TH77364A - Aryl-pyridine derivative as a inhibitor 11-beta-HSD1 - Google Patents
Aryl-pyridine derivative as a inhibitor 11-beta-HSD1Info
- Publication number
- TH77364A TH77364A TH501003445A TH0501003445A TH77364A TH 77364 A TH77364 A TH 77364A TH 501003445 A TH501003445 A TH 501003445A TH 0501003445 A TH0501003445 A TH 0501003445A TH 77364 A TH77364 A TH 77364A
- Authority
- TH
- Thailand
- Prior art keywords
- hsd1
- beta
- inhibitor
- aryl
- alkyl
- Prior art date
Links
- 102100015241 HSD11B1 Human genes 0.000 title 1
- 101710013483 HSD11B1 Proteins 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 230000002401 inhibitory effect Effects 0.000 title 1
- 239000000126 substance Substances 0.000 claims abstract 4
- 150000001875 compounds Chemical class 0.000 claims abstract 3
- 239000003814 drug Substances 0.000 claims abstract 3
- 229940079593 drugs Drugs 0.000 claims abstract 2
- 125000000217 alkyl group Chemical group 0.000 claims 3
- 150000002431 hydrogen Chemical group 0.000 claims 3
- 229910052739 hydrogen Inorganic materials 0.000 claims 3
- 239000001257 hydrogen Substances 0.000 claims 3
- 229910052736 halogen Chemical group 0.000 claims 2
- 150000002367 halogens Chemical group 0.000 claims 2
- 125000003545 alkoxy group Chemical group 0.000 claims 1
- 125000004103 aminoalkyl group Chemical group 0.000 claims 1
- 125000000753 cycloalkyl group Chemical group 0.000 claims 1
- -1 hydroxy, hydroxy Chemical group 0.000 claims 1
- 125000001624 naphthyl group Chemical group 0.000 claims 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 claims 1
- 125000004076 pyridyl group Chemical group 0.000 claims 1
- 125000001544 thienyl group Chemical group 0.000 claims 1
- 150000002148 esters Chemical class 0.000 abstract 2
- 239000000203 mixture Substances 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 239000011780 sodium chloride Substances 0.000 abstract 2
Abstract
DC60 (17/10/48) สารประกอบของสูตร (สูตรเคมี) (I) รวมทั้งเกลือและเอสเทอร์ของสารเหล่านี้ ที่ยอมรับได้ทางเภสัชกรรม ซึ่ง R1 ถึง R7, A, E และ G มี ความหมายตามที่กำหนดไว้ในข้อถือสิทธิ 1 สามารถถูกใช้ในรูปของสารผสมทางเภสัชกรรม สารประกอบของสูตร (สูตรเคมี) (I) รวมทั้งเกลือและเอสเทอร์ของสารเหล่านี้ ที่ยอมรับได้ทางเภสัชกรรม ซึ่ง R1 ถึง R7, A, E และ G มี ความหมายตามที่กำหนดไว้ในข้อถือสิทธิ 1 สามารถถูกใช้ในรูปของสารผสมทางเภสัชกรรม สิทธิบัตรยา DC60 (17/10/48) Compounds of formula (chemical formula) (I) as well as salts and esters of these substances. For which R1 to R7, A, E, and G have the meanings set forth in claim 1, they can be used as a pharmaceutical mixture. Compounds of the formula (chemical formula) (I) as well as their salts and esters. Acceptable pharmaceuticals of which R1 to R7, A, E, and G have the meanings set forth in claim 1, can be used as a pharmaceutical mix, drug patent.
Claims (1)
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TH77364A true TH77364A (en) | 2006-05-10 |
Family
ID=
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NO20073791L (en) | Pyrazolylaminopyridine derivatives useful as kinase inhibitors | |
| CR9314A (en) | DERIVATIVE OF SPIROCETAL AND USE OF THE SAME AS A MEDICINE FOR DIABETES | |
| ATE432272T1 (en) | AMINOPHENYL DERIVATIVES AS NEW INHIBITORS OF HISTONE DEACETYLASE | |
| CY1116885T1 (en) | Substituted cyclohexylmethyl derivatives | |
| TW200738684A (en) | Novel sulfated cyclic urea derivatives, preparation thereof and pharmaceutical use thereof as kinase inhibitors | |
| ATE500222T1 (en) | BENZAMIDE AND HETEROARE DERIVATIVES AS CETP INHIBITORS | |
| ATE543803T1 (en) | 3-Ä2-(3-AZYLAMINO-2-OXO-2H-PYRIDINE-1-YL)ACETYLAMINOÜ-4-OXOPENTANIC ACID DERIVATIVES AND THEIR USE AS CASPASE INHIBITORS | |
| UY29510A1 (en) | DERIVATIVES OF UREA, METHODS FOR ITS MANUFACTURING, AND USES OF THE SAME | |
| SE0400850D0 (en) | Novel Compounds | |
| NO20085317L (en) | Imidazoazepinonforbindelser | |
| DE502006008710D1 (en) | SUBSTITUTED TETRAHYDROISOCHINOLINES AS MMP INHIBITORS, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS A MEDICAMENT | |
| SG165381A1 (en) | Novel benzimidazole and benzothiazole derivatives, method for preparing same, use thereof as drugs, pharmaceutical compositions and novel use in particular as c-met inhibitors | |
| TH77364A (en) | Aryl-pyridine derivative as a inhibitor 11-beta-HSD1 | |
| EA201000720A1 (en) | 4,4-DESIGNED PIPERIDINES AS RENIN INHIBITORS | |
| ATE424394T1 (en) | 1H-INDOLE-3-CARBONIC ACID DERIVATIVES AND THEIR USE AS PPAR AGONISTS | |
| TH77088A (en) | Pyrimidine derivatives | |
| TH84138A (en) | N-formyl hydroxylamine compounds | |
| TH77591A (en) | 5-phenylthiazole derivatives (5-phenylthiazole derivatives) and their use as PI3 kinase inhibitors (PI3 Kinase inhibitors). | |
| TH83340A (en) | New compound | |
| TH87833A (en) | Perazolone derivatives | |
| TH75305A (en) | 7-phenylamino-4-quinolone-3-carboxylic acid derivatives, process for the preparation of these substances. And the use of these substances as drugs | |
| TH81547A (en) | Pyrimidine derivatives | |
| TH123699B (en) | Compound 4- [2- (2-fluoroximethyl) phenyl] piperidine | |
| TH97394A (en) | Aerylamide replaced with tetrazole | |
| TH98401A (en) | Material suspensions are stable in pharmaceuticals. |