TN2011000070A1 - Picolinamide derivatives as kinase inhibitors - Google Patents

Picolinamide derivatives as kinase inhibitors

Info

Publication number
TN2011000070A1
TN2011000070A1 TN2011000070A TN2011000070A TN2011000070A1 TN 2011000070 A1 TN2011000070 A1 TN 2011000070A1 TN 2011000070 A TN2011000070 A TN 2011000070A TN 2011000070 A TN2011000070 A TN 2011000070A TN 2011000070 A1 TN2011000070 A1 TN 2011000070A1
Authority
TN
Tunisia
Prior art keywords
kinase
compositions
compounds
kinase inhibitors
picolinamide
Prior art date
Application number
TN2011000070A
Other languages
French (fr)
Inventor
Wooseok Han
Jiong Lan
Gisele Nishiguchi
Matthew T Burger
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/EP2009/061205 external-priority patent/WO2010026124A1/en
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of TN2011000070A1 publication Critical patent/TN2011000070A1/en

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  • Pyridine Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

New picolinamide compounds, compositions and methods of inhibition of Provirus Integration of Maloney Kinase (PIM kinase) activity associated with tumorigenesis in a human or animal subject are provided. In certain embodiments, the compounds and compositions are effective to inhibit the activity of at least one PIM kinase. The new compounds and compositions may be used either alone or in combination with at least one additional agent for the treatment of a serine/threonine kinase- or receptor tyrosine kinase-mediated disorder, such as cancer.
TN2011000070A 2009-08-31 2011-02-11 Picolinamide derivatives as kinase inhibitors TN2011000070A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/EP2009/061205 WO2010026124A1 (en) 2008-09-02 2009-08-31 Picolinamide derivatives as kinase inhibitors

Publications (1)

Publication Number Publication Date
TN2011000070A1 true TN2011000070A1 (en) 2012-09-05

Family

ID=55024382

Family Applications (1)

Application Number Title Priority Date Filing Date
TN2011000070A TN2011000070A1 (en) 2009-08-31 2011-02-11 Picolinamide derivatives as kinase inhibitors

Country Status (1)

Country Link
TN (1) TN2011000070A1 (en)

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