TNSN03129A1 - HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING THEM, PHARMACEUTICAL USES THEREOF, AND MATERIALS FOR THEIR SYNTHESIS. - Google Patents

HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING THEM, PHARMACEUTICAL USES THEREOF, AND MATERIALS FOR THEIR SYNTHESIS.

Info

Publication number
TNSN03129A1
TNSN03129A1 TNPCT/US2002/018548A TNSN03129A TNSN03129A1 TN SN03129 A1 TNSN03129 A1 TN SN03129A1 TN SN03129 A TNSN03129 A TN SN03129A TN SN03129 A1 TNSN03129 A1 TN SN03129A1
Authority
TN
Tunisia
Prior art keywords
compositions containing
compounds
hiv protease
synthesis
materials
Prior art date
Application number
TNPCT/US2002/018548A
Other languages
French (fr)
Inventor
Stacie S Canon-Koch
Therese N Alexander
Mark Barvian
Gary Bolton
Fredrick E Boyer
Benjamin J Burke
Tod Holler
Tanya M Jewell
Josyula Vara Prasad
David J Kucera
Jeff Machak
Lennert J Mitchell
Sean T Murphy
Siegfried H Reich
Donald J Skalitzky
John H Tatlock
Michael D Varney
Scott C Virgil
Stephen T Worland
Michael Melnick
Maria A Linton
Stephen E Webber
Original Assignee
Agouron Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Agouron Pharma filed Critical Agouron Pharma
Publication of TNSN03129A1 publication Critical patent/TNSN03129A1/en

Links

Landscapes

  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

DES COMPOSES DE FORMULE (I), DANS LAQUELLE LES VARIABLES REPONDENT AUX DEFINITIONS FIGURANT DANS LE PRESENT MEMOIRE, QUI INHIBENT OU BLOQUENT AVANTAGEUSEMENT L'ACTIVITE BIOLOGIQUE DE LA PROTEASE DU VIH, SONT DECRIT. CES COMPOSES, AINSI QUE DES COMPOSITIONS PHARMACEUTIQUES CONTENANT CES COMPOSES, SONT UTILES POUR LE TRAITEMENT DE PATIENTS OU D'HOTES INFECTES PAR LE VIRUS VIH. DES INTERMEDIAIRES ET PROCEDES DE SYNTHESE POUR LA PREPARATION DE CES COMPOSES SONT EGALEMENT DECRITS.COMPOUNDS OF FORMULA (I), IN WHICH THE VARIABLES MEET THE DEFINITIONS APPEARING IN THIS MEMORY, WHICH INHIBIT OR BENEFIT BLOCK THE BIOLOGICAL ACTIVITY OF HIV PROTEASE, ARE DESCRIBED. THESE COMPOUNDS, AS WELL AS PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, ARE USEFUL FOR THE TREATMENT OF PATIENTS OR HOSTS INFECTED BY THE HIV VIRUS. INTERMEDIATES AND SYNTHESIS METHODS FOR THE PREPARATION OF THESE COMPOUNDS ARE ALSO DESCRIBED.

TNPCT/US2002/018548A 2001-06-11 2003-07-08 HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING THEM, PHARMACEUTICAL USES THEREOF, AND MATERIALS FOR THEIR SYNTHESIS. TNSN03129A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US29746001P 2001-06-11 2001-06-11

Publications (1)

Publication Number Publication Date
TNSN03129A1 true TNSN03129A1 (en) 2005-12-23

Family

ID=34078857

Family Applications (1)

Application Number Title Priority Date Filing Date
TNPCT/US2002/018548A TNSN03129A1 (en) 2001-06-11 2003-07-08 HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING THEM, PHARMACEUTICAL USES THEREOF, AND MATERIALS FOR THEIR SYNTHESIS.

Country Status (5)

Country Link
EC (2) ECSP034893A (en)
HN (1) HN2002000143A (en)
TN (1) TNSN03129A1 (en)
UA (1) UA77180C2 (en)
ZA (2) ZA200309040B (en)

Also Published As

Publication number Publication date
ECSP034893A (en) 2004-08-27
ECSP034892A (en) 2004-01-28
ZA200309041B (en) 2004-07-22
ZA200309040B (en) 2005-05-27
HN2002000143A (en) 2002-11-25
UA77180C2 (en) 2006-11-15

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