SV2003000931A - GLUTARAMIDE DERIVATIVES REPLACED WITH N-FENPROPILCICLOPENTILO AS NEP INHIBITORS FOR FSAD REF.PCS10967 - Google Patents

GLUTARAMIDE DERIVATIVES REPLACED WITH N-FENPROPILCICLOPENTILO AS NEP INHIBITORS FOR FSAD REF.PCS10967

Info

Publication number
SV2003000931A
SV2003000931A SV2002000931A SV2002000931A SV2003000931A SV 2003000931 A SV2003000931 A SV 2003000931A SV 2002000931 A SV2002000931 A SV 2002000931A SV 2002000931 A SV2002000931 A SV 2002000931A SV 2003000931 A SV2003000931 A SV 2003000931A
Authority
SV
El Salvador
Prior art keywords
optionally replaced
hydro
replaced
pcs10967
fenpropilciclopentilo
Prior art date
Application number
SV2002000931A
Other languages
Spanish (es)
Inventor
Adam Thomas Gillmore
Stephen Challenger
Andrew Simon Cook
David Cameron Pryde
Donald Stuart Middleton
Alan Stobie
Original Assignee
Donald Stuart Middleton
Alan Stobie
Pfizer, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0107750A external-priority patent/GB0107750D0/en
Priority claimed from GB0113113A external-priority patent/GB2376080B/en
Priority claimed from GB0120152A external-priority patent/GB0120152D0/en
Application filed by Donald Stuart Middleton, Alan Stobie, Pfizer, Inc. filed Critical Donald Stuart Middleton
Publication of SV2003000931A publication Critical patent/SV2003000931A/en

Links

Landscapes

  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)

Abstract

LA INVENCION SE REFIERE A COMPUESTOS DE FORMULA (I)PARA TRATAR, POR EJEMPLO, DISFUNCIOPN SEXUAL, EN LA QUE R1 ES ALQUILO C1-6 OPCIONALMENTE SUSTITUIDO, CARBOCICLICO OPCIONALMENTE SUSTITUIDO, HETEROCICLILO OPCIONALMENTE SUSTITUIDO, HIDROGENO, ALCOXI C1-6, -NR2R3 O -NR4SO2R5, X ES EL ENLACE -(CH2)N O-(C2)Q-O-(DONDE Y ESTA UNIDO AL OXIGENO); DONDE UNO O MAS ATOMOSD E HIDROGENO EN EL ENLACE X SE PUEDEN REEMPLAZAR INDEPENDIENTEMENTE POR ALCOXI C1-4; HIDROXI; HIDROXI(ALQUILO C1-3); CICLOALQUILO C3-7; CARBOCICLILO; HETEROCICLILO; O POR ALQUILO C1-4 OPCIONALMENTE SUSTITUIDO CON UNO O MAS GRUPOS FLUORO O FENILO; N ES 3,4,5,6 O 7; Y Q ES 2,3,4,5 O 6; Y ES FENILO O PIRIDILO, CADA UNO DE LOS CUALES PUEDE ESTAR SUSTITUIDO; O DOS GRUPOS R8 EN LOS TOMOS DE CARBONO ADYACENTES JUNTO CON LOS ATOMOS DE CARONO QUE LE INTERCONECTAN PUEDEN FORMAR UN ANILLO CARBOCICLICO O HETEROCICLICO, CONDENSADO DE 5 O 6 MIEMBROS, OPCIONALMENTE SUSTITUIDO, VER FORMULAS.THE INVENTION REFERS TO FORMULA COMPOUNDS (I) TO TREAT, FOR EXAMPLE, SEXUAL DYSFUNCTION, IN WHICH R1 IS RENT C1-6 OPTIONALLY REPLACED, OPTIONALLY REPLACED CARBOCICLIC OPTIONALLY REPLACED, HYDRO-C1, HYDRO-C1, HYDRO-C1, HYDRO-C2 -NR4SO2R5, X IS THE LINK - (CH2) N O- (C2) QO- (WHERE AND IS JOINED TO THE OXYGEN); WHERE ONE OR MORE ATOMOSD AND HYDROGEN IN LINK X CAN BE REPLACED INDEPENDENTLY BY ALCOXI C1-4; HYDROXY; HYDROXI (C1-3 RENT); C3-7 CYCLEALKYL; CARBOCICLYL; HETEROCICLILO; OR BY C1-4 RENTAL OPTIONALLY REPLACED WITH ONE OR MORE FLUORO OR PHENYLL GROUPS; N ES 3,4,5,6 O 7; And Q ES 2,3,4,5 O 6; AND IT IS PHENYLL OR PIRIDILE, EACH OF WHICH CAN BE REPLACED; OR TWO R8 GROUPS IN THE ADJACING CARBON TAKES AND THE INTERCONNECTING CARONOMOM ATOMS CAN FORM A CARBOCICLIC OR HETEROCICLICAL RING, CONDENSED WITH 5 OR 6 MEMBERS, OPTIONALLY REPLACED, SEE FORMULAS.

SV2002000931A 2001-03-28 2002-03-22 GLUTARAMIDE DERIVATIVES REPLACED WITH N-FENPROPILCICLOPENTILO AS NEP INHIBITORS FOR FSAD REF.PCS10967 SV2003000931A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0107750A GB0107750D0 (en) 2001-03-28 2001-03-28 Novel pharmaceuticals
GB0113113A GB2376080B (en) 2001-05-30 2001-05-30 Flowmeter proving device
GB0120152A GB0120152D0 (en) 2001-08-17 2001-08-17 Novel pharmaceuticals

Publications (1)

Publication Number Publication Date
SV2003000931A true SV2003000931A (en) 2003-03-12

Family

ID=40091711

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2002000931A SV2003000931A (en) 2001-03-28 2002-03-22 GLUTARAMIDE DERIVATIVES REPLACED WITH N-FENPROPILCICLOPENTILO AS NEP INHIBITORS FOR FSAD REF.PCS10967

Country Status (1)

Country Link
SV (1) SV2003000931A (en)

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