobicyclic substituted phenyl oxazolidinones
ID29452A (en) 4-OKSO-1,4-DIHYDRO-3-QUINOLINKARBOXAMIDE AS ANTIVIRUS AGENTS
DK459086D0 (en) quinazoline
DK345989A (en) quinoline
NZ233735A (en) Heterocyclic substituted aminophenol derivatives
ATE120955T1 (en) BENZYLIDENE-MALONONITRILE DERIVATIVES FOR INHIBITING PROLIFERATIVE PROCESSES IN MAMMAL CELLS.
MXPA02006329A (en) Substituted 8arylquinoline phosphodiesterase4 inhibitors.
NO20022976L (en) 2- (1H-indol-3yl) -2-oxoacetamides with antitumor activity
DK1042319T3 (en) dihydrobenzofuranes
ATE262509T1 (en) INDOLINE DERIVATIVES AS LIGHT PROTECTIVE AGENTS
DE60036558D1 (en) PHTHALAZINONE DERIVATIVES AS PDE 4 HEMMER
ATE264322T1 (en) ANTI-TUMOR DIHYDROQUINAZOLINE DERIVATIVES
TR200002757T2 (en) Indol derivatives with an anti-virus activity
TR200103685T2 (en) Optically active pyrolopyridazine derivatives
MA24197A1 (en) NEW FUNGARRESTINES
TR199801366T2 (en) �zooksasefem t�revleri.
ATE480533T1 (en) VARIOLINE DERIVATIVES AND THEIR USE AS CYTOSTATICS
GB9908021D0 (en) Pharmaceutical compounds
ATE69819T1 (en) 1-OXA-1-DETHIA CEPHALOSPORIN COMPOUNDS AND ANTIBACTERIAL AGENT CONTAINING THEM.
ATE243698T1 (en) 1,2-DIHYDRO-1-OXO-PYRAZINO(1,2-)INDOLE DERIVATIVES
YU74501A (en) Synthesis of 3-amino-3-aryl propionates
TR200300359T4 (en) Substituted novel (dihydro) benzoxazine and (dihydro) benzothiazine derivatives, their preparation methods and pharmaceutical compositions containing them