TNSN03129A1 - HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING THEM, PHARMACEUTICAL USES THEREOF, AND MATERIALS FOR THEIR SYNTHESIS. - Google Patents
HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING THEM, PHARMACEUTICAL USES THEREOF, AND MATERIALS FOR THEIR SYNTHESIS.Info
- Publication number
- TNSN03129A1 TNSN03129A1 TNPCT/US2002/018548A TNSN03129A TNSN03129A1 TN SN03129 A1 TNSN03129 A1 TN SN03129A1 TN SN03129 A TNSN03129 A TN SN03129A TN SN03129 A1 TNSN03129 A1 TN SN03129A1
- Authority
- TN
- Tunisia
- Prior art keywords
- compositions containing
- compounds
- hiv protease
- synthesis
- materials
- Prior art date
Links
Landscapes
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
DES COMPOSES DE FORMULE (I), DANS LAQUELLE LES VARIABLES REPONDENT AUX DEFINITIONS FIGURANT DANS LE PRESENT MEMOIRE, QUI INHIBENT OU BLOQUENT AVANTAGEUSEMENT L'ACTIVITE BIOLOGIQUE DE LA PROTEASE DU VIH, SONT DECRIT. CES COMPOSES, AINSI QUE DES COMPOSITIONS PHARMACEUTIQUES CONTENANT CES COMPOSES, SONT UTILES POUR LE TRAITEMENT DE PATIENTS OU D'HOTES INFECTES PAR LE VIRUS VIH. DES INTERMEDIAIRES ET PROCEDES DE SYNTHESE POUR LA PREPARATION DE CES COMPOSES SONT EGALEMENT DECRITS.COMPOUNDS OF FORMULA (I), IN WHICH THE VARIABLES MEET THE DEFINITIONS APPEARING IN THIS MEMORY, WHICH INHIBIT OR BENEFIT BLOCK THE BIOLOGICAL ACTIVITY OF HIV PROTEASE, ARE DESCRIBED. THESE COMPOUNDS, AS WELL AS PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, ARE USEFUL FOR THE TREATMENT OF PATIENTS OR HOSTS INFECTED BY THE HIV VIRUS. INTERMEDIATES AND SYNTHESIS METHODS FOR THE PREPARATION OF THESE COMPOUNDS ARE ALSO DESCRIBED.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US29746001P | 2001-06-11 | 2001-06-11 |
Publications (1)
Publication Number | Publication Date |
---|---|
TNSN03129A1 true TNSN03129A1 (en) | 2005-12-23 |
Family
ID=34078857
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TNPCT/US2002/018548A TNSN03129A1 (en) | 2001-06-11 | 2003-07-08 | HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING THEM, PHARMACEUTICAL USES THEREOF, AND MATERIALS FOR THEIR SYNTHESIS. |
Country Status (5)
Country | Link |
---|---|
EC (2) | ECSP034893A (en) |
HN (1) | HN2002000143A (en) |
TN (1) | TNSN03129A1 (en) |
UA (1) | UA77180C2 (en) |
ZA (2) | ZA200309040B (en) |
-
2002
- 2002-06-11 HN HN2002000143A patent/HN2002000143A/en unknown
- 2002-11-06 UA UA20031110768A patent/UA77180C2/en unknown
-
2003
- 2003-07-08 TN TNPCT/US2002/018548A patent/TNSN03129A1/en unknown
- 2003-11-20 ZA ZA200309040A patent/ZA200309040B/en unknown
- 2003-11-20 ZA ZA200309041A patent/ZA200309041B/en unknown
- 2003-12-11 EC EC2003004893A patent/ECSP034893A/en unknown
- 2003-12-11 EC EC2003004892A patent/ECSP034892A/en unknown
Also Published As
Publication number | Publication date |
---|---|
ECSP034893A (en) | 2004-08-27 |
ECSP034892A (en) | 2004-01-28 |
ZA200309041B (en) | 2004-07-22 |
ZA200309040B (en) | 2005-05-27 |
HN2002000143A (en) | 2002-11-25 |
UA77180C2 (en) | 2006-11-15 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
TNSN03130A1 (en) | HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING THEM, PHARMACEUTICAL USES THEREOF AND MATERIALS FOR THEIR SYNTHESIS | |
TNSN99253A1 (en) | CHEMICAL COMPOUNDS NOVEL MODULATORS OF CCR5, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM. | |
MA26877A1 (en) | AZETIDINE DERIVATIVES, THEIR PREPARATION AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
TNSN99053A1 (en) | ACID HYDROXAMIDES (4-ARYLSULFONYLAMINO) -TETRAHYDRO- PYRANNE-4-CARBOXYLIQUES), PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM | |
MA27774A1 (en) | PHOSPHATIDYLINOSITOL 3-KINASE INHIBITORS | |
ATE443043T1 (en) | PHENYLCARBOXAMIDE AS A BETA-SECRETASE INHIBITOR FOR THE TREATMENT OF ALZHEIMER'S | |
TNSN99055A1 (en) | NEW BICYCLIC HYDROXAMIC ACID DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
MA27908A1 (en) | THERAPEUTIC AGENTS USEFUL FOR THE TREATMENT OF PAIN | |
TNSN98025A1 (en) | ARYLSULFONYLHYDROXAMIC ACID DERIVATIVES, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM. | |
TNSN99006A1 (en) | 4- (2-CETO-1-BENZIMIDAZOLINYL) NOVEL PIPERIDINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
TNSN99156A1 (en) | NOVEL HYDROXYPIPECOLATE-HYDROXAMIC ACID DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
MA30089B1 (en) | (Arylsulfonyl) -PYRASOLOPIPERIDINES | |
MA26956A1 (en) | PYRIMIDINE-2,4,6, TRIONES INHIBITORS OF METALLOPROTEINASES. | |
BG100455A (en) | Hiv protease inhibitors | |
TNSN98084A1 (en) | DERIVATIVES OF SUBSTITUTED MACROLIDES IN POSITION C-4 | |
TNSN00092A1 (en) | NOVEL NPY ANTAGONIST COMPOUNDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM | |
TNSN98238A1 (en) | NEW MACROLIDES | |
TNSN00036A1 (en) | NOVEL OXAMIC ACIDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM. | |
MA28011A1 (en) | PIPERAZINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS | |
MA31894B1 (en) | Organic compositions | |
ATE517861T1 (en) | BENZYL ETHER AND BENZYLAMIN COMPOUNDS AS INHIBITORS OF BETA-SECRETASE FOR THE TREATMENT OF ALZHEIMER'S DISEASE | |
TNSN00235A1 (en) | NEW HETEROCYCLO-ALKYLSULFONYLPYRAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM | |
TNSN00250A1 (en) | NEW PCP INHIBITOR COMPOUNDS, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM | |
DE69518840D1 (en) | N-(3-amino-2-hydroxybutyl)sulfonamid-derivate as hiv-protease-inhibitoren | |
EA200200625A1 (en) | ANTIPICORNAVIRAL COMPOUNDS AND COMPOSITIONS, THEIR PHARMACEUTICAL APPLICATION AND SUBSTANCES FOR THEIR SYNTHESIS |